SMILES C(=O)(CCCCCOC)NCC1C2CN(C(CC(C=C)C)=O)C1C2 N1(C(C2(C)CC2(Cl)Cl)=O)CCC(CNC(=O)CC2C=CCCC2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(C2OCCC2C(F)(F)F)=O)CC(=O)C12CCC2 C(=O)(CCCSC)N(C1CC(NC(C(C2CCOC2)N(C(C)(C)C)CC)=O)C1)C.CO c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)ccncc1OC(C)C c1(C(=O)NCC2C(CNC(c3c(OC)cc(C)cn3)=O)C2)sccc1S(N)(=O)=O CC(O)CCCCCC(=O)N1CCC(NC(c2ccccn2)=O)CC(C)(C)C1 C1(CNC(=NCC)NC(c2ccc(F)cc2F)C)CCC(F)(F)C(=O)N1 c1(C2(C(=O)NC3C(CNC(C(C)n4cccn4)=O)CC3)CC2)ccc(F)cn1 C(=O)(C(CC)(CC)CO)NC(CC=C)CNC(C1OC2CCC1C2)=O N1(C(CCn2ccc(C)n2)=O)CC2(CCC2CNC(=O)CSc2nnnn2C)C1 N1(CC)CCC(C(=O)NCC(O)CC(=O)NCC)CC1 C#CC1CCC(C(=O)NC2CCC(NC(C3CC4CC3CC4O)=O)C2)CC1 C12(C(=O)NC(CC(=O)NC)C)COCC1CN(C(c1nc(=N)cc[nH]1)=O)C2 c1(CCC(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)C)ccncn1 c1(C(=O)OC)ncncc1NC(=O)NC1(c2nn[nH]n2)CCCC1C c1(SCCC(C(=O)O)c2ncco2)ccc(Br)c2c1CCCC2 C1(O)(C(=O)NCC2(C)CCN(C(C)=O)C2)CCCN(C(c2occc2Cl)=O)C1 C(=O)(N=c1[nH]nc(-c2ccc3c(c2)OCO3)s1)Nc1c(CC(C)C)cccc1 N1(Cc2cn(C(C)C)nn2)C(C)CN(C(=O)C(F)C2CCCC2)CC1C Cc1cc(F)ccc1C(=O)NCC1CCN(Cc2nc(Cl)ccc2F)C1 C1(CN(C(=O)CC2(NC(=O)CNC(=O)CCC3CCCC3)CC2)C)CCCO1 N1(C(CCCOCC)=O)CC2(NC(=O)Cc3cc[nH]c3)CCC1CC2 N1(C(C2C(C(C)C)(C(=O)O)C2)=O)CCn2c(cc3c(Cl)cccc23)C1 C1(C(=O)OC)CCCC(CC(C)C)N1CCCc1nc[nH]n1 C1(C(=O)NC2(C(=O)OC)CC2)CCN(C(=O)Cc2cc(C)on2)CC1 C1(COCC(=O)NCC(CN(C(C=C(COC)C)=O)C)O)CCCCO1 c1(CCC)ccc(C(N2CCC(N(CCC)C(c3ccoc3)=O)C2)=O)cc1 CCC(C)(CN=c1nc(N(CCC(O)C(C)(C)C)C)c2ncccc2[nH]1)C(N)=O N1(C(c2ccncc2Cl)C)CC(C)(Cc2ccc(Cl)cc2)CC1=O C1(C(C)(C)CNC(=O)CCn2ccnc2)CCCN1C(=O)CC(O)C1CCCC1 C1(NC(c2c(OC)ccs2)=O)CN(C(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 O(C=CC(=O)N(CCNC(=O)CN1CC(C)C1)CCOC)CC Cc1ccc(NCC(=O)NCCCN(C(C2(c3cncs3)CC2)=O)C2CC2)cc1 C1(C#N)(COC)CN(C(=O)C(CN2CCOCC2)OC)C1 c1(C(=O)NC2C(NC(c3scc(C)c3Cl)=O)C2)c(F)ccc(F)c1O C(=O)(C1=CCC(C)CC1)N1CCC(F)(CNC(C(C)C)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CCOC)(NC(c2ncc(OC)cc2F)=O)CC1 C(CC(O)C(=O)NCCCCCC1CC1)NC(c1scc(C)c1)=O c1(SCC(=O)N(C2CCN(C(C(CC)O)=O)CC2)CCO)ccc(C#N)cc1 c1(CCNC(c2nnnn2CCC2(C)CC2)CCC)cc(CC)no1 N1(C(CNC(C)=O)=O)CCC(OC(CCCOC(C)C)=O)C1C(F)(F)F O=C(CC(C(F)(F)F)NC(c1cnsc1)=O)NCCN1C(=O)CNC1=O C1(COC(c2ccc(Cl)c(Cl)c2)=O)CN(C(c2cccc(Cl)n2)=O)C(=O)CO1 CCC(C(=O)N1CC2CCC(C(N3CCN(C(C)CC)CC3)=O)(C2)C1)C(F)(F)F c1(C(=O)NC2(CNc3ncc(C)cc3[N+](=O)[O-])COC2)oc2c(C)cccc2c1C c1(CC(N2CCN(c3nc(C(F)F)nc(=N)[nH]3)CC2)=O)ccc([N+](=O)[O-])cc1F C12CCC3CN(CC3C1)C2.C1(C(=O)NC(c2nc(C3CC3)no2)C)CCC(C)(C)C1 C1(CNC(CCN(C)C(C2CC(CCC(N)=O)C2)=O)=O)CCCCC1 CCCCCC(O)CC(=O)NC1CC(C)N(C(=O)C(c2ccc(F)cn2)(F)F)C1 c1(C(=O)NC2CCN(C(CCSC)=O)CC2O)ccc2nc(C)c(=O)n(C)c2c1 c1(OC)ccc(C)cc1C(N1CCC(O)C1C(=O)Nc1ncc(O)cc1Cl)=O c1(CC)nonc1C(=O)NCC1(F)CC(NC(c2ccn(C(C)C)n2)=O)C1 N1(C(CCNC(c2nccs2)=O)=O)CCC2(CCCN(C(=O)OCC(F)(F)F)C2)C1 C#Cc1cc(C(=O)NC(CNC(=O)C(C)(C)n2cnnn2)(CC)CC)cc(F)c1 C(=O)(C(=O)CCC(C)C)N1CCC(C(C(=O)NCC(COC)(C)CO)C)CC1 Cn1cnc2cccc(C(=O)NCC(O)CNc3cncc(Cl)n3)c12 C#CC(C)N(C)N1CCN(c2ccccc2NS(=O)(=O)c2ccc(Cl)cc2)CC1 CCC(COC)C(=O)NC(c1ccccc1OC)CNC(c1sccc1SC)=O c1(C(CC)C)cc(C(=O)N(CCCCCNC(c2nsnc2O)=O)CC)on1 C1(C(N(CC(CN(C(=O)CCC2CC2)C)O)C)=O)CC12CCSCC2 c1(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3O)=O)C2)cc2cccnc2[nH]1 C1(NC(=O)CNC(C(c2ccccn2)N(C2CC(=O)C2)C)=O)CC(F)(F)C1 C1(C)(NC(C(C)OCC#C)=O)CCN(C(=O)Cc2ccc(F)c(Br)c2)CC1 C1(C(N2C(C)CC(CNC(=O)C(N)=O)CC2)=O)CN(C)C(=O)CCO1 N1(C(C(COC)C)=O)CCN(C(c2cn(C)nc2Cl)=O)C2CS(=O)(=O)CC12 CC1=NC(C)(C(=O)N(C)CC2CCCCN2C(C2CC(O)C2)=O)N1C N1(C(C2CCC(=O)NC2)=O)CCC2C(C1)CN2C(c1cn[nH]c1)=O N1(C(c2nc(CCC)sc2)=O)CC2CCN(C(c3noc(CC)c3C)=O)C2C1 C12(C#N)CCN(CC1)C(=O)C(=O)NCC2.c1(CN)cc(OC(F)(F)F)ccc1F C(=O)(CCCCC(C)C)N1C2CC(CNC(CC3(COC)CC3)=O)C1CC2 N1(C(C(CCC)C)=O)CC(C)(C)CC1C(=O)NC1(CC(=O)OC(C)C)CC1 C(C(=O)NCC(O)CCNC(=O)C(=O)NC1CC1)(C(C)C)NC(C(C)C)=O CC1(C)C(NC(=O)CC2CCCOC2)CCN1C(=O)C1=CSCS1 c1(C(=O)NCCCNC(C(CC)N2CCCC2=O)=O)cc(NC(C)=O)cnc1O c1(-c2ccc(CN3C(CN)CCCCC3)o2)c[nH]c2ccccc12 C=CC1CN(C(=O)C2=CCSC2)CC1NC(=O)CC1CSCCS1 C(CCC(=O)NC1(CO)CC1)SCC.C12(CC(O)C1)C(=O)N2C C1(C(N2CCC(CC=C)(NC(c3nnc(C(C)C)s3)=O)C2)=O)CCCCN1N=O C12(CNC(C3(NC(c4ccc(=N)[nH]c4)=O)CCSC3)=O)COC(C1)C(O)C2 C1(C(CC)NCC2CCC2c2ccccc2)Cc2ccccc2C1 c1(C(=O)OC2CCC(=O)NC2=O)cccc(S(=O)(=O)N2CCC(O)CC2)c1 N1(C(Cc2cn(C)nn2)=O)CCN(C(c2ccc(OCCF)cc2)=O)C(CO)C1 c1(C(N2CC(C)C(C)(CNC(c3ccc(F)o3)=O)C2)=O)cc2cccn2c(O)n1 CC(CC(F)(F)F)C(=O)NCC1(O)CCCN(C(C2CCCN2CC(F)(F)F)=O)C1 C=CCC(CC(=O)N1CCC2C(C(N)=O)C2C1)NC(=O)CCC1CCOC1 C1(CC(=O)NCCOCCCN(C)C(c2ccco2)=O)CC2CC1C2 c1(CCC)sc(C(N2CC(CNC(C3(C)CCCC3)=O)CC2C)=O)cc1CC O=C(C1=CCC2CCC1N2C(C1CCC2(CC2)C1)=O)NC1C(O)C2CCOC12 c1(C(N2Cc3ccncc3C2)C(=O)NC(C)C)cnc2sc(Br)cn12 C1(C)(NC(Cc2cn(C)nc2Cl)=O)CCCN(C(c2cc3cscc3s2)=O)C1 c1(C(=O)NC(C(=O)NC(CC#C)C(N)=O)COCC)c[nH]c2nccc-2c1 N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CCOC(C)(C)C1CO C(c1csc2ccccc12)=CC(=O)NCCNC(C1(Nc2cccs2)CC=CC1)=O C#CCCCCCC(=O)NCC1(O)CCN(C(=O)Cc2cn3c(n2)CCCC3)C1 c1(CN(CCN)CC)ccc2nonc2c1 N1(C(C2CC(C)N2C(C2CC(C)(C)CO2)=O)=O)CCN(CCO)CC1 c1(CC(N2CCCC(O)(CNC(C(C)=C(C)C)=O)C2)=O)cn(C)c2ccccc12 C1(CNC(C2(COC)CC(C)(C)C2)=O)CC(C)(C)CN1C(C1CC1COC)=O C(=O)(C1SCCc2sccc21)NC(CCCC)CNC(c1cnn(C)c1OC)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CCN2C(=O)CCC2=O)CC1 c1(OC)ncc(Cl)cc1NC(C1(F)CCN(C(C2(c3ccccc3)CC2)=O)C1)=O C1(CC(=O)NC2(CN(C(CCN(C(C)=O)C)=O)C)CC2)CCC(C2CC2)O1 c1(C(=O)NCC2N(C(C3OCCC(=O)C3)=O)CC(F)C2)cc[nH]c2nccc1-2 c1(CC(N2CC(O)(CN(C(CSCC(=O)OC)=O)C)C2)=O)cccc(C)c1 c1(C(=O)NC(C(=O)N(CC=C)CCOC)c2ccoc2)cnn(CCF)c1 C1(C(N(CC(C)C)CC(=O)NCC2(CO)CC3CC3C2)=O)CCCCOCC1 N1(C(C2C(COC)C2)=O)CC(F)(F)CC1CNC(=O)COC1(C)CCC1 C(=O)(CC1=CCOCC1)NC1C(CC)CN(C(=O)C#CC2CC2)CC1 C(CCCCCNC(C1(C)CC1(F)Cl)=O)NC(C=CCOC(C)(C)C)=O N1(S(CC)(=O)=O)CCCC1C(N1CC=CC1CN(C)CCn1cc(C)cn1)=O Cn1cc(Cl)c(C(=O)NCC(CO)NC(c2cccn2C)=O)n1 C(C)(C)(CC(=O)N1CC(CCNC(c2sccc2C2CC2)=O)(OC)C1)OC Cc1[nH]c2ccccc2c1C1=CCN(C(C2CC(C(F)(F)F)OC2=O)=O)CC1 N1(C(CCOCC#C)=O)CC(CNC(=O)CC2CC(F)(F)C2)N2CCC1C2 C1(C)(CNC(C2C(C)=C2)=O)CCCN1C(C1CC(C)OC1C)=O c1(-c2n(CCCC)nc(C(C)OC)n2)nn(-c2ccccc2)cc1[N+](=O)[O-] C#CCC(C)C(=O)NC(C)CNC(=O)COc1ccc(C(C)C)cc1 N1(C(c2c(C)nn(CCO)c2)=O)CCC2(C)CN(C(C3CCC(F)CC3)=O)CC12 Cc1ccc(C=CC(=O)NC2CC(F)(CNC(c3ccsn3)=O)C2)c(C)c1 C1(NC(c2cc(C)no2)=O)CCOCC1NC(c1cc(C)c(Br)s1)=O C1(CC=C)(NC(C2CCOCC2)=O)CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 C(=O)(CCCCC(=O)N1CC2(CCC(NC(C3CCCC3)=O)C2)C1)OC N1(C(CC2N(C(C3(C)CC4(CC4)C3)=O)C3C2CCC3)=O)CCC2CCC(C2)C1 c1(N2CCCC(N3C(=O)NCC3)C2)nc(=NCCC(F)F)[nH]c2c1CCCCC2 c1(C(=O)NC2CC(C(=O)NCc3ccc(Cl)nc3)C2)ccccc1C1CC1 N1(C(C=CC2N(C)CCC2)=O)CCCC(C)(C)C1CNC(c1cccc(N)n1)=O C1(COC)CN(C(=O)C(C(C)C)n2cncn2)CCN1C(c1ccco1)=O c1(C(=O)NCC2CCN2C(C2CC3C=CC2C3)=O)cc(F)ccc1Br C1(C(N2CC(CC)N(C(=O)CSC)CC2)=O)Cc2ccncc2C1 c1(OC)ccc(C)cc1C(=O)NC1CN(C(=O)C(F)(F)C(C)O)CCC1CO C1(CC)(CNC(C2CC2(C)C)=O)CN(C(=O)CNC(=O)C(c2cccnc2)O)C1 N1(C(CC(C=C)(C)C)=O)CCC2(CNC(c3coc(Cl)c3)=O)CCCCC12 C=CCCC(C)(C)C(=O)N1CCCC(NC(=O)Cc2ccc(CC(C)C)cc2)C1 Cn1cc(C(=O)OCCc2ccccn2)c(C2CCCO2)n1 S(=O)(=O)(c1nc2c(s1)CC(=O)CC2)Nc1cccc(C2C(C)(C)C2(C)C)c1 Cc1cc(C(N2CCCC(C(=O)N(C(C(N)=O)C3CC3)C)C2)=O)ncc1N C1(OCC)COCCC1CC(N1CCCC1CN(C(=O)C=CBr)C)=O C(C(=O)NC1(C)CC(NC(C2(CNC(C)=O)CCCC2)=O)C1)(C(C)C)NC(C)=O c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C2(C(=O)NCCONC(C3CC4(C3)CC43CC3)=O)CC2)c(F)cccc1F c1(C(N2CC(C=C)C(NC(c3cnc(C)[nH]3)=O)C2)=O)sc2ccccc2c1Cl C1(CNC(=O)Cc2cncs2)C=CC(NC(=O)CC2(CO)CCCC2)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnc2S)=O)C1)N1C(C)C(C)(C)CC1 CC(C)C(CCN(C(=O)C(C)(C)c1ncco1)C)NC(=O)CO C(=O)(C(CSC)OC)N(CCN(C(=O)C(C)CC1CCC1)CC)CC Cc1cc(C)c(C(=O)NCC(O)CN(C(=O)C(c2cccnc2)O)C)s1 C1(C(=O)NCC(CC(C)C)NC(c2c(C)nccc2)=O)CC2CCCCN2C1 c1(C(=O)NC2CCN(C(C(CC(C)C)N(C)C)=O)C2)cccc2c1OCC2(C)C c1(C(=O)NC(CNC(C2CC(CC(F)(F)F)C2)=O)C2CCC2)ccc(Cl)[nH]1 CC1(C)CCOC1C(=O)NCC1CC(O)CN1C(C1CCCOCC1)=O c1(CC)ncc(C(=O)NC(C2CCN(C(c3cc(OC)cs3)=O)C2)C)[nH]1 c1(C(N2CCN(C(C3CC(OCC)C3)=O)CC2)=O)ccc(Cl)nc1Cl Cc1cnc2c(cnn2CC(=O)NC2CCC(C)N(c3ncc(Br)cn3)C2)c1 c1(C(N2CC(NC(C3CCSC3)=O)CC3(C2)CC3)=O)cc2cc(Cl)cnc2o1 c1(OC)cc(C)nc(NC(C2CC(NCc3cccn3C)C2)=O)n1 N(C(=NCCC(C)C)NCC1CCC2(COC2)O1)CC(c1ccc(Cl)cc1)CC Cc1n[nH]c(C)c1CCC(N1CCC(C(C)NC(=O)Cc2ccc(F)cn2)C1)=O c1(C(=O)NCC2(F)CCN(C(C(C(C)C)C#N)=O)C2)ccsc1S(N)(=O)=O C1(N(C(=O)C(=O)NC(C)C)CC)CCCN(C(=O)C(c2cn(C)nc2C)C)CC1 Cc1cc(C(=O)N(CC(C)CNC(=O)C(O)C(F)(F)F)C)cc(C)c1F CN(C)N=Nc1ccccc1C(N1CCCN(C(=O)C(C)(C)CF)CC1CO)=O C1(c2cccc(OC)c2)CN(C(=O)COCCF)CCN1C(C1(C)C=CCC1)=O c1(C(N2C(CNC(CSCCC(C)C)=O)C=CC2)=O)cc(C(C)(C)C)ccc1O C1(N(C)C(c2cc(Cl)no2)=O)CCCN(C(c2cnc(O)nc2O)=O)CC1 c1(C(=O)NCC(C)(C)CNC(C2CC2C2CCC2)=O)c(Br)ccc2n[nH]cc12 c1(C(N(CC(C)N(C)C(C2CC(F)C(=O)N2)=O)C)=O)ncc2c(F)cccn12 C1(CC(=O)NCCN(c2nccc(-n3ccnc3)n2)CCC)CCC2CC2C1 C1(C(=O)NCCNC(Cc2ccn(C(C)C)n2)=O)COCCN1CC(F)(F)F N1(C(C2CC(CNC(C3COCC(C)O3)=O)OC2)=O)CCC(F)(F)C(O)C1 c1(CCC)ncc(C(N2CC(O)(CNC(c3coc(C)c3)=O)C2)=O)s1 C1(C(=O)NCC(CN(C(=O)Cn2nnnc2-c2ccccc2)C)O)OCC1(C)C CC(C)CC(C)CC(=O)NCCC1(O)CN(C(=O)C(C(C)C)N(C)C)C1 c1(CN2CC3CCC2C3)ccncc1Cl.C12CC1C(=O)N(C1CC1)C2=O n1(CC(=O)N(CC(C)NC(=O)COCC2CCOC2)CC)[nH]cnc1=N N1(C(c2c(OC)n(C)nc2)=O)CCC2CCCC(C1)N2C(C1CSCCS1)=O N1(C(=O)C2=NOCC2)CC2CCC(NC(=O)C(F)(F)CO)CC2C1 C=C=CC(C)C(=O)N1CC(F)CC1C(=O)N(C)OC C12(CNC(C3N(C(C4C(C)C4C)=O)CCOC3)=O)CCN(CC1)CC2 C12(CNC(C=CC)=O)CC1CN(C(=O)OC(C)(C)C)C2.c12ocnc1NC(=O)C2 Cc1cc(=NCC(C(C)C)N2CCC(C)CC2)[nH]c(N2CC(C)C(F)(F)C2)n1 C1(NC(CC2(COC)C=CCC2)=O)CC2CC(NC(=O)CC(=O)N(C)C)C1C2 C(=O)(C(C)(F)C(C)(C)F)NC1CC(F)(CNC(c2nc(C)nn2C)=O)C1 c1(CNCC2(C(N3C(C)C(=O)N(C)CC3)=O)CC2)cc(F)c(F)c(Cl)c1F C1(CCC)(NC(=O)COCC2CCOC2)CCN(C(c2cnc(OC)s2)=O)CC1 C1(C(=O)NCC(C)(C)CCO)(COC)CCCCCC1 c1(C(N(CC(CC)NC(C23CC(CO2)C3)=O)CC)=O)csc(C(C)C)n1 CCCC(C)(CC)C(=O)N1CC=CC(NC(=O)Cc2ccc(OC(F)F)cc2)C1 C1(C(=O)NCC=C)CC(F)(F)CN1Cc1ccc(C2CC2)cc1 N1(CCCNC(N=c2ccn(CC(=O)NCC)[nH]2)=O)Cc2ccccc2C1=O C1(CC(=O)NCC(CC=C)NC(c2[nH]cc3c2CCC3)=O)CCC(C)(C)CO1 C1(NC(N(C(C(C)C)CO)C(C)C)=O)COc2cccc(Br)c2C1 c1(C(=O)NCC2(C)CCC(NC(=O)CC3CCC3)C2)cc(Cl)ncc1O c1(Oc2nccc(CNC(C=CC(C)=O)=O)c2)ccc(C)cc1Br N1(C(C2=C(C)CCC2)=O)CCC2(CCC2CNC(C2CCOCC2(C)C)=O)CC1 N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC(C2CCN(C(C3CC=CCO3)=O)C2)CC1 C1(Cc2ccccc2)CCCC(Nc2nnc(C3(N)CCC3)s2)C1 N1(C(C(CCCC)(C)F)=O)Cc2n[nH]cc2C1C(=O)N1CCC(O)CC1 N1(C(C(c2cc(C)oc2C)C)=O)CC2CC1CN2C(c1ncoc1C(F)(F)F)=O N1(C(C(CCF)NC(c2nn(C)c(Cl)c2)=O)=O)CCOCC(C)(C)C1 c1(OC)nc(=NCC2CN(C(c3nc(O)sc3C)=O)CCCO2)[nH]c2[nH]cnc12 c1(CC(=O)NCCN(C(=O)C2=CCOCC2)C2CC2)cc2ccccc2o1 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(C2CC3OC2C2CC32)=O)C2CCCC12 C(C1CCC(C)CC1)=C(C)C(N1CC(O)(C(C)NC(c2ncoc2C)=O)C1)=O CC1CC2CN(C(C3CSCCN3C(c3cnc(O)o3)=O)=O)CCN2C1 c1(-c2scc(NCC(C3CCCC3)N)n2)cccc(F)c1 c1(CN(CCC(=O)O)C(=O)C(C2(O)CCCC2)F)c(F)cc(OC(F)F)cc1F c1(C(=O)NC(CCCCNC(C(CC)N(C)C)=O)C)nn(C)c(C)c1Br CCCCCC(=O)NCC(C)(C1CCC1)NC(=O)CC1CCC=CCC1 n1(CC)nccc1C=CC(=O)NC(C1(O)CN(C(C2CC(C)OC2C)=O)C1)C c1(C(N(C2CCN(C(c3nncs3)=O)C2)CCC)=O)cc(F)cc2cnccc12 C1(CC(=O)NC2CCN(CCCn3cnnc3)CC2)CC2CCC1C2 CC1C2CN(C(=O)C(C)(C3CCCO3)C3CC3(F)F)CC12.C1(CC=S)CCC1 CC1CC(C(=O)NC(C)(C)CCNC(c2csc(=N)[nH]2)=O)CO1 C1(C(N2CCC(F)(CNC(CC3(OCC)CC3)=O)C2)=O)C2CCC(F)(F)C12 c1(CNC(C2=CCCC2C)=O)nn(C)c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 C(C(CO)C(F)(F)F)NC(C1N(C(c2c(CNC(N)=O)cco2)=O)CC=C1)=O C(=O)(C1=NOC2(CCC2)C1)NC1C(OC)CN(C(C2CCCCC23CCC3)=O)C1 Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CN2C(=O)CCC2=O)cc(N)c1 CC1CCN(C(c2cccnc2)=O)CC1NC(C1CNC(=O)N1)=O N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2CC3CCC3C2)=O)CC(C)(C)C1 C1(CC)(NC(C23CSC(C2)C3)=O)CCN(C(=O)C(C(C)C)n2ccc(C)n2)CC1 C1(C#N)(C(N2CCC(C)(C(=O)NCC(=O)NC(C)(C)C)C2)=O)CC2CC2C1 N1(c2ccnc(OC)n2)CC2CCCN(C(c3cc(Cl)ccc3F)=O)C2C1 C=CCC(C(=O)NC1COC(C)(C)C1)NC(C1CC(=O)C1)=O c1(C(=O)NCC(C2(O)CN(C(CCOC(C)C)=O)C2)(C)C)cscc1C#N C(=O)(C(C)CCCC(C)C)N1CCC(CNC(C(CC2CCC2)OC)=O)C1(C)C CCC(CCOC)C(=O)NCCOCC(=O)NCc1cc(C)sc1C c1(C(N2CCC(C(C(=O)N(C)CCOCCO)(C)C)C2)=O)cccc2cc[nH]c12 C(C(=O)NCC1CCC1)(N(C(=O)COC1(C)CCC1)C)C1CC1.C1CCC1 C1(NC(C=CC(C)C)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 CN1CCOCC1C(N1CC(N(C)C(c2ccc(C3CCCOC3)cc2)=O)C1)=O C(CC1CCC1)(C(=O)N1CC(O)(CCNC(=O)CCc2cc[nH]n2)C1)NC(C)=O CC(CCl)CS(=O)(=O)NC1CCCC2OCCC12 c1(N2CCCC(CCNC(C(C)(C)CF)=O)CC2)nccn2nnnc12 Cc1ccccc1-n1ncc(C(=O)NCC2(CNC(C3CC3F)=O)CCCC2)n1 c1(C2(C)CC2)cccc(CNC(=O)NCC2CC2CC(=O)O)c1 C(CO)(C(=O)NCCn1cc(CNC(=O)C(C)O)nn1)OC c1(OCC(C)C)ccc(NC(=O)C2=CCOC2)cc1.C12(CC1)C(=O)OCC2C c1(OC)ccc(C(N2CCC(O)C(C(N3CC(OC)C(OC)C3)=O)C2)=O)cc1Br N(C1CCCc2ccccc21)N1CCN(C(C2CC(C(=O)OC)OCC2)=O)CC1 c1(CN2CC(C(C)NC(=O)NC(C)(C)C)OCC2)cc(C#N)n(C)c1 C(CS(=O)(=O)CC)NC(c1n(CC=C)nnn1)(C)CC1CCCOC1 Cc1cncc(C(=O)NC2CCCN(C(=O)Cc3ccnn3C3CCC3)C2C)c1Cl n1(C(C)C(=O)NCC2CCC2NC(C2(C)CC2)=O)ccc(C(F)(F)F)n1 CC(CC(=O)NCC1CCCC1NC(c1ncccc1N(C)C)=O)C(C)(C)C N1(C(COc2cn(C)nc2)=O)CCC(O)C(NC(=O)C#CC2CCC2)C1 Cc1ncc(Br)cc1C(=O)NC(CNC(=O)CC1(C)CCCO1)CO c1(COC(C23C(CN(Cc4ccc(COC(C)=O)o4)C2)C3)=O)cc(Br)ncc1Cl c1(C(N(CC(C)(C)CNC(c2cocn2)=O)C)=O)nc2ccc(CO)cn2c1N c1(OC)cccc2c1OCC2NC(=O)C(C)(c1ccccc1)N(C)C CC12CN(C1)N2CCC1CCCCN1.c1(CCCC2CCOCC2)cccnc1 N1(C(CC(C=C)C)=O)CC2(CC2)CC1C(=O)NCc1ccncc1C N1(C(C2OCCC(NC(CCCN(C(C)C)C)=O)C2)=O)CC2(CCOC(=O)N2)C1 Cc1ccc2oc(C(N3CCCC(CN(C(=O)C=CC(N)=O)C)C3)=O)cc2c1 c1(C(N(CCCNC(C(CC)COC)=O)C)=O)cc2cc(Br)cn2c(O)n1 c1(C(N2C(C(=O)Nc3c(CC)cccn3)CC3CC32)=O)cccc(C(F)F)c1F C1(C)(C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)CCCO1 CC(C)C(C)C(=O)NC1CCC(CCNC(C2(CO)CCOCC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)C1CC2(C(N(C(C)CN)C)=O)C(C1)C2C Cc1cc(C(=O)NC(C)(CNC(C2CC(C)(C)CN2C)=O)C2CC2)nc(O)n1 CCS(=O)(=O)CCNC(C1CCC(CNC(=O)C(CO)NC(N)=O)O1)=O CC(C)CC(C(=O)O)N1C2CC(F)(C2)C1=O.CSC.N(C)C CCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2CSC2)CC1C c1(CN(C)C)cn(C2COCC2NC(=O)C(N)COC(C)(C)C)nn1 C1(C(=O)NCC2CC(O)(CNC(c3c(COC)cco3)=O)C2)CC(=O)N(C)C1 N1(C(C(CCCC)NC(=O)CN(C)CCC)=O)CCOC(C2(C)N=N2)C1 c1(OC)ccc(-c2ccc(CNC(c3cc(Cl)cnc3Br)=O)nc2)c(F)n1 N1(C(c2cc(C)oc2)=O)CC(NC(c2ccccc2CC(C)(C)C)=O)CC1C C(N=c1cc(NCCN(C2CC2)CC2CC2)nc[nH]1)C1OCC(C)(C)C1 N1(C(C2(C#N)CCC2)=O)CC2C=CC1C(C(=O)NCC1CC3(CCC3)C1)C2 C(=O)(CC(C)(C)NC(=O)CSc1ccc(CN)cc1)NC C1(NC(=O)CNC(C2CCCC2F)=O)CCn2ncnc2C1 CN1CCC(O)C(NC(C2CN(C)CCN2C(c2ccc(C#N)n2C)=O)=O)C1 C1(NC(C2C(C)(C)CC2)=O)CCCN(CCNC(=O)C2=CCSC2)C1 c1(C(=O)NCCCNC(COCC=C)=O)cc(F)cc(C)c1N c1(C(=O)NCC2C(NC(C(CCC)N(C)C)=O)C2)cc(C)c(CC)nc1O c1(C(N2CC(F)(C(N3CCC(O)C3)=O)C2)=O)cccc(Cn2ccnc2)c1 C(C(CC(=O)OC)C(F)(F)F)NC(c1n(CC=C)nnn1)(C)CC1CCCC1 N1(C(c2ccc(C)s2)=O)C(C(=O)NC2CC=CC2)C2CC(F)C1C2 c1(CN(C(C2CCN2C(=O)CC2CCOC2)=O)CC)occc1C S(=O)(=O)(c1ccc(Br)cc1Cl)N.c1(-c2ccc(C)cc2)ncnc([SH2]c2nncs2)c1N C(=O)(CC(CN(C)C)C(F)F)NCC1N(C(CCCOC(C)C)=O)CC(C)(C)C1 CCC(C)C(C(=O)N1CC(CSC)(OC)C1)NC(=O)CN(C)CCOC N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)N(C(c1cnn(CC)c1Br)=O)C2 C(Cn1cncn1)(C(=O)N1CCCCO1)NC(C1CN(C)C(=O)C1)=O C(CCCCC(=O)NC(C)(CNC(c1c(C)c[nH]c1CC(N)=O)=O)CO)SC c1(C(=O)OCC)ccnc(NC2(c3ccccc3)CCN(C(=O)CO)C2)c1[N+](=O)[O-] CCCC(C(=O)NCC1(OC)CCOC1)NC(N)=O.c12ccsc1C(=O)NC2 c1(C(=O)NC2(CO)CN(C(c3occ(C(N)=O)c3)=O)C2)csc2c1CCCC2 CCCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NNCCC.CC CCC(C)(C)CC(=O)NC1CCCC(NC(c2cnn(C3CC3)c2C)=O)C1 Cc1cccc2c(CC(=O)NC3CCC(NC(=O)C(C)(C)C(F)F)C3)c[nH]c12 c1(NC(C#C)=O)cccc(C(F)(F)F)c1Br.C12(C)CCCN1C(=O)OC2 C12(NC(c3cncc(C(C)=O)c3)=O)CCN(C(C3CCSCC3)=O)CC1C2 C1(CN(C(c2ccc(C#N)s2)=O)CC)CCN(C(C2CCC(F)C2)=O)CC1 C1(C(N2CC(NC(C)=O)C2)=O)(CC)CCN(C(C2CC=CCC2)=O)C1 C(=O)(CC(C)C)NC(CCN(CCC(=O)N(CCC1CC1)CC)CCCOC)=O Cc1nn(CC(=O)NCC2CCN(C(c3ncncc3Cl)=O)C2)c(=O)n1C N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(C2(O)CCC2)=O)C1C C#Cc1cccc(C(C(=O)NCCC)N(C2CCCCCC2)CC(C)C)n1 Cc1c(C(N2CCC(NC(=O)C=Cc3nnc(C(C)C)o3)CC2)=O)ccn1C C#CC1(N(C)C)CN(C(C2(C(C)NC(C3C=C(C)CS3)=O)CC2)=O)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)CC2CC)nnc2ccccc2n1 C1(C(N2CC(CS(N)(=O)=O)C2)C)CCOC1=O c1(C(=O)C(N2CCN(C(C3CCCO3)=O)C(CO)C2)=O)ccc(F)c(F)c1F Cc1ccc(C(=O)NCC2(CNC(C3CCN(c4ncccn4)C3)=O)CC2)nc1 CCCC(C(=O)OC)C(=O)N1CCC(N(C(c2scnc2C)=O)CC)C1 c1(C(C(N)=O)N(CC(Cc2ccccc2)OC)C(C)C)ccc(Cl)cc1 CC1(C(=O)NCCCCCCCc2ccccc2)CCCN(C(N)=O)C1 Nc1c(C(=O)NC(CNC(=O)C=CCN2CCCC2)CO)cccc1Br c1(C(CC)NC(=O)NCc2cc(Br)ccc2OC)cc2ccccc2s1 N1(C(C(CO)NC(N)=O)=O)CC2CC(NC(C3(O)CCSC3)=O)C2C1 S(=O)(=O)(c1ccc2c(c1)CCC2)Nc1ncc(-c2ccc(C)cc2)cc1C C(CN=c1cc(NCc2nnc(C)o2)nc(C(C)C)[nH]1)NC(=O)NCC c1(CNC2CCC(C)SC2)ncnc2c1CCC2 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(c2cc(C(F)F)on2)=O)C(C)C1 CC1CC(C(N2CCC(CF)(NC(c3ccnc(N(C)C)n3)=O)C2)=O)CC(=O)N1 c1(C(N(CC(C)NC(=O)CP(C)(C)=O)C)=O)ccc(-c2cccs2)nc1O C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(c2ncc(C)c(C)c2)=O)CC1 N1(Cc2nc(C)on2)CCCC1C1CCCCN1C(c1ccnn1CC(C)C)=O c1(NC2CC3N(C)C(CC3)C2)ccc(S(=O)(=O)N(C2(C)CCOC2)C)cn1 O=C1CC(C(N2CCC2CNC(C2(F)CCCC2)=O)=O)CC(=O)N1 c1(C(=O)NCC(C)NC(c2cc(C3(C)CC3)n[nH]2)=O)ncn2c1CCCC2 N1(C(C(C)OCC=C)=O)CC(C)(C(=O)N(CC(F)F)C)CC1(C)C Cc1[nH]c2ccccc2c1C(=O)N(C)CCNC(c1cncc(Cl)c1Cl)=O C1(OCC(=O)NCC(C)C)CC(CNCC(c2ccc(F)cc2)O)C1(C)C C1(NC(C2C(C)N(C)CC2)=O)CC(F)CN(C(C2(F)CC=CC2)=O)C1 c1(C(C)C)nnnn1CC(N1CCCC1CNC(C1COC1)=O)=O N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CN(C(=O)COCC(C)(C)C)CC2C1 c1(C(N2CC(C)OC(CCNC(c3ccc(F)s3)=O)C2)=O)n[nH]c2c1CSCC2 c1(C(=O)NCC(CC)NC(=O)C(C)(F)C(C)(C)F)cc(OC)c(OC)cc1C Fc1cccc2nc(N3CCCC3c3ncc(-c4ccccc4)[nH]3)oc12 c1(C(N2CC3C(NC(CCC(N)=O)=O)C3C2)=O)ccc2c(c1)CCCC(=O)N2 N1(C(C=C(C)C)=O)CCOCC1C(C)NC(=O)Cc1ccc(C2CCC2)cc1 c1(C(N2CC(NC(=O)Cc3nnc(O)s3)C(F)C2)=O)ccc(F)c(C(F)(F)F)c1 CC(C)C(F)(CNC(c1cncnc1)=O)C(=O)N1CCC2(CC(F)C2)C1 c1(OC)ncc(Br)c(N(CCCCN(C)C(C2CCCC(O)C2)=O)C)n1 C(CC(C(=O)N(C1(NC(=O)Cn2nnc(-c3ccsc3)n2)CC1)C)OC)N(C)C CC1(CCO)CCN1C(c1n[nH]cc1CNC(=O)Cn1ncnn1)=O c1(C(=O)NCC2CC(COC)CN2C(=O)COC(C)=O)cc(=O)n(C)cn1 c1(C(N2CC(CNC(c3cc[nH]n3)=O)C3C2C3)=O)cc2ccc(Cl)c(F)c2o1 c1(CN2C(CCC(=O)Nc3nccnc3Cl)CCC2)ccc(O)c2ncccc12 c1(C(=O)NC(C)CN(C(=O)C(C)C(C)O)C)ccc([N+](=O)[O-])[nH]1 c1(OCC(=O)OC(C)C(=O)Nc2ccc(N)cc2)c(Cl)cccc1Cl N1(C(CN(CCC)C)=O)CC2CCC1C2NC(c1cc(C(=O)OC)on1)=O N1(C(=O)CCCCC(F)F)CCC2(CCN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 C1(C(C)NC(c2coc(CNC(=O)CC3CCC4CC34)n2)=O)CC(O)C(O)C1 c1(NC(C2C(NC(C(CC)NC(N)=O)=O)CCO2)=O)cnc(F)nc1 Cc1c(C(=O)OCCCCOCCOC(=O)CC23COCC(C2)C3)cccc1C#N C#Cc1ccc(OC)c(C(=O)NCC2(C)CCC(NC(=O)Cc3cnsc3)C2)c1 N1(C(C2CCCC(F)(F)C2)C)CC2C3CCC(C3)C2(C)C1 C12(C(N(C)CCNC(=O)COCc3ccncc3)=O)CC3CCC(CC(C3)C1)C2 C1(C(N(CCN(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)C)C)=O)OC2CCCCC2C1C N1(C(C(=O)NCCC#N)C2C(C)C2)CCCC(NC(=O)NS(C)(=O)=O)C1 C1(C(=O)NC2(CNC(c3c(C)c(N)ccc3)=O)CCCC2)CCCCC(C)(C)C1 C(=O)(C1CC(C)(C)C1)N(CCC)CCNC(c1ccccc1)=O CCCC(C)(C)CC(=O)N1CCC(=CCNC(=O)C(=C2CCCCC2)F)CC1 CCCC(CC)CC(=O)NCCC1CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1 CC1(C)CCN(C(c2c(N)cccc2Cl)=O)CC1NC(c1cccnc1)=O CC1CCC(NC(c2cnn3ccsc23)=O)CN1C(=O)CC12CC(C1)C2 c1(OC(CC)CNC(C2(C)CCSCC2)=O)cccc(C)c1 c1(C(C)=O)c(NC(c2cc(OCC(F)(F)F)nc(Cl)c2)=O)cccc1C C(=O)(C1CCOc2ccccc21)NCC1C(NC(CCCN=[N+]=[N-])=O)CCCC1 C(CN(C)C(C1CN(CC(C)C)C1)=O)(CO)(CO)NC(COCCC=C)=O CCCCC(=O)NCC1(O)CC(C(N2CCOCC2)=O)C1 c1(C(=O)NCCC2(O)CCCN(C(CN(C)C)=O)C2)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(NNC(=O)Cc1ccccc1)NCC(C(C)c1ccccc1)O C1(C(=O)NC(CNC(CCCC)=O)CC)COCC(=O)N1C(C)C CCC(C)(C(=O)NCc1ccc(C(N2CCC2)=O)nc1)C(C)=O C(C(=O)NC(c1cnc[nH]1)C)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O N1(C(c2c(OC)ccs2)=O)CCCC2CN(C(c3cnc(C)cn3)=O)CC12 N1(C(c2c(CC)nn[nH]2)=O)CCC(CNC(C2(C#N)CC=CC2)=O)C(CC)C1 O=C(CC1COc2cc(O)ccc21)N1CCC(N(CCO)C(C2CC(O)C2)=O)C1 N1(C(CCN(C(=O)CC(C)(C)CCC)CC#C)=O)CC2(CCC2)CC1C c1(C(=O)NCC2(NC(C(C(C)C)c3ccc(F)cc3)=O)CC2)ccccc1C#N C(=O)(CC(C)CNC(=O)CN1CCN(C(=O)Cc2nocc2C)CC1)NC Cc1ncc(CC(=O)N(CCN(C)C(C2(C3CC3)CC2)=O)C(C)C)o1 c1(OC)ncc(C(=O)NCCC2CN(C(C3(C(F)F)CC3)=O)CCO2)cn1 C(=O)(CCCC(C)(F)F)N(C)CC1(NC(C(C)CC=Cc2ccccc2)=O)CC1 C1(NC(c2cnc(C)o2)=O)CCC(C)N(C(c2cc(C(N)=O)cc(F)c2)=O)C1 N1(C(C2C(C)CCS2)=O)C2CCC1CN(C(C1(c3ccsc3)CC1)=O)C2 C(=O)(CC1OCc2cc(Cl)ccc21)N1CCCC(CC)(NC(c2cnsc2)=O)C1 c1(C(=O)NCCN(C(C(C=CCCC)O)=O)Cc2ccccc2)ccncc1O N1(C(CCCCOCCOCCOC)=O)C(c2cn(C(C)CO)nn2)COC1(C)C C1(NC(Cc2ccc(C)s2)=O)CCCN(C(c2cn(C(C)C)nc2C2CC2)=O)CC1 N1(C(C(C=C)(C)CCOC)=O)CCCC2(CCCN2C(=O)Cc2coc(C)n2)C1 c1(C(=O)NC(C)CCCNC(C2CN(C)C(=O)N2)=O)ccc2cn(C)nc2c1 c1(C(N2CCN(C(c3nccc(C)c3O)=O)C(C)C2)=O)cccc2ccnn12 n1(CCC(N2CC(COC)(NC(=O)CC3CCCOC3)C2)=O)nc(C)nc1C C1(COC)CN(C(c2ccc(Cl)nc2N)=O)CCN1C(C1CNC(=O)N1)=O CC(C)C(F)(F)CC(=O)N1CC2CCC1C2NC(c1ccc(CN(C)C)nc1)=O N1(C(C2(CC#C)CCOC2)=O)CCC(CNC(=O)Cn2ccnn2)C(F)(F)CC1 C1(CNC(C2CC3(CC(=C)C3)C2)=O)CC2CCC(C1)N2C(c1scnc1C)=O CCC(C)CC(=O)NCCOC1CCN(C(=O)C(C)CC2CCCCC2)CC1 n1(CC(=O)NCC=C(C)Cl)cc(C(C2CCOCC2)C)nn1 CC(C)C(C)CC(=O)N1CCCN(C(=O)CCC2CCN(C)CC2)CC1 C1(C(=O)NCC(C)CO)CCCCN1C(=O)CN(C)C=O.c1(N)ccccc1 CN1CCN(C(c2coc(C#N)c2)=O)C(CNC(c2n[nH]cc2Br)=O)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2)=O)cnc2n1CCS2 C1(CNC(CCCCOC)=O)C(C2CC2)CCN1C(=O)CC(C)(C)OC(C)=O CC(C)CC(=O)C(=O)N(C1CCN(C(=O)C(C)C2CCCO2)CC1)C C1(CNC(c2c(OCC)nccc2C)=O)CC12CCN(C(C1CCCO1)=O)CC2 c1(C(N2CCOC(CCO)C2)C(=O)NCCC)ccc2ccc(Br)cc2c1 C(S(=O)(=O)C(F)F)C1N(C(C2(n3cc(CN)nn3)CC2)=O)CC1.N#CCCCN n1(CCCC)ncc(C(=O)NCC2CCN2C(=O)CC(C)O)c1CC N1(C(C2C(C)N(C(=O)COCCCN(C)C)CC2)=O)CCC2(CC(N(C)C)C2)C1 C(C)(CNC(=O)Cc1ccnn1C)(CC(C)C)NC(C(C=CCCC)O)=O CC(CCCc1ccccc1)C(=O)N1CC(NC(C2CC=CC2)=O)C(C(F)F)C1 C=C=CCC(=O)N1CCC(C(F)C(=O)N(C)CC2(O)CCC2)C1 c1(C(=O)NC2CC(CCNC(C3C(C=C)OCC3)=O)C2)ccc(C(C)=O)cc1C C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CSCc2ccccc2)C(C)(C)C1 CCC(C)(C#N)C(=O)NC(CNC(c1cc(O)cc(F)c1)=O)C(C)(C)C N1(C(C2(CC)COC2)=O)CCC2(CC1)CN(C(=O)CC1CCCN1CC)CCO2 c1(C(N2CCCC(CNC(C3C(C)CC(C)O3)=O)C2)=O)cnn2c1C(=O)NCC2 CCCCCC(O)CC(=O)NCCN1CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 CC(=O)CC(C)C(=O)NC1CC2CC1CN2C(=O)CSc1ccccn1 C(c1cn(C)nn1)=C(C(=O)NC(C1(O)CCN(C(c2ccc(=N)[nH]n2)=O)C1)C)F C1(CNC(CCCSCC)=O)CCCN(C(c2ccc(CC)s2)=O)C1 N#CC1CCCC(C(=O)NCCCCCCNC(=O)Cc2ccc(CO)cc2)C1 C12(C(=O)NC3C(C)CCN(C(C4CCOC4)=O)C3)CC3CC(C)(C1)CC(C)(C3)C2 C(CC(F)F)(C(=O)N1CCC(O)(CO)C1)NC(c1nc(=N)[nH]cc1)=O C1(C)(CNC(CNC(=O)OCC)=O)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(n2cc(C(C)OCC3CCOC3)nn2)CN(C(c2cn(C)nn2)=O)CC1C c1(C(N2CC(n3cc(NC(N)=O)nn3)C2)C)nnc2ccccn12 S(=O)(=O)(c1c(Br)cc(F)c(Cl)c1F)SCC(CC)N(CC(=O)O)C c1(OC)cccc2c1OCC(C(=O)N1CC=CC(NC(=O)C(F)C(F)(F)F)C1)=C2 N1(C(c2cc(C)c(O)nc2)=O)CCC(C2CC2)C1CNC(=O)CN(C)S(N)(=O)=O C1(NC(CC2CC(C)C2)=O)CCCC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 O=C1CCC(CNC(=O)CN2CCC(n3ccnc3)C2)C1 C(=O)(C1CCCc2nn[nH]c21)NC1CC(NC(c2c(CC)nns2)=O)C1 c1(CNC(c2nn(C)cc2Br)c2n(CCC)nnn2)c(Cl)n[nH]c1C c1(C(N2CCC(O)(CCNC(CC(C)(C)C3CC3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(=O)NCCOCC(=O)NC)C(C)OCCN1C(C1CC2(C1)CC21CC1)=O C(=O)(C(=O)C(C)(C)CC)N1CC(CCC=C)(C(=O)NC2CCCN(C)C2)C1 N1(C(CCC)C(=O)NCc2cccc3ccccc23)Cc2ccccc2CCC1C N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCCN2C(c2cccc(O)c2)=O)C1 c1(CNc2c3cc(C)[nH]c3ccc2)nccc(=NCCC(C)N(C)C)[nH]1 C1(C(C(=O)NCCCCNC(=O)C(C)c2ccco2)OCC)CC(F)(F)C1 C1(C(=O)NCCCN(CCCNC(c2c[nH]nc2C(F)(F)F)=O)C)CNC(=O)N1 N1(CCN(C)C(=O)NC2ON=C(C(C)C)C2)CCc2ccccc21 c1(C(N2C(C)C(C)C2)=O)cc2oc(Br)cc2[nH]1 c1(CC(N2C(CCNC(C=NOC)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 c1(OC2(C(=O)NCC(=O)OCC)CCN(C(=O)CCOC)C2)cccc(CC)c1 CCCC(C(=O)N(C(C(=O)N1CCOCC1)C(C)CC)C)C(C)C C1(O)(C(=O)NCCF)CCN(C(c2ccc(-c3ccccc3)cc2)=O)C1 c1(CCC)sc(C(N2CCOC(CNC(=O)CCc3cccs3)C2)=O)cc1CC c1(C(C(N2CC(CNC(C(C)CO)=O)C2)=O)C)cccc(Br)c1 c1(C(N2C(C(=O)NCc3ccccc3F)CC(=O)C2)=O)cnn2c1OCC2 CC(C)CC(CNC(C1(c2cc[nH]n2)CCC1)=O)NC(C1CC(F)C1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(C(CCC)OC)=O)C(CC)C1 C(C(C(C)C)C(C)C)N(C(CCC(=O)OC)=O)CCN C12(C(=O)NC3(CCNC(=O)Cn4cc(Cl)cn4)CCCC3)CCCCC1OCC2 CCCC(O)CC(=O)NCC1CCCCCN1C(c1cnn(C(C)C)c1N)=O c1(C(N2CC(NC(c3c(C)cnnc3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C2 C1(COC)(NC(c2c[nH]c(Br)c2)=O)CCN(C(=O)C(C)c2ccsc2)CC1 C(C1OCCc2sc(F)cc21)NC(=NCC)NCC1CCN1CC N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(=O)CCO2)=O)C(C)(C)C1 CC(C)C(C(=O)NCc1nnnn1C)C(C)NC(=O)C(=O)C(C)(C)C Cc1cc(C)c(S(=O)(=O)Nc2ncc(CCNc3ncco3)s2)c(C)c1 C1(C(=O)NC(CC=C)CO)(CNC(C2CC3C=CC2O3)=O)CCCCC1 c1(C(=O)NC(C2CC(NC(C(C)OCCCC)=O)C2)C)cccc2c1OCC2 N1(Cc2c(OC)cc(N(C)C)cc2)CCCC2(CCCN(C(C3(F)CC3)=O)C2)C1 N1(C(C(C)c2cc[nH]n2)=O)CCCCC12CC(NC(=O)Cc1nc[nH]n1)C2 c1(C(N2CC(CC)C(NC(c3scnc3C)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(CCCNC(=O)OC)N(CCNC(C(C1CCOC1)OC)=O)C(C)C Cc1ccc(Cl)c(C(=O)N(C2CCCCN(C(=O)C#CC3(C)CC3)C2)C)c1 N1(C(C(c2cccc(C)n2)(F)F)=O)CCCCC(CNC(=O)CCC(C)C)CC1 C1(NC(=O)NCCCNC)CN(C(c2ccc(OC)nc2)=O)CC1C(F)F N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 N1(C(CC(=O)OCC)=O)CCCCC(C(=O)Nc2cc(Cl)ccc2OCC)C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCCNC(c1ccn(C(F)F)n1)=O c1(C(N(C2CN(C(=O)C(F)(F)C3CC3)CC2O)C)=O)cn(C)[nH]c1=N C1(C(=O)NCC(CO)NC(c2csc(C(F)F)n2)=O)CCCCS1 c1(CNC(c2cnn(C)c2F)c2n(CC)nnn2)cc2ncccc2s1 C=CCC(C(=O)OCC)NC(=O)C(O)C1CCC1.C(C)(C)(C)O N1(C(C=CC(C)C)=O)CCC2(NC(c3cc(Cl)c(Br)[nH]3)=O)CC2C1 c1(CN(c2nccs2)C(CN2CC(Br)=C(C)CC2)=O)cnc2c(c1)C(=O)NCC2 c1(C(N(CC(C)(C)C)CCOC)=O)ccc(Cl)c2c1OCCO2 C1(NC(C(C)OCCC(C)C)=O)CCCC12CCN(C(=O)C=CS(C)(=O)=O)CC2 c1(OC)ccc(C(c2nnnn2C2CCC2)NC23CC(F)(C2)C3)cn1 C1(C(N(CCC(F)(F)F)C)=O)CCC2CCC1N2C(c1ccsn1)=O C1(NC(c2cnc(C(F)(F)F)s2)=O)COCCN(C(C23CCCCC2C3)=O)C1 C1(NCC)CC2CC3CC(C2)CC1C3.n1(CCCS)cc(C(C)(C)C(C)C)nn1 c1(N2C(C(=O)Nc3ccc(C)nc3I)C=CC2)nc(C)c2cc(Br)ccc2n1 Cc1ccc(CC(=O)Nc2cccc(C3(N)CCC3)c2)nc1 C(=O)(CC1COc2ccccc21)NCCC1(NC(c2c(C)cnn2C)=O)CCC1 C=C(C)C(CC(=O)NC1CCCC(NC(=O)C=C2CCCCC2(C)C)C1)OCC C(=O)(C1OCCc2ccccc21)NCC(C(C)C)NC(C1CC2CC1C1CC21)=O C(=O)(C(C)CCOC)NC(C(CO)NC(c1c(CC)ncs1)=O)C c1(C(N2CCCC(NC(C3(C)CCC34CCC4)=O)C2)=O)ncc2ccccn12 C1(C(=O)NCCC2CCOC2)(CC)CCCN(C(=O)CC2CCCC2)C1 C(=O)(C(C(C)(F)F)c1ccccc1)N1C(C(C)C)C(NC(=O)CCC(N)=O)CC1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CCC(=O)N(C)C1 C#CC1CC2CCC1N(C(c1cc(COC)on1)C(=O)NC1COC1)C2 N1(C(c2ccc(C#C)cc2)=O)CC2CCN(C(=O)CCCn3cccn3)C2C1 NC1c2ccccc2CC12CCN(C(c1cc(Cl)cc(Br)c1Cl)=O)CC2 C=Cn1nccc1C(=O)NCC(F)CNC(=O)C=Cc1ccc(Br)s1 C1(C)(COC)CCCN(C(=O)CC(C)(C)N(C)C(c2ncc(F)cc2N)=O)C1 c1(OC)cc(C(=O)NC2CCN(C(C34CCC3CC4)=O)CC2C)c(F)c(Cl)c1 c1(C(N2CCC(NC(=O)CC3CC4(CC4)C3)C2)=O)cc2cccn2c(O)n1 C(=O)(CC(CNC=O)CC(C)C)N1CC(OC)(CNC(c2ccc(Cl)cc2)=O)C1 CC(C)C(O)C(C)C(=O)N1CCCC(C)(C)C1C(=O)NCC(Cl)=CCl N1(C(CC2CCCC(C)C2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)CC1 CC(CCC(C)(C)C)C(=O)NCC1CCN1C(c1ccc2c(c1O)CCC2)=O C1(CNC(Cc2cn(C)nc2)=O)CCN(C(c2ccnc(CO)n2)=O)CC1(F)F N1(C(=O)CCCN2CCOC2=O)CC(C2CN(C(=O)CC3COCC3O)C2)C1 c1(CC(=O)NCCN(C(c2csc(Cl)c2)=O)C2CC2)coc2ccccc12 CCC(CC)C(F)C(=O)NCCC1CC(NC(=O)C(c2ccccc2F)C)C1 c1(C(N(C2CCCN(C(c3ccncc3)=O)CC2)C)=O)cc(Cl)cc2c1CCC2 C1(C(=O)NC2CC(CCC(=O)NCC3C(C(=O)OC)C3)C2)CC(C)(C)CO1 CC1=C(C(=O)N2CCCC(CCC(=O)NC3CCN(C)CC3C)C2)SCCO1 CC(C)C(C)C(CNC(=O)CC1CC(C)(C)CO1)Nc1nccc(C(F)(F)F)n1 CCN=c1ccc(C(N2CC(NC(=O)C=Cc3ncc[nH]3)CC(C)C2)=O)c[nH]1 C(=O)(CCCC(=O)NCc1cccs1)NCCN(C(=O)CN1CCSCC1)CC c1(CC)ccc(F)c(C(=O)NC2CC(CCNC(=O)CC=C(C)C)C2)c1F c1(OC)cc(O)ncc1C(=O)NC1CCC(C)N(C(=O)Cc2ccnc(O)c2)C1 N1(C(c2ccc(C)nn2)=O)CCOCC(C(N2CCC(O)CC2C)=O)C1 c1(CC(=O)NCC(CNC(c2ccc(OC)c(O)c2)=O)O)ccn2cncc2c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(C1)CN(C(c1cnncc1O)=O)CCO2 C1(NC(c2c[nH]c(=N)s2)=O)CCCOC1C1CCN(C(=O)COCCCF)CC1 N1(c2c(C)cncn2)CC2CC(NC(=O)C(C)C3CCOC3)CC1C2 c1(CC(=O)N(CCC)CCNC(C2CC2(C)C(C)C)=O)ccc(OC(C)=O)cn1 C1(OC)CCC1C(=O)NCC1CC1NC(=O)CNC(c1ccco1)=O n1(CC)ncc(C(N2CCCC(CCNC(=O)Cc3cncnc3O)C2)=O)c1Cl CC1CCC(CC(=O)NCC2(CNC(c3cnc(C4CCC4)s3)=O)CCCC2)O1 CC(C)(C)CC(O)C(=O)NC1CCC1C(N1CCCC(O)(C(N)=O)C1)=O CCC(CC)C(C(=O)N1CCSCC1C(=O)NC1CCn2nccc2C1)OC C1(C(=O)NC2C(OC)CN(C(CN(CCC)C)=O)C2)CCc2nn(C)cc2C1 c1(OC)cc(O)ncc1C(N1CCC(NC(C2CC2C(N)=O)=O)C12CC2)=O C=CCC(CC)C(=O)NCc1cc(C)c(C(N2CCCC2C(O)CC)=O)o1 c1(C(N(CC(CN(C(C2C(C)CCC2)=O)C)O)C)=O)cc(C2CC2)ccn1 c1(C(=O)NCC2CN(C(CC(C)C)=O)CC23CC3)occ2c1CCOC2 CCC(CCCC(=O)N(CC(C)(F)F)C)NC(c1cc(CO)n(C)n1)=O CC1(C)OC(C)(C)C1C(=O)NC1CC1NC(c1cnoc1-c1ccoc1)=O c1(SCC)ccc(Cl)cc1C(=O)NCCCNC(c1cc(C#N)no1)=O C1(C(N2CC(C)(NC(c3coc(C4CC4)n3)=O)C2)=O)CC(C2CC2)C1 C1(F)(C(=O)NCC(C)(C2CC2)NC(c2csc(=N)[nH]2)=O)CCC(F)(F)CC1 C1(C)(C(=O)Nc2cccc(NC(C#CC(C)(C)C)=O)c2)CCCNS1(=O)=O C1(C(=O)NCC2C(CNC(CSCC=C)=O)C2)CCC(N=c2cncc[nH]2)CC1 Cc1ccc(Br)c(CN(C(=O)CCC2CCC(=O)NC2)C)c1 C(=O)(CC(=O)N1CCCC1C(C)(C)NC(C1CNC(=O)N1)=O)NC c1(C(=O)NCCCCCNC(CSC(C)C)=O)ccc(C2CCCO2)cc1 C(=O)(CCCC(C)(C)C#N)NC1(C(N(CCCCC=C)C)=O)CC1C c1(C(N2CC3(C(NC(C(C)OC)=O)CCC3)C2)=O)cc2cc(C)ccc2nc1C CCC(O)(CC)CCNC(C1CCCN(C(C2(O)CCCCCC2)=O)CC1)=O C1(C(N(CC(CN(C(CCNC(=O)OCC)=O)C)O)C)=O)CCCC(C)CC1 c1(OC)ccc([N+](=O)[O-])cc1C(=O)OCCN(S(C)(=O)=O)C C1(N(C(C(C=CC)O)=O)C)CC2CCC(C1)N2C(=O)C(c1ccc(C(C)=O)s1)=O N1(C(c2c(N)nccn2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C(C2CCC2)C1 N1(c2c(C)c(O)ncn2)CCC2CCC(C1)N2C(C(C)(C)C)=O C12(CC(=O)NC3CN(CC(=C)C)CC3(C)C)CC3CC(CC(C3)C1)C2 C1(NC(CCSCCCC)=O)CC1C1CCCN(C(C2(CC)CCCC2)=O)C1 c1(C(CNC(CC2(C#N)CC2)=O)NC(C2CC2(F)F)=O)cc(F)cc(Cl)c1 S(=O)(=O)(c1ccc(F)cc1Cl)NC1CCC(NC(c2ccc(C)c(Br)c2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)C(C)C#N)C)cccc2scnc12 Cc1c(CC(=O)NOCCCCC(=O)NC2CCC2)cnn1C C(=O)(CCN1C(=O)CCc2ccccc21)N(CC(C)N(C)C(C1CC(O)C1)=O)C Cc1ncc2ccccc2c1C(=O)NC1CC(C)CN(C(C2(C#N)CCC2)=O)C1 Cc1ccc(C)c2c(C)c(C(N3CCCN(C(=O)C(O)C(F)F)C(C)C3)=O)oc12 c1(CN2CCCC(C(N(C)CC3(OC)CC3)=O)C2)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)NCC2C(NC(CN(CCCCCC)C)=O)C2)c(Cl)ccc(F)c1C N1(C(C(C#C)(C)C)=O)CC2(C1)OC1(C)CC2(NC(c2ccn3ncnc3c2)=O)C1 c1(C(=O)NC(C)(CNC(=O)CCc2cnc(O)[nH]2)CO)cnc2[nH]cnc2c1 Cc1cc(C(=O)N(C)CC2(CNC(C3CC4CC4C3)=O)CC2)c2c(c1)CCO2 C#CCC(CC(=O)NCC1CC1C(C)C)NC(C12CCC(C1)OC2C)=O c1(C(=O)NCC2N(C(C(CC3CC3)OC)=O)CC2)ccc2nc(N(C)C)sc2c1 C(=O)(CC(C)C(=O)NCCCCC(N1CC(=O)NCC1C(N)=O)=O)OC Cc1cn(CC(=O)NC2CCC2NC(C2CCc3nncn3C2)=O)c(=O)nc1O C(=O)(CC(C)(O)C(F)(F)F)N(C1CN(C(c2cnc(C(C)(C)C)o2)=O)C1)C CC1CCC(C2CCC2)CN1C(=O)C(=O)Nc1ccc(S(C)=O)cc1 C1(CNC(C(C)C2CC2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C12CCC2 C1(CNC(C2CCN(C(C)C)CC2)=O)CC2(CCO1)CC(F)(F)C2 N1(C(C(CC(=C)C)OC)=O)CCC(CCNC(C2CC(O)C(F)C2)=O)C(F)(F)C1 N1(C(C(CCN(C)C)NC(C2CCC=CCCC2)=O)=O)CCC(C)(C2CC2)C1 c1(OC)cccc2c1OCC(C(=O)NCCCCCNC(=O)CC(C)OC)C2 C1(CC#C)CCNCC1.c1(OCCN(C=O)C)ccccc1C(C)C c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)CC2)=O)cnn(CC(C)C)c1C N1(C(C(c2ccc(Cl)s2)C)=O)CCN(CC2CN(C(C3CC3(C)C)=O)C2)CC1 CCS(=O)c1ccccc1C(=O)NCC1CC(F)CN1C(=O)CN1CC2CC2C1 c1(C(N2CCCC(F)(CNC(C(CC)OC)=O)C2)=O)cc2cc(F)ccc2cn1 C1(C)(C(=O)NCC(CC=C)NC(C2CC(O)(CC#C)C2)=O)CCC(=O)N(C)C1 C(CCCCCNC(=O)COC1CCCCC1C)N(C(c1c(C)occ1)=O)C c1(C(=O)NCC2N(C(c3c(C)nc(C)[nH]3)=O)CCCC2)cc(Cl)n[nH]c1=N CC(Cc1nccn1C)N=c1[nH]c(=N)[nH]c(=NC2CCC(S(C)(=O)=O)C2)[nH]1 C1(CNS(CC(=O)OC)(=O)=O)CN(C(C2(c3cccs3)CC2)=O)CC1(C)C N1(C(C(C(C)O)C)=O)CC2CC(NC(c3cc4n(n3)CCO4)=O)C2C1 CC#CCCC(=O)N(CC(=O)N(C)CC1CCCS1)C(C)C Cc1[nH]c2c(C(N3CC4C(C3)N4c3ncnc4ccccc34)=O)cccc2c1C N1(C(C(C)OCCOCC)=O)CC2(CC(NC(c3coc(C)n3)=O)C2)C1 CC(O)CC(C)(C)CNC(c1ccc(CNC(C2COCC2C(N)=O)=O)s1)=O C1(O)(CCNC(CN(CC)CC)=O)CCN(C(=O)Cn2cccc(N)c2=O)CC1 C(=O)(CCS(C)=O)NCC(C(C)C)NC(c1n(C(C)C)ncn1)=O Cc1coc(C(=O)NC(C)CCN(C(=O)CSCc2ccccn2)C)c1C N1(C(C2C(C)CCO2)=O)CC2OCCN(C(c3cc4cccc(F)c4o3)=O)C2C1 Cc1cc(C(N2CC(NC(c3cnnn3C3CC3)=O)CC(C)C2)=O)c(F)cc1Cl c1(C(N2CC(NC(C(C(COC)C)C)=O)C2)=O)cncc([N+](=O)[O-])c1 c1(C(CNC(CCOC)=O)NC(=O)COCC(=O)OC(C)(C)C)ccccc1 N1(C(C2CC=C(C)CC2)=O)CC2(CCN(C(C3CC(F)C3)=O)CC2)C1 N1(C(CCNC(=O)CO)=O)CC=CC1C(=O)NCC1(F)CCC1 C12(NC(CCCCOC)=O)CCN(C(=O)C(=Cc3cscn3)F)CC1C2 c1(C(=O)NCC2(OCC)CC2)cc(CNC(C2CCCC2SC)=O)nn1C N1(C(=O)C(F)(F)c2cncs2)CCC(c2cccc(C(F)(F)F)c2)CC1 CC1=NOC2(C1)CC(C(=O)NC1CCN(C(C3CCC(=O)O3)=O)C1C)C2 C1(NC(c2c(N)n(CCO)nc2)=O)CS(=O)(=O)CC1NC(c1ccc(F)o1)=O c1(COC)nc(NCc2ccoc2C)cc(N(C)CCc2nccs2)n1 c1(C(N(CCCNC(=O)CC(C)OC)CC)=O)cc(F)ccc1C(F)F C(CC(CC)(CC)NC(C1C2CCC(F)(F)C12)=O)NC(C1CCCN(CC)C1)=O C1(F)(CNC(=O)CC2CC2c2ccoc2)CC(CNC(=O)Cn2cnnn2)C1 C#Cc1cc(C(=O)N(C2CCN(C(=O)C=COCC)C2)C)ccc1C Cc1ccc(Cl)c(N)c1C(=O)NCCCN(C(=O)C1=NOCC1)C C(C(CC(=O)NCC1C=CCN1C(c1cc[nH]n1)=O)C(F)(F)F)N(C)C C(=O)(C(C)(COC)CC)NCC(CC)Nc1ccccn1.c12cccc(c1)OC2 C12CCC(CC1)NC2=O.c1(NC(C2(CC(C)=O)CC2)=O)cncnc1O C1(NC(c2cnns2)=O)CC(F)CN(C(C2CCS(=O)(=O)N2)=O)C1 C1(C(N2C(CNC(=O)CC(=O)NC3CC3)C=CC2)=O)CC(=O)N(C2CCCC2)C1 Cc1cc(C(=O)NC(CCN(C)C(C2CC=CCO2)=O)C(C)(C)C)ccc1C#N C1(NC(CCCCN(C)C(C2CC(=O)OC2(C)C)=O)=O)CCC(=O)NC1=O C1(C(=O)NC(CCCNC(C(C)N(C(C)=O)C)=O)(C)C)CCC2(CC1)OCCO2 CS(=O)(=O)C1CCCCN(C(=NCC2CC2)NCc2nsc3ccccc23)C1 c1(N2CC(C)OC(CCO)C2)nc(NCc2nc(CO)cs2)c2ncn(C)c2n1 N1(C(=O)CC2CCCN2C(c2cc(CCO)[nH]n2)=O)CCC(O)C1C(F)(F)F C1(N(C(=O)CCNC(=O)NC)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 C1(N(C(CSCCOC)=O)CCO)CCN(C(C2(C)CC=CC2)=O)C1 N1(CC)CCCc2cc(CN(C(=O)CCCC(F)(F)F)CCO)ccc21 c1(C2(C(=O)NC(C3CN(C(=O)CC4CC4)CCO3)C)CC2)c(Cl)cccc1Cl C1(C)(C(=O)NC(C)CN(C(=O)CNC(=O)OC(C)(C)C)C)CCC(=O)C1 c1(C(=O)NC(C(=O)N(C2C(C)CCC2)C)(C)C)ccc(CC#N)cc1 C1(CC)C(C(N2CCC(NC(N)=O)CC2)=O)CCN1C(=O)Cn1nccc1C c1(NC(=O)Cc2cn(CCNC(COCCOC)=O)nn2)cccc(OC(F)F)c1 c1(C(=O)NC2CC(C(=O)NC(C)C(N)=O)C2)ccccc1Cl C=C(CNC(c1cnoc1-c1cccs1)=O)CCNC(C1(CC)CCOC1)=O c1(COC2CCN(C)CC2)cnn2c1CN(C(=O)C(Cl)=CCl)CC2 C1(C(N(C(C)CCNC(=O)CCC(=O)c2ccncc2)C)=O)CCCCC1(C)C CCC(C)C(CC(=O)N1CCC12CC(O)C2)NC(=O)CC1CCCO1 c1(CC(=O)NC(C2CSC2)C)c(C)ncnc1C N1(C(c2cccc(NC)n2)=O)CCOCC(NC(=O)C(C2CCCCCC2)O)C1 C1(NC(c2c(CC)c[nH]c2)=O)CCC(C)N(C(=O)CCOCC(F)(F)C(F)F)C1 C(=O)(C(CO)C(F)(F)F)N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCCC1 N1(C(c2c(C)c[nH]c2)=O)CCS(=O)(=O)C(CCNC(=O)CCOC2CC2)C1 Cc1cc(C(=O)NCC2(F)CCCN(C(c3cnc[nH]c3=N)=O)C2)nc(O)n1 Cc1c(F)ccc(CN2CC3CC3(C(=O)Nc3cc(Br)cnc3O)C2)c1F c1(OC)cccc(C(N2CC3CC(NC(c4cc(O)cc(F)c4)=O)C2C3)=O)c1N C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(c2nn[nH]n2)CC)(CC)C1 C1(C(=O)OCC)NC(=O)N(c2cccc(NC(=O)C(=O)N(C)CCOC)c2)C1=O C(=O)(C1CCCc2nn[nH]c21)NC1C2CN(Cc3cnn4ccn(C)c43)CC21 C1(O)(CCNC(c2c(C(C)C)con2)=O)CCN(C(n2nnc(=O)[nH]2)=O)C1 N1(C(c2ccc(=N)[nH]n2)=O)CCC(NC(=O)COCC2CCOCC2)C(F)C1 C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)N1CC(N(OC)C)C1 C12CC3CC(C1C3)C2=O.Cc1nccnc1C1CN(C(=O)NC(C2CC2)C2CC2)C1 Cc1ccc2c(C(=O)NCC3(C)CCN(C(C4CNC(=O)C4)=O)C3)coc2c1 CC(CC(=O)NCC1CC(C)N(C(c2n[nH]c3c2CCC3)=O)C1)CC(F)(F)F C(C(C)(C)CC(=O)NCC(N1CCN(C)CC1)(C)C)N(C)C(=O)OC(C)(C)C N1(C(C2CCCN(C)C2)=O)CCC2(CCCN(C(=O)CCCCBr)C2)C1 C1(NC(=O)Cc2nc3c([nH]2)CCCC3)CCN(C(c2ccco2)=O)CCC1CO C(C(N=[N+]=[N-])C(=O)NCC1CC(NC(C2CNC(=O)O2)=O)C1)OCC c1(C(N2CC(CNC(c3cccc(C#C)c3F)=O)C2)=O)c(F)c(F)cc(F)c1F CC(=O)C(C)(C)CC(=O)NCC(C1CCCCC1)NC(=O)CSC1CC1 c1(NC(C(=O)NCC(C(C)(C)C)OC)=O)ccc2c(c1)NC(=O)CS2 Nc1cc(C(=O)NC2CCN(C(C3(C4CC4)CCC3)=O)C2)cc(Cl)n1 Cc1cc(C(=O)NCC2(C3CC3)CC2)ccc1C#N.C12CCCC1NC2=O C(C(CC(=O)N1CCCCC1CNC(=O)CC(C)(C)C#N)C(F)F)N(C)C1CC1 C(C(=O)NCC=CCNC(c1c(-n2cccn2)cccc1F)=O)(C(C)(C)C)SC Cc1nc2ccccc2nc1NC(C1C=CC(NCc2cccs2)C1)=O N1(C(c2ncc(C)cc2C)=O)CCCC2(CCCN2C(=O)CC2CCC2(C)C)C1 n1(CC(=O)NCCN(C(=O)CC23CCCC2C3)C(C)C)c(O)nnc1O [N-]=[N+]=NC1CC(C(N2CCS(=O)(=O)CC2)=O)N(C(=O)OC(C)(C)C)C1 N1(C(C=CC(=O)OCC)=O)CCCC(C(=O)NC2C=C(C)CCC2)C1CC Cc1cnn(CC(N2CC(NC(=O)C(F)(F)C3(O)CCCC3)C2)=O)c1 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2(NC(=O)CN=S(C)(C)=O)CC2)C1 C12(NC(Cc3cn(CC)nn3)=O)CCCC1(F)CN(C(C1(SC)CCC1)=O)C2 c1(OCCC(=O)NCCCC2CN(C(=O)CCF)CCO2)ccc(F)cc1F c1(OC)cc(NC(C2CCN(Cc3cccc(O)c3F)C2)=O)ccc1I c1(NC(C2CC(O)CN2S(=O)(=O)CC2CC2)=O)cc(Cl)c(Br)c(Cl)c1 c1(N2CCC(CCOC)(NC(=O)CNC(N)=O)CC2)ncnc(C)c1C#N CCC1=NOC(CC(=O)NC(C)(C)C(C)NC(c2ccncc2OC)=O)C1 CCCC(CC)C(=O)NC1(CNC(c2cnoc2C)=O)CCCCC1 N1(C(CCCC(C)O)=O)CCCCC(C2CN(C(C3CC3F)=O)C2)C1 Cc1cc(F)c(CC(=O)Nc2cccc(C(=O)NC(C)(C)C)c2)cc1F c1(C(N(CCOCC)Cc2cncn2C)=O)cn2ccncc2n1 C=CCC(C)(C(=O)NCC(C1CC1)N(C(=O)CCC(C)OC)C)N(C)C N1(C(C(C)OCC2CC2)=O)CC(=O)CCC1C(N1CCC12CC(C(N)=O)C2)=O c1(COC(CC2(SC)CC2)=O)c(N(C)C)n(C)c2c(C)cccc12 C1(NC(CN2CCC(C)CC2)=O)CCC12CCN(C(C1CCS(=O)CC1)=O)CC2 CCCCC(O)C(=O)Nc1ccc(C(C)NC(c2csc(CC)n2)=O)cc1 C(c1cncn1C)=CC(=O)N(C(C)C(N1CCC(N2CCCC2)C1)=O)C1CC1 CCCCCC(F)C(=O)NCC(C)(C)CC(=O)NCCN(CCC)CCC n1(CC)ncc(Br)c1C(=O)NC1CC(F)(CNC(=O)CCNC(C)=O)C1 C1(CNC(Cc2c(C(C)C)cccc2)=O)C2CN(Cc3cn[nH]c3)CC12 O=C(N=c1ccc(C2CC2)n[nH]1)NC1CCCC(N2CCOCC2)C1 c1(C(=O)NC2COCCN(c3ncnc(CC)c3F)C2)ccc2nsnc2c1 Cc1cc(C(N2CC(NC(c3c(Cl)cnn3C)=O)C(CC(C)(C)C)C2)=O)sc1C c1(NC(C)C(=O)NC2CC(CNC(=O)CCn3ccnn3)C2)ccc(C#N)cc1 Cn1cc(C(=O)NCC23CC2CN(C(=O)COc2ccc(Cl)cc2)C3)ncc1=O N1(C(CCNC(=O)OCC)=O)CCC2(CNC(c3cnn[nH]3)=O)CCCCC12 c1(OCCCOC)ccccc1-c1nc(-c2ccc(CO)nc2)no1 C(=O)(CCCC(C)(C)C)N(CC(=O)NCC1CC1Cl)C CCCC(C)(C)C(=O)NC(C1CN(C(c2cc(CC)on2)=O)C1)C c1(NC(C2COCC2C(=O)O)=O)ccc(OC2CCCCO2)cc1 c1(C(C)=O)ccccc1C(N1CCC(NC(C2(C)C=CCCC2)=O)C1)=O Cn1nc(C(=O)NC2CCCCC2CNC(=O)COC2CC2)c2c1CCCC2O C1(CCC(=O)NCCN(C(=O)Cc2nonc2C)CC)COC(C)(C)O1 C1(NC(COCC(=O)OC)=O)CCOCC1NC(=O)CCc1ccccc1C Cc1nc2cccc(C(N3CC(Cn4cc(Cn5cncn5)nn4)C3)=O)n2n1 C1(F)(CNC(C(C)NC(CC)=O)=O)CCN(C(c2ccccc2C(=O)OC)=O)C1 c1(C(=O)NCC2C(NC(=O)CCC3CCCC3)CCCC2)cnc2ccccn12 c1(CC(N2CC(O)CC(NC(C3(OC)CC3)=O)C2)=O)ccc2cccnc2c1 CC1CC(=O)NC(C(N2CCCCC2CCC(=O)N(CCCO)CCCO)=O)C1 c1(C(=O)NCCC(=O)OC)ccc2[nH]ccc2c1.C1=CC(=O)N2C1CCC2 N1(C(C(C)CC2CC2)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2CC1 c1(NC(C(c2cccnc2)NC(=O)OC(C)(C)C)=O)cc2c(nc1O)CCCC2 c1(C(=O)NCC2N(C(c3n(CC)ncc3)=O)CC=C2)cc([N+](=O)[O-])cc(C)c1Cl C(=O)(CC(C)C(F)(F)F)N1CCC(CCOC)(NC(C2CCC2C)=O)C1 N1(C(c2c(C#C)cnn2C)=O)CCCC(C2(NC(C3CCS3(=O)=O)=O)CC2)C1 c1(C(=O)NC(CCCCNC(C(CC)COC)=O)C)cnc2c(c1)COC2 Cc1cc(C)c(C(=O)NC2CC3CCC2N(C(c2snc(O)c2Cl)=O)C3)cc1N N1(C(C2C(C(=O)NCC(=C)C)C2)=O)CCCC(CC)(CO)C1 C1(CC)CC(C(N2CC(NC(c3cccnc3CC)=O)CC(C)C2)=O)CC(=O)N1 O=C1Cc2ccc(C(=O)NC3(CO)CCN(C(=O)CC4=CCCCC4)C3)cc2N1 C1(NC(C(C)C2CC2)=O)CCCCN(C(c2scnc2C2CC2)=O)C1 N1(C(c2c(C)cc(CNC(=O)CC3CC3(C)C)o2)=O)CCOC(C)C1C N1(CC(=O)NC(C2CCN(C(C(COC)C)=O)C2)(C)C)CCN(C)CC1 O=C1CCC(c2ccccc2)(C(=O)N(C(=O)C(F)(F)F)CC2CCS(=O)CC2)CN1 N1(C(C(C(C)C)c2cnc(C)s2)=O)CCCC(NC(=O)COCC2CCC2)CC1 O=C1CC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCOCC2)CN1 c1(CC)cc(C(=O)N(CC(O)CN(C)C(c2cncnc2)=O)C)cc(Cl)c1 Cn1nc2c(c1C(=O)NC1CC3CN(C(c4ccns4)=O)CC13)CCCC2 C1(OC(c2ccc(CN3C(=O)CCC3=O)cc2)=O)CCC2(CCOC2)C1 c1(C(c2n(C(C)(C)C)nnn2)NCCC2(CS(C)(=O)=O)CC2)ccc(Cl)c(F)c1 C1(SCC(N2CCC(C(=O)OCC)CC2)=O)CC(c2ccc(C)cc2)=NO1 C1(C(=O)NC(CNC(c2cccc(OC)n2)=O)CO)Cc2ccccc2C(=O)O1 C(=O)(C1=CC2(CCN(C(=O)CN3CCN(C)CC3)C2)C1)NC(CCCC)C C12CN(CCO1)C(=O)NC2=O.N1(C(=O)NC2C3COCC23)CCOCC1 N1(C(c2n(CC)nnc2C)=O)CCCN(C(=O)CP(C)(C)=O)CC1C C1(C(N(C2CCN(C(c3ccn(C)c3)=O)CC2)CC2CC2)=O)CCC(C)(F)CC1 CC(C(O)C(=O)N(C(C)CCNC(=O)CCOCC(F)F)C)c1ccccc1F C1(CC(NOCCC)=O)CC(NC(=O)C(O)C2CC2)C1(C)C N1(C(C2CC(C(C)C)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(CC(F)F)C1 C1(CC(=O)NCC(C)(C)OCC(=O)NCC2CCCCO2)CC(=O)NC1=O C(=O)(CC1CS(=O)(=O)c2ccccc21)N1CCC(N(C(=O)C=CCF)CC)CC1 S(=O)(=O)(c1ccc(N(C)CC2CCCC2)c(Cl)c1)NCCC1CCC(C)O1 CCC(Cc1cccc(C)c1)C(=O)NC1CC1NC(c1ccc(SC)cc1)=O C1(C(N2CC(CNC(C3(C(C)C)COC3)=O)C2)=O)COCCN1CC(F)F N1(C(c2c(CC)non2)=O)CCC(F)(CNC(c2cnc(O)o2)=O)C1 C1(CC(=O)NCC2(NC(c3c(C)[nH]cc3)=O)CCOC2)CCCC12CC2 Cc1nc(C)n(CC2CCCCN2C(=O)Nc2sccc2C(F)(F)F)n1 C1(c2cccnc2)(C(=O)NC2CC(NC(C3C4COCC34)=O)C2)CC(F)(F)C1 C1(NC(C(COC)OC)=O)CCC2(CC1)CN(C(c1ccccc1C)=O)CCO2 N1(C(C(CC)OCC)=O)CCC(CO)(CNC(=O)CCC(=O)NC)C1 c1(C(N2CCCC(NC(C(C)(C(C)C)NC(C)=O)=O)C2)=O)c(F)ccc(Cl)c1N c1(OC)ncc(CNC(c2cc(-c3cccnc3)ccc2C)=O)cc1Cl C1(C(=O)Nc2cccc(C(C)C)c2)(OC)CCN(C(=O)C=Cc2ccncn2)C1 N1(C(C2C(C)CCOC2)=O)CCC(C)(C(N2CCC2CC2CC2)=O)CC1 N1(C(C2CC(=C)C2)=O)CCCC1(C(=O)N(CCS(C)(=O)=O)C)CC Cc1ocnc1C(c1nnnn1Cc1cccs1)NCCc1ccc(Cl)s1 c1(C(N2CC(NC(c3c(CC)nn(C)c3)=O)C(O)C2)=O)cn2cc(Cl)cnc2n1 n1(CCC)ccc(=NC(=O)C2(CCNC(C3CC=CC3)=O)CCC2)[nH]1 C1(C(=O)NCC2CC(CF)C2)C=CCN(C(c2ncc[nH]2)=O)C1 C1(NC(N2CCCC(NC(=O)CCc3ncccn3)C2)=O)CCCC12OCCO2 C#CC1CN(C(=O)C(O)C=C)CCN1C(=O)COC1CCCC1 c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CCn3cncn3)C2)cnc1C C1(NC(=O)CC2(CO)CC2)CN(C(c2cccc3c2OCO3)=O)C2(CCOC2)C1 C1(NC(COCCCCC)=O)CCCCC1CNC(=O)C=CS(C)=O C(=O)(C1=C(Cl)CCOC1)NCCCNC(CC(C)n1cc(Br)cn1)=O N1(C(C(CC=C)C)=O)CC(CNC(c2cnn(C3CCCC3)c2C)=O)C(C)(C)C1 C1(C(=O)Nc2c(C)cccc2)CC2(CC2)CN1C(=O)CC1CCCOC1 Cc1n[nH]c(C)c1C(=O)NCC(C)CC(=O)NC1(C)CC(C)(C)C1 c1(C(=O)NCCCCN(CCCNC(C2(C)CCCO2)=O)C)cn(C)c(C(F)F)n1 C(=O)(CCC(=O)NN(C)C)NC1CC2(C(C(N(C(C(C)SC)C)C)=O)C2)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CCC2(CCC2)CN1C(=O)COCCF C1(CC)CCCN(C(=O)C(C)OCCC(C)C)C1C(=O)NCc1ccncc1Cl c1(C(C(=O)NC(C(C)NC(c2c(CCC)nns2)=O)C)(F)F)ccc(F)cc1 Cc1coc2ccc(C(N3CC(NC(=O)C(O)CC(N)=O)CC3CO)=O)cc12 C(=O)(CC(O)C(C)C)N1CC(N2C(c3onc(OCC)n3)COCC2)C1 N1(C(C(CSC)C)=O)C(CNC(=O)CCCc2ccc(Cl)cc2)CC2CCCC12 C1(C(=O)NC2CN(C)C2)C2CC1N(C(c1cccnc1Br)=O)C2 c1(C(N2CCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc(Oc2ccccc2)cn1 C1(CC(=O)NCCCCN(C(c2c(C(C)C)nn(C)c2)=O)C)CCC2(CCC2)O1 N1(C(c2ccc(=N)[nH]n2)=O)CCN(C(=O)CNC(=O)C2CC2)C2CCCCC12 C1(N(C(=O)CC2CC(F)C2)CC)CCCN(C(=O)COC(C)(C)C(F)(F)F)CC1 CCC(C)(C)CCCC(=O)N1CCC(=CCNC(C2CC2F)=O)CC1 Cc1c(O)ccc(C(=O)Nc2ccc(NC(c3cccs3)=O)cc2)c1C C1(CNC(C(c2cccc(Cl)c2)OC)=O)CC2CC2N1C(=O)C(C)(F)F C#Cc1ccc(Cl)c(C(=O)NCc2cc(F)ccc2N2CCCC2)c1 Cc1ccc(C)c(CC(=O)NC(C)CNC(c2ccccc2SCCO)=O)c1 C1(c2cccc(CC)c2)NC(=O)N(CC(C)C)C(C(C)F)=C1C(=O)OC C(C(C(=O)NC(CC)C(=O)NCC1=NOCC1)N(C)C)OC Cc1cccc(C(N2CCCCC2C(=O)NC(C)(CO)C(F)(F)F)=O)c1F S(=O)(=O)(c1ccc(C(=O)NC23CC(C2)N(C(=O)CC(C)COC)C3)cc1)NC C1(C(N2CCN(CCNC(C3(OC)CCC3)=O)CC2)=O)CC(C2CCC2)C1 c1(C(N(CC(O)CN(C)C(C2CC23CCCC3)=O)C)=O)cccc(F)c1C#N C1(C(=O)NCCCCN(C(=O)COCCCF)CC)CSCN1C(C)=O N1(C(C(C)OC2CCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CC2CC(C1)C2(C)C N1(C(C)=O)CCC(NC(=O)Cc2ccccc2-c2ccccc2CO)C(F)C1 CC(C)CCC(F)C(=O)N1CCC(C(=O)NCC2CC3C=CC2O3)C12CC2 C1(C(=O)NCCN(C(c2cnc(C)n2C)=O)CC)CCC(=O)CC1C N1(C(CC=CC)=O)CC(NC(C2CC(=O)N(CCOC)C2)=O)C(O)C1 C(c1ccc(C2CC2)cc1)=CC(=O)NC1CN(C(C2CC(N(C)C)C2)=O)C2C1C2 c1(C(C)=O)ccc(CC(N2CCN(C(=O)Cc3cnc(C)[nH]3)CC2)=O)cc1 c1(C(=O)NC2CCC(N(C)C(c3ccc(=O)oc3)=O)C2)cc2ncccc2o1 CCN=C(NCC1CCCN1c1cnccn1)N1CCC(OCCOCC)CC1 c1(NC(C2CCN(Cc3c(Cl)cncc3Cl)CC2O)=O)cc(Cl)ncc1C(F)F c1(C(=O)NCCN(C(C=CC(=O)NC2CC2)=O)C2CC2)cc(F)cc2nc[nH]c12 c1(CC)cnsc1C(N1CC=CC1C(=O)NC(c1snnc1C)C)=O c1(CONC(Cc2cc(OC)c(Br)cc2)=O)cc(OC)c(OC)c(I)c1 C1(NC(=O)NC(C(=O)O)C2CCC2)CC(O)(C(F)(F)F)C1 Cn1nnc2cc(C(=O)NCC3(C)CN(Cc4cc(Cl)cnc4F)C3)ccc12 C1(NC(c2cc(C3CC3)nc(O)c2)=O)CS(=O)(=O)CC1NC(c1ccccn1)=O Cc1ccc(CC(N2CCOC(CN(C(=O)CC3CCOC3)C)C2)=O)cc1F Cc1ccc(C(=O)NCC2CN(C(c3cccnn3)=O)CC2C(F)(F)F)c(C)n1 CCC(C)(CNC(=O)C=CC(=O)OC)C(=O)NCc1nc(COC)n[nH]1 S(=O)(=O)(c1[nH]c(=NCC2CC(n3ccnn3)C2)ccc1Br)NCC(COC)C N1(C(CCNC(=O)C=CCl)=O)CC2CC(C1)N(C(C1CCOC1C(F)(F)F)=O)C2 N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC(F)C(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 N1(C(CN(C(C2CN(C(C)C)C2)=O)CC2CC2)=O)CCCC(F)(F)C1 N1(C(C(F)=C(C)C)=O)CCC2(CCCCC2NC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(OC(c2nc(CN=c3[nH]ncs3)cc(O)n2)C)ccc(F)c2c1C(=O)CC2C c1(C(N2CCC(C(C)NC(c3cc(C)cc(C)c3)=O)C2)=O)cscc1S(C)(=O)=O C(=O)(C(C)CC(C)C)N(CC(CNC(C=Cc1cc(C)no1)=O)(C)C)C C1(CS(=O)(=O)NCC(c2ccc(F)cc2F)(C)O)CC2C(C1)C2(F)F C1(CNC(c2cccc(C)c2F)=O)CN(C(c2cnc(O)n2C)=O)C2(CCC2)C1 c1(C(N2CCCC(N(C(CCCC(C)=O)=O)CCO)C2)=O)cc2c(s1)CCSC2 CCC(C)(C)C(=O)NC(CN(C)C(c1c[nH]c(=N)s1)=O)Cc1ccccc1 C1(C(=O)NCCNC(C2CN(C(c3csc(C)n3)=O)C2)=O)CN=C2N=CNN2C1 c1(C(=O)NCC2CN(C(CC(C)F)=O)C3(C2)CCC3)cc2ccccc2cc1F C=CCCCC(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)CN(C)C(C)C c1(C(N2CC(CC(C)NC(c3cnnc(O)c3)=O)C2)=O)cc2c(O)cccc2[nH]1 C(=O)(CCCC(F)(F)CO)N1CCC(C(C)NC(c2nn(C)cc2Cl)=O)C1 C(CC(C)(C)C)(c1n(CC=C)nnn1)(C1CC1)NCc1c(C)ccnc1C c1(C(=O)NC2CCN(C(C3C4COCC34)=O)CC2F)ccc(F)c(Cl)c1F Cc1ccc(C(C)NC(=O)C(C)N(c2ccncc2F)C(C)C)cc1 c1(C(C)C)ccc(C(=O)NC2CCCC(NC(=O)C(O)CN3CCCC3)C2)cn1 N1(C(C(c2c(NC(C)=O)cccc2)(F)F)=O)CCC(O)(CNC(=O)C(C)C)CC1 c1(C(=O)NC2(CNC(C3C(SC)CCC3)=O)CC2)cc(N)cnc1Cl c1(C(=O)NC2(C(=O)NC(CCCC)CCCC)CCC2)cccn2cncc12 C(=O)(CC(F)(F)C(F)(F)F)N1CC2C(CNC(c3c(SC)nccn3)=O)C2C1 c1(OC)cnccc1C(=O)NCCC1CC(NC(=O)CC(C)n2ccc(C)n2)C1 N1(C(C(CCOC)(C)C)=O)CCCC2(CC(NC(C3(F)CCOCC3)=O)C2)C1 c1(C(=O)NC2CCCN(Cn3cccn3)C2)ccc(F)c(S(=O)(=O)N2CCC2)c1 C1(C2CCN(C(c3n[nH]cc3C(F)(F)F)=O)C2)(NC(c2ccc(Cl)cc2)=O)CC1 C12(CNC(C(CC)(C)C#N)=O)CCCC(CN1C(c1ccc3nc[nH]c3c1)=O)C2 c1(C(N(C2(CCCCNC(=O)C=CC(F)(F)F)CC2)C)=O)cc(CO)[nH]n1 CC1CC(NC(=O)CSc2nncs2)CN1c1cc(-n2ccnc2)ncn1 N1(C(C2(CC#C)CCCO2)=O)CCOC(C2CN(C(c3csc(S)n3)=O)C2)C1 N1(C(C(CNC(c2ccc(C)s2)=O)C)=O)CCc2ccncc21 n1(C(C)C)cc(C(=O)NCC(O)CNC(=O)CCCCN2CCCC2)c(Br)n1 Cc1ccc2c(C(N3CCC(C(C)NC(c4occc4F)=O)CC3)=O)csc2c1 c1(C(N2CC(NC(C(C)n3cccc3)=O)(CO)C2)=O)cc2c(cn1)CCCC2 C#CCC(CC(F)F)C(=O)NCSC.C1(=O)CCC(=O)NCC(C2CC2)N1C Cc1c(C(=O)NCC2CC2NC(C2(C(F)F)CC2)=O)noc1-c1ccccc1 c1(CC(=O)NC(CNC(COCc2onc(C)n2)=O)(C)C2CC2)cc(Cl)n(C)n1 C(=O)(CCN(OC)C(=O)C(C)C(O)C(C)C)N(C1(COC)CCCC1)C1CC1 c1(C(=O)NC(C(C)NC(COCC=C)=O)C)cc(O)c(F)cc1N C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)NCC1(O)CCC(C)(C)C1)N(C)C c1(-c2ccc(CNC(C3CCOC3c3nc[nH]n3)=O)s2)ccc(Cl)cc1 c1(CC)cnn(C)c1C(=O)NC(C)CCNC(=O)C(c1ccccc1)OC c1(C(N(CC)CC2CCN(C(C3(CO)CC3)=O)CC2)=O)cc2sc(Cl)cc2s1 c1(C(=O)NCC(C)CNC(C2CC2Br)=O)cn2ccccc2n1 c1(CC)ncnc(CC)c1C(=O)NC(C)CCN(C(=O)CC(C)c1ccco1)C CC1(C)CCN(C(C2CC=CCO2)=O)C1CNC(=O)COCc1ccncc1 c1(CNC(=NC)NCC2(N3CCOCC3)CCC2)cccc(C(C)OC)c1 c1(C(N(C2CN(C(c3c(C)nns3)=O)C2)C)=O)cncc2ccccc12 c1(CCN(C)CCO)cn(CC(=O)N(C)CCN2CCOC2=O)nn1 O=C(C#CC1CC1)NCCC1CSCCN1C(=O)CSc1ccccc1 N1(C(C(C)SCC)=O)CCC(C)(C)C1CNC(c1c[nH]nc1-c1ccncc1)=O c1(C(C)OC(c2cc(COC)no2)=O)ccc(F)cc1 c1(C(=O)NCC2CCC(NC(c3c(C)nsc3C)=O)C2)c(Cl)cncc1Cl C1(CNC(c2ccc(C)cn2)=O)CCN(C(C2C=CCC2)=O)C1(C)C c1(C(N(c2cnn(C)c2)Cc2c(C)non2)=O)ncccc1Br C1(NC(C(C(C)O)N(C)C)=O)CCC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 c1(C(=O)NC)cccc(C(N2CC(NC(=O)CC3CCN(C)C3)C(C)C2)=O)c1 C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(c2ncc(Br)c(C)n2)CC1 N1(CC(c2cccc(SC)c2)NCC(C)C)CCCC(C)(C#N)C1 N1(Cc2cc(C(=O)OC)[nH]c2)CCN(C(c2cc(Cl)nc(Cl)c2)=O)C(CC#N)C1 N1(C(C(C(C=C)C)C)=O)CCc2ccc(CNC(c3cnsn3)=O)cc2CC1 C(=O)(C1=CCCCC1)NC1(C)CN(C(C2CCC23CCCO3)=O)C1 c1(OC)ncc(Cl)cc1C(=O)N(CCCN(C(=O)Cc1ccco1)C)C C1(CC(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)CC2C=CCC2)CC1 N1(C(C2ON=C(C(=O)OC)C2)=O)CCCC2CN(C(C3CC(C(C)C)C3)=O)CC12 C1(NC(CCCCOCC)=O)CN(C(=O)C(C)n2cncn2)CC(F)(F)C1 C(CC(=O)NCC12CCC(CC1O)C2)(C(F)(F)F)NC(C1C(C)SCCC1)=O N1(C(c2[nH]cc(C)c2)=O)CCC(C)C(CC(=O)NCC(=O)NCCO)C1 N1(C(c2c(COC)noc2)=O)CC(C)CCC1CNC(=O)C(F)(F)C1CCCC1 CC1(C)OC(C(=O)NCC(C)(F)CNC(c2csnn2)=O)C(C)(C)O1 C1(C)(CNC(CCc2onc(CC)n2)=O)CCCN(C(c2c(C)nsc2C)=O)C1 N#CC1CCCN(c2nnc(-c3ccccc3F)n2CC2=CCCCC2)C1 N1(C(=O)CC2CC=CC2)CC2(C1)CN(C(C1CC13CCOCC3)=O)CCO2 N1(C(COCCOCC#C)=O)CCC2OCCN(C(c3ccsc3C#N)=O)C2C1 C1(NC(=O)CCCn2cc(-c3ncc(F)cn3)nn2)CC2CC(C1)C(=O)N2 N1(C(c2cc(OC)ncc2)=O)CC(CNC(C2CC(=O)NC(=O)C2)=O)C(C)(C)C1 C1(CNC(C2(NC(C3C(C)=CCS3)=O)CCCC2)=O)CCCC(F)C1 c1(C(N2C(CNC(c3c(C)ccs3)=O)CCC2)=O)c2c(nn1C)CCC2 c1(OC)c(CC(N2CCOCC(NC(c3cc(F)n[nH]3)=O)C2)=O)cccc1C#N C1(CNC(=O)NC(c2c(F)cccc2I)C(=O)O)CCc2c(O)cccc2C1 c1(SC)ccccc1C(C)NC(=O)NC1CCN(c2ccc(Br)cc2)C1 N1(C(CCN(C(=O)CCc2ccncn2)C(C)C)=O)CCC2(C1)CC2(F)F S(=O)(=O)(CCC(=O)N1CCC(O)(CCNC(=O)CCC=CC(C)C)C1)NC c1(C(=O)NCCCN(C(=O)Cc2ccnnc2O)CC)cncc(OC)n1 N1(C(C)=O)CCC2(CC1)CN(C(=O)C1CC1)C2.C(=O)(C(C)CC=Cc1ccccc1)O Cc1[nH]nc2ccc(C(N3CCCC(F)(CNC(=O)CSC(C)C)C3)=O)c(Cl)c12 c1(C(=O)NCC2(F)CCC(NC(C)=O)C2)c(OC(F)F)cccc1Cl CC1CCN(C(=O)C(=O)Cc2cccs2)CC1CNC(C1(C)CCCS1(=O)=O)=O N1(C(C(N2CCCC(C)C2)=O)=O)CCC2CC1CN2C(C1CCC=CCC1)=O c1(C(N2CCC(NC(CCN(C)CC)=O)CC2C2CC2)=O)cc(C)c(C)nc1C CCC(CNC(c1cc(COC(C)(C)C)on1)=O)(CC)NC(=O)C(C)N(C)C O=C(C#CC1CCOC1)NCC1CCCCN(C(c2cc3cnccc3[nH]2)=O)C1 c1(NCC(C)CO)ccc(S(=O)(=O)NCc2cc(Cl)n(C)n2)cc1C#N CC1CC(c2ccsc2)CN1CC(=O)Nc1ccccc1.c12ccc(cc1)COC2 C1(NC(C(CN(C)C)c2ccccc2)=O)(CO)CCCN(C(=O)CSC(F)F)C1 c1(OCC(=O)NCC2CC(F)(CNC(C=C)=O)C2)cc(F)ccc1F CCC(C(=O)NCC#CC(N1CCC(C2CCC2)C1)=O)C(C)(C)CC C(=O)(C#CC(=O)N(C)C)NCC1CCN(C(C(CC)F)=O)C1 c1(C(=O)NCC(CN(C(C(CC)n2nccc2C)=O)C)C)ccnc(OC)c1 c1(CCC(=O)NC2CC(NC(CCC3CCCN(C)C3)=O)C2)c(O)cccc1F C#Cc1ccc(C)c(NC(=O)C(CCC=C)NC(=O)CC(CC)OC)c1 c1(C(=O)NCC2CC(NC(C3OCCCO3)=O)C2)ccc(-c2ccccn2)o1 CCC(N=c1nc2sccc2c(NCc2nc(C)c(C)o2)[nH]1)C(C)CN(C)C N1(C(C(C2CCCN(C(C3CC(=O)CC(=O)N3)=O)C2)C)=O)CCCN(C)CC1C N1(C(CN2CC(C)(OC)C2)=O)CCC2CCN(C(=O)CCC(C)SC)C2C1 C(C)(CCN(C(=O)C(C)n1cnnn1)C)NC(COCC)=O C1(C(=O)NC(C(=O)NCCC2CCCCCC2)C2CCC2)C2CCC(F)C12 N1(C(CN(C)CC)=O)CCC(NC(=O)CCNc2ccc(C)cc2)C(C)C1 CC(=O)CCCC(=O)NCC1CN(C(=O)CCOC2CCCC2)CC1C CCCCCC(CC)C(=O)N1CCC(CC(C)NC(c2csc(C)c2N)=O)CC1 Cc1ccc(C(N2CCN(C(c3conc3C)=O)C(C3CC3)C2)=O)cc1Br N1(C(CC2(OC)CC2)=O)CCC2(CCC2)C(NC(=O)CN2CC(=O)NC2=O)C1 c1(C(=O)Nc2cccc(S(C)=O)c2)cc2c(s1)C(C)(C)CCC2 c1(C(N2CC(CC=C)(NC(=O)COC3CCOC3)C2)=O)ncnc2sccc12 N1(C(CC(C)(C)OC)=O)CCCC12CCCN(C(C1(CC3CCC3)CC1)=O)C2 Cc1cc(C(N2CCC(N(C)C(c3ocnc3C)=O)C2)=O)c(C(F)(F)F)o1 CC(CO)C(=O)N(CC(C)N(C)C(c1ccc(C(F)(F)F)s1)=O)C c1(OC)ccc(C=CC(=O)NC(C2CCCN(C(c3csnc3Cl)=O)C2)C)cc1 c1(C(N2CCC(NC(C3OCCN(C)C3)=O)C(F)C2)=O)cnc2[nH]ccc2n1 c1(C(=O)NCCCCC2CN(C(C3CCN(C)C3=O)=O)C2)cc(Cl)c(F)cc1F C(CC1CCC1)(C(=O)N1CCC(Cn2ccnn2)C1)NC(=O)C=CC(F)F CC1(NCC2(C(F)(F)F)CC(F)(F)C2)CCOC12CC2(F)F C1(C)(Cc2ccc[nH]2)C(=O)N1.c1(C(=O)OC)csc(SC(C)C(=O)N(C)CC)n1 c1(CNC(=O)CC(CC2CN(C(COCCOC(C)(C)C)=O)C2)C)ccc(F)cc1 N1(C(c2cncc(C(=O)OC)c2)=O)CC=C(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(=O)NCC(C)NC(c2ccc[n+]([O-])c2)=O)c[nH]c2nccc(Br)c12 CCCCC(CNC(=O)C=Cc1cccn1C)NC(=O)C(CN(C)C)N(C)C N1(C2CCC(=O)NCC2)CCc2ncnc(O)c2C1 c1(C(N(C2CCCN(C(c3ccccc3C(N)=O)=O)C2)CC)=O)cc[nH]c(=N)c1 c1(C(N2CCCC(NC(CCC#CC)=O)C2C)=O)oc2ccccc2c1COC C(=O)(C(C)(C)C(F)F)N1CC=CC(C(=O)NC(COC)C(C)C)C1 C1(CNC(CC2(OC)CCCC2)=O)CCC2(CN(C(C3CC4CCC4C3)=O)C2)O1 c1(C(N2C(C(=O)OC)C=CCC2)C(=O)Nc2ccccc2)csc2cncn12 c1(OC)cc(CN2CCC(C)(C(=O)NCCCN3CCCCC3)CC2)ccc1Cl c1(C(=O)NCC2(CO)CCN(C(c3c(C#C)c[nH]n3)=O)CC2)cc(Cl)cc(C#C)c1 N1(C(C(CC)Cc2ccccc2)=O)CCCN(C(C2CCCSC2)=O)CC1 c1(NC(=O)Nc2ccc(OCC(F)(F)F)cc2)cccc(F)c1F C1(C(=O)NC2CN(C(C(CC)SC)=O)CC2(C)C)CCc2nncn2CC1 Cc1c(C(N2CCC(F)(CNC(C3(CCO)CC3)=O)C2)=O)ccc2ccccc12 C1(OC(=N)O)CCN(C(C2(N(C)C(C3C=CCC3)=O)CC2)=O)C1 CCCCC(=O)C(=O)NCC=CCC(=O)NCCC(C)c1cn[nH]c1 Cc1[nH]nc(C(=O)NC2COCCC2C(N2CC(C#N)C2)=O)c1Cl Cc1cccc(OC(C)C(=O)NC2CCC(NC(C3CCCC3CF)=O)CC2)c1 CC1(C)C(c2ccccc2)CN1C(=O)Cc1nc(C2CC2)cs1 CC(c1ccsc1)=CC(=O)NC1COCCC1NC(=O)C(C)(C)c1ncco1 C1(C(C(=O)N(CC(CC)NC(C2(COC(C)C)CC2)=O)C)O)CCOCC1 C1(CC(N2CCC(NC(C(C(C)C)(C)C)=O)CC2)=O)Oc2ccccc2NC1=O C1(C(=O)OC)(C(N2CC(CO)(NC(=O)C(C(C)C)N(C)C)C2)=O)CC2(CCC2)C1 c1(N(C)C)ccc(C(=O)Nc2nc(CC(=O)Nc3cnc(Cl)cn3)cs2)cc1F Cc1cc(C(N2CCC(C(=O)NCC3C4COCC34)C23CC3)=O)cnc1C C1(C(=O)NC2CCSC23CN(C(C2CCOC2)=O)C3)CC(c2cccnc2)=NO1 N1(C(CCc2cnc(C)s2)=O)CCOC(C(C)NC(=O)COCC(C)(C)C)C1 CC(c1ccccc1)=CC(=O)NCC1CCC(C)CN1C(=O)CSCC(F)(F)F CC(C(=O)N(CC(C)(C)NC(=O)CC1CCCC(C#N)C1)C)C(C)(C)C C#CCC(C)C(=O)NCC(C1CC1)NC(c1ccc(Cn2ccnc2)cc1)=O c1(N(CCCNC(C2CCCN2C2CCCC2)=O)CC)ccncc1C#N c1(C(N2C(C3CCN(C(CC(CC)OC)=O)CC3)CCC2)=O)cc(F)ccc1N c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)C(C)OCCC(C)C)nc1 C1(CC(=O)NCCC(=O)N(CC)CC)CN(C(c2ccon2)=O)C(C)(C)C1 c1(C(N2CCC3(C(C(=O)NCC4C(C)(C)COC4)C3)C2)=O)ccn2ccnc2c1 C(=O)(C1=CCOCC1)N1CCC(NC(=O)NC)C1.C123CC1CCN2C3=O C=CCC(C(=O)N1CC(CNC(=O)C=C(C2CC2)C2CC2)C(O)C1)C(C)C CCC(CCC(=O)NCC1(COC)CCN(C(=O)C2=C(Cl)CC2)C1)OC c1(N(C2CN(C(=O)CC3CCOCC3)C2)C)nc(-c2ccsc2)ns1 N1(C(c2ccc(F)cc2)=O)CCC(O)C(NC(c2cnc(C(F)(F)F)s2)=O)C1 Cn1c(O)nc2cc(C(=O)NCCC3=CCCCCC3)ccc12 c1(OCCC2C(C(N(c3c(C(CC)C)cccc3)CC)=O)C2)nc(C)ncc1F C1(C(=O)NCC(C)(C)NC(C(c2ccc(F)c(Cl)c2)C)=O)CCc2ncnn2C1 C1(C(=O)NCc2nccc(C)c2)CC12CCN(C(=O)Nc1ccccc1)C2 c1(OCCOC)cc(C)ccc1CNC(=O)NCCC1CC(F)C(=O)N1 N1(C(c2c(C)coc2C(C)(C)C)=O)CCC(C)C(NC(C2C3(CC3)C23CC3)=O)C1 C(=O)(CC(C)(C)c1cccc(Br)c1)NC(C(CO)NC(C(F)=CC)=O)C C(C(=O)NC1CN(C(=O)Cc2conc2C)CC1C)(C(C)C)(C(C)C)NC(C)=O N1(C(c2c(N)non2)=O)CCCC12CCN(C(C1CCc3ncnn3C1)=O)CC2 C1(C(N(CC(=O)NCCc2coc(C)n2)CC#C)=O)CCOC1C(C)C C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)C2=CCSC2)CC12CCOCC2 CC(=O)CCCC(=O)NC(CNC(=O)COc1cccnc1)C(C)C C1(NC(C(c2ccccc2F)(C)OC)=O)CCC(C)N(C(=O)C2=COCCC2)C1 S(=O)(=O)(c1ccc(Br)cc1N1CC2CCCN2C(C(C)C)C1)N(CC(C)C#N)C C12(C(=O)NCCC(C)N(C(c3cnn(C(C)C)n3)=O)C)CCC(CC1)C(C)(C)O2 c1(NC(N2C(C(=O)Nc3ncc(C)cc3O)CC2)=O)ncc([N+](=O)[O-])cc1Br C1(CNC(C=CCCC)=O)CCCN1C(=O)C(C)c1cncs1 CC(F)(F)CCCC(=O)NC(C)(CNC(C1C2COCC12)=O)C1CC1 c1(C(N2CC(N(C(c3cnc(C)s3)=O)C)C(F)C2)=O)cnn2ccncc12 c1(C(C)NC(=O)NCC(C=C)(F)F)cccnc1F C1(CC(=O)NCCCCN(C)C(C2CCCC2O)=O)CCNC1=O c1(C(=O)NNc2cccc(Cl)n2)ccc2c(c1)CNCCN2 C1(NC(C2C(C)(C)CO2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(C(C)OCOC)=O)C2)cncc(-c2ccoc2)c1 c1(NC(C2N(C(C=C(C)C3CC3)=O)CC(F)C2)=O)cccc(N=[N+]=[N-])c1 CC(=O)CCN=C(NCC#Cc1ccccc1Cl)NCc1noc(C(C)(C)C)n1 N1(C(c2n(C)cnc2)=O)CCCC(CNC(=O)CCc2ccc(Br)cn2)C1 Cn1ccc2ccnc(C(N3CCC3CNC(C3CC4CCC(C3)S4)=O)=O)c12 CC(CC(=O)NC12CCC(CC1)N(C(=O)C(c1ccc(Cl)s1)C)C2)CC(F)(F)F C(=O)(CCCCCCC(=O)OC)N1C(CNC(CCC=CC)=O)CCCC1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CC(NC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCCC2(C1)CN(C(=O)CSCc1ccccc1)C2 C1(C(=O)NCc2ncc(CC)s2)(NC(=O)CCC2CCCC2)CCCC1C CC(CCCC(=O)NC1(C)CCCN(C(c2ccc[nH]2)=O)C1)c1ccccc1 c1(C(C)=O)ccc(CNC(=O)N(C2CS(=O)(=O)CC2O)CCO)c(F)c1 c1(CC)cc(C(=O)NCC2C(CC)CCN2C(C2C=CCC2)=O)oc1CC C1(NC(C(Br)=C(C)C)=O)CC2CCC(C1C)N2C(c1ccc(CO)cc1)=O C(=O)(C(CNC(=O)CCc1nccn1C)N(C)C)N(CCOCC)C c1(C(=O)NCC2(O)CCCN(C(CNC(=O)OC)=O)C2)cc2cc(Cl)ncc2[nH]1 c1(C(N(CC(CC)(C)Cl)c2ccccc2)=O)cc(C(F)(F)F)cn1C CCCCCCC(CC)C(=O)NC1CC1CNC(=O)Cc1cc(SC)nn1C c1(C(=O)NC(C(N2CC(C)CC(OC)C2)=O)C(C)CC)cccc2[nH]ncc12 N1(C2CCC(NC(=O)NC(C)C(=O)N(C)C)C2)CCN(Cc2ccccn2)CC1 CCCC(O)CC(=O)NC(C)CNC(c1cn(-c2cccc(F)c2)nc1C)=O c1(C(=O)NC(CC)CN(C)C(c2c(C)coc2COC)=O)ccc(F)cc1N N(C1CCc2cccn21)C(C1(C)N(Cc2ccc(C)o2)CC1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C1CN(C(Cn2nc(C)n(C)c2=O)=O)C1)C C1(F)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CCN(C)CC1 CCCCC(C(=O)NC(CN(C)C)C(=O)NCCC(C)(C)N(C)C)N(C)C S1(=O)(=O)C(C(F)(F)F)N1.n1(CCC(=O)OCC)cc(C2(O)COC2)nn1 C1(C2CN(C(=O)CCCNC(c3ccsc3)=O)C2)(NC(CN(C(C)C)C)=O)CC1 C#Cc1cccc(C(=O)N(CC(=O)NCC2CC2Cl)C(C)C)c1C CC1Cc2sc(C(=O)NC3CC(NC(c4cnc(O)cc4O)=O)C3)cc2C(C)C1 CC1=CC(C(=O)NCc2ncoc2CCNC(=O)CC(C)C2CC2)SC1 c1(C(c2n(CC(=C)C)nnn2)NCC(Cc2ccco2)CO)cncc(C=C)c1 c1(CC)ccc(OCC(=O)NCCOC2CN(C(c3csnn3)=O)C2)cc1 Cc1cc(NC(C(C)NC(C2(C)CC3(CC3)C2)=O)C(C)C)nc(C(F)(F)F)n1 C(=O)(C(F)(F)C(F)F)N1CCC(N(c2cnc[nH]2)C(=O)COC(F)F)C1 S(=O)(=O)(c1cccc(=NC(C)c2ccccc2Br)[nH]1)NCc1cc(OC)no1 c1(C(=O)NCC(CC)NC(C2(COC)CC=CCC2)=O)cnc2cccnn12 Cc1ccc(F)cc1C(N1CCC(O)(C(=O)NC(C2CCOC2)C)C1)=O C1(C(=O)NCC(CC)(CC)NC(=O)CCCN(C)N=O)CCC2(CCCO2)CC1 C1(CCNC(COc2ccc(C)cc2)=O)C(C)CCCN1C(c1nnn(C)n1)=O C1(NC(C(CC)OC)=O)CC(N=c2cc(Cl)nc(S(C)(=O)=O)[nH]2)C12CCC2 C1(NC(C2CCN(C(=O)C(=O)Nc3ccc(Cl)cc3)C2)C)CN2CCC1CC2 CC(C)C(C)(C)C(=O)NC(CNC(=O)C(C)OCC1CC1)CO c1(NCC)cncc(C(=O)NC(C2CN(C(C3CCC(C(N)=O)O3)=O)C2)C)c1 C(=O)(C(C)(C)CF)N(CCCCCNC(C1C(C)(C(C)C)C1)=O)C c1(C(=O)NC2C(CNC(c3ccc(C4CC4)s3)=O)C2)cccc2nc(S)oc12 C(=O)(C(C)(C)C(=O)N(CC(C)N(C)C(c1cc(SC)oc1C)=O)C)NC C1(NC(COc2cccc(C#C)c2)=O)CC2CN(C(C3(C)CC3)=O)CC2C1 c1(CNC(CCC2(NC(CC(C)n3cccc3)=O)CCCC2)=O)cccc(F)c1 C1(C(N(CCCNC(=O)C(C)(F)F)CC)=O)CCCCC12CCC2 c1(C(=O)NCCC=C(C)C)ccc(C2CC2)o1 C1(CC(=O)NCC2N(C(c3c(COC)scc3)=O)CC2)CCCCC1F C(CN=c1nc2sccc2c(N(C)Cc2cc[nH]n2)[nH]1)n1c(C)ncc1 C1(NC(c2cnccc2Cl)=O)CN(C(=O)CCCCC2CC2)C2(CCCCC2)C1 CC1c2cc(Cl)c(Cl)cc2CCN1C(c1cncc(C(N)=O)c1)=O C(=O)(C(F)CC(CC)CC)NCC1CCC(NC(C(C)OCCCC)=O)C1 C1(N(C)C(=O)Nc2cccc(C(F)C(F)(F)F)c2F)CC(C)(C)OC(C)(C)C1 C=CC(C)(O)CC(=O)N(C(C(=O)O)C(C)C)C(C1(O)CCCCCC1)C1CC1 C1(NC(c2cc(C)nc(C)c2)=O)CCC12CCN(C(=O)C1=COCCC1)CC2 Cc1c(Cl)ccc2[nH]c(C(=O)NCC(F)CNC(c3c[nH]c(=N)o3)=O)cc12 c1(NC(C2(COC)CN(C(=O)Cc3ccc(C)cc3)C2)=O)nccc2occc12 C1(C(C)C)CN(C(c2cncnc2)=O)CCN1C(=O)Cc1cccc(Br)c1 Cc1cccnc1CC(=O)NC(C)C(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O c1(-c2c(C)cccc2)nc(=NC2CN(C(C3CCCOC3)=O)CC(C)(C)C2)s[nH]1 c1(C(C)C(N2CCC(N(C(=O)C=CCOC(C)(C)C)C)C2)=O)cccc(F)c1 C(=O)(C(C)C(C)NC(=O)C(CCSC)NC(c1cc(C2CC2)on1)=O)OC Cc1cccc2[nH]c(C(N3CC(O)CC3C(=O)NCCc3nn[nH]n3)=O)cc12 c1(C(=O)NC2CN(C(=O)C(=O)C=Cc3cccs3)C2)ccc(-n2ccnc2)nc1 C#CCC(CC#C)C(=O)N(C1CC2CCC(C1)N2C(C12COCC1C2)=O)C N1(C(c2ncc(C)nc2)=O)CC2CC(NC(c3cncc(Cl)c3Cl)=O)CC2C1 Cc1c(NC(=O)CC2CCCC2NC(=O)CNC=O)cnn1CCO CCC(C(=O)NCC1(F)CCN(C(c2c(OC)ccnc2O)=O)C1)C(C)(F)F CN(C1CCCC1O)N(CC1CCOCC1)CCC(F)F N1(C(CCCCN(C(C)=O)C)=O)CCN(C(C2CCCC(O)C2)=O)CC12CC2 C1(CNC(C2OCC(C)(C)C2)=O)CCN(C(c2cnsc2)=O)C12CCC2 c1(COCCC=C)ccc(SC(C)C(=O)OC)cc1 C1(NC(C(CC)C)=O)(CNC(c2cc(OC)ncc2F)=O)Cc2ccccc2C1 c1(C(=O)NC(CC)CNC(=O)C(CC)C(F)(F)F)cnc(P(C)(C)=O)cn1 c1(C(=O)NCC(C)N(C(c2csc(C(C)OC)n2)=O)CC)ccnnc1O c1(CCCN=C(NC(CC)C)NCc2nnn(C)n2)c[nH]c2ccc(F)cc12 N12CCC(CC1)C(=O)NC(C)CN(C)CC2=O.c1(C2C(C(N)=O)C2)cccs1 c1(NC(c2ncn(CCNC(CC(C)SC)=O)c2)=O)cccnc1C Cc1cc(CC(=O)NCCC(O)CNC(c2cccn2-c2ccccc2)=O)n[nH]1 CCC(CC(=O)NCC1CC2CCC1N(C(C1(C)CCC1)=O)C2)C(F)F CCC(CC)C(=O)N1CCNC(C(N2CCC(N3CCCC3)CC2)=O)C1 C#CCC(C(=O)NCC=Cc1ccccc1)NC(=O)C(C)CC=CCOC c1(OC)ccc(F)c(C(=O)NCC(F)CNC(C2CCSCC2)=O)c1F c1(C(N2C(CNC(CC(C)c3cccnc3)=O)C=CC2)=O)ccn2ccnc2c1 Cc1ncc2ccc(C(=O)NC3CC4CC(NC(c5ccncn5)=O)CC34)cn12 CC1(C)CCCC1CNC(C1OCCC1NC(=O)C(O)c1ccco1)=O C(CC(C)CC)(C(=O)NCc1nnn(C)n1)NC(C=CC)=O O=C(CCCC(F)(F)CO)NCCC1CCCN(C(=O)CC2CCCC2)C1 c1(C(=O)NCC23C(CN(C(Cc4cnc(C)s4)=O)C2)C3)cnc2[nH]cc(C)c2c1 C1(C)(CNC(C=COCC)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(NC(c2ccc(C(F)F)c(Cl)c2)=O)CN(C(=O)C#CC2CC2)CC2(CCC2)C1 C1(CC)CN(C(C2CCCSC2C)=O)CC1C(=O)NCC(C)(C)C(N)=O C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)C(NC(C)=O)=Cc2cccs2)C1)NC N1(CC(N2CCN(C3CCN(Cc4ccc(F)cn4)C3)CC2)=O)C(=O)CNC1=O c1(C(=O)NC2C(F)CCN(C(c3cn(CC=C)nn3)=O)C2)cscc1S(C)(=O)=O C1(C(=O)NCCc2cn(CC)nn2)C=CCN(C(=O)CCn2ccnn2)C1 c1(C(=O)NC(CC)CCOC)cccnc1CNC(=O)CC1CC2CC2C1 c1(NC(C2N(C(c3cnn(C)c3C(F)(F)F)=O)CCOC2)=O)ncc(Cl)cc1F C(C(CC(=O)NC1CCCNC1=O)C1CCC1)NC(c1cc(C2CC2)on1)=O N1(CC)CCC(C(N2CCC(n3cc(NC(c4ccccc4)=O)nn3)C2)=O)CC1 c1(CC(=O)OCCCC2(C(=O)NCCNC(C)=O)CC2)ccn(C(F)(F)F)n1 n1(CC)nc(C)cc1C(=O)NC1C=CC(CNC(=O)CCCOC(C)(C)C)C1 c1(C(NNC(N2CCCS2(=O)=O)=O)=O)cc2c(s1)-c1ccccc1OC2 C1(NC(C(COC)(F)F)=O)CCN(C(c2c(F)cncc2Br)=O)CC1C N1(C(COCc2n(C)ccn2)=O)CCC2CC2(NC(=O)CCCN=[N+]=[N-])CC1 N1(C(C(C)N(C(C)=O)C)=O)C2CC=C(C(=O)N(CCCN=[N+]=[N-])C)C1CC2 C=CC1(CC(N2CC(O)CC2CNC(=O)C(C)(C)c2ccsc2)=O)CCCCC1 C1(NC(c2ccc(OCCF)cn2)=O)CC2CC1CN2C(=O)C(O)c1ccsc1 C(CO)(CCCCNC(c1ccc(SC(F)(F)F)cc1)=O)NC(CCSC)=O c1(C(=O)NC2C(C(=O)NCc3c(OC)cccc3)C2)cccc(Cl)c1OC c1(CNC2C(C(N(CC(O)CO)C(C)C)=O)C2)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CC(NC(=O)Cc3cc(C)no3)CC2C)=O)cc(C)c1 c1(C(=O)NCC2C3CC2N(C(=O)CCCc2ccncc2)C3)cc(F)cnc1O C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(=O)Cc1[nH]cnc1C C1(Cc2cn[nH]c2)C(=O)OC(=O)CCN1C.c1cn[nH]c1.C1CCN1.C1(O)CCC1 c1(C(N(CC(CNC(CC2(OC)CC2)=O)O)C)=O)c(Br)cnn1C C1(C(N(C)CC2(NC(=O)Cn3ccc(Br)n3)CC2)=O)CCc2nn[nH]c2C1 c1(CC)cnn(C)c1C(C(=O)NC(C)C(=O)OCC)N(C(C)CCC)C1CC1 C1(c2nnnn2C(C)(C)CC)(NCC(=C)Br)CCC(P(C)(C)=O)C1 c1(C(N(CCC(C)NC(CS(CC)=O)=O)C)=O)nc2ccccn2c1F CC1CN(C(=O)CCc2cnn[nH]2)CC(C)N(C(=O)CC23CCC(CC2)CC3)C1 c1(CC)c(C(=O)NCC23CC(NC(=O)C(C)C(F)F)(C2)C3)[nH]c2ccccc12 c1(OC)nc(C(=O)NCC2CCCCN2C(=O)C=Cc2nnn(C)n2)sc1C N1(C(c2nn(CC)c(O)c2)=O)CC2CCCC(C1)N(C(c1ccns1)=O)C2 C(CC(O)C(F)(F)F)NC1CN(C(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)C1 CCC(C)CC(C)C(=O)N1C2CCC1CN(C(c1n[nH]c(C(C)(C)C)n1)=O)C2 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCC(C)NC(C1CC(CCC)C1)=O)C N1(C(C(c2c(C)cccc2C)O)=O)CCOCC(F)(CNC(=O)C2CC2)C1 C1(NC(CN(CCC)C)=O)C(CNC(=O)CCOCC)C1(C)C C1(NC(CC=C)=O)CN(C(=O)Cc2ccc(C)c(C)c2)C2(CCCOC2)C1 c1(C(N2CCC(O)(C(C)NC(c3ccnn3C)=O)CC2)=O)ccc(F)c(Cl)c1N CC(CCC(C)(C)C)C(=O)NCC1CCCCN1C(c1cnoc1)=O Cc1cnc(C(=O)NCC(CO)NC(c2csc(C)c2C)=O)cc1Br N1(C(C(F)=C(C)C)=O)CCN(C(=O)CCC(N)=O)C(CF)C1 C12(C(=O)NCC3(CNC(C(C)NC(N)=O)=O)CC3)CCC(C)(CO1)C2 c1(C(N(CCCCCCNC(C2COCCO2)=O)C)=O)cncc(C(C)(C)C)c1 C1(C(N2CCC(NC(c3c(CC)con3)=O)(CF)C2)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NC(C2CCCN2C(C23CCC2CC3)=O)C)c(C(F)(F)F)o1 C1(NC(C(C)C2CC2)=O)COC2(CNC(c3c[nH]ccc3=N)=O)CC1C2 C(C1CCC(c2nnnn2C(C)C)(NC(c2c(Cl)cccc2Cl)C)C1)=CC(=O)OC CC1(CNC(c2ccncc2)=O)CCCN1C(=O)COC1CC1(F)F C12(CNC(C(C)SCC)=O)CC(NC(c3cnc(CC)[nH]3)=O)(C1)C(C)(C)O2 c1(CCC(=O)NCC2CCC(NC(COCC=C)=O)CC2)ccc(C(F)F)cc1 C1(NC(c2cccc(OC)c2)c2ccc(OC(F)F)cc2)CCC2(CNC2)OC1 C12(CNC(CCCNS(C)(=O)=O)=O)COC(CNC(=O)C(F)=C3CCC3)(C1)C2 Cc1cc(C(=O)NCCc2ocnc2CNC(C2CCCC23CC3)=O)nc(O)c1 Cc1c(CC(N2CC=CC(NC(c3cnns3)=O)C2)=O)ncn1C Cc1cc(F)ccc1CC(=O)N(CCCNC(C1CC1C(F)(F)F)=O)C c1(C2(NC(N3C(C)(C)C(c4ccccc4F)CC3)=O)CC2)ccc(F)c(F)c1F CC1CC(NC(c2ccc(F)s2)=O)CCN1C(C1CC2CC2CC1C)=O c1(C(=O)NCCC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc(O)nc(O)c1 C(=O)(C(O)C(C)(C)C)N1CC(O)(C(C)NC(C2CC(N3CCOCC3)C2)=O)C1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2c[nH]nc2OC)=O)C1 Cc1ccc(C(=O)NCCC2(O)CCN(C(=O)C(C)P(C)(C)=O)CC2)nc1O C1(NC(c2cncc(N)n2)=O)CCCCN(C(c2cncc(C(F)(F)F)n2)=O)C1 O=C(C#CC1CCCO1)NC(c1cccc(Cl)c1)CNC(c1cnc(O)o1)=O c1(C(N(CCn2cc(CC3CCC4(CC4)C3)nn2)CC)=O)cccc(OC)c1Cl N1(C(CCCNC(C2CC(C)(C)C2)=O)=O)CCCN(C2CC2)CC1 c1(C(=O)NCCCN(C(=O)Cc2ccn(C)n2)C)cncc(OCC(F)F)c1 c1(CNC(=O)NC(C)CCC(F)(F)F)cnc2ccccn12 O=C(C1OCCn2ccnc21)NC12CC1CN(C(=O)Cc1cnn(C(F)F)c1)C2 C1(C(=O)NC(c2csnn2)C)CC2(CCN(C(=O)CN3CCNC3=O)C2)C1 N1(C(C(C2CCN(C(C3OCCOC3C)=O)C2)C)=O)CC2(CCC2)C1 c1(C(C(=O)NC)N(C2CN(C(=O)OC(C)(C)C)C2)C)ccccc1[N+](=O)[O-] CC1CCC(CNC(=O)CCSC(F)(F)F)CN1C(c1nnc(O)nc1O)=O C1(CNC(C(CCN(C)C)O)=O)(NC(=O)Cc2ccc(Cl)s2)CCCCC1C n1(CCC(=O)NC(CC)CNC(C2Cc3nnsc3S2)=O)c(C)cc(O)cc1=O C(=O)(C(O)C1=CCCCC1)NC1(CNC(c2cc(F)c[nH]2)=O)CC(OC)C1 c1(COCC)nc(N2CCC(C(C)NC(=O)C(C)CCN(C)C)CC2)cc(Cl)n1 c1(OC)cccc(C(F)F)c1C(=O)NCC1(NC(=O)C(CC(C)C)N(C)C)CC1 C(=O)(C(CCC1CCC1)NC(c1cccnn1)=O)N1C(C)CC1 C1(OC)CCC2(CCN(C(=O)C(C(C)(C)C)NC(=O)C(=O)NC3CC3)C2)C1 C1(C(=O)NCC(CNC(=O)C(F)(F)c2nccs2)OC)CC2CCCC12 c1(OCC)ccc(C(=O)NCC2(N(C(=O)C=CCO)C3CC3)CCOC2)cc1 N1(C(C(C)CN2CCOCC2)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC12 C(CC(C)C)(CC(C)C)NC(CCC(C)NC(c1c(OC)nn(C)c1)=O)=O N1(C(c2c(CC)cnn2C)C(=O)NCC2CCCO2)CCN(C)CC1CC(C)C c1(OC)ccc(CCC(N2CCC(C)(CC(=O)Nc3cc(O)ccn3)C2)=O)cn1 c1(C(=O)NC(C2CCCN(C(=O)CC3CCCOC3)C2)C)cnc2cccnn12 CCCCCCC(C)CC(=O)N1CCCCC(NC(=O)C(C2CCC2)OC)C1 N1(C(CC=C=C)=O)CCC2(CC(NC(=O)C(C)CSC)C2)C1 c1(SC)ccc(N)cc1C(=O)N(C)CC1(O)CCN(C(=O)C2CC2)CC1 c1(C(=O)OC)cc(SC)ccc1NC(N1CC(C(F)(F)F)CC1C)=O c1(C(=O)NC2(CCCC(=O)N3CC(C(CC)C)C3)CCC2)cc(O)ncn1 CC1CCN(C(C2CCC=CC2NC(=O)Cc2cnoc2)=O)CC1O c1(CSC(C(C)O)C)nc2cc(Cl)ccc2n1C C(=O)(NN1CCCC1C(=O)NC1(C)CS(=O)(=O)C1)c1cc(C)c(C)o1 Cc1cc(N)c([N+](=O)[O-])c(N2CCOC(CC(F)(F)F)C2)n1 c1(C(C)C)c(C(=O)NCC2CC3CC3N2C(=O)CO)cnc2ncnn12 C1(C(N(CCCC#C)C)=O)(NC(c2[nH]cc(C)c2C)=O)CCC(C)(C)C1 C#Cc1ccc(F)c(NCC(O)CCc2ccccc2)c1 C=Cn1nccc1C(=O)NCC1CC1CNC(C1(Cl)CC12CCC2)=O S(=O)(=O)(c1cccc(C(C)C)c1)Nc1c(C)ccc(C(=O)OC)c1 C12(NC(C34CC(COC)(OC3)C4)=O)CCC(CC1NC(=O)Cn1cc(C)cn1)C2 Cc1ccc(C(N2CC(NC(=O)CC34CCC(CC3)C4)CC(C)C2)=O)c(F)c1C c1(Cn2c(C(c3nnnn3C(C)C)NCc3c(C)ncs3)ccc2)cccc(F)c1 C(=O)(C(C)(CO)NC(c1ccc(C)cn1)=O)NCC(CCC)O C1(COC)(NC(=O)C=Cc2cnc[nH]2)CN(C(=O)C(Cc2ccsc2)NC=O)C1 c1(C(N2C(C)(CNC(=O)CS(N)(=O)=O)CCC2)=O)ccc2oncc2c1 CC(c1ccccc1)=CC(=O)N(C)CC1CCCN1C(=O)CCc1cnc(O)[nH]1 C1(NC(c2ccsn2)=O)C=CCCC1C(=O)NC1COCC1F Cn1cc(C(N2C(CNC(C3CCCC3O)=O)CC3CC23)=O)c2cccnc12 C1(NC(c2ccc(C)c(Br)c2)=O)CN(C(C2COC2)=O)C2(CCC2)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2CC(NC(c3ncccc3OC)=O)CC2C1 C(=O)(CC(C)CCCCCC)N1CC(CCC)N(C(c2ccn(CC)n2)=O)CC1 c1(C(=O)NCCOCCNC(C2(C)N(C)CCC2)=O)ccc(=O)n(C(C)(C)C)n1 C12(NC(CN(C(CC=CC=C)=O)C)=O)CC3CC(CC1C3)C2 CCC(Cc1cn(CC(C2CC(C)N(C(=O)OC(C)(C)C)C2)O)nn1)C(=O)O c1(-c2nc(C3(C(C)C)CNC(=O)C3)on2)cc(F)ccc1F N1(C(C(=O)NCCCC)=O)CCC2CCN(C=O)CC2C1.c1(C(CN)=O)cnc[nH]1 C1(NC(C(CC)CN(C)C)=O)CC2CC1CN(C(C1CC(CC(C)(C)C)C1)=O)C2 C1(CNC(C(N2CCCCC2=O)C)=O)CN(C(C2COCCO2)=O)CCC1C c1(OC)nc(N2CCC(C)(NC(=O)CC3CC(F)(F)C3)CC2)cc(C)n1 c1(CN2C(C(N3CCOCC3C(F)(F)F)=O)CC(C)C2)ccc(Br)cc1[N+](=O)[O-] C(=O)(N=c1ncnc2[nH][nH]c(Br)c1-2)c1c(-c2cccc(C)c2)cccc1 C1(CC(=O)NCCOC2CCOC2)CCCN1C(C1(CCO)CC1)=O N#Cc1ncc(C(=O)NCCN(C2CCCCCC2)C(c2ccoc2Cl)=O)s1 CC1(NC(c2ncsc2Br)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(NCC(=Cc2ccc(Br)s2)C)nc2ccc(Br)c(C)n2n1 CC1CN(C(=O)C=Cc2ccc[nH]2)CCN1C(C1CC(=C2CCC2)C1)=O CCCCC(CC)CC(c1nnnn1C)NCCCc1nnc(C)s1 C1(C(N2CCC(N(C(C(CC)n3cncn3)=O)C)C2)=O)(OC)CCC(C)(C)CC1 c1(CCC(=O)NC2C(C)N(C(c3csnn3)=O)CC2)nc2cnccc2[nH]1 C1(C(N2CC(N(C)CC)C2)=O)CCC(C(C)C)N1C(=O)COCC(F)F c1(C(=O)NCC2(C)CCN(C(C34CC3C4)=O)C2)ccc2ccncc2c1.CCCC c1(CN2C(C(=O)Nc3c(C(N)=O)ccs3)C=CC2)cnc2[nH]ccc2c1 C1(NC(c2ccnnc2S)=O)CCN(C(c2cn(C(F)F)cn2)=O)CCC1CO C1(C(N2CC3C(NC(=O)C(O)C4CCC4)(C3)C2)=O)CC2(CCCCC2)C1 C1(C(=O)NC2C3CN(C(C4CNC(=O)N4)=O)C2C3)CC2COCCN2C1 c1(OC)ccncc1C(=O)NC1CC1NC(=O)CC(C)c1cccnc1 N1(C(COC2(C)CCCC2)=O)CC2(NC(=O)CCc3cncc(F)c3)CC1C2 N1(C(CC(C)F)=O)CCC2(CC1)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 c1(CCOC)n[nH]c(=NC(=O)C2(C#N)CC3C=CC2C3)s1 c1(C(=O)NC(CNC(CC(C)CF)=O)(C)C2CCC2)cccc2ncccc12 C(=O)(CCCC(F)F)N(C1CCN(C(C(C)O)=O)C1)CCO C(CC(=O)N1CC(O)CCO1)C1N(C(Cc2cc(C)[nH]n2)=O)CCCC1 c1(C(=O)NC2CCCC(CNC)C2)nn2c(c1I)CCCC2 c1(OC)ccc(CN(C)CCN(C(=O)CC2CCCC(C)C2)C)cc1 C1(C(N2CCC(CC)C2)=O)(CC)CCN(C(c2csc(CO)n2)=O)C1 N1(C(C)C)CCCC1C(=O)NC(C(=O)NCc1cccnc1)C1CC1 c1(-c2c(C(=O)NCC3CN(C(CCC)=O)C(C)C3)cccn2)ccc(F)c(F)c1 c1(CC(=O)NCCN(C(C)C)C(C2CCC(C)O2)=O)cccc(Cl)c1Cl C12(CNC(c3cn(C)c4c3cccn4)=O)CCCCC1N(C(=O)C=CBr)CC2 CC(C)CC(C(=O)NCC1CC12CC2)ONC(=O)C(C)N1CCCCC1 CN=c1[nH]c(=NCC2CCCCN2CCO)[nH]c(=NC2CCCCCC2SC)[nH]1 c1(C(N2C(C)CCC(NC(CC(=O)NC)=O)C2)=O)cccc2c(C)c(C)[nH]c12 c1(CC)cc(NC(=O)CC(C)CNC(c2ncoc2C)=O)cc(C)c1 C1(CC(=O)NCC2(C)N(C(COC)=O)CCC2)CC(c2ccccc2)=NO1 C1(c2nnnn2C2CC(F)(F)C2)(NC2(CC)CC2)CCCC(CC2CC2)C1 Cc1cc(C)n(CC(N2CC(C(C)NC(c3cnn(CC(C)C)c3C)=O)C2)=O)n1 CCC(CC(=O)N1CCCCC1c1cn(Cc2[nH]nnc2C)nn1)C(C)C N1(C(c2nc(C)sc2)=O)CCC2(CCCN2C(c2ccc(F)cc2Br)=O)C1 c1(OC)cc(OC)cc(CN2CC3CC3(C(N3CCCCC3CCCO)=O)C2)c1 c1(OC)cc(CNC(C2C=CCN2C(=O)CCC2CCCC2)=O)ccc1F Cc1cccc(OC(C)C(C)NCc2ncc(C3OCCO3)s2)c1 C1(CNC(COCC)=O)CC(CNC(c2sccc2Br)=O)CO1 C(C1=NOC(C)C1)N(CC(F)C(=O)C(C1(C(CC)=O)CC1)=O)C.C c1(C(=O)NCC2CC2NC(C2CCOCC2)=O)cccc(F)c1F c1(SCC(N2CCC(O)C2c2ccccc2)=O)cc(Cl)nc(Cl)c1 c1(CC)oc(C(N2CCC(CNC(C3(C)CCCS3)=O)C2)=O)cc1C(=O)OC N1(C(C=C(COC)C)=O)CCOC2(C1)CN(C(c1cncc3c[nH]nc13)=O)C2 S(=O)(=O)(c1ccc(N2CCN(C=O)CC2)c(Cl)c1)NCc1c(C)cc(Br)cc1C c1(SC)ncc(C(N2CC3CC(NC(=O)CCc4ccsc4)C2C3)=O)c(O)n1 c1(C(=O)NCCN(C)C(c2cccc(F)c2)=O)ccccc1OC(C)(C)C Cn1ncc2c1CC(CCC(=O)NCCC1CC(NC(=O)C(F)F)C1)CC2 c1(CSCC)cccc(C2(C)CC2)c1.C(C)(CCNC(C1CCC1)=O)N(C=O)C Cc1ccc(-n2nc(COc3ccc(C(C)(C)C)cc3)nc2-c2ccc[nH]2)cc1Cl N1(C(CCNC(C2CCC2)=O)=O)CCC2(NC(C3C=CCC3)=O)CCCCCC12 N1(Cc2ccccc2)CC2(CC(NCC3COC4(CCCC4)O3)c3nccn32)C1 N1(C(C(CC)NC(C)=O)=O)CC2CCC1CN2c1nccc(SC)n1 C1(C(=O)O)(CNCCc2ccc(C)nc2)CCCCCCC1 Cc1cnc(C(=O)NCC#CCNC(=O)C(C(C)(C)C)n2ccnn2)cc1C#N C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CC2(C1)CC(NC(=O)C(Cl)=CCl)C2 c1(SCC(=O)N(C2CCCN(C(=O)C(F)(F)COC)C2)CC)ccc(O)cc1 c1(C(=O)NCCC2CCCN(C(c3sc(Cl)nc3Cl)=O)C2)cc(Br)c(O)c(Br)c1 C1(C(=O)NC(C2(CNC(=O)C(c3ccc(F)cc3)(F)F)CC2)C)CCS(=O)(=O)C1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(=O)CC2CNC(=O)C2)C1 N1(C(CC2C(CC)C2)=O)CCC(CC(=O)NCCC(C)C(C)(C)C)C1(C)C CC(CC(=O)N1CC(O)(CNC(=O)C=CCN2CCC2)C1)c1cnn(C)c1 c1(C2C(C(=O)NCC(c3cccc(Cl)c3)CO)CNC2)ncc2c(n1)CCC2 C1(N(C(=O)OC)C)CCCN(Cc2ccccc2)C1=O.c12nc(n[nH]1)NC2=O N1(C(CCOC)=O)CCCC(C2CCCCN2C(=O)C(C)OCC)C1 c1(N2CCC(C)C2)nc(N(C)Cc2cc(Br)cn2C)c2c(n1)CSC2 c1(OC)ccc(CN2CC(F)CC2C(=O)NCC2CNC(=O)CO2)c(Cl)c1OC Cc1nc(C(=O)OC(C)(C)C)ccc1C(=O)O.C1C(C)(C)CC(=O)NCC1 C1(C)(CNC(C=COCC)=O)CN(C(=O)COCc2nc(C3CC3)no2)CC1C N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 CCC(C)CCCC(=O)NC(Cc1ccc(Cl)cc1Cl)C(=O)NCCOC(C)C c1(C(N(C(C)CNC(c2c(Cl)cccc2Cl)=O)C)=O)cc(F)cc2ccncc12 C(=O)(CC(C(F)(F)F)c1nccn1C)NC(CC)CNC(=O)CCOCC(C)C C1(C(N2CC(NC(C3=C(C)OCC3)=O)C(O)CC2)=O)CCOCC12CCCCC2 Cc1ncccc1CN1CCOCC1C(=O)Nc1cc(-c2cccc(Br)c2)no1 C1(NC(C(COC)C)=O)CN(C(C2(Cc3ccc(F)cc3)CCC2)=O)CC1O N1(C(C(=O)NC(CC)C)CCCc2ccccc2)CCc2c(F)ccc(O)c2C1 Cc1cc(C(=O)O)c(-c2nccn2Cc2ccc(C(N)=O)cc2)cc1C C(=O)(C(C)C(CC)CC)NC1(C2CN(C(c3cc(CC)c(C)cc3)=O)C2)CC1 N1(C(C2CCCN2C(c2cc(Br)no2)=O)=O)CCC(NC(C2CCOC2)=O)CC1 c1(CC)ccc(N)c(C(=O)NCC2CN(C(c3ncncc3Br)=O)C2)c1 C1(NC(=O)CCOCC(F)(F)F)CN(C(C2CCCNS2(=O)=O)=O)CC1C1CC1 c1(OCC)cccc(CN2CC(C(=O)OCC)C2C(=O)OC(C)(C)C)c1 N1(C(C2CCCN(Cc3onc(CCCC)n3)CC2)=O)CCOC2COCCC12 C1(NC(C=C(C)C(F)F)=O)CCCC12CCN(c1nccnc1C#N)CC2 N1(C(CCC(C)NC(CC2(CSC)CC2)=O)=O)CCn2c(cnc2C)C1 N1(C(C(CC)N(C)C)=O)CC(OC)CC1CCNC(c1ccc(C)o1)=O CC(C)C(C(=O)N1CCCC(C)C1)NS(=O)(=O)C1(C)CC1 C(=O)(CCCCC(=O)N1CC2(COC(CNC(=O)C(F)(F)CO)C2)C1)OC N1(C(C2CC(C#N)(O)C2)=O)CCc2ccccc2C1CNC(C1CC=CCC1)=O N1(C(=O)C(=O)NC2CCC(N3C(C)CCC3C)CC2)CCC2NCCCC2C1 C(C1CCCCCC1)=CC(=O)NCC(C)(C)CNC(=O)COCCF c1(CC)ccnc(C(N2CCOCC2CNC(=O)CCN(C)CC)=O)c1 C1(C(=O)NCC(C#C)CC)CCN(C(=O)C2=CCCCC2)CC1C N1(C(C(C)OCCC#C)=O)CCN(C(=O)C(C)(C)CF)CC1C1CCCC1 C1(C(=O)NC2CCC(CNC(C3CC=CCC3)=O)C2)Cc2cscc2C1 N1(C(C(CC)C#N)=O)CCCN(C(=O)C(O)Cc2c(F)cccc2Cl)CCC1 C(CC(CC)C(=O)N(C)CC1(NC(c2oc(C3CC3)nc2C)=O)CC1)=CC C1(CC(=O)N(C)Cc2ccc(Br)c(Cl)c2)(OC)CC2NCCC12 c1(C(=O)Nc2cnncc2Br)[nH]c2ccccc2c1-c1cn[nH]c1 C(=O)(CCCCCOCCCSCCN(CC)CC)NC1(CN)CCOCC1 N1(C(C2C(C)(C)C2(C)C)=O)C(C(=O)NC(C2CCOC2)CO)CCC12CC2 C1(NC(C(CC2CN(C(c3c(C)n[nH]c3)=O)C2)F)=O)CC2CC1CC21CC1 Cc1c(C(=O)NCC2CC2NC(=O)C2=COCCO2)nc2sccn12 C1(NC(c2scc(C)c2)=O)CCCCC1C(=O)NCCC1CCCCC1O C(C(=O)N(CC(C)O)CCNC(c1c(C)ncnc1O)=O)(C(F)(F)F)OC(C)=O C1(NC(COC)=O)(CNC(=O)CCCc2coc(C3CC3)n2)CCC(F)(F)CC1 N1(C(C(=Cc2ccccc2)OC)=O)CCN(C(C2CCNC2=O)=O)CC1C1CC1 C1(O)(Cc2cnc(NC(C3CC(C)(C(=O)OC)C3)=O)s2)CCN(C(=O)OC)C1 N1(C(c2ccc(OC(C)C)cc2)=O)CC2CC(NC(=O)CCCN=[N+]=[N-])C1C2 C1(NC(C(C)CN(C)C)=O)CCCCC12CCN(C(=O)CC13COCC(C1)C3)C2 Cc1ncnc(C)c1OCC(=O)N(C)CC1(NC(c2ccoc2C)=O)CC1 c1(C(N(C(C#C)C)CCCC)=O)ccoc1CNC(C1CCCC1)=O N1(C(CNC(CCC)=O)=O)CC2(CCC2)CC1C(=O)NC(c1ccc(C)nc1)C c1(C(=O)NC(C2CCCC2)CNC(CN(CCC#C)C)=O)c(N)sc2c1CCC2 C1(NC(C(c2ccc(F)cc2F)C)=O)CN(NC(=O)CSC(F)(F)F)CC12CCC2 c1(NC2C(OC)CCOC2)nc(N(CC(C)(C)C)C)nc2c1cnn2C c1(OC)cc(F)c(C(c2nnnn2-c2ccc(Cl)cc2F)NCC(N)=O)cc1Br Cn1cc(C(=O)N(C2CCCC2)CCNC(C2C3CC3C3CC23)=O)c(O)nc1=O C1(CCNC(C(C)(C)F)=O)CSCCN1C(=O)C(c1ccccc1)C1CCCC1 C(CSC)(C(=O)N1CC(C(C(=O)N(C)Cc2cc(C)cs2)OC)C1)OC C1(CC)CCOC2(CCN(C(=O)CCC(=O)N(CC)CC)CC2)C1.C1(C)C(=O)N1 c1(C(=O)NCCC(CC)(C)NC(=O)C(C)NC(C)=O)cc(C)c(F)cn1 c1(CNC(CCSC)=O)cccc(C(=O)NCC2CN(C)CCO2)n1 c1(C(=O)NCC2CCC(NC(c3c(C)cc(Br)o3)=O)C2)ccc2n[nH]cc2c1 C(=O)(C(=O)N1CC(OCCC(=O)N(CCO)CCN(C)C)C1)NCC.C(C(F)F)O c1(OC)c(Br)ccc(CNC2CCC(C(=O)Nc3ccc(C#N)c(Cl)c3)C2)c1F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(=O)C(C)OC)C2 C1(CNC(c2cnc[nH]2)=O)C2CCC(C2)N1C(=O)C=CC1CCCCC1 C1(NC(=O)NC2(C)CC(F)(F)C2)CCCC23OCCC2CC13 O=[N+]([O-])c1cc[n+]([O-])cc1NCc1cnc(C(F)(F)F)c(F)c1 CN1C(=O)CSC1=CC(=O)NC1CC(C)(NC(C2CC3(C2)C(F)(F)C32CC2)=O)C1 CC(C)S(=O)(=O)CC(=O)N(CCCCNC(c1ccc(C(F)F)c(F)c1)=O)C C1(CN(C(C2CCC(NC(CNC(C(CC)C)=O)=O)C2)=O)C)CCCC1(C)C c1(C(N2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)ccc(F)c(C(C)(C)C#N)c1 C1(C)(C(N2CCC(N(CCC)C(c3ncoc3COC)=O)C2)=O)CCC(=O)N1 c1(-c2cc(C(=O)O)cc(OCC(=O)N(C)C)c2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 N1(C(c2nccc(CC)c2)=O)CCCC2(C1)CN(C(=O)C(C)CC(=O)OC)C2 C1(CNC(CN(C)CC)=O)C=CCN1C(=O)Cc1ccc(C)s1 C1(C(N(C2CCCN(C(C=CCCC)=O)C2)CC)=O)Cc2ccc(F)cc2C1 C1(C(=O)NC2CN(C(COCCCCCC)=O)CC2(C)C)CNc2ccnn2C1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(=O)NC)=O)C2)nn(C)cc1[N+](=O)[O-] C1(NC(C=C(C)C)=O)CC(C)CN(C(c2cccc(-c3ccco3)c2)=O)C1 N1(C(c2ncn(C(C)C)n2)=O)CCC(C2CC2)C1CNC(C1(C)CCOCC1)=O CCC(O)CC(=O)NC1(C(N2CCN(C(C)=O)CC2)=O)CC1 C1(CC)CN(C(c2cccc(N)c2O)=O)CCN1C(=O)CC(C)c1cccnc1 N1(CC(N2CCC(N(C(CC=C)=O)CCC)CC2)=O)CCCC2(CC2)S1(=O)=O c1(N(C(N(C)C)=O)C)cccc(N(CCC2CCCCC2)C2CC2)c1 C[Si]1(C)CCC(N)(C(=O)NCCCc2ncc(-c3ccccc3)[nH]2)C1 C12(NC(CS(=O)(=O)N(C)C)=O)CCCC1CN(C(C1(F)CC3(CCC3)C1)=O)C2 CCC(C(=O)N1CCCCC1C(N1CCCC(O)CC1)=O)C(C)(C)CC N1(C(c2c(CNC(CC3(N(C)C)CC3)=O)cco2)=O)CC(C)(CO)CC1(C)C N1(C(C2(C=C)CCOCC2)=O)CCN(C(=O)C(O)CC2CCCCC2)CCC1C c1(NCCN2C(C)COCC2)ccc(S(=O)(=O)NCCN2CC=CC2)cc1C#N c1(C(=O)NCC2(O)CCN(C(CC(CC)C)=O)C2)ccc(S(=O)(=O)N(C)C)o1 CCC(C)(C)C(C(=O)N1CCC(NC(c2cnc(C)n2C)=O)C1)OC c1(NC(C)=O)ccc(C(=O)NC2CCC(C)N(C(=O)C(=O)NC(C)C)C2)c(Cl)c1 c1(C(=O)NC2C(CNC(C(C)OCC)=O)CC2)cnnc(C2CC2)c1 CCC(C(=O)N1CCC(NC(c2ccccc2C(C)(F)F)=O)CC1)C(C)O C#CCCCC(=O)N(C)CC1C2CN(C(=O)CCc3cccc(OCC)c3)CC12 Cc1cc(N(C)CCN(C(c2cn(C3CCOCC3)nn2)=O)C(C)C)nc(Cl)n1 C1(C(N2CCC(CC(C)NC(C3CC(=O)N(C)C3)=O)CC2)=O)C(F)(F)C12CCC2 c1(C(c2noc(-c3sc(CN)nc3Cl)n2)C)cccc(Cc2cccc(F)c2)c1 Cn1nc(C(F)F)c(CN2CCC3(CC3C(N3CCC(C)(O)C3)=O)C2)c1Cl C(=O)(CCC(CC)CC)NC(c1ccc(C)nc1)c1nnnn1CCCSCC c1(C(N2CC(N(C(C3(CC)CCC3)=O)C)C(C)CC2)=O)oc2ccccc2c1Cl C(CC(=O)OC)N(CCNCC(C)N(C(=O)CN(C)C(N)=O)C)C N1(C(C(CC2CN(C(=O)CSc3nc[nH]n3)C2)F)=O)CCC(C2CC2)C1 N1(C(CC(C)NC(CCNC(=O)OCC)=O)=O)CC2(CC(C)CO2)C1 C(=O)(C(C)(CC)C(=O)NC(C)(C)CCCNC(c1cc(C(F)F)[nH]n1)=O)OCC c1(OC)cccc(Cl)c1C(N1CC(OC)CC(NC(=O)C(C)(C)CF)C1)=O C(C(=O)NCC1CN(C(c2ccncc2N(C)C)=O)CC1O)(C(C)(C)C)N(C)C Cc1cc(-c2cn(CC3CCCN(C(=O)CN4CCNC(=O)C4)C3)nn2)n(C)n1 C1(CNC(NCC(C)(C)C)=NCC2CCCSCC2)CC2(C1)C(F)(F)C21CC1 C1(C)(CC)C=C(C(=O)NCC(c2ccc(F)cn2)(F)F)C1 c1(COC)ncc(C(=O)NC2CCCC2CNC(=O)CCc2ccn(C)n2)s1 N1(C(C2(c3cc(NC(C)=O)[nH]c3)CCC2)=O)CCN(C(C)=O)C(C2CCCC2)C1 N1(C(C#CC(C)C)=O)CCC(O)(CN(C(=O)COCC2CCCC2)C)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(=O)CC2CC2)CC1CO C(=O)(CC(O)C(Cl)(Cl)Cl)NC(CC)CN(C(=O)C=Cc1ccc(C)cn1)C C12(NC(C3N=C(C)SC3)=O)CCCN(C(c3ccncc3OC(C)C)=O)CC1C2 C1(CNC(c2c(C)n(CC(C)(C)O)nc2)=O)CC2CCCCC2N1C(=O)CO C(=O)(C(C)C(O)C(C)C)NCC(C1CCCC1)NC(c1cc(C)ncc1C)=O c1(C(=O)NCc2cc(OC)nn2C)ccc2c(n1)CN(C(C1CCO1)=O)CC2 c1(COC)ccc(Cl)c(F)c1Cl.N12CC(CC(F)C1)C(=O)Nc1ncc(cn1)C2 N1(C(CCOCCC)=O)CCC(CCNC(C2CCC(c3cc[nH]n3)O2)=O)C1 c1(C(=O)NC2CCN(CC(=O)NC)CC2O)cccc2nc(C)sc12 C(C(CC(=O)N1CC=CC(O)C1)C1CCC1)N(C(CC)C(=O)NOC(F)F)C N1(C(C=CS(C)=O)=O)CC(CNC(=O)Cc2ccc(Cl)nc2)CC(C)(C)C1 C1(NC(c2ccccn2)=O)CCN(S(=O)(=O)CC2CCC3(CC3)C2)CC1 N1(C(Cc2nc(CC)sc2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C1(C)C c1(CC(=O)NC(C)CCNC(C2CC2(Cl)Cl)=O)cccc2ccccc12 C(=O)(C1=CC2(CN(C(c3cn(CCO)nn3)=O)C2)OC1)N1C(CO)CCC(C)C1 c1(NCCNC(C(CC(C)C)NC(C)=O)=O)ncnc2c1nnn2CC1CC1 CCC(C(=O)NCC1CCN(C(=O)C(C)(C2CCOCC2)OC)CC1)C(F)(F)F n1(CC)cc(C(N2CC(O)(CNC(=O)COC(c3nccn3C)C)C2)=O)nn1 CN1N=C(CC(=O)NC(CNC(C2(Br)CC2(C)C)=O)C2CCC2)CC1=O C1(C(N(C)Cc2cn[nH]c2)=O)COCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC(C)N(C(c2c(CC)nns2)=O)C)cnc2c(c1)N(C)CCO2 Cc1nn(C)cc1CC(=O)NCCc1ccc(CNC(C2CC2F)=O)cc1 c1(N(C2CNCCC2(F)F)C(C2CC3(CCC3)CN2)=O)ncnc2c(Br)c[nH]c12 C1(C)(CC)C=C(C(=O)NCCN(CCCN(C)C)C(c2[nH]c(C)nc2C)=O)C1 CC(C)CC(CNC(=O)COC1CC1)NC(c1ccoc1)=O Cc1nn(CCNC(c2ccc(C(=O)O)s2)=O)c(C)c1Br.c12cccc(c1)CC2 c1(C(N(CCNC(=O)C(C)C(C)O)CC)=O)c(OC)ccc(OC)c1N c1(C(=O)NCCOC(CNC(C(C)=C(C)C)=O)(C)C)csc(C)c1C n1(CC)nccc1C=CC(N1CCOCC1CNC(C1CC1CCOC)=O)=O CC1(C#CC(=O)NC2CN(C(=O)C(O)c3ccsc3)C2)CCCO1 C(=O)(C1=CC2CCC(C1)C2)NCCC1CC(NC(CSc2n(C)ccn2)=O)C1 C1(C(=O)NCCC2CN(C(C=C(C)C(C)(C)C)=O)C2)CCC2(CC1)OCCO2 c1(C(=O)NC2CC3(CN(C(CC(=O)OCC)=O)C3)OC2)cnc2snc(C)c2c1 C(C(O)CC(=O)N(CCCN(C)C(C1CC(c2cccc(Cl)c2)C1)=O)C)N(C)C C=Cc1cncc(C(=O)NCC2CN(C(c3conc3CC)=O)CC2C)c1 C1(C(N(CCOCC)C)=O)C2CCN(C(c3cc(OC)cnn3)=O)CC12 CC1(CF)CN(C(C2CCCN2C(=O)C(C)(O)C2CCC2)=O)C1 N1(C(c2c(C)csn2)=O)CC(C(=O)NCC(c2ccncc2)C)C2(CC2)C1 CCC(CC(=O)NC(Cc1cn(-c2ccsc2OC)nn1)C(=O)OC)C1CCC1 C(c1ccnc(Cl)c1)=CC(N1CC2C(CN(C)C)C2C1)=O c1(NC(C)=O)cccc(C(=O)NC2CCN(C(=O)CN3CCOCC3)C2C)c1 CC1C2CCC(C2)C1C(=O)NCCCN(C(=O)C=Cc1ccc[nH]1)C CC1CCC(Cl)=C(C(=O)NC2C3CC2N(C(=O)CCC(=O)c2ccccn2)C3)C1 Cc1nc(C#N)c(NCCC(=O)N(C)CCNC(=O)C(C(C)C)c2cccs2)o1 c1(OC)cc(C(=O)NC2COCC2NC(=O)CCC(C)(F)F)ccc1C#N N1(C(C(C)N(C(C)=O)C)=O)CC2(COC(CNC(C34CCCN3CCC4)=O)C2)C1 C(=O)(C1=CC2(CN(C(=O)C(C(C)CC)OC)C2)OC1)NCc1c(CC)n[nH]c1 c1(OC)ncc(C(=O)NCC(C2CCCN2C(C2CC2CN(C)C)=O)(C)C)s1 c1(C(=O)NC(C2(O)CN(c3cnc(C#N)cn3)C2)C)cc(F)c(F)cc1Cl C1(CNC(C2C(COC)CCC2)=O)(NC(c2cccc(OC)c2)=O)CCCCC1 N1(C(C2CCCCS2(=O)=O)=O)CCCN(C(c2ccc(C3CC3)c(F)c2)=O)CCC1 n1(CC)cc(NC(=O)CC2CCCN2C(=O)Cc2n[nH]c(C)n2)c(C)n1 N1(C(c2nc(=NC)[nH]c(C)c2)=O)CC2CCCC(N(C)C(C3CC3C)=O)C2C1 CON(C(=O)c1oc(CNC(=O)C(C)CC#N)nc1C)C(C)C c1(C(N2CC(OC)C(NC(C3(F)CC=CCC3)=O)C2)=O)cn(C)c(=O)nc1O c1(C(=O)NCC(CC=C)NC(C2CC(C(=O)OC)C2)=O)cc(C)ccc1Br c1(COC(c2cccc3occc23)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(C(N2CCC(NC(=O)CN3CCS(=O)(=O)CC3)C2)=O)nccc2c[nH]nc12 n1(CC(=O)NC2C(NC(c3c(C)oc(Cl)n3)=O)CCC2)ccc(=O)n(C)c1=O C1(O)(CNC(c2c(C)snc2)=O)CC2CCC(C1)N2C(C1(O)CCCCCC1)=O c1(C(=O)N(C2CCCC2)CCNC(C2CCOC2)=O)ocnc1C1CC1 C1(CC(N2CCC(N(C(COCC)=O)C)C3(C2)CC3)=O)Cn2ccnc2NC1=O CCCC(O)CC(=O)NCC1CC(O)CN1C(c1cc(Cl)cnn1)=O C(=O)(CC1=NNC(=O)C1)NC(CC)CN(C(=O)CCn1c(C)csc1=O)C N1(C(C2(CC=C)CCC2)=O)CCC(CO)(CNC(C2(C)CCCOC2)=O)C1 C(=O)(C1=NOCC1)NC1(CC=C)CN(C(C2CC23CC(OCC)C3)=O)C1 Cn1cc(CN2CCC3(CC3C(=O)NCCCC(F)(F)F)C2)c2ccccc12 N1CC2(CCCC2C(=O)NCc2ccc(C)o2)C1.C(=O)(COCCOCCO)N C12(CNC(Cc3cccc(COC)c3)=O)CCC1CN(C(C1(C#N)CC1)=O)C2 C1(OC)CCC2(C(=O)NC3CCCCC3N(C)C(C3C4COCC34)=O)CC12 C1(C(C(=O)OC)O)CCN(C(=O)Nc2cccc(-n3cncn3)c2)CC1 C(CNC(c1ncoc1C(C)C)=O)(C(C)(C)C)NC(C1C(CC(C)C)C1)=O Cc1cc2nc(NCC(C)(C3CC3)NC(C3CCCS3)=O)cc(=O)n2o1 O=S(=O)(c1cccnc1NC(c1cc(Cl)ccc1F)CO)NC(CO)CCF n1(CC(=O)NC(C2CCNCC2)C)ccc2ccc(-c3ccc(F)cc3C#N)cc12 c1(NC(C2(CC)CCCN2C(=O)C(C)=C2CCCC2)=O)ccc(CO)cc1O N1(C(c2cc(C)sc2C)=O)CCCC(CO)(NC(c2cc(O)ncn2)=O)C1 N1(C(C(c2cccnc2)C)=O)CC(NC(=O)CCC(F)(F)F)C2(CCC2)C1 c1(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cc(F)cc(F)c1 C1(C(N2CCC(N(C(CC(=C)C)=O)CC)C2)=O)CN(C)CCO1 C1(C(=O)NC(C2(O)CN(C(=O)Cc3cnc[nH]3)C2)C)CCC2(CCC2)C1 C1(N(C(=O)Cc2cc[nH]n2)CC)CCCN(C(c2ocnc2C2CC2)=O)C1 c1(C(C)(C)C)ccc(SCC(N2CC3CC2C3NC(C2(F)CCOC2)=O)=O)cc1 O=C(CCCCCn1cc(CC2C3CCCCCC23)nn1)N1CC2(CCOC2)C1 CC1CCN(C(C2C3CCC23)=O)CC1N(C(=O)CCC(N)=O)C c1(C(N2CCOCC2(C)C2CC2)C(=O)NC(CC)C)ncc(Br)cc1C C=CC(C)(CC)C(=O)N1CC(CNC(=O)COCC2CC2)C(SC)C1 C1(N(C)C(C2CC(CCO)C2)=O)CCN(C(c2ccc(CO)cc2)=O)CC12CC2 N1(C(C(C(C)C)C(C)NC(=O)C=CC(F)(F)F)=O)CCC2(CC1)CN(C)C2 Cc1ccc(Cl)c(N)c1C(N1CC2OCC(NC(=O)CCc3cccs3)C2C1)=O N1(C(Cc2cn(C)nn2)=O)CCCC(CNC(C2(C#N)CCC2)=O)C1 c1(CC)nc2ccccc2cc1NC(=O)C(N1CCC2CCCCC2C1)=O Cc1ccc(S(=O)(=O)N2CCC(CN3CC4(CC(C(=O)O)C4)C3)CC2)cc1 N1(C(c2cc(OC)no2)=O)CCC(CC(C)NC(C23CSCC2C3)=O)CC1 C1(F)(CNC(C2C(CC)C2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(CN(C2CCN(C)CC2)Cc2c(C)nn[nH]2)cccc(Cl)c1 C(C(C)(O)C(C)(C)C)NC(C1(C#C)CN(C(=O)C2=NOC(C)C2)C1)=O C1(C(N2CCCC(C)(O)C2)C(=O)NC(C(=O)OC)C)CC2C(C1)C2(F)F Cc1cccc2c1CC(C(=O)Nc1cc(F)cc(F)c1CO)N2 C1(C(N(CCC)CCNC(C2(C)CC3(CC3)C2)=O)=O)CCN2CCOCC12 C1(NC(C2C(C)(C)C2)=O)CN(Cc2ncccc2F)CC1F C#Cc1cccc(C(=O)NC(CNC(c2cnn3ccsc23)=O)CC(C)C)c1F N1(C(CSC(C)C)=O)CCC2(CCN(C(C3CCc4n[nH]cc4C3)=O)CC2)C1 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2COC(C)C2)=O)C1C CC(CC(=O)N1CCCC(CO)(NC(=O)CC2SC(=N)NC2=O)C1)CC(C)(C)C Cc1ncc(CC(=O)NC2(CNC(C3COC(=O)N3)=O)CC2)[nH]1 c1(C(=O)NC2(CC(=O)NCC(CC(=O)NC)C)CCC2)cncc(F)c1C C1(NC(C(CC)OC)=O)C2CC3CN(C(C4(CC)CC(OC)C4)=O)C1C3C2 c1(C(N(C2CN(C(C=CC=CC)=O)C2)C)=O)c[nH]c2ccc(OC)cc2c1=O c1(C(N2CCC(C(C(=O)NC(C(=O)NC)C)C)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(c2cc(C(C)(C)C)on2)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C12CC2 N1(C(C2OCCC(C)C2)=O)CC2(CC2)CC1C(=O)NC1CC1CN(C)C c1(CN2C(C(N3CCCC(CO)C3)=O)CC(F)C2)cc(Cl)c(O)c(Br)c1 C(=O)(CCN(C(=O)CNC(N)=O)CC1CC1)NCCCCC C1(O)(CNC(c2cc(C)nnc2)=O)CCCN(C(c2ccc(C(F)(F)F)s2)=O)C1 c1(C(=O)NCC(CO)NC(=O)COC2CCS(=O)(=O)C2)ccc(Cl)c(F)c1F CCCCCC(F)C(=O)NCC(=O)NCC(=O)NCc1cnn(C(C)C)c1 CC(CN=C(NC1CCC1)N(C)Cc1ccc2c(c1)OCO2)C(C)(C)C c1(C(N(CCCNC(c2ncc[nH]2)=O)CCO)=O)cc2n(n1)CC(F)C2 Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)N2CC3CC3C2)cnn1 S(=O)(=O)(c1ccn(C)n1)N1C(C)C(c2ccccc2)CC1 C1(C(=O)NCC2C(C)CN(C(=O)C=CBr)C2)C2C3CC4C1C1C2CC3C41 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CC(CNC(c2c(OC)scc2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCN(CC2(NC(=O)C(CC)SC)CC2)CC1 C(c1ccncc1)=CC(=O)NCC(C(=O)NCC1(CO)CCCCO1)OC C1(NC(C(C)OCC#C)=O)CCN(C(c2cc(F)c(Cl)cc2F)=O)CC1(C)C N1(C(C2(F)CN(C(C3SCCS3)=O)C2)=O)CC2(CCC2)CC1CO C(CC(C)CC)(C(=O)NC(c1nccc(O)n1)C)NC(C1CC(CCC)C1)=O N1(C(C(F)OC)=O)CC(NC(=O)CSc2ccnc(C(F)(F)F)c2)CC1(C)C C1(C(=O)NC(CC)C(N)=O)CN(C(c2ccc(O)cc2)=O)CC1F C#CC1CN(C(c2nccn2C)=O)CCN1C(c1csc(C(C)=O)n1)=O Cc1c(C(N2CCC3CCC(C2)N3C)=O)[nH]c2ccc(Br)cc12 C(=O)(C(C)(C)C(C)C)NCC(C1CC1)NC(C1CN(CC(C)C)C(=O)C1)=O C1(C(=O)NC(C)C=CC(=O)NCC(=O)N(C)O)CCCC(=O)CC1 CC(C(C)(C)NC(c1cnn(CCO)c1)=O)NC(=O)CCOC1CCOC1 C1(NC(c2n(CCC)nnn2)c2ccnn2C2CCCCC2)CC=C(C)CC1 c1(C2(C(=O)NC3CCN(C(COCCC#C)=O)C3)CC2)ccc(F)cc1O CCCC(C)(CC)C(=O)NC(CN(C(=O)C(=O)NCCNC(C)=O)CC)CC Cc1ccncc1C(=O)NCC=CCC(=O)NCc1cncc(F)c1 N1(C(CCCCN(C(C)C)C)=O)CCC(NC(=O)C(c2cnn(C)c2)C)C(F)C1 N1(C(C(C)n2ccnc2)=O)CCC2C(CCCN2C(c2cc[nH]c(=N)c2N)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCCN2C(=O)CSC(F)(F)F)(C)C)C1 C(=O)(C(=O)CCC(C)C)N1CCC(C(C)NC(c2c(C)nn(CCO)c2)=O)C1 n1(CC)nc(CCCN2CCCCC2)nc1C1CC1F c1(C(=O)NC2CCC(NC(C(C(C)C)F)=O)CC2)cccn(C2CCSC2)c1=O N1(C(C(c2cncnc2)C)=O)CCC(C)(C)C1C(=O)NC1CC2CCCCC12 C1(NC(C(CC=C)NC(=O)CC2CCOC2=O)=O)CCCCCC1C(N)=O C1(C(N(CCNC(C(C(C)C)C)=O)CC2CC2)=O)CCN(C)S1(=O)=O C1(C(=O)Nc2cn(CC)nn2)CCN(Cc2c(Br)cc(Br)cc2Br)CC1O Cc1ccc(O)c(C(N2CCC3CC23C(N2CCC2CN=[N+]=[N-])=O)=O)c1 C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCC(=O)N1C)=O C1(C(N2CCC(C)(NC(C3CCC(F)C3)=O)C2)=O)(COC)CCCCC1 C#Cc1cc(C(=O)NC2CCC2NC(C2CCCCN2CCCC)=O)cc(F)c1 Cn1c(=O)ccn(CC(=O)NC2C=CCN(C(C3CCNC3=O)=O)C2)c1=O C1(CN(C)C(N)=O)CCN(C(C2(NC(C3(C)CC3(F)Cl)=O)CC2)=O)CC1.C(N)(=O)N C(=O)(CCCCCNC(c1cnn(C)c1)=O)NC(CC(=O)NC)C N1(C(COC)=O)CCC1CNC(C1CC1C)=O c1(CC)c(C(=O)N(C2CC(NC(=O)CC(C)C3CC3)C2)C)cccc1C CC(C(=O)N(CC(C)CNC(=O)COCC1CCOC1)C)OCCN(C)C C1(CCC2N(C(C(C)c3ccsc3)=O)CCC2)CCCCN1C(=O)CNC=O c1(C(N2CCCC(NC(c3cc(C)ns3)=O)CC2)=O)c(F)ccc(F)c1Cl N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(=O)C(O)C(C)CC)C2)C1 c1(C(=O)NCCCCC=C)ccc2c(c1)CN(C(=O)C=CCC)CC2 c1(OC)cccc(C(C)CC(=O)N(CC(C)CNC(c2ncccc2F)=O)C)c1 C1(CC(=O)NCCC(C)NC(c2cn3c(n2)SCC3)=O)CC2C=CC1CC2 C(=O)(C1CCCc2ccnn21)NC1C(NC(C(C(C(C)C)O)C)=O)CCCC1 C1(C(=O)NCC(CCOC)NC(=O)C=CCN2CCOCC2)CC2(CCCO2)C1 C1(C(=O)NCCC(C)NC(C(CC)NC(C)=O)=O)CCC2(CC2)C1 N(C1CCCc2ccc(Cl)cc21)Cc1c(O)cccc1O S(=O)(=O)(c1cc(C(=O)O)co1)N1CCN(C(=O)C(O)CC(F)F)CC1 C1(NC(C(C2(O)CCCCC2)NC(=O)CCCF)=O)CCN(C2CC2)C1=O CCCC(O)C(=O)NC1CN(C(=O)CN2CCC(O)CC2)CC1SC c1(N(CC(CNC(C2CCC(C(C)C)CC2)=O)C)C)ncc([N+](=O)[O-])cc1F CC1(NC(c2cnc(-c3ccc(Br)s3)nc2)=O)CC2CCC1CC2=O C1(C2CCC2)(C(=O)NC(CCCNC(c2n(CCOC)ncc2)=O)C)CC1 N1(C(C(C)N(C(c2cnc(CC)o2)=O)C2CC2)=O)CC2C(C)C2C1 CN=c1nc(C(=O)NCCCCNC(c2cncn2C)=O)cc(C)[nH]1 C1(CNC(C(CSC)OC)=O)(CNC(C2(C(C)C)CCOCC2)=O)CC12CCC2 c1(NCCCc2ccc(OC)c(N)c2)cc(=NCC2(SC)CC2)[nH]cn1 N1(C(C(CC)(C)OC)=O)CC(S(=O)(=O)N2CCN(CC=C(Cl)Cl)CC2)C1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2C(C)C)ccc(Br)c(F)c1C C#CCCCC(C)C(=O)NCc1cc(C(=O)NC(C)CC#CC)n(C)n1 c1(C(=O)NC2COC2)nnn2c1CN(C(c1ccc(Cl)nn1)=O)CC2 C1(Nc2cnc3cc(C)nn3c2)C2Cc3cc(F)ccc3C12 C(=O)(C(C)(C)C(N)=O)N(C)CCN1CCN(C(=O)CCc2ccccc2F)CC1 c1(C(N(CCC(=O)N(C(CC)C(=O)O)C)C(C)C)=O)cnc(O)nc1O N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)C(C)OCC3CCCO3)C2C1 CCC(C(C)C)C(C(=O)Nc1cccc(OC)c1)N1CCSC(C)C1 C(CC(CNC(C1CCS1(=O)=O)=O)NC(c1ccc(NC(C)=O)s1)=O)OC C1(O)(CN(C)C(c2ccc(SC(F)(F)F)s2)=O)CCN(C(C2(N(C)C)CC2)=O)C1 Cc1[nH]c(=N)ccc1C=CC(N1CCC1CNC(c1cc2c([nH]1)CCCC2)=O)=O N1(C(C(C(=O)OCC)(C)C)=O)CC2(CCCC(CNC(=O)CC3(C)CCC3)O2)C1 C=C=CC1CCN(CC(=O)Nc2sc3c(c2C(=O)O)CCC3)CC1 CCCCC(F)C(=O)NCCCC(O)C(=O)NCC1CC2(CCC2)CO1 C(C(C)C(C)C(=O)NC1COCCN(C(=O)Cc2c(C)noc2Cl)C1)OC c1(C(=O)NC2C(NC(CC(C)N3CCCC3=O)=O)CC2)cccc(F)c1 c1(NC(C(CCC)C)=O)ccc([N+](=O)[O-])c(N2CCC(C(C)OC)C2)c1 S(=O)(=O)(c1cnccc1N1CCCC2(CCCC2)C1)NC(C)CCN(C)C Cc1ccc(-c2ncc[nH]2)cc1C(=O)NCc1cc(C(N)=O)co1 Cc1cc2cc(NC(c3sccc3NS(=O)(=O)CC3CCC3)=O)ccc2[nH]1 N1(C(C2CC(=O)NCC2)=O)CC2CC(NC(C3CCC4(C3)CC4(F)F)=O)C(C2)C1 C1(C)(C(=O)NCC2N(C(C3N(C(C)C)C(=O)CC3)=O)CCCC2)CCN(C)CC1 c1(CNC(c2ccc[nH]2)=O)nc2c(s1)CCN(C(C1CC3C=CC1C3)=O)C2 Cc1cncc(C(=O)NCc2ccccc2CN(C)C(c2nnn(C)c2C)=O)n1 N1(C(CC=C)=O)CC2CCCC(C1)N(C(c1ccc(-c3nncn3C)cc1)=O)C2 N1(C(CCCC(C)C)=O)CC(NC(C2CCCS2(=O)=O)=O)C(N=[N+]=[N-])C1 N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2C(CNC(c3cnoc3C3CC3)=O)C2C1 CC1CCC(C(=O)NCC(C2CCCCC2)NC(=O)Cc2cncnc2)O1 N(C1c2ccccc2CC1NC(=O)COc1ccccc1)C(CCS(C)(=O)=O)=O N1(C(C(C2CC2)OC)=O)CC(NC(=O)CC2CC2(C)C)C2CCCC12 N1(C(CCCC)C(N)=O)CCC(C2CC(=O)N(Cc3cnn(C(C)C)c3)C2)CC1 CCC(C)(COC)C(=O)NCC(O)CN(C(=O)Cc1csc(-c2ccco2)n1)C C1(NC(c2c(C)ccs2)=O)CN(C(=O)Cc2ccc3nc[nH]c3c2)CC1C1CC1 c1(C(=O)NCC(CN(C)C(c2cnc(O)o2)=O)O)ccc(CC2CCC2)cc1 C1(NC(C2(C(CC)=O)CC2)=O)CCOC(C(=O)NOCc2nnc(C)s2)C1 C12(CNC(C(N3CC(C)C3(C)C)=O)=O)CC3CC(C1)CC(O)(C3)C2 O(N(C)C(=O)CN=C(NCC1CC1)N1CCC(C(C)C)C1)CC c1(C(N2CCC(CN(C(C(CCC)OC)=O)C)C2)=O)nnc(O)c(Br)c1O CCC(CO)C(=O)NC(Cc1ccccc1)CCNC(=O)CCn1ccnn1 C(C(CN=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C(F)(F)F)NC(C=Cc1n(C)cnc1)=O C1(C(=O)NCCNC(C2C(C)C2)=O)CCCN(C(=O)CC2COC(=O)N2)C1 C12(C(=O)NCC=C(C(=O)NCCC(C)OC)C)CC(C#N)(C1)C2 NS(=O)(=O)c1ccc(C(N2CC(NC(c3cnc4[nH]ncc4c3)=O)C2)=O)cc1Cl c1(OC)cc(N)c(C(=O)NCC2CCCCN2C(C2CC3C=CC2C3)=O)cc1F c1(NC(c2cccc(CNC(C(CN(C)C)N(C)C)=O)c2)=O)cccc(F)c1O c1(C(N2CC3(F)C(NC(C=CC)=O)(CCC3)C2)=O)ccc2c(c1)C(=O)N(C)C2=O C(=O)(C1CCc2nccn21)NC1CCCCCN(C(C(CC)(CC)CO)=O)C1 C1(NC(=NCC)NCC(c2ccc(F)cc2)(F)F)CC1C1CCCC1 C(=O)(CC(C)CC(=O)N1CCN(C(c2[nH]cc(C)c2C)=O)CC1C(C)C)OC C#Cc1ccccc1CC(N1CCC(C)(C)C1CNC(=O)CCC=C)=O c1(C(=O)NCC(c2ccccc2)NC(CC=CC)=O)nn[nH]c1Cl c1(OC)cc(C(=O)NCCC2CCC(NC(c3cc(CO)n(C)n3)=O)C2)ncn1 C1(NC(CC2N(C)CC=CC2)=O)CCCCCC1NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC2N(C(c3c(Cl)ccc(C)c3)=O)CC2)c(F)ccc2c1OCC2 CC1(C)CCCN(C(c2ccc(C#N)cc2)=O)C1C(=O)NCCC12CCCC1C2 Cc1cc(C(N2CC3CC2CN3C(c2cn3ccnc3s2)=O)=O)cnc1C Cc1nc(C(=O)NCC(C)N(C(=O)C(C)(O)C2CC2)C)sc1C c1(C(N2CC(NC(c3cccc(OC)c3F)=O)C2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)(C)C(=O)N(CCN=[N+]=[N-])C)cc2cccnc2[nH]1 C1(CC)CCN(C(c2cnn(C)c2)=O)C(C(=O)NCC2(CO)CC=CC2)C1 N1(C(c2c(C)n(-c3cccc(Br)c3)nn2)=O)CCC2(CCCO2)C1 C1(CNC(C2N(C(CNC(CC(C)C)=O)=O)CCC2)=O)CCCC1(C)C c1(C(N(CCCNC(CNC(C)=O)=O)C2CC2)=O)cscc1C#N Cc1nn(C)cc1Cc1cn(CCCOc2cccc(C(=O)O)c2)nn1 C1(C(=O)NCC2CC(NC(CCc3ccc(NC)cc3)=O)C2)CC(=O)NC(=O)N1 Cc1cc(C(=O)NC2CC2NC(=O)C(O)c2ccsc2)cnc1OC(F)F c1(CN(C)C(C2C=CCC2)=O)cnn2c1CN(c1ncnc3c1nnn3C)CC2 c1(C(N2CC(O)(CCNC(C3CC(OC)C3)=O)C2)=O)cc2c(OC)cccc2s1 CC1(C)CC(C(N2CCCC(C(N)=O)CC2)=O)CCN1C(=O)Cn1cc(Cl)cn1 C1(N(C(c2cc(OC)c(OC)cc2)=O)CCNC(C)=O)CCCN2CCCC12 C#CCC(C(=O)OC)NC(=O)C(Cc1ccco1)NC(c1cc(CCC)on1)=O c1(C(=O)NC(CC=CC)C(=O)NC(CCC)CCO)ccc2[nH]ccc2n1 c1(C(=O)NC2CC(CNC(C(C)OC)=O)CC2O)cc(C)c(C)c(C)c1 C1(NC(c2ccc(C#N)o2)=O)CN(C(c2coc(Br)c2)=O)CC2CC12 C12(NC(CCCc3onc(CC)n3)=O)CCN(C(c3c[nH]nc3C)=O)CC1C2 c1(C(N2CC(OC)C(NC(c3ccco3)=O)C2)=O)c(F)cc(Cl)cc1Cl C12(C(N3CC(C)N(C(=O)C(C)(C)N(C)C)CC3)=O)C3C4C1C1C2C3C41C(N)=O c1(N2CCC(NC(c3cn(C(C)C)nc3)=O)C(F)C2)ncc2c(ncn2C)n1 O=C(N=c1ccc2nnc(C(F)(F)F)n2[nH]1)c1ccc(Cl)o1 C1(C(=O)NCC(C(CC)C)C)CC2(CCN1C(C1COCCC1C)=O)CC2 C(C(CNC(=O)C(C)OCCC(C)C)S(C)(=O)=O)NC(c1ccc(OC)cc1)=O N1(C(c2c(C)cccn2)=O)CC2(C1)CN(C(c1cc(Br)cn1C)=O)CCO2 C(=O)(N=c1cc(C)n(C2CCCC2)[nH]1)C1C(SCc2c(F)ncc(C)c2)CCC1 C12(C(N3C(CNC(C4CC5CC(=O)C4C5)=O)CCC3)=O)CCCC1CS(=O)(=O)C2 C1(NC(c2nc(C#C)sc2)=O)CC2CC1N(C(=O)CCC(=C)C)C2 c1(CC(=O)N(CCn2cc(-c3sc(C)nc3C)nn2)CC)ccc(C)nc1Cl C1(CNC(CCC(C)SC)=O)CCN(C(=O)COC2(C)CCC2)CC1O C1(C(=O)Nc2cnc(OC)nc2)N(C(=O)C(O)Cn2cncn2)CCCC1(C)C c1(C(N(CC(C)CNC(=O)CCN2C(=O)CCC2=O)C)=O)c(N)sc2c1CCC2 C(=O)(C1OC(=O)c2ccccc21)NCC1CC(NC(c2ccncc2)=O)C(O)C1 C1(O)(CC(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)[nH]n2)=O)COC(C)(C)C1 N1(C(C(C(C)(C)C)OC)=O)CCN(C(c2csc(C)c2C)=O)CC(C)C1 N1(C(C2N(CC)C(=O)CC2)=O)CCC(C2CCN(C(C3(SC)CC3)=O)CC2)C1 CC1(C)COC(C(=O)NC2CCC(NC(c3cc(Br)co3)=O)C2)CO1 C(C)(C(CC(=O)N1CCSCC1)NC(C1(C)CC1C)=O)OC C(Cc1cnc[nH]1)(C(=O)N(Cc1ccccc1)OC)NC(CCC=C=C)=O C1(C(N(CC(O)CNC(=O)C2=C(Cl)CCC2)C)=O)CCc2c(nnn2C)C1 C#CC1(C(=O)NC(CO)CCC)CCN(C(c2ccc[nH]2)=O)C1 c1(C(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)ccn2[nH]c(=N)nc2c1 c1(C(N2CCC(CNC(C(C)=C(CC)C)=O)CC2)=O)cc2c(s1)CCC(CC)C2 c1(CNC(=NC)NCc2cc(C3CC3)nn2C(C)C)ccc2c(c1)C(=O)OC2 N1(c2n(CC(C)C)c(-c3cc(C4CC4)[nH]n3)nn2)CCOC(C)(C2CC2)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1N(C(C(CC)F)=O)CC(O)C1O c1(C(=O)NC2(C)CC(NC(c3n(CC)nnc3)=O)C2)cc(Cl)ccc1Br c1(C(=O)NCC(=C)CCNC(C2COC(C)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2c(C)nc(C)n2O)=O)CC1C C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)c1cccc(NC(c2ccc(C)c(C)n2)=O)n1 N1(C(C2C(C)(C)CC2)=O)CCC(C)(CNC(=O)C(O)C2CCCC2)C1 CN1CCN(C(c2ccsc2C#N)=O)CC1C(=O)NCC(O)C1CCC1 C1(OC)CC2(CCC(C(N3CCN(C4CN(S(=O)(=O)C5CC5)C4)CC3)=O)CC2)C1 C1(NCC2C(NC(c3c(C)nsc3)=O)CCC2)CCCN(c2cc(O)ncn2)C1 C(C(C)CCCO)NC(C1(CC)CN(C(C=C(CCC)C)=O)C1)=O c1(C(N2CC(CN(C)C(C3CCCSC3)=O)C2)=O)nc(=O)cc(N)[nH]1 c1(OC)ccc(C)c(C(=O)N(CCNC(c2ccc([N+](=O)[O-])s2)=O)CC2CC2)c1 c1(C(=O)NC(C2(O)CN(C(c3nc(C(C)OC)sc3)=O)C2)C)ccccc1Cl C1(N(C(CNC(=O)NC)=O)C)CN(C(C2(n3cccc3)CCCC2)=O)CC12CC2 S(=O)(=O)(c1ccc(Cl)c2nonc12)N1C(CC(=O)OC)COC(C(F)(F)F)C1 CC1(NC(=O)C(F)=CC2CC2)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 N1(C(c2cn(CC)nn2)=O)CCOC(C(=O)NCCc2ncccc2F)C1 N1(CCC)CCCCC1C(=O)NCCC(CSc1ncc[nH]1)NC(=O)CSCC N1(C(C(C)SC)=O)C2CCCC1CC(NC(C1(C(F)F)CCC1)=O)C2 N1(C(C(=O)NCC=C)C)CCC(NC(c2cn(C)nc2C(F)F)=O)C(C)(C)C1 Cc1ccc(C=CC(=O)N(CCCNC(C2CC3C=CC2C3)=O)C2CC2)s1 c1(NC(CC2N(C(CN(CC)CC)=O)CC2)=O)ccc(F)cc1F c1(-c2nc(C(CCC)C)nn2C2CSC2)cc2ccc(Br)cc2s1 CCC(CC(F)F)C(=O)NC(c1ccccc1)CNC(=O)Cc1cn[nH]c1 Cn1nc(CNC(C2C=CCC2)=O)c2c1CCN(C(C1(C#N)CCC1)=O)C2 C1(C(N2C(c3ccc(OC)cc3)CNCC2)=O)CCC2(CCC2)OC1 c1(C(=O)Nc2cccc(C(=O)Nc3c(C)cc(CC)s3)c2)cc(Cl)c(Cl)nc1Cl C1(NC(c2n[nH]c3c2CCSC3)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 CC1CCCC(C(=O)NC(C2CN(C(c3cccc(F)c3)=O)C2)C)CC1 CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1c(Cl)cnn1C)=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC(C1F)N2C(C1CC(C)(O)C1)=O CC(C)CC(C(=O)NC(CN=[N+]=[N-])C(=O)NCC1CC12CC2(F)F)C(C)C c1(C(=O)NC2CN(C(C(C(C)C)(C)O)=O)CC2F)noc2c1CC(C)(C)CC2 N1(C(c2cnn[nH]2)=O)CC2C(NC(=O)C(F)(F)c3nccs3)C2C1 c1(NC(C(N2CCC(C(C)O)C2)=O)=O)ccc(F)cc1OC(F)F c1(C2(C(=O)NC3(CC=C)CCN(C(=O)C(F)(F)CO)C3)CC2)c(F)cccc1F n1(CC(=O)NCCCNC(=O)CC2CCCCC2F)c(=O)cnc2ccccc12 S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1CCN(C(C2CCC(Br)CC2)=O)CC1 Cc1ccsc1C=CC(=O)NCC(F)CNCC1CN(c2nnnn2C)C1 N1(CC)CCOCC1CC(=O)NC1CCCC1NC(c1cnn(CC(F)F)c1)=O N1(C(C2(COC)CCC(=O)N2)=O)CCN(C(=O)CN2CCCC2)CC(C)(C)C1 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnsc2)=O)ccc2c(c1)NS(=O)(=O)C2 c1(OC)ccc(CN(C2CS(=O)(=O)CC2O)Cc2nc(C(C)C)nn2C)cc1Br CCC(C)(CNC(c1sccc1C)=O)C(=O)N(CC(C)COC)C N1(C(CC(C(F)F)NC(c2c(OC)csc2)=O)=O)CCc2cccnc2C1 CCCCC(CCCC)C(=O)NCCC(C)NC(C1C=CC1C(=O)OC)=O n1(CCC)cccc1C(=O)NCC(=O)NCC1CC12CC2 C(CCCC(=O)NCC(c1ccc(C)cc1)NC(=O)C=C(C)C(F)F)(OC)OC c1(OCC)cccnc1C(=O)NCC1CCCN(C(C2(O)CCOC2)=O)C1 c1(OCC(=O)NC(CNC(C(C)=C2CCCC2)=O)CC(C)C)c(F)cccc1F CCCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)N1CC2(CCC2O)C1 N1(C(c2cccc(N)c2Br)=O)CCC2(CCN(C(c3ccccn3)=O)CC2)C1 c1(C(=O)NC(C(=O)NC2CCC(OC)C2)CCF)cc2cccnn2c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCCC2(CCN(C(c3cnc(Br)s3)=O)C2)C1 C1(C(=O)NCCNC(=O)OC)CN(C(c2ccc(C#N)cn2)=O)CCN1C C1(C(=O)NCC2CC(C)N(C(C3CC=CC3)=O)C2)CCS(=O)(=O)C(C)C1 C(=O)(C1Cc2c(Cl)cccc21)NCC1C(C)CN(C(=O)CCOCC2CC2)CC1 C1(CNC(C(C)OCC=C)=O)CCC2CN(C(=O)C(C#N)CC)CC12 c1(C(N(CC#CC)C)=O)ccc(CNC(=O)C(C)c2cccs2)cn1 CC(CC(=O)NCC(C)C(N1CCC(C(N)=O)CC1)=O)CC(C)(C)C O=c1[nH]cc(C(c2nnnn2C2CC2)NCC2CC23CC3)c2ccccc12 Clc1cccc2c(CNC3CCC(c4cccc(Br)c4)C3)csc12 c1(C(=O)NCC2(NC(N)=O)CCOC2)cccc(NC(=O)C=CCO)c1 C1(OC)CCCC(NC(c2cc(C(N3CC(N4CCN(C)CC4)C3)=O)[nH]n2)=O)C1 c1(C(N2CCC(NC(C(CN(C)C)N(C)C)=O)C2)=O)cc(F)c2[nH]nnc2c1 C1(COC(c2cccc(CC)n2)=O)CN(C(=O)OC(C)(C)C)C(C)(C)C1 n1(CCC(=O)NCC(C)NC(C2C3CNC(=O)C23)=O)ncc2c1CCCC2 c1(OC)ccc(C(=O)NC(CNC(c2coc3c2COC3)=O)C2CCC2)cc1O c1(C(=O)NCC(C2CCN(C(=O)C=CS(C)=O)CC2)C)cc2c(=O)[nH]ccn2n1 C1(N(C(CC)=O)C)CCCN(C(=O)C=Cc2ccc(I)o2)CC1 CCC(C)(COC)C(=O)N1CCCC(CO)(CNC(=O)C(O)CC2CC2)C1 c1(NC(C)=O)ccc(C(N2CCN(C(=O)CC3=CCCC3)CC2CF)=O)cc1F C(C)(C(C)(C)C(=O)NC1CCN(C(N)=O)CC1)NC(CSCCC)=O c1(NC(NCC(CC)(C)CO)=NCc2cccs2)cc(C)c(Br)cn1 C1(N(CC(c2ccccc2Cl)(C)C)C)CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(CNC(C(C)=C2CCC2)=O)C(C)C(C)C)nn(C)cc1[N+](=O)[O-] c1(CC(N2CCN(C(CCC=CC)=O)C(SC)C2)=O)cccc2c1OC(C)(C)C2 c1(C2CCN(Cc3c(F)ccc(C)c3)CC2)cc2c(s1)CCCC2 c1(C(=O)NC2C(NC(C(=O)NC(C)C)=O)CC2)cocc1Br c1(OC(c2ccc(CC)cc2)c2ccc(Cl)cc2)ccnc(O)c1C=O C1(CNC(c2ccsc2C(F)F)=O)CC2(CCN(c3nnc(O)s3)C2)CO1 Cc1cc(Br)c(C(=O)NCC2C3CN(C(c4coc(C#N)c4)=O)CC23)s1 CC(C)CS(=O)(=O)CC(=O)NCC1CSCC(CO)C1 C1(NC(C(c2cccc(F)c2)OC)=O)CC2(C1)CC2NC(=O)C1=CCCC1 C(=O)(C(C)C(C)(F)F)N(C1CCN(C(CCn2c(C)ccc2C)=O)CC1)C C(C(C)C(F)C(=O)N(C)CC1OCCC1(C)C)NC(C(CC)C#N)=O C=Cn1nncc1C(=O)NC1(C2CCCN2C(=O)C(C)OCCOCC)CC1 C(N=c1nc2scnc2c(N2CC3CC3(CO)C2)[nH]1)C1(C)C(C)(C)C1 N1(Cc2cn(CCC)nn2)CCN(C(=O)Nc2ccnn2Cc2nnc(C)o2)CC1 Cc1ccc(C(=O)NCC(N2CCOC(c3nnn(C)n3)C2)=O)cc1Cl Cn1ncc2c(NCc3cn4c(n3)COCC4)[nH]c(=NCCC3CCOC3)nc12 C(CC(O)C(F)F)NC(C(COC(C)C)NC(c1c(C)noc1)=O)=O c1(OC)ccc(S(=O)(=O)N2CC(C)CC2C(=O)N=c2cc(Cl)n(C)[nH]2)cc1Br c12ccccc1S2.N1(C(=O)NC(C)(C)C)CCN(CC)CC1.C12CN(C1)C2 S(=O)(=O)(c1cc(C(N2CC(NC(=O)CC(C)(C)C#N)C(C)C2)=O)n(C)c1)NC Cc1ncc(C(N2CCCC2CCNC(=O)CC(O)C(C)C)=O)cc1N C=CC1CCN(C(=O)C(CCC2CC2)NC(c2cnc(C)nc2)=O)C1 C12(C(=O)NC(C3CCCO3)CC)CCC(NC(C3CC(CSC)C3)=O)(CC1)CO2 C1(N(C(C=CCCCCC)=O)C)CCCC(NC(=O)COCc2scnc2C)C1 C(N=c1nc(N2CCC(N3CC(O)C3)C2)c2[nH]ccc2[nH]1)C1CCN(C(C)C)C1 C1(NC(C(CCNC(C(N)=O)=O)O)=O)C2C3CCC(C3)C12 N1(C(C(CSC)O)=O)CCCC(C(=O)N(CC(C)O)C)C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCCCCC1Cc1cccs1 c1(CC(N2CCC(C(=O)NCCC(C)F)CC2)=O)cnc(C)c(C)n1 Cc1nn(CCC#N)c(C)c1NC(c1cscc1C(F)(F)F)=O c1(C(C(=O)OC)N(C(=O)CCCSC)C(C)=O)ccc2c(c1)Cc1ccccc1-2 c1(OCCNC(c2n(CC)nnc2)c2nnnn2C2CC2)cc(F)ccc1C CC(C)C1=CCC(C(N2CCC2Cn2cc(C3(C)CC4CC4C3)nn2)=O)CC1 c1(OCC)cccc(C)c1C(c1nnnn1C)Nc1cn(CC2CC2)cn1 C1(C(N2CC(NC(CC(=O)NCC)=O)C(C)CC2)=O)CCC(C2CCC2)CC1 c1(OC)ccc(F)c(F)c1CN1CCC(CC(=O)NC(C)CC#N)CC1 C1(CNC(C=C(C)CNC(c2ccc(F)s2)=O)=O)CCCCS1 c1(C(N2C(C(C)NC(c3cnc(OCC)s3)=O)CCCC2)=O)ccc(F)cc1C N1(C(C2(C)CCCS2)=O)CCN(CCNC(c2ncccc2Br)=O)CC1 CC#CC1CCN(C(C2CCC(CNC(=O)C3=CCCC3C)C2)=O)C1 c1(C(N2C(C)(C)CC(CNC(C3CCSC3)=O)C2)=O)c(Cl)oc2ccccc12 C(=O)(NNc1cc(I)ccn1)NC(CC(=O)O)CC1CC1 C(=O)(C1=COCCO1)N1C(C2CCN(C(CN(C(COC)=O)C)=O)CC2)CCC1 c1(NC(CC(C)(C)n2cc(-c3ncoc3C3CC3)nn2)=O)ccc(Cl)cc1CO N1(C(C)CNC(=O)CC2CC2(C)C)CCN(C(N)=O)CC1.N12CC(C1)C2=O N1(C(C(C)(C)c2ccno2)=O)CC(NC(C2(CCO)CC2)=O)C(N=[N+]=[N-])C1 C=CCC(CC(=O)NC1CN(CC)C1)NC(=O)C(C)COC c1(C(=O)NCC2C(C)CN(C(c3ccsc3)=O)CC2)cnc2ncnn2c1N CC(C)(C)C(CNC(=O)CCN1CCCCC1)NC(C12CCCC1(C(N)=O)C2)=O C(CC(F)CN=[N+]=[N-])NC(C(C)(CO)NC(CC1ON=C(C)C1)=O)=O c1(C(=O)NC2(COC)CCN(C(C(CCC)OCC)=O)C2)cccc2c1COC2 c1(OC)cc(C)c(C(N2CC3CC2CN(C(C2(C)CC2Br)=O)C3)=O)cc1OC c1(NCC(C)NC(=O)NCC2N(S(CC)(=O)=O)CCC2)ccccc1Cl N1(C(c2c(C)nns2)=O)CCC(C)(CC(=O)NCCNC(=O)CO)C1 C1(C(=O)NCC#C)CC12CCN(Cc1ncc(Cl)cc1Cl)CC2 C1(C(=O)NC(C)CC2CN(C(c3ccc(C(F)(F)F)s3)=O)C2)CC2CCC2C1 c1(C(N2C(C#N)CC(F)(F)C2)=O)csc2c1CCN(Cc1ccc(Br)cc1Br)C2 C1(C(=O)NC2(C(N(CC)Cc3cnn(C)c3)=O)CCCC2)CC2(CCO1)CC2 c1(C(=O)NC2CC(C)(Nc3ncc(C)c(C)n3)C2)ccc2c(c1)NC(=O)C2 N1(C(=O)NC(c2cccc(C)c2)CN(C)C)C2C=CCC1CC2 C(CCCCCC(=O)N(C1CCCCC1O)C)NC(CCC(C)(C)N(C)C)=O C1(CNC(C2(OCC)CCC2)=O)CCN(C(c2coc(C(N)=O)c2)=O)C12CCC2 Cc1cccc(NC(=O)C(C)(C)NC(=O)CCN2CCOC2=O)c1C C(=O)(C(F)(CNC(=O)CC1(O)CCCOC1)C(C)C)NC1CC(CC(=O)OC)C1 C(C)(C)(C(=O)NCCN(C)C(C1(O)CC(c2ccccc2)C1)=O)OC(C)C C1(CCC)CCCCC1CNC(C1CCCC1CC(=O)OC)=O.C1(=O)CCCN1 c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2C2CC2)=O)ccc([N+](=O)[O-])cn1 C1(NC(c2cncc(F)c2)=O)CCCCN(C(C2CCC23CCC3)=O)C1 C12(CNC(C=CCC)=O)CCC(CC1)N(C(=O)C(C)(Cl)Cl)C2 c1(CN(C(CN(CCC)C)=O)C)ccccc1CNC(=O)C=CCOCCO CC1CCN(C(=O)CC2CCSC2)C1CNC(c1nccc(C(F)(F)F)n1)=O c1(OC)ncnc(C(=O)NC2(CN(C(=O)CCOc3ccccc3)C)CC2)c1F C(c1c(C)noc1C)=CC(=O)NCC(CCOC)NC(c1cc(C(N)=O)c[nH]1)=O C1(C(N(CCCN(C)C(c2ccc(C(N)=O)cc2)=O)C)=O)CC2CCCCC2O1 CCC(CC(=O)N1CCCCC1C1CCN(CC2CCS(=O)(=O)C2)C1)C(C)(C)C C(=O)(C(CC(C)C)C(N)=O)NC(C(N1CC2(CC(OC)C2)C1)=O)c1ccoc1 Cc1ccc(F)c(C(=O)NCCC2C(C)CCCN2C(=O)COCCCF)c1Cl CCCCCCCCOCC(=O)NC(C1(O)CCN(C(C2(F)CC=CC2)=O)C1)C c1(C(=O)Nc2cc(C(F)(F)F)c(Cl)cc2Cl)c[nH]c(=O)c2ccnn12 c1(C2C(NC(C(C)N(CC(C)C)C(=O)CN(C)C3CC3)=O)C2)ccccc1 c1(C(=O)NC(c2nocc2C(=O)NCCC2CCCN2C)C)cncc(O)c1 c1(OC)c(C(N2CCC(O)C(NC(c3csc(C(C)C)n3)=O)C2)=O)c(C)nn1C N1(C(c2cccc(NCC)c2)=O)CCOCC(C)(CNC(=O)C(C)OC)C1 c1(C(c2nnnn2CC(C)C(=O)OC)(CC)NCCCOC)cc(Br)cs1 C1(NC(C(C)Sc2ccccc2)=O)CC(F)CN(C(=O)C(C)N(C)C)C1 c1(C(=O)NC(COC)CNC(=O)CC2CC=CCC2)cc([N+](=O)[O-])no1 Cc1cn2c(n1)CCC(C(=O)NCC(C)(C)NC(c1ccc(S(C)(=O)=O)o1)=O)C2 CC1CCCc2nc(C(=O)OCC3(C(C)NC(=O)OC(C)(C)C)CC3)cn21 C1(C(=O)NCC2(CC=C)CCCC2)CC(C)(C)CN1C(=O)C(CC)CC Cc1[nH]nc(C(C)C)c1C(=O)NC(C)C(CO)NC(C1CCCS1)=O C1(N(C(c2ccccc2)C(C)C)C(Cc2cc(C)no2)=O)C2CCC1CNC2 Cc1nnccc1C(=O)NC1COCCC1NC(c1cc[nH]c1C1CCCC1)=O CCC(C)(C(=O)N1CCC(N(C)C(c2cc(OC)c(C3CC3)nn2)=O)C1)C(F)F Cc1ccnc(CNC(C2CCC(=O)NC2c2ccccc2)=O)c1F CC1(CNC(C2CCN(c3cc(-c4cscc4CO)ccn3)CC2)=O)CCNC1=O C(=O)(CCC(=O)NC1CC(CNC(c2coc(Cl)n2)=O)C1)NCCC C(CN=C(NCC1(C)CCCCC1O)NCCc1c(F)cccc1Cl)OCC=C N1(C(C(C)n2ccnn2)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)CC1 C12(CNC(c3cc(C)[nH]n3)=O)CC1CN(C(C1C3CC4C(C3)C14)=O)C2 C(=O)(C1CCCc2ccnn21)NCCN(C(CC(C)P(C)(C)=O)=O)C n1(CC)nnnc1NC(C1CN(C(=O)C=CC2CC2)C1)=O c1(N(CCNC(C=CCC)=O)CC2CC2)cc(C2CC2)ncn1 c1(C(C)=O)ccc(C(=O)NCCC2CC(NC(c3c[nH]c(Br)c3)=O)C2)o1 C(C(C(=O)NCC1CC(F)(F)CO1)C(C)C)NC(C(COCC)C)=O Cc1scc(C(=O)NC(C)CNC(=O)C(c2ccc(Cl)cc2)C)c1N CCC(CN(C)C(C1CC(NC(C)=O)C1)=O)N(C)C.C12(CC1)C(=O)N2 c1(CC(=O)NC2CC2CNC(=O)CCC2CC2)c(F)cccc1Br CCCC(CC)C(C(=O)NC1CCC(F)(F)CC1)N(C)Cc1ccc(F)cc1C CC1(NC(c2nccn2C2CCC2)c2nnnn2C2CCC2)CCOC1C1CC1 c1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccoc3)C2)cc2cccnn2c1 c1(C(C(=O)NCC(F)F)N(CCCn2ccnc2)CC)ncc(C(C)(C)C)o1 c1(C(=O)NC(CN(C(=O)CS(N)(=O)=O)CC)C)ccc(-n2cccn2)c(Cl)c1 C1(CNC(CN2CCC(=O)NC2=O)=O)CC2CCCC2N1C(=O)C(F)=C1CCC1 c1(C(=O)C2CC2)cc(Cl)cnn1.C12CC(C1)C(=O)NC1CC(C1)C(=O)NC2C c1(CCC(=O)N(C)CC2CCSCC2)nc2ccccc2[nH]1 Cc1ccc(OCCC(N2CCOCC2c2ccccc2Br)=O)cc1 C1(C(N2C(CNC(c3nc(C)n(C)c3)=O)C=CC2)=O)CC(O)c2ccccc2O1 O=C(CCCCC(F)(F)F)NC1(CO)CN(C(C2(C3CCCO3)CCC2)=O)C1 C12(C(=O)NC3C(NC(CN(C)C(N)=O)=O)COC3)CCN(CC1)CC2 C1(NC(C(C)(C)CO)=O)COCCN(C(=O)CC(=O)Nc2ccc(N)cc2)C1 c1(C(=O)N(CCC2CC2)CC2CC2)cccc(C2CC2)c1 CC1CC(C(=O)NCC2CC3CN(C(=O)C(C)=C4CCC4)CC23)=NO1 Cn1ncc(C(N2CC(NC(=O)C=Cc3cc[nH]n3)C(O)C2)=O)c1N c1(C(=O)NCC2(NC(c3ccc(-n4ccnc4)cc3)=O)CCC2)cncc(O)c1 N1(C(CC=CC=C)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)nn1C)=O C1(CC(C)C)CCCN1C(=O)CCn1cc(CCN2CCNCC2)nn1 N1(C(C(CC)F)=O)CC2C3CCC(C(NC(=O)Cn4cc([N+](=O)[O-])cn4)C3)C2C1 c1(NCCC2(C)CC2(Cl)Cl)cc(S(=O)(=O)N(CCCCO)CC2CC2)ccc1C#N N1(C(CN(C(=O)C=Cc2ccoc2)CC#C)=O)CCC(c2ncco2)C1 C(CCN=C(NCCCCl)N1CCC(Nc2cccc(C(F)(F)F)n2)C1)SC C1(C)(NC(C2C(C)=CCS2)=O)CCCC1NC(c1c[nH]c(=N)s1)=O CC1(C)CC1(C)CN1CC(C(=O)OC2CN(C(=O)OC)C2)C1 CCCCCC(O)C(=O)NC1CN(c2cc(C(=O)OC)nc(C)n2)CC2(CC2)C1 c1(C(N2CCCCC(NC(=O)C(F)CC3CC3)C2)=O)cc(O)nc2c1CCCN2 CC(C)(F)C(C)(F)C(=O)N1CC(NC(c2cc(N)cnc2Br)=O)C(C)(C)C1 Cc1cccc(C(N2CCC(NC(c3cnn(C(C)(C)C)c3)=O)C(O)C2)=O)c1I C1(O)(CNC(c2nn(C)nc2Br)=O)CSCC1(C)C CC1(F)CCC(NC(=O)CN2CC(Oc3ccc(F)cc3)C2)CC1 c1(C(=O)NCc2nnnn2CC2CCOC2)cc(CNC2CC2)ccn1 c1(C(=O)NC2(CNC(C3CCC(C(=O)OC)C3)=O)CC2)[nH]c2cc(C)ccc2c1C c1(NC2C3N(C(c4ccc(C)cn4)=O)CC(CC3)C2)nc(C)c([N+](=O)[O-])cc1Cl C1(C(N2C(C(=O)OC)CC2C)=O)CC2CC2N1C(c1ccc(C)cn1)=O CCCCCCC(COC(C1CC=C1C(=O)OC(C)(C)C)=O)CC CCS(=O)CC(=O)N(C1CCCC1)CCNC(c1ccc(Cl)cc1)=O CCC(CC(=O)N(C1CCOC1)CCF)NC(c1cc(C)on1)=O N1(C(C2CCC=CO2)=O)CCCC(O)(Cn2cc(-c3cccnn3)nn2)CC1 N1(C(C(C)OCCCC)=O)CCC(C(C)(C)C(=O)N(C)Cc2ncc(C)o2)C1 N1(C(CC2CN(C(C(n3c(C)ccn3)C)=O)CC2C)=O)CC2C=CC1CC2 C1(CC(=O)NC2CCN(C(CCCC=C)=O)CC2)SC2=NCCN2C1=O CC1=NNC(=O)C1CC(=O)NC(CNC(C1(C(F)(F)F)CCOCC1)=O)C(C)C C(=O)(C1Cc2ccccc21)N1CC2C(CNC(C3(F)C(C)(C)C3(C)C)=O)(CC2)C1 C(=O)(CCCCC(N)=O)NCC(CNC(c1ccc(OC)c(Br)c1)=O)(C)O n1(CC)nncc1C(=O)NC1COCC1NC(=O)COC1CCOC1 Cc1sc(Cl)nc1C(=O)NC1CC1NC(=O)CC(O)c1cnc(Cl)s1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCN(C(=O)CC(c3ccccc3F)C)C2C1 Cc1cn(C)nc1C(=O)NC(C1CCN(C(=O)CCc2nc(C)c(C)o2)CC1)C C1(C)(C(=O)OC)CCN(C(=O)CC2CCCCO2)C1.n1(CC(=O)OCC)cc(C)nn1 c1(N2CCC(N(C(c3ncncc3C(=O)O)=O)CC)C2)c(Cl)cncc1[N+](=O)[O-] C(C(C)(C)C#CC(=O)NC(C)Cc1ccccn1)NC(c1cc(COC)on1)=O C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)C(c2cncn2C)O)CC1 N1(C(c2cnc(C)s2)=O)CC=C(C(=O)NC2(C(F)F)CCC2)C1 c1(C(=O)NC(CC(C)NC(CSCCCC)=O)C)cc(C)c(C)c2ncccc12 C1(C(N2CCN(CCNC(C3C(C)C3C)=O)CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(=O)NC2CCC(F)(CNC(C3C(C)C3)=O)C2)cnc2c(c1)COCC2 c1(CC)ocnc1C(=O)N(CC(=O)NC(C)C(C)n1cncn1)CC N(C(=NCCc1ncccc1F)Nc1cccc(F)c1)CC(COC)C CC(C)C(C)CCNC(C1CCC(C2CC2)N1C(=O)C=Cc1ccn(C)c1)=O N1(C(C2CCC(OC)CC2)=O)CCCC2C1CCN2c1nc(SC)ncc1Br Clc1cccnc1CNC(c1ccccc1)CC1COCCO1 CC1=C(C(=O)N2CCSCC2CCNC(=O)C(C)n2cccn2)CCO1 CCC(C)(C)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CSC1 Cc1cnc(C(N2CCN(C(c3cccnc3C)=O)C(C3CC3)C2)=O)c(F)c1 C1(C(c2cn(C(C(=O)N(C3CCCC3)C(C)C)C)nn2)N(C)C)CC2CCC1CC2 N1(C(c2n(C)c(=O)ccc2)=O)CCOC2(C1)CN(C(c1ccc(F)cc1Cl)=O)C2 C1(C(N2C3(CNC(CCN(S(C)(=O)=O)C)=O)CC(C2)C3)=O)CCC2(CCC2)O1 c1(NC)cnncc1C(=O)NC(C)CCNC(c1sc(CO)nc1C)=O c1(C(N2CCCC(CNC(N)=O)C2)C(=O)NC)ccc(OC)c2oc(C)cc12 c1(NC(C2CN(C(c3cc(Br)cnc3Cl)=O)CCC2O)=O)ccc(Br)c(Cl)c1Cl c1(C(CC(=O)NC2C(CNC(c3cnc(OC)s3)=O)COC2)O)ccc(F)cc1 c1(C(N2CCN(C(C3C(=C)CC3)=O)CC2CCO)=O)ccc2c(c1)B(O)OC2 c1(OC)cc(OC)c(C(N2CCOC(C(C)NC(=O)CCCN(C)C)C2)=O)cn1 c1(C(N2CCC(C3CCCN3C(C3CCCS3)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCCNC(C(C(=O)OCC)OC)=O)cncc(Cl)c1C C1(NCc2cc(C(=O)OCC)cn2C)CCC2(CC1)CNCCO2 C1(C(N(C2CCN(C(C3CN(S(C)(=O)=O)C3)=O)CC2)CC)=O)C2CCC1CC2 Cc1cc(C(N2CCCC(C(=O)NCc3cccc(F)c3Cl)CC2)=O)ccc1O CC1C(C(=O)N2CC(C)C(C)(C(=O)N(CCC(C)C)CCO)C2)=NOC1C Cc1cnccc1C(=O)NC1CCC(N(C(=O)C(C(C)O)NC(N)=O)C)CC1 c1(C(=O)Nc2ccc(-c3cc4sccc4s3)cn2)cnc(OC2CCOC2)c(Cl)c1 Cc1cncc(-c2ccc(N3CCN(C(C4CNC(=O)C4)=O)CC3)cn2)c1 C1(C(=O)NC(CN(C(c2cc3sccc3[nH]2)=O)CC)C)CCc2[nH]nc(O)c2C1 c1(OC)ccc(C(=O)NC(CCN(C(=O)CCCC(F)F)C)C(C)(C)C)c(C)c1 CCS(=O)(=O)Cc1cn(CCC2CC(NC(c3snnc3C)=O)C2)nn1 C1(C(=O)NC2CN(C(c3ccc(C)cc3F)=O)CC3C2C3)CCc2c[nH]nc2C1 c1(C(=O)NCCC2CN(C(=O)CC3CC4CC4C3)CCCO2)ccc(F)c(Cl)c1 C1(C#N)(C(N2CCCC(O)(CNC(CCC(C)OC)=O)C2)=O)CCN(C)CC1 c1(C(=O)NCC2CCC2NC(=O)C(c2cccc(Cl)c2)O)ccc(Cl)c(F)c1 Nc1c(Cl)c(C(=O)NCC2CCC2NC(=O)C=Cc2ccco2)cc(F)c1Cl c1(C(N2C(CNC(C3CC3CF)=O)CCCC2)=O)ccc(F)cc1OC(F)F C1(NC(C=CC)=O)CCN(C(C2CCCC3(C2)CC3(F)F)=O)CC(C)(C)C1 C1(C(N2CC(C)C(C)C2C)=O)CC2CCC(C1)N2C(=O)CCC1CCCOC1 c1(C(=O)NC(C)CNC(=O)CCSc2ccccc2Cl)cc(O)cc(O)n1 S(=O)(=O)(c1[nH]c(=NC(Cc2ccncc2)CO)ccc1Br)NCC1(C)CC1 C1(Oc2ccccc2)CCN(C(N2CCC(C)C(O)C2)=O)CCC1C(=O)O c1(OC)cccn2ncc(C(=O)NC3CN(C(=O)C(C)OC)CC3N=[N+]=[N-])c12 N1(C(C=CSC)=O)CCC(C2(O)CC(NC(=O)C(C3CCC(=O)N3)C)C2)CC1 C1(CC#C)(C(=O)NCCCCCN(C)C)CCN(C(=O)C(C)CO)C1 C1(COC)CN(C(C23CC2CNC3=O)=O)CCN1C(c1cn(C2CC2)cn1)=O C(=O)(C(C(C)(C)O)NC(C1CC1C(F)F)=O)NCc1nnn(C)n1 C(CCNC(C1C2CCCC12)=O)(C(=O)N1CCC(C(C)(C)O)CC1)OC N1(C(C=C(CC)C)=O)CCN2C(=O)C(NC(=O)CC3CCN(OC)CC3)CC2C1 CC1(C)C(NC(=O)C(=O)NC2CC3C=CC2CC3)CS1(=O)=O Cc1cc(Sc2ccccc2)nc(N2CCCCC2)n1.C12(C#N)CN(C1)CNC2=O C1(C(=O)NCC2CCC(NC(c3c(C)nccc3)=O)C2)CC2CS(=O)(=O)CC2C1 N1(C(C=CC(C)C)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(CO)C1 c1(C(=O)NC2C=CC(CNC(C3CC=CCC3)=O)C2)cc(F)cnc1O C(=O)(C1OCCc2ccccc21)N1CC(CN(C(COC(CC)C)=O)C)C1 c1(C(=O)NC2CCN(C(CC)=O)C2c2ccccc2)nn(C)c(=O)cc1C C(C1CCNc2ccccc21)NC(C12CC(C(=O)OC)C(C1)C2)=O N1(C(CC2CCCC(NC(C3C(C)CC3)=O)C2)=O)CCC2(CSC2)C1 C1(C(=O)Nc2c(C)ccc(-c3ccccn3)c2)CCN(C)C12CCCNC2 CN=c1cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)cc[nH]1 C12(C(=O)NC3(C#C)CCCOC3)CCC(CC1)N(C(C1(OC)CCSC1)=O)C2 CC(C)(C)C(CNC(=O)C=Cc1cnc[nH]1)NC(=O)CSCc1cscn1 C12(c3cn(CC(=O)NC(CC)C(=O)NCCOC)nn3)CCC(CC1)N2C(C)=O N1(C(C2C(C(C)C)CCO2)=O)CC2(C1)CN(C(c1ncccc1N(C)C)=O)C2 N1(C(Cc2c(OC)cccc2)=O)CCC(NC(C2CN(S(C)(=O)=O)C2)=O)C(F)C1 C1(CC(=O)NCCN(C(c2c(NC)nccc2)=O)CC)CCCC(OC)C1 N1(C(C(CCOCC)NC(c2cnsc2)=O)=O)CC(C(N)=O)CCC1C C(CCCC(=O)NC1(CC(=O)NCc2cccnn2)CC1)(OC)OC N1(CCC)CC(C)CCC1C.n12cnnc1C(=O)NCC2=O.C(C(C)C)SCC C1(NC(c2c(CNC(=O)CC3CCOC3)cco2)=O)CCCC2(CC2)C1 n1(CC(=O)NC2(CC(=O)NC3C(NC(C)=O)CCC3)CC2)ccccc1=O c1(C(C)Nc2ccc(N3CCOCC3)nc2)cc(F)cc(Cl)c1 C1(NC(C=CCCCC#C)=O)CCN(C(=O)CCc2c(C)c[nH]c2C)CC1 c1(CC(=O)NC2C(CNC(CCSC)=O)CC2)ccc(OC(C)C)cc1 C1(CN2C(c3ncc(Cl)cn3)CCC2)CC2C=CCC(C1)C2 n1(CCC(=O)NCCC2(NC(=O)CSc3cn[nH]c3)CC2)ncc2ccccc12 c1(C(N2CC(NS(CC=C)(=O)=O)C(C=CC)C2)=O)ccc2nc[nH]c2n1 C12(C(=O)NCC(CNC(C3COC3)=O)OC)CCC(C1)S(=O)(=O)CC2 C12(CNC(COC(C)C)=O)CCC1CCN2C(c1cc(-c2ccccn2)no1)=O N1(C(=O)OC(C)(C)C)CC2CC(C1)N(C(c1c(OC(C)(C)C)nnc(=N)[nH]1)=O)C2 C1(C)(C(=O)NCC(CNC(CCc2c(C)nccc2)=O)CO)CCN(C)CC1 Cc1ccnc2c(C(=O)NC3CN(C(C4Cc5ccc(F)cc5O4)=O)C3)cnn12 c1(C(N2CCC(C(C)NC(c3cscc3C(F)F)=O)C2)=O)ccc([N+](=O)[O-])s1 NS(=O)(=O)CCCCc1cn(CC2CN(C(=O)CN(C3CCOC3)CCO)C2)nn1 C1(C(c2n(CCOC)nnn2)NCC2(OC)CCOC2)CC2(C1)OCCO2 C1(NC(=O)COCC2CCOCC2)CCN(C(=O)CN2CCCC2)CC1CO N1(Cc2c(=N)cc[nH]c2)CCc2sc(C(=O)Nc3cc(Br)c(F)cc3Br)cc2C1 c1(C(=O)NCC2CCCN(C(C3C=CCC3)=O)C2)c(Cl)ccc2ncccc12 N1(CC)CCC2(CC1)CN(C(=O)CC(=O)NCCCOc1ccon1)CC(C)O2 C1(C(=O)NC2CCCC(NC(c3c(OC)c[nH]n3)=O)C2)CCCCC(F)(F)C1 c1(C(c2nnnn2CCCC2CC2)NCCCCC=C)nn(C)c(Cl)c1Br CCC(C)CCC(=O)NC1(CO)CCCN(C(c2ncc[nH]c2=O)=O)C1 C1(OC)CC2(C1)NC(=O)N(Cc1cnc3n1CC(NC(=O)C(F)(F)F)CC3)C2=O C(=O)(C(O)CCCNC(=O)Cn1ncnn1)NCC(COC)C C(=O)(C(CC)C(C)C)NC1(CC=C)CCN(C(c2cnc(Cl)[nH]2)=O)C1 N1(C(c2c(CC)n(CC(C)C)nc2)=O)CC(NC(C2CC(O)C2)=O)C(C)(C)C1 c1(C(=O)O)ccc2c(n1)CN(C(C1CC3(CCC1OC(F)(F)F)CC3)=O)CC2 c1(C(C)C)ccc([N+](=O)[O-])cc1NC(=O)CCCCCF CCCCCCC(C)C(=O)N(C1(CC(N2CCC3(CCC3)C2)=O)CC1)C Cc1ccn(CC(=O)NCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C)c(=O)c1 C(=O)(C1=CNC2=NCCC2=C1)NCC(CCNC(c1c(SC)cnn1C)=O)(C)C c1(C(C(N2CCC(NC(CC(C)(C)OC)=O)C2)=O)C)cc(Br)ccc1C c1(C(N2CCC(CS(=O)(=O)NC)C2)C(=O)NC(CC)(C)C)cc(C)co1 C=C(C)CCCC(=O)NC1CCCC1NC(=O)Cn1nc(C)n(C)c1=O CC(C)(C)C(CNC(C1(Cc2cnn[nH]2)CCOCC1)=O)NC(C1CSC1)=O C1(NC(CCCCNC(C)=O)=O)COC2(C1)CN(CCOc1ccccc1C)C2 c1(OCC)cccc(C(=O)NCc2cccc(NC(=O)COC(C)(C)C)c2)c1 CN1C2CCC1CN(C(=O)C(CCF)NC(=O)C#CC(C)(C)C)C2 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(C2(CO)CCC2)=O)CC1F C1(C(=O)Nc2c(C)scc2)CN(C(=O)CNC(N)=O)CC1C C=CCC(C)(CC)C(=O)NC1CCCC1NC(=O)CCC(C)(F)F Cc1ccccc1C(C)CC(=O)NC1(C(=O)N(C)C)CC1.c12cnc(s1)[nH]c2=O C(CCC(=O)NCCN(C(=O)CNC(=O)CC1CCCCC1)C1CC1)OCCC C1(NC(c2c(C)n(C)cc2)=O)CC=C(C(=O)NC2COCCN(C)C2)C1 N1(C(C=NOC)=O)CC2CC1CC2NC(=O)Cn1nc(C(F)F)cc1C C1(NC(Cc2cc(C)[nH]n2)=O)CC2CC(NC(c3noc(C4CC4)c3C)=O)CC12 c1(C(=O)NC2COCCN(C(c3nncc(C)c3)=O)C2)cccc2oc(O)nc12 C1(CNC(=O)CO)CN(C(c2cnn3ccsc23)=O)C2(CCOCC2)C1 C1(N(C(=O)CCC2CC2(C)C)C)CCC(N=c2[nH]nc(C(N)=O)s2)CC1 c1(CC)c(C(=O)Nc2cnn(CC(N)=O)c2)ccn1C.C12(CC1)CC=CC(=O)N2 C1(CNC(c2c(C)cno2)=O)CC2CCC1N2C(c1cccc(C)c1O)=O C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)(OC)SC)CC1c1cnn(C)c1 c1(N2CC3CCC(O)C3C2)nc2ccccc2nc1N1CCC(F)C2(CCC2)C1 C1(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CN2CCN1CC2 c1(C(N(CCCNC(=O)C#CC2CC2)CC)=O)ccc(F)c(C)c1C#N c1(OC)cc(CN2CCC(C)(C(=O)NCc3cccc(F)n3)C2)c(Br)cn1 O=C(C1CCCc2ccccc21)NC1CC(NCc2cn3cc(F)ccc3n2)C1 N1(C(C=CC)=O)CCC(C(N)=O)(CNC(=O)CCC2CCC(C(N)=O)O2)C1 N1(C(C(=Cc2ccc(F)cc2)C)=O)CCC2CCN(C(C(C)(C)C(F)(F)F)=O)C2C1 c1(OCC)cnc(C(N2CCC3(NC(=O)CC4CCCCC4)CC3C2)=O)c(Cl)c1 N1(C(C(CCC)N(C)C)=O)CC2CCC2(NC(=O)C=CCOCCOC)C1 C1(C(=O)NC(c2cn(CC)nc2CNC2CC2(CC)CC)=O)CC(C2CC2)=NO1 CCCCCCC(C)C(=O)N1CC2CCCN(C(=O)C3=CCCS3)C2C1 C1(C(=O)NC2(C(N(C)CC3(C)CCCO3)=O)CC2(C)C)C2CCCC(=O)C12 c1(-n2c(-c3[nH]cc4c3CCC4)nc(C(C3CC3)OCC)n2)ccc(C)c(Cl)c1N c1(C(=O)NC(CC)CNC(c2cnnc(O)c2)=O)ccc2oc(O)nc2n1 C1(NC(=O)CCc2ccnc(Cl)c2)CCCC(NC(C23CCCC2C3)=O)C1 C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1CN(C(CC2C(CC)C2)=O)C1 N1(C(CC=C)=O)CCCCC1C1CCCN1C(c1cc(OC)ccc1N)=O c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)CCC)cn(C(F)F)c(C)n1 C=Cc1cncc(C(=O)N(C2CCCN(C(=O)CSCCC(C)C)C2)CC)c1 C(=O)(CN1C(=O)COc2ccc(Cl)cc21)NC(C(C)(C)C)CNC(=O)CCCF C1(C(=O)NCC2(N(C)C)CC2)CC(NC(=O)C(F)C2CCOC2)C1 c1(SC)ncc(N)c(C(=O)NC(C)CC(C)NC(=O)CN2CC3CC3C2)n1 c1(C(=O)NCC(CC)NC(C2(C(F)F)CC2)=O)sc2ccccc2c1CS(C)=O c1(-c2nc(C)sc2)cccc(C(=O)N(CC(C)NC(C2CCCN(C)C2)=O)C)c1 C12(NC(C(c3ccc(F)cc3)C)=O)CC1CN(C(=O)C(c1cccnc1)C)C2 N1(C(=O)CC2CCCC2)CCC2C(C1)CN2C(=O)CC(C1CC1)C1CCC1.C1CCC1 c1(C(N2CCC(C(=O)NCCCCC#C)C(O)C2)=O)ccc(O)c([N+](=O)[O-])c1 c1(CNC(c2n(CC)ccn2)=O)cccc(CNC(=O)CC2CN(C)CC2O)c1 N1(C(CC(C)=C(C)C)=O)CCOC(CNC(=O)C(C)(F)c2ccon2)C1 CN1CC=C(C(=O)NC(C2CN(C(c3cccc(N(C)C)n3)=O)CCO2)C)C1 c1(C(N2C(C3CCN(C(C(C)OCC#C)=O)C3)CCC2)=O)nnn(C)c1CC C1(CNC(C2C3(CC(NC(C4C5CCCOC45)=O)C3)C2)=O)CC2(C1)CC(O)C2 C(CC(C)(C)C(=O)NCc1nn(C)cc1CO)NC(C1CC(OC)(OC)C1)=O C(=O)(C1=NN2CCCN=C2N1)NCC1CCC(NC(c2cc(C)nc(C)c2)=O)C1 C1(C(=O)OC)(COC)CCN(C(=S)NC2CC2)C1 c1(C(=O)NCC(C)NC(c2c(C)n(C)nc2Cl)=O)cc2cc(Cl)sc2[nH]1 C1(C(C)C)C(=O)N1.c1(OCC)nc(C(=O)NC2CCCC2NCC)ns1 O=C(NNc1ccc2c(c1)CCO2)C1CCC(c2nc[nH]n2)O1 c1(OCC)cccc(C(=O)NC2(CNC(C3OC(C)CC3C)=O)CC2)c1N C(C(C)(C)CC(=O)N1CCCC(F)C1)NC(CCc1ccn(C)n1)=O C1(CC(=O)NCCSCC#C)CC2(CC2)CN1C(=O)C(C)OCOC N1(C(C2CCCN(C(C=CC(C)C)=O)C2C)=O)CCN2CC(F)CC2C1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(F)(F)C2)=O)C12CC2 C1(C(N2C(C)(C(N3CCC(OC)C3)=O)CC2)=O)C2CCC(C2)C1C Nc1cnc(Cl)cc1C(N1CC(CNC(c2ccc(F)cc2Cl)=O)C(F)(F)C1)=O C12(NC(c3c(NC)nccc3)=O)CCC(CC1NC(c1cc(C(N)=O)[nH]n1)=O)C2 C=CCC(CNC(=O)C(N1CCCCC1)C)C(=O)NC1CN(C)CC12CC2 c1(CC)noc(C)c1CNC(=O)CN(C1CC(C#N)C1)C(C1C2CCC(F)C12)=O n1(CC(F)F)ncc(CN(C2CC2)CC2CCOC2)n1 c1(C(=O)NCC(C)(C)OCCNC(C(C)OCCC#C)=O)ccccc1Cl c1(C(=O)NCC(CNC(C2C(CCCC)C2)=O)OC)cccc(C2OCCO2)c1 c1(C(=O)NCCC(C)N(C(C=C(C)C)=O)C)cc(C(F)(F)F)nn1C c1(CCCN2CCCC(CS(=O)(=O)NC)C2)c(Cl)cccc1[N+](=O)[O-] CCCC(C)(O)CC(=O)N1CCC(NC(c2ccnn2CC(F)(F)F)=O)C(O)C1 Cc1cnccc1C(=O)NCC1(C)CCCN1C(=O)CNC(c1ccccn1)=O Cc1c(CC(N2CCCC(Nc3cncc(Cl)n3)C2)=O)cnn1C c1(-c2c(C(=O)NC)nccc2)ccc(S(=O)(=O)N2CCC23CCCCC3)cc1 CC1CC2CN(C(=O)C(O)C3CC3)CC2N1C(C12CCC(CC1)C2(C)C)=O C1(C(=O)NCC(N(OC)C)=O)CCC2CCC1N2C(=O)CN1CCCNC1=O C1(CN(CCN(CCCOC)C)C)CCCN(C)C1c1cncn1C CC(C)C(F)(CNC(=O)C(N)=O)C(=O)NCC1(n2ccnn2)CC1 c1(C(=O)NC2CN(C(C(CC)n3nccc3C)=O)C2)ncccc1C(F)(F)F c1(CNC(COC(F)F)COCC)c2c(nn1C)CCC2 CC(C)C(C)C(CNC(c1cccc(F)c1)=O)NC(c1coc(Cl)c1)=O c1(SC)ccccc1C(=O)NC1CCCCC1CNC(=O)CCS(C)=O Cc1nc(C#N)ccc1NC(C1C2CCC(C2)N1C(c1sccc1Cl)=O)=O Cc1cc(C(=O)NC2CN(C(=O)COC3CC=CC3)CC2(C)C)cc([N+](=O)[O-])c1 c1(CC)cc(C(=O)NCC2CCCCC2NC(C2C=C(C)CS2)=O)n(C)n1 c1(-c2scc(COC)c2)cc(C(=O)Nc2cc(F)c(Cl)cc2I)c2nccn2c1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C2C(NC(=O)CSc3cn[nH]c3)CC(C2)C1 c1(C(=O)NCC(C(C)(C)C)NC(c2cc(C)sc2)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCCC(N(C(=O)CN2CC3CC3C2)C)C1 C12(CNC(c3cc(C(C)C)ncn3)=O)CCC1C1(CC2)OCCO1 N1(C(C)=O)CCCCC1CC(=O)NC(C)(C)CCN(C)C(C1CC(CF)C1)=O C1(NC(c2ccc(CC)[nH]2)=O)CCCN(C(=O)C(C)(C)n2cnc(C)c2)CC1 c1(-c2cc(C)cc(C)c2)ccc2c(c1)CCN(C(=O)CNC(N)=O)C2 C#CCCCCCC(=O)N1CCC2(NC(C3CC(OC)C3)=O)CC2C1 N1(C(Cn2c(C)cc(C)n2)=O)CCC(CO)C(NC(c2cnc(S)nc2)=O)C1 N1(C(C(C)(C)O)=O)CCc2c(C(=O)NCc3ncccn3)cccc2C1 C12(NC(C(CC#C)O)=O)CCC(CC1)N(C(c1cc(O)ncc1Br)=O)C2 c1(C(N2CC3C(CNC(c4cccc(C)n4)=O)(C3)C2)=O)oc2ccccc2c1C Cc1nn(C)c(Cl)c1C(N1CC(CO)C(C)(C)C1)C(=O)Nc1cccc(Cl)c1C C1(C(=O)OC)CCCC(OC)OC(=O)CCN1C.C(C)(C)(C)OC Cc1cnn2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3cnn(C)c3)C)nc12 N1(C(C(C)Nc2nccs2)=O)CCC2(C1)CN(C(c1ccc(F)cn1)=O)C2 C(CCCN=c1[nH]c(=NCC23CCC(CO2)C3)c2ccccc2[nH]1)OC C1(OC)CC(NC(c2c(C)[nH]c(C)c2C)=O)C12CCN(C(C1CSC1)=O)CC2 C(CCCCC(=O)NCC1CCN(C(=O)CCS(C)=O)C1)=CC C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)C(=O)Cc1ccccc1 c1(C(N(C(CN(C(CN(CCC)C)=O)C)C)C)=O)cc(=O)c2ccc(Cl)cc2o1 c1(C(N2CCN(C3CCN(C(C(CC)C)=O)C3)CC2)=O)coc2c1C(=O)CCC2 c1(C(=O)NCCCCN(C(=O)CCCC2(C)N=N2)C)cnn2ccncc12 N1(C(c2cc(C)c(C)s2)C(=O)NCC=C)CCNC(=O)CC12CCOCC2 C12(C(CNC(=O)COc3ccccc3)NC(C3CCCO3)=O)CCC(CC1)C2 c1(C(C(=O)NC2CCC2)N(CCC(N)=O)C)cc(Cl)ncc1Br.c1(CN)nnn(C)n1 N1(C(c2c(CC)onc2)=O)CCC(C2(O)CCN(C(=O)C(C)(C)C)CC2)CC1 CCC(C(=O)NCC1CC2(C1)CN(C(=O)CC(C)=C(C)C)C2)C(C)O C(=O)(CCCC(=O)NC1CCC(N(C(=O)Cn2nnc(C(C)C)n2)C)C1)OCC C1(NC(c2ccc(-n3c(C)nnn3)cc2F)=O)CCNC2(CCC2)C1 c1(NC(N2CCC(c3scc(C)n3)C2)=O)cc(F)c(N2CCOCC2)c(F)c1 N1(C(CN2C(C)CC2)=O)CC2C(CNC(=O)C=Cc3ccc(C(N)=O)o3)C2C1 Cc1nc2cc(C(=O)NC3CCN(C(c4ncsc4C)=O)C(C)C3)cnc2[nH]1 CCS(=O)(=O)C=CC(=O)NCCCCC1CN(c2ncc(C#N)cc2F)C1 c1(OC)ccnc(-c2nc(SCCNC(=O)CN3CCN(S(C)(=O)=O)CC3)cs2)n1 n1(C(CC)(C)C)nnnc1C(c1cnc(C2CC2)s1)NCCCN1CC(C)(C)C1 c1(C(N2CCC(C(C)NC(COCC)=O)C2)=O)cc(NC)ccc1Cl N1(C(c2cnc(C(C)=O)s2)=O)CCC(C(C)NC(C2(F)CCOC2C)=O)CC1 c1(C(N(C2CN(C(C3(C)CC3F)=O)C2)C)=O)cc2oc(Br)cc2[nH]1 c1(N2CCC(CCOC)(NC(c3cnc(O)n3C)=O)C2)nc2cccnc2s1 c1(C(C)NC(c2ccsn2)C)nnnn1C1CC1 Cc1nc2c(C(N3CCN(C(=O)C4=CCC4)CC3CC3CC3)=O)ccnc2n1C CC(C)C(O)C(=O)NCc1nc(CNC(C2CCCN(C)C2)=O)cs1 Cc1cc(C(N2CC(C3CN(C(=O)C(F)(F)C(F)F)C3)C2)=O)c(N)c([N+](=O)[O-])c1 C(CCCCC(=O)NC1C2CC1N(C(=O)Cc1cnc(C)s1)C2)NC(C)=O C(=O)(C(F)Cc1ccccc1)NC1C(NC(=O)CN2CCC2)C1 N1(C(c2c(C)nsc2Br)=O)CCC2(C1)CN(C(=O)CSCCC#N)C2 c1(OC)cc(C(N2CCC(C(=O)NCc3cncn3C(C)C)C2)=O)ncn1 C1(CCNC(C(CCOC)C)=O)CCCN(C(c2ncn(C(C)C)n2)=O)CC1 c1(CC)onc(C(N2CC3C(CC(=O)N(CC(O)CN(C)C)C)C3C2)=O)c1C C(=O)(C#CC1CCCCC1)N1CC(NC(CCCCCCC)=O)C2(C1)CCC2 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NCC2CCN(C(N)=O)C2)CC1(C)C C1(CNC(C(C)=CC2CC2)=O)CC(C)CN(C(=O)Cc2ccnc(C)c2)C1 N1(C(CCN(C)CCO)=O)CC2(C1)C(NC(C1CC3CC3C1)=O)CCS2(=O)=O c1(C(=O)NC(CC)(C)CNC(=O)CSc2cccs2)cnccc1Cl N1(C(=O)Cc2ccccc2F)CC2CCN(C(=O)CCC3CC3(Cl)Cl)C2C1 c1(CN(C(CO)CO)CC)ccnc(-c2ccc(-c3nn[nH]n3)cn2)c1 N1(C(c2nccc(OC)c2)=O)CCCN(C(C2CC=CCC2)=O)CC1CO c1(OCC(=O)N(CCCCCNC(=O)CNS(C)(=O)=O)C)cccc(F)n1 C1(CN(C(C2CS(=O)(=O)C2)=O)CC)CCN(C(=O)CC2CCCCC2)CC1 C1(CCCC)CN(C(C23CC(F)(C2)C3)=O)CCN1C(=O)CCC1CC(F)(F)C1 N1(C(CCC=C)=O)CC(O)CC1C(=O)NC(CC)C(C)(C)C N1(CCCOCC)CCC(C(C)NC(=O)C(C2CCCC2)OC)CC1 c1(OCC)cccc(C(=O)NC2CC(O)CN(C(=O)CCCF)C2)c1N c1(C(=O)NC2C(CNC(c3c(Br)cn(CC)n3)=O)C2)cccc2[nH]ncc12 N1(c2cc(NCC(C)(F)C(C)(C)F)nc(C)n2)CCN2CCCC2C1 c1(C(N2CCC(C(=O)NC3C(CN(C)C)CCC3)CC2)=O)ccc(N)c(F)n1 C1(C(C)C)CN(C(c2cnn(C)c2)=O)CCCN1C(c1cnc(O)c(F)c1)=O C1(NCCCCCC)CCN(C(c2cc(C(=O)OC)no2)C(=O)NC)CCO1 c1(NC(C)=O)ccnc(CC(=O)N(C)C)c1 C1(NC(C(C(C)C)C)=O)CN(C(c2cc(-c3ccccc3F)[nH]n2)=O)CC1(C)C C1(OC)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C)n1)=O c1(CN2C(C)CCC2C(=O)Nc2cc(O)n[nH]2)cc(Br)cc(Cl)c1O C1(NC(c2cncc(OC)c2)=O)CC1C1CCN(C(C2(CC(F)F)CC2)=O)CC1 C(=O)(C(C(=O)NC1(C(=O)NC(c2ncc[nH]2)C)CCN(C)C1)OC)OCC C1(CNC(C(C(C)(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cncs1 N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)Cn2ccccc2=O)C(C)C1 CCC(CC(=O)N1CCN(C(c2nccc(C)n2)=O)CC1CCO)CC(F)(F)F C12(NC(C(c3ccccc3F)C)=O)CCCC1N(C(=O)CCC(N)=O)CC2 N1(C(C)=O)CCc2c(NC(c3cc(-n4nnnc4C)cc(F)c3)=O)cccc2C1 N1(C(C2C(C)=CCC=C2)=O)CCC(O)C(C(=O)Nc2cncc(Cl)c2Br)C1 c1(NC(c2c(NC(C=C(C)C(=O)O)=O)nc(Cl)cc2)=O)cc(C)cc([N+](=O)[O-])c1 C(=O)(C(CO)N(C)C)NCCN(C(=O)COCC1CCCOC1)CCC c1(OCC)cc(Cl)ccc1C(=O)NC1(CCNC(=O)Cc2ccon2)CC1 c1(C(N2C3(C)CCC(C2)C3)=O)ccc(S(=O)(=O)N2CCC3(CC(F)C3)C2)cc1 C1(CNC(C(C)OCCC=C)=O)(CO)CCN(C(C2(c3ccno3)CC2)=O)CC1 Cc1ccc(-n2nc(C(=O)N(C3CCC4(CC3)CC4)C)c(C)n2)c(C)c1 CCCCCC(O)CC(=O)NCC1CC(C(N2CCOC(C)C2C)=O)C1 C1(C)(C(=O)NCC2CC(NC(C3(SCC)CC3)=O)C2)CCCC1(F)F CCC(C)CCCCC(=O)N(CC(=O)NCC(F)(F)C(F)F)C(C)C c1(CC)cc(OC)cc(C(=O)NCC2CN(C(=O)C(C)(COC)CC)CCO2)c1 c1(C(=O)NC(C)CCCNC(c2ccoc2)=O)ccnc2ccccc12 C1(C(=O)NC2C(C)(C(F)F)C2)(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(-c2onc(-c3cc(C)cc(C)c3)n2)cnn2c1CCCC2 Cc1ccc(C(N2CC(NC(=O)C(C)(C)c3cnc[nH]3)C(C)C2)=O)c(O)c1C Cc1nc(=NCCC2CCC(NC(c3nc(F)ccc3Cl)=O)C2)[nH]cc1Br C1(CC(=O)NCCC2(NC(c3ccc(Cl)[nH]3)=O)CC2)CCCCC1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)CCCc2ccc(SC)cc2)CC1(C)C c1(CC(=O)N(C)CC2N(C(C(CC)=CC)=O)CCOC2)cccc(C)c1Cl C1(NC(c2cc(C(C)=O)[nH]n2)=O)CC(C)CN(C(C2CC3CCC(C2)S3)=O)C1 c1(COC)cc(C(=O)NC(C)(C)CN(C(=O)CCCn2cccn2)C)no1 c1(CCC(=O)N(CC(C)NC(=O)CC2CCC(C)CO2)C)ccc(Br)cc1 C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)N1CC(N(C(CC(CC)C(F)F)=O)C)C1 c1(C(=O)NCCN(C(C2CCC(=O)O2)=O)CC)c(C(F)(F)F)nn2ccccc12 c1(C(=O)NCC(c2ccccc2)NC(C=C(C)C2CC2)=O)ccnnc1S CC1CN(C(=O)C=Cc2ccc(Cl)cc2F)CCCN1C(=O)C(CO)N(C)C N1(C(C(=O)Nc2ncc[nH]2)=O)CCC2(CCN(C(c3ccc4c(c3)CC4)=O)C2)C1 N1(C(c2ccc(Br)cc2CCO)=O)CC2CCCC(C1)N2C(c1cncnc1)=O C1(COC)CCN(C(=O)C(F)(F)c2cccnc2)CC1.CCC1C(=O)N1CC c1(C(N2CCN(C(C=C(C)C(C)C)=O)C3C2C3)=O)cnc2c(c1)CCCO2 N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)C(C)N(C)C)C2)C1 C(N=c1nn[nH]n1C)C1(F)CC(NC(C(C)C2CC2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C)(C)CC1C(=O)NC12CC(F)(C1)C2 N1(C(C=CCC)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1c1ncc[nH]1 c1(CC(=O)NCC(C(C)C)NC(CC(CC)SC)=O)ccc2ncccc2c1 N1(C(C(C=C)C)=O)CC2CC(C(=O)NC(C(C)C)c3ncc[nH]3)C(C2)C1 c1(C(=O)NCC(CO)NC(C2(OCC)CCCC2)=O)cccc2c1NCC2 C(C1CN(C(C2CNC(=O)C2)=O)CC1C(=O)N(CCC(=O)NC)CC)=CC N1(CC)CC(C(=O)NCCOCCN(C)C(c2sccc2C#N)=O)CC1=O C1(C(N2CC(NC(c3cc(O)nc(O)n3)=O)(CO)C2)=O)COc2ccccc2O1 c1(C(=O)NC(CNC(C2(C)C(C)C2)=O)C)cc(C(F)(F)F)ncc1N c1(C(N2CC(CNC(C3(OC)CCCOC3)=O)C(C)C2)=O)ccc(C)c(F)c1N C(=O)(CCC(=O)NC1CC(N(C)C(C2COCCN2CC2CCC2)=O)C1)N(C)C C(=O)(C1=CCS(=O)(=O)C1)NCC(CNC(Cc1ccn(C(C)C)n1)=O)(C)O C(CC)(C(=O)NC(C)C(CO)NC(c1ccc(C2CC2)s1)=O)=CC C(=O)(C(O)C(F)(F)F)N1CCN(CC(=O)NCC(C)(C)O)CC1 C1(CCNC(c2cc(C3CC3)ncn2)=O)CSCCN1C(=O)CC1C=CCC1 c1(NCC2CN(C(C(C)OC)=O)CC2(C)C)nc2c(cc1C#N)CCC(C)C2 CC(C)C(C(=O)NC(CCF)C(=O)NC1CC2CC2C1)C1CCC1 Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)c2c(n1)CCCC2 c1(CC)ncc(Br)cc1NC(C1CN(C(c2ccc(O)cn2)=O)C1)=O c1(C(N2CC(NC(c3ccnc(OC)n3)=O)CC2(C)C)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC2CCCC2N2CCCC2)ccc2[nH]ccc2c1 C(=O)(C(C)(C)CC(=O)Nc1cccc(NC(c2sccc2F)=O)c1)OC c1(C(=O)NCC2CCCCC2NC(=O)CCc2cncs2)cnc2ccoc2c1 N1(C(c2ccc(NC)cc2)=O)CCC(C)(NC(=O)C(O)CC2CC2)CC1 CC1CCCCC1CC(=O)NCC1CN(C(=O)CCc2ccccc2F)CCO1 C(CN=c1[nH]nco1)(c1ccccc1F)NC(C1CCCCC1O)=O c1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CC2)cccc2c1CCCC2=O c1(C(N2CCC(O)C2)C(=O)NC(CC)(C)C)sc(S(N)(=O)=O)c(OC)c1OC C1(NC(Cc2nc(C(C)C)sc2)=O)CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2 C(CC(=O)N1CC(C)CCCC1C)(C(F)(F)F)NC(C(CCC)C)=O CC(CNC(c1n[nH]cc1C(F)(F)F)=O)CN=c1cc(C(C)(C)C)nc(Cl)[nH]1 C=C(C)C1OCCC1C(=O)NCCCC(C)NC(c1cc(C(N)=O)cn1C)=O N1(C(c2occ(C(N)=O)c2)=O)CCC(O)(C2(NC(=O)Cc3ccsc3)CC2)CC1 CCC(CC)(C(=O)N(C)CCOCCNC(C1CC2CCCC2C1)=O)OC c1(C(N2C(CNC(c3cccnc3)=O)COCC2)=O)nccn2cnnc12 Cc1cccc(C)c1C(N1CSCC1C(c1ccccc1)=O)=O CCC(F)C(=O)N(CCNC(=O)C(C)(C)c1ccccc1)C1CC1 CCC(CCC(=O)NC1CC(=O)NC1=O)NC(C1CCC=CCC1)=O c1(CNC(=O)CNC(=O)CNc2ccsn2)ccc(O)c(F)c1 N1(C2C(C)OCC2)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1c1cccs1)=O N1(C(c2c(C)ncs2)=O)CC2CC1CCN2C(c1cc(CO)on1)=O c1(C(N2CC(N(C)C(c3cnc(Cl)s3)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)o1 C(C)(C)(C(=O)NCC1(F)CN(C(=O)CC2(C)CCCO2)C1)OC(C)=O C(=O)(CCCCCC(=O)NCCCC(C)NC(C1CCS1(=O)=O)=O)OCC c1(C(=O)NC2CN(C(C3C(c4c(C)nn[nH]4)C3(C)C)=O)C2)c[nH]c2cnccc12 N1(C(=O)C#CC2CC2)CC(CO)C2(CCN(C(C3CCC=CCC3)=O)CC2)C1 N1(C(C(C#C)(C)C)=O)CCC2CCN(C(c3c(SC)cccc3F)=O)CC2C1 Cc1ccn(CC(=O)NCC2(O)CN(C(=O)Cc3ccccn3)C2)c(=O)c1 C12(NC(C(CCC#C)O)=O)CC(C)(C1)OC21CN(C(=O)C(CC)SC)C1 OC1CCN(C(=NCCCC2C=CCC2)NCCF)CC1 Cc1ccc(CC(=O)NCCOc2ccc(C(=O)NC3CCCC3)cc2)cc1C C(C1COCc2ccccc21)NC(=NCC=C)NCC1CCS(=O)(=O)C1 c1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)cc2ccncc2s1 N1(C(C2(SC)CCC2)=O)CCC2(CC(NC(c3ccnc(C(C)C)n3)=O)CO2)C1 C(=O)(C(C)(F)C(=O)NC1CCC(C(=O)NCc2cnsc2)C1)OC c1(C(N(CCCN(C(=O)Cc2c[nH]nc2O)C)C)=O)nn(CC(F)(F)F)cc1Cl N1(C(C=CCC)=O)CCC2(COCC(CNC(=O)CCC3CC(F)(F)C3)O2)C1 C(=O)(C(CCC(C)C)NC(=O)CC(C)C(C)C)NCc1c(C)ncs1 C1(C(=O)NC2(CNC(=O)C(C)Cn3ccnc3)CC(OC)C2)CCCCCCC1 c1(OCC(=O)NC2C(NC(C3CC(C)(C(=O)OC)C3)=O)COC2)ccccc1C c1(C(=O)NCCN(C(=O)C=Cc2ccoc2)CCC)cccc2c1nnn2C N1(C(C(C)OCCC#C)=O)CCC(C)(CNC(C2(C(=O)OCC)CC2)=O)CC1 C(CC(C)C(F)F)NC(C1CCC(CNC(c2c(C)snn2)=O)C1)=O c1(C(=O)NCC2(NC(CC=C)=O)CC2)nnn(C2CC2)c1C(F)F C(C(C)(C(=O)NCC(O)(CO)CO)NC(=O)Cn1cnnc1)SC N1(C(c2c(CCNC(C(C)=CC3CC3)=O)n[nH]c2)=O)CCC(CC2CC2)CC1 c1(C(N2CCOCC(NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc2c(s1)CCC2=O C(=O)(C(C)(C)C(=O)N(C)C)NCC(CCC)NC(c1cnn(C(C)C)c1F)=O n1(CC(=O)N(C)CC2N(C(c3c(OC)csc3)=O)CCCC2)ncc(C)cc1=O Fc1c(C(F)CNC(=O)CCn2cc(I)cn2)cccc1Cl C1(C)(CNC(C2(c3cc(C)on3)CC2)=O)CCN(C(=O)C=C2CCN(C)CC2)C1 CCCCCCC(=O)NC(C)CCC(=O)N(CC)Cc1cccnc1 C1(CC(N2CC(NC(c3n(CC)ncc3)=O)C2)=O)CCCC2(CC2)C1 c1(OC)c(NC(c2cccc(I)c2)c2ccc(F)cc2)nnn1-c1ccccc1 N1(C(C(C)O)=O)CC2CN(C(=O)CCn3ccnn3)C2C1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(OC)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C12CCCCC1NC2=O.CCCCSCC(=O)N(C)CC1(COC)CC1 c1(CC(=O)NC(C(=O)OC)Cc2cn(C(C)C(=O)O)nn2)cncc(C(C)C)c1 c1(COC(c2cc(F)c3cn[nH]c3c2)=O)ccc2nc(Cl)sc2c1 c1(CNC(CC2(CNC(C(CC=CCC)C)=O)CC2)=O)ccc(NC)c(C)c1 c1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)ncc2[nH]ncc2n1 c1(C(=O)NCC(CC)(C)NC(c2csc(C)c2)=O)cn2c(n1)C(C)CCC2 C1(CNC(C2C(OCC)C2)=O)CCCN(C(=O)CN(C2CCSC2)C)CC1 c1(C(=O)NCCCCC(C)NC(c2nc(OC)c(C)s2)=O)cc(N)c(O)c(F)c1 c1(C(=O)NC2CCN(C(C3CCNC3=O)=O)CC2F)nc2ccccc2[nH]1 C(=O)(C(C)CCCC(C)C)N1CCC(C(N(CC(CC)(O)CC)C)=O)C1(C)C C(CNC(C1CCCN(C)C1)=O)(CC(=O)NCc1c[nH]nc1C(C)C)OC N1(C(CCOCCOCC)=O)CCC2(CCCN(C(=O)CN(C)CC)C2)CC1 O=C1CN(CCc2cc(Cc3ccccc3)on2)C(=O)N1Cc1ccccc1 c1(-c2cn(OCCOC)nn2)ccnnc1C CCC(C)CCC(=O)N1CC2CC(N(C)C(c3cnn(C)c3C)=O)C1C2 c1(C(=O)NC2C(CNC(C=Cc3ccc(C)s3)=O)CC2)cnc2[nH]cnc2c1 c1(C(C(N2CC(CCNC(CCCCOC)=O)C(C)C2)=O)=O)ccc(F)c(Cl)c1 c1(C(N(C2CCCN(C(c3scc(OC)c3OC)=O)C2)CC)=O)cncnc1C C1(n2cc(CCCNC(c3nn(C)c(C(N)=O)c3)=O)nn2)CCCC(F)(F)CC1 C1(C)(C(=O)OC)CC(OC)CN1C(=O)CCc1ccncc1 c1(C(N2CCC(CN(C)C(c3cnsn3)=O)C2)=O)cnnc(C2CC2)c1 c1(C(=O)NC2CC3(CN(C(CCC(=O)NC)=O)C3)C2)cc(N)c(Br)c(F)c1 n1(CCC(=O)N(C2CN(C(c3cccs3)=O)CC2O)C)sc2ccccc2c1=O C1(C(N2C3(CNC(c4cc(C(F)(F)F)no4)=O)CC(C2)C3)=O)CCCNS1(=O)=O CC1CN(C(c2ccc(CN(C)C)[nH]2)=O)CCC1NC(=O)C(O)C1CCC1 C1(C(=O)Nc2ncc(C#N)s2)CN(Cc2cccc(-c3ccco3)n2)CCC1O c1(C(=O)NCCOC2CN(C(C3(CC)COC3)=O)C2)cc2ccccc2n1C Cc1c(C(=O)NCC2CCC2NC(=O)C(C)(F)F)sc(Cl)c1Cl C=CCCC(C(=O)NCC1(OC)CN(C(c2ncn(C)n2)=O)C1)c1ccccc1 c1(OC)cccc(-n2c(SC3CC(F)C(=O)N3)nnc2-c2ccco2)c1 CC1CC(=O)NCC1C(=O)NCCCCCNC(c1cscc1C(N)=O)=O C1(CC(=O)NC2CCN(C)C2=O)CC(C)(C)CN1C(=O)Cc1csnn1 N1(C(c2c(CC)[nH]cc2)=O)C(C(=O)NCC(C(C)(C)C)OC)CC2CC12 CCC(C)CC(=O)NCC(CC(=O)NCc1cccnc1O)OC c1(OC)cc(CN(c2cc(NCc3ncc(Br)s3)ncn2)C)ccn1 c1(OC)ccc2cc(C(N3CCCC3)NC(=O)C=C3SCC(=O)N3C)c(Cl)nc2c1 C1(C(=O)NCCN2CCNC2=O)CC12CCN(C(=O)CC1CCCCC1)C2 C1(CNC(c2c(C)nccn2)=O)CCC(C)(C)CN1C(C1C(C)C1(F)F)=O CC1(C)Cc2cc(Br)ccc2C1NC(C1CCC2(CC1)CSC2)=O N1(C(=O)NCC(C(F)(F)F)c2ccccc2)CC2(CCSCC2)C1 Cc1cc(C)c(C(=O)NCC2CC(C)CN(C(=O)Cc3ncoc3C)C2)cn1 N1(C(C2N(CC)CCOC2)=O)CC2CCCC(C1)N2C(=O)Cn1cnnn1 c1(CNC(C2(SC)CC2)=O)ncc(C(=O)N(C2CCCC(O)C2)C)cn1 Cc1cc(C(=O)NC2CC2NC(=O)CC23CCCC2C3)no1 Cc1cc(Nc2nc(F)ccc2F)c(F)cc1F C=C1CCN(C(=O)CCNC(C)=O)C(C(=O)NCCC(F)(F)CC)C1 c1(CNCC2CC(C)SCC2)cnc2sc(Br)cn12 c1(C(=O)NCC2(F)CC(NC(C3(C4CCCO4)CCCC3)=O)C2)cccc(=O)o1 Cc1ncc(N)cc1C(=O)NCC(O)CN(C)C(c1csc(Br)n1)=O CCCCC(F)C(=O)NCCC(C)(C)C(=O)NCCC(=O)NCC(C)C C1(SCCOCCN(C(CN(C(C)=O)C)=O)C)CCCN1C(=O)Cn1cccn1 C(=O)(CCN=c1ccc(C)c[nH]1)OC.C1(=O)C(C)N1CCC1(CC)CC1 N1(Cc2cnn(CC)c2C)CCCCC(c2ccccc2)C1 S(=O)(=O)(CCc1ccccc1)N(C(C1C=CCC1)=O)C1CC1 Cn1cnn(CCC(=O)NCC2CN(C(C3CCCC3)=O)C3CC23)c1=O c1(C(=O)NC2CN(C(c3scc(C(N)=O)c3)=O)C(CO)C2)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(=O)CC2(O)CCCOC2)=O)CCC2CC1C(=O)O2 CC1CCOCCN1N1CCCC(Oc2ccc(F)cc2)C1 C12(NC(C3CC3NC(c3nc(N(C)C)oc3)=O)=O)CCC(COC)(CC1)C2 C1(C(NOCCC=C)=O)C(C)CCN1C(=O)NC1(n2cccc2)CC1 C1(C(=O)Nc2cc(O)nc(C(F)F)n2)CC12CCN(Cc1cccnc1O)CC2 C(C(=O)N1OC2C=CC1CC2)NC(CONC(=O)Cc1ccc(F)c(F)c1)=O C1(C(=O)NCC(=O)NC2CC(OCC(c3ccccc3)C)C2)CCC2(CCC2)O1 c1(SCC(N2C(c3cn(CC4CC(=O)OC4)nn3)CCC2)=O)cccc(Cl)c1 Cc1ccc(Cl)cc1C(C)N(C1CCN(C(c2ccccc2)C)CC1)CC1CC1 N1(C(c2ccc(OC)o2)=O)CC(C(=O)NC2CC23CCOCC3)C2(CCC2)C1 C(=O)(CC(C(C)C)C(C)C)NCC(CNC(C(CC(C)C)OC)=O)C c1(C(=O)NC2(C)CCN(C(CC3N(C(C)C)CCC3)=O)C2)ccc(N)c(SC)c1 c1(SCCn2cc(C(N3CCOCC3)(C)C)nn2)cnn2c1CCC2 c1(C(=O)OC)ncnc(SC)c1OCCOCCNC(=O)NCCCOC C(CC(C)C)(C(=O)NCCc1ccoc1)NC(C(CC)OCC)=O N1(C(CSC(=N)N)=O)CC2ON=C(CCNCC(=C3CCSCC3)F)C2C1 CC1(C)CCC=C(C(=O)NCCCC(C)(C)NC(=O)CCc2cnco2)C1 CC1CC2(CCN(C(=O)CCCN3CCCC3)CC2)CN1C(C12CCC1C2)=O C1(C(=O)Nc2cccc(NC(c3n(CCC)ccc3)=O)c2)CC12CC(C)(C)C2 Cc1cc2[nH]c(C(=O)NCC3CC(C)(C)CN3C(=O)CSCC#N)cc2o1 C(CN=c1[nH]c(=NCC(C)(C)CC(C)C)[nH]c2cccnc12)SCC=C c1(C(=O)NCCCCN(CCCNC(=O)CC2C=CCCC2)C)cc(Cl)cn1C N1(C(C(C)SC)=O)CCC(C(C)(C)C)(COCCNC(=O)CCn2ccnn2)C1 Cc1nc(=NCC(CC(C)C)NC(=O)CCC2CC2(Cl)Cl)s[nH]1 CC1CC(F)(F)CN1C(=O)C(=O)NCC(c1cc(F)cc(Cl)c1)N CCC(C)C(O)C(=O)N1CC(F)CC1CNC(c1sccc1C1CC1)=O c1(C(=O)NCC2CN(C(C(C)(C)OC)=O)CC2C)cc2cnccc2cc1F CC1CN(N2CCCCC2c2cncnc2)CCC1(F)F c1(CC(N2CCCOC(CC)C2)C(=O)NCCSCC)cc(F)c(F)c(F)c1F Cc1cc(CN(C)C)nc(NC(C2CC(F)C2)=O)n1 Cc1nc(C(C)C)ccc1C(=O)NCC12CCC1CN(C(c1ccccn1)=O)C2 c1(NC(C2C(NC(CC(=O)N(C)C)=O)C2)=O)ccc(Cl)cc1 CN1CCN(C(=O)CC2(C)OCCO2)C(C(=O)NCCC2CCC(C)(C)O2)C1 C=C(Br)CCC(=O)NCC1(n2ccnn2)CC1.c12cn(nn1)C1CN(C1)C2=O Cn1cc(CC(N2CCC2CNC(c2cncnc2O)=O)=O)c(Cl)n1 N1(C(c2c(OC)cc(F)cc2)=O)CC2CCN(Cc3occc3OC)C2C1 C1(NC(C(C)(C)OC(C)=O)=O)COCCC1NC(c1cnc(C(F)(F)F)nc1)=O N1(C(C)=O)CC2CCC1CN2N1C(C(=O)OC)CCC1C1CC1 N1(C(CCC=CCC=C)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC12 c1(NC(C(CC)(C)C)=O)ccc(OC)cc1O.C12CN(CC1F)C(=O)N2C c1(NS(CC)(=O)=O)cccc(F)c1C(=O)Nc1cc(OC)cc(Br)c1 C1(C(=O)NCCC(CCNC(c2n(CC)cnn2)=O)C)CCCC(C)(C)CC1 c1(OC)cccc(C2CC(C)CN2C(N2CC3(CCC3)C2)=O)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2C)=O)cc(C)c(C)cc1C c1(OC)cc(C(=O)NC23CCN(C(=O)Cc4cnoc4)CC2C3)ccc1OC C1(NC(N2CC(c3ccccc3)(C(=O)OC)C2)=O)CC2CCC1N(C)C2 Cc1nc(C)n(CC(=O)NCC2CC2CC(=O)NCc2cnco2)n1 C12(C(=O)NC3C(CNC(C4=C(C)CCC4)=O)CCCC3)CC3CC(CC(C3)C1)C2 C1(NC(CCC=C=C)=O)CCCCCN(C(c2ncc(Br)cc2F)=O)C1 C1COCCN1CCOC.c1(SN2CCC(N(C(C)=O)CC)C2)ccccc1Cl N1(CCC(=O)NC2C(NC(=O)CNC(c3ccoc3)=O)C2)CCCCC1 C=C(Cl)CC(C(=O)NCC(N1CCCC1)C)NC(=O)CSCCCN C1(NC(C2(NC(=O)COCC3CCC3)CC(CO)C2)=O)CC(C2CCC2)C1 C1(CC(=O)NC2CC(C(C)NC(C(C)CN(C)C)=O)C2)OCCCC1(C)C C1(C(=O)NC(c2ccc(O)cc2)C)C(O)CCN1C(c1ccc(F)cc1)=O c1(NCC(C2CCC2)OCC)ncccc1S(=O)(=O)NCC1COCC1O N1(C(CC(CC)C)=O)CCC2(CCC2)C(NC(C2CN(C)C(=O)N2)=O)C1 CC(C)C(=O)C(=O)NC1CCOCC1C(=O)NC(C1CCCC1)C CON=C(C(=O)NCC1CCN(C(=O)CC(C)(C)O)C(C)C1)c1ccco1 C(C(CCC)C(=O)NCCC(C)c1cn[nH]c1)NC(C=CCC)=O C=C=C(C)CC(=O)NC1COCC1C(=O)NCCCC(=C)C c1(CC)c[nH]nc1C(=O)NCCCN1CCC(NC(c2cc(Cl)c[nH]2)=O)C1 c1(C(=O)NCCCOc2nnc(C)s2)ccc(C(F)C(F)(F)F)cc1 n1(CCCOC(C)C)nc(-c2cccc(OC)c2)nc1C1CC1CF N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(=O)C(C)n2cccn2)CC1C c1(C(C(=O)NC2COC2)N(C)Cc2c(C)noc2C)ccc(S(N)(=O)=O)s1 C(CC(C(C)(C)C)NC(C1CCC1)=O)N(C(=O)C(c1ccc(O)cc1)(C)C)C C1(C(=O)NCc2nc(CNC(C(C)n3ccnn3)=O)sc2)CC(=O)NC(=O)C1 C1(NC(c2cccc(OC)c2F)=O)CC2CC(NC(C3CC=CCC3)=O)CC2C1 O=C(NNc1ccnc(Cl)c1)NCCCCCCc1ccccc1 C1(C(=O)OC)CN(C(c2onc(C)c2I)=O)CC2(CCC2)O1 N1(C(C(=O)NCc2ccccc2)C2(CC)CC2)CCC2CCCC2C1 C1(NC(C(CCOCC)NC(=O)CC2CCC(=O)CC2)=O)CCOCC1(C)C C(C(N=[N+]=[N-])C(=O)N1CCC(CN(c2nc(C)cc(C)n2)C)CC1)OCC C(CC(=O)NCC(O)CNC(=O)CCCOc1ccc(C)cc1)(C(F)(F)F)OC C(CN=c1ccnc(N2CCC(n3ccnc3)C2)[nH]1)OC1CCN(C(COC)=O)C1 CN1CCCC1(C)C(=O)NCC1CCN(C(c2cc(Br)c[nH]2)=O)C1 C1(C(N(C(C)C)CCN(C)C(c2cc(Cl)n(C)n2)=O)=O)CCN(C)C(=O)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(CCCC#C)=O C1(C(N(C)Cc2nnc(CC)o2)=O)CCCN1NC(=O)COCCC(C)C n1(CC(C)C)ccc(CNC(c2nnnn2C2CCCC2)C2CCSCC2)n1 CCC(C)(C)C(C)CC(=O)NC(C1CCCN1C(C1CC(S(C)(=O)=O)C1)=O)(C)C C(CC(=O)NC1(CCCF)CC1)N(C(=O)CN(C)C)CC C1(CC(=O)NC(CCC=C)C)CCCC(NC(c2cccnc2O)=O)C1 CC(C)(C)C(C(=O)NCc1cc[nH]n1)NC(c1cn[nH]c1)=O C1(C(CNC(C)CCC2CCCO2)(C)C)CCN(C(=O)OC(C)(C)C)CC1 C1(NC(C(C)(C)OC)=O)CCCCC1CNC(=O)Cc1ccc(C(=O)OC)cc1 c1(CC=C)cc(-c2nc(-c3cscn3)nn2C)cc(OC)c1OC c1(CNC(c2cnc(CS(C)(=O)=O)s2)=O)ccc(Cl)cc1Br C1(NC(c2cc(NC(C)=O)ncc2)=O)CN(C(C23CCC2C3)=O)CC2(CCC2)C1 c1(C(N2CCC(C(CNC(COCCC)=O)(C)O)CC2)=O)c(F)cc(O)cc1F c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)(C)C2CCC2)cc(F)c(C)cc1N C1(CNC(C=Cc2n(C)ncc2)=O)CCN(C(c2cc[nH]c2)=O)CCC1(F)F N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOCC(C)(C)C)C)CC1 Cc1nn(C)cc1CNC(C1CC(O)CN1C(=O)Cc1cnn(C)c1)=O Cn1nccc1CCNC(=O)CCC1CC(NC(C2CCC2C#N)=O)C1 C12(NC(c3c(Cl)c(C)n(C)n3)=O)CCCN(C(=O)C(N)=O)CC1C2 C(CC(C(=O)N(C1(C)CC1)C)NC(C1CCS1(=O)=O)=O)OC c1(NC)ccc(C(=O)NC2CCC2NC(=O)C(c2c(C)cccc2C)O)cc1F C12(CNC(CC(C)(C)OC)=O)CN(C(=O)C=C3CCOCC3)CC1(C(F)(F)F)C2 Cc1cc[nH]c1C(=O)NCC1CCC(NC(=O)CSc2n[nH]c(O)n2)C1 N1(C(Cc2c(CC)con2)=O)CC2CCC2(CC(=O)NCc2cnccc2Cl)C1 C1(C2CCC2)(CNC(=O)C(N2CCC(N3CC=CC3)C2)=O)CCNCC1 N1(C(C(CC)N(C)C(c2cccnc2N)=O)=O)CCOC(CN(C)CC)C1 c1(C(=O)NCC2(C#N)CCOCC2)ccc2c(n1)CN(C(C1C=CCC1)=O)CC2 C1(C(N2CCC(NC(C(C(CC)C)OC)=O)C2(C)C)=O)CCn2ccnc2C1 N1(C(c2ncn(C(C)(C)C)n2)=O)CC(C2CN(C(c3coc(C4CC4)n3)=O)C2)C1 c1(CC(N2CC(CC)C2)=O)nc2ncccn2n1.C12(C)CC(C1)C(=O)N(C)C2 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1ncc(C)[nH]1 c1(C(N2CC3(CC(NC(c4cnc(C)c(N)c4)=O)C3)C2)=O)cccc2c1OCC2 C=C1CN2C(=O)CCC2(C(=O)NCCCCCN(C)C(C2CCNC(=O)C2)=O)C1 C(C(C)(C(C)C)NC(c1cnn(C)n1)=O)NC(C(Cc1ccccc1)OC)=O c1(C(=O)NCc2ccccc2Br)nc2ccccn2c1-c1cccc2c1OCC2 C1(C(=O)NCC(CCNC(C=CC)=O)O)N(C(=O)OC(C)(C)C)CCC12CC2 C=C(C)CC(C(=O)NCC(c1ccco1)O)NC(c1sccc1C)=O C12(CNC(c3[nH]cc(C)c3)=O)CCCN(C(=O)COc3cccc(C)c3F)C1C2 C1(C(N2CC3(CN(C(C4C(C)(Br)C4)=O)C3)C2)=O)Cc2ccccc2N1 CCC(CNC(c1ccc(C(C)(C)O)cc1)c1nnnn1C1CCCC1)CCO C1(C(=O)NCC(CN(C)C)O)COCCN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CCC2(CC1)CN(C(c1cnco1)=O)CCO2 c1(C(=O)NCCCCNC(CC2(OC)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(Cc2cn(CCCCOC(C)=O)nn2)=O)COC2CCCCC2C1 c1(CN2CC(C(C)C)C(C)C2)ccc(C(c2ccccc2)=O)c(Cl)c1 C1(CC)CN(C(C2CCC2(C)C)=O)CCC1NC(=O)CCCn1cncn1 c1(NCC(c2ccccc2)NC(c2ccc(C)[nH]2)=O)cc(O)ncn1 CC1CN2CCN1C(C(=O)NCC#CCNC(C1CCOC(=O)N1)=O)C2 N1(C(c2cc(C)oc2C)=O)C2CCCC1CC(NC(c1ccnc(C)c1N)=O)C2 c1(C(=O)NCC2(C)CCC(NC(COCCOC)=O)C2)nc(C)ncc1Br N12CCCC(C)(CC1)C2.Cc1nc(C(C)C)oc1CCNC(=O)OC(C)(C)C c1(SC)ccc(C(=O)NC(C)C(C)NC(c2ncnc(O)c2F)=O)cc1[N+](=O)[O-] c1(C(C)C)ccc2occ(C(=O)NCC3CN(C(=O)C(F)C(C)C)CC3C)c2c1 c1(C(=O)NC2CCCC(N(C)C(c3ccc(F)s3)=O)C2)csc2ncnc(O)c12 N1(C(CCOC(C)=O)=O)CCC2CC2(C(=O)Nc2cccc(CCF)c2)CC1 C(C)(C)(CC(F)(F)CC)NC(C(OC)NS(C)(=O)=O)=O C1(c2n(CCOC)nc(-c3ccc(C(C)(F)F)nc3O)n2)COC2CCCCC12 N1(C(c2cccc(OC)n2)=O)CC(C)CCC1C(=O)NCc1sccc1C N(C(=NCCN1CCOC1=O)N1CCCC2(CCOC2)C1)C1CCS(=O)(=O)C1 C(C(=O)Nc1ccc(-n2cnnn2)cc1)(C(C)C)OCC(C)C c1(C(N(C(C)(CN(C)C)NC(=O)OC(C)(C)C)C)=O)ccc(C(F)(F)F)c(Cl)c1 C1(NC(=O)CCc2csc3ccccc23)Cc2nc3ccccc3n2C1 c1(C(=O)NC2C(CNC(CCCOCC=C)=O)CCC2)cncc(N(C)C)c1 Cc1cccc(C)c1C(=O)NCC(=O)N(CCC(C)NC(=O)C(C)C(C)C)C c1(N2CCC(c3c(OC)cccn3)C2)nc(N2CCC(C#N)C2)c2sccc2n1 C1(C(=O)NCC(=O)NCC(F)F)COCCC1NC(C1SCCS1)=O c1(OC)cc(OC)cc(C(=O)NC(C)CN(C)C(c2c(C)ccnc2Cl)=O)c1 Cc1cccc2[nH]cc(C(=O)NC3(C)CN(C(=O)Cc4n[nH]c(=N)s4)C3)c12 c1(CCCC(=O)NC(C)CN(C(=O)CCN2CCCCC2)C)ccc(O)cc1 c1(C(=O)NCC(CNC(C(CC=C)(C)C)=O)C(F)(F)F)cc2nc[nH]c2cn1 C1(OC)CC2CCC(C1)N2C(c1coc(C(C)NC(c2ccc(C)o2)=O)n1)=O O(NC(=O)CC1(N(C)C(c2c[nH]cc2C(C)C)=O)CC1)CC(C)C C(=O)(C#CC1CCCO1)N1C2CC(CNC(C=C(C)C(C)(C)C)=O)C(C2)C1 CCC(CC)(CCNC(=O)C(SC)SC)NC(=O)CCSc1ccccn1 N1(CC(=O)NCC(=C)CCNC(=O)C(C)(C)F)CCC(OCC(F)F)CC1 C(=O)(C(C)CC1CCCCC1)NC1CC(NC(C(c2ccccc2)OCC)=O)C1 c1(C(N2CCC(C)(NC(C(CC(C)(C)C)O)=O)C2)=O)cc2ccccc2nc1O c1(OC)cnc(C(=O)NC(C)(C)CCNC(C2(CO)CC2(F)F)=O)nc1 N1(C(C)=O)CCC(c2nnnn2C)(NC2CC(=O)N(C)C2)CC1 CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1NC(C1Cc2cscc2C1)=O C1(C(=O)NCc2cc(OC)ns2)CN(C(C2CCCC2)=O)CC12CC2 C(C1(O)CCc2cc(F)ccc21)NC(N1CC(C)(C)C(C(N)=O)CC1)=O Cc1cc(C(=O)Nc2ccc(NC(C)(C)C)cc2)c2c(O)nn(C)c2n1 c1(C(=O)NCC2(CNC(c3cc(CC)no3)=O)CC2(F)F)cc(CC)oc1C CCC(C)(CC)C(=O)N1CCN(C2CN(C(=O)COCCCF)C2)CC1 N1(CCNC(=O)Nc2ccc(CN3CCCC3)cc2)CCOCC12CCC2 C#CCC(C)C(=O)NC1CCCC1CNC(c1occc1-c1ccccc1)=O C#CC1(O)CN(C(=O)CC2(NC(=O)Cc3cncs3)CCC2)C1 N1(C(=O)Nc2cccc(Nc3cccc(OC)n3)n2)CCCC(C)(F)C1 CCCCC(C(=O)NCC12CC1CN(C(=O)C(CO)N(C)C)C2)N(C)C Cn1ccc2cc(CC(N3CCC3CNC(=O)CCCc3ncco3)=O)ccc12 c1(CC)nc(C)ncc1C(=O)NC1CCCC(NC(=O)CC(C)(C)C#N)CC1 CN1CCN(C(C2CCCN2C2CC2)=O)C(C(N2CC3CC2CN3C)=O)C1 N1(C(C=CC(C)NC(C(C)C2CCC2)=O)=O)CCOCC12CC2 C1(C(=O)NC(Cc2cc(C)[nH]n2)C)C2CCN(C(C3(CO)CC3)=O)CC12 c1(C(N2CCCC(O)(CNC(CS(CC)=O)=O)C2)=O)cc(Br)c(C)nc1O C(=O)(C(COC)CC(C)C)NCCCOCC(C)(C)NC(C1(CC)CCOC1)=O C1(NC(c2c(CC)noc2)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1O C1(CNC(C(C)(C)n2cccn2)=O)CN(C(=O)CCC2OCCO2)C2(CCC2)C1 CN1N=C(CC(=O)NC2CC3COCC(C2)N3C(=O)CSC(F)(F)F)CC1=O C12(C(N3C(CNC(=O)CSc4ccncc4)CC(OC)C3)=O)CCCC1C2(F)F c1(C(=O)NC2CC(CNC(C=CCOCCOC)=O)C2)c[nH]c2nc(Cl)ccc12 N1(C(=O)CC2CCCN(C(c3ccc(O)cn3)=O)C2)CCC2(CCCO2)CC1 N1(C(C2CC(=O)NCC2)=O)CC(NC(c2c(Br)cncc2Br)=O)C(F)(F)C1 C(CC(C)C)(C(=O)NC1CCN(C(=O)C(C)CC(N)=O)CC1C)NC(C)=O C(=O)(C1=CCCSC1)N1CCC(CNC(CCc2ccc(=N)[nH]c2)=O)CC1 N1(C(C2C(OC)CC2)=O)C(C(N2CCC(O)C2)=O)C2CC(O)C1C2 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCNC(c1cc(Cl)cs1)=O N1(C(C(CSC)C)=O)CC(NC(c2ccn(C)c2)=O)C(c2nccn2C)C1 C1(CC)CN(C(=O)C(O)C2CC2)CCN1C(c1ccc(C(C)(F)F)cn1)=O c1(C(N2C(C(=O)NCCCNC(=O)OC)C(C)CC2)=O)ccc(F)c(C)c1F C1(NC(c2c(C)nsc2)=O)CC2(C1)CC2NC(=O)CCn1ccnn1 N1(C(CCC=C)=O)CC(=O)N(C)CC1C(=O)OC.c12cn(nn1)C2c1csc(Br)n1 C1(C)(CNC(c2c(C)n(C)nn2)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C1(C(N2CC3C(CNC(=O)CCc4ccoc4)(C3)C2)=O)CCC(F)(F)CC1 c1(C(=O)NCCN(C(C23CC(F)C2C3)=O)CC)ccc(CO)cc1F C(=O)(CC(CC(C)C)NC(=O)Cc1sccc1C)Nc1c(C)ccc(C)c1 C(CC(C)CC)(C(=O)N1CCn2cnnc2C1)NC(c1cncc(C#C)c1)=O c1(OCC(=O)NCCCC2(NC(C(C=C)O)=O)CC2)ccc(F)cn1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)NCC#CC)CC(C)C c1(C)nc2cc(C)cc(C)c2[nH]1.C1(C)C2(CC2)C12CC2.CN=C1NN2CCC(N1)C2 O=C1CCC(C(=O)N2CC3CC3(C(=O)Nc3nccc(C(F)F)c3F)C2)=NN1 C(C(C)(CO)NC(=O)OC(C)(C)C)N(C(C1(CCNC)CC1)=O)C CN1CCN(C(C2N(C(c3ccc(C#N)cn3)=O)CC23CCCC3)=O)CC12CC2 c1(CN(C(C2(n3cc(Cn4c(C)nc(C)n4)nn3)CC2)=O)C)ncc(Cl)cc1Cl C1(NC(C2(C)CCC(F)(F)CC2)=O)Cc2ccccc2C1NC(C1CCC1)=O C(=O)(C(C)CC(C)C)N1C(CNC(CCC(=O)NCCC)=O)CCCC1 c1(CC)ccccc1C(=O)NCC1CCN(C(C2C3CCCC23)=O)C1 N1(C(C2N(C(c3cc(C)sc3N)=O)CCCCCC2)=O)CCC(C2=NOCC2)C1 C(N=c1[nH]c(Cl)ncc1C(=O)OC)C1CN(C(CN(CCC)C)=O)CC1(C)C CC(C)C(CNC(=O)Cc1ccc2c(c1)CC2)C(=O)NC1CCC(=O)NC1 N1(CC)CC(NC(=NC)NCC2(C)CCCO2)CC1=O CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CC2)=O)CC1C C(C)(CCC(=O)N1CCCC1(C)CNC(=O)CCc1cnco1)OCC C1(C(N2CC(NC(C3C(C=C)C3)=O)CC2(C)C)=O)CCC(=C(F)F)CC1 CN1CCc2nc(O)c(C(=O)NCC(O)CCNC(C3CC3C(N)=O)=O)cc2C1 C(=O)(CC(C)C(F)(F)F)NCC1(C(=O)NCC23CCCC2CCO3)CCCC1 C1(C(N(C(C(N2CC(O)(C(C)C)C2)=O)C2CC2)C)=O)CC2(CC2)CN1C N1(C(CC(C)c2cnn(C)c2)=O)CCN(C(=O)Cc2cnoc2)C(CCO)C1 C1(NC(c2nc(CCC)oc2)=O)CCCC(N=c2[nH]nc(COC)s2)C1 c1(C(N2CC(CC(C)NC(=O)C(O)c3ccsc3)C2)=O)cnc2c(c1)COC2 C(=O)(C(CCC1CCCOC1)N1CCOC(COC(C)=O)C1)NCC(C)C C#CCC(C(=O)N(C1CCN(C(C2(C3CC3)CC2)=O)CC1)CC(C)C)C1CC1 c1(C(=O)OC)cc2c(s1)CN(C(=O)C(C1CCCCCC1)C)CC2 C1(C(=O)Nc2c(Oc3ccc(C)cc3)cccc2)CC2CSCC(C1)C2 N1(C(c2[nH]nnc2C2CC2)=O)CCC(N(CCO)C(c2snc(O)c2Cl)=O)CC1 C1(NC(c2c(C)csc2Cl)=O)CN(C(=O)C(F)C(F)(F)F)CC1(C)C c1(C(=O)NCCOCCNC(C(CC#C)CC#C)=O)ccc2[nH]ccc2c1F C(=O)(C(F)(CNC(C1(O)CCC1)=O)C(C)C)NC1C(C(C)O)CCC1 C1(CNC(C=CC=CC)=O)CN(C(c2cccc(-n3cccc3)n2)=O)CCC1C C=CC(CCC)CC(=O)NC1(C)CCCC1NC(=O)CCc1cc(Cl)cs1 CC1N(C(=O)CCC2CCCN2C(C2CC3CCCC3C2)=O)CCC1(C)C C1(CCCNC(C(CC)N(CC)CC)=O)CCCN(C(c2ccc(C)o2)=O)C1 C(=O)(CC(C)(O)c1ccccc1)NCCOC(CC)C(=O)N1CC(NC(C)=O)C1 CON(C)C1CCN(CC2CCS(=O)(=O)C2)CC1 Cc1nc(C(=O)N(C2CCC(NC(=O)C(C)(C)n3ccnn3)C2)C)c(C)o1 Cc1cn2c(n1)CCC(n1cc(CNC3CNC(=O)C34CC4)nn1)C2 C1(C(=O)NC(CNC(C(C)=C(C)C)=O)C)(C(F)F)CC1(F)F C1(NC(c2cc(Cl)ccn2)=O)COC2(CNC(C3(C(F)(F)F)CCC3)=O)CC1C2 c1(SCC)c(NC(C2CCOCC2)(C)C)cccc1F Cn1c(C(N2CCCCC2C2(NC(=O)C=CBr)CC2)=O)ccc1C1COCCO1 CCC1=NOC(C(=O)NC(CO)C(=O)NCCc2ccon2)C1 c1(C(=O)NCC2N(C(C3(C)CC4CC4C3)=O)CCC2)cnc2[nH]nnc2c1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(=O)CC2(C)CC(F)(F)C2)C)n(C)n1 S(=O)(=O)(c1cccc(=NCC(C)(C)C(C)O)[nH]1)N(CCOCC=C)C N1(C(Cn2c(C)ncc2)=O)CCC2(CCCN(C(=O)CC3CCCOCC3)C2)C1 c1(OC)ccc(CN2CCCC(C(=O)NC3CCC(F)(F)C3)CC2)c(Br)c1 c1(CN2CCC(CC(=O)CCn3c(C)ncc3)C2)nc(-c2nccs2)nn1C C1(C(=O)NCC(Cc2ccccc2)NC(c2ccoc2)=O)CCC12CCOCC2 c1(C(=O)NC2C(NC(=O)CC3CCOC3)C2)cc2n(n1)CC1(CC1)CO2 C=CCCC(C(=O)N1CC(N(C)C)C(C)C1)NC(c1cc(C2CC2)on1)=O N1(C(c2c(=N)[nH][nH]c2)=O)CCC(F)CC1C(=O)NCC1CC2CCCC2C1 C1(NC(COC)=O)CN(C(c2cccc(C#N)c2)=O)Cc2ccnn2C1 C1(C(=O)OC)(CC)CCCN1C(C)=O.C12CCCN1NC2=O C1(CNC(CCCN(CCCC)CCCC)=O)CC(NC(=O)C(C)O)C(O)C1 C(CS(=O)(=O)CC(=O)NCC1(C(=O)NC2CCC(=O)N2)CC1)OC C1(CCC)(NC(c2cc(CN(C)C)on2)=O)CCN(C(=O)CC(C)C)CC1 C1(CNC(c2cc(C)oc2)=O)CC(F)(F)CN1C(c1coc(C)n1)=O N1(C(CC2(OC)CC2)=O)CC(F)(F)CC1CNC(c1cnc(-c2cccs2)s1)=O C1(OC)CC(N(C)C(c2ccccc2F)c2nn[nH]n2)C12CCC2 N1(C(C(C2CN(C(=O)CCCc3ncco3)C2)OC)=O)CC2CCC(C1)C2C#N c1(C(N2CCC3(CCN(c4ncccn4)C3)C2)=O)cc(Br)cc2cn[nH]c12 C1(C(C)C)(C(=O)NCc2cccc(O)c2)CCN(C(c2ccc(C(N)=O)s2)=O)C1 N1(C(C=CC=CC)=O)CCC(NC(c2ccn(CCO)c2C)=O)C1CC C1(CCC(=O)NCC=C(Cl)Cl)CCN(C(=O)C(C2(O)CCCC2)F)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(=CCNC(C2CCC(=O)N(C)C2)=O)CC1 N1(C(C(n2ccc(C)n2)C)=O)CC(NC(c2cc(C)sn2)=O)C(n2cccn2)C1 C1(NC(C2C(C)C2)=O)CC(N=c2[nH]ccc(C#N)c2[N+](=O)[O-])C12CCC2 C1(CCO)(CNC(c2n(CC=C)nnn2)c2csc(Br)n2)CCCCC1 c1(C2CC(C(N(CCN(C(C(c3ccccc3)C)=O)C)C)=O)C2)ccc(Cl)cc1 C1(C#N)(C(N2CC(O)C2)=O)CC2CC2C1.C12CCN(CC1)C2=O.C1(C(C)=O)CCCSS1 C12(C(=O)NCCCCCN(C(CC(=O)NCC#C)=O)C)CCC(CC)(C1)OC2 c1(C(N(C2CCN(C(Cc3c(OC)nccc3)=O)C2)C)=O)cccc(F)c1Cl C(C)(CO)(C(C)(C)O)NC(c1c(C)nc(CNC(C2CC(C)(C)CO2)=O)o1)=O c1(C(=O)NC(CN(C(C(F)OC)=O)C)C)cc(N)cc(O)c1 c1(C(N2CC3CC(NC(COCCOCC)=O)C3C2)=O)c(C)nc(O)nc1C c1(C(=O)OCC)ccc(S(=O)(=O)Nc2cn(C3CCCCNC3=O)nn2)n1C C(=O)(C1=NOC(C)C1)N(CC(C)NC(=O)CS(C)(=O)=O)CC c1(C(N2C(CCc3cn(CC(=O)O)nn3)CCC2)=O)ccc(-c2nccs2)cc1 c1(CC)nonc1C(=O)N(CC(C)(C)CNC(c1cnc(C2CC2)o1)=O)CC N1(CC)CC(C(=O)OC)CC1C(=O)Nc1cc(NCCc2ccnc(C)c2)sn1 Cc1cc2cc(NC(c3ccc(OC4CNC4)cc3)=O)ccc2[nH]1 C(N=c1[nH]c(N2CCCC2c2ccc(Cl)cc2)nc2c1CSC2)c1cc(C)ns1 CC(C)CCC(=O)NCC1(NC(=O)CC2CCCN2C)CCOCC1 CC1C2CCC(C2)C1C(=O)NC1CC2(C1)CC2NC(=O)CC1CCC(C)(C)C1 C(CCCC(C)(C)C(=O)NNC(=O)CCCC1CCC1)NC(c1c(C)occ1)=O C1(C(N(C)CCOCCNC(=O)CSc2nccs2)=O)CCSCC1 c1(CN2CCC(c3nc(C)on3)CC2)cc2c(cc1Br)OCO2.C12CC1NC2=O C(=O)(C1=C(Cl)CCCC1)N(CCC(=O)NCC1CC(O)C1(C)C)C C(=O)(C1=CC2C=CC1C2)NCC1CCN(C(Cn2c(C)ccc2C)=O)C1(C)C c1(C(N2CC(CN(C(CCC=C=C)=O)C)OCC2)=O)ccc(F)c(F)c1F C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)CN1CSCCSC1 N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)C2CC12 C1(OC)CCCCC1N=c1cccc(S(=O)(=O)NCc2cncn2C)[nH]1 CN1CCOC(C)C1.C1(C(=O)N)C2CC1N(C(C13CC(CN1C1CC1)C3)=O)C2 CN1CCC(C(=O)NC2(C)CCN(C(=O)CC3(C)CC3(F)F)CC2)S1(=O)=O N1(C(C2CCC(CC)CC2)=O)CCC2CN(C(=O)C3=CCCSC3)C2C1 C(C1(C)CCOCC1)=CC(=O)NCC1N(C(C2C(OCC)C2C)=O)CCC1C C12(NC(C=CC)=O)CC3CC(C1)CC(NC(=O)C(C)CSc1ccccc1)(C3)C2 c1(NC(=O)NCC2CCCC2F)ccc(Cc2cn(CC(N)=O)nn2)cc1 C12(C(=O)NCC3CCC(NC(c4c(C)cnn4C)=O)C3)CCC(N=[N+]=[N-])(CC1)C2 C(CNC(=O)Cc1ccc(OC)cc1C)(C(C)C(C)C)NC(CS(=O)(=O)NC)=O C=CCC(CNC(=O)C(C)(C)C(O)C(C)C)C(=O)NOCC(N)=O Cc1ccc(F)cc1CC(=O)NC1(C)CC(NC(=O)CN2CCCCS2(=O)=O)C1 c1(NC(C(CCSC)NC(=O)CC2CCCC23CC3)=O)ccc(O)c(Cl)c1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(F)(F)C1 CC1OC(=O)NC1C(=O)NCC12CC1CN(C(=O)CN(C)C(=O)C1CC1)C2 CC1CC(C(=O)NCC2CCCC2NC(c2ccc(C(F)F)cn2)=O)CCC1=O C#Cc1ccc(COC(C2(c3ccccc3)CNC(=O)C2)=O)nc1 C(=O)(CCC(=O)C(C)(C)C)N1CCCC(C(=O)Nc2c(C)ccc(OC)c2)C1 c1(C(=O)NC2CCC(CNC(=O)C=Cc3cc[nH]c3)C2)cnnc(O)c1 N(CCC=O)(CCN(C)CC)OCCOCCOCCC(=O)O C1(NC(c2cn(CC)nc2C)=O)CCCC12CN(C(c1sccc1COC)=O)C2 CC1CCCN(C(C2C3CCC2CC3)=O)C1CNC(=O)CN(C1CCC1)C C1(CNC(c2ccc(NC(C)=O)s2)=O)CC2CCC1N2C(=O)C(C)c1ccsc1 N1(C(C2(CC=C)CCCCC2)=O)CC2(CC(NC(c3ccc(C)s3)=O)CO2)C1 c1(CCC(=O)N(C(C)CNC(=O)CC2CCC(=O)N2)C)nc2ccccc2s1 C1(CNC(CNC(CCCCC)=O)=O)CC2(CCC2)CN1C(C1CC1C(C)O)=O N1(C(C2(C)CC2Br)=O)CCC2(COC(CNC(c3c(F)cccc3F)=O)C2)C1 C1(CN(c2cc(N3CC(C)OC(C)C3)ncn2)C2CC2)CC(F)(F)C12CCC2 c1(NC(C(C)OC(c2c(C)n[nH]c2)=O)=O)ncccc1C(F)(F)F c1(-c2nc(CC(CC)C)nn2C(C2CCC2)C)ccc(F)c2occc12 C1(NC(=O)Cc2ccncc2)CCC2(CC1)CCN(C(=O)CC1CC1)CC2 c1(C(=O)NCCOC(C2C(C)(C(F)F)C2)=O)ccc(CN)cc1.c1(O)ccccc1Cl c1(C(N2CCC(NC(C3CC4(C3)CC4(F)F)=O)C(F)C2)=O)cc[nH]c2nccc1-2 C1(NC(C(C)CC(F)F)=O)(CNC(c2ccc(F)cc2N)=O)CC2CCC1CC2 C(=O)(C1=CC(O)CCC1)N1CCC(C(=O)NCCNC(=O)OC(C)(C)C)C1 C(=O)(C(CC=CC)NC(c1c[nH]c(=NC)o1)=O)N(CCOCC=C)C N1(C(c2c(CNC(c3c(OC)nn(C)c3)=O)occ2)=O)CC(O)C(N=[N+]=[N-])C1 C1(CNC(Cc2ccc(CC)cc2)=O)COCCN(C(c2cnc(C)nc2)=O)C1 c1(CC)nc(CCNC(=O)CCOCCN(C)C(c2ccccn2)=O)n[nH]1 C1(CC)CCCCC1C(=O)NC(C)(CNC(=O)CCOCC(C)C)CC CCCC(C(=O)NCC(=O)N(CC(=O)NC(C)C)C1CC1)NC(N)=O N1(C(=O)C2=CCCC2)CCC2OCCN(C(C3CC4CCC(C3)S4)=O)C2C1 Cc1cc(C(=O)NC(C)CN(C(=O)Cn2nccn2)C)n(C(F)F)n1 C1(CC)CC(NC(=O)C(C2CCC2)OC)C1.C1(=O)C=CC(C)N1CC C(=O)(C#CC1CCCCC1)N1CCC(=CCNC(=O)Cc2csc(Cl)c2)CC1 C(C1=NOC2(COC2)C1)C(=O)Nc1cccc(C(=O)NCC(=O)OC)c1 c1(OCC(=C)C)ccccc1C(=O)NC1CC(NC(c2n[nH]cc2Cl)=O)C1 C(C1CN(C(c2sc(O)nc2C)=O)CC1C(N1CCCC1CC1CCC1)=O)=CC C1(NC(CC=CC)=O)CCCCCN(C(=O)C(=Cc2cnc[nH]2)C)C1 c1(C(=O)Nc2scc(C(=O)NCC3CCOC3)n2)ccc(I)c(Cl)c1 C1(C(N(C(C)CO)CC)=O)COC2(CCN(C(c3ccno3)=O)CC2)C1 C12(C(N3C(C=C)CC3)=O)CCC(CN(C(C3(C)CCCC3(F)F)=O)C1)C2 C(c1nnn(C)n1)=CC(=O)N(CCCCN(C(=O)CCCN1CCCC1)C)C Cc1cc(C)c(CNC(C2C=CCN(C(=O)C(=O)C3CCCC3)C2)=O)s1 C1(CNC(C2CCN(C(CC)=O)C2)=O)CC(F)(F)CN1C(=O)CCN1CCCC1 N1(C(C(CCCC)O)=O)CCC2CN(C(=O)C(O)CC)CC2CC1 N1(C(=O)NCc2cc(N3CCOC3=O)ccc2F)CCC2(CCNC2=O)CC1 C(=O)(C(C)(CC)CCC)N1CCC(CCC(=O)NCC2CCN(CCC)C2)C1 C1(C(=O)NC(CCCOC)(C)C)CC(C)CN(C(c2sccc2C)=O)C1 C1(NC(c2ccnc(Cl)c2Cl)c2n(CC)nnn2)CC2CC(OC)C2C1 c1(CCNC(C(C)C2CCCO2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(C(C)C(C)C(=O)OC)NC(=O)NCC(COC)(C)C Nc1ccc(C(=O)NCC2CCN(C(=O)Cc3cccnc3F)C2)nc1 O(NC(=O)C(C)CNC(C1(F)CCOCC1)=O)CCC C12(CNC(CCCNC(C(C(C)C)OC)=O)=O)CCCC(CO1)C2 C1(C(=O)NCC(C)(C)OCCNC(C2(CC)CC2)=O)CCCCN1C C1(OC)CC(NC(=O)OC)CN(C(C23CCCC2(C(=O)O)C3)=O)C1 Cc1cc(C(N2CCCCC2CNC(c2nccnc2C(F)(F)F)=O)=O)ccn1 c1(OC)cc(C)c(C(=O)NC2CC(F)CN(C(=O)C=CCN3CCCC3)C2)cn1 C(C(NC(=O)NCCOCC1CC1)OC1CCC1)OC C1(CN(C)C)CC2CCC(C1)C2.c12ccsc1C(=O)NCC(C)(CO)NC2 C1(CC(=O)NCC2(C#C)CCCC2)C2CCCC2N1C(=O)C1=C(C)OCC1 c1(C(C(N2CC(C(C)NC(=O)CCC3CCCN3C)C2)=O)O)ccc(F)cc1 C1(CC)(CC)C(OC)CC1N(C(=O)CC1(OC)CCOCC1)C N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 CCCCCCC(C(=O)N1CCC2C(NC(c3ccc(OC)s3)=O)CC12)N(C)C c1(CN2C(C(=O)NCCCCO)CC(O)C2)cnc2cc[nH]c2c1 N1(C(c2ccc(C(=O)OC)o2)=O)CCC(C(=O)NCC2(SC)CCOCC2)CC1 C(=O)(C(CNC(=O)Cc1ccccc1C)C(C)C)NCC(C#C)C(C)C N1(C(c2ccn(C3CC3(F)F)n2)C(=O)Nc2c(C)cccc2)CC2CC2C2CC12 c1(C(=O)NCC2(F)CC(NC(c3c(C)ccs3)=O)C2)cnc2nccn2c1 CCCC(C)(O)C(=O)N1CCC(CN(C(=O)CCOCC)C)C1 C1(C(N2CC(F)(CNC(C3CC(C4CCC4)C3)=O)C2)=O)CCCC1C1CC1 CCCCN=C(NCCC1(O)CCCOC1)NC(C)CC C1(C(C(=O)NCCC(C)NC(c2cc(C)nn2C2CC2)=O)C)CCC(C)(C)CC1 C1(C)(C(=O)NCC=CC(N2CC(OC(=O)NC)C2)=O)CCC(=O)NC1 C1(NC(C2(C)C=CCC2)=O)CN(C(=O)CC2OCCO2)CC2(CCOCC2)C1 CCCCS(=O)(=O)c1ccc(C(=O)NC(C)C(C)NC(=O)CCCC(N)=O)cc1 C1(NC(c2onc(C)c2C)=O)COC2C(NC(c3ccnnc3)=O)COC12 Cc1cc(NC(C2CCCS2(=O)=O)=O)ccc1NC(=O)CCN1CCN(C)CC1 N1(C(C(C)C#N)=O)CC2CCCC(C1)N2C(C1CCn2cnnc2C1)=O C1(CCC=C)(C(=O)NC(C2CCOC2)CC)CN(C(=O)C(C)=CC2CC2)C1 C1(NC(C2COCCO2)=O)CN(C(=O)CC2COCCO2)CC12CCCC2 c1(N2CCC(CSC)(NCC(=O)OC(C)(C)C)CC2)cc(C)c(C(=O)O)cn1 Cc1cccc(OCC(=O)NCCCC(C)NC(c2ccn(C(F)F)n2)=O)c1C C(=O)(C1CCCc2scnc21)NC1(C)CN(C(c2cc(C)c(N)cc2Cl)=O)C1 Cc1nn(C)c(Cl)c1C(=O)NC1CC(CO)N(C(C2CC23CC3)=O)C1 c1(CC(N2CCCC(Cn3cc(C4(C)CCCC4)nn3)C2)=O)cc(F)cc(F)c1 C1(OC)CN(C(=O)CCC(C)C)CC1NC(c1ccc(C(F)(F)F)cn1)=O C(CC(C)C)(C(=O)NCC1(NC(C2CCCC(C)(C)C2)=O)CCOCC1)OC N1(C(c2cc[nH]n2)=O)CCCC(NC(C23CSCC2C3)=O)CC1 C1(NC(c2cc(OC)nn2C)=O)C(C)(C)CN(C(=O)CP(C)(C)=O)CC1(C)C S(=O)(=O)(CC(=O)NC1CCC(C(=O)N(C)CC2CC2(F)F)CC1)NC C(CC(=O)NCC1(C)CCCN(C(c2cc(C#N)[nH]c2C)=O)C1)(C(C)C)OCC N1(CC#CCOCC)C(=O)c2ccccc2C1=O.C1(C(F)(F)F)CN1 N1(C(COCCCC)=O)CCCC(C)C1CNC(c1cnc(O)n1C)=O c1(CC(N2CC(CNC(c3ccc(OCCO)cc3)=O)C2)=O)ccc(F)cc1O C(=O)(CCCCCC(C)O)NC(CC(C)C)CNC(c1ccc(C(N)=O)o1)=O C1(C(N2CCC(C)C2CNC(C23CC2C3)=O)=O)C2C3CCC(C3)C12 N1(C(c2nc(CC)sc2)=O)CC(C)OC2(CCN(C(C3CC(C)(O)C3)=O)CC2)C1 c1(CNC(C(CC)=CC)=O)cc(O)nc(CNC(=O)C(F)CC2CC2)n1 CC1CCCCC1CC(=O)NCCCN(C)Cc1csc(Br)c1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCCCCCCNC(=O)Cc1cnoc1 S(=O)(=O)(c1c(C)cccc1Cl)N1CCC(NC(CCC=C(C)C)=O)C1 C1(CNC(CNS(CCCC)(=O)=O)=O)CN(C)CCN1C(c1cccnc1Cl)=O c1(C(=O)NC2(C3CN(C(C4CC(CF)C4)=O)C3)CC2)cc2c(F)cccc2s1 c1(C(N(CC(C)NC(CNC(C(CC)C)=O)=O)C)=O)cccc(OC(C)C)c1F c1(C(=O)NCC2(CF)CC2)csnc1-c1ccccc1 Cc1cc(C(N2CCCC2CN(C(=O)CSc2cnn(C)c2)C)=O)on1 C(=O)(C(C(C)C)N1CCCC1=O)NCC(CNC(C(C)C)=O)F C#CCCCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1ccc(F)c(C)c1 C1(CCOC)(NC(=O)CCCF)CCN(C(c2cnn(CC3CC3)c2)=O)C1 c1(C(=O)NC2(C)CN(C(c3c(C)n[nH]c3)=O)C2)ccc2c(n1)CCC(C)C2 N1(C(C2C(C)CCC2)=O)CCCN(CCNC(c2cccnc2C(F)F)=O)CC1 Cc1cocc1C(=O)NCC.C(C(C)CC1CCCC1)NC(C1CC1)=O Cc1cccc(CC(=O)NCC(C2CC2)NC(c2conc2C)=O)c1Br Cc1cnc(CNC(C2CC(NCc3ccc(CN(C)C)cc3)C2)=O)cc1C c1(N(C)Cc2cc(Cl)cc(Cl)c2)nc(N2Cc3ncsc3C2)nc2c1CSC2 C#CCCCCCC(=O)NCC1CN(C(=O)Cc2cc(F)cc(C#N)c2)C1 Cc1noc(C)c1C(C)C(=O)NC1CN(C(c2conc2C2CCC2)=O)CC1C Nc1cncnc1C(=O)NCCc1n[nH]cc1C(=O)NC1CC(CO)C2CC12 Cc1ccnc(NC(C2CC(F)CN(C(=O)Cc3cc(Br)cc(Br)c3)C2)=O)c1Br CCC(C(=O)N(C)CCn1cc(-c2c[nH]c3nccc-3c2)nn1)C(F)(F)F Cc1cc(F)cc(Cl)c1NCC1CN(C(=O)OC(C)(C)C)C1 C(=O)(C(C)C(=O)OC)NCCN(C(C1CCC(c2ccccc2)O1)=O)CC CC1CN(C(c2cnc(Cl)cn2)=O)CC1CNC(=O)CC1CCC(C)CC1 Cc1ccnc(C)c1CNC(=O)CC1CCCCN1C(=O)CCP(C)(C)=O C(=O)(C(C)(C)C)NCC1CN(C(CN(C)C(c2ccns2)=O)=O)C1 C12(C(=O)NCC3(O)CN(C(C4CC5(C(C(=O)OC)C5)C4)=O)C3)CCCN(CC1)C2 N1(C(CC=C)=O)CCC2(CC1)CC(NC(=O)C(C)C(O)CCCC)C2 c1(OC)cccc(C(C)C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)c1 c1(C(N(CCCNC(C2Cc3nncn3C2)=O)CC)=O)cc2sccc2n1C C(=O)(C(F)(F)Cc1ccccc1)NCC1N(C(C(c2nc(C)sc2)=O)=O)CC1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(=O)CN2CCCC2C)c(Cl)c1 C1(CC(=O)N(C(C)CCNC(C2CCC(F)C2)=O)C)Cc2ccccc2N1 c1(CC(=O)NC23CC(C2)N(C(=O)C(F)CC2CCC2)C3)cccc2c1OCCO2 c1(CC2CCCN(CC(=O)CCC3CCNCC3)C2)cc(F)ccc1F C1(NC(c2ccc(Cl)o2)=O)CN(C(C2CCC2)=O)CCC12CCC2 N1(C2CCCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)COCC(=O)OC)CC1=O C1(CC(=O)N(C2CCCC2)CCCNC(C(COC)C)=O)CCN(C)C1=O c1(C(N(C(CNC(C)=O)C2CC2)C)=O)ccc([N+](=O)[O-])cc1O c1(CC)cc(C(=O)NC(C2CN(C(=O)CCc3cnn[nH]3)CCO2)C)cc(O)n1 c1(C(=O)NCCN(CC)CC)c(Cl)cc(OC)cc1Cl c1(C(=O)NC2CCN(C(c3c(C)nsc3C)=O)C2)cccc(C(N)=O)c1C C1(c2cn(CC3N(C(c4ncn(CCOC)n4)=O)CCC3)nn2)COCCOC1 C1(C(=O)NC2CC(C)(NC(=O)CCCc3nncn3C)C2)(OC)CCSC1 C#CC1(C(=O)NC2CC(F)(CNC(c3nccnc3C)=O)C2)CCOCC1 C12(C(N(CC(C)(C)C)C)=O)CC(CCO1)N(C(c1sccc1Cl)=O)C2 CC(CNC(=O)C=Cc1cn(C)nn1)CC(=O)N1CCCC(CC(N)=O)C1 C1(C(=O)NCC(C)(Cn2cccn2)NC(=O)Cc2nnc(O)s2)CC12CC(O)C2 N1(C(C(CCN(C)C)O)=O)CC(C(N2CC3(CCC(=O)N3)C2)=O)CC12CCC2 C(N=c1[nH]c(=NCC(C)N2CCC2)[nH]c2c1COC2)c1nn(CC)nc1Br.N(C)C C(=O)(C(C)N(OC)C(=O)CC1C2CN(C(=O)CC3CCC=CCC3)CC12)OC C1(CNC(C(C2CCC2)OCC)=O)CCOC1C(=O)NC1(n2ccnn2)CC1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)n[nH]c2CC)=O)cnc(C(F)(F)F)cn1 N1(C(c2cccc(C#C)c2Cl)=O)CCC2CN(C(C3CCCS3(=O)=O)=O)CCC12 c1(OC)ccc(C(C)NC(C2CC(F)(F)C2(C)C)=O)c(F)c1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC12CN(C(=O)CCc1cccc(C)c1)C2 c1(C(=O)NC2CN(C(c3cc(Br)ncc3F)=O)CC2O)cc(F)c(Br)cc1F N1(C(C(C)OCC)=O)CCC(C)(NC(=O)Cc2cnn(Cc3ccccc3)c2)C1 CCCCC(C(=O)NCC1CCCC(=O)N1)NC(=O)Cc1cc(C)nn1C C12(C(=O)Nc3ncccn3)CCC(NC(=O)Cc3ccc(F)cn3)(CC1)CC2 C1(NC(CCc2cn(-c3c(OC)ccnc3)nn2)=O)CCCN(C(C)=O)C1C C(=O)(C1CCCc2nncn21)N1CCCC(CN(C(=O)C2=COCCO2)CC)C1 CC1(CNC(=O)CC2CCNC2=O)CCCN(C(C2CC(C#N)C2)=O)C1 c1(CNC(c2cnc(CC3CC3)n2C)c2n(CCC)nnn2)ccccc1SC C(=O)(C(CC)C(=O)NC1(C)CCN(C(c2ccn(CC(C)C)n2)=O)C1)OCC CCCCC(CC(=O)N1CC(C(=O)N(C)C)C1)NC(=O)CCc1cnccn1 CCC(CC(=O)NCc1cccc(OC)c1)NC(=O)CC(C)(C)OC N1(CCN(CCN(C(C=CC)=O)C)C)CCC(O)C1 C(=O)(C1=CCC2(COC2)OC1)N1CC(O)CCC(NC(=O)C=CC2CCCC2)C1 CC1CCC(C(=O)NCC(N2CCCCCCC2)c2ccccc2)C(C)C1 N1(C(c2cn(CC=C)nc2)=O)CC(CNC(c2cc(CCC)on2)=O)C(C)C1 CC(C(=O)OC(C)(C)C)C(=O)NCCC(C)N(C(=O)CCCn1ccnn1)C CC(C(=O)NC(C1CCCC1)CNC(c1ccc(-n2cnnn2)cn1)=O)C(F)F C1(CNC(C(C(C)C)n2ccc(C)c2)=O)CN(C(c2cc(F)c[nH]2)=O)CC12CC2 c1(C(=O)NC(CC)(C)CNC(c2cc(COC)on2)=O)ccc2c(c1)CCCC2 C1(C(N(CCCCCNC(c2ccc(C#C)cn2)=O)C)=O)CCC2(CCC2)OC1 c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 C1(C(=O)NCC(C2CC(C)(C)C2)O)CCCN(C(C2CC23CCC3)=O)C1 N1(C(C(C)Oc2ccc(Cl)cc2)=O)CCC2(CC2NC(C2CCCO2)=O)C1 Cc1c(C(=O)NCC2CC(C)N(C(=O)CCSC(F)(F)F)C2)cccc1Br C1(F)(NC(C(C)OCCOCC)=O)CCN(C(=O)Cc2cnn(C)c2C(F)F)C1 Cc1cc(C(=O)NCC2CC2NC(=O)CN2CCS(=O)CC2)nc(N(C)C)n1 c1(NC(c2n(C)ncc2CNC(=O)CN2CC(C)(C)C2)=O)cnc2[nH]cnc2c1 CCCCC(C)CCC(=O)NC(C(N1CCC2(CCC(O)C2)C1)=O)C1CCCC1 c1(OC)ccc(CCC(=O)NC2CCOCC2NC(=O)C(C)=CC2CC2)cc1O c1(C(N2CCN(CC)CC2)C(=O)NC)cccc(OC)c1Br.N12CCCC(C1)C2 c1(C(=O)NC(C)CNC(=O)Cc2cnn(C)c2)ccc2nc(O)[nH]c2n1 C1(NC(c2cc(C(C)(C)C)no2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(F)F CC(C)(C)CC(=O)NCC(c1cccc(Cl)c1)NC(=O)CN1CSCCSC1 N1(C(COCC(=O)NC)=O)CCC(C)C(NC(c2cc(Cl)cs2)=O)C1C N1(CC)CC(NC(=O)C(C2(O)CN(C(C3CC=C(C)CC3)=O)C2)F)CC1=O c1(C(=O)NCCC(C)NC(c2csc(SC(C)(C)C)n2)=O)cc(O)c(F)cc1N N1(C(Cc2cccc(OC)c2)=O)CC(NC(=O)C(F)C2CC2)CC12CCC2 C1(C(N2CC3C(CNC(C(C(C)C)NC=O)=O)(C3)C2)=O)CC2(CCCCC2)C1 CCCC(F)C(=O)N1CCSCC1CCNC(c1ncoc1C(C)C)=O Fc1ccc2ncnc(N3CC4(CO)CC4(C(F)(F)F)C3)c2c1 N1(C(=O)OC(C)(C)C)CC2(CCC2)OCC1CNCC1Cc2nccn2C1 CCC(C#N)C(=O)N(C1CN(C(c2snc(Cl)c2Cl)=O)C1)C c1(C(=O)NCc2ncc(OC)nc2)c(C)ccc(C)c1O N1(Cc2c(C(=O)OCC)n[nH]c2)CCC(F)(C(=O)Nc2cccc(Cl)c2O)CC1 N1(C(C2C(=C)C2)=O)CCC(CC)(NC(c2cc(C)cnc2F)=O)CC1 CCC(C)C(C(=O)NC1(C)CC(C(=O)NCC2CCOC2)C1)NC=O Cc1cc(NC(c2nc(C(=O)Nc3ccc(C(F)(F)F)nc3)cs2)=O)ncc1Cl C1(CCC)CCCN(C(C2(C)CCN(C(c3nn(C)cc3Cl)=O)C2)=O)C1 N1(C(COCCOCC)=O)CC2CCC1C2NC(=O)C(C)Sc1nncn1C c1(OC(C(=O)NCCC(c2cccc(OC)c2)C)C)ccc(C#N)cc1 N1(S(c2cc(NC(C)=O)c(F)cc2)(=O)=O)CCc2occc2C1C(=O)O c1(OC)c(N2CCC(=CCNC(=O)CC3CSCCS3)CC2)ncnc1Cl c1(CNC(=O)NCc2c(OC)ccc(C)c2)cc(F)c(Br)c(F)c1 c1(C(=O)NC2(C)CCN(C(C34CC(F)(C3)C4)=O)C2)cccc(Br)c1Cl c1(N2CCC(CNC(CCC(C)OC)=O)C(C)C2)cnc(C#N)c(C#N)n1 C1(C(C)C)(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)CNC(=O)C1 C1(CC)CN(C(=O)C2=CCCCC2)CCC1(C)C.C12(O)CCCN(C1)C2=O C1(NC(C2(COC)CCCC2)=O)CCCC(CNC(=O)Cn2ncnn2)C1 CCCCCC(c1ccccc1)NC1CC(n2cc(CN)nn2)C1 c1(C(N(C)CC2(O)CN(C(C(CC3CCC3)OC)=O)C2)=O)ccc(OCF)cc1 N(C1c2ccccc2OC1C)C(=O)NCC(CC)(CC)C(N)=O c1(C(C)(C)C)ccnc2c(C(=O)Nc3cc(Cl)cc(F)c3O)cnn12 C1(C(CC)O)COCCN1C(=O)C(O)C1CC1 N1(C(C2(SC)CN(C(CCOCC#C)=O)C2)=O)CCCC(C)(C)C1C C1(O)(C(C(=O)NC(c2ccccc2)CCC)NC)CCCCC1 C1(C(=O)NCC(C)CC(C)O)(CNC(c2c(CC)ocn2)=O)CCCCC1 CON(CCC(=O)NCCN1CC(c2cncc(F)c2)C1)C(=O)Cc1ccccc1 C12(C(=O)NC(C(=O)OCC)CC)CC1CN(C(C1CC13CCCC3)=O)C2 C1(NC(Cn2ncc(CC)c2)=O)CN(C(=O)CCC(=O)c2ccccn2)CC1O c1(C(=O)NC(CNC(=O)COc2cccnc2)CO)cn(C(F)F)nc1C(F)F Cc1c(C)c(C)c(C(=O)NCC(C)(O)CN2CCOCC2)c(C)c1C C(C)(CCC(=O)NCC(CC(C)C)NC(=O)C(O)Cc1ccccc1)OCC C1(CNC(c2ccccc2)=O)CCCN1C(c1csc(C(F)F)n1)=O C(=O)(C1=NN(C)C(=O)CC1)N(C(C)C)CCN(C)C(C1COCC1(C)C)=O CC(CC(=O)N1C2CCC1CN(C(c1cnn(C)c1Cl)=O)C2)CC(F)(F)F C1(C(N(CCCNC(CCC=C=C)=O)CCO)=O)CCC2CCCCN12 C1(NC(c2c(C(C)NC(=O)CN3CCNC(=O)C3)noc2)=O)CCC12CCCC2 C#CCC(O)C(=O)N(CC(C)CN(C)C)C.C1C(C)C(=O)N1 CC(C)CC(C(N)=O)NC(C1(F)CCCN(C(c2cn(C(C)C)cn2)=O)C1)=O c1(SCC(=O)NC2CCC(NC(c3ncc(Cl)s3)=O)C2)ccccn1 C(CC(=O)NC1CC(F)CN(C(c2cccc(F)c2F)=O)C1)(C(F)(F)F)OC C1(CC)(NC(=O)CC(C)(C)O)CCN(C(=O)COC2CCOC2)CC1 CC(C)CC(CC(=O)NC1CCCC1O)NC(=O)CC(O)C(C)C CC(O)C(C)C(=O)NCCCC(C)(C)NC(=O)CCNC(c1ccccc1)=O N1(Cc2ccc(C#C)s2)CCC2(CC1)CC2C(=O)Nc1cccc(I)c1 C12(CNCC)CCC(CC1)N2C(C1(c2cn(CC(=O)OC)nn2)CCCCC1)=O c1(C(C)C(=O)NCC(=C2CN(C(=O)C(F)(F)C3CC3)C2)F)ccc(F)cc1F C1(CNC(c2ccc(OC)cc2)=O)CCN(C(=O)C(O)c2cnc[nH]2)CC1(F)F C(=O)(C(F)(F)C(C(C)C)NC(C1CCCCC1CC(F)(F)F)=O)OC C=CC(CC)CC(=O)N1CC(CNC(=O)CC(=O)NCC(F)(F)F)C(C)C1 N1(C(c2c(C)csc2)=O)CCC(C(=O)NCc2cnnn2C)C(C)(C)C1 N1(c2snc(CC)n2)CCC2CCC(C1)N2C(=O)CCc1nc[nH]n1 C1(C(N(CC(N2CCC(C#C)C2)=O)CCOC)=O)CCCCCN1C CC1(C(=O)NC2CC(NC(=O)CCCNC(=O)C3CC3)C2)COc2ccccc2O1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(C2CC(C(C)C)=NO2)=O)C1(C)C C(=O)(CC(C(F)(F)F)NC(c1c[nH]c(=NC)o1)=O)N(CC(C)OC)CC CC1(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(C(=O)OC)c(NC(=O)C(C)NC(=O)Nc2cccc(OC)c2)ncn1C c1(NC(C2CCCCN(C(C(C)OCC#C)=O)C2)=O)c(C)cccc1[N+](=O)[O-] C1(NC(CCC(C)SC)=O)CCOC12CCN(C(c1cc(C(N)=O)[nH]n1)=O)CC2 CCC(O)C(C)C(=O)NC1(CCNC(c2c(C)coc2C2CC2)=O)CCCC1 C1(C(=O)NC(C2(O)CCN(c3snc(CC)n3)CC2)C)Cc2ccccc2O1 N1(C(C2(COC)CC2)=O)CC(NC(c2cnn(C(C)C)c2N)=O)C(SC)C1 c1(C(=O)NCC(CC=C)NC(=O)C(CCO)N(C)C)ccc(F)c(O)c1F c1(CC)cc(C(N2CCCC2CNC(=O)C(C)(C)CNC(C)=O)=O)ccc1OC C1(CC)CN(C(=O)CC2CC(OC)C2)CCC1CNC(c1ncc(F)cc1F)=O c1(C2(C(=O)NC3C(CNC(CN(C(C)=O)C)=O)C3)CCC2)c(F)cccc1F N1(C(CN(C)CC)=O)CCCC(N(C(=O)Cc2ccc(F)c(C)c2)CC)CC1 c1(C(N2CC(CNC(C3C(CCC)C3)=O)OCC2)=O)cc(C)c(O)nn1 c1(C(N(C)CC2OCCN(C(CC(C)O)=O)C2)=O)ccc(F)cc1C1CC1 C(CCCCCC(=O)NC1CC12CCC(NC(C1(C)C=CCCC1)=O)CC2)SC n1(CC(=O)NCC(C)NC(C=CSC)=O)c2ccccc2c(=O)c2ccccc12 N1(C(COCC(=O)OC)=O)CC(NC(C2CC(C)CC(C)(C)C2)=O)C(C2CC2)C1 N1(C(c2nc(OCC)sn2)=O)CCN(C(c2cc3occc3s2)=O)CC1C C1(CSCc2nc(-c3ccccc3)no2)CCN(Cc2n(C)nnn2)CC1 Cc1nc2cccc(C(=O)NCCCNC(C3CCCSC3C)=O)c2[nH]1 C(CCCCS(=O)(=O)CC)N1C(CNC(CCCC(=C)C)=O)CN(C)CC1 C1(CNC(C2CC(CC)(CC)C2)=O)(NC(=O)C(C)C2CCOC2)CCCCC1C c1(C(C(=O)NC(C)COC(C)(C)C)O)ccc(C#N)cc1.CC1C=CC(=O)N1 c1(NC(C2(F)CN(C(C3CC3(F)Cl)=O)C2)=O)ccc2nn[nH]c2c1 C1(C(=O)NCC(=O)NC2CCCCC2)C2CC(O)C(C2)N1C(C1CCCC1)=O C1(C)(CC)CC(NC(C2(CO)CCCC2)=O)CN1C(c1ccc(C)o1)=O c1(C(=O)NCC#CCNC(CNC(C(CC)C)=O)=O)cnc(Cl)n1C C1(CCNC(CCC=C)=O)CN(C(=O)CCCn2ccnc2C)CCS1(=O)=O c12ccc(cc1)CS(=O)(=O)N2.n1(CCCCC)cc(-c2noc(C(F)F)n2)nn1 c1(C(CNC(=O)C(F)=CCCF)NC(c2ccc(CO)s2)=O)ccccc1 C1(NC(Cc2c(C)ccs2)=O)CCN(C(C2(O)CCC2)=O)CCC1CO n1(C(CC)CC)ncc(C(=O)NC2CCN(C(c3cnc(Cl)s3)=O)C2)c1C1CC1 C1(NC(c2[nH]cc(C)c2)=O)CC1C1CCN(C(c2ccncc2Br)=O)CC1 CCC(C)C(=O)C(=O)NC(CCC1CC1)C(=O)N(C)Cc1nc(C)cs1 N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(=O)C(C#N)CC2CC2)CC1 N1(CC(N2CC(C(C(=O)NC34CCC(CC3)C4)OC)C2)=O)C(C)CCC1C c1(C(=O)NCC(CC)(C)NC(c2cc(C3CC3)on2)=O)ccc(OCCF)cn1 C(CCCCC(=O)NC1CC1C(=O)NC1CC1c1cccnc1)NC(C)=O c1(C2N(CC(C3(COC(C)=O)CCCC3)=O)CCOC2)cccc(F)c1F C1(C(N2CCC(O)(CCNC(C3CCCCS3)=O)CC2)=O)CCCCC12CCC2 c1(CNC(C2(C)CCCO2)=O)cccnc1CNC(C1CCCC1(C)C)=O C(=O)(CC1OCc2ccccc21)N1CC=C(CNC(C2CCCC2(F)F)=O)CC1 C1(c2cn(C(COC)COC)nn2)CN(C(C2CCCC2O)=O)CCO1 C(=O)(C(C)CC(=O)N1C(CNC(c2ccc(F)cc2F)=O)CC2CC12)OC c1(C(=O)NC(CC)CNC(=O)C(C)c2ncco2)cc(C)ccc1Br C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(c2coc(C3CC3)n2)=O)C(C)(C)C1 C1(O)(CNC(=O)CC(F)F)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1 Cc1cc(C(=O)N(C)CC2(CNC(c3nc(C4CC4)cs3)=O)CC2)n(C(F)F)n1 C#CC1(C(=O)NCc2cc(C(=O)NCC(C)(O)C(F)F)n(C)n2)CC(=O)C1 C1(NC(c2cc(CCC)nn2C)=O)(CO)CCCN(C(c2ccc(C)nn2)=O)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)CN2CCCCCC2)CC1C N1(C(CCC(C)OCC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 CCC(CC)C(O)CNC(=O)CC1COCCN1C(=O)CCP(C)(C)=O c1(C(=O)NC2(CC=C)CN(C(C3CC3c3ccc(Cl)s3)=O)C2)ccc(F)cc1Cl C1(CNC(C(C)(C)C2CCCCO2)=O)NCCC1C1CC1 C1(CC(=O)N(CC(C)NC(C(C)C(C)(C)C)=O)C)CCCCCC1(F)F c1(OC)cccc(CCC(=O)NCCN(C(=O)CCOCC(C)C)C2CC2)c1F c1(COCC)ccc(NCCCNC(=O)C(F)(F)CN(C)C)cc1Cl c1(C(=O)NC2CN(Cc3nccc(OC)n3)CC2F)cnc2cccc(Cl)c2c1 C1(C(=O)NCCC(C)(C)NC(c2cc(C(=O)OC)[nH]c2)=O)CC2CCCC2C1 c1(C(N2CCN(C)CC2)C(N2CCC(O)(C(=O)OC)C2)=O)cccc([N+](=O)[O-])c1 CC1CCCC(n2nc(CCCCN(C)C)nc2-c2cc(Br)nn2C)C1 c1(CC(=O)N(CC(C)(C)CNC(=O)C(C)=C(C)C)CC)cccc(C#N)c1OC C(=O)(CC(CC)N(C)C(c1ccsc1C#N)=O)N(CCCO)CC#C C=CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C(C)OC(C)=O C(C(CC)(CC)CC)NC(c1ccc(CC)nc1)=O c1(C(=O)NCCOCCNC(C(CC=C)(F)F)=O)c(Cl)ccc(OC)c1F C(=O)(C(C)C(C)(F)F)NC(CC)CNC(=O)Cn1cc(Cl)c(C(F)(F)F)n1 C(c1ccccc1C#N)=CC(N1CCCC(N2CCN(C(CC)=O)CC2C)C1)=O C(=O)(C1CCCc2cncn21)NC1CN(C(C(F)=CCC)=O)C2C1CCC2 c1(N2CC(C)C(N(C)C)C2)cc(N2CCSC(C)C2)nc(C2CC2)n1 C12(CNC(CC3(OC)CC3)=O)CCCC1N(C(=O)CC13CCCC1C3)CC2 N1(C(c2c(C)nsc2)=O)CCCCC1C1(CNC(C2CC2CF)=O)CCOCC1 C1(C(=O)NC(CCC)C(N)=O)(CC)CCCN(C(=O)Cn2nnc(C)n2)C1 c1(OC)cncnc1C(=O)NCC(CC1CC1)C(=O)N1CC2(CC2)C1 N1(C(C2N(C(CC3C(C)OCC3)=O)CCOCC2)=O)CCCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)N(C3CCN(C)CC3)CC(F)(F)F)ccc2n1 C1(OC)CCN(C(C2CSCN2C(c2ncc[nH]2)=O)=O)CC1(C)C c1(NC(C(CSC)(C)NC(=O)CC2CC(F)(F)C2)=O)cc(C)cnc1C C#CCCN=C(NCc1ccc(CN2CCCC2)cc1)NC(c1ccccn1)C C=C(C)CCCC(=O)NC(C1CCCCC1)CNC(c1cncc(O)c1)=O N1(CC)CCC2(C(=O)Nc3occ4c3CCC4)CCCCCC12.C(=O)(C)N1CC1 N1(C(=O)C(c2cccc(Cl)c2)NC2CC(CC)C2)CCCOCC1(C)C C(=O)(C=C1SCC(=O)N1C)NC1CCN(C2CN(C(C3N(C)CCC3)=O)C2)CC1 Cc1cccc(C)c1NC(=O)C(c1ccoc1)NC(=O)CN(C)C(N)=O N1(C(C2CC23CCC3)=O)CCC2(CCCN2C(c2cccc(Cl)c2O)=O)C1 c1(C(N(C2CC(NC(=O)CCc3csc(Br)c3)C2)C)=O)cnccn1 N1(C(C=C(CC)CC)=O)CC2CCCC(CNC(=O)C=CC(C)C)C2C1 CC1(CNC(C2(F)CC=CC2)=O)CC(NC(=O)CCc2ccc(Br)s2)C1 N12CCc3ccc(cc3CC1)N(C(=O)C1CC1)C(=O)CC2=O.C(C)(C)(C)OC C1(C(=O)NCC(COC)OC)CN(C(=O)C(C)(C)OC)CCO1 Fc1c(CNc2ccc(-c3ccc(C(F)(F)F)cc3)s2)ccnc1Br Cc1cnc2n1CC(C(=O)NCC(C1CCC1)NC(=O)C(F)(F)C(F)(F)F)CC2 CC1(C)CC(NC(=O)C=CC2CCOCC2)CN1C(c1cc(CO)ccn1)=O c1(C(N(C)CC2CCCN2c2ccnc(C3CC3)n2)=O)nnc(O)nc1O Cc1nc(C2CC2)ccc1C(=O)N(CCNC(C1CC(=O)N1)=O)C1CC1 Cc1cc(C(=O)NC2CC(F)CN(C(C3CC3C)=O)C2)n2ncnc2n1 c1(C(C(=O)NCc2cccs2)N(C2COCC2(C)C)C)cnc2ccnn2c1 Cc1cc(C)n2nc(C(N3CCCC3C3(O)CN(C(=O)CN(C)C)C3)=O)cc2n1 c1(N(CC(C)(C)OC(C)=O)C(=O)C2CC2)cc(C2CC2C)on1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C)CC1CNC(c1ccnc(C(F)F)c1)=O n1(CCC)ncnc1CNC(=O)N(C1CCN(C)C1)CCOC C#Cc1cc(C(N2CCC(NC(=O)C(=O)Nc3ccc(C)cc3)C2)=O)cc(F)c1 c1(N(C)C)ncc(C(=O)NCCCC(C)NC(c2ccncn2)=O)cc1Cl c1(C(C(=O)N(CC(=O)N(C)C)C)NC(C(C)C)=O)cccc(C(F)(F)F)c1 c1(Cc2n(CC)nnn2)ccc(F)cc1.C(C(=O)N(C1(C)CC1)C)OC N1(C(C2C(=C)C2C(=O)OC)=O)CCOC(C)C1C(N1CC(F)(F)CC1C)=O C1(C(=O)NC(c2csnn2)C)CCC2CCC1N2C(c1ccncc1)=O Cc1csc2c(=NCC3(C)CCN(C(=O)Nc4c(Cl)cccc4Cl)C3)[nH]cnc12 C(C(=O)N(CC(C)N(C(=O)COc1ccc(OC)cc1)C)C)(C(C)(C)C)SC C1(C(N2C(Cn3cc(-c4nc(C)sc4)nn3)CC2)=O)CCC2CC2CC1 C1(N(C(c2cnc(Cl)[nH]2)=O)CC)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)CO)C2)cncc2ncn(C)c12 n1(CC=C)cc(C(=O)NCC2CN(C(C3(C(=O)NC)CCC3)=O)C2)nn1 CS(C)(=O)=NCCNC(=O)N(C(c1ccccc1)C(F)F)CCO N1(Cc2c(OC)nccc2)CC2CCC(NC(c3ccc(O)nc3)=O)CC2C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(n2cc(-c3cccc(C)c3)nn2)CC1 CN(OC1CCCC1)C(=O)C(C1CCCO1)NC(c1cc(O)ccc1F)=O C1(NC(C2C(CC)C2)=O)CN(C(c2ccc3ncnn3c2)=O)CC(C)(C)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 c1(C(CNC(C2(C)CCN(C)C2)=O)NC(C2(C(N)=O)CC2)=O)cc(F)cc(Cl)c1 Cc1cc(O)c(C(=O)NC2CCCC(CNC(=O)Cc3cnc[nH]3)C2)nn1 C1(CNC(CC=CC=C)=O)CCCN(C(C2CCCCS2(=O)=O)=O)CC1 Cc1ccc2nsnc2c1C(=O)NCCCCN(C(=O)CCCC(C)C)C CN1CCCCC1C(=O)NC1CN(C(=O)CCc2cccc(O)c2)CC1O C(=O)(C(C(C)(C)C)NC(N)=O)NCC(C)NC(c1cccc(NS(C)(=O)=O)c1)=O CC(C)C#CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cccnc1)C c1(C(=O)NC(C)CNC(C2CC(O)C2)=O)cc(C(N)=O)[nH]n1 N1(Cc2c(C)c(Br)cnc2)CC2OCCN(OC(C3(c4cccs4)CC3)=O)C2C1 C#CC1(C(=O)NCC(O)CC(=O)NCC(c2ccccn2)C)CCCCC1 C1(CNC(C(C)C(F)F)=O)CN(C(c2cccc(Br)c2Cl)=O)CC12CC2 C(=O)(CC1=CCN(C(=O)C(C)(C)OC(C)C)CC1)N(CC)CC1CCC1 N1(C(CN(C(=O)OC)C)=O)CCC(C(N2CCCC2c2ccon2)=O)C1 CCCCCC(O)C(=O)N(C1CCC(NC(=O)CCCNS(C)(=O)=O)CC1)C N1(C(CSC)=O)CC2CCC(C1)C2CNC(=O)CCCc1ccc(Cl)nc1 N1(C(C(C(C)C)(C)O)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CCC2 C1(CC(N2CC(c3c(C)con3)C2)=O)CC2(CC2)CN1C(=O)C=Cc1cncn1C CC1COC2(CCCC2)CN1C(=O)CCn1cc(CC2CCCNC2)nn1 CCC(C)(CC)C(=O)NC(C)CCNC(c1cccn1Cc1cccs1)=O Cc1cc(=NC(=O)C(=O)N2CC(O)(C(C)NC(=O)CC(C)C3CCCC3)C2)[nH]o1 c1(N(CCCC)C(=O)NCC2CCOC(c3nccn3C)C2)ccc(Br)cc1 CC(C)(CCC(=O)NCC1(O)CCN(C(c2ccc(Cl)nc2N)=O)C1)[N+](=O)[O-] C(=O)(C1CCCc2sc(C)nc21)NC1C2C(NC(C(F)=CC)=O)CC(CC2)C1 c1(OC)ccc(-c2cccc(OC)c2F)c(CN2CCC(O)(CN(C)C)C2)c1 c1(C(N2C3(CN(C(CC(=O)NCC)=O)C3)CC2)=O)ccc(S(C)=O)cc1 CCCCCCCCCN(C1CC2(CNC2)C1)C(=O)COC1CCCC1 c1(C(=O)NC(c2nccs2)Cc2ccccc2)coc2c(F)c(Cl)ccc12 C(CC(C)(C)C)(C(=O)NC1CCOC(CNC(c2c[nH]nc2OC)=O)C1)OC Cc1nc2cncc(C(N3CC=CC3CNC(=O)COCC3CCCC3)=O)c2[nH]1 c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CC2)ccn2ccnc2c1 CC1CN(C(=O)C(C(C)O)NC(c2cc(Cl)cn2C)=O)CC1F N1(CCCCN(C(=O)Cc2ccoc2)CC2CC2)CCCCC1 C1(C)(CNC(CCn2ccc(C)n2)=O)CN(C(c2c[nH]c(C#N)c2)=O)CCO1 C(c1ccc(Cl)nc1)=C(C)C(=O)NC1CCC(CNC(c2ccncc2F)=O)C1 c1(NC(CNC(CC2CCCC(C)(C)O2)=O)=O)ccc2c(c1)OCO2 C12(NC(C3C(C)(C)COC3)=O)CCCC(NC(c3cnccc3Cl)=O)(C1)C2 N1(CC2CCC2)CCOCC1.c12ccc(s1)NC(=O)C1C(C1)NC2=O C=C(C)C(C)(C)C(=O)N(CCC(C(C)C)NC(=O)CCc1ccc[nH]1)C S(=O)(=O)(c1cccnc1)NCCC(=O)NC(c1ccc(F)cc1F)(C(=O)OC)C C(=O)(C1=CC2(CCN(C(c3c(F)cccc3F)=O)C2)C1)N(CC(C)C)C N1(C(C(CC)(C)F)=O)CCC(CNC(=O)CC2(CO)CC2)C(F)(F)CC1 c1(N(CC(Cl)Cl)C)[nH]c(=NCc2ccccc2C2CCC2)nc2scnc12 C1(CCOC)(NC(=O)Cn2ncccc2=O)CCN(C(c2ccnn2C)=O)CC1 CC1(C2CN(C(C3CCCN(C(=O)C(=O)NCC(F)F)CC3)=O)C2)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CCC(CNC(=O)C3=COCC3)C1)S2(=O)=O C1(CNC(C(CC)OCC)=O)C(C2CC2)CCN1C(=O)CC1(COC)CC1 C=C(C)CC(C(=O)NC(C)C(C)C(=O)OC)NC(c1cccc(C)n1)=O C(C(C)(C(=O)NCCCOC(F)(F)F)NC(=O)C(C)N=[N+]=[N-])SC c1(C(N2CC(CC(C)NC(c3c(Cl)ccnc3F)=O)C2)=O)n[nH]c2ccccc12 Cc1cc(C(=O)N(c2ccccc2)CC2COC(=O)O2)nc(C2CC2)n1 N1(C(C(C)(C)c2ccns2)=O)CCC(F)(F)C(CNC(C2CC3CC3C2)=O)C1 CC1CC=C(C(=O)N2CCC(C(=O)NCCC3OCCC3C)C(O)C2)CC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)COCCCF)CC(C)C1 C(=O)(C(C(C)CC(C)(C)C)N1CCC(F)(F)CC1C)NCCC c1(OC)cc2c(c(OC)c1OC)CN(C(CC(C)CO)C(=O)NCC1CCC1)CC2 c1(C(N2CCC(CNC(C34CCC(C3)C4)=O)C23CC3)=O)cc2ncccc2o1 Cc1ccc2c(CC(N3CC(NC(=O)CC4(O)CCOC4)C3)=O)coc2c1 c1(C(=O)NC(C(CO)NC(CC2C(C)=NNC2=O)=O)C)c[nH]c(C)c(Cl)c1=O C1(C(=O)Nc2ncccc2OC)CC(F)CN(C(C2(CC)COC2)=O)C1 c1(C(N2CCCC(F)(CNC(C=CCC)=O)C2)=O)c(OC)ncc(Cl)c1C CN1CCN(C)C2(CCCN(C(C(=O)NC3CC3)C3=CCCCCC3)C2)C1 C1(C)(C(=O)NCCC(CNC(COCCSC)=O)O)CCCCC1 c1(C(N(CCNC(CCSCCC)=O)C)=O)coc2cc(OC)ccc12 N1(CC(=O)NCc2onc(CCC)n2)CCN(C(=O)CCc2cc(Cl)cs2)CC1 C1(CC(=O)NCc2c(C(N(CC(C(=O)OC)C)C)=O)n[nH]c2)CC(C)(C)CO1 N1(C(C(c2ccccc2)C)=O)CC(F)CC1CN(C(=O)C=CSc1nc[nH]n1)C C1(NC(=O)CC2CC(F)(F)C2)CC(NC(c2csc([N+](=O)[O-])c2)=O)C12CCC2 CC1CC2(CCN(C(=O)CC3(O)CCOC3)CC2)CN1C(=O)CCc1nc[nH]n1 c1(CNC(C2C(NC(c3cc(C)sn3)=O)CCO2)=O)ccc(C2CC2)cc1 c1(C(C(=O)Nc2nnn(C)n2)N(CCCC(O)CO)CC)ccc(C(=O)OC)nc1 c1(CC(=O)OC)cn(CCOn2cc(-c3ccc(C)cc3F)nn2)nc1C#N c1(C(=O)NCCC2CCN(C(C3(O)CCSC3)=O)CC2)cc(O)nc(C2CC2)n1 C(=O)(CCC(=O)NCCC1CCCCN1C(=O)C=Cc1cnc(C)s1)NCCC c1(C(N2C3CCN(C(C(CC)(F)F)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(CCCNC(C)=O)=O)CCC2CCN(C(=O)C3CC3)C2C1 c1(C(N2CCN(C(C3CCN(CC#C)CC3)=O)C(C)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCCCCN(C)C)NCC(C(=O)NC(CC#C)C(N)=O)O c1(C(N2CC(NC(c3cc(CC)cc(Cl)c3)=O)C2)=O)c(C)ccc2nsnc12 Cc1cnc2c(C(=O)NC(C)CC3CN(C(C4CCC(C)(C)C4)=O)C3)cccn12 c1(C(=O)NC2CCC(CCNC(c3c(Cl)cn(C)n3)=O)C2)nc2cnccc2s1 C1(CCC)CN(C(=O)CN(CC(=O)NC(C)C)C)CCN1C(=O)C1=CC(C)CC1 N1(C(C(=O)N(C)C)=O)CCN(C(c2sncc2Br)=O)C(CO)C1 C1(CCC)(NC(=O)C(C)CC(C)C)CCCN(C(=O)C=Cc2ccc(SC)s2)C1 c1(C(=O)OC)sc(C(N2CCS(=O)(=O)CC2)=O)c2c1CCCC2 N1(C(C=C(C)C(F)F)=O)CCC2C(CCN2C(=O)C(c2ccc(Cl)cc2)C)C1 C1(CC(NOCC#C)=O)CC(NC(=O)Cc2cccs2)C1(C)C c1(-c2cn(C3CC4(C(=O)NCCCCC)C3C4)nn2)c(F)cncc1F N1(C(Cc2c(C)ccnc2)=O)CCC2(CCCC2NC(C2CCOCC2)=O)C1 C1(C(N(C2CC(F)(F)C2)C)=O)CCN(C(C2(C#N)CCC2)=O)C1 c1(CNC(CC)=O)ccc2c(c1)CCCC2NC(C12CC(C)(C1)OC21CCC1)=O n1(CC)c(C)c(C(=O)NC2CN(C(=O)CC3CC3)C3CC23)c2cc(OC)ccc12 C1(NC(C)=O)CCC12CN(C(c1cc(-c3cccc(F)c3F)on1)=O)C2 Nc1cc(F)c(O)cc1C(=O)NC1CCC(CCNC(=O)CC(=O)NC2CC2)C1 C12(CNC(CN(CCOC)C)=O)CCCC1N(C(=O)COCC(F)F)CCC2 CCC(CC(C)O)NC(C12CC(NC(=O)C(OC)OC)(C1)C2)=O C1(C(=O)NC2C3(CC(NC(C4CN(C(C)C)C4)=O)C3)C2)CC(=O)NC(=O)N1 CCC(CC(=O)N1CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1C(C)C)C(F)F CCCC(CNC(=O)C(C)c1ccco1)NC(c1cnc(C)[nH]1)=O c1(NS(c2c(C(C)=O)c(F)ccc2)(=O)=O)ccc2c(S(N)(=O)=O)cccc2c1 C1(C)(CNC(CCN(C(c2cn(CCC)nc2)=O)C)=O)CCCCC1 c1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)ccnn1-c1ccccc1 N1(C(C(C)NC(CC)=O)=O)CCC(N(CCCC)C(C2(F)CC=CC2)=O)CC1 C1(CNC(c2ncn(CC)n2)=O)CC(O)C(O)CC1C(=O)NCCN1CC=CC1 C1(C(=O)OC)CCCCCCN1C(c1cnccc1OC)=O C1(C(=O)Nc2c(C)cccc2)CCN(C(=O)C2CCNC(=O)C2)O1 C1(C(C)NC(c2c(CC)scc2)=O)CCN(C(=O)CCOC)CC1 C(=O)(C(CC(C)C)n1ccnc1)NC(CC)CNC(=O)C=CC(c1cccnc1)=O C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(c2cc(C)n(C(C)C)n2)=O)C)C1 c1(C(N2CC(CNC(c3ccc(CC)s3)=O)C(C)C2)=O)ccc(OC)cc1C C1(C(N(CCOC)CCF)=O)CN(C(c2cnsc2)=O)CC1F C1(NC(C(C)(C)n2cccn2)=O)CCCC2CN(C(=O)Cc3c[nH]nc3O)CC12 C1(C(=O)NCCCN(C(c2c(OC)nsc2)=O)C)CCC(=O)N(C2CC2)C1 N1(C(C23CC(n4cc(C(CC)(O)CC)nn4)C2C3)=O)CCC(C#N)(C(C)C)CC1 Cc1cc(Cl)c(C(=O)NC2CCN(C(c3ccc(Br)cc3)=O)C2)cn1 C1(NC(CC(C(C)C)O)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CCC1CO c12ccccc1OCC(C)NC(=O)C1CN(CC1CC)C(=O)N2.O(C(F)F)CC C(=O)(C(CNC(C1CC1C(C)(C)C)=O)N(C)C)NC(c1nc[nH]n1)CC C12(C(N(CCCNC(C3CCCN3c3ncccn3)=O)C)=O)CCCN(CC1)C2 N1(C(CCC2CC(C)C2)=O)CCC2CCN(C(=O)C=CC(F)F)CC12 c1(CC(=O)OCC(N2CC(c3ccccc3)(OC)C2)=O)csc2ccccc12 Cc1cc(C(=O)Nc2cc(C(F)(F)F)cc(Br)c2O)c2c(C3CC3)noc2n1 c1nc2ccc(N3CCC(C4CCc5nccn5C4)CC3)nc2s1 C1(NC(CC2OCC(C)(C)C2)=O)CCN(c2nnc(CO)s2)C12CCC2 N1(C(c2ncn(CC)c2)=O)CCC(CNC(C2CCCN2C)=O)C(O)C1 C1(O)(CNC(=O)CN2CCCCC2)CCCN(C(c2cncn2C2CC2)=O)C1 C1(NC(CC2ON=C(C)C2)=O)C2CC3C1C3C2C(=O)NCCN1CCCCC1=O C1(NC(C=COCC)=O)C2CC1CN(C(=O)Cc1cc(C)nn1C1CCC1)C2 C(=O)(CC1=CCN(C)CC1)NCC(C(=O)NC(CC)(C)CN(C)C)C Cc1n[nH]c(C)c1CC(C)C(=O)NCC1(NC(=O)CC23CCC(CC2)C3)CC1 N1(C(C=CC=CCC)=O)CC(C(N2CC(N=[N+]=[N-])C2)=O)CC1(C)C C1(NC(=O)C(F)CC2CN(C(=O)CCC(F)(F)F)C2)CCC=CCCC1 C1(C(=O)NC(C(=O)NCCCC(F)F)Cc2cc[nH]n2)CC2C=CC1O2 CCCC(C)CC(=O)NC(Cc1ccco1)C(=O)N(C)CC CC1CC(NC(c2csc3nccn23)=O)CCN1C(c1ccncc1)=O CC(C)(C(=O)NCCOC1CCN(C(c2c[nH]c(=N)s2)=O)C1)N1CCCC1 c1(C(=O)NCC2C(C(=O)NCC(CC3CC3)OC)CCC2)cncn1C c1(NC(C2CCCC2)=O)cccc(Cl)c1NC1CC(=O)N(c2ccc(Cl)c(F)c2)C1 c1(CNC(N2CCC(CO)C(c3ccccc3)C2)=O)noc2c1CCCCC2 C1(C(=O)NCc2cn(C3CC(NC(C(C=CC)O)=O)C3)nn2)CCC(CO)CC1 CC(C)C(CC(=O)NC1C(O)CC1O)NC(C1CCC1C#N)=O c1(C(N2C(C(C)(C)NC(C(F)=CC)=O)CCC2)=O)cc(F)c(F)cc1O C1(CC)C(C(=O)NCC2CC3CC(C2)C3)CCN1C(=O)C=NOC N1(C(CCCC#C)=O)CC2(CNC(C3CCCS(=O)(=O)C3)=O)CC(F)(C1)C2 C1(CN(C)C(c2ccc(Cl)[nH]2)=O)CCCCN1C(=O)CSc1nncn1C(C)C C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCCc1cc(CC)no1)C(C)C C1(NC(c2c(C)nc[nH]2)=O)COCCN(C(C2CC3CCC2CC3)=O)C1 C1(COC)CN(C(=O)C(C)CC(F)F)CCN1C(C1(c2ccncc2)CCC1)=O C(CNC(=O)CC1(NC(C2CC2CC(C)C)=O)CC1)(C(C)(C)C)OC C(=O)(CCCCCC#N)NC(C(C)O)C(=O)NCc1ccc(Cl)cn1 CCCC(C(=O)NC(C(=O)NCCN(C)CCOC)C(C)OC)OC CCCCC(CC(=O)N1CCOCC(CC)C1)NC(C1(n2cccc2)CC1)=O N1(C(CN(CC)CC)=O)CC2CCCC(NC(c3ccncc3F)=O)C2C1 CCC(N=c1cc(NCC(C)C#N)nc(C(F)(F)F)[nH]1)C1CCCC1 c1(OC)ncc(C(N2CCC(NC(=O)CNC3CC3)C(C)C2)=O)cc1Cl C1(C(=O)NCCC(C)c2cn[nH]c2)(NC(C)=O)CCC1.C1C(=O)N1.C1C(=O)N1 N1(C(CCC2C(C)(C)C2)=O)C(CNC(C2COC(=O)N2)=O)CC2CCCC12 N1(C(CSc2n(C(C)C)cnn2)=O)CC(NC(=O)CCn2cnnn2)CC1C N1(C(C=CC)=O)CCN(C(c2cc(C)c(C#N)cn2)=O)CC12CCC2 C1(C(C)C)C(C(=O)N(C)Cc2cccnc2)CCN1C(=O)C(O)C1CCC1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CC(Nc2ncccn2)C12CCC2 N1(C2CC2)CC2CN(C3COC3)CC2C1.CC(C)C(C=O)NC(c1ccccc1)=O CC(O)C(C)(C)C(=O)N1CCC(N(C(=O)CC2(CS(C)(=O)=O)CC2)C)CC1 c1(C(=O)NCCCN(C(C(C=C)O)=O)C2CC2)nnn(Cc2cc(C)no2)c1C c1(OC)c(C(=O)NCCN(C(C2CCOCC2C)=O)C(C)C)cc(F)cc1F c1(C(N(CCCNC(Cc2nc(C)oc2)=O)C2CC2)=O)snc(O)c1Cl Cc1cc(F)cnc1C(=O)NC(c1cn(CC2(C(C)(F)F)CC2)nn1)C c1(OC)ccc(C)cc1-n1cc(CNC(=O)C(C)SC)nn1 C(C(=O)N1CCC(=CNC(=O)COc2nc(O)nc(O)n2)CC1)(C(C)C)NC(C)=O C(=O)(C1CCC(=O)c2ccccc21)NCC1N(C(C2(C)CSC2)=O)C2CCC1C2 C1(SCC)CCC(C(N2CCC(C)(CNC(C3(F)CC3)=O)C2)=O)CC1 N1(C(C23CN(C(CCN(C)CCO)=O)C(C2)CO3)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NC(C2CN(C(c3cc(C)no3)=O)C2)C)c(O)cc(F)cc1F c1(OC)cc(Cl)ccc1C(=O)NC1C2CCN(C(=O)C(O)Cc3ccccc3)C12 N1(C(C(n2c(C)ccn2)C)=O)CC2(CC2)CC1CNC(c1cc(Cl)cs1)=O Cc1cc(Br)cc(C)c1CC(=O)NCC1CCC(F)(F)CO1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CCNC(c1cnc(O)cc1OC)=O C1(F)(C(N(C2CCN(C)C2)CC)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1 C#CCCC(O)C(=O)NCC1CCC1NC(c1cccc(C(F)(F)F)c1)=O n1(C(c2ccncc2)OC(F)(F)F)nc(C2CCC2)nc1C1CCN1C1CCCC1 c1(CC)cc(C(=O)N(C(C)CNC(C2CC(CF)C2)=O)C)c(Br)s1 c1(NC(CCC2CCCN(C(Cc3c(C)ocn3)=O)C2)=O)ccc(O)c(CO)c1 C1(C(=O)NC(C(=O)Nc2cccc(C)c2)Cn2cccn2)CCCC2(CC2)C1 CCCCC(CNC(c1cc(F)n[nH]1)=O)NC(=O)CCC1CCCCN1C c1(SC)ncc(N)c(C(N2CC3C(N(C)C(c4ccc(F)s4)=O)C3C2)=O)n1 c1(N2CCC(NC(c3cccc(=O)o3)=O)C(F)C2)ncnc2[nH]ccc12 C1(C(=O)NC2CCC(NC(c3n(CC)ccc3)=O)C2)CCCS1(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1C1(NC(c2cnn(C(C)C)c2)=O)CC1 CCCCCCC(=O)NC1CN(C(C2C=CCCC2)=O)CCC1C C(=O)(N=c1c(Br)c[nH]cc1I)C1CCC(NC(c2cccc3[nH]ncc23)=O)C1 N12CCC3(CC1)CC3NC(=O)CC=CC=CC2.C(=O)(CCN1CCCC1)C(C)=O N1(C(c2cncc(OC)n2)=O)CC2CCCC1(CNC(=O)C(C)(O)C(C)C)C2 C1(CN=[N+]=[N-])CCCN(C(c2cc(CNC(=O)Cn3ccnn3)no2)=O)C1 Cc1cnc(Cl)c(C(=O)NCC2(O)CCCN(C(=O)CNC=O)C2)c1 Cc1nc(C2CCC2)oc1C(=O)NC(C1CCCN1C(c1ccc(CO)s1)=O)C C1(OC)CN(C(=O)C2=CCCCO2)C(C)(CNC(=O)Cc2sccc2C)C1 c1(NC2C(C)C2C)ccc(S(=O)(=O)NCC2CC(C)(C)C2)c(Br)c1 C1(C(N2CCC(c3cnn[nH]3)C2)=O)(OC)CCN(C(c2nc[nH]n2)=O)C1 Cc1ccc(C(N2CC3(CNC(=O)Cc4csc(Cl)c4)CC2CO3)=O)nc1F c1(N(C2CCCNC2)C(c2ccc(OC)cc2C)=O)ncnc2ccccc12 Cn1cnc2cc(C(=O)NCCCOCCCNC(c3ccsn3)=O)ccc12 C1(CNC(=O)CCc2nccn2C)CCN(CC2N(C)CC(O)C2)C1(C)C C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2(CC2)CN1C(=O)CCc1nc(O)n[nH]1 C1(OC)CN(C(=O)CN2CCCCC2=O)CC1NC(C1OCCC1(C)C)=O c1(OC)ccc(C(N2CC(NC(CC(N)=O)c3cn(CCO)nn3)C2)=O)cn1 c1(OCC(=O)N(C2CN(C(CCSCC)=O)CC2F)C)ccc(Cl)cc1F C(=O)(C1c2ccccc2C2CC1C2)NC1(CN(C(=O)C(C2CC2)N(C)C)C)CC1 c1(C(=O)NCC2N(C(COC)=O)CCC2C2CC2)ccc2[nH]c(=O)c(=O)[nH]c2c1 c1(C(CC)(C)C)ccc(S(=O)(=O)N2CC(NCc3cncnc3)C(C)C2)cc1 CCCC(CC(=O)NC(c1cnc[nH]1)C)NC(=O)CC1CC1 N1(C(CC)C(=O)NCCNC(=O)CCCCSC)CCC(CO)(CF)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 Nc1ccc(F)c(C(N2CCC3C(NC(c4cnsc4)=O)C3CC2)=O)c1F c1(C(=O)NC(C)(C)CC(=O)N2CCNCC2)cc2c(cc1O)CCCC2 N1(C(c2c(CC)cns2)=O)CC2CC(C1)CN(C(c1conc1C(C)C)=O)C2 C(CCCCC(=O)N(CC(O)CN(C)C(c1cn2ccsc2n1)=O)C)=CCCC Cc1ccc2nc(C)c(CN=c3ccnc(N(CC(=O)NCC4CC4)C)[nH]3)n2c1 CCCS(=O)(=O)CC(=O)NC1(CNC(c2csc(Cl)c2OC)=O)CCCCC1C CCCCCC(F)C(=O)N1CCC(NC(=O)C=CC(=O)N(C)C)C1C1CC1 C(C(C)C(=O)NC(C1(O)CN(C(=O)C=C2CCC2)C1)C)OC c1(C(C)OC(c2c[nH]nc2-c2ccco2)=O)ccc(F)c(OCC2CC2)c1 c1(C(=O)NC)ccc(C=CC(=O)NCCN(C(=O)C(C)(C)O)CC2CC2)cc1 C1(C(=O)NCC2C(NC(CNC(CC(C)(C)C)=O)=O)C2)Cc2c[nH]cc2S1(=O)=O CCCC(C)CC(=O)NOCCOc1cc(OC(F)F)ncn1 C1(C(N(CCN(C(c2nc(C)oc2)=O)C(C)C)C)=O)CCOCC12CCCC2 C1(C2CCN(C(=O)Cc3cccc(F)c3F)C2)(NC(C(C(COC)C)C)=O)CC1 C1(N(C(C)C(N)=O)C(=O)CC2CCCCC2)CCNCC12CC2 CCC(CNC(=O)C(C)NC(c1ccc(CO)s1)=O)C(C)(F)F N1(C(c2nn(CC)nc2C)=O)CCC(C2CCN(C(=O)CC(C)O)C2)C1 C1(OC)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CCOCC2 N1(CC2CC(C)=C(C)CC2)CC2CCC1CN(CCSC[Si](C)(C)C)C2 N1(C(C2(C(=O)OCC)CC2)=O)CCC(O)(CNC(c2cc(Cl)c(C)cn2)=O)CC1 c1(CC)cc(C(N2CCC(C)C2CNC(C2CCOC2)=O)=O)c2c(c1)CCO2 c1(C(CNC(COCC=C)=O)NC(c2cc(CC)[nH]n2)=O)cccc(Cl)c1 N1(C(CC(C)(C)CNC(c2ccncc2Cl)=O)=O)CC2(C)CC1CCO2 c1(C(=O)NCC2CC(NC(C3CCC(=O)NC3)=O)C2)cnc2c(c1)CNC(=O)N2 CC(C)CC(=O)C(=O)N1C2CCC1C(C(N1CCOC(C3CC3)CC1)=O)C2 N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)C(C)c2ccon2)CC(O)C1 Cn1cc(Nc2ccc(O)cn2)nc1C(N1CCC(C)(C(=O)N(C)C)C1)=O CC(O)CC(=O)N(CCn1cc(CCC2CCOC2)nn1)C1CC1 c1(OCC)cnc(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cn1 O=C(C1=CC2CCC=CCCC12)NCC1CC(O)CN1C(=O)C=Cc1nccs1 C(=O)(CCN=c1[nH]ccs1)NC1CN(C(C(c2c(C)n[nH]c2C)C)=O)CC2C1C2 c1(C(N2CC(O)(CNC(C(CSC)C)=O)C2)=O)cc(CO)cc(C(F)(F)F)c1 N1(C(C=CCOC)=O)CCC2CC1CN(C(=O)C1=CCCOC1)C2 c1(C(=O)NC2CCC(C(=O)Nc3scc(C)n3)C2)snc(Cl)c1Cl C1(C)(NC(C2CCC(CNC(c3ncn(CC)n3)=O)O2)=O)CC2(CCC2)C1 C=C(Br)CCC(=O)N1CC(NC(=O)CCN2CCCCC2=O)C(SC)C1 N#CC1(C(=O)NC(c2cccc(Cl)c2)CNC(=O)CSCC(N)=O)CCCO1 c1(OC)nsc(OC)c1C(=O)NC1CCC(NC(=O)C(C)NC(N)=O)CC1 C(=O)(C(C)(C)C(=O)NCC1COCC1NC(=O)C1=CCCCO1)N(C)C C(=O)(C#CC1(C)COC1)NC(C(=O)NCC(C#C)CC)C1(C)CC1 c1(NC(C(C(C)OC)NC(c2ccsc2C)=O)=O)ccc(C)nc1O N1(C(CCNC(CN2C(C)CCC2)=O)=O)CCC2CC12CO C1(CCCNC(c2cnc(C)[nH]2)=O)CCCCN1C(c1nnsc1C)=O c1(C(N2CC(C)C(NC(=O)C(c3cccnc3)C)C2)=O)ccc2nnn(O)c2c1 CC1c2ccccc2CC1C(=O)NC1(CCNC(c2nc(Cl)cs2)=O)CC1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C)C)C(=O)C1)CC2 c1(C(N2C(C)CCC(NC(C(C)SCCCC)=O)C2)=O)ccnc2cc[nH]c12 C1(O)(CC(=O)NCC2CC3CCC2N3C(C2CC2C2CCC2)=O)CCCCCC1 C(N=c1[nH]c(=NC2CCCC(C)C2)[nH]c2cccnc12)c1ccc(C(C)C)cc1 c1(CC(=O)NC(CC=C)CNC(c2ncncc2Br)=O)cc(F)ccc1F CC1COC2(C1)CN(C(=O)CC1C3CCCC3N1C(=O)C(C)S(N)(=O)=O)C2 N1(C(C2CCCOCC2)C(=O)NCCC#N)CCC(C2CC2)CC1 CC1Cc2ccccc2N(C(=O)NCc2ccnn2-c2ccccc2)C1C c1(C(N(CCCNC(COCCC)=O)C(C)C)=O)cnc2ccccc2c1OC C1(CNC(C(C)SC(C)C)=O)CCC2(CN(C(=O)CN3CC(C)(C)C3)C2)O1 c1(NC(CC)=O)cccc(C(=O)NC2CN(C(=O)CCNC(N)=O)C3CC23)c1 C1(C(=O)NCC2(CN(C(CC(C)C)=O)C)CC2)CC(=O)N(c2ccccc2F)C1 Cc1ncccc1C(=O)NC(Cc1cn[nH]c1)C(=O)N1CC(CN(C)C)C1 N1(C(CC2CC(C)(C)OC2)=O)C2CCC1C1CC1(NC(=O)CNC(N)=O)C2 C1(NC(=O)C(O)Cc2cnc[nH]2)CCC(NC(=O)CCCC2CCCCC2)CC1 N1(C(C(c2ccc(C)o2)C)=O)CCC2OCCN(C(c3nc(C)sc3C)=O)C2C1 C1(C(=O)NCC(C(C)O)C)CCC(C)(C)N(C(C2CC2(C)C)=O)C1 Cc1ccc([N+](=O)[O-])cc1C(=O)NC(Cn1cc(CC(C)(C)C)nn1)CC(C)C C1(NC(c2c(C(C)C)cccc2)=O)CCCCN(Cc2nc(=O)n(C)[nH]2)C1 c1(C(N(C)CC2CCCN(C(C(=O)NC)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 CN(C)NC(=O)CCC(=O)NC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(OCC(COCC)=O)ccc(C(F)(F)F)cc1OC(F)F c1(N2C(C3(NC(C(C)NC(C)=O)=O)CC3)CCC2)ncc([N+](=O)[O-])cc1Br C(=O)(CC(C)CC(C)(C)C)NC1CC(NC(C2CC(C)(OC)C2)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(c2nc(Cl)ccc2N)=O)cc(C)c1Cl C(C(CCNC(C1CCCN1C(=O)CCN1CCOCC1)=O)OC)OC C(N=c1[nH]c(=NCc2cnsc2)c2c(F)cccc2[nH]1)C12C(F)(F)C1CCCC2 CS(=O)(=O)c1cccc(OCCCOC(=O)NC2CC2)c1 c1(N2Cc3n(cc(C)n3)CC2)nc(=NCc2cnc[nH]2)[nH]c2c1CCCCC2 CC#CCCC(=O)NC1CC(NC(c2ccccc2C(C)=O)=O)C1 N1(C(C2OCCC(C)C2)=O)CC2(CCCN(C(=O)C(C)(C)CN(C)C)C2)C1 N1(C(c2cc(CNC(CCNC(C)=O)=O)oc2)=O)CCN(CCF)CC1 c1(C(=O)NC(c2ccc(F)cc2)CNC(C(C)c2ccsc2)=O)cc(F)n(C)n1 C(=O)(CCCC(C)(F)F)N(CC(O)CN(C(=O)Cc1n[nH]c(=N)s1)C)C C123CCC(CC1)(C2)n1cc(nn1)C(C1CC1)N(C)C3=O.C(=O)(CC(CC)SC)OC C#CC1(C(=O)NCC(C)(O)CC)CCN(C(=O)Cc2csc(C)c2)C1 c1(-n2ncc(NC(N(c3cc(C)sc3)C3CC3)=O)c2)cc2cn[nH]c2cn1 C1(Cc2cn(CCCNC(C(C)n3cccn3)=O)nn2)CN(C(N)=O)CCO1 c1(SC)cc(C)c(C(=O)NC2CC(CNC(=O)CC3CC3)C2)s1 c1(C(N2CCC(C(=O)NCCCCC#C)(CO)C2)=O)nccc(C)c1N C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1cc(F)ccc1C(F)F)=O)C2 Cc1ccc(C(=O)NC(c2cn(C(C)C)nc2C)=O)nn1.C1(F)(CN)CC(C(=O)O)C1 N1(C(C2CCN(C(c3cnns3)=O)C23CC3)=O)CCc2ccccc2C1 c1(C(N(C2CN(C(=O)C(C)(C)C(F)F)CC2O)C)=O)cc(C(F)(F)F)ncc1F n1(C(C)C)cc(Br)cc1C(=O)N(CC(=O)O)Cc1noc(-c2ccccc2)n1 N1(C(C(c2ccc(C)o2)C)=O)CCN(C)CC1CNC(c1nscc1C)=O C(=O)(CS(=O)(=O)C(C)C)NCc1c(C2CCN(C(C(CC)(C)O)=O)C2)n[nH]c1 N1(C(c2c(C(C)C)nn(C)c2)=O)CCCCC(NC(C2CC(=C3CCC3)C2)=O)C1 N1(C(c2ncc(C#C)cc2C)=O)CCOC2(C1)CN(C(=O)C(CC)SC)C2 N1(C(C=CC(=O)OCC)=O)C2CCC1CC(F)(CNC(=O)C(C1CC1)N(C)C)C2 C1(CNC(C2(OC)CC2)=O)CCN(C(=O)CNS(C)(=O)=O)CC1C C(CN=c1[nH]c(N2CCNC(=O)CC2)nc2c1CSC2)(c1cccc(C)c1)OC C12(C(=O)NCC3CCN(C(C4C(C)(C)C4(F)F)=O)CC3)CC=CCN1CCC2 c1(NC(CC)CNC(c2ccc(C(C)(C)C)cn2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl C(=O)(C(C)(C)C(N)=O)NCC(C(C)C)NC(c1cc(C(C)=O)sc1)=O C(=O)(C(CCC1CC1)NC(=O)C(C1CCOCC1)C)NCc1ccc(CC)s1 C12(C(=O)NCC(C)(O)CNC(=O)CCc3ccc(Cl)nc3)CCCCC1C2(F)F c1(N2CCC(CNC(CCCC(C)(C)C)=O)C(C)(C)C2)[nH]cnc2nc(Cl)cc1-2 c1(C(=O)Nc2cccc(OCCC=C)c2)cccc(Cl)c1-n1cncn1 CC1(C)CC(C(N2CCCC2CC(N)=O)=O)CN1C(=O)CC1CCCCC1 C1(C(CNCC(CN(CCCC)CC)(C)C)O)CCC(C)CC1 C1(CC(=O)NCC(O)CNC(=O)C(O)c2ccco2)CCC(O)C1 n1(CCCS(C)(=O)=O)nc(C(=O)O)c2ccccc2c1=O c1(CC)ncnc(N2CC3(CC3)CC2CNC(=O)CCCc2ccsc2)c1F c1(CCC)[nH]ccc1C(N1CC(CNC(=O)CCc2cnc(C)s2)(COC)C1)=O N1(C(CCCOCC=C)=O)CCC2(CC1)CCN(C(C1C(C)C1(F)F)=O)CC2C C1(NC(=O)C2CC2)CCCC(C(=O)NCCNC(c2cncn2C2CC2)=O)CC1 c1(CC(=O)NC2CC3(NC(=O)CC=C(Cl)Cl)COC2C3)n[nH]c2c1CCCC2 N(C1CCCc2c[nH]nc21)C(C12N(C(C(C)CC(F)(F)F)=O)CC(C1)C2)=O C1(CC#C)(C(=O)NCC2C3CN(C(c4nonc4N)=O)CC23)CCCCC1 c1(C(N(C2CCN(CCO)C2)CCC)=O)ncccc1Br.C1(SC)CCCO1 Cc1cc(Br)cc(C)c1C(=O)OCC(C1C=CC=CC=C1)=O C1(CNC(=O)CC2CCSC2)CN(C(C2(c3ccno3)CC2)=O)CCC1(F)F C1(CC=C)CCCCN1C(C1(Cn2cc(CCCO)nn2)CC1)=O C1(C(=O)NCC(CCC)OC)CCN(Cc2cccn2CC)C1c1ccccc1 c1(C(=O)NCC2C(NC(CCC3N(C)CCC3)=O)CCCC2)ccc(C#N)cn1 c1(C(N2CC(CNC(c3c(OC)ccnc3)=O)C2)=O)cc(O)cc(O)c1 C1(NC(c2c(C)cc(CNC(CS(CC)=O)=O)o2)=O)C2CCCC1CC2 c1(OC)cc(C(N2CCN(C(=O)C(C)(C)C3(C)CC3(F)F)CC2C)=O)nc(C)c1 Cc1cccc([N+](=O)[O-])c1CNC(C1(Cc2cccs2)CCC1)=O N1(C(CCC(C)OC)=O)CCCC2CN(C(c3cncc4sccc34)=O)CC12 c1(C(N(C(C)CN(C)C(C2(C)CC=CCC2)=O)C)=O)ccc2c(O)n[nH]c2c1 N1(C(c2cnc(OC)s2)=O)CCC2C(C1)NC(=O)CCN2C(=O)CSCCOC C(=O)(CCCCC(=O)NCc1ccoc1C(N1CCC(C)(O)CC1)=O)OC CC(C)(C)C(O)C(=O)N1CCCC(CCC(=O)NCC2(C)CCC(O)CC2)C1 c1(C(=O)NC2C(NC(C3CN(C(C)=O)C3)=O)C2)nc(C(C)(C)C)no1 c1(C(=O)NC2CCOC2C(F)(F)F)cn(-c2cccnc2)nn1 c1(NC2CCC(CC)C2)ncc(C)cc1S(=O)(=O)NCc1cnsc1 N1(C(C2CCC(C)N2C(c2cc(I)cnc2Cl)=O)=O)CCNC2(CCC2)C1 c1(C(=O)NC2(C)CN(C(c3cc(CC)ncn3)=O)C2)cn(C)c2ncccc12 C1(C(=O)NCCCCN(C(C(C)N2CCC2)=O)C)CC12CCC1(CC1)CC2 c1(SCC(C(=O)NCCC)N2CCCC2C(C)(C)OCC)ccc(F)cc1 N1(C(N)=O)CCCC(NC(C2(O)CCN(CCCNCC3C4COCC34)C2)=O)C1 c1(CN(C(c2scc(C(=O)OC)n2)C(=O)NC(C)C(=O)OC)C)ccc(Br)cc1 C=CCCC(C)(C)CNC(=O)C(CC(C)C)ONC(c1cc(C)nnc1O)=O C1(C(N(C2CCN(C(C34CCCCC3C4)=O)C2)CC#C)=O)CCCN1C=O CC1CCCC1NC(c1n[nH]cc1CNC(=O)CCOC1CCCC1)=O C1(C(=O)NCC(N(C)C(C23CC=CC(C2)OC3)=O)C2CC2)CC2(C1)CC2(F)F CC1CC(C(=O)NCC2(C(=O)NC3(CF)CC3)CC2)=NO1 Cc1ccc(CCC(=O)NCC2(NC(=O)C(C)n3ccnc3)CC2)cc1C C1(CNC(C2(C)CCC2)=O)CN(C(=O)CCCc2ccccc2)CCC12CCC2 Nc1c(F)ccc(F)c1C(N1CCC2CC2(NC(c2cnc(O)s2)=O)CC1)=O CC(O)CCCCCC(=O)NC12CC1CN(C(c1cnc3cnccc3c1)=O)C2 C12(CNC(CCOCCNC(c3ccn(C)n3)=O)=O)CCC(CC1)CC2 c1(CNC(C2C(NCc3cc(C)oc3C)C2)=O)ccc(Cl)c(Cl)c1 N1(C(=O)Cn2cc(C(F)(F)F)nn2)CCN(C(=O)C2=CCCC2)C(CCO)C1 C=CC(C)(C)C(=O)NC(C)CCNC(=O)CC1CCC(C2CC2)O1 C12(CNC(C3CCCN(C(C(CC)C)=O)C3)=O)CCC(CC1)CN2C(C)=O N1(C(C(CSC)C)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)C1 N1(C(c2ccncc2)C(=O)NC)CCN(CC(C)O)CC1 C(C(COC)CC(=O)NCCC1(C)CCN(C(C2CC(C3CC3)=NO2)=O)C1)OC c1(C(CNCc2c(F)ccc(C)c2Br)C)ccc(S(N)(=O)=O)cc1 C(N=c1[nH]c(Cl)ncc1F)C1C(NC(C2CCC(CN(C)C)O2)=O)CCC1 C=CC(C)CC(=O)NCc1cccc(C(=O)NCC2CC(OCC)C2)n1 C1(NC(c2cc(C3CCCC3)no2)=O)CCN(C(=O)Cc2ccsc2)C1 N1(C(C(F)OC)=O)CCC(NC(=O)C(C2CCCCC2)OC)C(C)(C)C1 N1(C(C(=O)NCCC2CC(C)(C)C2)=O)CCCSCC1C1CCC1 c1(OC)c(C(=O)N(CC(C)NC(c2cocc2C(N)=O)=O)C)cnn1C c1(NC(CN(C(c2cnc(C)n2C)=O)C)C)ccc([N+](=O)[O-])cc1S(C)(=O)=O CC1CC(NC(C2(CCF)CC2)=O)CCN1C(=O)CCN1CCCS1(=O)=O CC1=NNC(=O)C1CC(=O)NCc1cn(CC(=O)NC(C)Cn2cncn2)nn1 c1(C(N(C2CCN(C(C3CC(C)OC3C)=O)C2)CC)=O)cncc(O)c1 C(=O)(C(CC(F)F)NC(=O)CCC(C)(C)F)NCCCN(OC)C C(=O)(CC(C)C(=O)N1CCN(C(=O)C=Cc2scnc2C)CC1C(C)(C)C)OC c1(CC)noc(CC)c1CC(=O)NCC1(COC)CN(C(=O)C(CC)N(C)C)C1 N1(C(C2OCCC(NC(c3ccc(C#C)o3)=O)C2)=O)CCCC(C=C)C1 C=CC1OCCC1C(=O)NCCC1(NC(=O)C(n2nccc2C)C)CCC1 N1(C(C=Cc2ncn(C)c2)=O)CC(C2CC2)(C(=O)NCCc2nncs2)C1 CC1CC(NC(C2C=CCC2)=O)CCN1CC(O)CC1OCCCO1 C#CC1CC2(CC(C(=O)OC(C(=O)N(C(C(OC)OC)C(C)C)C)=O)C2)C1 C1(CCC)CN(C(c2nc(C)nn2C)=O)CCN1C(=O)C1=CCCC1C c1(C(=O)NCC2N(C(CC(CC)O)=O)CCOC2)cccc2c1CCCO2 c1(NC(C)CCS(C)(=O)=O)ncnc2c1cnn2CCC#N C(=O)(CCCC(=O)OC(C)(C)C)N(C1CCN(C(c2cc(F)n[nH]2)=O)CC1)CC C(CCCCCNC(c1cscc1Cl)=O)NC(=O)CC1CC1C1CCCC1 CCC(C(C)C)C(C(=O)NCCOC)N(C(CC(C)C)C(N)=O)C CC1(C(=O)NCC2COCCN2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC(=O)NC1 C1(CC)C(=O)NCCN1CC(c1ccc(C(c2ccccc2)C)cc1)=O C1(C(=O)NC(CC#C)CO)CN(C(C2(Cl)CC2(F)F)=O)CCO1 c1(C(N2CCC(C)SCC2)=O)cc(O)nc2c1CN(C(=O)CCC(F)(F)F)CC2 N1(C(c2n(C)cnc2)=O)CC(CNC(=O)C(O)CC(F)F)CC12CCC2 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1C(C)C(NC(C1(CCO)CC1)=O)C2 C1(C(C(C)(F)F)NC2CCOC2C2CC2)CCCCCC1 Cc1ncc2n1CCN(C(=O)CC1CCN(C(C3CNC(=O)C3)=O)C1)C2 CCCC(CCCNC(c1cc(Cl)n(C)n1)=O)NC(=O)C1=CCOC1 c1(CC)ccc(O)c(C(=O)N(C)CC2CCCC3CC23)c1.C12(CC1)CCNC2=O C1(C)(COC)CC(NC(c2csc(=N)[nH]2)=O)CN1C(c1cn(C)nc1OC)=O N1(C(C=CCC(C)(C)NC(C2CC3CCC(C2)O3)=O)=O)CC(S(N)(=O)=O)C1 Cc1ccc(C(=O)NCCCNC(=O)C(O)C2CCC2)o1 c1(C(N(C2CC(NC(c3c(O)cccc3F)=O)C2)C)=O)ccc([N+](=O)[O-])s1 Cc1cc(NC2(CCNC(c3n[nH]c4c3CCC4)=O)CCC2)n2ncc(C)c2n1 C=CCC(CC=C)ONC(=O)NC(=O)CCC(C)NCC1CC12CCC2 C1(N(C(C(C)=C(CC)C)=O)C)CN(C(c2occc2C(C)C)=O)CC1F N1(C(c2c(C)coc2)=O)CCC(CO)(CNC(=O)C(O)C2CCCC2)C1 c1(C(C(=O)NCC2CCCO2)N(CCC)C)n[nH]c(C2CC2)n1 O=S(=O)(c1ccc(Br)cc1)N1CCC(O)(c2ccc(F)c(F)c2)CC1 c1(N(C(c2cc(F)ccn2)C(=O)NCCCC)C)cc(Br)cc([N+](=O)[O-])c1 N1(C(CC(C)CNC(C2CCS2(=O)=O)=O)=O)CCC2(CC1)CC2C#N C(=O)(CS(=O)(=O)CC(=O)NC1CCCN(C(=O)C(C)CC(C)C)CC1)OC Cc1ncc(N)cc1C(=O)NCC(C)(O)CNC(=O)CC(C)n1cccn1 Cc1nc2ccc(C(N3CCC(C)CC3)C(=O)NC(=O)CC3CC(CF)C3)cc2s1 N1(C(C2CC(C)(C)OC2)=O)CCCC(C2(NC(=O)C#CC3CCCCO3)CC2)C1 C(C)(N=c1[nH]c(=NCC2CCSC2)[nH]c2c1COC2)c1n(CC)ncc1 Cc1cc(C(N2CCC(C)(CNC(C3(Br)CC3)=O)C2)=O)ccc1C(F)(F)F c1(C(N(C(CNC(c2c(SC)csc2)=O)C)C)=O)cnn2ccc(C)cc12 C(=O)(CS(=O)(=O)CCC(F)(F)F)NCCC(C)N(C(CN(C(=O)OC)C)=O)C CCCC(C(=O)N(CCC(=O)NC1(C2CCC2)CC1)OC)N(C)C C1(CCC)C(=O)NCCN1C(=O)C(C)=CCNC(=O)CS(=O)(=O)NC C1(C)(NC(CC(CC)OC)=O)CCC(NC(=O)COCC2(F)CC2)CC1 C1(N(C)C)CCC(C(=O)NCC(CNC(=O)C(c2cccc(Cl)c2)O)CO)CC1 c1(C(=O)NC23C(CN(C(C4N(S(C)(=O)=O)CC4)=O)C2)C3)cc(N)ccc1Cl c1(C(N(C2CCC(NC(=O)C3=CCC3)CC2)CC)=O)ccc2c(c1)NC(=O)C2=O c1(C(=O)NCCSCc2cn(CC3COCCO3)nn2)[nH]nc2ncnc(O)c12 N1(C(c2n(CC)nc(C)c2)=O)CC2CCCCC2(NC(=O)C(C)n2ccnn2)C1 C(C(C)(C(F)(F)F)c1ccccc1)OC.N12CCC(CC1C)NC2=O C1(OC)(NC(C2(NC(C)C(=O)NC3CCCCC3)CCC2)=O)CCOC1 c1(CNC(c2c(CCNC(C3CC(N(C)C)C3)=O)n[nH]c2)=O)ncc[nH]c1=O C1(CC)CCCCC1C(=O)NCC(O)CNC(=O)CSc1cccc(F)c1 CC1(C(=O)Nc2ccc[n+]([O-])c2)CCCN(C(CNC2CCC(C3CC3)C2)=O)C1 C=C(C)CCCC(=O)N1CC2(CC2)CC1C(N1CC(F)CC(F)C1)=O Cc1ncc(CCC(=O)NCC(C)C(=O)NCC2CC(N(C)C)C2)o1 C(=O)(CC(C)(O)C(F)(F)F)NCC1C2CN(C(c3cccc(C)c3N)=O)C1C2 C1(NC(C=CCN(C(C(c2ccccc2)C)=O)C)=O)CC(C)CC(C)(C)C1 C1(C(=O)NC2(C)CN(C(C3=C(C)CCC3)=O)C2)COc2ccccc2O1 C1(C(N2CC(CNC(N3CCC(CC(=O)OCC)C3)=O)C2)=O)(CF)CCOCC1 N1(C(C=NOC)=O)CCN(C(=O)C(C)CO)CCC1C N1(C(CCCCNC(N)=O)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C1(NC(C2(C)CCCOC2)=O)CC(C(N2CCC3(CC2)N=N3)=O)C12CCC2 c1(C(=O)NC2C(NC(=O)Cc3ccccc3)COC2)c(F)ccc(F)c1Br Cc1nn(C)c2nc(C(=O)N(CC(C)NC(=O)C(C)Cc3cnc[nH]3)C)ccc12 N1(C(c2cccc(CNC(C3CCN(CC)C3)=O)n2)=O)CCNC(=O)C1C C(C1=CCCN(C(C2C3CC4C(C3)C24)=O)C1)NC(CCOCCN(C)C)=O C1(NC(C2ON=C(C)C2)=O)C2CC3CN(C(=O)CCP(C)(C)=O)C1C3C2 n1(CCC)nc(C)cc1C(=O)NC1CC(NC(=O)C(C)C(C)O)C(O)C1 c1(C(c2nnnn2CC=CC2CCCO2)NC2CC(=C)C2)ccc(Br)cc1OC c1(N2CCC(N)C2)cc(F)cc(F)c1.N12CC(C3CC13)C2=O.C=CC12CCC1C2 N1(C(c2cc(C)nc(C)n2)=O)CCC2(CC1)CC(C(N1CCOC3CC13)=O)CO2 CC1CN(C(=O)CN2CCCC2C)CC1NC(C1CC1C#N)=O CC1CN(C(c2sccc2CC#N)=O)CCN1C(=O)CCCC(=O)NC1CC1 N1(C(C2CC3(CCCO3)C2)=O)CCN(C(C2CCCC2O)=O)CC(O)C1 c1(C(=O)NC2C3CN(Cc4cc(C)c(Cl)c(C)c4)CC32)oc2ccccc2c1C N1(C(=O)OC(C)(C)C)CC2OCCN(C(C3CN(CC(F)(F)F)C3)=O)C2C1 C1(CC=C)(NC(=O)C(CN(C)C)N(C)C)CCN(C(C2(C(N)=O)CCC2)=O)C1 S(=O)(=O)(CCC(=O)N(CCN(C(=O)Cc1ccn(CC(C)C)n1)CC)CC)NC Cc1n[nH]cc1CC(=O)NC1(C(=O)NCC2(C3CC3)CCCO2)CC1(C)C C(C)(C)(CCC(=O)NC1CN(C(=O)C(F)(F)c2cccnc2)CC12CC2)N(C)C C1(C(N(CC(O)CO)C(C)C)=O)CCC(CNC(C2CC2C(C)C)=O)CC1 C1(NC(=O)CSc2ccccc2)CCN(C(C2(O)CCSC2)=O)CCC1(F)F c1(CCC)ccc(-n2nc(CCCOc3ccccc3)nc2C2CCCO2)cc1 C1(C(=O)NC2CC(CSC)C2)CN(C(c2cocc2C(N)=O)=O)CCO1 c1(C(N2CC(C)C(NC(C3CCC(C)=C(C)C3)=O)C2)=O)cnc(O)c(Cl)c1 CN1CCCC(C(=O)NC(C2CCCCC2)CNC(C2CCCC2O)=O)C1 N1(C(C)=O)CC2CC(NC(=O)Nc3ccc(NS(C)(=O)=O)n(C)c3=O)C(C2)C1 Cn1cc(S(=O)(=O)N2CCCC2)cc1C(N1CCC(O)C1)=O N1(C(C2(CSC)CCC2)=O)CCC2(CCC(NC(=O)CN(CC(=O)NC)C)C2)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1(C(=O)NCCCn2c(C)nnc2)CCOCC1 Cc1[nH]nc2c1CN(C(=O)CC1CN(Cc3cccc(Br)c3CBr)CCO1)CC2 c1(NC(=O)C(=O)N(C(c2ccc(Br)cc2)CC)CCC)ccc(OCC)cc1 C1(CCOC)(NC(c2ccc(CC)nc2)=O)CCN(C(C2(C)CCOC2)=O)CC1 c1(N2CCC(NC(C(CC)=CC)=O)(CF)C2)nc(C(F)(F)F)nc2ccccc12 c1(NCC(CCOC)NC(=O)OC(C)(C)C)c(C)nn2c1CCCC2C Cc1c(O)ccc(CN(C)CC2CCCN(C(c3c(O)cccc3O)=O)C2)c1O CC1CN(C(C2COCCOC2)=O)CC1CNC(=O)CC1CCCS1(=O)=O Cc1ccc(C(=O)NCCC2(C)CCN(C(=O)C(C)C(F)(F)F)C2)n(C)c1=O c1(C(=O)NCC(CC(=O)NCC2CC2)OC)coc2ccccc12 N1(C(C2C(NC(c3c(C)nccc3)=O)CCCCC2)=O)CC(C)c2ncccc21 CC(C)C(C(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)NS(N)(=O)=O N(C(=NCC#Cc1ccccc1)NC(c1ccc(SC)cc1)C)CCC(=O)NC C1(NC(c2cn3c(Cl)cccc3n2)=O)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 CC1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC(C(=O)NCC(c2cn(C)cn2)O)O1 N1(C(Cc2cccc(C)c2F)=O)CC2CCN(C(c3ncccc3Cl)=O)C2C1 N1(C(C(C)OCC(C)C)=O)CC2(CC(NC(C3CCCC34CC4)=O)C2)C1 c1(C(=O)NC2CC(F)(CNC(c3sccc3Cl)=O)C2)cc(Br)ccn1 c1(CNC(=O)Nc2ccc(N3CCOCC3)cn2)cc(C(F)F)cc(Br)c1 N1(C(c2ccc(CCC(=O)O)s2)=O)CC2(C(=O)O)CCC2(C(=O)OC2CC2)C1 c1(NC(C)C)cc(C(N2CCC(CN(C(=O)C(F)(F)C(C)O)C)C2)=O)ccc1F C(CNC(=O)Cn1cc(Cl)cn1)(CCC)NC(C(C)=C(CC)C)=O c1(OC)ccc(CCN(CCS(=O)(=O)N(C)C)C)c(C)c1.C(CCOC)N c1(C(N2CCC(C(C)NC(COCC=C)=O)C2)=O)cccnc1N(C)C N1(C(C=C(CCC)C)=O)CC(NC(C2(c3ccc(Cl)cc3)CC2)=O)CC(C)(C)C1 N1(C(C(N(C)C)C2CC2)=O)CC(NC(=O)COC2(C)CCC2)CC12CCOCC2 CCCC(CC)N=c1[nH]c(=NCC(=O)NC2CCS(=O)(=O)C2)[nH]c2c1COCC2 N1(CC)CCN(CCC(=O)NC2(CNC(c3cccc(COC)c3)=O)CC2)CC1 c1(C(=O)NC(CN(C(C2CC(N3CCCC3)C2)=O)CC)C)ccnc2ncnn12 C#Cc1ccc(C(=O)NC(C)CN(C(=O)CCOc2c(F)cccc2Cl)C)nc1 c1(C(=O)NCCCCCCNC(c2n(C)nnc2)=O)ccc(F)cc1O Cc1cc(=NC(=O)C2CCN(C(=O)C(C)S(C)(=O)=O)CC2C)[nH]n1C c1(CNC(=O)CC2C=CCC2)ccccc1CNC(c1cnccn1)=O C1(C(=O)NCCc2ccn(C)n2)CC2CCC(C1)N2C(c1ccccc1O)=O N1(C(c2cscc2Cl)=O)CCC(F)(F)C(Cn2cc(CCCO)nn2)C1 C1(CNC(CSCC)=O)CC2CC2N1C(=O)C(C)Cc1cnc[nH]1 Cc1nc(C)c(C(=O)NCC2COCC2NC(C2CCCN(C)C2)=O)o1 N1(C(c2cn(CC)nc2C)=O)CCC(NC(c2cc[nH]c2C2CC2)=O)C(CO)C1 C(=O)(C(F)(CNC(=O)C(C)CC(N)=O)C(C)C)NC(c1nc[nH]n1)CC c1(C(N2CCN(C(C(CSC)C)=O)CC2CCO)=O)ccc2ncccc2c1Cl c1(C(=O)NC2C(NC(c3c(C)c(O)ccc3)=O)CC2)nc(C)n2ccccc12 CCC(C(=O)N1CC(N(C(=O)OC(C)(C)C)CC2CC2)C1)C1CCOCC1 c1(C(C(N2C(CNC(c3c(C)snn3)=O)CCCC2)=O)=O)cc(F)c(F)cc1F C1(C(=O)Nc2c(C)noc2C(C)C)CC(C)(C)CCN1C(=O)OC(C)(C)C N(C1CCc2cccc3cccc1c23)C(=O)NCC1CCC(O)C1 c1(NC(c2c(C)c(Cl)ccc2)=O)nc2ccc(O)nc2s1 C1(C(=O)NC2C(NC(c3n(C=C)ncc3)=O)CCCC2)CC2(C1)CC(C(=O)OC)C2 C(CCN=C(NCCc1cnc(C)s1)N1CCOC(C2CCCO2)C1)OCC Cc1nn(C)c(C)c1CCC(=O)NC1(C2CN(C(=O)CC3CC(C)C3)C2)CC1 C1(NC(=O)Cc2ncccn2)CN(C(C2CCCS2)=O)CC12COC2 C1(C)(C(N2CC3C(NC(C(C)C)=O)(C3)C2)=O)CCCCC1(F)F C#Cc1cc(C(=O)NC2CCCC2NC(C2CN(S(=O)(=O)CC)C2)=O)cc(N)c1 Cc1nn(C(F)F)c(C)c1CC(=O)NC1CCN(C(C23COCC2C3)=O)C12CC2 C(=O)(C1CCc2ccccc21)NC1CCCN(C(C2CN(C)C(=O)C2)=O)CCC1 S(=O)(=O)(c1cccc(F)c1)Nc1c(CNC(=O)OC(C)(C)C)nc2n1CCCC2 c1(C(=O)NC2C(CNC(C3C(OC(C)(C)C)C3)=O)CCC2)c(F)cc(Cl)cc1F N1(C(C=CC(C)(C)NC(c2n[nH]cc2Cl)=O)=O)CCCNC(=O)CC1 C(=O)(C1=NOC(C)(C)C1)NCCC1(NC(CC2CCCC(C)C2)=O)CCC1 N1(c2nnc(C(CC)(C)C)o2)CCC(NC(=O)CC(C)C2CC2)C(C)(C)C1 n1(CC)nc(C(N2CCC(CNC(c3ccn(CCF)n3)=O)C2)=O)cc1C N1(C(C(C2CCCC2)OC)=O)CC(NC(c2coc(C)c2)=O)C2(CCC2)C1 c1(C(N2CC3CC2CN3C(C2CC(F)(CO)C2)=O)=O)ccc2ncnn2c1 c1(OC)cc(C(F)(F)F)[nH]c(=NCCCN(C(=O)C(CC2CCCC2)OC)C)n1 C(N=c1cc(Cl)nc[nH]1)C1C(NC(C(c2cccnc2)C)=O)CCC1 C1(C(=O)NC2CC(F)(CNC(C(CCC)C)=O)C2)COc2cccc(OC)c2C1 c1(OC)cccc(C(=O)NC2CN(C(=O)CC3CC(C)=NO3)CC2O)c1C c1(C(N2CCN(C(=O)Cc3cncs3)CC2C2CCC2)=O)cc2ccncc2o1 C1(C(=O)NC2C(NC(CC(CC)c3ccccc3)=O)COC2)CCS(=O)(=O)CC1 N1(c2c(C)c(NCc3ccnc(Cl)c3)ncn2)CC2CCC1CN2CCO Cn1cc(C(N2CC(NC(=O)Cc3ccccc3CO)C2)=O)c(O)nc1=O c1(CC(=O)NCCC(C)(C)NC(C(CO)N(C)C)=O)ccc(Cl)c2cccnc12 S(=O)(=O)(c1cc(C)c(F)c(Br)c1)NCC1(OCC)CCCCCC1 Cc1csc(C(C(F)(F)F)NC(=O)CCC2CC(C(=O)O)C2)n1 c1(C(c2n(C(C)C)nnn2)N)ccc(Cl)cc1NCCC1CCCOC1.OCF C1(N(C(=O)C(Cl)=CCl)C)CCCCN(C(C2(CO)CC2(F)F)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(C(C)NC(c2cnccn2)=O)OCC1 CCCCC(CNC(=O)Cc1c[nH]nc1C)NC(C1CCC(=O)N1C1CC1)=O C(=O)(CC(C)CNC(c1cnc[nH]c1=N)=O)N(CCOC)CC1CC1 C1(F)(C(=O)NCCc2cnc(C)[nH]2)CCN(C(c2sncc2C)=O)CC1 C1(C(N(CCNC(=O)CS(=O)(=O)C(C)C)CC)=O)CC(c2cccc(F)c2)=NO1 c1(CC(=O)NCC(C)NC(c2scc(C(=O)OC)c2)=O)ccc(C(C)(C)C)cc1 N1(C(CCC)=O)CCC(NC(=O)CSc2nc(C)no2)C(c2ccccc2)CC1 C1(C(F)F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccn2)C1 C1(C(=O)NC2CCC(C(N(CCN(C)C)CC)=O)C2)C2(CC2)C12CC2 C(=O)(C(N)CCC(=O)O)N1CCCC(C(=O)NCc2ccccc2)(CN)C1 CC1CCNC(=O)C1NC(c1cc(CNC(c2cc(Cl)ns2)=O)ccn1)=O N1(C(C2=C(C)OCC2)=O)CCCC2(CC(NC(=O)CSc3ccccn3)CO2)C1 c1(C(c2nnnn2C2COC2)Nc2ncn(C)n2)c(Br)ccc2c1OCO2 c1(C(N(CC(C)(C)NC(C(COCC)C)=O)C)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(CCN1C(=O)COc2ccccc21)N1C(C)C(O)CCC1 C1(NC(C(C=CCCC)O)=O)CN(C(c2cc(F)n(C)n2)=O)C2(CCOCC2)C1 CCC(C)CC(=O)C(=O)NC(C(N1CCCCC(C)(F)C1)=O)C1(O)CCC1 C(=O)(CC(CC(C)C)NC(=O)Cc1cccnc1C)NCC(CCC)C C1(C(=O)NC2C(OCC)CCC2)CC12CCN(C(c1cc(CO)n(C)n1)=O)C2 Cc1coc2c(C(=O)N(C)CCN(C)C(c3cnn(C(C)(C)C)c3)=O)cccc12 C#CC1CC2CCC1N(C(=O)CC1CC1CNC(=O)Cc1cc(C)[nH]n1)C2 C1(NC(=O)C=CC=C(Cl)Cl)CC2CC(C1)N(c1cc(C3CCCC3)ncn1)C2 c1(CNC2C(C(C)C(=O)NCC(c3ccsc3)O)CCC2)ccc(F)c(Cl)c1 C(=O)(CCC1=CCCCC1)N1C(C)(CNC(CCc2n(C)ccc2)=O)CCC1 C(C(C)(C)CCC#N)(c1nnnn1CCCSC)NCCC(=O)N(CC)CC N1(C(CCC(=C)C)=O)CCN(C(c2ccc(Cl)c(OC)c2F)=O)C2COCC12 c1(C(N2CC(NC(C(C(C)(C)O)F)=O)CC23CCC3)=O)cc2c(Cl)cccc2s1 C(=O)(C(F)(CC)C(=O)OC)N1CCC(C)(CNC(c2c(CC)cco2)=O)C1 c1(C(C)=O)cncc(C(=O)NCC2(CNC(c3sc(N(C)C)nc3Cl)=O)CCC2)c1 N1(C(C(C)(CO)OC)=O)CCN(C(C2OCCCO2)=O)C(CF)C1 N1(C(C2C(CCC)C2)=O)CCC(C(F)C(=O)NCCN(C)C2CC2)C1 C1(CCC)CCC(C(=O)NCC=CCNC(=O)C(n2nccc2C)C)CC1 C(=O)(C1=CSCCO1)NCC1N(C(c2cc(C3(C)CC3)on2)=O)CC1 C(N=c1[nH]cnc2ccsc12)C1(F)CCN(C(C2CC23CC3)=O)CC1 c1(CC)oc2ccccc2c1CNCc1ccc(CNC(=O)OC(C)C)cc1 CC1(C(N2CCC(C(F)(F)CO)C2)=O)CC(c2ccccc2)=NO1 Cc1cc(N2CCC(CC(=O)NCc3sccc3C(=O)O)CC2)nc(C)n1 c1(CSC)ccc(C(=O)N(CCC(C)NC(C2(C)CC(C)=NO2)=O)C)cc1 N1(C(C2C3CCCC23)=O)CCCN(C(c2ccoc2C2CC2)=O)C(CO)C1 C1(C(=O)NCc2cc(C)no2)CC(F)CN(C(=O)Cn2ccc(C)n2)C1 N1(C(C(Cn2ccnn2)NC(CC(C)C(F)(F)F)=O)=O)CCOC2(CCCC2)C1 c1(OC)cccc(C(N2CC3CCC(C2)N3C(=O)CP(C)(C)=O)=O)c1[N+](=O)[O-] c1(OC)cccc(C(=O)NCC(C(C)C(C)C)NC(c2c[nH]nc2OC)=O)c1F c1(C(N2CCC(O)(C(C)NC(COCC#C)=O)C2)=O)cc(CC)nnc1C C=C(Cl)CCC(=O)NC1CCOCC1C(=O)NCCCn1ccnc1C c1(CC)ccc(F)cc1C(N1CC(OC)CC1CNC(c1nocc1C)=O)=O CON1CC(C(N2CCN(CC(N3CCOC(CF)C3)=O)CC2)=O)CC1=O c1(SC)ccc(CCC(=O)N(C(C)(C)CO)CC2(C)CC2(Cl)Cl)cc1 C1(C#N)(C(=O)NCCN(C)C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 C(=O)(C1=CC(O)C(NC(=O)C2=NOC(C)C2)C1)NC(c1nc(C)[nH]n1)(C)C c1(NC(c2cnc(-c3ccc(C4CC4)cc3)cn2)=O)cccc2ccccc12 c1(C(=O)NC2C(CNC(c3c(C)coc3)=O)COC2)sc2ccc(C)cc2c1C Cc1ccc(C(C(=O)N2CC(N3CCC(C)CC3)C2)C2CC2)cc1.O C=CC1CN(C(=O)CCC#N)CC1NC(C1CC(CC)=NO1)=O C1(NC(C(C)=C(C)C)=O)CN(C(=O)CCC(F)F)CC1C1CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1CN(C(c2c(OCC=C)cccn2)=O)CCC1 N1(C(CSCC#C)=O)CCC2(CCCN(C(c3c[nH]c(C(=O)OC)c3)=O)C2)C1 C(=O)(CCCCCC(C)O)NC1(C2CN(C(c3c(NC)cncc3)=O)C2)CC1 C(C(N=c1[nH]nc(C2CC2)o1)C1CC1)NC(C(=O)Nc1ccc(C)c(C)c1)=O c1(OC)ncc(CN2CCCC2CCC(=O)NCc2cccnc2)cc1Cl C1(NC(c2c(SC)scc2)=O)C=CCN(C(=O)CCOC(C)CC(C)C)C1 C1(CNC(C2COc3ccccc3O2)=O)CC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 n1(CC(=O)NCC2(COC)CN(C(=O)C=CC3CCOC3)C2)ccccc1=O CCC(C)(C)CC(=O)NC12CCC1CN(C(c1ccc(N(C)C)cn1)=O)C2 C(N=c1ccc(Br)c(S(=O)(=O)N2CCCC(C)(C)C2)[nH]1)C1CCCN(C(C)=O)C1 N1(C(CC2(C(=C)F)CCC2)=O)CC2(CCC2NC(=O)C(Br)=C(C)C)C1 C1(C(N2CC(CNC(c3c(=N)cc[nH]c3)=O)OCC2)=O)CCC12CCOCC2 C=CCC(C)(C)CC(=O)NCC1CCC(CNC(c2cc(F)ccc2F)=O)CC1 N1(C(C(=O)NCC)=O)CC2CC(C(N3CCN(C)C(=O)C3C)=O)C(C2)C1 c1(C(=O)NCCCOc2cccc(C)c2)cc(Cl)c(Cl)c(Cl)c1 C1(OC)CC(C(=O)NC(CNC(C2CN(CC(F)(F)F)C2)=O)CO)CC1OC Cn1nc2ccccc2c1CN=c1ccnc(NCCCN2CCCOCC2)[nH]1 C(=O)(C1=NOC(CN)C1)N(C(CNC(=O)Cc1cccc(F)c1Cl)C1CC1)C N1(C(c2ccc(OC)nn2)=O)CCC2CN(Cc3ccccc3C)CC12 CCC(CC(=O)N(C1CN(C(=O)CC2C(C)(C)C2(C)C)CCC1O)C)C(F)F N1(CCCNC(C(C)c2ccsc2)=O)CCC(NC(=O)CCc2cnccn2)C1 c1(C(=O)NCCCCCNC(C2CC3CCCC3C2)=O)ccc2ncccc2n1 c1(CC)ccc(C(=O)NC(CSC)C(=O)N(C(C)C(C)C)C2CC2)[nH]1 N1(C(C2(C)CC3CCC2O3)=O)CCC2(CC1)CN(C(c1ccc(N)c(Cl)c1)=O)C2 C(=O)(CC(=O)N1CCC(C(F)C(=O)NCCNC(N)=O)C1)OC N1(C(C(C)OCCC)=O)CCCCCCC1C(=O)NCc1csc(C(=O)OC)n1 c1(C(=O)NC(C)CCCCNC(=O)C(O)CN(C)C)cc(Cl)c(Cl)n1C C1(C)(CNC(c2nccc(C)c2)=O)CCN(C(c2coc(Br)n2)=O)CC1 CC1(C)CCCC(CC(N2CC(NC(=O)CNC(N)=O)C(F)C2)=O)O1 c1(CC(N2C(CO)CC(NC(COCCCC)=O)C2)=O)cnc2ncccn12 N1(C(CCc2n[nH]c(=N)s2)=O)CCCC(Oc2ccccn2)C1 N1(Cc2onc(CCCC)n2)CCC2CCC(C1)N2C(=O)CCNC(N)=O N1(C(CN(C(=O)C(CC)C(F)(F)F)CCC)=O)CC(C)CCCC1C Cc1ccc2ncccc2c1C(=O)NC1CN(C(=O)CCC(C)CN(C)C)C1 CN1CCN(C(=O)C(O)C(F)(F)F)CC1CNC(c1scnc1Cl)=O c1(C(C)C)ccc(C(=O)NCC2COC(CNC(c3cn[nH]c3)=O)C2)o1 c1(CC(=O)NCC2CC(OC)CN2C(=O)C2=CCCS2)ccc(F)c(Cl)c1 c1(C(=O)NCC(CC)(C)NC(C2CC3C=CC2C3)=O)n[nH]c2nccc(Cl)c12 Cc1cc2c(C(=O)N(CCCN(C)C(c3ccnc(F)c3N)=O)C)cccc2o1 CCC(C)(CCNC(C1CC2(CC2)CO1)=O)NC(=O)CCC1CCC1 N1(C(c2ccnc(C)n2)=O)CC2CCC1C(CNC(C1CNC(=O)CC1C)=O)C2 c1(SCc2ccc(-c3n(C(CC)(C)C(=O)O)ccn3)cc2)ccc(C)c(N)c1 N1(C(c2ccc(C(C)C)s2)=O)CC2CCC1C(NC(C1(Br)CC1)=O)C2 C1(C(N(CC=C)C)=O)CCCN1NC(=O)CCCN(C)C Cc1c(F)ccc(C(=O)NCC2CC(O)CN2C(c2ccc(Cl)c(N)c2)=O)c1F C1(OC)CN(C(=O)CC(F)(F)CC)C(C)(CNC(c2cc[n+]([O-])cc2)=O)C1 N1(C(CCc2onc(NC)n2)=O)CC(CNC(=O)C(C)O)OC2(CCC2)C1 c1(C(c2nnnn2CCCC2CC2)NCC(C)(C)SC)n[nH]c(C)c1C N1(C(c2c(CCC)cccc2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC1CO c1(CNC(C2(F)CN(C(CC(C)C)=O)C2)=O)cc2ccc(C#N)cc2[nH]1 n1(CC(N2CCN(C(=O)Cn3nnc(=O)[nH]3)C(CO)C2)=O)ccc2ccccc12 c1(C(=O)NCC2N(C(CCCC#C)=O)CC(OC)C2)c(C)ccc2ncccc12 N1(C(c2cnn(C)n2)=O)CCOCC(F)(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(CC(C)NC(CSCC)=O)C1 N1(C(C2C(OCC)C2)=O)CCOC(C)(CNC(c2cnc(C)cc2C)=O)C1 c1(CNC(C(C)CC2CC2)=O)ccccc1CN(C(=O)C(C)OC1COC1)C N1(C(COCCCC#C)=O)CCCC(CNC(=O)C(N2CCCCCC2)C)C1 Cc1nc(C(C)C)oc1C(=O)NC(c1ccccc1)CNC(=O)CC(C)C C(=O)(C(C)(C)Cc1nn[nH]n1)N(C(C1(C)CC1)C)C N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(C2(C(=O)NCCC#N)CCC2)=O)CC1 Cc1cc(C(c2nc(-c3ccn(C)n3)nn2C2CCC2)C)ccc1Br C(=O)(C#CC1(C)CC1)NCCCN(C(=O)C(C1CCC(C(C)(C)C)CC1)O)C CC1C2CCC(C2)C1C(=O)NCC1(O)CC(C(=O)NC2(C3CCCO3)CC2)C1 N1(C(CCC)=O)CCC(NC(c2cc(C)ccc2OC)=O)C(C(C)C)C1 C1(C(N2CC(F)(CNC(C3CC=C(C)CC3)=O)C2)=O)Cc2ccncc2N1 N1(C(=O)CC2C=CCC2)CCC2(CC2)CC1C(N1CC(N2CC(O)C2)C1)=O n1(CC(=O)NC2C3CN(C(c4c(N)cccc4F)=O)CC32)ccc2ccccc12 C(=O)(C(F)(F)C(F)(F)F)N1CCCC(C(=O)Nc2cc(O)ncn2)CC1 N1(C(c2nccc(C)n2)=O)CCN(C(c2nc(Br)cnc2N)=O)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(C)N(C(C2CN(C)C(=O)N2)=O)CC1 c1(CC(=O)NC2CN(C(=O)C=C3CCC3)CC23CCC3)cc(Cl)ccc1[N+](=O)[O-] CC1(C)CC(C)(CNC(C2CCCC2C(F)F)=O)CN1C(C1C(C)(C)C1(C)C)=O N(C1CCCn2nccc21)C(C(CCSC)NC(c1c(OC)cnnc1)=O)=O Cc1cn2c(n1)CCC(C(=O)NC1CCCN(C(c3cc(Cl)c[nH]3)=O)C1C)C2 C1(OC)CC2CCC1(C(=O)NCC(C1CCCCN1C(=O)C1=CCC1)(C)C)C2 c1(C2CCCN(CCCCCBr)C2)nnc2n1CCCC2 c1(CNC(COCC)=O)ccc2c(c1)CCN(C(=O)C(COC)NC(C)=O)C2 C1(C)(C(=O)NC2(CC(=O)OC)CC2)CCCN(C(=O)C(C)C(F)F)C1 C(CC(C(=O)N(C1CCCCCC1)CCNC(=O)CP(C)(C)=O)NC=O)SC n1(C2(C(=O)NC3CCC(NC(c4c(C)[nH]cc4)=O)C3)CC2)cc(C#N)cn1 CC(C)C(O)C(F)(F)C(=O)N1CCC(NC(=O)CC2CCC2)C(O)C1 N1(C(C(CC#C)O)=O)CCC2CN(C(=O)CCc3nc(C)cs3)CCC12 Cn1nccc1C(=O)NC(c1ccccc1)CNC(=O)CC1CCC1(F)F N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(CNC(C2(CC)CCCO2)=O)CC1C C1(CNC(COCC(=O)NC)=O)CN(C(C2CCC2C#N)=O)C2CCN1C2 C(=O)(CCC(=O)NC(C)CNC(=O)CN1CCSCC1)OC O=C(C1=CCCCCC1)NCCC1CCCN(C(C2CC=CCC2)=O)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc3cc(F)ccc3[nH]2)=O)C1 N1(C(C2(SC)CC2)=O)CC(C)(C)C(NC(C2CCC(C)(F)CC2)=O)C(C)(C)C1 C(=O)(C1=NOC2(CCN(C(c3ncccc3F)=O)C2)C1)N1CCC(C(=O)OC)C1 N1(C(C(CC)(C)CNC(c2cscn2)=O)=O)CCCC(O)(C2CC2)C1 c1(SC)c(CCNCC(C)(C)NC(=O)C=Cc2cocn2)cccc1C c1(NC(C)CC2CC2)ncccc1S(=O)(=O)N1CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NCC2C(NC(c3cc(COC)on3)=O)CCCC2)ccc(C)c(C)c1 Nc1c(Cl)ccc(F)c1C(=O)NC1CC(CNC(c2ccn3c2CSCC3)=O)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCCC(NC(C2CC3CC2C3)=O)C1C c1(N2CCCC(CC=CC)CC2)nc(N2CCC3CCC(C2)S3)nc2scnc12 C=CCCC(CO)NC(C1CCN(C(=O)CN(C)CCC)C1)=O CC(C)C(O)C(C)(C)C(=O)N1CCOC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1C2CC(NC(c3cn(C)c(Br)c3)=O)(C2)C1 N1(CC(=O)NCCN2CCOC2=O)CCCCC1C(=O)NCC1CCC1 c1(C(=O)NCCNC(CCOc2ccc(C)cc2)=O)ccc(F)c2cnccc12 c1(C(C(=O)NCCC2CCCN(C(C(C)(C)CO)=O)C2)O)cc(F)cc(F)c1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCCCC1NC(C1CC(F)C1)=O C=CCCC(C(=O)NN(C(=O)C(COC)OCCOCC)C1CC1)NC(C)=O C1(CNC(C(C)c2cc[nH]n2)=O)CN(C(c2cc(C3CC3)ncn2)=O)CC1(F)F C=C1CCN(C(c2n[nH]cc2C)=O)C(C(=O)NC(CO)C2CCC2)C1 c1(OC)ccccc1CC(N1CC(NC(=O)C(C(C)C)NOC(F)(F)F)C1)=O C(=O)(CC1=CCN(C)CC1)N(CCN(C(C)C)C(C1CC(Cl)(Cl)C1)=O)C Cc1ccc(Cl)cc1C(N1CCCCC(NC(=O)Cc2c(C)cnn2C)C1)=O N1(C(CCC(C)O)=O)CCC(C)(CNC(c2ccnn2C2CCC2)=O)CC1 C1(CNC(C(CC2CC2)NC(C(N2CCOCC2)C)=O)=O)CC2(CC2)C(=O)O1 CC1CN(C(=O)CC(C)(C)CNC(C23CCC(CO)(CC2)C3)=O)CCC1N(C)C CCC(C)CCN=C(NCCN1CCOCC1)NCc1ccc(C#N)cc1 C12(C(=O)NCCN(C(C(C)=CC)=O)C3CCCC3)CCC(OC)C1C2 c1(CC)ccc(C(=O)NC2CN(C(=O)CSC(F)F)CC2OC)cc1 N1(c2n(CCC=C)c(C(=O)NC(C)=O)nn2)Cc2c(CO)ccc(F)c2C1.CCO c1(C(C(=O)NC2(C(NOCC(C)C)=O)CC2)C)ccn(C)c1 C123CCCC1N(CC2)C3=O.c1(NC(CNC=O)=O)cccc(Cn2cccn2)c1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CC(C)n2cccn2)cnc2c(c1)NCC2 c1(CC(=O)NC(CCN(C(C2(CC#C)CCCC2)=O)C)C)c(F)cccc1Cl c1(NC(=O)OC2CC(SC)C2)ccc2cc(OC(C)C)ccc2c1 c1(C(=O)NC(C)CCNC(c2ncccc2C2CC2)=O)cnc2[nH]ncc2c1 c1(C(N2CC3C(NC(c4ccc(CC)s4)=O)(C3)C2)=O)ccc(S(N)(=O)=O)o1 C=CCCCC(C)(C)C(=O)NC1CC2(C1)CN(C(=O)C(N1CCCCCC1)C)C2 c1(C(C)C)c(C(=O)NCC(C2CC2)NC(c2cn(C)c(O)n2)=O)cccc1F c1(CN(C)C)cc(C(N2CC(CNC(=O)Cc3nncn3C)C2)=O)no1 c1(C(N2CCN(C(c3ccccc3)C(=O)O)CC2)=O)cc(O)nc(O)n1.CCl CCC(C)C(CNC(=O)CCC(C)(C)NC(c1cnn(C)c1OC)=O)CO C1(C(N2CCN(C(C=C(C)C)=O)C(C3CCC3)C2)=O)CC(C)CC(C)(C)C1 c1(-c2n(CCC)ncc2)ccc(-c2nccn2CCC2NC(=O)NC2=O)nc1C C1(CNC(C2C(CCC)C2)=O)CC(F)CN1C(=O)C(Cc1ccccc1)OC c1(C(=O)NC2CC(F)(CNC(c3c(NCC)scn3)=O)C2)cc(C)nn1C1CC1 C(C(=O)N(C1CN(C)C1)C)(C(C)C)NC(c1cc(C)no1)=O C1(NC(C(C(C)C)SCC)=O)CCCC2CN(C(=O)C=Cc3cccnc3)CC12 c1(NC2CN(C(C=Cc3n(C)cnc3)=O)CC23CCC3)ncc2c(n1)CCOC2 N1(C(COCC=C)=O)CCC(CO)C(NC(=O)CNC(=O)C(CC)CC)C1 C1(CC(=O)NCC(C)N(C(c2cc(CC)n(CCO)n2)=O)C)CCC(C)(C)CC1 c1(-c2cc(C(=O)NC34CC(NC(C(CC)C)=O)(C3)C4)no2)cc(C)ccc1C c1(C(=O)NC(C)C(=O)NC2CCC2C(=O)NCc2ccccc2)coc(O)n1 C(C(C)(CC)NC(c1ccn(C(F)F)c1)=O)NC(CCN(CCCCC)C(C)C)=O c1(OC)coc(C(=O)N(CCCN(C)C(c2cc(C)cnc2Cl)=O)C)cc1=O C#Cc1cccc(NC(=O)CC=CC)c1.C1(=O)CC(=O)N(C)CCCN1 Cc1cc(Cl)ccc1NC(C1CC1n1cnc(C(F)(F)F)n1)=O.C1(=O)C(C)N1CC C1(NC(C(N2CCC(O)CC2)C)=O)CC1C1CCCN(C(C2(C)COC2)=O)C1 CCCC(CCCNC(C1CC12CC(O)C2)=O)NC(=O)CCOC(C)=O C1(N(C(C(=O)NCCSC)C2CC2(Br)Br)CC=C)CCCCC1 c1(C(N2CC(NC(C3CCN(C4CCCCC4)C3)=O)C2)=O)ccnc(C2CC2)n1 Cc1cccc2c(C(=O)NCCC3CN(C(c4cnn5c4CCC5)=O)C3)c[nH]c12 CC1(C)CN(C(C2CC23CC(NC(=O)CCc2nncs2)C3)=O)CCO1 C1(NC(C(c2n(C)ncc2)(F)F)=O)CCC(CNC(=O)C(F)C2CCC2)CC1 c1(CC(N2CCC(C)C2CNC(C2(CCN(C)C)CC2)=O)=O)ccc(O)c(F)c1 c1(C(=O)NCCC2CCN(C)C2=O)cc2cccnc2nc1O C1(NC(Cc2c(C)scc2)=O)CN(C(=O)C(C)OC2CCOC2)C2CCCC12 Cc1cnc(NCCc2cnco2)c(S(=O)(=O)NCC(N2CCCC2)C)c1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC(C)(C)CNC(c1ccccc1)=O c1(C(CNC(C=CC(C)C)=O)NC(c2cn(C(C)(C)C)nn2)=O)cccc(Cl)c1 C(C)(N=c1[nH]c2c(c(=NC(C)CCSC)[nH]1)SCC2)c1c(OC)nccc1 CC1=NOC(C(=O)NCC2CN(C(c3coc(C(F)F)n3)=O)C2)C1C C1(CNC(COCC#C)=O)COCC2(CCN(C(c3cccc(F)c3F)=O)C2)O1 C(=O)(NNC(=O)C(N)=O)N(C)CCn1cc(Br)cn1 N1(C(C(C)=CC)=O)CCCC(NC(=O)C(c2c(C)noc2C)CC)CCC1 c1(NC(=O)NC(Cc2cnc[nH]2)CO)cccc(NC(C2CCC(F)C2)=O)c1 N1(C(CCC(C)OC)=O)CC(F)(F)CC1CNC(C1(C)CCNC(=O)C1)=O c1(C(=O)NCCC2COCCN2C(C23CSCC2C3)=O)nccc2c[nH]nc12 c1(CC)ccc(C(=O)NC2(CF)CCN(C(c3sc(F)cc3Cl)=O)C2)cc1F N1(CC(=O)N(CC(=O)NCC2C=CCN2C)CC)CCCCC1C C1(NC(c2cnccc2Cl)=O)CN(C(C23CCCC2(C(N)=O)C3)=O)CC12CCC2 C1(NC(C(c2cn(C)nc2)(F)F)=O)CCCN(C(c2cscc2F)=O)C1 C1(C(=O)NCCN(C(c2cccc(C)c2C)=O)CC)CCc2ncccc2C1 C(CN=c1cc(C)c(S(=O)(=O)NCC2CCN2C)c[nH]1)=CCCC CCCCC(C(=O)NC1C2CN(Cc3ccc(OC)cc3O)CC12)NC(N)=O n1(CCOC)cccc(C(=O)NC(C)CNC(=O)C(C2CCCC2)OC)c1=O C(CC(O)CC(=O)NCC1CCCN(C(c2scnc2Cl)=O)C1)SC N1(C(CC2CCC(=O)NC2=O)=O)CCCCC(NC(=O)COCCF)CC1 CC1CN(C(=O)CS(=O)(=O)CCO)CCCN1C(=O)C=C1CC1 C1(C2CCN(C(=O)C(O)P(C)(C)=O)C2)(NC(CC2(OC)CCCCC2)=O)CC1 C(=O)(C(C(C)(C)C)NC(C1CC(CC)(CC)C1)=O)N1CCC(C(C#C)C)CC1 c1(CC)c(C(=O)NCC2CCCCN2C(=O)Cc2cnsc2)cnn1C C1(C(=O)NCCCN(C(C2CCC(N(C)C)CC2)=O)CC)CCCN(CC)C1.N(C)C N1(C(C(C=C)C)=O)CCN(C2CN(C(c3conc3COC)=O)C2)CC1 c1(C(=O)NC2C(NC(CCCC)=O)CCCCC2)cc(S(=O)(=O)N(C)C)c[nH]1 CC(C)CC(CNC(C1CC1(C)C(F)F)=O)NC(c1cc(Cl)no1)=O Cc1ccc(C(C)CC(N2CCC(O)(CNC(c3ccc(Cl)o3)=O)C2)=O)cc1 C(C)(CCC(=O)NCCN(C1CCCCC1)C(C1(C#N)CC=CC1)=O)SC c1(C(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc2nccn12 C1(C(=O)NC(C2(O)CN(C(CCC)=O)C2)C)CCc2nnc(O)n2C1 CCC1C(=O)Nc2ccc(C(=O)NC3CC[Si](C)(C)C3)cc21 c1(C(=O)NCC2(C(C)(C)C)CCN(C(CC(CC)OC)=O)C2)c(C)oc(C)c1C c1(C(=O)NC2CC3C(NC(=O)CC4CC5CCC4O5)C3C2)ccc2ccoc2c1 c1(CC)ccc(F)cc1C(=O)NC1CCN(C(c2cnc(N)c(N)c2)=O)CC1O CC(C)CC(C)C(=O)NCC(C)=CC(=O)N(CC(C)(C)O)C n1(CCC)cc(C(=O)NCC(C)NC(c2coc(C(=O)OC)n2)=O)c(C)n1 c1(CCC)ccccc1S(=O)(=O)N1CC23CCCC2(CO)C13 c1(C(=O)NC2C3CCN(C(c4cccc(OC)c4C)=O)C32)nccc2cc[nH]c12 c1(C(=O)NCC(CN(C)C(C2(Br)CC2(C)C)=O)O)ccc2c(c1)COCO2 C(CC(=O)N(CCNC(C1CC(CC(F)(F)F)C1)=O)CCOC1CC1)N(CC)CC c1(C(=O)NCCC23C(CN(C(CC(=O)OC)=O)C2)CC3)cnc2n1C(C)CCC2 c1(C(=O)NC(C(C)NC(c2c(C)nccn2)=O)CO)c(Br)sc(C)c1C C1(C(=O)NCCNC(CC23CC(C)(OC2)C3)=O)CC1C1CC(F)(F)C1 C(=O)(CCCN(C)N=O)NCC1CCN(C(c2cnc(CC(C)C)s2)=O)CC1C CC1CN(C(=O)C(F)(F)C2(O)CCC2)CC(CCNC(C2CCCC2)=O)O1 c1(CC(=O)NS(=O)(=O)CCCn2cnnn2)cc(Cl)nc(Cl)c1 C#CCC(C(=O)N1CCC(N(C(=O)Cc2csnn2)C)C1)C1CC1 N1(C(C2C(C)C2)=O)CCN(C(c2cn(C(C)(C)C)nn2)c2ccccc2)CC1C CP(C)(=O)c1ccc(C(=O)NCC2CC(CNC(=O)C(F)=CC3CC3)CO2)nc1 N1(C(CNC(CN(C)C)=O)=O)CCOC(C(=O)N(CC(C)(O)C2CC2)C)CC1 N1(C(C2CC(OCC)C2)=O)CCCCC(NC(c2sccc2-n2cnnn2)=O)C1 CC1CN(C(C2(Cl)CC2)=O)CCC1NC(=O)C=Cc1cn[nH]c1 C#CCCCCC(=O)NCC1(F)CCN(C(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NC2CC(CC(=O)NC(CCOC)(C)C)C2(C)C)cc[nH]c2nccc1-2 c1(CCC(C)C)cccc(NC(=O)C(=O)N(CC(C)O)C)n1 N1(C(C(COCC)C)=O)CCC(O)C(NC(=O)C(C)(C)CSC)C1 c1(C(N2C(C(=O)NC(c3nc(C)on3)C)CCCC2)=O)coc2ccccc12 c1(NC(C2C3CC2N(Cc2ccc(N4CCOCC4)cc2Br)C3)=O)cnc(O)nc1O C(=O)(C(C)(C(C)C)OC)N(CCCNC(c1cccc(SCC)c1)=O)C c1(OC)cccc(Cl)c1CC(N1CCN(c2cc(F)ncn2)C(CCO)C1)=O C1(NC(CCC)=O)CC2CC1N(C(c1nn(C3CC3)nc1C)=O)C2 C12(NC(=O)C=CCN3CCCCC3)CCCN(C(=O)CCC3CCOC3)CC1C2 c1(C(=O)NCCN(CCC)C(C2CN(C)CC2C)=O)ccnc2ccsc12 N1(C(CC(CCC)O)=O)CC2CCN(C(c3cn(C)c4ncccc34)=O)C(C2)C1 N1(C(c2cc(C)c(F)cc2)C(=O)NCC(C)C)CC=CCC12CCOCC2 n1(CC(=O)NC(C)C(C)NC(=O)CNC=O)cc(CO)nn1 CC(C)C(C)(CNC(C1CC2CCC1C2)=O)NC(=O)Cn1cc(C(F)(F)F)nn1 C1(NC(c2nc(C(N)=O)sc2)=O)(CNC(c2cncc(F)c2)=O)CC2CCC1C2 C=C1COc2c(C(=O)NCC(C3CCCC3)NC(c3sccc3C)=O)cnn2C1 C1(NC(=O)OCC)CCc2nc(NC(=O)C(c3ccc(CC)cc3)N)ncc2C1 CC1CC=C(C(=O)NCC(Cc2ccccc2)NC(C2CCOC(C)C2)=O)CC1 Cc1ccccc1C(C(C)(C)C)NC(c1ccccc1OC1CCNCC1)=O c1(CC)ncc(C(=O)NCC(C2CC2)N(CC(C)(C)CC2CCOCC2)C)[nH]1 C(=O)(C(C)(C)C(=O)NC(CCN(C)C(C1Cc2nccn2C1)=O)C(C)C)OC CCCCC(CNC(=O)Cc1nncn1C)NC(c1cn(CC2CCC2)nn1)=O CCCC(C)(O)CC(=O)NC1CC2(C1)CC(C(N1CCOC(C)(C)C1)=O)C2 N1(C(C(C)OC)=O)CCn2nnc(C(=O)Nc3cncs3)c2C1 C(=O)(C(C)(O)CCC)N1CC(CCC)C(NC(c2c(C)nsc2C)=O)C1 c1(C(=O)NC23CC(CC(=O)NC4C(OC)C(O)C4)(C2)C3)cnn(C)c1C#N C1(C)(CNC(CCCC)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 C1(NC(C(C=C)C)=O)CC2CC(C1)CN(C(=O)CCc1cccc(C)c1)C2 Cc1ccc(C)c(C(=O)N(C2(C(=O)NCC3CSC3)CC2)C)n1 CC1CCN(C(c2nc(C3CC3)cs2)=O)CC1NC(c1ccc(C(C)(C)C)[nH]1)=O c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)cc(Cl)c1O Cc1nn(C)c(=O)c(C(N2CC3(C2)C(NC(=O)C(N)=O)CCS3(=O)=O)=O)c1C C(=O)(C(O)C(C)(C)C)NC(CCNC(c1c(COC)cccn1)=O)C CC(C)CC(C(=O)NC(CNC(c1ccn2ccnc2n1)=O)C(C)(C)C)C(C)C C1(NC(c2c(CC)n(C)nc2)=O)CC2CC(NC(=O)C(F)(F)C(O)C3CC3)C1C2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(C(C)C(=O)NCCC(C)F)C1 CC(C)C(O)CC(=O)NC(C)(C(=O)NCC1(S(C)=O)CC1)C1CCC1 c1(C(N2CCC3(CC2)CN(C(=O)CC2CC2)C3)=O)c[nH]c2cccc([N+](=O)[O-])c12 C12C3CN(CC13)C(=O)C=CC2=O.C1(C(=O)NC2CCCC2)CC=CCO1 C12(NC(c3cc(OCC)cc(F)c3)=O)CCN(C(=O)COC)CCC1C2 C1(NC(COC(CC)C)=O)CC2CCC1(C(=O)NCC(=O)N(C)C)C2 Cc1cnc2n1C(C(=O)N(CC(O)CNC(=O)CSCC(N)=O)C)CCC2 c1(C(N2CCC3(C(C(N4CC(O)(CC)C4)=O)C3)C2)=O)c[nH]c2ncccc12 C(C(CC=C)C(=O)N(CC(=O)NC)C(C)C)NC(CCCOCCC=C)=O c1(N2CCN(C(C3CCC(C)(CC)O3)=O)CC2)ncc([N+](=O)[O-])cc1CO C12(NC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c3cc(O)ccc3F)=O)CC1C2 C(CCN=c1nc(C(=O)N(C)C)cc(SC)[nH]1)N(C(C(C(CC)CC)C)=O)C C1(C(N(CC)CC)=O)CCN2CCOCC12.c1(CCC=O)ccc(C2CCCC2)o1 Nc1ccc(C(N2CCCCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c(F)c1 C(=O)(C(C)(C)CNC(c1ccn(C)c1C)=O)NCCCOC C=CCC(C(=O)N1CCC(CNC2CCN(c3ccccc3)C2)CC1)NC(C)=O C1(C(=O)NC2CC(CCNC(c3cc(CO)c(C)o3)=O)C2)(COC)CCNC1=O C(=O)(C1=NOCC1)NCC(CNC(C1CC(N(C)CC)C1)=O)C c1(C(N(CC(=O)NCCN(CCCC)C)CCC)=O)sccc1Cl C=CCC(CNC(=O)CCCF)C(=O)N(C(C)CSC)C c1(NCC(=O)NC2CC(NC(CC)=O)C2(C)C)ccc(C)c(S(=O)(=O)NCC)c1 C#CCC(CC(=O)NC(c1cnsc1)C)NC(=O)C(C)=C(C)CC N1(C(C2(CC)CCN(C(c3cc(C)cc(O)n3)=O)C2)=O)C2CCC1CC(F)C2 C1(CNC(CN(C2CCC2)C)=O)CC(C)(C)CN1C(C1C=CCCC1)=O C1(NC(C23OC(C)C(C2)C3)=O)COCCN(C(=O)CCS(C)(=O)=O)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(CNC(=O)CC1CCCC1(F)F)CO N1(C(C(=O)NC2C(COC)C2)=O)CCCc2sccc2C1 Cc1cc(Cl)c(C(=O)NCC2C3CN(C(C4(C)CC(C#N)C4)=O)CC23)cc1C C1(NC(c2cc(C)cc(O)n2)=O)CCCCCN(C(=O)CSc2ccncc2)C1 Cc1cc(C(=O)NC2CC(F)CN(C(=O)Cn3cncn3)C2)ccc1S(C)(=O)=O N1(C(CNC(=O)C(N2CCC(c3ccccc3Br)C2)=O)=O)CCCNCC1 C1(NC(c2ccsc2)=O)COC2C(NC(C3CC4CCC3CC4)=O)COC12 c1(C(=O)NC(C)CCN(C(=O)CC2(C(F)(F)F)CC2)C)ccsc1Cl c1(CN(C(CN(C(c2cnccn2)=O)CC)=O)C)cnnn1C CC1(C)CC1(CO)CNC(=O)CCCOC1CNC1 C1(O)(CCNC(c2cc(CF)on2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(C(N2C(Cn3cc(C(C)(C)O)nn3)CC(O)C2)=O)csc2c(F)cccc12 N1(Cc2c(CN3CCC(N)CC3)cccc2)CCC2(C=Cc3ccccc32)CC1 C=C(C)C1CN(C(C2COC3(COC3)C2)=O)CCO1 S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(C(=O)Nc2c(C)ccc(Br)c2)nc1 C(=O)(CC(F)(F)F)N(C1CC(F)(CNC(C(C)OCC=C)=O)C1)CC(F)(F)F C1(C(=O)NC(C2CN(C(CN(C(C)=O)C)=O)C2)CO)CCCCC1 C#CCCCCCC(C(=O)Nc1ccc(Cl)cc1F)N1CCC(C(=O)OC)CC1C N12CC=CC(C1)NC(=O)C2=O.c1(NC(c2cn(CC)nn2)=O)ccc(F)cc1 c1(NC(c2cc(O)ccc2O)=O)c(-c2ccc(OC(F)F)nc2)ccc2c1OCO2 c1(CN(CCC)C(=O)NC2CC(C(=O)OC)C2(C)C)ccc(Cl)cc1Cl C1(C(N2CCC(CNC(CC(C)(C)F)=O)CC2)=O)Cc2nncn2C1 C#CCC(C)(C(=O)NC1CCCC1(C)N(C)C)NC(=O)C(COC)SC C1(CC)CN(C(c2cccc(Br)c2)=O)CCN1C(c1cc(C)cc(Cl)c1)=O C1(C(=O)NC2(C(=O)NC3C=CCCC3)C(C)C2)(CC2CC2)CC(=O)C1 Cc1cc(F)c(C(N2CCC(NCc3cn4ccsc4n3)C(C)C2)=O)c(F)c1 Cc1ccc2sc(C(=O)N(C(C)CNC(c3c(C)cnnc3O)=O)C)c(C)c2c1 c1(CNC(C)C(=O)NCC2CCCO2)cccc(C(=O)OC(C)(C)C)c1 CCC(CC(=O)NCCN1CCCCC1)NC(=O)C(C)NC(C)=O C1(CNC(CCNS(CC)(=O)=O)=O)COCC1NC(=O)Cc1ccsc1C C1(C2CCC2)(CNC(CC(C)C)c2nc(C3CC3)no2)CCC1 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1(C)CCOC1)C2 c1(CC(=O)NCCC2CCN(C(C3(CC)CCC3)=O)C2)cc(F)ncc1Br O=S1(=O)CCCN1c1ccc(-n2cc(C3CCCCC3)nn2)cc1 C1(CC)(NC(c2cn(C)c(=O)cn2)=O)CCN(C(=O)CSc2nccn2C)CC1 C(=O)(CCCCCNC(N)=O)N1C(CNC(C(C(C)OC)O)=O)CC2CC21 CC(CCNC(=O)NCC=C1CCSCC1)C(C)(C)C c1(C(=O)NCC(=O)NCC(C)N(C(=O)CCOCC(F)F)C)ccncc1 CCC(C)CC(C)N(C(c1ccncc1C)C(=O)NCCC#N)C C1(NC(c2c(Cl)cn(CC)n2)=O)CCCCN(C(C2CC(OC)C(OC)C2)=O)C1 C(C(=O)N(CC1CC1)OC)C1CCN(C(c2ccc(CC)s2)=O)CC1 N1(C(CN2CCC(C)C2)=O)CCC(O)CC1C(=O)NCC1(O)CCCCCC1 CCCCC(CC)CC(CNC(=O)NCCOCC1CCOC1)CC O=C1CN(C(=O)C2=C(F)CSC2)c2ccccc2N1.N1CCc2ncccc2C1=O C1(C(N2C(C3(NC(C4C(=O)NCC4)=O)CC3)CCC2)=O)Cc2cccnc2C1 CN1N=C(C(=O)N2CCC(C(=O)NCCn3ncnn3)C2C2CC2)CCC1=O c1(NC(C)=O)cccc(C(C)NC2CCOC(c3ccccn3)C2)c1 c1(N(C)C)ccc(Br)cc1CNC1CCC(CNC(=O)C(C)OC(C)(C)C)C1 N1(C(C2(CC)COC2)=O)CCC(C)(NC(c2cnc(C)nc2)=O)CC1 C1(C(N2CC(CO)C(O)C2)=O)CCC2CCC1N2C(=O)CCn1ccnc1 C=CC1CC(N=c2[nH]c3c(c(=NCc4nc(O)c5c(n4)CCC5)[nH]2)CCC3)CCO1 C1(NC(c2csc(-c3ccccc3)n2)=O)C2CN(C(=O)COCCCF)CC12 c1(CNC(C2(NC(C(COC)N(C)C)=O)CC2C)=O)ccncc1Cl C1(NC2(C=O)CCSC2)(CO)CCCCC1.C1(NC(C)=O)CC1CC(C)C N1(C(C2C(C)C2)=O)CCC(F)C(NC(c2ccc(CCF)cc2)=O)C1 C1(C(=O)NCC(CNC(C(C)(C)F)=O)CO)CCC2(CCC2)CC1 N1(C(C(C2CCOCC2)C)=O)CC(F)(F)CC1CNC(=O)C(C)(C)c1cncnc1 CC1(C)CC(CNC(=O)CCCc2ccsc2)CN1C(c1c[nH]cc(Cl)c1=O)=O c1(C(N2CCC(CC(N3CC4C(C3)C4(F)F)=O)C2)=O)cccc([N+](=O)[O-])c1O CC1COCCN(C(=O)CC2(NC(C3CC(=O)CS3)=O)CCC2)C1 Cc1cc(Cl)c(C(N2CC3CC(NC(c4ccc(F)cn4)=O)C3C2)=O)cc1N C(=O)(C(C)(C)CCS(C)(=O)=O)NC12C(CN(C(CCC=CC(C)C)=O)C1)CCC2 c1(C(N(C)CC2CN(C(C3(F)CCOC3)=O)CCO2)=O)ccc2nn[nH]c2n1 N1(C(c2ccc(C#N)s2)=O)CC(NC(c2cc3ccncc3[nH]2)=O)CCC(O)C1 CCCCC(O)CNC(=O)C(Cc1cc[nH]n1)NC(c1coc(CC)n1)=O CCC(C)(C(=O)N1CC2CCC(C1)N2C(=O)Cc1ccc2sccc2c1)C(F)F N1(c2c(Br)cnc(C(C)C)n2)CC2CC(NC(C3CC=CCC3)=O)CC2C1 C12(C(=O)NCC(C)CN(C(=O)Cc3ccc(C#N)cc3)C)CCC(C)(CO1)C2 c1(C(=O)NCC2C(NC(C3CC(C)(C)OCC3)=O)COC2)cc(F)cc(N)c1F N1(C(c2cc(OC)ncc2)=O)CC2CCC(C1)C(NC(C1CC13CCCC3)=O)C2 C(=O)(C(Cc1ccccc1)C(F)(F)F)NCC(C)N(C(C(C)OC)=O)C c1(C(=O)NCCC2CC(NC(c3nc(COC)oc3)=O)C2)cccc(Br)c1 c1(C(=O)OC)cc(Br)c(C)cc1F.C12CN(C(=O)OC(C)(C)C)CC1NC2=O C(=O)(C1CCc2nnc(C)n21)NC1CC(NC(CC(C(=O)OC)(C)O)=O)C1 Cc1cc(-c2ccnc(CC(=O)NCC34CCN(CC3)C4)c2)ccn1 c1(-c2ccc(C)o2)cc(C(N2CC(OC)C(NC(=O)CS(C)(=O)=O)C2)=O)sc1C C=C(C)CC(C(=O)NC(CNC(=O)C(COC(C)C)NC(C)=O)CC)OC CC(CNC(C1CCC1(F)F)=O)CC(=O)NC(C(=O)OC)C1CC1 Cc1cn2c(n1)C(C(=O)N(C)CC1CCCN(C(c3ccnnc3)=O)C1)CCC2 N1(C(c2c(NC)cccc2)=O)CC2CC1CN2CCc1ccns1 C12(C(=O)NCCCCSC)CCC(CN(C(=O)C(C)(C)C(=O)N(C)C)C1)C2 n1(CC(N2CC3C(CNC(c4cnn(C)n4)=O)(C3)C2)=O)ccc(O)nc1=O c1(C(=O)NCCCn2cc(-c3cc(C)c(F)cc3)nn2)ccc([N+](=O)[O-])cc1 Cc1ccc(Br)c(-n2cc(CONC(c3cc(Cl)cnn3)=O)nn2)c1 N1(C(CCc2scc(C)n2)=O)CCCC(NC(C2CN(C3COC3)C2)=O)C1 C#CC1CN(C(=O)C(C)C(C)O)CCN1C(=O)Cc1cc(F)ccc1Cl C(N=c1[nH]c2c(c(=NCC3(C)CCN(C)CC3)[nH]1)COC2)C1(OC)CCSCC1 C(CN=c1[nH]c2c(c(=NCc3csc(Cl)c3)[nH]1)SCC2)(S(C)=O)OC c1(C(N2CCC(N(C(=O)CCN(C)CC)CC)CC2)=O)cnc2n1CCC(C)C2 N1(C(N(CCc2ccc(C)cc2)C)=O)CCC2CSCC2C1 N(C(=NCC1CCCCO1)NC1CCOC1)C(c1ccc(Cl)o1)c1ccccc1 C(=O)(C1=NOCC1)NCc1cc(C(N(C2CC2)CC)=O)no1 c1(C(=O)NC(C)CN(C)C(c2nccc(Cl)c2F)=O)ccn2c1CS(=O)(=O)CC2 N1(C(C2CCN(C(c3c(C)nn(C)c3C)=O)CC2)=O)CCc2cccc(C)c21 C1(C(N2C3(C(=O)NCCC(C=C)C)CC(C2)C3)=O)CC2CCCC2C1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CSC1)NC(CC)C(C)CN(C)C N1(C(COCCOC)=O)CCN(C)C(C(N2CCCC2CF)=O)C1 C(C(O)C(F)(F)F)N(C)C(=O)NCc1nc(-c2cc(Br)cs2)cs1 C1(C(=O)NCc2cc(COC)on2)CCC(O)CN1C(c1ccccc1F)=O CCC(CC(=O)NCC1CN(C(=O)CC2(C)NC(=O)NC2=O)CC1(F)F)C(C)C c1(CCC)nc(C(=O)NC2COCC2NC(=O)C(C)CN(C)C)co1 C1(C(=O)NC2CC(CNC(C(C)(F)c3ccccc3)=O)C2)Cc2ccccc2S1 C1(C(=O)NCC(C=C)O)CC(=C)CCN1C(=O)C(CC)NC(C)=O CCCC(F)(F)C(=O)N(CC(N1CCC(C)C1C)=O)C CC(=O)CC(C)(C)C(=O)N1CC2C(CNC(=O)CSCC(F)(F)F)C2C1 c1(C(N(CCCCO)C)=O)cccc(CNC(=O)CC2(O)CCOC2)c1 C1(C(=O)NC2CC(CCNC(=O)CCc3cc(C)[nH]n3)C2)(CC)CC(F)(F)C1 O=C(CCS(=O)(=O)c1ccc(Br)cc1)NC1COCC1O c1(C(N(CC(CNC(CCCN(C(C)=O)C)=O)O)C)=O)ccc2oc(S)nc2c1 CCCCCC(CC)C(=O)N1CC(C(=O)Nc2cc(Cl)ccc2F)CC(C)(C)C1 c1(CCC(=O)N(C2CC(NC(c3cncc(O)c3)=O)C2)C)c(F)cccc1Cl Cc1c(CC(=O)NCC(C)CNC(=O)CCc2ccc(O)nc2)cnn1C CCCC(C(=O)NCC1(C(N)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)C1)N(C)C c1(SCC(=O)NC(CNC(C(C)NC(C)=O)=O)C)nccn1C.C(C)(C)(C)NC=O CC(C)CC(=O)C(=O)NC(c1ccc(SC(F)F)cc1)C CCCC(C)(C)CC(=O)N1CC2(C1)CN(C(=O)C(C1CCC1)OC)C2 c1(C(N2C(C(CCC)C)CCC2)=O)cc(Br)c(I)s1 c1(C(=O)NC(CC(C)C)CNC(=O)C=C2CCCCC2)ccc(N)cc1Cl N1(C(C2C(OC)CN(C(c3cc(C)nc(C)c3)=O)C2)=O)CCC(C)(C2CC2)C1 c1(C(=O)NC2CC3CN(C(c4ccc(CC)cc4)=O)CC32)cc2ccccn2c1 CC(C)(C(O)CO)NC(=O)CC1CCN(C(=O)CCNC(N)=O)C1 C1(NC(C2C(NC(c3ccc[n+]([O-])c3)=O)CCO2)=O)CCn2ccnc2C1 Cc1cc(F)cnc1C(N1C2CCC(C2)C1CNC(=O)C(O)Cc1cnc[nH]1)=O c1(C(=O)NC(CC)C(O)C(=O)OC)c2c(nn1C)CCC2 c1(CC(=O)OC)ccc(NNC(=O)C2CCN(C(c3cnc[nH]3)=O)CC2)cc1 c1(CC)ncnc(CC)c1C(=O)NCCCCCCNC(=O)C(C)OCC(C)C c1(C(N2CCC(NC(C3(CC=C)CCOC3)=O)C2)=O)ccc(C)nc1C N1(C(C(COC)(C)O)=O)C2CCC(C2)C1CNC(=O)Cc1ccc(OC)cc1 N1(C(c2n(C(CC)C)ncc2)=O)CCC2(C1)CN(C(=O)C(F)=C(C)C)C2 C1(CNC(CNC(=O)OC)=O)CC2CCC1N2C(=O)C(C1CCOCC1)C Cc1nn(C)c(CNc2cccc(SCc3ccccc3)c2)c1Cl c1(C(=O)NCCC2N(C(Cc3n(C)ccn3)=O)CCC2)c(F)ccc2[nH]ccc12 C1(CC(N2CC(OCCNC(C(C)Cn3ccnc3)=O)C2)=O)COCC1(C)C c1(C(=O)OCC)ocnc1C(=O)NC1CCC(NCC2=CC=C(CC)C2)C1 C1(C(N)=O)CN(C(c2cnnc(C3CC3)c2)=O)CCC1NC(=O)CO C(=O)(C(C)(C)O)NC1CC(CC(=O)N(CCC(N)=O)CC)C1 CC1CC(NC(c2ccc(C(C)(C)C)s2)=O)CN(C(=O)C2=CCCSC2)C1 c1(CC(=O)NCc2cccc(NC(C(C=C)(C)C)=O)c2)ccc2c(c1)CC(=O)N2 C1(C(C)O)CCC(F)C1.C1(OCCOCCO)CN(C=O)C1.C1(=O)CO1 C1(O)(CC)CCCN(C(C(=O)NCCCF)C(C2CCC2)OC)C1 C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CNC(C2CCCC3(CCC3)C2)=O)C1 C1(CNC(COCC(=C)C)=O)CC2CCC1N2C(=O)CC1CCN(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CC2CCC1(CNC(=O)COC)C2 C=CCC(CC(=O)N1CC(N(C)C)C1)NC(=O)CC(=O)OCC(C)C C12(C(=O)NCCOCCN(C(=O)C(C)NC(c3ccccc3)=O)C)COCC1C2 C(=O)(C1=NOC(CNC(c2occc2C(C)C)=O)C1)N1CC(C)(OCC)C1 c1(OC)nscc1C(=O)NC1CC(F)(CNC(C2CC2(C)C(F)(F)F)=O)C1 c1(C(=O)NC(c2ccc(Cl)c(Cl)c2)CC(=O)OC)ccc(C)cc1C N1(C(c2ccc(F)s2)C(=O)NCC(=C)C)CCCC(O)(CC(=O)N(C)C)C1 C(=O)(C(O)CC[S+](C)C)N1CC(CN(C)C(c2cccc3ccoc23)=O)OCC1 N1(C(CCC(N)=O)=O)CC2CCN(C(=O)C3CC3)CC12 c1(C(N2CCC(n3cc(C(C)OCC)nn3)C2)=O)cc2c(C)ccc(Br)c2[nH]1 c1(C(=O)NC2CC(C(C)O)C2)cccc2nn(C)cc12 C1(CNC(C2C(CCC)C2)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1(F)F C1(NC(c2ccn(C(C)(C)C)n2)=O)CN(C(=O)Cn2ccnn2)CC1n1ccnn1 c1(-c2cn(C3CCN(C(=O)CSC4CC5CC5C4)C3)nn2)cccc2ccsc12 c1(C(N2CC(C)(NC(C(c3ccnn3C)C)=O)C2)=O)cnc2ccccn2c1=O N1(C(C(Cc2cn[nH]c2)NC(c2cc(C(C)C)no2)=O)=O)CCc2nn[nH]c2C1 c1(C(=O)Nc2cc(C(=O)OC)sc2)cc(O)nc2[nH]c(=N)ccc12 C1(C(=O)NC2CC(C)(NC(c3ccc(O)c(N)n3)=O)C2)CCC2(CCC2)OC1 N1(C(c2cnn(CCF)c2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCC12 C=CC(CC)CC(=O)N1CCOC(CN(C(=O)C(F)(F)CC2CC2)C)C1 C1(C(=O)NC2C(NC(c3ccc(CN(C)C)[nH]3)=O)CCC2)CN2CCCN1CC2 C(C)(C)(CCN=c1ccnc(S(C)(=O)=O)[nH]1)NC(CC(COC)C)=O C(=O)(CC(C)CNC(=O)C(C)(C)OC)N1C(C)(CCC)CC1 c1(SCC(=O)NCC2CN(C(CC=CC=C)=O)C3C2C3)ccc(F)c(F)c1 Cc1ccnc(O)c1C(=O)NCC(C)(C)NC(=O)C(c1cccc(Cl)c1)C C1(OC)CC(CC(N2CCC(N(C(=O)CN(C)S(N)(=O)=O)C)CC2)=O)C1(C)C N1(C(CCc2n(C)ccn2)=O)CCOCC1CNC(C1CCCN1C(N)=O)=O C(=O)(C(C)(C)C(F)(F)F)N1CC(C)(C)C(CNC(=O)C(F)=C2CCC2)C1 CN1CCN(C(c2scnc2C(F)F)=O)CC1CNC(c1cc(C(N)=O)[nH]n1)=O N1(C(CNC(CC)=O)=O)CC(NC(=O)C(=O)NC(C)C)C1 C1(C(=O)OC)CC2CN(C(=O)NC(c3ccc(C(C)C)cc3)C)CC2C1 C(=O)(C(CC(F)F)C1CCC1)NCC1CCC(CNC(C2CN(C)C2)=O)CC1 C1(CC(=O)NCCCCCN(C(c2cc(COC)sc2)=O)C)CCCNC(=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C(F)C1)=O C1(C(=O)Nc2c(CC)noc2)CN(C(=O)C(CC)NC(N)=O)CCO1 c1(NCCNC(CCCC)=O)ccc(S(=O)(=O)NC2CCCC(F)(F)C2)cc1F c1(C(N2CCCN(CCNC(C3CCSC3)=O)CC2)=O)cccc2c1CCC2=O N1(C(CC2(C=C)CCC2)=O)CCC(NC(c2cc(C)oc2CC)=O)C(O)C1 c1(CNC(C(n2ccc(C)n2)C)=O)ncccc1C(=O)NOCC1CCCN1C N1(C(CC2CC(CC)OCC2)=O)CC2(CCN(C(=O)C=C(C)c3cccs3)C2)C1 c1(C(N2CC3CC(NC(C4(C5CC5)CC4)=O)C(C3)C2)=O)cnn2c1OCCC2 C1(C#C)(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)C(CC(C)(C)C)OC)CC1 C1(Cc2cn(C(C)CNC(C3C4CCCC34)=O)nn2)SC(=N)NC1=O N1(C(C(C(C)O)N(C)C)=O)CC2CC(C1)CN(C(c1cc(O)cs1)=O)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCCCC(NC(c2cncs2)=O)CC1 c1(CCCC)ccc(C(N2CC3CC2(CNC(C2CC4CCC2O4)=O)C3)=O)cc1 C(N=c1[nH]cnc(Cl)c1Br)C1OCC(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 N1(C(CN2CCC(OC)C2)=O)CCC(=CCNC(=O)Cn2cnc(C#N)n2)CC1 C1(C(N2CCC(NC(=O)CCc3ccc(Cl)s3)(CF)C2)=O)CCC(F)(F)CC1 C12(CC(=O)N(CCNC(C3(CC=C)CC=CC3)=O)C)CCCCC1C2(F)F O=C1CC(CC(=O)NC2CN(C(=O)CSc3ccccc3)C2)CCCN1 c1(CCC)ccc(C(=O)NC(C)CCCNC(=O)CC(C)C(C)C)cc1[N+](=O)[O-] C1(C)(CNC(c2ccc(CNC(CN3CC(C)(C)C3)=O)o2)=O)CCCC1O C12(NC(C(C)=CC)=O)CCC(CNC(c3cc(C)n(CC)n3)=O)(CC1)OC2 C12CCC(CC1)C(=O)NC2.N1(C(C2C(OC)CCC2)=O)CCSC(C)C1 c1(C(N(CCNC(C2(C)C(C)(C)C2)=O)C2CC2)=O)ccc(F)cc1 Cc1cc(NC2CN(C(=O)CSC(C)=O)C2)cc(NC(=O)OC(C)(C)C)c1 C1(N(C)C(C2CCCOCC2)=O)CN(C(c2cscc2F)=O)CC12CC2 N1(C(C)C)CCCC(C(=O)NCC2CC(NC(=O)C(C)(O)C3CCC3)C2)C1 Cc1cc(F)ccc1-n1cc(O)c(C(=O)NC2CCn3nccc3C2)n1 c1(C(=O)NC2C(NC(=O)CN3C(=O)CNC3=O)CC2)c(F)cccc1F Cc1cnc2n1CCCC2CNC(=O)C(CC(C)C)NC(c1ccc(F)cc1)=O c1(CC)noc(C(=O)NCCNC(C2CCN(c3ccc(C)cc3)C2=O)=O)c1C CC1CN(C(=O)C2=C(Cl)CC2)CCN1C(=O)C(F)(F)C1CCCCC1 c1(C(=O)NC2CC(NC(c3cnc(C)o3)=O)C2)sc(Cc2ccccc2)nc1C c1(C(N2C(C)CC(NC(c3ccoc3)=O)C2)=O)cc2c(nn1)CCCC2 Cc1nc(C)c(C(=O)N(C2CCN(C(C3CCOC3)=O)C2)C)o1 C1(C(=O)NC2C3CN(C(C(c4ccccc4)OC)=O)C2C3)CC2CCC1CC2 C1(CC)C(C(=O)NOCC2CCCO2)CCCN1C(C1COCC(C)O1)=O N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(C2CC3CCCC23)=O)CC1C c1(CC)cnn(CCNC(C2(c3cccnc3)CC2)=O)c1.C1(=O)COCCN1 C(CC(O)CNC(c1ccsc1NC(C1CCC1)=O)=O)NC(c1ccncc1)=O c1(C(=O)NC(C)CCCNC(C2(Cl)CC23CCC3)=O)cnc2ccoc2c1 Cc1cc(C(=O)NC2CCCC(C(=O)NC3CC4(CCCC4)C3)CC2)cc(C)c1 Cc1ccn2cc(C(=O)NC(C3CCN(C(=O)C(F)CC4CCC4)C3)C)nc2c1 Cc1cc(P(C)(C)=O)oc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C n1(CC)ncnc1CSc1cccs1.o1[nH]c(=O)o1 c1(N2CCCC(NC(C(C)(F)F)=O)C2)ncc2c(n1)NC(=O)C2 c1(CC)ncccc1C(=O)N(CC(=O)Nc1ccc(OC)cc1)CCN(C)C C1(O)(C(C)NC(C(C)=C(C)C)=O)CCN(C(=O)CN(S(C)(=O)=O)C)C1 [N-]=[N+]=NC1CC(C(N2CCC(CC3CC3)CC2)=O)N(C(=O)C(O)C(F)(F)F)C1 Cc1cn2cc(C(=O)N(C)CC3CCCCN3C(=O)C(C)n3ccnc3)sc2n1 C1(C(=O)NCC=CCNC(C(C2CCC(C)(C)CC2)C)=O)CC(C(C)(C)C)=NO1 C(C)(C(F)(F)C(F)(F)F)N.c1(OC)ccc(Cl)cc1CC(C(=O)C(=O)N)=O Cc1cnc(NC(c2ccccc2F)(C)C)c(S(=O)(=O)N2CC3CCOC3C2)c1 N1(C(C2CCCC(C)(C)O2)=O)CCC2CCCC(C1)N2C(=O)CS(C)(=O)=O c1(C(=O)NC2COCCN(C(=O)CC3CCC3)C2)ccc2c(c1)S(=O)(=O)NC=N2 C1(N(C(c2c(SC)ccs2)=O)C)CCCN(C(=O)C(C2CC(F)(F)C2)O)C1 Cc1nc2ccc(C(N3CC4CC(C3)N4C(=O)CCC(C)CN(C)C)=O)cc2[nH]1 C(CC(C)C(=O)NCC(CC(C)C)NC(c1c(Cl)n[nH]c1C)=O)OC C=CCC(CCC=C)NC(=O)CN(C(=O)C(C=C)CC)C(C)C C1(C(=O)NCC2(C)N=C(C)SC2)CC2(C1)CN(C(c1cc(C)sn1)=O)C2 C1(C)(C(N(CCCCCC=C)C)=O)CCCN(C(=O)C(C)(C)NC(C)=O)C1 Cc1nn(C)c(Br)c1C(N1CCCC1C(c1ccccc1)O)=O CS(=O)(=O)c1ccc(-c2ccnc(CNCCCCCCCCCCO)c2)cc1 Cc1coc(C)c1CNC(C1(NC(=O)C(F)OC(F)(F)F)CC(O)C1)=O CC1(C)CCCCC1C(N1CCCCC1C1CCCN(C(=O)C2=CCCC2)C1)=O N1(C(C(CCOCCO)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(C)(C)CC1 N1(c2nccc(=N)[nH]2)CCC2(CC1)CC2C(N1CC2C(C(=O)O)C2C1)=O c1(CC)cc(C)ccc1C(=O)NC(CNC(=O)C=CCN1CCOCC1)(CC)CC C(CNC(C1CCC1CNC(=O)CC1OCCC1C)=O)(C(F)(F)F)OC N1(C(C2(CCC)CCC2)=O)CC2CCC(CNC(=O)C(F)C(C)(F)F)C2C1 c1(C(=O)NCCOC(CNC(c2ccn(C)c2)=O)(C)C)cncc(P(C)(C)=O)c1 C12(OCC)CCC(CNC(c3ccc(Oc4ccc(Br)cn4)cc3)CO)(CC1)C2 c1(C(=O)NCC(CC=C)NC(=O)C(C)CCOC)ccc(Cn2ccnn2)cc1 C1(O)(C(=O)NC2C(NC(C(C)(C)SC)=O)CCOC2)CCc2ccccc2C1 c1(C(=O)NCCCCCNC(C(C)C(F)F)=O)cc(N)c2ncccc2c1 C=C(C)C1OCCC1C(=O)NCC1CN(C(c2ccc(F)c(C)c2)=O)CC12CC2 Cc1cc(CN(c2nnnn2C2CCOCC2)C)cc(C)c1.C1CCS1 C1(OC)CCC2(C(=O)NCC(C)CNC(=O)CCSC3CCCC3)CC12 C1(CNC(C2(SCC)CC2)=O)CN(C(c2ccc(C(C)F)cc2)=O)CCO1 C1(NC(Cc2c(C)con2)=O)CCN(C(c2nnsc2C)=O)C(C)C1 c1(C(=O)NC2CCCN(C(CCCN=[N+]=[N-])=O)C2)n[nH]c2ccc(Cl)cc12 CC1CC(NC(c2c[nH]c(=N)nc2O)=O)CCN1C(=O)Cc1ccccc1CO S(=O)(=O)(c1ccc(NCC(O)C2(Cl)CC2)c(Cl)c1)NC1C2(CC(OC)C2)C1 C(=O)(C1=CC(C)CC1)NCC1CC(NC(COCCCC)=O)C1 CC1CC(NC(c2cccc(=O)n2C)=O)CCN1C(c1cc(F)c[nH]1)=O N1(C(CSCCC=C)=O)CCC(CO)(NC(c2oc(C3CC3)nc2C(F)F)=O)C1 C1(C(N(C(C(=O)NCc2c(C)nco2)C)C)=O)CC(O)CN1C c1(CC(=O)NC2CCCC(NC(C3(C)CC(C)(C)C3)=O)C2)cc(O)nc(O)n1 Cc1nn2ncccc2c1C(N1CC2CCC(C1)N2C(=O)CN1CCC(C)C1)=O C1(CNC(c2n(C(C)C)ncc2Cl)=O)COC(C)(C)CN1C(=O)Cc1cscn1 C1(NC(c2nnc(C)s2)=O)CC(C)N(C(=O)CNc2nccs2)C1 N1(C(C=C2CCC(C)C2)=O)CCC2(CCCN(C(c3cnc[nH]c3=N)=O)C2)C1 O=C1CN(CC(=O)NCC2(O)CCN(C(=O)CNC(=O)CC3CCCC3)C2)CCN1 Cc1cccc(Cl)c1CC(=O)Nc1cccc(NC(=O)C(C)CN(C)C)c1 c1(C(N)=O)c(NC(C2CC23CN(C(C2CC(O)C2)=O)C3)=O)cccc1Br C(=O)(C(F)C(F)(F)F)NC(C(=O)NCCc1ccn(C)n1)Cc1cnc[nH]1 c1(C2(C)CC2CNC2CCC(CNC(=O)CN3CCOCC3)C2)ccccc1 C1(NC(C2CCC(=O)N2)=O)CC2CN(C(=O)CCc3nc[nH]n3)CC12 N1(CC)CC(NC(C(=O)CCC(C)NCc2ccoc2)=O)CC1=O C1(CC(=O)NCC2CN(C(c3cccc(N)c3)=O)C2)COC2(CCC2)CO1 c1(C(=O)NC2CC(C(=O)Nc3cccc(OC)c3)C2)ccc(C)cc1Cl c1(OC)ccc(CC(=O)NC(C2CCN(C(C3CC(=C(F)F)C3)=O)C2)C)c(Cl)c1 C1(C(=O)NCC(CC)Nc2ncc(C#C)cn2)CCC2(CCC2)CC1 C(=O)(C(CC1CCC1)NC(=O)NCC1(CCO)CCCC1)OC(C)(C)C.CO c1(OC(C)C)ccc(Cl)cc1C(=O)NCC1CCN(C(c2cn[nH]c2)=O)C1(C)C n1(C(CC)C)ccc(=NC(=O)CC(O)CNC(C2(O)CCC2)=O)[nH]1 c1(C(N2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)=O)ccc2ncsc2c1 c1(C(C(=O)NCC2(C(N)=O)CN(C(C3C(C)OCC3)=O)C2)(C)C)ccc(N)cc1 c1(CC(C(=O)N(CCSC)CC)NC(=O)CNC(=O)C2CC2)ccc(Cl)cc1Cl C1(C(N2CCC(NC(CC)=O)C2)=O)CC2(CCN1C(=O)C#CC1CCC1)CC2 C1(N(C(C=C(C)Cl)=O)Cc2ccccc2)CCCN(C(=O)CC2CC2(Cl)Cl)C1 Cn1cc2c(n1)CCC(C(=O)NCCOCCCNC(c1cncc(Br)c1)=O)C2 N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CC2CNC(=O)C=CC=C(Cl)Cl CON(CCC(=O)N1CCOC(C)(C)C1C)C(=O)c1ncnc(O)c1F c1(C(N2CCC(CNC3CC4(C(=O)OC)CC34)C23CC3)=O)ccccc1[N+](=O)[O-] c1(OC(C(=O)N(c2c(C)cc(Br)cc2)N2CCOCC2)C)cc(Cl)c(Cl)cc1Cl C1(C(=O)OCC)CC2(C(=O)NC3CC(CCS(C)(=O)=O)C3)CC1C2 N1(c2n(C3CN(C(C)C)C(=O)CC3)nnn2)CC2CC(F)CC2C1 O=C1CCC(C(=O)NC2COCC2NC(c2ccoc2)=O)CN1 C(=O)(C(F)(F)c1nccs1)NCC1N(CC(=O)Nc2ccccn2)CC1 CCC(CC(C)C)C(=O)N1CCC2C(C1)CN2C(c1cncc(C)c1)=O c1(CNC(CC(C)(C)O)=O)ccc(CNC(C2CC(=O)OC2(C)C)=O)cc1F c1(C(=O)NCC(C)NC(CCNC(COC)=O)=O)nccc(Cl)c1O C1(CNC(COC(CC)C)=O)CCC(CNC(=O)C(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NC2(CO)CC(O)C2)CC2(CCN(C(C3OC4CCC3C4)=O)C2)C1 Cc1nc2c(s1)C(NC(CCCCCC(=O)NC(C)(C)C)=O)CCC2 Cn1ncc2nc[nH]c(=NC3CCCN(CC4(c5ccccc5)CC4(C)C)C3)c12 C(=O)(C(CC(C)C)C(N)=O)NCC1(F)CCN(C(c2c(CCC)nco2)=O)C1 c1(C(N(CCOC)CCNC(=O)C(O)CC(F)F)=O)cn2ccnc2cn1 CCCC(CC)CC(=O)N(C1CN(C(=O)COC2CCC(F)(F)CC2)C1)C C1(N(c2cn[nH]c2)C(C2CCCO2)=O)CCCC12CCNCC2 c1(C(=O)NC2CN(C(C3(OC)CCS(=O)(=O)C3)=O)C2)cc2nn[nH]c2cc1F c1(C(=O)NCC2CCC(NC(C3CC4(CSC4)C3)=O)C2)cccc2cnnn12 C(CCSc1ccccc1)(C(=O)NCC1CCCC1(F)F)NC(=O)OC(C)(C)C C=C1CC(N=c2[nH]c(=NC(CCC)CCO)[nH]c3cccc(F)c23)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(=O)CC2(c3ccccc3)CC2)C1 N1(C(C=CC(=O)N(C)C)=O)CCC(C(C)(C)NC(C2(C)CCCCO2)=O)CC1 C1(C(N(CCC(C)NC(c2ccc(SC(F)(F)F)o2)=O)C)=O)CCCOC1 c1(C(=O)NC(CNC(CC2CC(OC)C2)=O)C)ccc(CO)cc1 C1(CN=C(NC(CC)CC)NC2CCc3nccn3C2)CC(F)(F)CCC1(C)C C1(CC(=O)N(CCOC(C)(C)CNC(=O)CCOC2CC2)C)CC(F)(F)C1 C1(CCNC(C=CCC)=O)CN(C(c2cc(N)ccc2Cl)=O)CCS1(=O)=O c1(C(=O)OC(C)C)ccc(CNC(c2cnc(C(C)C)o2)=O)cn1 Cc1cc(=NC(C)c2nncs2)[nH]c(=NCc2cnc(C(F)(F)F)s2)[nH]1 CC1CCC(CC(=O)NCC2COCCN2C(c2cc(CN(C)C)c[nH]2)=O)CC1 c1(OC)ccc(OC)c(CC(N2CCN(C(=O)C(O)C(C)C)CC2C(F)F)=O)c1 Cc1cc(F)cc(C(N2CCC(CNC(=O)CCCc3ccccn3)C2)=O)c1C N1(C(CCC2C(C)(C)C2)=O)CCC(F)C(NC(=O)C2=COCCC2)C1 S(=O)(=O)(c1ccc(F)cc1)N1C(C(=O)Nc2c(OC)cccc2)CCCC1 c1(CCC(=O)NCC2C=CCN2C(C2CCC(=O)N2)=O)ccc(F)cc1Br C(=O)(C1=C(c2ccccc2)CCCC1)NCCNC(c1csc(C)c1C1CC1)=O c1(C(=O)NC(CC)CNC(=O)CSc2nncs2)coc2c(C)cccc12 C1(F)(C(N(CCN(C(C(C)CSCc2cccnc2)=O)C)C)=O)CC2(CCC2)C1 CC1CCn2ncc(C(=O)NCC3CC(F)CN3C(=O)C#CC3CCCO3)c2C1 c1(C(=O)OCc2nc(C(=O)OCC)c(NC)s2)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NCC2C(OC)CN(C(=O)COCCOC)C2)ccc2[nH]ccc2c1F N1(C(c2cc(-n3ccnc3)no2)=O)CCOCC1c1cn(CC2CCCO2)nn1 N1(C(C(C)C(C)O)=O)CCC(F)(F)C(CNC(=O)CC2CCCCN2C)C1 CCC(CC)(CCNC(=O)C1=CC(C)(C)C1)NC(=O)CC1CCCC1C c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)c(F)c3)=O)C2)ccc2c(c1)NC(=O)C2 c1(C(N2CCC(C)(NC(C3C(C(C)O)C3)=O)C2)=O)ccc(Cl)c(C#N)n1 S(=O)(=O)(CCC(=O)NCC1C(C)CCCN1C(=O)C(C1CCC(=O)N1)C)NC Cc1ncc2ccc(C(=O)NCCCNC(=O)COC3CCN(C)CC3)cn12 C(c1ccc(C)nc1)=CC(=O)NC(COC)C1(C)CC1 Cc1cc(C(N2CCCC(C(N3CCN(CC4CCCO4)CC3)=O)C2)=O)cnn1 c1(CC)c[nH]cc1C(N1CC(N(C)C(c2cc(C(C)C)[nH]n2)=O)C1)=O N1(C(CSC(C)C)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC1CC(F)F C1(C#N)(C(N(C(C)CNC(=O)C=Cc2ccc(Br)s2)CC)=O)CCOC1 CC(C)C(C)CC(=O)NCc1ccc(C(=O)NC2CC(=O)N(C3CC3)C2)cc1 N1(C(C)C(=O)Oc2ccccc2)CC(COC(c2cnccn2)=O)OCC1=O c1(CC)cncc(C(=O)NC2CC(OCC(=O)NC(C)(CC)C(N)=O)C2)c1 N1(C(C=Cc2occ(C)n2)=O)CC2CC(NC(C3CC(C)(C)C3)=O)CC2C1 c1(CN2CCC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(F)c(S(C)(=O)=O)c1 C1(OC)CN(C(C2(CNC(c3ccc(C)nc3)=O)CC3(CC3)C2)=O)CC1F c1(C(=O)NC2CC(CNC(C3C(C)CC3)=O)C2)cc(C(N)=O)co1 C(C(C(=O)NCC(C)(O)CO)NC(=O)C(C)NC(C)C)OC(C)C c1(C(N(C)Cc2cc(I)ccc2F)=O)cnc2ncn(C)c2n1 S(=O)(=O)(c1cccc(NC(=O)CNC(=O)C(c2ccn(C)c2)N)c1)N(C)CC C1(C(=O)NC(C(N2CC(C(C)OC)C2)=O)c2ccco2)CC(C)(C)CCO1 c1(OC)ccncc1-c1nc(-c2ccsc2)nn1CCc1ccccc1 c1(C(N(C2CCCN(C(=O)C(C)(C)C3CCCO3)C2)CC)=O)cn(C)nc1O c1(CNC(=NCCF)NC2CCN(CC3CC3)C2)cccc2c1OCC2 C(=O)(C1=CCC(NC(=O)CCc2ccn(C)n2)C1)NC1(C)CC(C(=O)OC)C1 c1(NC(c2ccc(OC3CCC3)nc2)=O)ncc(Br)nc1C(=O)NCCCO S(=O)(=O)(c1ccc(NCCc2ccccc2Br)c(F)c1)NCc1scc(CC)c1 C1(C(=O)NC2CCN(C(C(C(C)OC)N(C)C)=O)CC2)C2CCC(F)(F)C12 N1(C(CN(C)C(C2(CC(C)=O)CCCC2)=O)=O)CCN(C(c2cnccn2)=O)CC1 Cc1cccc(F)c1C(=O)NCC1CC(C)N(C(=O)Cn2cc(N)cn2)C1 CCCS(=O)(=O)NC(C)C(=O)NCCC1(OC)CN(C(C2(O)CCSC2)=O)C1 N(C(=NCCC1(C)OCCO1)NC1CC(c2ccc(C)cc2C)C1)CC1C(=C)C1 C(=O)(C1=NOC(C2(O)COC2)C1)N1CC(NC(C(C)(C)N2CCOCC2)=O)C1 c1(CN2CCC(CCNC(c3cnc4n3CCS4)=O)C2)cc(O)nc(C2CC2)n1 C1(C(N(C(c2cn(-c3cccc(C)c3N)nn2)C)C)=O)CN(C)C(=O)CCO1 C1(C)(C(=O)NC)CCCN(C(=O)C)C1.Cc1ccc(C(=O)O)cn1.N12CCCC1C2 c1(NC2CN(C(C(n3cc(C(=O)OC)nn3)C)=O)CC2OC)ccc(C#N)cc1 c1(C(=O)NCCNC(C2C(OC(C)C)C2)=O)cccc(Oc2ccccc2)c1 C(=O)(C(CC(C)C)NC(=O)NCC1CC(OC(F)(F)F)C1)NCC(=C)C C(=O)(C(C)(C)C(O)C(C)C)NCC1C(NC(Cn2nc(C)c(Cl)c2C)=O)CC1 Cc1cc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc(C)c1F N1(C(C(C)c2ccco2)=O)CC(C)(NC(=O)C(F)Cc2ccccc2)C1 c1(C(=O)Nc2n[nH]cc2COc2ccccc2C(=O)O)ccc(OC(F)F)nc1 c1(C(=O)OCC)ccc(N(CC(C)CNC(=O)Cc2ccoc2)C)nc1 [N-]=[N+]=NCCCCNC(c1csc(CNC(=O)C(O)C2CC2)c1)=O N1(C(c2ccn(CC)c2C)=O)CCCC(C2CC2NC(c2ccc(F)s2)=O)C1 c1(N2CC3(C(NC(C4N(C)C(=O)CC4)=O)CCS3)C2)nc(Cl)nc2ccccc12 C1(C(=O)OC)CCC2(CCOCC2)N(C(=O)Cn2cc(-c3cn(C)cn3)nn2)C1 c1(OC)nccc(C(=O)NCC2CN(C(c3c[nH]c(-c4ccccc4)c3)=O)C2)n1 N1(C(NNC(C)C(F)(F)F)=O)CC2OCCN(Cc3ccccc3)C2C1 N1(c2ncc(C#N)cc2F)CC2CCCC(NC(=O)C=CCO)C2C1 CC1(C(=O)NC(CNC(c2ncc(F)cc2N)=O)C2CC2)CCCCC1(F)F C1(CNC(c2c(F)ccc(C)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)C2(CCC2)C1 C12(NC(CC(C)(C)O)=O)CCOCC1CN(C(c1ccnc(F)c1O)=O)C2 N1(C(c2cncnc2)C(=O)NCC2CCCCC2)CCC2(CC1)C(O)CC2O C1(NC(c2c(OC)n[nH]c2)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 N1(C(CCCN(C(=O)OCC)C)=O)CCCCC1C(=O)CN(C)C n1(CC)c(CN2CCC(C3CCOC3)C2)nc2cc(Cl)ccc12 N1(C(CC(C)n2ccnc2)=O)CCC(C)(CCNC(C2(CO)COC2)=O)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccncc1Br c1(C(=O)NCCC2CCC(NC(c3cc(Cl)cs3)=O)C2)cc(F)c(O)c(F)c1 CC1CN(C(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CCC(C)(C)C2)=O)CC2(CCC2)O1 C(=O)(C(C)(C)C(=O)OC)NC(CN(C(CCCC=C)=O)CC)C S(=O)(=O)(c1ccccc1C1(C)N=N1)NCC=CCCC c1(OC)cncc(C(=O)NCCOC(C)(C)CNC(C2CCCC2O)=O)c1C C1(OCCNC(=O)Cc2cscn2)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 CC1(C)CN(C(=O)C2=CCSC2)CCC1NC(=O)CC1SC(=N)NC1=O C1(NC(C2C(C)C2C)=O)CN(C(c2cc(F)c(Cl)cc2Cl)=O)Cc2nccn2C1 CCCC(CC)CCC(=O)NCC1(C(=O)N(C)CCc2ncon2)CC1 CC(C)C(F)(CNC(=O)C(C)(C)C(C)(C)C)C(=O)NC(C)CS(N)(=O)=O N1(C(C23CC(NC(C4OCCC(=O)C4)=O)(C2)C3)=O)CC(F)C(F)(F)C1 C1(NC(=O)NCC(=O)NC(CNC(C2(CO)CCCC2)=O)CO)CCCCC1 C(=O)(C1=CC(O)C(NC(=O)C(=O)NC2CC2)C1)N(C)C.C12CC(C1)NC2=O N1(C(COCCC)=O)CCN(CC(C)(C)NC(C2CC2C)=O)CC1 c1(C(N(CC(C)NC(=O)Cc2coc(-c3ccccc3)n2)C)=O)ncccc1Cl CC1(CNC(c2cc(C3CCC3)on2)=O)CCCN1C(c1sccc1F)=O N1(C(CCOC)=O)CCCC1C(=O)NCc1cnn(CCCl)c1 c1(C(CNC(N(C)Cc2ccn(C)c2)=O)(C)O)cccc(Cl)c1 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(O)(CNC(c2nc(C)sc2C)=O)CC1 c1(NC(CC2CCN(C(c3c(C)scc3)=O)C2)=O)ccc(Br)cc1O c1(C(N2CCCC(N(C(CC3(C=C)CC3)=O)C)C2)=O)cc(C)nc2c1cnn2C CC1COc2ccc(C(=O)NC3CC4C3CCN4C(=O)C=Cc3ccco3)cc21 C1(O)(CNC(C(C)=CC2CC2)=O)CCCN(C(c2ccc(O)nn2)=O)CC1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C3CC3F)=O)C2)nc1 c1(C(N2CC(CNC(C=CCOCCOC)=O)C2)=O)csc(CCP(C)(C)=O)n1 C(=O)(C1=NOC2(CCN(C(c3cnc(OCCN)cn3)=O)CC2)C1)N(C)C1CC1 c1(C(N2C(CNC(c3ccc[n+]([O-])c3)=O)CC2)=O)cccc(Cl)c1O n1(CC)c(C(=O)NCC2CCN2C(=O)Cc2csc(NC=O)n2)cnc1O c1(C(=O)NCC(CN(C(C(c2cnccn2)C)=O)C)O)cc(-c2ccco2)on1 c1(SC)cc(C(N2CCC(N(C(=O)CC(C)C3CC3)C)C2)=O)cc(Cl)c1 Cc1nsc2ncc(C(=O)NCC(n3cc(CC4CCCCN4C)nn3)C)cc12 c1(CCC(=O)NCC2(CN(C(C(C=CC)O)=O)C3CC3)CC2)ccc(=N)[nH]c1 Cc1cc(-c2cn(CC3CCN(C(C4C5C(=O)OCC45Br)=O)C3)nn2)ccc1F Cc1ccc(CC(N2CCC(C)CC2CNC(=O)CC2COCCO2)=O)cc1C C(C(C)(C)CCO)NC(c1cccc(Cl)c1)c1n(CCC(=O)OCC)nnn1 N1(C(CC(COC)C)=O)CC2(CCN2C(c2nccc(OC)c2O)=O)C1 N1(C(C(c2cn(C)nn2)NC(C(CC=C)C)=O)=O)CC2(CCOC2)C1 C(=O)(C1=C(C)CCOC1)NC(CCNC(C1CC(C)=C(C)CC1)=O)(C)C N1(C(c2cnc(C)[nH]2)=O)CCC(O)C(C(=O)NC(c2ccccc2C)C)C1 N1(CC(c2onc(-c3ccc(C)cc3)n2)N(C)C)Cc2ccccc2C(C(N)=O)C1 c1(C(C)=O)cc(NC(C2CC3CC3N2Cc2cn(C)cn2)=O)ccc1F N1(C(C2(CCCC)CC2)=O)CC2C(NC(=O)C(C)OCc3ccccc3)C2C1 CCC(C)(O)C(=O)NC(C1CCN(C(C23COCC(C2)C3)=O)CC1)C C#CCC(C)(C(=O)N1CC(Cc2ccco2)C1)NC(=O)C(C)S(C)(=O)=O N1(C(C(C2(OC)CCCC2)(F)F)=O)CCC(NC(=O)C(C)(C)C)C(F)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NCC1CN(C(CC(C)SC)=O)C1 c1(OC)ccc(CNC(CN2CCC(COC)C2)=O)cc1.C12(CC1)C(=O)NC2 C1(CC=C)(NC(c2ncc(C)cc2C(F)(F)F)=O)CCCN(C(C2(O)CC2)=O)C1 c1(C(=O)NCC2C(NC(c3cc(OC)n[nH]3)=O)C2)cc(F)cc([N+](=O)[O-])c1 CCCC(CCC)=CC(=O)NC1(CC)CN(C(C2(OCC)CCOCC2)=O)C1 N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 Cc1nc(C(=O)C(=O)NC2CCC2NC(c2ccsc2Cl)=O)cs1 C1(C(N(CC(CNC(C(C)OCC)=O)C)C)=O)Cc2cc(C)ccc2S1 C(=O)(CC(O)CNC(=O)CCCOC(C)(C)C)NC1CC(C)(C(=O)OCC)C1 Cc1cc(CCC(=O)NC2CC2NC(=O)CCc2ncc(F)cn2)cc(C)n1 CC1=CCSC1C(=O)NC1COCC1CNC(c1ccc(C)s1)=O CCCCCC(CC)C(=O)NC1CC1NC(c1cn(C)c(C)cc1=O)=O Cc1cccc(OCC(N2CC(C)(NC(c3cnsc3C)=O)C2)=O)c1 C(=O)(C1CCCc2nc[nH]c21)N(CCC(C(C)(C)C)NC(c1cncs1)=O)C C1(NC(C(C2CCOC2)OC)=O)Cc2ccccc2C1N=c1[nH]nc(C)s1 C1(NC(C(Cn2cncn2)NC(CC2(C)CCOC2)=O)=O)CCN(C2CC2)C1=O c1(CC(=O)N(CCCC(=O)O)C)ccccc1O C(=O)(CC(CC(C)C)NC(c1c(C)ccnc1O)=O)NC(C=C)C1CC1 N1(C(C(CC=CC)NC(C2CC2OC(C)=O)=O)=O)CCCN(C=O)CC1 C(C)(CC1CCC1)(C(=O)N(CCNC(=O)CCCCO)C1CC1)OC C#Cc1ccc(C(=O)NC23CCN(C(=O)Cc4nocc4C)CC2C3)nc1 c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cnn(CCC(C)C)c1C c1(CC2CC(NCC3CCCC(=O)N3)C2)ccc2c(c1)OCO2 c1(OC)cc(C(=O)NCC(O)CN(C(=O)C(C)(C)C(C)C)C)cc(OC)n1 c1(C(=O)NCC2OCCC(NC(c3cc(C)ns3)=O)C2)cc(S(N)(=O)=O)co1 c1(CC)cc(C(N2CCCOC(CNC(C3SCCS3)=O)C2)=O)c2c(c1)CCO2 Cc1c(CC(=O)N(CCCn2cc(C(O)C3CC3)nn2)C2CC2)cnn1C c1(CC(N2CCN(C(C(CC)CO)=O)CC2)=O)cccc2cccnc12 C1(C(N2CCC(NC(Cc3n[nH]c(=NC)s3)=O)C2)=O)CCS(=O)(=O)C12CCC2 CC1=CCC(CN(C(=O)CC2CCN(C(=O)C(c3ccccc3)C)C2)C(C)C)CC1 c1(NC(c2cccc(OC)c2)C)ccc(S(=O)(=O)NC2CCS(=O)C2)c(Br)c1 CC1(C2CCC(=O)N(CCNS(=O)(=O)CC3CCC4(CCCC4)O3)C2)CC1 C1(C)(NC(c2c(C)con2)=O)CCN(C(C2(F)CCOC2C)=O)CC1 C(CCF)(C(=O)N1CC(O)C(O)CO1)NC(C1C(C)(C)C1)=O c1(C(N(C2CCN(C(C(C(C)(C)C)N(C)C)=O)C2)CCO)=O)cc(Cl)c(F)cc1F C(=O)(C1=CC2CCCCCC12)c1c(C)nc(CN2CC(C)(C)CC2C(=O)O)s1 C1(C(N2CC3C(CNC(CCn4ncc(C)c4)=O)(C3)C2)=O)CC12CCSCC2 c1(C(=O)NC(CC(C)C)(C)CNC(C2CCCC2)=O)cccc2cc(O)ncc12 c1(C(CNC(=O)CNC(=O)CN(C)C)NC(C(C)SCC)=O)ccc(F)cc1F c1(C(C)=O)ncn(C(c2ncc(Br)s2)C)n1 C1(C(N(C)CC2(NC(=O)Cc3cccnc3)CC2)=O)CCCC12OCCO2 c1(NC(C2CCN(C(c3ccno3)=O)C2)=O)cccc(OCCF)c1 C(C(C)(C)C(=O)NC(C1CCOC1)CNC(=O)CCc1cccc(Cl)c1)OC c1(C(=O)NC(CC)CN(C)C(c2cncc(C)n2)=O)cnc(N(C)C)c(Cl)c1 c1(C(C(=O)NC2COC2)N(C(C(=O)OC)C)C)ccoc1C C1(NC(C=C(C)Cl)=O)CC2CCC(C1C)N2C(C1CCCCCC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CC2(CCCC2NC(=O)CCC(C)(C)C)C1 Cc1cn2cc(C(N3CC4CCC3C(CNC(=O)C(F)(F)C3CC3)C4)=O)nc2s1 c1(N2CC(C)OC(C3CC3)C2)nccc(=NCc2cnc(O)nc2O)[nH]1 C(CCCCNC(=O)C(F)(F)c1ccccc1)CCC(=O)O.c12cn(nn1)CC2 CC1(C)CN(C(=O)Cn2[nH]cnc2=N)CCC1NC(c1[nH]nc2ncccc12)=O c1(CNC(C2CC(NC(Cc3c(C)n[nH]c3)=O)C(O)C2)=O)ccc(N)c(F)c1 Cc1cnc2nccc(C(=O)NC3CC(C)N(C(=O)Cc4sccc4C)C3)c2c1 n1(CC#C)cccc1C(=O)NC(C1CCCCC1)CNC(c1cscc1Cl)=O CCC(Cc1ccccc1C)C(=O)NC1CC(NC(=O)C=Cc2ccoc2)C1 C1(C(CC)O)CCCN1CC(=O)N(C1CC(F)(F)C1)C1CC1 C=CC1CCN(C(C2CN(C(=O)C(CO)OC)CC2CCC)=O)C1 C1(C)(NC(C(CCC)C)=O)CCCN(C(C2CCN(C(=O)OC)CC2)=O)C1 C1(CNC(C2(C)CS(=O)(=O)C2)=O)CC2(CO1)CN(C(c1ccc(CO)cc1)=O)C2 CCC(C)C(=O)NCC(=O)NC(C(=O)NC(C)Cn1cc(C)cn1)C1CC1 c1(CSCC)cccnc1C(=O)N(C1CN(C(=O)CSC2CCCCO2)C1)C C12(CCNC(c3cc(CC)c(CC)o3)=O)CCC(C1)N(C(=O)C(=O)N(C)C)C2 C1(C(=O)NC(CNC(c2oc(CC)c(C)c2)=O)CC)CC2C(C1)C2(F)F CC(C(F)(F)F)NC(=O)C(F)CC1CN(C(c2coc(CO)c2)=O)C1 CCCC(CCC)CCCC(=O)NC(C)(C)CNC(=O)C(C)(C)COCC N1(C(C2(C(C)C)COC2)=O)CCC2(CCCN2C(=O)CCc2cncc(O)c2)C1 Cc1c(C(=O)OC)[nH]c2ccccc12.c12ccccc1NC2C.C1CCCCC1 N1(C(CCC=C=C)=O)CC23CCCC2(C1)CN(C(C1CNC(=O)C1)=O)C3 c1(CC)ncccc1C(=O)NCC1(O)CN(C(c2cncc(N(C)C)c2)=O)C1 N1(C(CCC)=O)Cc2ccccc2CC1CNC(c1nnn(C)c1C(F)(F)F)=O c1(OC)cc(C(N2CCC(SCC(c3cccc(Cl)c3)=O)C2)=O)n(C)c1 N1(C(C(CCC)C)=O)CCC2CCN(C(=O)C(F)C(F)(F)F)C2C1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(C)(CNC(=O)C(C)(C)CF)C1 CCCCC(C)(F)C(=O)N1CC(C)C(C)(C(N2C3CCC2CC(CO)C3)=O)C1 N1(C(CCC(C)OCC)=O)CCCC2(C1)CN(C(=O)CC1CCOC1)C2 C1(COC)(NC(C2CC3CC3C2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 CC1CCSC1C(=O)NCCNC(=O)CNC(=O)CNC(=O)CCc1ccccc1 C(=O)(CC(C(F)F)NC(C1CCCN1C)=O)NCC1(C)N=C(C)SC1 C=CCC(C)(C)C(=O)N1CCC(C(=O)N(CCCC)CCCO)C(C)C1 N1(C(C(CC)SC)=O)CC(NC(c2ncc(C)cc2C)=O)C(S(C)(=O)=O)C1 c1(SC)cccc(CNC(c2cc(C3CC3)n[nH]2)c2nnnn2C)c1 C12(CC)CCN(C1)C(=O)C1C(COC1)C(=O)N2.C1(C(=O)OC)(SC)CCC1 Cc1ccc(CC(=O)NC23CC(C2)N(C(=O)CNC(=O)CCCCO)C3)c(F)c1 c1(C(=O)NC(CCCNC(C2CCC(C)C2)=O)(C)C)cc2ncccc2[nH]1 C(CC(=O)NCc1cc(C2CC2)on1)(CC(C)C)NC(CSCC#C)=O c1(CC(=O)OCc2cccc3c2CCCC3)ccc(Cl)c2cccnc12 C1(NC(C2CCC(NC(c3c(COC)nn[nH]3)=O)C2)=O)CCCCC1CO C1(NC(C(COC(C)C)NC(C)=O)=O)CN(C(=O)C(F)(F)CO)CC1C Cc1ncc(NC(C2CCN(C(=O)CCc3ccccn3)C2(C)C)=O)c(C)c1C CN=c1[nH]c(C(N2CCCC(CNC(C3ON=C(C)C3C)=O)C2)=O)cs1 c1(CC)ncc(NC(N(C)CCC2CC2)=O)o1 N1(C(c2nc(CC)sc2)=O)CCCN(C(=O)CCCC(C)(F)F)CC1C N1(C(C2(C3N(c4n(CC)nnn4)CCC3)CC2)=O)CCN(c2cc(Cl)ncn2)CC1 CCCCCCC(C)C(=O)N(CCC(=O)NCCc1ccccc1)C1CC1 C1(NC(C(C)n2cnnn2)=O)(CNC(=O)C(C)C(F)(F)F)CCC(C)(C)CC1 c1(N(CC(=O)NC2(CNC(=O)C(C)(C)F)CCCC2)C)ccc(Cl)cc1 CN1CC=C(CC(=O)N2CC3CCC(C(=O)NCC(=O)NC4CCCC4)(C3)C2)CC1 c1(CC(N)=O)ccc(C(=O)NCC(O)CCNC(=O)CNc2ccccc2)cc1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1CN(CC(=O)NCC(C)C)CC1C S(=O)(=O)(c1ccc(=NCCCN=c2cc[nH]cc2)[nH]c1)NCC(CC)C(C)(F)F c1(NC(CN(CC(C)O)CC2(Br)C(C)C2C)=O)ccccc1 N1(C(C=C(C)c2ccco2)=O)CC(CCNC(c2ncsc2C)=O)OC(C)C1 c1(CC(=O)NC2CN(C(c3c(C(C)C)cccc3)=O)C2)cc2c(cc1Br)OCO2 n1(CC)ccc2ccc(NC(=O)C(n3cc(CC4CCCCN4C)nn3)C)cc12 N1(CCC(C)NCC23CCC(C(=O)OCC)(C2)CO3)C(=O)c2ccccc2C1=O C1(C(=O)NCC(C2CCN(C(=O)CSC(F)F)CC2)O)CC2(CCC2)C1 c1(C(N(CCOC)CCNC(C2C3CCC2CC3)=O)=O)cccc(C)c1Br N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)C2 c1(C(N2CCN(C(c3c(C)nn(C)c3C)=O)C(C)C2)=O)ccc(C#N)c(Cl)c1 c1(OC)ccccc1NC(c1ccc(-n2ccnc2)nc1)c1nnnn1C N1(S(Cc2nc(C3C(C)CCO3)on2)(=O)=O)CCCCC1c1ccc(F)cc1 N1(C(CNS(CCOCC)(=O)=O)=O)CCN(C(=O)C(C2CC2)OC)CC1C(C)C C1(C)(C(=O)NCC(C)N(C(C2CCN(CC)C2)=O)C)CCNC1=O C12(C(=O)NCC3(O)CC(CNC(C4CS(=O)(=O)C4)=O)C3)CCC(CC1)CO2 C(=O)(C(CC(C)C)C(N)=O)NC1C(CNC(c2cc(C)c(O)nn2)=O)CC1 CC1CC(NC(C2CC3(C2)CC(F)C3)=O)CCN1C(=O)CCSc1nnnn1C c1(CCNC(C2N(C(CCN3CC(=O)NCC3)=O)CCC2)=O)c[nH]cc(F)c1=O CC1(C)CC(O)(CC(N2CCC(O)(CNC(=O)CCc3ncco3)C2)=O)CO1 N1(C(C2C=CC=CC=C2)=O)CC2CCN(C(C3CC(C(F)(F)F)C3)=O)C2C1 Cc1cc(C(=O)N(C)CCN(C(c2c[nH]nc2C)=O)C(C)C)ccc1Cl c1(C(=O)NCC(CC=C)NC(c2cccc(C(C)C)n2)=O)c(C)ccc(C)c1O N1(C(c2c(C)oc(C#N)c2)=O)CC2CN(C(=O)C=Cc3cncc(F)c3)CC2C1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(C)(NC(c2ccc(OC)cc2F)=O)C1 N1(C(c2cc(C)nn2C)=O)CCN(C(=O)CN=S(C)(C)=O)CC1CC(F)F Brc1ccccc1C1(NCc2noc(Cc3ccco3)n2)CC1 C1(C(=O)OC)CCN(C(=O)CC2CCN2C(=O)Cc2ccon2)O1 c1(C(N2CCC(=CBr)CC2)C(=O)NC(C(=O)OC)C)ccc(OC(F)F)cc1Br C1(NC(CC2(OCC)CCC2)=O)CCN(C(=O)C(C)OC)CC1F N1(c2nnc(CCC)s2)CC2(COC(CNC(C3(CC)CCC3)=O)C2)C1 n1(CC(C)NC(c2cn[nH]c2)=O)cc(CNC(C2(O)CCSC2)=O)nn1 N1(C(CCCCCC)=O)CCOC2(C1)CN(C(C1(F)CCCC1)=O)C2 C(C)(C(CC)CC)NC(c1c(CNC(c2ccc(CC)s2)=O)c[nH]n1)=O N1(Cc2cn(C)nn2)CC2C3CCC(C2C1)N(C(c1ccc2ncsc2c1)=O)C3 CC(CNC(=O)CCc1cnn[nH]1)C(=O)NCc1nc(C2CC2)n[nH]1 C1(NC(c2cnsc2)=O)CN(C(c2cnc[nH]2)=O)CC1C1CC1 c1(OC)cccc(CC(=O)NCCC2CN(C(=O)CC34CCCC3C4)C2)c1Cl N1(C(CN(C2CCC2)C)=O)CC2(CC(NC(C3(C)COCCO3)=O)C2)C1 C1(NC(CC2CN(C)C2)=O)CN(C(C2(C)CNC(=O)C2)=O)CC1C(F)(F)F CC1CCCCCC1NC(C1OCCC1NC(C1CCCC1O)=O)=O Cc1ccc(F)c(N)c1C(=O)NCC(C)N(C)C(C1C(F)(F)C12CCC2)=O N#Cc1ccc(C(=O)NCC2(F)CCN(C(c3ccc(Cl)cn3)=O)CC2)cc1Cl CCC(CCC(=O)Nc1cnccc1CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CN(C)C(c2c(Cl)n[nH]c2C)=O)CC1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CC#C)(C(=O)NCC2(OC)CN(C)C2)C1 c1(OC)ccc(N=c2scc(CC3CCCO3)n2-c2cccc(C(F)F)c2)cc1 C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC2C(CN(C)C)C2)COCC1 C=CC(C)(O)C(=O)NCC1CC(F)CN1C(=O)C(C)OC(C)=O c1(C(=O)NC2(C)CC(NC(C(C)=C3CCC3)=O)C2)cc(S(C)(=O)=O)ccc1C C1(NC(C(c2cc(N(C)C)cs2)N(CC(CC)CC)C)=O)CCC(F)(F)CC1 C1(O)(CC(=O)NC2CC(C(C(=O)NC(C(CC)C)C)F)C2)CCOCC1 C1(NC(=O)CCCC2CCCCC2)CN(C(C2CC(O)C2)=O)CCC1C(F)(F)F c1(C(=O)NCC2CC(C(=O)NCC(F)CO)C2)ccc2cccnc2n1 C(=O)(C#CCNC(=O)CN(C)C)NC(C#C)(C)C1CC1 c1(C(C)=O)ccc(NC(C2CCCN2CCOCc2ccccc2)=O)cc1 C1(NC(CNC(C)=O)=O)CCN(C(c2ccc3cn(C)nc3c2)=O)CC(C)(C)C1 C1(=CC(=O)NCC(CNC(c2c(C)nsc2Br)=O)C)CCCCC1(C)C CC(C)C(CNC(=O)C=Cc1ccccc1)C(=O)N1CC2CC2C2CC12 c1(NC(C2CC(NC(c3cccc4ncsc34)=O)C2)=O)cccn2ncnc12 C(=O)(C1Cc2c(Cl)cccc21)NCC1C(C)CCN1C(c1ccc(O)nc1Cl)=O N1(C(c2c[nH]c(=NC)s2)=O)CC2(CO)CC1(C(=O)NCC(O)CF)C2 c1(C(=O)NC2(CC=C)CCN(C(COCCCC#C)=O)C2)cnc(F)cc1C O(NC(=O)C(C)CC1CCCC1)CC(=O)NCC(CCCC)OC N1(C(C=C(C)c2ccco2)=O)CCC2CCN(C(c3oc(C)cc3C)=O)CC2C1 c1(C(C(=O)NC(C)C(C)NC(=O)C(F)(F)C(C)(C)O)(C)C)c[nH]c2ccccc12 CC1(C)CC(=O)OC1CNC(=O)C=CCNC(c1cccc(F)c1O)=O c1(OC)ccccc1CCNC(c1cncc(-c2ccncc2)n1)=O C1(C(C(=O)NCC2(C(C)NC(COC)=O)CC2)F)CCOCC1 N1(c2n(CC(=C)C)c(CC(F)(F)F)nn2)CCCN(S(N)(=O)=O)CC1 Nc1sc2c(c1C(=O)NCC1CC1CNC(c1ccc(=O)oc1)=O)CCC2 C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)C(C2CCC2)OCC)CC1C C1(CNC(C2N(C(C)C)CCC2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)C1 C(=O)(C(=O)CCC(C)(C)C)NCCN(C(=O)C=Cc1ccncc1)CC N1(C(c2cccc(C)c2N)=O)CC2CC1CCC2NC(=O)CC(C)C n1(SCC)nc(C(=O)NCC2(CCNC(=O)C(CC)OC)CC2)c(C)n1 CCC(CC)C(=O)N1CC(CN(C)Cc2ccc(-c3ccccc3)o2)C1 c1(OC)cc(C)ccc1C(N1CC(F)(C(=O)NCC2COCCO2)C1)=O N1(C(C(C)n2ccnc2)=O)CC2CCC(NC(c3ncc4ccccn34)=O)C2C1 Cn1ccc2ccc(CNc3ccc(NC(c4c[nH]c(=O)cn4)=O)cc3F)cc12 c1(C(N2CC(NC(C(CC)(C)CC)=O)C(N=[N+]=[N-])C2)=O)ccc(F)c2c1CCC2 C1(NC(C(CSC)O)=O)C2CN(C(=O)CCOCC(C)C)CC12 C1(O)(C(C)NC(C)=O)CCN(C(c2cccnc2-c2ccncc2)=O)C1 C1(C(N2CCC(=CCNC(c3cnc(C)[nH]3)=O)CC2)=O)CC2(C1)CC(C)C2 N1(C(C(C)OCCC#C)=O)CCC2(C1)CN(C(=O)Cc1sc(C3CC3)nc1C)C2 Cc1nc(-n2nc(C3CC=CCC3)nc2-c2cnn(CC(F)(F)F)c2)n(C)n1 N1(C(CC=C)=O)CCC2CCCN(C(c3nc4ncc(Br)cc4[nH]3)=O)C2C1 N1(C(c2ccc(OC)c(O)c2)=O)CCCC2C1CCCN2C(C12CSC(C1)C2)=O C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)N(CC=C)C c1(C(N2CC(CCNC(c3ocnc3C3CCC3)=O)C2)=O)cccc2ncnn12 c1(C(=O)NC2CC(NC(c3c(F)cccc3F)=O)C2)ccc2c(c1)C(=O)CC2 N1(C(C2C(C=C)C2)=O)CCN(CCN(C)C(c2cncc(COC)c2)=O)CC1 CCCC(O)CC(=O)NC(C)(CNC(c1cn(CC)nn1)=O)CC(C)C C1(CC(=O)NC2(CCF)CCC2)(OC)CN(C(=O)CNC(C)=O)C1 C1(C(C)C)CC(c2nnnn2C2CCOC2)(NCC2(CO)CCCC2)C1 C1(NC(CCOCC)=O)CC2CC(NC(C3(C(F)(F)F)CC(F)(F)C3)=O)C2C1 c1(OCCNC(=O)NCCCCn2ccnn2)ccc(O)cc1 c1(C(=O)NC23CCC(C(=O)NCC4(O)CCCC4)(CC2)C3)c(F)cccc1Cl C(=O)(CC(C(F)F)N(C)C)NCC1C(C(C)C)NCC1 N1(C(C(CCOC)OC)=O)CCCCCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 Cc1noc(C)c1C=CC(=O)NCC(C(C)C)NC(=O)CC1CCOC1=O C(CC(=O)NCC1COC(C)(C)C1)(C(F)(F)F)NC(CC=CC(C)(C)C)=O C1(NC(c2ncc(N)nc2)=O)(CO)CCCN(C(C2CC(F)(CO)C2)=O)C1 CC(CN(C)C(C1CC2(CC2)C1)=O)C(=O)NC(C)C(C)(C)O CCS(=O)CC(=O)N(C)CC1(O)CN(C(=O)COc2cccc(OC)c2)C1 C(=O)(C(=O)Nc1ncc[nH]1)N(CCCNC)C N1(C(CC2N(C(C(C)(C)n3cccn3)=O)C3C2CCC3)=O)CC2COC(=O)C2C1 CC1(C)CCN(CC(=O)NC(C)(C)CCCNC(=O)CC2CSCCO2)CC1 Cc1ccc2c(c1)CC(C(N1CCC3CCC(NC(=O)CCC(F)F)C1C3)=O)S2 c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CN(C(c1coc3c1CSC3)=O)C2 c1(-c2ccc(CCCC)nc2)cccn2ncc(C(=O)NCCC(C)C)c12 n1(CC)nnc(C)c1C(=O)NCCC1COCCN1C(c1cn(C)[nH]c1=N)=O C(=O)(CC(F)(F)C(C)C)NCC(C(C)C)(C)NC(c1cncc2c1CCC2)=O C1(CC)CCOCC1(c1nnnn1-c1ccccc1)NC1CCC=CCC1 N1(C(CCN(C(CC(CC)C2CC2)=O)CCO)=O)CCC(O)C(C)C1 c1(OC)ccc(C)cc1C(=O)NC1CCN(C(=O)CC2CCCC(C)C2)C(C)C1 N1(C(C2SCCS2)=O)CCN(C(c2cccc(F)c2O)=O)C(CC(F)F)C1 C=CCCCCC(=O)N(CC(C)NC(C1CC2(CC(OC)C2)C1)=O)C C(C)(CCC(=O)NCC1CCC(C(=O)NC2(c3cnn(C)c3C)CC2)C1)SC c1(C(N2CCC(OCCNC(C3CCC(C)C3)=O)C2)=O)cccnc1S C1(CC=C)(C(=O)NC(c2cnc(F)cn2)C)CNCCO1 CCC(CC(=O)NCCCCc1ncc[nH]1)NC(C1CCCSC1)=O C(=O)(CC1CC(=O)Nc2ccccc21)NC1(C)CC(NC(C2CC=CCO2)=O)C1 N1(C(CC(C(CC)C)NC(=O)C(CCOC)OC)=O)CCC2C(=O)NCC2C1 N1(CC(Cc2ccccc2)OC)CC2CCCN(C(=O)CC3COCCO3)C2C1 C12(C(N3CCCC(NC(=O)Cn4nnc(C5CC5)n4)C3)=O)COCC(C1)OC2 C1(C(=O)NC(=O)CSCc2cn(CC(CC)C)nn2)CCCC2(CC2)C1.C1(=O)CN1 N1(C(CCC)=O)CCC2C(NC(c3ccc(C4(C)CC4)cc3)=O)C12 C=CCC(C(=O)N1CC(CCNC(c2scc(C)c2C)=O)(OC)C1)C(C)C c1(CS(=O)CI)nc(-c2cncc(F)c2)nn1-c1cccc(Cl)c1 n1(COC)nccc1C(N1CCCC1CC(=O)NC1CC(F)C1)=O C1(CNC(CCSCC)=O)CC(C)N(C(=O)C=Cc2cn[nH]c2)C1 C(=O)(C(CCC1CCC1)NC(C1CC2(CC2)CO1)=O)NCC1CCC(C)C1 N1(C(C(=O)NCCOC)=O)CCC(CNC(=O)C(c2cncnc2)C)C1(C)C N1(C(C(C2CC2)OCC)=O)CCN(C(=O)Cc2ccnc(OC)c2)C(C#N)C1 N1(C(c2ccc(OC(C)C)nn2)=O)CC2CCCC1C2CO c1(OCC)ccc(CN2CC(NC(C3CCCC3C)=O)C(F)C2)cc1Br Cc1nc2ccnn2c(C)c1C(N1CCN(C(=O)CC(C)CF)CC1C)=O N1(C(C2CCN(CCCC#C)CC2)=O)CCCC(O)(c2ccccc2)C1 Cc1cc(Cl)c(C(N2CCCC2CN(C)C(C2CCC(=O)N2C)=O)=O)s1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C=C)(C(N2CCOC3CCCC23)=O)C1 C1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)CCn2c(O)nnc2C1 C(=O)(C(C)C(C)NC(C1CC(OC2CC2)C1)=O)NCCSC(C)C C(CCCC(=O)OC)OCCN(C(CONC(c1nc(OC)oc1)=O)=O)C c1(C(N(C(C)CCNC(=O)C(F)(Cl)c2ccccc2)C)=O)ccnc2ccsc12 C1(C(N(C2CC(F)(F)C2)C)=O)CCCCN(C(=O)Cn2cccn2)C1 C1(CNC(c2c(C)coc2)=O)CCN(C(c2cn(C)ccc2=O)=O)CC1C CC1(C)CCC(NC(=O)CN(C)CCO)(NC(=O)CC2COC3CC2C3)CC1 c1(C(C(=O)NCC(C)C)N(C(c2ccc(C)cc2)C)C)cn2ccc(Br)cc2n1 N1(C(CC(C(F)(F)F)OC)=O)CC2CC(NC(c3cnsn3)=O)CC(C2)C1 c1(OC)cccc(CC(=O)NC(C)CNC(c2ccc(SC)o2)=O)c1F C1(CCC)CN(C(=O)CCc2cccs2)CCN1C(=O)COCC1CCOC1 c1(OC)ccc(C(=O)NC(C)CCNC(c2c(C(C)C)cccc2F)=O)c(F)c1 c1(OC)ccc(C(C)C(=O)NCC(C)(C2CC2)NC(=O)Cc2cn[nH]c2)c(C)c1 N1(CCC(=O)NC(C(C)(C)C)CNC(C2(C)CC3CC3C2)=O)CCSC(C)(C)C1 N1(C(C2(COC)CC2(F)F)=O)CCN(C(c2cc(C(=O)OC)on2)=O)C(CF)C1 C1(c2n(C3(C)CC3)nnn2)(NCCSCC2CCOC2)CSCCSC1 C(=O)(C#CC1CC1)NCC(CNC(c1oc(Br)cc1C)=O)OC Cc1[nH]nc(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)c1C c1(OCC)cccc(CC(=O)NCCC(C)NC(=O)CCc2ccoc2)n1 c1(C(=O)NCC2(F)CC(CNC(C3(CO)CCC3)=O)C2)cnc2c(n1)CCCC2 C(=O)(CCCCNC(=O)CC1CC(F)(F)C1)N1C(C(CC)O)CCC1 c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C(F)C2)=O)c(Cl)cccc1Cl Cc1nc(C)c(CC(=O)NC2(CNC(=O)CC3CCC(=O)N3)CC(F)(F)C2)s1 N1(C(C(=O)NCC(F)F)=O)CCCC2(CNC(=O)C3=CCCS3)CCCC12 N1(C(CSC(C)C)=O)CC2CCOCC2(NC(=O)C=CC2CCCCC2)C1 c1(CCC(=O)NCCC(C)N(C(CCCCOC)=O)C)nc2ccccc2[nH]1 N1(C(C2CC(C)(C)OC(C)(C)C2)=O)Cc2ccnc(Cl)c2C1 C1(OC)CN(C(C2CCCC(C)C2)=O)CCC1NC(c1ccncc1Cl)=O C(C1=CCN(C(=O)CCOc2cccc(Br)c2)CC1)NC(C1CC=CC1)=O c1(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)cc2n(c1)CCCC2 CCC(O)C(C)C(=O)N1CCC(NC(=O)CNc2ccc(C#N)cc2)C(C)C1 C1(C(N(CC(C)(C)NC(c2oc(C)c(Br)c2)=O)C)=O)C2CCCCCCC12 N1(C(CC(COC)C)=O)CCC(NC(c2cnsn2)=O)C(OC)C1 c1(NCC)cccnc1C(N1CCC(C)(NC(c2ncc(Cl)n2C)=O)C1)=O Nc1c(C(N2CCN(C(c3cnccn3)=O)C3CC23)=O)cccc1F C(C(=O)NOCC)(C1CCCC1)NC(C(CC)SCC(C)C)=O.c1(C)cccnc1 C1(NC(CS(=O)(=O)NCC)=O)COCCN(C(=O)C(N2CCCCC2=O)C)C1 c1(C(N(C)CC2C3CN(C(C=C(COC)C)=O)CC32)=O)c(C)[nH]c2ncccc12 C1(C(N(C)CC2CN(C(C3(n4nccn4)CC3)=O)CCO2)=O)CC2(CCCC2)CO1 c1(C(=O)NC2CC(CNC(COC)=O)C(O)C2)ccc2c(C)noc2n1 c1(C(C(N2CC(CNC(c3c(C)ccnn3)=O)C2)=O)C)c(F)cccc1F Cc1cc(C)c(CNC(=O)CC2CN(Cc3cc(Cl)nc(Cl)c3)CCO2)c(C)c1 C(=O)(C(C)(C)CN(C)C)NCC1CCN(CC)C1.C12CCC1C(=O)NC2 C1(C)(C(=O)NC2CCC(NC(c3ncn(C)n3)=O)C2)CC2(CC2)C1 C1(C2CCC2)(C(N(CCOC)CCNC(C2(C)CC(C)(C)C2)=O)=O)CC1(F)F C1(=O)NNC(=O)NC12CC(CF)C2.c1(C2C(C(=O)OC)C2)ccccc1 C1(NC(=O)Cn2cnnc2)CCCCCC1NC(c1ccc(OC(F)F)cn1)=O C=CC1(C(=O)NCCc2nc(CC)no2)CCN(C(=O)CCn2ccnc2C)C1 C(=O)(C(F)(F)C(F)(F)F)NC1CCCC(NC(CCC(=C)Br)=O)CC1 Cn1ccc(=O)c(C(N2CCN(C3CCN(C(=O)Cc4cc[nH]n4)C3)CC2)=O)c1 C1(C(=O)NCC(C)CNC(c2nnc(C(F)(F)F)s2)=O)CCCC(C)CC1 CCCCCC(C)(C)C(=O)N(C)CCNC(c1c(C)sc(C)c1C#N)=O N1(C(C2CC(C)C2)=O)C2CCC1CN(C(c1ccnc(N3CCCC3)n1)=O)CC2 c1(C(=O)NCCN(C(=O)C(C2CCCC2)OCC)CCC)cccs1 c1(C(=O)NC(C)CCNC(C2CC3(C2)CC3(F)F)=O)ccc2n[nH]cc2c1Cl C(CCCCNC(=O)CC(C)N(C)C)N(C(C=CC(C)C)=O)C c1(C(=O)NCc2scc(C(=O)NCC=CCCOC)c2)ccc(C)c(O)n1 c1(NC(C2(CO)CCN(C(C3CC(OCC)C3)=O)C2)=O)nc(OC)ccc1C CN1CCc2ccc(C(=O)NC3CC3CNC(c3cc4cnccc4o3)=O)cc21 c1(C(C(=O)NC2CCN(C(c3ncc(C)s3)=O)C2)O)ccc(F)cc1 N1(C(c2n(C)c(S)nc2)=O)CCOC2CN(C(c3ccc4nc[nH]c4n3)=O)CC12 c1(C(=O)NCC=CCNC(C2(CCC=C)CC2)=O)cnn(CC2CCOCC2)c1 C1(C(=O)NCC2CCCCN2C(c2ccc(CN(C)C)o2)=O)CCCCC12CC2 N1(C(C2=CCCC2C)=O)CCC(C2(O)CN(C(c3cc[nH]c3)=O)C2)CC1 c1(CC(=O)NC2CCC(COCCS(C)(=O)=O)C2)cc(Br)ccc1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2nc(CC)sc2N)=O)CC1O c1(NCCC=CC=C)ccc(S(=O)(=O)N2CCC(C3CCCCO3)C2)cc1F C1(C(=O)NC2CCCC2)CCCN(CC(=O)NCCN2CC3CCC2C3)CC1 N1(C(C2CCN(C(C(=Cc3ccco3)C)=O)C2)=O)CCc2ncncc2C1 C1(NC=O)CCCN(C(c2cocc2C)=O)C1.C12CCCN1N(CC)C2.C(C)(=O)O C12(OC)CCC(CNC(c3cc(C)c(Br)cc3F)=O)(CC1)CC2 C1(NC(c2c(CC)oc(C)c2)=O)CC(F)CN(C(c2ccc(C(C)O)cc2)=O)C1 N1(C(C(C)Oc2cccnc2)=O)CC(NC(=O)CSc2nncs2)C(C)(C)C1 CC(C#N)C(=O)N(CC(C)C(=O)NCc1nnnn1C1CC1)C C1(CNC(CCCOC(C)=O)=O)CN(C(=O)CCCCC(F)F)C2(CCC2)C1 c1(C(c2n(CCC(=O)OC)nnn2)NCC2(Br)CC2)ccnc(C2CC2)n1 CC1(N2CCCC2)CCC(NC(=O)CCSc2cccc(Br)c2)CC1 C1(C(N2CCC(OCC#C)C2)=O)CNC(=O)CN1C(=O)C(CC)CC Cc1csc(Cl)c1C(=O)NCC(O)CN(C(=O)C(C)C1CCCC1)C c1(-c2onc(CC3(O)CC(C(=O)OC)C3)n2)nc2cc(Br)ccc2[nH]1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(NC(c1cn(C)nc1O)=O)C2 N1(C(c2c(C)cc(F)s2)=O)CC2CCC(C1)N2C(c1cscc1C#N)=O c1(N(CCCC(=O)OCC(=O)NC(C#N)C2CC2)C)ccc(-n2cccn2)cc1 CCC(CNC(c1cnc(C(C)C)[nH]1)=O)(CC)NC(=O)C(C)N1CCC1 C1(C(N(CC(C)CNC(=O)CN(CC(C)(C)C)C)C)=O)CCS(=O)(=O)C(C)C1 Cc1cnc(C(=O)NC(CCC2CCC2)C(=O)Nc2cnc(F)cc2C)c(F)c1 c1(CC(=O)NC2CN(C(C(OC)OC)=O)CC(C)C2)ccc2sccc2c1 C1(O)(CNC(C2C(C(N)=O)C2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)CC1 C#CCC(O)C(=O)NCCCN1CCN(C(c2ccc(CC(C)C)nc2)=O)CC1 C1(NC(C(C2CCN(C(c3c(CC)nns3)=O)CC2)C)=O)CC2(C1)CN(C)C2 Cc1oc2ccccc2c1C(NC(=NCCF)NCCOc1ncnn1C)C CCS(=O)CC(=O)N1CC(C(N)=O)(CNC(=O)Cc2cccc(Br)c2)C1 C(=O)(C1=CCN(C(C2COCCN2C)=O)C1)NCCC(C)N(C)C C(=O)(C(CC1CCCCC1)CC)N(CC(C)(C)NC(C(C=C)O)=O)C N(C1c2ccccc2CC1NC(=O)Cc1ccc(CO)cc1)C(C(CC#C)C)=O N1(C(c2c(C)nn(C)c2)=O)CCCC(C2CN(c3ccnc(C(C)(C)C)n3)C2)C1 c1(C(N(CCOCCNC(CC(CC)(C)C)=O)C)=O)cc2ccncc2s1 Cc1nc(CC(=O)NC2(C)CC(NC(c3csc(C4CCCN4C)n3)=O)C2)n[nH]1 C1(NC(c2c(C(C)C)nn(C)c2)=O)CCCN(C(c2occc2C2CC2)=O)CC1 C1(NC(Cn2cc(C3(C)CC3)nn2)=O)CCOC12CCCCC2 c1(C(N2CCC(O)(C(=O)Nc3n(C)nnc3)C2)=O)coc2ccccc12 CC1(C)C2CCC(C2)C1C(=O)NCCCNC(c1ccc(N)c(F)n1)=O c1(CCC(=O)NC(CCNC(C(C(C)C)SCC)=O)C)cnc(C)nc1O C=CCC(C)(C)CC(=O)NCC1(C)CC(F)(F)CN1C(=O)C1=CSCS1 N1(CCCC(=O)N(C2CCN(C(c3c(CC)noc3)=O)C2)CC)C(=O)CCC1=O S(=O)(=O)(c1cnccc1N1CCC(S(N)(=O)=O)C1)N(CC(OC)OC)CCOC c1(C(=O)N(Cc2ccncc2)Cc2ccsc2)csc(-c2ccco2)n1 c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NCC=CCl C(=O)(C1=CCCO1)N(C(CNC(C1(C#C)CC1)=O)C)C C1(C(=O)NC2CN(C(=O)Cc3ccccn3)C2)CCCCN1CCO c1(SCC(=O)NCC(CO)NC(C2C(C)(Br)C2)=O)nnnn1C1CC1 C1(CNC(Cc2c(C(C)C)con2)=O)CC(C)(C)CN1C(C1CCSCC1)=O C(=O)(CC(CN=C(NCc1ccc(Br)c(F)c1)NC(C)C)C(C)C)OC N1(C(C(C(C)O)(C)C)=O)CCC(C(=O)NCCC(F)(F)F)C(C)(C)C1 CC1OC2(C(=O)NCC(C3CC3)N(C(=O)CC3CCC4CC34)C)CCC1CC2 c1(OC)ncccc1CC(=O)NCC1CCN(C(c2n[nH]c(C)c2C)=O)CC1 CCCCC(CC(=O)N1CCCC1C#N)NC(C1CCN(OC)CC1)=O n1(C(C)C)ncc(C(=O)NCCCNC(c2nn[nH]c2C(F)(F)F)=O)c1F c1(N2CC(C(C)NC(=O)CN3CCC(O)CC3)OCC2)ccn2nccc2n1 Cc1c(C(=O)N(C2CCCC(NC(=O)CN3CCC(F)CC3)C2)C)c[nH]c1C#N Cc1c(C(N2CCOC(c3cccnc3)C2)=O)nnn1C1CCOC1 CCCCC(CNC(c1cccnc1)=O)NC(=O)C(c1cccc(OC)c1)C C(C(C)(C)CC(F)F)NC(C(c1n(C)ncc1)NC(C1CCCSC1)=O)=O N1(C(C2C(C)CC2)=O)CCC2(CC2)CC1C(=O)NCc1ccnc(CO)c1 N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnc(O)n2CC)=O)C(C)C1C C(=O)(C#CC(C)(C)CNC(c1ncoc1C1CC1)=O)NCC1(N(C)C)CCC1 Cc1sc(C)c2sc(C(=O)NC3CN(C(C45CCC(CO4)C5)=O)C3)cc12 N1(C(CCn2ncn(C)c2=O)=O)CC(NC(c2sc(C#N)cc2Cl)=O)C(C)(C)C1 n1(CC)nccc1C1OCCC1CNC(c1cc(C)[nH]n1)=O C(=O)(CC(C=C)CCC)N1CC2C(CNC(Cc3ccc(CC=C)cc3)=O)C2C1 N1(CC2CN(C(C(N3CCC(C)C3)=O)=O)C2)CCN(C(C2CSCCS2)=O)CC1 c1(C(N2CCN(Cc3cc(C)c(O)cc3C)C3C2C3)=O)c[nH]c2ncc(Br)cc12 C1(CC(=O)NC(c2ccnn2C)C)C2CCCC2N1C(=O)C=CCO c1(C(=O)NC2CC3CN(C(COCCC)=O)C(C2)C3)ccc2c(c1)C(=O)NCC2 CCC(C)CC(=O)N(C1CCCN(C(=O)Cc2cnn(CC)c2)C1)C C1=NC(NC(CO)CC(O)C(C)(C)C)=C(C(=O)OC(F)(F)F)NC1 c1(C(=O)NCCn2cc(-c3c(C(=O)OCC)n[nH]c3)nn2)c(C)cccc1Cl C1(C(N2C(CNC(C3(C(=O)OCC)CCC3)=O)CCC2)=O)C(Cl)(Cl)C12CC2 N1(C(c2c(C)cc(C)c(Br)c2)=O)C(C)Cc2cc(F)ccc2C1C C1(C(N(C)CC2CN(C(c3nc(C)[nH]c3C(F)(F)F)=O)C2)=O)CC1C1CCCC1 C1(NC(C=C(C)C)=O)CS(=O)(=O)C12CCN(C(C1C(C#N)C1(C)C)=O)CC2 C1(CCNC(C2C(C)CCO2)=O)CSCCN1C(=O)C=Cc1cn(C)nn1 CC1(C)COCCC1NC(=O)C=CC1CCCN1C(=O)CCN1CCCCC1 C(=O)(C1CCCc2cccnc21)N1CC2(CN(C(C(c3n(C)ccc3)=O)=O)C2)C1 c1(C(=O)NCC(C2CC2)NC(C2CC(CC)(CC)C2)=O)ccc2c(n1)OCCO2 C1(C(N2CCC(C=C)C2)=O)CCN(C(=O)C(CC)CC=CC)CC1C N1(C(C(C2CC2)SC)=O)CCC=C(C(=O)NCCOCC(C)C)C1 C(=O)(N=c1ccnc2[nH][nH]cc1-2)C1C(C(NC2CCc3c(Cl)cccc32)=O)C1 C(=O)(C(C)C(C)NC(c1cnnc(C)c1)=O)NCc1occ(C)n1 N1(C(C(C)=C2CCC2)=O)CCC(n2cc(CNC(C34CSC(C3)C4)=O)nn2)CC1 c1(CN(C(=O)C(C)N(C)C)C)cnn2c1CN(C(=O)CCCc1nccs1)CC2 C(=O)(C1CCCn2cc(C)nc21)NC(CC)CNC(C1(O)CCCCCC1)=O N1(C(CCSCC(=O)OC)=O)CC(NC(=O)C(C)(C)c2ccncc2)CC1C c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC2C)cnc(Cl)cc1N N1(C(c2ccc(C)nc2)=O)CCN(C(=O)Cc2ccc(C)o2)CC1CCO c1(N2CCC(CC=C)C2)nc(NC(c2ccc(Cl)cc2)C(C)C)nc2c1CCC2 c1(C(=O)NCC(CNC(=O)COc2ccccc2O)OC)coc2c1CSC2 c1(OC)ccc(C(=O)NC2(CCNC(=O)C3=NOC(C)C3C)CC2)c(F)c1Cl CC(C)C(CO)C(=O)NC(CNC(c1cc(C(F)(F)F)nn1C)=O)C(C)(C)C N1(CC)CC(C(N2CCC(N(C(=O)CC3(OC)CCCCC3)C)C2)=O)CCC1=O C1(CN2CCN(c3ncn(Cc4ccccc4)c3)C2)CCC2(CCC2)O1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(c1ccc(NC(=O)OC)cc1)=O)CO CC1=C(C(=O)N2CCN(C(=O)CCCOc3ccccc3)C3CCC23)CCCC1 C12(CNC(c3nnc(C)s3)=O)CCCC1CCN2C(=O)Cn1ccc([N+](=O)[O-])n1 N1(C(Cc2c(C)ncnc2C)=O)CCC2(CC1)CC(NC(C1C=CCCC1)=O)C2 O=C(C1=NN(c2ccc(Cl)cc2)C(=O)CC1)N1CC2OCCOC2C1 C1(NC(=O)Cn2cc(C3(O)CCC3)nn2)CCOC12CCC2 c1(O)ccc([N+](=O)[O-])cc1C.C1(C(CNC)CC)CCCC1 c1(C(=O)NC2CC(C(=O)NCCSCC)C2)ccc(S(C)(=O)=O)cc1Cl Cc1nc(CC(=O)NCCC2CCC(NC(c3cc(F)cs3)=O)C2)cs1 N(C(=NCCCN1CCOCC1)NCc1nc(C2CC2)n[nH]1)CC1N(C)CCC1 c1(C(=O)NC(C)C(C)NC(=O)C=CCn2cncn2)c[nH]nc1C(F)(F)F N1(C(c2[nH]cc(C)c2)=O)CCC(NC(c2cc3n(n2)CCC3)=O)C(F)C1 C1(NC(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cc(F)ccc2C)C(C)C1 S(=O)(=O)(c1cccc2c1OCC2)NC1C(C)COCC1 C1(C(=O)NCCOCCn2cc(CCCOC)nn2)CC2(C1)CS(=O)(=O)C2 n1(CC(=O)NCCCCNC(CC2C(C)(C)C2)=O)cnc([N+](=O)[O-])n1 CC(CN(C)C)CC(=O)NCC1(NC(c2cncnc2)=O)CCOC1 Cc1cccc(N(C(c2cc(Br)ccn2)C(=O)NCCCC2CC2)C)c1 C(=O)(CCCC(C)(C)NC(=O)CCc1cncs1)NCC1(CC)CCOC1 C1(CNC(c2c(C)nccc2)=O)CCC2CN(C(C3COCOC3)=O)CC12 n1(C2CN(C(=O)NCC3N(S(C)(=O)=O)CCC3)C2)ncc([N+](=O)[O-])n1 CC1(O)CCCN(C(c2cc(CC3CCC3)[nH]n2)=O)CC1 C1(C(=O)NCc2ncc(Br)s2)CN(Cc2ccncc2O)CCC1O C(=O)(CC(CC)C(C)C)NCCCCC(C)NC(c1ccc(OCC)nc1)=O N1(c2n(Cc3ccccc3)c(C3CCCCO3)nn2)CCCC(O)CC1 c1(NCC(C)S(C)=O)nccc(=NCC(O)CN2CCCCCC2)[nH]1 C12(NC(c3cc(SC)oc3)=O)CCCC1N(C(C1CCc3nccn3C1)=O)CC2 C1(OC)CC(C(N2CCC(N(C(=O)Cc3ccns3)C)C2)=O)N(S(C)(=O)=O)C1 c1(OC)coc(C(=O)NCC2CC2CNC(=O)CCc2ccccc2O)cc1=O C(C)(C(=O)N=c1ccn(C(C)(C)C)[nH]1)N(C(=O)CCCC(=O)N(C)C)CCC c1(C(C(=O)N(N2CCCC2)CCC)N(CCC#N)C2CC2)cccc(C#N)n1 c1(OC)ccc(C(N2CCOCC(CNC(c3sccc3C)=O)C2)=O)c(OC)c1 C1(C(=O)NC(CCC)C)CCCN(C(c2cnn(C)c2N)=O)C1C N1(C(c2ncccn2)=O)CC(C(N2CCn3ccnc3C2)=O)CC2OCCC12 CC(C)C(C(C)NC(c1csc(-c2cccs2)n1)=O)NC(=O)CC1OCCO1 C1(S(=O)(=O)Nc2nnc(C34CC(CO3)C4)o2)(COC)CC1C CC1CC(CC(=O)NCc2cnccc2Cl)CN1C(C1(C)CC(C#N)C1)=O N1(C(C2N(C(C(SC)SC)=O)C(C)C2)=O)CC(C)(C#N)C1 Cc1cnc(NCC2C3CCCC23)[nH]c1=N N1(C(CCC#C)=O)CCCC2(C1)C(NC(=O)CCC1CCCCC1)CCN2C c1(N2CCN(Cc3c(C)nc(C)[nH]3)CC2C)ncnc2cnn(C)c12 C(C(C)(C)CNC(=O)CC(C)C1CC1)N(C(C=C(COC)C)=O)CC N1(C(C(CCC)CCC)=O)CCC(C2CCCN(C(c3cncn3C)=O)C2)CC1 C1(C(=O)NCCCNC(CCSCCC)=O)CCCN1C1CCCC1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1NC(=O)CC1(O)CCC1 CN1CCN(CC(=O)NCCC2CN(C(C3(C(F)F)CCCO3)=O)CCO2)CC1 C1(NC(c2cnc(CC(C)C)s2)=O)CN(C(c2nccn2C)=O)C2CC12 c1(-c2cc(F)cc(-n3cccn3)c2)cccc2c1oc1ccccc21 C(CC(C)C(=O)N(CC(C)NC(c1cccn1Cc1ccccn1)=O)C)OC C=CC1(C(=O)NC2CCC(NC(=O)COCCc3cccs3)CC2)CCCCC1 CC1C2CCC(C2)C1C(=O)NCc1nc(C(=O)N(c2ccccc2)C)co1 N1(C(c2scc(COC)c2)=O)CCC(C2CN(C(C3CC34CCOC4)=O)C2)CC1 N1(C(CCC=CC)=O)CCC2(CCN(C(=O)COC(F)F)CC2)C(C)C1 c1(CC)ncoc1C(=O)N(CC(=O)N(CC(O)CO)C)CC(C)C c1(SC)cc(C(=O)NCC2CC2CNC(=O)CCc2ccncn2)oc1C C(c1cc2ccccc2o1)=CC(=O)NC1CCCCN(C(=O)C2=COCC2)CC1 C1(C(=O)Nc2cccc(NC(C3C(COC)C3)=O)c2)CCC2(CCCCC2)C1 c1(C(=O)NCC(=O)NCCCCCn2cc(CCOC)nn2)ccc(Cl)cc1Br c1(CC)nc(=N)[nH]cc1C(=O)NCCCC(C)NC(c1coc(Br)n1)=O C(=O)(CC(C)CC(C)(C)C)NCCN(C(C#CC(C)C)=O)C1CCCCCC1 CCC(C)CC(=O)C(=O)NCC1CCC2(CCC2)C1NC(=O)C(C)=CC(C)(C)C C1(CC(=O)NCCCn2cc(CN3CC4CC4C3)nn2)CCC2C(CC1)C2(F)F c1(NC(C(C)C)=O)ccc(Cl)c(C(=O)NC2C=CCN(C(C3(C)COC3)=O)C2)c1 CC(C)(CNC(=O)C(CCC1CC1)NC(=O)CC1OCCCO1)C(F)F CC1CN(C(c2cn(C)nn2)=O)CCC1C(=O)NCCc1nccc(O)n1 C=CCC(C(=O)NCC(C(C)C)NC(C1CCCC1CC)=O)N(C)C C(C1CCN(C(C2(F)CC=CC2)=O)CC1)=CC(=O)NCC1CC=CC1 c1(C(N2CCC=C(C(=O)NCc3cc(Br)ccn3)C2)=O)ccc2ccccc2c1 C=C(Br)CCC(=O)NCC1(COC)CCN(C(c2cn(C)c(O)n2)=O)C1 N1(C(=O)NCCc2nc(-c3ncccn3)no2)CC2C=C(Br)C2C1 c1(OC)c(C(=O)NC2CC2C(=O)NCC2CCCC(NC(C)=O)C2)csc1C C1(NC(C2(CNC(C(C3CCOCC3)C)=O)CC3(CC3)C2)=O)CCCCCC1F CC(CC(=O)N(C(C)CCNC(c1[nH]ccc1C1CC1)=O)C)c1ccco1 CCC(C(=O)OC)C(=O)N(C(C)(C)CC(=O)N(C1CC1(C)C)C)C Cc1c(N)ccc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)c1C C1(NC(C=C(COC)C)=O)CC(F)CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(CC(N2CCCCC2=O)C)=O)CN(C(=O)Cn2cnnc2)CC1N=[N+]=[N-] c1(CC(C(C)C)C)ccc(C(=O)NCCNC(=O)CCc2ncc(F)cn2)cc1 CC(C)CC(C(=O)NC1CCN(C(=O)C=CCF)CC1O)c1ccc(Cl)cc1 c1(C(N(C2CCCC2)CCC)=O)ccc(CCNCc2ccc(C3CC3)o2)cc1 C1(C(=O)OCC)CCCN(C(=O)CC2(C)CCN2C(c2cn(C)nn2)=O)C1 CCC(CC(F)(F)F)C(=O)NC12CC(CNC(c3cnn4c3N(C)CC4)=O)(C1)C2 Cc1ccc(C(N2CCC(C(C)NC(=O)C=C3CCSCC3)C2)=O)c(N)c1F C(=O)(CC(F)(F)C(C)C)N(C1CCCN(C(c2cc(C3CC3)cs2)=O)CC1)CC Cc1cc(C(F)F)nn1CC(=O)NC1(CNC(C2(C)CCC(=O)C2)=O)CC1 c1(C(=O)NCC2CC3CCC2N3C(c2ccoc2)=O)cccc2c1C(=O)CCN2 N1(C(C(C)S(C)(=O)=O)=O)CCCC2CN(c3nccc(-n4ccnc4)n3)CCC12 C1(NC(CCCC(C)=O)=O)CCN(C(=O)C=Cc2ccc(SC)cc2)CC1(C)C C1(C(N(C)CC2CCCCN2S(C)(=O)=O)=O)COC(C)(C)O1 c1(-n2cc(-c3n(C)ncc3Cl)nn2)cc2ccccc2nc1O c1(C(=O)NCCCC(C)(C)NC(c2cncc(C)n2)=O)cc(C)c(C)c(C)c1 c1(C(=O)NC(C)(C)CNC(C2CCCN2)=O)ccnc(C(=O)NCCOC)c1.CC c1(C(C(=O)NCC(CO)NC(C=CCCC)=O)C)ccc2ccccc2c1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)CC2CC2)CC(C)(C)C1 C1(C)(C(N(C2CC3CCC2CC3)C)=O)CC12CCN(CCc1ccccc1)CC2 C1(N(C(C(C2CCOC2)OC)=O)Cc2ccccc2)CCN(CC2CCC2)CC1 C12(C(=O)NCC3COCCN(C(CNS(C)(=O)=O)=O)C3)CCCCC1OCC2 N1(C(C2(C)CCCS2)=O)CCCCC(NC(=O)CNC(N)=O)CC1 c1(C(N2CC(CCCCNC(C(C=C)(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(C#N)c1 c1(C(N2CCC(C(C)NC(CC(C)SC)=O)CC2)=O)ncc(F)c2ccccc12 C(C1=Cc2ccccc2OC1)=CC(=O)N(C1CN(C(CSC(C)C)=O)CC1O)C C(=O)(C#Cc1ccccc1)NCc1cccc(C(N2C(CC)CC(O)C2)=O)c1 C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)Cc3c(F)cccc3Cl)CC2C1 CC1CN(C(c2c(Cl)cnn2C)=O)CCC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C2(CCNC(C(CC)CC)=O)CCCC2)=O)CCN2CC(C)CC2C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2(CC(CNC(=O)C(C)C3(O)CCC3)C2)C1 C(C(CNC(c1ccc(C2CCOC2)s1)=O)C(F)(F)F)NC(c1cnsc1)=O c1(C(N2CCC(CNC(C34CC(F)(C3)C4)=O)C(F)(F)C2)=O)ccc2oncc2c1 CC(F)(F)CCC(=O)NC1CCCC1NC(=O)Cn1ccnn1 S(=O)(=O)(c1c[nH]c2ccc([N+](=O)[O-])cc12)NC(c1c(Br)sc(C)c1C)=O c1(C(=O)NCC(CC=C)NC(c2ccon2)=O)ccnc(CC(C)C)n1 CC(C)C(O)C(C)C(=O)NCc1cc(C(=O)NCC2(C)CCC(=O)N2)no1 n1(CCO)nc(C2CC2)nc1-c1ccc(C(F)(F)F)o1 C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(c1cnc(O)o1)=O CCCC(C)(O)CC(=O)N(C)CC=CC(N1CCOCC(C)C1)=O c1(NC(C(CCC)C)C)ccc(S(=O)(=O)NCC2(C)CC2)c(Cl)c1 c1(OC)ccc(C(C)(C)C)cc1NC(C1CCCN(C(=O)NC2CCCO2)C1)=O C(=O)(C(COC)C(F)(F)F)NCC1CC(NC(C2C(CCC)CCC2)=O)C1 c1(OC)cccc(C(=O)NC(C2CCCCN2C(=O)CNc2ccccc2)C)c1 c1(N(C)CCN2CCCCC2)nccc(=NCCNC2CCCS2)[nH]1 C1(CC(=O)N(C2CCN(C(=O)Cc3csc(Br)c3)C2)C)CCC(O)C1 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)C)ccc2sccc2c1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC12CC2)NCCC(=O)NCC#C C1(COC)(NC(c2cc(OC)ns2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 C(CC(C)(C)C(=O)N1CC2(NC(=O)C(C)OC3CCCCC3)CC1C2)SC N1(C(c2cc(SC)c(F)cc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1cn[nH]c1 c1(N(C)C)ccccc1C(N1CCC(CNC(c2cnc(C3CC3)[nH]2)=O)C1)=O N1(C(C(=O)NC(C)Cc2cc(O)cc(Br)c2)=O)CCC(=C(F)F)CC1 Cc1cc(NC(=O)CN(C)C(c2ncnn2C)=O)ccc1O c1(C(=O)NC2CC(O)(CNC(c3c(C)cc(F)s3)=O)C2)cn2cccc(C)c2n1 N1(C(CCOCCOC)=O)CC(NC(C2CCC(=O)O2)=O)C2(CCC2)C1 CC1=NOC(=O)C1CC(=O)NCC1(O)CC(NC(C2(O)COC2)=O)C1 C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C12CC2 S(=O)(=O)(C1CCOC1)NC(CC(=O)OC(C)(C)C)Cc1ccccc1 C12(C(N(C)CC3CCN(C(c4ccc(C#N)[nH]4)=O)CC3)=O)CCC(C)(C1)OC2 N1(C(C2C(CNC(C=C(CC)CC)=O)OCC2)=O)CCOCC1CCC CCS(=O)(=O)CC(=O)NC1C2CN(C(c3ccc(C)nc3O)=O)CC12 N12CCC3(CC1)CC3C2=O.c1(C(=O)O)ccc(-c2cn(CCCN(C)C)nn2)nc1 n1(CC(=O)NC(C2(O)CN(C(c3c(N)cccc3Cl)=O)C2)C)cnc([N+](=O)[O-])n1 c1(C(C)C)noc2ncc(C(=O)NC(C)CCNc3ncnc(O)c3Br)cc12 C1(NC(Cc2c(C)occ2)=O)CCCN(C(=O)CCn2cccnc2=O)CCC1 N1(C(C(CCOC)NC(=O)Cn2nccn2)=O)CCOC(C)CC1 c1(C(N2CCCC(C(N(CC(=O)NC)C)=O)C2)=O)cc2c(C)cc(OC)cc2[nH]1 CC1CN(C(c2sc(Br)cc2F)=O)CCN1C(=O)Cc1ccc(F)cn1 c1(OC)ccc2c(=NC(C)C3CC4(CCC4)C3)[nH]c(=NCc3cccs3)[nH]c2c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)C2)csc2nccn12 c1(C(N2CC(NC(C3C(CC)CCO3)=O)C(C)C2)=O)c(N)cc(Cl)cc1F C(C)(C)(CCN(C)C)NC(CSCC#C)=O.C1(C2CCC2)C(=O)N1 c1(NCC(Cc2ccc(C)cc2)OC)nc2cnc(Cl)cc2s1 C(CN=c1[nH]c2c(c(=NCC3COCC(C)O3)[nH]1)CCC2)c1nc(C)oc1C Cn1c(C(=O)NCC2CN(C(C3CS(=O)(=O)C3)=O)CCO2)cnc1Cl c1(OC)cc2[nH]c(C(N3CC(C)CCCC3C(=O)O)=O)cc2c(Cl)c1OC CC1CCN(C(=O)CC2CC(F)(F)C2)CC1CC(N1CCCN(CCO)CC1)=O c1(C(=O)NC(C(=O)N(CC=C)CC=C)c2ccoc2)ccnnc1O c1(C(=O)NC(C)(CNC(=O)Cc2c[nH]ccc2=O)C2CC2)ccc2snnc2c1 C1(C)(CNC(C2C(OCC)CCC2)=O)CCCN(C(c2conc2CC)=O)C1 c1(OC)ccc2c(=NCc3ccc[nH]3)[nH]c(=NCc3csc(O)n3)[nH]c2c1 Cc1cc(C(=O)NCCCOCCNC(c2coc(Br)n2)=O)nnc1C CC(=O)CCCC(=O)N1CCCC(CNC(=O)C(O)Cc2[nH]cnc2C)C1 C12(NC(C(=O)N(CCNC(C)=O)F)C)CC(CO)(C1)OC2(C)C.S(C)(=O)(=O)N N1(C(C(CCC)NC(C)=O)=O)CCN(C(C2CN(C)C2)=O)CC1CF c1(C(N2C(C)(C(=O)NC(C3(CO)CC3)C)CCC2)=O)ccc2cncn2c1 c1(CN2C(C(N3CCC(c4ccc(Cl)s4)C3)=O)CC(O)C2)cccc2cc[nH]c12 CC(N=c1ccc(C#N)n[nH]1)C1CCCN(C(=O)CC(c2ccccc2F)C)C1 N1(C(c2cc(C)c(F)nc2)=O)CCC(C2CC2)C1CNC(c1c(C)noc1C)=O c1(N(c2ccccc2)C(=O)CCc2cncs2)ccc(C(=O)CF)cc1 C1(CC(=O)N(CCC)CCNC(c2cc(C(F)(F)F)no2)=O)CN(C)CC1O c1(OC)cc(C)c(CN2CC(C(=O)Nc3nc(Br)c(Br)cc3Br)C2)cc1OC c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C)sn3)=O)C2)cc(Cl)c(N)c(Cl)c1 c1(OCC)nccc(C)c1C(N1CCC(NC(c2csnc2Cl)=O)C(O)C1)=O C1(C(=O)OC)CC2(C1)C(C(=O)Nc1c(Cl)cc(OC)cc1Cl)C21CCC1 C1(n2cc(Sc3ccc(C)cc3)nn2)CCCN(C(=O)C2=NOC(C)C2)CC1 N1(C(c2ccn(C)n2)=O)CCN(Cc2cnco2)CC1Cc1ccccc1 CCCN=C(NCC1CCCSC1)NCC(C)(C)Oc1ccccc1 c1(C(=O)NC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCC2CCCC2NC(=O)CNc2ccc(Cl)cn2)CCC(=O)N1 N1(C(CC=C(C)C)=O)CCC2CN(C(c3cc(S(C)(=O)=O)cs3)=O)CC2C1 N1(C(CCCSC)=O)CCN2CCN(C(c3ncnn3C(C)C)=O)CC2C1 c1(C(C)OCC)cn(C2c3ccccc3N(C(C3CC34CC4)=O)C2(C)C)nn1 N1(C(CC(=C=C)C)=O)CCC(O)(C2(NC(c3cn(C4CC4)cn3)=O)CC2)CC1 C(c1ccncc1)=CC(=O)N(C1CCC(NC(c2cncn2C(F)(F)F)=O)C1)C c1(C(N2CC(C)OC(C)C2)C)ccc(S(=O)(=O)N2CCCN(C)CC2C)cc1 C(=O)(C(F)(F)CC(C)C)NCCC1CCC(NC(C(C)=C2CCCC2)=O)C1 C#CCCC(O)CCNC(=O)C(C)(C)CNC(C1CC=CCC1)=O C1(NC(c2cccc(C3CCC3)c2)c2n(CCOC)nnn2)COCCC1(F)F C1(CCC)(NC(C2CCOC(=O)N2)=O)CCN(C(=O)C(C)(C)OC(C)C)CC1 Cc1n[nH]cc1CC(N1CCC(N(C(C2CCOC2C2CC2)=O)CC2CC2)C1)=O C1(C#N)(CNC(C(CCSC)NC(=O)CC2COCC(C)O2)=O)CC(C)(C)C1 C1(C(=O)NC(CN(C(c2ccc(OC(C)C)cn2)=O)C)(C)C)COCCC1(F)F N1(C(C2C(=C)CC2)=O)CCC(CO)C(NC(=O)COCC(c2ccccc2)=O)C1 C(=O)(CCCCCO)NC(C)CNC(=O)CCN1CCCCC1 Cc1cc(C(=O)NC2CC2CNC(c2cc3ncccc3o2)=O)c2c(c1)CCC2 c1(CN2CC3C(C(=O)Nc4c(OC)cc(Cl)cc4)C3C2)ccc(OC)c(C#N)c1 n1(CC)ccc(C(N2CCOC(CCNC(c3ccc(Cl)[nH]3)=O)C2)=O)c1C c1(C(=O)OC)cn(C)nc1C(=O)NCC1(NC(C2CCCC2(C)C)=O)CC1 c1(C(N(C)CC2(CNC(C3C(CCOC)C3)=O)CC2)=O)cc(Cl)no1 N1(C(c2cc(C(C)(C)C)on2)=O)CCC(O)(CCNC(C23CCC(CC2)O3)=O)C1 CC(C(C(=O)NC1CCOCC1)N(C1CC(=O)NC1=O)C1CC1)C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC(O)(CN(C)C(c2cc(C(C)(C)C)n[nH]2)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1(CO)CCN(C(C2C=CCS2)=O)C1 Cc1nn2cc(C(=O)NC3CC4CCC3N4C(C3C(C)C3C)=O)nc2s1 CC(C(=O)NC1CCCCC1CNC(c1cc2c(s1)CCC2)=O)C(C)(C)C C12(NC(=O)CC34CCC(CC3)C4)CCOCC1CN(C(=O)C(F)(F)C(F)(F)F)C2 Cc1cc(F)cnc1C(=O)NC12COC(C1)C(NC(=O)CCc1nccs1)C2 c1(C(=O)NC23CC(NC(c4ccn(C(F)F)n4)=O)(C2)C3)cc([N+](=O)[O-])ccc1O CC1=NC(C(=O)NCCCOCCNC(c2ocnc2C(F)F)=O)CS1 c1(CC)cnc(O)c(C(=O)NC2CCN(C(=O)CN(S(C)(=O)=O)C)C2C)c1 N1(C(NNC(c2nc(Cl)c(Br)cc2F)=O)=O)CCCC2CCCN2C1=O N1(C(CC(=O)OCC)=O)CC(C)CN(C(C2CCCN2C(C)=O)=O)CC1C C1(C(N2C(C(=O)NC3CCC(O)C3)CC3CC32)=O)CCc2ccccc2C1 N1(Cc2n(C(C)(C)C)ncc2)CCC2CN(C(c3ccc(Cl)nc3)=O)CCC12 c1(COC)cncc(C(=O)NC2CCCC2NC(=O)CCCc2cc[nH]n2)c1 C=C(C)CC(C(=O)NCCCc1cnn[nH]1)NC(C1OCCC1(C)C)=O N1(C(C(c2n(C)ccc2)=O)=O)CC2CC2(C(N2CCOCC2CN(C)C)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCC1C(CNC(Cc2cc(C)c(O)cc2)=O)C1 c1(OC)nccc(C(=O)NC2CC(NC(c3ccnc(OC)c3F)=O)C2)c1F C1(NC(C(CSC)C)=O)CCCN(C(c2csc(-c3ccc(C)o3)n2)=O)C1 N1(C(C(=O)NCCOC)c2ccsn2)CC(C)C12CCOCC2 N1(C(CCCC2C(C)C2)=O)CCC(C)(CCNC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(=O)NC2CCC(C)N(C(c3ccc(C#N)[nH]3)=O)C2)ccc2c(c1)CCOC2 C(CCC[Si](C)(C)C)N(C)C(c1ccc(Br)cc1CC#N)=O Cc1cccn2cc(CC(=O)NCC(C(C)C)NC(C3CC(=O)C3)=O)nc12 N1(C(=O)Cc2ccc(Cl)cc2)CCC2(CCCN2C(=O)COC2CCCC2)C1 N1(C(CC)=O)CCc2c(CNC(c3cc(Cl)c(C)cn3)=O)cccc2C1 C(CC(O)C(=O)N1CCC(C(N2CCC(COC(C)=O)C2)=O)(CO)C1)SC C1(CC(=O)NCC2CC(NC(=O)CCSC3CCCC3)C2)(OC)CCC1 c1(C(N(C2CCN(C(C3(CCCC)CC3)=O)C2)C)=O)ccc(Cl)cc1C c1(C(c2n(CC)nnn2)NCc2cnn(CC(F)(F)F)c2)cc(C)c(C)nn1 c1(C(=O)NCC(C)N(C(c2cccc(NC(C)C)c2)=O)C)cnc2occc2c1 c1(C(=O)N(c2ccccc2)CCC2CN(C(=O)CC3CCC3)C2)n[nH]cc1CO N1(C(CCSC)=O)CC2CC1CN(C(C1OCCC1C(C)C)=O)C2 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2)[nH]c(C)nc1C CC1OC2(CNC(c3ccns3)=O)CC1(NC(=O)CCn1ccnn1)C2 c1(C(=O)OCCSCC2(OCC)CCOC2)cc([N+](=O)[O-])ccc1N1CCCC1 C(=O)(CC1=NNC(=O)C1)N1C(CCCC)CN(C(C2(C)CCCS2(=O)=O)=O)CC1 C1(NC(C2N(CC)CC2)=O)CCC2(CC1)CC2NC(c1ccoc1)=O C(CCN=C(NCCn1cncn1)N1CC(C)N(C)C(C)C1)SC c1(C(N(CC(N2CC(CNc3ccccn3)C2)=O)C)=O)cccnc1S C(=O)(CCC(C)(F)F)N(C1CCN(C(CC(C)O)=O)CC1)Cc1ccccn1 N1(C(CS(C)(=O)=O)=O)CC2CC(O)C1C2NC(=O)CNC(C1CCC1)=O C(=O)(CCC(C)NC(c1cn(C2CC2)nn1)=O)N(CC)CC1CCC1 N1(C(C2(F)CCN(C(CC(CC)C)=O)C2)=O)CCC(CO)C(C)(C)C1 c1(CC)ccc(C(=O)Nc2ccccc2COCC(F)(F)F)cc1C#N c1(C(=O)NC(COC)C#N)cc(Cl)cc(Cl)c1F CCCCC(C)C(=O)N(C1CC2CCC(C1)N2)C(C)(C)C(N)=O C1(NC(c2n(C)ccn2)=O)CCN(C2CCN(C(=O)CC3CC3(C)C)C2)CC1 CC(C)CC(CNC(=O)CN1CC=CC1)C(=O)NCCNC1(C2CC2)CC1 C1(CNC(CCCCNC(C2CC(C#C)(O)C2)=O)=O)OCC2CCC1C2 C12(CNC(CCCCC=CC)=O)CCC(CC1)N(C(=O)C(C)OC)C2 c1(NC(CC=C)CC)[nH]c(=NCC2CCC23CCOCC3)nc2c1ncn2C C1(NC(=O)OCCOCC)CN2CC3CC2(CO1)C3 C1(OCCOC(c2[nH]cc(C#N)c2)=O)CCS(=O)(=O)CC1 N1(C(C2CNC(=O)N2)=O)CCC(CO)(CNC(c2cnc(Cl)s2)=O)C1 c1(C(=O)NCCc2cccc(C)c2)cc(Br)c(C)c([N+](=O)[O-])c1 C1(NC(c2ccc(CNC(c3cccc(C)c3)=O)cn2)=O)C(C)CCCC1C C1(CNC(CSC(C)C)=O)CCN(C(=O)CCc2cncs2)CC1C c1(C(=O)NC2C3(CC(NC(C(CC#C)O)=O)C3)C2)cccc2ccsc12 C1(C(=O)OCC(c2scc(C(C)=O)c2)=O)CC(C2CCCCC2)CN1C c1(C(=O)NCCOC2CCN(C(c3c(C)snn3)=O)C2)ccc2c(c1)NCCC2 N1(C(c2n(C)nc(Br)c2)=O)CCC2(CC1)CC(NC(=O)C1=CCCOC1)CO2 N1(C(CCc2n(C)ncc2)=O)CCC2C(C1)CN2C(C1CC1c1nc[nH]n1)=O c1(CNC(C2(CNC(CCC3C(C)C3)=O)CC(F)(F)C2)=O)cnc2ccccn12 CCCC(C)(CC)C(=O)N1CCC(=O)C(c2nn[nH]n2)C1.CC(C)(C)O N#Cc1ncccc1NC(C1CC(F)(F)CN1C(c1ccco1)=O)=O N1(C(C2C=CC(NC(CCOC)=O)C2)=O)CC2COC(=O)C2C1 C1(NC(c2scc(C(=O)NCCC(=O)NCCCO)n2)=O)C2CCC3C(C2)CC13 c1(OC)ccc(C(=O)Nc2ccc(CS(C)(=N)=O)c(Cl)c2)cc1Br N1(C(CCNC(=O)OC)=O)CC2CCC2(CCNC(c2c(C)nn(C)c2C)=O)C1 C1(NC(c2c(C)sc(O)n2)=O)CC2CC(NC(=O)CC(=O)N(C)C)CC2C1 N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)C(C)CCN(C)C)CC(O)C1 c1(C(=O)NC2CN(C(c3n(CC)ccn3)=O)C(C)CC2)cnn2cnnc2c1 Cc1cccc(CNC(=O)CCN(c2ccccc2O)Cc2ncc(Cl)n2C)c1 Cc1cc(NCC2(C)CCN(C(=O)C(C)C(C)(C)C)CC2)c(F)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)N(C1CC2CN(C(c3n(CC(C)C)ncc3)=O)C1C2)C c1(C(=O)NC(CC(C)NC(=O)OC(C)(C)C)C)cncc(CC2CCOCC2)c1 C1(C)(C(=O)NCCC(CCNC(c2ncn(CC)c2)=O)C)CCC(C)=C(C)C1 CCCCC(C)CCC(=O)NCC1OCCC1C(=O)NC1CC(N2CCCC2)C1 c1(NC(CN(C2CN(Cc3ccc(O)cc3)C2)C)=O)ccc(OC(C)(C)C)cc1 c1(C(c2ccccc2)NC(c2c(C)non2)=O)ccc(S(N)(=O)=O)cc1 CC(C)(O)CCCCCC(=O)NCCN(CCOCCO)C(C1CC2CC1C2)=O N1(C(C(N2CCC(O)CC2)C)=O)CCCC(NC(c2cc(F)ccc2N)=O)CC1 C1(NC(COC(C)C)=O)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)CC12 Nc1cnc(C(=O)NCCC2CCCN(C(=O)CN3CCC(F)CC3)C2)c(Cl)c1 C1(C(=O)NCCOc2ncccc2C(F)(F)F)COc2cc(O)ccc2C1 C1(C(=O)NCC2(CC(=O)NCC3CCC(C)(C)O3)CC2)CC2(CCO1)CC2 C(=O)(CC(C(F)F)NC(=O)C(C)=C(C)C)NC(C=C)C N1(C(C=CCC)=O)CC(C(F)(F)F)OCC1CNC(c1occc1CC)=O Cc1[nH]cc(C(=O)NC2CC3CCC2(NC(c2ccsc2)=O)C3)c(=O)c1Cl CN1CC2CCN(C(c3ccoc3CNC(c3sccc3Cl)=O)=O)C2C1 C1(NC(c2cc(Cl)c[nH]2)=O)CN(C(=O)C(F)(F)c2ccncc2)CC12CC2 Cc1ccn(CC(=O)NC(C)C(C)NC(c2cccs2)=O)n1 c1(C(CC)NC(=O)C(C2CCCO2)NC(=O)COCC(F)(F)F)ccccc1 CCC(CC(=O)NC12CC1CN(C(=O)CCc1ccc(F)nc1)C2)CC(C)C Cc1cc(O)c(C(=O)NCCC(C)NC(=O)CC2C=CCC2)cc1Br C(CCC(C)(C)C(=O)NCC1CC(C(=O)NCC2CCCC2)=NO1)OC N1(C(CC(=C)C)=O)CC2(CCN(C(c3cnn(CC(F)(F)F)c3N)=O)CC2)C1 c1(C(C)=O)ccc(C(=O)NCC(C2CC2)NC(=O)CCn2ccc(=N)[nH]2)nc1 c1(C(N(CC)CC2CCCN2C(C2(C)CCCN2C)=O)=O)ccn(C)c(=O)c1 C1(C(=O)NCc2cc(C(=O)NCC(C)F)no2)COCC1(C)C N1(C(C(CCF)NC(C=C(CC)CC)=O)=O)CCc2ccsc2C1 C1(C(C)C)(N(CCCCn2ccnc2)C(=O)NC2CC3CC3C2)CCN(C)C1 N(C1C(=O)NCc2ccccc21)C(C1CCCN(C(CC(C)N(C)C)=O)C1)=O N1(C(C(N2CCC(c3c(OC)cccc3)CC2)=O)=O)CCCC2(CNC(=O)C2)C1 c1(CC(N2CC3C(CN(C(C(C)NC(CC)=O)=O)C)C3C2)=O)cccc(F)c1O CCC(C)(CNC(=O)C(Cc1cnc[nH]1)NC(c1ccc(=N)[nH]n1)=O)C(N)=O N1(C(C=C(C)c2cccs2)=O)CCC(C)C(NC(C2CCCS(=O)(=O)C2)=O)C1C C1(C2CNC2=O)CCCN(C(=O)C(C)=CC=CC)C1.C(C)(=O)OC C1(C(=O)NC2(CNC(CCC)=O)CCCCC2)CCc2nn[nH]c2C1 C1(NC(C(C2CC(F)(F)C2)OC)=O)C=CCN(C(c2ccc(CO)nc2)=O)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2C1CCCN2C(C1CCS1(=O)=O)=O CCC(CN(C)C)C(=O)N(C(C(=O)N(CC(C1CCCC1)O)C)C1CC1)C C1(NC(C2(CC=C)CCC2)=O)CC2CCC1C(NC(c1csc(C(C)=O)n1)=O)C2 n1(CC(N2CC(C)(CCC(N3C(CCC)CCCC3)=O)C2)=O)ccc(O)nc1=O N1(C(C(C)N(C(C)=O)C)=O)CC2(C1)SCCC2NC(=O)CSC(F)(F)F C(c1ccccc1)=CC(C(=O)NC1CC(C)(NC(c2cc(C)on2)=O)C1)C c1(C(N(C)Cc2ccccc2CNC(C2CCSC2)=O)=O)ccc2occc2n1 c1(OC)cc(F)ccc1CCNC(c1nnnn1CCCC1CC1)c1ccon1 C=C(C)C1OCCC1C(=O)NCCOCCNC(c1ncoc1-c1ccon1)=O CN1CCc2[nH]nc(C(N3CCCC(CCNC(C4(C#N)CCC4)=O)C3)=O)c2C1 c1(C(N2CCC(C)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)cc2sccc2s1 N1(C(C2ON=C(CC)C2)=O)CC2CCCC1(CNC(=O)Cn1cccnc1=O)C2 C1(OCC)(CNC(C23CCC(SC)C2C3)c2nnnn2C)CCCOC1 CCCCCC(=O)NC(c1nocc1C(=O)NCC1CCOC1)C C(=O)(CCCC(F)(F)CO)N1CC(NC(C(c2cccc(C)c2F)O)=O)C(O)C1 C(CC(O)C(=O)NCC1(F)CC(NC(c2cc(C(F)F)ncn2)=O)C1)N(C)C c1(OC(C)C)cc(NC(C2CC3CC3N2C(=O)C=CC2CC2)=O)c(F)cn1 c1(C(=O)NC(C)CCCNC(C2COCCC2(F)F)=O)ccn2ncccc12 C(=O)(CCC(=O)NC1(CNC(C2CC3C=CC2C3)=O)CCCCC1)OC Cc1ccc(Cl)c(N)c1C(=O)NC(C1CCCN(C(=O)CSS(C)(=O)=O)C1)C c1(C(=O)NC2CN(C(c3cc(Cl)ncc3F)=O)CC23CC3)cc(Br)cc(Br)c1O Nc1c(F)cc(F)c(F)c1C(=O)NC1CCN(C(C2(C3CCC3)CC2(F)F)=O)C1 CC1CCC(CNC(c2ccc(O)cc2)=O)N(C(=O)Cn2cc(Cl)cn2)C1 Cc1cnc2cc(C(=O)NC3COCC3CNC(c3cc[nH]n3)=O)nn2c1 c1(CN2C(=O)CNC(=O)C=CC2)ccc(F)cc1SC.c1(N)ccc(Cl)cc1.CO c1(C(C(=O)N(CC(C)CN(C)C)CC=C)C)ccc(Cl)c(Cl)c1.C(=O)(CC1CC1)NC Cc1cc([N+](=O)[O-])cnc1NC(=O)NCCc1ccc2nc(OC)ccc2c1 C1(CNC(c2n(CC)ccn2)=O)CCC2(CN(C(=O)CC3CCCCN3C)C2)O1 C1(NC(CS(=O)(=O)NC)=O)CCN(C(c2cc(C)[nH]c(=NC)n2)=O)CCC1CO c1(NCc2cccc3c2NC(=O)C3)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CNC(CC(CC)C)=O)CCN(C(c2ccnc(C)c2)=O)C1(C)C c1(CCC(=O)NC(CC#CC)C(=O)OC)ccc([N+](=O)[O-])cc1Cl CN(CCCC(=O)N1CC(CCNC(=O)CCc2cccnc2Cl)C1)N=O CCCCCCCCC(C)C(=O)NCC1CN(C(c2cncnc2C)=O)C1 c1(C(=O)NC(c2cccnc2)C(=O)N(CC)Cc2ccccn2)ccnnc1O C(=O)(C(C)(C)C1CCCCO1)N1CC(CNC(C=C(C)C(C)C)=O)C1 c1(CC(=O)NC2CCCN(C(C(C=C)O)=O)C2C)nc(F)c(F)cc1F Cc1cc(N)c(C(=O)NC(CNC(c2cc(C)c(C)s2)=O)CO)c(F)c1 n1(CC)cc(Cl)c(C(c2nnnn2C2(C)CC2)NC(c2ccccc2F)C)n1 c1(C(N(CCNC(C2(C)CC2(F)Cl)=O)C2CC2)=O)ccc(F)c2[nH]ccc12 c1(C(=O)NCC(CN(C(C2CCCN(CCC)C2)=O)CC)(C)C)cccc(F)c1O O=S(=O)(c1ccc(Cl)cc1Cl)N(c1nc2ccccc2o1)C1CC1 c1(C(N2C(CCCNC(C3CN4CCN3CC4)=O)CCC2)=O)cc(F)ccc1F S(=O)(=O)(c1[nH]c(=NCC23CCC(CC2)C3)ccc1Br)NC(C(C)C)CCO CCCCC(C)C(=O)NCC(O)CCNC(c1cccc(C(=O)NCCC)c1)=O C1(C(N2CCC=C(CNC(C3CC(=O)NC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1ccc(CC(=O)NCC2(C(=O)Nc3ccc(OC(F)F)nc3)CC2)c(C)c1 N1(C(Cn2c(CCC)ncc2)=O)CC2CC1CN2C(=O)C(=O)Nc1ccccc1 c1(OC)cc(C)c(Cl)cc1C(=O)N(CC(C)(C)NC(=O)Cc1ccsc1C)C CC(=NOCC#N)C(=O)NCC(C)C(=O)N(C)Cc1cocn1 C=C1Cn2c(C(N3CCC(CF)(NC(=O)C=CC4CCOCC4)C3)=O)nnc2S1 C(=O)(CC(C(F)F)C(C)(C)C)NC1C(C)(C)CN(C(=O)CCCC2CCC2)CC1 c1(CC(=O)N(C2CCCN(C(CC(C)(O)C3CC3)=O)C2)CCF)ccc(Cl)cc1F c1(NC(N2CCN(C(C(C)C)=O)CC2)=O)ccc(S(C)(=O)=O)cc1C(F)(F)F C1(NC(C2CC(=O)N2)=O)CN(C(c2c[nH]c(-c3ccncc3)n2)=O)CC12CCC2 CCCC(C)CC(=O)NCc1cc(C)c(C(=O)N(CC(CC)OC)C)o1 C1(CNC(C(CC)SC)=O)CC(C)(C)CN1C(=O)CCc1nnc(S)n1C c1(CN(C(C(=O)OC)C)C)ccc(SCc2sc(C3CCCCC3)nc2C)cc1 C#CC1(C(=O)NC2CCC(O)C(O)C2)CCN(C(=O)C(C)n2ccnc2)C1 c1(NC(c2cncc(-c3ccc(OC)cc3F)n2)=O)cc(Cl)c(Br)cc1F Cc1ccc(CN=C(NCC2CCCO2)NC2CC=CCC2)c(Cl)c1 C(CC(C(=O)NCC(O)CN(C)C)NC(=O)CC1CCCCC1)=CC O=C(C1CCCc2scnc21)NC1CN(C(C2CCC3CC23)=O)C1 C(=O)(C(C)(O)CC(F)F)N1CCN(CCN(C)C(C2CCCN2C=O)=O)CC1 C1(CNC(c2ccc(C)c(C)n2)=O)C2CCCC1N(c1ncc(I)cn1)C2 c1(CNC(CCN(CCC)C)=O)cnn(C)c1C(=O)NCCC(C)CO c1(C(=O)NCC2(F)CC(NC(CC(C)OC)=O)C2)cc(SC(F)(F)F)oc1C c1(C(N(C2CN(C(c3ccc(C4CCCO4)[nH]3)=O)C2)C)=O)cc(N)cc(O)n1 c1(NC(C(C(C)C)C)CNC(C2CCOCC2)=O)nc2c(cc1C#N)CCCC2 C1(CNC(c2c(C)nn(C)c2)=O)N(C(=O)CSc2nncn2C2CC2)CCC1(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC(N(C(c2ccc[nH]2)=O)CC)CC1 C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)CCc2cn(C)cn2)C1 S(=O)(=O)(c1cnn(CC(F)(F)F)c1)NC(C(=O)NC)CC(C)C C1(CCNC(C(C)=C(C)C)=O)CCCN(C(=O)CC2COCC2O)CC1 N1(C(CC=C=C)=O)CCN(C(c2ccc(Br)c(C)c2N)=O)C(C)C1C C1(C(=O)NCC2CCN2C(c2cnco2)=O)COCC1C(F)F N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NCC(F)(F)CO)CC1 CC(C)(C)CCCCC(=O)NCCC1(C)CCN(C(=O)COC2CCCC2)CC1 C(=O)(C1CCc2c[nH]nc21)N(C(C)CNC(=O)CNC(c1ccco1)=O)C.CC#N C(=O)(CC(C)(C)CN(C)C)NCC1N(C(C2C(=C)C2)=O)CCC1C C1(C)(C(=O)NC2CN(C(C3(OC)CCCCC3)=O)CC2C)CC(O)CN1C c1(C(=O)NC2CN(C(CC(=O)OC)=O)C2)cn2c(n1)CCCC2 C1(C(N2CC(SC)C(NC(=O)Cc3cncs3)C2)=O)C2CCC3(COC(=O)C13)O2 c1(C(=O)OCC2(c3ccc(OCC)cc3)CC2)nc(F)ccc1Cl C1(C(=O)Nc2cccc(C(c3ccccc3)C#N)c2)CC2C=CC1CCC2 c1(C(=O)NC2CC2(F)F)cnc2c(c1)CCN(S(=O)(=O)c1cccnc1)C2 N1(S(Cc2c(OC)cccc2)(=O)=O)C2CCC1CC(CC(C)O)C2 Cc1cn(C)nc1C(N1CCC1C(=O)NCc1nnc(O)o1)=O C12(C(N3CCC(N(C(C(CC=C)C(C)C)=O)C)C3)=O)C3CCC(CC13)C2(F)F N1(C(c2c(NC(CC)=O)cccc2)=O)CCCC(N=c2[nH]nc(O)s2)CC1 C1(NC(c2cn(CC)nn2)=O)CCCN(C(c2ccnc(C(F)(F)F)c2)=O)C1C Cc1cc(C(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)cs1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)CC2COCCOC2)C(C(F)F)C1 CCC(CC)N(CCC(=O)NC(C1CCCC1)CNC(C)=O)C C12(NC(CNC(=O)OC)=O)CCC1CN(C(C13CCC(OC)C1CC3)=O)C2 Cc1nc(Cl)ccc1CNC(c1csc(C)c1C)c1nnnn1C1CCOCC1 c1(C(N2CCC(C)(C(N3CCC(C#N)C3)=O)C2)=O)cccc2[nH]ccc12 C1(NC(c2cc[n+]([O-])cc2)=O)CCC2(CC1)CN(C(=O)C1CCc3c[nH]nc31)C2 C(=O)(C(CNC(=O)CN=[N+]=[N-])C(C)(C)C)NCC1(C)ON=C(C)C1 c1(C(=O)NC(CNC(C=C(CC)CC)=O)CO)cn2ccc(OC)cc2n1 N1(C(Cn2cc(C(=C)C)c(C(=O)O)n2)=O)CC(C)(C)C(O)C(C)(C)C1 C1(C(=O)NC2(C(=O)NC(CC(=O)OC)C3CC3)CC2C)CCCCCC1 N1(C(c2ccn(C)n2)C(=O)NC2(C)CC2)CC2CC1C(F)(F)C2 N1(C(c2cc(C)oc2C)=O)CC2(CNC(=O)Cc3sc(S)nc3C)CCC1C2 CC(C)CC(C(=O)N1CC(NC(C2CC23CCCCC3)=O)C2(CC2)C1)NC(N)=O c1(NC(c2cncc(Br)c2)c2n(CCCC)nnn2)cc(Cl)cc2c1OCC2 C1(NC(c2cn3c(n2)CCCC3)=O)CC2CCC1CN2C(=O)CC1CC1(Cl)Cl C1(CNC(C2(CC#C)CCCO2)=O)C(C)CCN1C(=O)Cc1ccc(F)cn1 Nc1c(C(=O)NC23CCN(C(=O)CCCF)CC2C3)cc(F)cc1Cl Cc1cnc2[nH]cc(CN3CCC(C(=O)NC(=O)CNC(N)=O)C(F)C3)c2c1 c1(C(=O)NC)ccc2c(c1)CN(C(=O)C(=O)N(C)CC1CC1)C2 N1(C(=O)CCCC(F)(F)F)CCC2(COCCN2C(c2cc[nH]n2)=O)C1 c1(CC)c(C(N2CCOC(CCNC(c3[nH]cnc3C#N)=O)C2)=O)cnn1CC c1(CC(=O)NC23C(CN(C(c4cnc(SC)s4)=O)C2)C3)cn2c(C)csc2n1 c1(C(=O)NCCc2c(C(N(CCC3CC3)CC)=O)c[nH]n2)[nH]ccc(=O)c1C Cc1ccc(C(N2CC(C)(NC(c3ccc(Cl)c(C)c3Cl)=O)C2)=O)c(F)c1F CC1(C)CCC(C(N2CC(NC(=O)Cc3ccc(Br)cc3)C(O)C2)=O)CO1 c1(C(CO)NC(c2ncc(-c3ccccc3)o2)=O)ccc(OC(F)(F)F)cc1 C1(CC(=O)N(C2(C(=O)NC3CCC4(CC4)C3)CC2)C)CC2CCC1O2 C1(NC(=O)NCCc2ncc(CC)s2)CCN(c2cc(C)nn2C)C1=O N1(C(c2c(C)[nH]cc2)=O)CC(N(C)C(c2ccc(-c3ccco3)s2)=O)C2(CC2)C1 c1(C2C(C(N(CCNC(CCC=CC)=O)C)=O)C2)ccccc1Br O(NC(=O)C(CC1CC1)NC(C1CC(=O)NC(C)C1)=O)CC(=C)C N1(C(c2cc(C)nn2C)=O)CCN(C(=O)C(c2ccc(=O)n(C)c2)(C)C)C2CC12 S(=O)(=O)(c1ccc(F)c(C(N2CCC(CNC(C)=O)(OC)CC2)=O)c1F)NC C(C)(CC#CC)NC(CCN(CC=C)C(C1CCNC1=O)=O)=O c1(NC(C2(O)CN(C(Cc3cn(CC)nc3)=O)C2)C)ncc(C)c(SC)n1 c1(NC(CCC(CC)NC(C2(C#C)CC(=O)C2)=O)=O)ccc2c(c1)OCC2 c1(C(N(C2CN(C(CCCN(CC)CC)=O)C2)C)=O)ccc(CC2CCC2)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C(C(C)CC)N(C)C(C1CCCC(CF)C1)=O)NCCCCCC#C c1(C(=O)NC(CN(C(CCOCC#C)=O)C)(C)C)cc2c(CC)cccc2[nH]1 C1(NC(c2cccc(OC)c2)=O)CC(F)CN(C(C2CC(O)C2)=O)C1 C(CC(F)F)(C(=O)NC(c1nn[nH]n1)C1CC1)N(C(C1C(=C)C1)=O)C CC1(CNC(=O)C2CC2)CC(F)(F)CN1C(=O)C(=O)Nc1ccc(Cl)cc1 C(=O)(C1=NOC(c2ccccc2)C1)NCC(C)NC(C=C(CC)C)=O N1(C(C2N(C(=O)CCN3CCCCC3)CCN(C)C2)=O)CC2(CNC(=O)OC2)C1 Cc1cc(NC(C23CCC2C3)=O)ccc1NC(c1cc2n(n1)CCC2)=O C1(CCC)C(=O)NCCN1C(C1(NC(=O)CC(C)(C)CC)CC1)=O c1(C(N2CC(C(=O)NCc3cc(Cl)ccc3Cl)OCC2)=O)c(F)ccc(Cl)c1Cl C1(C(=O)NCCCCCCNC(c2c(C)cccc2F)=O)CC2COCCN2C1 C1(CCC(C)(C)NC(=O)C(F)F)CCCCN1C(=O)C=CC1CCCC1 c1(OC)ccc2occ(C(=O)NCC3(C)CCN(C(=O)CCNC(C)=O)C3)c2c1 N1(C(c2ccc(=NC)[nH]c2)=O)CCC=C(C(=O)N2CCC(OC)CC2)C1 c1(OCCC(=O)NCCCNC(c2c(N)nccn2)=O)ccc(F)cc1Cl N1(C(c2ccc(=N)[nH]c2)=O)CCCC2(CCCCC2NC(c2ccc(Cl)o2)=O)C1 Cc1cc(N(C(C)(C)CNC(c2nnn(C(C)(C)C)n2)=O)C)nc(CO)n1 C12(C(=O)NCC3N(C(COCC(=O)NC)=O)CC3)CCCCC(=O)N1CCC2 C1(C(=O)NCCCC)CC12CN(Cc1ccc(C(=O)OC)nc1)C2 C=C(C)CC(C)C(=O)N1CCC(O)(CCNC(=O)C(F)=C2CCCC2)C1 C=C(C)CCCC(=O)NCC1CN(C(c2sccc2C)=O)C2CC12 N1(C(C(CCC)O)=O)CC(O)(C2CCN(C(=O)CSc3nc[nH]n3)CC2)C1 N1(C(CC(C)SC)=O)CC2(C=C(C(=O)N3CC4(CC(F)C4)C3)CO2)C1 C(C(=O)NCCC(C)NC(c1ccnc(N2CCCC2)n1)=O)(C(C)C)OC C1(C(N2CC(N(C(=O)CCC3OCCO3)C)C2)=O)CS(=O)(=O)CC(=O)N1 C1(C(N2C(C)(COC)CCC2)=O)CC(NC(C2CC(O)C2)=O)C12CCC2 CC(C)(O)C#CC(=O)NC1(C(N2CC(N3CCCC3=O)C2)=O)CCCC1 Cc1nc(NC(C2C3CC2N(C(c2nc(C)c(Br)s2)=O)C3)=O)ccc1Br CC1CCN(C(=O)CN(C)C(c2cncn(C)c2=O)=O)C(C)C1 C1(CNC(COCc2cc(C)on2)=O)C(C)CCN1C(c1ccc(C#N)s1)=O C(CC)(CCC(=O)N1CCCC1C1CCOC1)NC(C(CC)=CCCC)=O c1(NC(N2CC(CCl)C2)=O)ccc(CCN(CCO)CS(=O)(=O)Cc2ccc(F)cc2)cc1 C1(C(=O)NC(C2CCCCC2)C(=O)NCC2(SC)CCC2)CC(O)C(F)C1 C1(C2(O)CCC2)(C(=O)NCC(C)(O)CNC(c2cc(C3CCC3)no2)=O)CC1 N1(C(C23CC(CN(C(C(C(C)C)SC)=O)C2)C3)=O)CCC2(CCCN2C(C)=O)C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CN(C(c2cc3c(s2)CCC3)=O)C(C)(C)C1 N1(C(CC2C(C)CCCC2)=O)CCC(C=CC(=O)NC2CN3CCC2CC3)CC1 CC1(C)CCn2cc(C(=O)NC3CN(C(C45CC(F)(C4)C5)=O)CCC3F)nc2C1 c1(C(=O)NC(C2CCN(C(=O)CCOCC(F)(F)F)C2)C)ccn(C)c(=O)c1 N1(C(C(CCCCC)O)=O)CCC2(C)CN(C(c3cc(N)ccc3C)=O)CC12 c1(NC(C2CCC(C)N2C(C2CC2C2CC2)=O)=O)cc(Cl)nc(Cl)c1 C1(C(=O)NC2CC(CNC(CSCC(N)=O)=O)C2)C2COCC12 c1(C(=O)NCC2(OCC)CN(C(=O)CCc3cnco3)C2)ccc(C)nc1 C1(NC(=O)C(F)F)C=CC(C(N2CCC(C(F)(F)F)C2)=O)C1 c1(NC(=O)CC2CN(C(C3CC3F)=O)C2)cccnc1I N1(CC)OCC(NC(=O)C(c2cn(C)nn2)NC(=O)CC(C)COC)C1=O Cc1cnncc1C(N1CC=CC1C(=O)NCC(C)(C)N(C)C)=O C1(CNC(C(C#C)(C)C)=O)COCCN(C(c2cccnc2OCC)=O)C1 CC1(C)CC(c2ccccc2)N(C(=O)C(c2cc(F)cc(F)c2)F)C1 c1(CN2CC(CNC(c3ncn(C)c3)=O)C2)nccc(OCC(F)(F)F)n1 C1(NC(C2(CC)CCCC2O)=O)CCN(C(=O)CCN2CCOCC2)CC1OC c1(C(=O)NC(C)CN(C(=O)Cc2ccc(Cl)cc2)C)ccc(Cl)nc1N CC(C(C)(C)C)=CC(=O)N(CCC(=O)NCC(CC1CC1)CO)C1CC1 [N-]=[N+]=NC1CCC(C(N2CCCCC2C(=O)NCc2cc(O)ccc2F)=O)C1 C1(NC(C2CCC(C)O2)=O)CC2CCC(C1F)N2C(C1COCCOC1)=O C1(CC=C)(NC(=O)CC(C)C2CC2)CCN(C(C2(C)CC(C)(C)C2)=O)C1 N1(C(CNC(=O)OC(C)(C)C)=O)CCC(NC(=O)C#CC2CC2)C1C1CC1 N1(C(CCNC(COC)=O)=O)CCC2CCCC(C1)N2C(=O)CCC(F)(F)F C1(C(N(C(CNC(c2scc(C)c2)=O)C2CC2)C)=O)CC(C)CC(=O)N1 c1(CC)[nH]nc(C(=O)NCCCCN(C(=O)CC2C(C)(C)C2(C)C)C)c1Br N1(C(C2C(C)C2)=O)CC2OCC(NC(c3ccsc3S(N)(=O)=O)=O)C2C1 N1(C(C=CC)=O)CCN(C)CC1CNC(c1cncc(C#N)c1)=O C1(N(C)C)CCCN(CCC(=O)N(CCNC(=O)Cc2cncn2C)C2CC2)C1 CC(C)CC(C(=O)NC1CC2CC(C1)N(C(c1cccc(Cl)c1F)=O)C2)C(N)=O N1(C(CCNC(c2nc3c(s2)CCCC3)=O)=O)CCC(C2(O)CC2)C1 C1(C(N2CCC(C)(CCO)C2)=O)(NC(C(C)OCC=C)=O)CCC(C)(C)C1 C(=O)(CCCCCN(C)C)NCCC(C)NC(c1n[nH]c(=N)[nH]1)=O CCN=c1nc(C(N2CCCC2CN(C(=O)CC(C)F)C)=O)cc(C)[nH]1 C1(CCC)CN(C(=O)COCC2CCCCC2)CC1C(=O)NCc1ccnn1C c1(C(N2CCC(C)(NC(CCOCC#C)=O)C2)=O)cc2c(s1)CCC(C)C2 CCCCCCCCC(C)C(=O)NCC1CC(NC(=O)C(O)CCn2cncn2)C1 c1(CCC(=O)NC(C(C)NC(=O)CSc2ccccn2)(C)C)cc(F)ccc1F C1(C(=O)NC(C)C(C)NC(c2cncc(N)c2)=O)(OC)CCCCCCC1 C1(CNC(c2ccc(CC)nc2)=O)COC(C)(C)CN1C(=O)C=C(C)C(C)(C)C c1(OC)ccc(Br)nc1NC(c1nc(-c2cnn(CCF)c2)cs1)=O C1(n2cc(CS(=O)(=O)CCNC(=O)C=CCO)nn2)(C(=O)OC)CCOCC1 CC(C)CS(=O)(=O)CCC(=O)N1CCC1CNC(=O)Cc1cccc(F)c1O C1(C(C)C)CN(C(=O)C(C)C2(O)CCC2)CCN1C(C1CC1C(F)(F)F)=O C(=O)(C(S(C)(=O)=O)C1CC1)NC1C(C)CN(C(c2csc(C(C)(C)C)n2)=O)C1 c1(NC(C2OCCN(Cc3ccc(C)cc3F)C2)=O)cccc2nc(O)oc12 S(=O)(=O)(c1cc2cncc(Br)c2s1)NC(Cn1c(=O)cc(C)nc1C)=O N1(C(C(CCC)(C)C)=O)CCC(NC(C2(C)CCCS2(=O)=O)=O)CC(O)C1 c1(C(=O)NCCCCNC(C(c2ccc(F)cc2)C)=O)cc(S(C)(=O)=O)cs1 N1(C(c2ccc(N(CCC)CC)cc2)=O)CC(NC(=O)CC(C)COC)C(C)(C)C1 c1(OCC(=O)O)ccc(CCNC2CCC(C(=O)Nc3ccc(Cl)cn3)C2)cc1 c1(OC)c(C)ccc(C(=O)NC(C)CCNC(=O)C(C(C)C)N(C)C)c1F c1(OC)ccc(-c2nc(CCN3CCCCC3)nn2CC(C)C)nc1OC N1(C(C2CC2CCC)=O)CCN(C(=O)COCc2ccccc2)C2(CC2)C1 c1(C(=O)NCC(C)(CO)NC(C(CSC)C)=O)ncnc2cc[nH]c12 c1(C(N2CC(O)CC(NC(CN(CC)CC)=O)C2)=O)ccc(OC)c(OC)c1Cl c1(C(=O)NC2CN(C(CC=C)=O)CC2F)cc(OC)c(OCC)c(Br)c1 c1(C(=O)NCC(C)NC(c2ncc(Cl)n2C)=O)c(C#N)cnn1C C1(NC(C2CC(F)(F)C2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cn1)(F)F)C2 c1(C(N(CCNC(c2nc(OC)ccc2OC)=O)CC)=O)c(C)cc(C)cc1N C1(C(c2ccccc2)N(C2CC(OC)C2)C)CCCC(C)(C)C1 C1(NC(C(CNC(C2(CC(C)C)CC2)=O)O)=O)CCN2CCC1C2 c1(C(C)=O)cc(F)ccc1C(=O)O.c1(CNCC)nccn1C1CC1 C(C)(C)(CC(=O)NCCCC1(NC(C2CC(C)OC2=O)=O)CC1)SC c1(CC(=O)N(CC(CNC(C(C)=C(CC)C)=O)O)C)ccc2nn[nH]c2c1 c1(C(N(CCC)CCNC(=O)C(C)Cn2ccc(C)n2)=O)ccc(O)c(Cl)c1 c12cc(on1)C2.C1(Cn2ccnc2)CCN(C2CC2)C1 CC1CN(C(c2cc(O)cc(O)n2)=O)CCC1NC(c1ccc(C(N)=O)nc1)=O c1(N(C)CC2CCN(C(C(C(C)O)(F)F)=O)C2)nc(Cl)nc2c1COCC2 C1(CNC(=O)CC(F)(F)F)CN(C(=O)COC2CCCOC2)CCCO1 Cc1cc(O)cc(=O)n1C(C)C(=O)NCCC1CN(C(C2(CF)CC2)=O)CCO1 C(=O)(CCCCN1CCOCC1)NC(CC(C)NC(C1C2CCC(=O)C12)=O)C c1(OCC)ncccc1CC(=O)NCCNC(C1CC(=O)N(CC(F)(F)F)C1)=O C=C(C)C(C)(C)C(=O)NCC(C)CN(C)C(C1CCNC1=O)=O Cc1ccc(C2OCCCC2NCC(=O)OCCCCCc2ccccc2)cc1 c1(C(=O)NCC2CCCN(C(c3cc(C)ncn3)=O)C2)cc2ccccc2o1 N1(C(c2c(C)coc2)=O)CC2CCN(C(C3CCC(=O)N3)=O)CCC2C1 c1(C(=O)NCC2C(NC(c3nc(C)[nH]n3)=O)CCC2)nn(C)c2ccc(F)cc12 CCC(CC)CC(=O)NCc1nc(CNC(=O)Cc2ccc(O)c(C)c2)cs1 CCCC(C)(C)CC(=O)NCC(CC(F)(F)F)NC(c1[nH]c(C2CC2)nc1C)=O C=CC1OCCC1N=c1nc2c(ncn2C)c(N2CCN(CCOC)CC2)[nH]1 C1(CNC(C2(OCC)CCOC2)=O)CC2CCC1N2C(c1cnc(C(C)C)o1)=O CC(C)C(CCN(C)C(c1occc1C1CC1)=O)NC(=O)C=C1CC1 C1(CC(=O)NCC(C2CCC2)NC(=O)CCC2CCC2)CCCO1 C(=O)(CC(C(F)F)C(C)(C)C)NC1CC2CN(c3snc(C)c3C#N)CC21 C1(CNC(COCCC=C)=O)CN(C(C2C3CC4C(C3=O)C24)=O)C2CCCCC12 C1(C(=O)NC(C(C)C)C(C)C)CN(C(c2cccc(CO)c2)=O)CCN1C N1(C(C(c2cncnc2)C)=O)CCC2CC12C(=O)NCCC(C)C(F)F C(C)(CCC(=O)NC1CCS(=O)(=O)C1)NC(C=C(CCC)C)=O N1(C(C(C)(O)C2CCC2)=O)CCCCC(CNC(c2ncsc2Br)=O)C1 C12(C(=O)NCc3c(C(=O)NC(CCC(=C)C)C)nco3)CCCC1CCC2 CC(CC(=O)NCC1(C)CCN(c2nnn(C)n2)C1)CC(C)(C)C C=CCC(C)(C)NC(=O)C(C1CN(C(=O)C(C2CCCC2)OC)C1)OC Cc1nonc1CC(=O)NCc1cn(CCNC(=O)CN2CCCC2C)nn1 C=CCC(C)C(=O)NCc1cc(C(N2CCC(NC(C)=O)C2)=O)n(C)n1 C1(CC#C)(C(=O)OCCC(CO)NC(=O)NC(C)(C)C)CCOC1 N1(Cc2ccc(CC(=O)OC)[nH]2)CCNC(=O)C1C C1(NC(Cc2c(C)oc(C(F)(F)F)n2)=O)CC2(C1)CC(NC(C1(C)CSC1)=O)C2 C#CC1(C(N2CCC(c3nc[nH]n3)C2)=O)CCN(C(c2cnc(OC)nc2)=O)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCCn2ccnc2)CCCC(F)(F)C1 c1(C(N2CC(NC(C(C)O)=O)C(c3ccccc3F)C2)=O)nc2c(s1)CCC2 c1(NC(C2N(Cc3c(C)noc3C)CCC2)=O)ncc(Br)nc1CO CC(C(C)(C)CN(C)C)NC(C1(CNC(c2cccnc2O)=O)CC1)=O N1(C(C2(C(C)C)COC2)=O)CCCCCC(N=c2[nH]n(C)cc2[N+](=O)[O-])C1 c1(C(=O)NC(C)CNC(=O)CCNC(c2ccco2)=O)cccc(Br)c1O c1(C(=O)NC(CC)CC)conc1C(C)NC(=O)COc1ccsc1 c1(CC)ccc(C(N2CC(CNC(C3CCC3)=O)C(c3ccccc3)C2)=O)cc1 Cc1c(C(N2CCCC2C(N2CCSCC2)=O)=O)cccc1O CC(CC(N)=O)C(=O)N(C)CC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(NC(C2(C)CCN(C(c3ncn4ccccc34)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C=C(C)C(C)C)=O)CC=CCC1C(=O)NC(CO)C(C)(C)C C12(C(N3CC4(N(C(c5cc(C)on5)=O)CC4)C3)=O)CCCCC1OCC2 c1(OC)ccc(Cl)cc1CC(N1CC2CC(NC(C3CC(O)C3)=O)C1C2)=O c1(CN2CCC(N(CC(=O)N(C)C(c3ccccc3)=O)C)C2)ccc(Cl)s1 C(CCS(C)(=O)=O)(C(=O)OC(C)C)c1c(-n2cc(CCC(CC)O)nn2)ccs1 n1(CC(N2CC(C(C)NC(c3cn(C4COC4)nn3)=O)C2)=O)cccnc1=O C(c1cccc([N+](=O)[O-])c1)=CC(=O)N(C)CC1CN(C(C(F)OC)=O)CC12CC2 CC1(C)CC(CO)CN(C(=O)C(C2(C)CC2)NC(c2ccc(C#N)cn2)=O)C1 C1(C(N(C(c2cnnn2C)C)C)=O)C(O)CCN1C(C1CCCSC1C)=O C1(COCC(=O)N(C2CC(NC(C3CCC(O)C3)=O)C2)C)CCOCC1 Cc1cc(Cl)c(C(=O)NCC(C)CNC(=O)CN(C)Cc2ccccc2)cc1N c1(OC)c(CN2CCC(C(=O)Nc3nccs3)C(O)C2)ccc(Br)c1F c1(C(N(CC(C)N(C(CCOCC)=O)C)C)=O)cn(C(F)F)cn1 c1(OC)ccc(C2(CC(=O)OC)CC2)cc1NC(=O)CNC(=O)OCN N1(C(c2cc(CCNC(CCN(C)CC)=O)on2)=O)CC2CCCC2(CSC)C1 C(CNC(=O)C(F)(F)CO)(N=c1nc(C2CC2)[nH]s1)c1cccc(N(C)C)c1 C(=O)(C(C(C)C)c1ccc(F)cc1)Nc1c(C(=O)NC)ccs1 CCCC(C(=O)NCC12CC1CN(C(=O)C(=Cc1cccnc1)F)C2)OCC c1(COC)cccnc1C(=O)NC(CNC(C1(C)CCCC1O)=O)CC(C)C N1(C(c2ccc(=N)[nH]c2)=O)CC2(NC(c3cc(-c4ccns4)on3)=O)CCC1C2 n1(CC(=O)NC2C(CC)CN(C(=O)Cc3cncs3)CC2)cc2ccccc2n1 C1(CC)CN(C(c2coc(C(F)F)n2)=O)CCC1NC(c1nc(=O)n(C)[nH]1)=O C1(C)(C(N2CCC(OC)(CNC(=O)C(C)NC(N)=O)C2)=O)CCC(=O)NC1 C1(CNC(c2c(C)c(N)ccc2)=O)(NC(=O)C=C2CCC2)CCC(F)(F)CC1 C(=O)(CCCCCNCC(=O)OC(C)C)OCC CC(C#N)CCC(=O)NC1(C)CN(C(=O)CCc2ccc(Cl)c(F)c2)C1 C1(NC(C2CN(CC)C2)=O)CCCC(C(=O)NCC2(C(=O)OC)CCCC2)C1 c1(C(N2CCc3ccc(Br)cc3C2)C(=O)NC)ccc2c(c1)OCC(=O)N2 C(=O)(C(CC1CC1)NC1CC(C)(C)C1)N(C(C)C(=O)NC)CC Cc1cc(N)c(C(N2CC(C3(NC(=O)C(C)OCCN(C)C)CC3)C2)=O)nc1C Cc1nc(NC(C2CCCN(Cc3ccccn3)C2)=O)nc2ccccc12 c1(C(N2C(C(=O)Nc3c(C(C)C)ccnc3)CC(F)C2)=O)csc2ccccc12 N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)C(C)(C)SC)CC1C(C)C C(=O)(C1=CCCC1)N(C1CN(C(=O)CCc2cccnc2)CC1F)C CCC(CC)CCC(=O)NCCOC1CCN(C(c2cnccc2Cl)=O)C1 CC1Cc2c[nH]nc2C(C(=O)NC2(CCNC(c3c(Cl)nn(C)c3Cl)=O)CC2)C1 c1(C(=O)NCC2C(NC(=O)CCc3ccccn3)CCC2)cn2c(n1)SCC2 C1(C(=O)NCC2OCCCN(C(c3nc(C)n(C)n3)=O)C2)CCC(N=[N+]=[N-])CC1 C1(NC(C2(CC)CCN(C(c3cncc(C#C)c3)=O)C2)=O)CC1C1CCCCC1 C1(NC(Cc2c(C)nn(C)c2)=O)CCN(C(=O)Cc2ccno2)C12CC2 c1(C(N(C2CCN(C(=O)CO)CC2)CCOC)=O)ccc2cc(C)ccc2n1 n1(CC)c(CNC(=O)C(CNC(=O)CCC2(C)CCC(=O)N2)N(C)C)cnc1C c1(CNC(c2c(C)[nH]nc2C(F)(F)Cl)=O)cccc(Cl)c1O c1(OC)cc(CN2CC3CCN(C(=O)C(C)S)C3C2)cc(F)c1OC C1(CC)CN(C(C2CC2C(F)(F)F)=O)CCN1C(=O)C1=CC(C)(C)C1 CC1(NC(=O)NC(CCCC2CC2)c2nc(-c3nc[nH]n3)no2)CCCC(=O)N1 C=CCC(C(=O)NC1CN(C(=O)CC23CCC(CC2)OC3)C(C)(C)C1)C(C)C C=Cc1cnn(C)c1C(=O)NCC1CCC(C)CN1C(=O)CC1CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCC2C(NC(=O)C(C)COC)C2C1 C(CCNC(=O)OC(C)C)(C(C)C)Oc1ccc(COCC)cc1 CC(C)CC(F)C(=O)N1CCCCC1C1CCN(C(c2ccc(O)nn2)=O)CC1 C1(C(N2CCC(CNC(c3cc(SC)oc3)=O)C2)=O)CCc2ncnn2C1 C1(N(C(C2C(C(C)C)CCO2)=O)C)CCN(C(C23CC(C2)C(C)O3)=O)CC1 CCC(COC(C12C(NC(=O)OC(C)(C)C)C3CC1C2C3)=O)(CC)C(N)=O C1(NC(c2cnco2)=O)CN(C(C23CCCC2C3(F)F)=O)C2CCCC12 C(=O)(CC(C)P(C)(C)=O)NCCCN(C(C1ON=C(CC)C1)=O)CCO C1(NC(COCCNC(Cc2cc(C)sc2)=O)=O)CC2C=CC1C2 C1(CC(=O)NCCN2CCNC2=O)COCCN1C(c1cc(=O)cco1)=O Cc1ncsc1C(=O)NCCC(C)NC(c1ncoc1-c1cccs1)=O Cc1cn2cc(C(=O)N(CC(C)(C)CNC(=O)Cn3ncnn3)C)nc2s1 C1(NC(CCCOCC)=O)COC2CN(C(=O)Cc3ccc(C)nc3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(O)CC(C)C)C)cc2c(s1)CCCCC2 Cc1c(F)c(CN2CC3OCCC3(C(=O)O)C2)cc(Br)c1F C#CC1CC2CCC1N(C(c1cnn(CCNC(C3CCCOC3)=O)c1)=O)C2 C1(OC)CC(NC(=O)CCC(=O)N(C)C)CN(C(c2cn(CCF)nn2)=O)C1 N1(C(c2cn(C)nc2)=O)CC2CC1CC2NC(c1cccn(C2CCC2)c1=O)=O CC(C)(C)C(C(=O)N1CCC12CN(C(=O)CC1NC(=O)NC1=O)C2)n1ccnn1 Fc1ccccc1C(C(F)(F)F)Nc1ccc(OC2CCCCC2)cn1 N1(C(C)=O)CC2CC1CN2C(=O)C(C(C)O)NC(=O)CC(C)C(F)F C(=O)(CCCCC(N)=O)NCC(CCOC)NC(C1(c2ccccc2F)CC1)=O c1(C(=O)NC(C2(O)CCN(C(C3(CC4CCC4)CC3)=O)C2)C)cc2ccsc2s1 N1(CCC(N2CCC(N(C(=O)CCc3ccc(C)s3)CC)C2)=O)CCOCC1=O C1(c2ccccc2)(NC(C2CC2(Cl)Cl)=O)CCN(C(c2ccc(O)nc2)=O)CC1 C12(NC(CCCCCN(C(C(C(C)(C)C)OC)=O)C)=O)CCC(CC1)C2(C)C N1(Cc2onc(CC)n2)CCC(NC(C2C(C)OC(C)C2C)=O)CC1C C(=O)(CCC(F)(F)F)NC(CC)COC.C1(=O)C(N(C)C)CCN1C N1(C(c2ccn(CC)n2)=O)CC2CCC(C1CO)N2CC.C12(CC)CCN1C2=O C1(CCC)CC(C(=O)NCC2C3CN(Cc4ccc(F)cc4)CC23)CCO1 C1(CNC(c2n(CCOC)ncc2)=O)C2CC2CN1C(c1cc(C)nn1C)=O C1(NC(CCC(=O)NCCC2CC2)=O)CCN(C(=O)CC(F)(F)F)CCC1(F)F Cc1ccc(F)c(C(=O)NCC2CC2C(=O)NCc2nn[nH]n2)n1 c1(SCC(c2cc(C)n(C3CCS(=O)(=O)C3)c2C)=O)cc2ccccc2n1C C(C(CC(C)C)C(=O)NCC1CCCCC1(C)C)NC(c1c(NC)cncc1)=O c1(C(=O)OCC)noc2c1CN(C(=O)NC1CC(=O)N(C3CCOCC3)C1)CC2 N(C1CS(=O)(=O)Cc2ccccc21)C(c1c2nc(C)sc2ccc1)C1CC1 Cc1nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(=O)C(N1C(=O)CCC1=O)C N1(C(c2nc(CC)oc2)=O)CC(N(C)C(c2cc(Br)c(C)s2)=O)C(F)C1 N1(C(c2cc(Cl)ncn2)=O)CCC2(CCC(C(N3CCC3)=O)C2)CC1 N1(C(CCC=C)=O)CCCC1(CNC(=O)COC1CCCOC1)COC O=C(CC(C(F)F)NC(c1ccccc1F)=O)NCCCC1CCCCO1 Fc1ccc(CNC(=NCCN2CCCC2)NCC2CCC23CCC3)c(F)c1 C(C)(C)(C(=O)NC1CCN(C(C2CC2C(C)C)=O)C1)NC(=O)OC N1(C(c2nc(C)c(C)n2C)C(=O)NCCCOC)C2CCC1CC(CCO)C2 N#Cc1nccc2cc(NC(c3ccc(Cl)c(C(F)(F)F)c3)C(N)=O)ccc12 C(=O)(C1=CCC(NC(=O)CC2CCCOC2)C1)NCCOCC CCCCC(=O)C(=O)NCC1CC1CC(=O)N(CC)Cc1nncn1C C(=O)(CCCC(C)(C)C)N(CC(C)(C)C(=O)NCCC1CCCC1O)C C=CCC(CC(C)C)C(=O)N1CCC(CNC(=O)C(CC)(CC)CC)C12CC2 N1(C(Cn2cnc(C#N)n2)=O)CCOC2(CCN(C(c3csnc3Cl)=O)CC2)C1 c1(OC)cccc(Br)c1C(N1CCN(C(=O)Cc2ccon2)C(CO)C1)=O n1(CC(=O)N(CC(O)CN(C)C(c2csnn2)=O)C)ccc(Br)cc1=O C(C(C)(O)C(=O)NC1C=CC(CC(N2CCC(C)(O)C2)=O)C1)OC C1(CCC(=O)NCCCCC#C)CCCCN(C(=O)C(CC(C)C)N(C)C)C1 C1(C(=O)NCc2cccc(C(NOCC=CC)=O)n2)CC2C(C1)C2(C)C N1(C(CCOCC#C)=O)CCC(=CCNC(=O)C(F)=CCC)CC1 CCCCC(C(=O)NCC1(NC(=O)C(F)(F)CCn2cccn2)CCC1)N(C)C C1(C)(C(N2CC(NC(CC3C=NN(C)C3=O)=O)C3(C2)CC3)=O)CCS(=O)(=O)CC1 C1(CNC(c2ncc(CC)s2)=O)CCN(C(=O)CC2=CCCCC2)C12CCC2 C1(CCNC(=NCCC=C)NCC2(OC)CCCC2)CCc2ccccc2C1 C1(NC(CNC(=O)OC)=O)CCCCC1N=c1[nH]ccnc1F C(=O)(C1CCCc2scnc21)NCC1CN(C(c2nc(OC)c(F)cn2)=O)C1 N1(C(C(CC)F)=O)CCC2(CC1)CC2CNC(=O)CSCc1ccccc1 C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cn2ccnn2)CC(C)(C)CCO1 C1(C(=O)NCC2C(C)CN(C(C3(C)CC4CCC3C4)=O)C2)Cc2ccccc2C1 c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)cccc(Br)c1Cl C1(CC=C)(NC(=O)CCOCC)CCCN(C(C2(C(=O)N(C)C)CC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1CCCC(C)(C(=O)NCCC2CC(F)(F)C2)C1 N1(C(C=C(C)C)=O)CC(F)(F)CC1C(=O)NCC(O)C1(Cl)CC1 N1(C(C2CCCC(NC(c3ccc(Cl)o3)=O)C2)=O)CC2C3CCC(C3)C2C1 C(C(C)(O)CNC(CN)=O)N(C(=O)NC)C1CC1.c1(C2(C)C(C(=O)N)C2)ccccc1 C(=O)(C(CNC(C1COCCC1C)=O)C(C)(C)C)NCc1cncc(CC)c1 c1(C(N2CC(C(=O)NC(CCOC)(C)C)C(O)CC2)=O)cnn2cccnc12 c1(C(C)=O)cc(C(=O)N(CC(C)NC(c2ccc(C(F)(F)F)o2)=O)C)oc1C Cc1cc(C(N2CCCC2(C)CNC(=O)Cn2ncnn2)=O)cc2ccoc12 C1(NC(c2ncc(CC)cn2)=O)CC1C1CCN(C(=O)CC(C)(C)C)CC1 O=C(C1=C(Cl)CCC1)NCCOC1CCN(C(C2CC2c2ccncc2)=O)CC1 N1(C(CC2(C)CCC2)=O)CCN(C(=O)CCC2CC2)C(CC(F)F)C1 c1(C(=O)NCC(CCNC(C=CCCC)=O)O)cc(CCC)c(C)s1 CC(N=[N+]=[N-])C(=O)N(C)CC1CCCCN1C(=O)CCCC1CC1 CCC(O)C(C)C(=O)NC1(COC)CN(C(=O)C2=CCCS2)C1 C1(NC(C(F)=CCC)=O)CC(OC)CN(C(=O)C(=O)NCCCCCCCC)C1 Cc1cc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC(OC(F)F)C2)nn1C N1(CCCC(=O)NC(CNC(C2C(CC)C2)=O)(CC)CC)CCc2ccccc21 C1(C(N2C(CCC)COCC2)=O)CCC(C)(C)N(C(C2(C)C=CCCC2)=O)C1 C1(O)(CCc2ccc(NC(C(C)OCC=C)=O)cc2)CCN(C(=O)COCC)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCN(C(=O)CCc2ncc(F)cn2)CC1F c1(OC)cc2ccccc2cc1C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1 O=C(C1COc2ccccc21)NC1CN(C(c2cc3c(s2)CCCC3)=O)CC1F C(=O)(C(C)C(C)NC(c1oc(CNC(C2CC(=O)C2)=O)nc1C)=O)OC Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)CS(C)(=O)=O)C12CCC2 C(c1ccc(Cl)s1)=C(C#N)C(=O)NCCOCCS c1(CNC(C2CCS(=O)CC2)c2n(C3(C)CC3)nnn2)ccnc(F)c1F C1(NC(C(C)c2cccs2)=O)Cc2ccccc2C1NC(=O)CCc1nc[nH]n1 c1(C(C(=O)N(CC(C)NC(C2COC2)=O)C)C)ccc(Cl)cc1 C1(CNC(c2cnc3nccn3c2)=O)CN(C(c2ccco2)=O)C2COCC2O1 C(CC(=O)N1CC(OC(=N)O)C1)N(C(=O)C(C)C1CCC1)CC=C N1(C(c2n(C)c(Br)nc2)=O)CCCC(CC(N2CCCC(C)(C(=O)O)C2)=O)CC1 C1(NC(C2C3CC4C(C3)C24)=O)CC2CC(C1)N(C(c1ccn3nncc3c1)=O)C2 c1(OC)cc(F)c(F)cc1NC(=O)CCCN(C)C(c1cnc(O)n1CC)=O N1(C(C2=C(C)CCC2)=O)CC2CC(NC(=O)COc3cc(Cl)ccc3Cl)CC1C2 C1(NC(CN2CC(C)C2)=O)CC(C)CN(C(C2(F)C(C)(C)C2(C)C)=O)C1 C(=O)(C(F)CCC(C)(C)C)NC1(C(=O)NCC(c2n(C)ncc2)O)CC(F)C1 C(CO)(C(C)(C)CO)NC(C1(C(C)NC(=O)CC2CNC(=O)O2)CC1)=O c1(C(N)=O)cc([N+](=O)[O-])cnc1N1CCCCC(NC(=O)C(C)n2ccnc2)C1 C1(NC(CCN(C)CCO)=O)COC2(C1)CN(C(c1ccns1)=O)C2 C=CC1(C(=O)NC2CC(NC(C3(C)CC4CC4C3)=O)C(O)C2)CCOCC1 CCC(C(=O)N1CC(CNC(=O)CN2CCCC2=O)C2(CC2)C1)C(F)(F)F C=CC(C)(CCOC)C(=O)NCC1(F)CCN(C(c2cn3ccnc3s2)=O)C1 C1(CN(C)C)CCC(C(N2CCC(CNC(=O)Cc3coc(C(F)F)n3)C2)=O)O1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2COCCOC2)=O)C12CC2)=O C1(C(c2cccc(CC)c2)N2CCC(OCC)C2)(NC(C)(C)C)CCOCC1 CCCC(O)C(=O)NCC1(C(=O)NCCSCC(C)C)CC=CC1 C(=O)(N=c1ccn(-c2ccc(F)cn2)[nH]1)C1CC2(CC(NC(=O)OC)C2)C1 c1(C(N2CC(C(C(=O)NCC3CCC3CO)OC)C2)=O)csc(Cl)n1 N1(C(c2c(C(C)C)ncs2)=O)CCC(CNC(C2(O)COC2)=O)C(C)C1 C1(=O)C(C)CCN1.C1C(O)CN1C(CN(C)CC)=O.C(C)(C)(C)OC(=O)N.CC C1(CNC(=O)CSc2nc[nH]n2)CCCCN1C(=O)Cc1ccco1 N1(C(C(C=CC)O)=O)CC(O)CC1(C)C(=O)NOCc1ccccc1 Cc1cc(N(C)C)ccc1C(=O)NC12CCC(C1)N(C(c1cc(F)n[nH]1)=O)C2 CC1(C)OC(=O)NC1NC(=O)C(=O)NC1CN(C(C2(OC(F)F)CCC2)=O)C1 C(CCC(C)CC(=O)N(CC(O)CNC(c1cnc[nH]c1=N)=O)C)=C(C)C c1(CNC(C(CC)C#N)=O)ccc2c(c1)CCC2NC(c1ccccc1OC)=O CC1OC2CCC1(NC(=O)CC1COC(C(=O)Nc3cccc(=O)n3C)C1)C2 Nc1cccc(C(N2C3CCC2C(NC(=O)C(c2ccccc2Cl)O)C3)=O)c1O N1(C(C(C)OCC)=O)CCCC1(C)C(=O)NCCN(C1CCCC1)C C(=O)(C(CO)C(C)(C)C)NC1C(NC(C2CCN(S(CCC)(=O)=O)CC2)=O)C1 C(N=c1[nH]c2c(c(=NC3CCC4CC34)[nH]1)CCCC2)c1c(Cl)cc(Br)cc1 c1(C(C)C)cc(C(=O)Nc2cnn(C(=O)NC3(CC4CC4)CCC3)c2)no1.CCSC C(N=c1[nH]c(=NC2CCCCC2C#N)[nH]c2c1COC2)c1c(C)ncs1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C2CCCCC2)=O)cccc2cnnn12 c1(C(=O)NCC(C)(CO)NC(CC2(OC)CCC2)=O)nc(C)[nH]c1C(F)(F)F C(C#Cc1cn(CC2CC(F)(F)C2)nn1)NC(CC1C(C)CCCC1)=O c1(C(C)(C)C)ncc2c(n1)CCN(C(c1c(F)cc(Br)cc1Cl)=O)C2 N1(C(Cn2ccc(C)n2)=O)CCC(F)(CNC(=O)CN(C2CCSC2)C)C1 N1(C(c2c(CN)nn3c2CCCC3)=O)CC(S)CC12CCOCC2 c1(C(=O)NCCCOCC(C)C)ccc(CNC(C2CN(C3COC3)C2)=O)cn1 C1(CNC(C(C)(C2CCC2)NC(CCSC)=O)=O)C2CCCCCC12 CN1CCCC(O)(CC(=O)NCC(C)(C2CC2)NC(c2ccnc(CO)c2)=O)C1 c1(C(=O)NC2(CCNC(C(C(C)(C)C)NC(N)=O)=O)CC2)cc2c(s1)CCC2=O Cc1ccc2c(C(=O)NCC3CCCCC3NC(=O)CS(C)(=O)=O)coc2c1 N1(C(c2c(C)ncs2)=O)CC(CNC(=O)CCCCN(C)C(C)C)CCC1C Cc1cc(C(=O)NC2CCCC23CN(C(C2CCN(C)C2=O)=O)C3)c(O)nc1C Cc1ccc2snc(C(=O)NCCC(O)CNC(=O)CCc3nc[nH]n3)c2c1 C1(C(=O)NCC2CC(NC(COCCC#C)=O)C2(C)C)CCCCC1N=[N+]=[N-] c1(C(=O)OCC)nc(C)sc1NC(C1CCC(NC(C2(Br)CCC2)=O)CC1)=O c1(C(=O)NCC2CC(C(=O)NCC(C3CCCCC3)C)C2)ccccn1 N1(C(C2(OC)CCCCC2)=O)CCCCC(NC(C2OCCOC2(C)C)=O)C1 C1(C(NOCCC)=O)CCCCN(C(C2CCN2CC)=O)C1 C12CN(CCO1)C2=O.c1(C2(N(C(COCCCN(C)C)=O)C)CC2)cc[nH]n1 N1(C(C(CCSC)O)=O)CCc2[nH]nc(CNC(=O)C(C)SC)c2C1 c1(C(=O)NCC2C(NC(C=Cc3n(CC)ccn3)=O)C2)ncc(Cl)cc1Cl N1(C(C2CCC(C(N)=O)C2)=O)CCCN(C(c2sccc2N(C)C)=O)CC1CO C(=O)(C(=O)CC(C)C)N1C(C(CNC(C2CC(C)(CC)C2)=O)(C)C)CCC1 N1(C(c2c(OC)nsc2)=O)CC(C)(C(=O)NCCn2cnnc2)CC1(C)C C1(CNC(CCC)=O)CN(C(c2cc(N)ccn2)=O)CC(C(F)(F)F)O1 C1(CNC(c2c(C(C)(C)C)ncs2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(N(CC(=O)NCC2(CO)CN(C(C(COC)O)=O)C2)C)ccccc1[N+](=O)[O-] c1(C(C(=O)NC(CNC(C2(COCC)CC2)=O)CO)CO)ccc(Cl)cc1 CN1CCCCC(CNC(=O)CCCNC(=O)CCCn2cccc2)C1 Cc1cc(CCC(=O)NC23CC(CNC(C4CC45CC5(F)F)=O)(C2)C3)cc(C)n1 C(=O)(C(C)(C)CC(=O)OC)N1CCN(C(CN(S(CC)(=O)=O)C)=O)C(C(C)C)C1 N1(C(c2n(CC=C)ccc2)=O)CC(NC(c2cc(Br)c(C)cn2)=O)CC(C)C1 CCCCCC(=O)NCC(N1CC(NC(=O)C(C)CN2CCOCC2)C(C)C1)=O C1(C(=O)NC(CCC)CO)COCCN(C(c2cnc(Br)s2)=O)C1 C=CCC(C(=O)NC1COCC1NC(=O)CCc1ccc(Cl)cc1F)C(C)C c1(OC)ccnc(C(=O)NCCC(C(C)C)NC(=O)CC2COCCO2)c1OC Cc1cnc[nH]c1=NCCC1CCCN(C(=O)C(O)C(C)C)C1 N1(C(C(C)NC(C)=O)=O)CC2CC(C1)N(c1ncc3ccsc3n1)C2 C1(CC)CCN(C(C2CCSCC2)=O)C1C(=O)Nc1ccccc1O C(=O)(C(C)(C)CC(=O)N1CCCC(N(C(=O)CC2(C)CCCO2)C)C1)OC N1(C(c2cncnc2)=O)CCCC2(CCCN(C(c3ccnc(Br)c3Cl)=O)C2)C1 C1(C2(O)CCCOC2)(CNC(c2n(C)nc(C3CCC3)c2)=O)CC1 N1(C(=O)C=Cc2cc[nH]n2)CCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])(c2nn[nH]n2)C1 C1(C(=O)NCCCOCC#C)CCN(C(=O)C2(C)CC2(C)C)O1 c1(C(N2C(C(N3CCC(C(=O)OC)C3)=O)CC3CC32)=O)cc(Br)c(O)c(Br)c1 c1(C(=O)NC2CCN(C(CCCSC)=O)C2)cc2cc(C#N)ncc2[nH]1 C(=O)(CC(F)(F)C(F)F)N1C(CNC(C2CC2C(F)(F)F)=O)CC1 n1(CC(=O)NCC(C)CN(C(=O)C(c2cncnc2)C)C)cc(S(C)(=O)=O)cn1 C1(C(N2CC(CC(C(=O)N(CCCC(C)O)C)F)C2)=O)NC(=O)OC1(C)C Cc1cc2c(C(N3CCC(C)(CNC(=O)C(C)O)C3)=O)nccn2n1 N1(C(CNC(=O)OCC)=O)CC(NC(c2csc(C(C)(F)F)n2)=O)C2(CCC2)C1 C1(C(N2C(C(=O)NC)CC2)=O)CCCC1NC(c1csc(CO)n1)=O C1(NC(=O)CSCC2CCCCO2)CCCN(C(=O)Cc2ccccc2)C1 C12(C(=O)NC3CCC(N(C)C(c4nc(Cl)cs4)=O)C3)CCN(CC1)S(=O)(=O)C2 C1(CC(=O)NC(C2CCN(C(C(C)NC(CC)=O)=O)C2)C)C(=O)ON=C1C CC(CC(N)=O)C(=O)N1CCN(C(=O)CC2CC(C3CC3)C2)C(C2CCCC2)C1 CC(CS(C)(=O)=O)C(=O)NCc1cccc(NC(=O)CCC2CCCN2C)c1 C1(c2cn(C(C)C(=O)N3CCCC3)nn2)(N(C)C)CCN(C(=O)C(F)F)CC1 N1(C(C(C)(C(F)(F)F)OC)=O)CCC2(COCCO2)C1 N1(C(C2(C)C(C)OCC2)=O)CCCC(NC(=O)CSc2ccncc2)CCC1 C1(NC(C=Cc2cc(OC)ns2)=O)COC2(CCN(C(c3cnc(O)s3)=O)C2)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(C1CN(C(CC(C)(C)SC)=O)C1)C CC(CCOc1ccccc1)C(=O)NC1CC(NC(=O)Cn2cnnc2)CC1O N1(C(CN(CCOC)C)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 C=CC1CN(C(=O)CC(CC2CC2)NC(C2CCC2C#N)=O)CC1O c1(C(=O)NC(CN(C)C(C2CC(C)(F)C2)=O)(C)C)ccn(C2CCCC2)n1 c1(-n2cc(COC)nn2)ccc(NC(c2ccc(Br)cc2)(C)C(=O)O)cc1F C1(NC(CC(=O)NCC#C)=O)CC2CC1N(C(C1(N(C)C)CCOCC1)=O)C2 Cc1cc(C(=O)NC2CC3(C2)CC3C(N2CCOC(C)(C3CC3)C2)=O)cc(C)n1 N1(C(C(C)N2CCCC2)=O)CCCC(O)(CNC(C2(C)CC=CC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)o2)=O)ccccc1Br CC1CCN(C(C2(n3ccnn3)CC2)=O)CC1NC(c1ccc(Br)s1)=O c1(C(=O)NCCCC(C)NC(=O)C=Cc2cc[nH]n2)cccc(-n2cccn2)c1 N1(C(Cc2n(C)c(S)nn2)=O)CCC2CCCC(C1)N2C(C1CCOCC1)=O c1(CC(=O)NCCSCc2cn(C3CC3)nn2)cccnc1OC(F)F C1(C)(CC(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)CC(F)(F)C1 Cn1cc(Br)c(C(N2C3CCC2CC(NC(=O)CCC#N)C3)=O)cc1=O N1(C(=O)C=CC2CCOC2)CCN(C(c2cc(C3CCCC3)no2)=O)C(CO)C1 C(=O)(C(C)c1ccsn1)N(CCCNC(C1(C(F)(F)F)CC1)=O)CC C1(CC)CN(C(C2C3CC(=O)CC23)=O)CC1C(=O)N(C)CC1CCCN1CC C1(NC(C2CC(C(F)F)(OC)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(N2CCC(CNC(C(C)SCC)=O)C2)nc(C)ncc1F c1(C2(C(C)NC(c3cncc(F)c3)C)CCC2)ccc(Cl)cc1 N1(C(c2c(C)cn(C)n2)=O)CCCC2C1CCN2C(C1CN2CCN1C(C)C2)=O C1(C(=O)NC(CNC(=O)NC)C2CC2)CCCCC1Nc1ccccc1 C1(C(N2CCC(CC)(CC)C2)=O)CN(C(c2cc(C#N)cs2)=O)C(C)(C)C1 c1(C(=O)OC)cnc(O)c2ccsc12.C12CC13CCN(CC3)C2=O C1(NC(C(F)=CCC)=O)CCCC1NC(c1oncc1CC)=O C(=O)(CC(COC)COC)N(C1CCN(C(=O)CC2CCOC2C)CC1)CC#C O=C1Cc2cc(C(N3CCC4(C3)CN(C(C3CCCSC3)=O)C4)=O)ccc2CN1 C=C1CCC(C(=O)N(CCC(=O)N2CCC2C(C)O)C2CC2)CC1 c1(C(=O)NCC2=CCN(C(CC(=C)C)=O)CC2)cccc2c1ncn2C N1(C(C=Cc2c(C)ccnc2)=O)CCC(NC(c2ncn(C)n2)=O)CC(C)(C)C1 C(C1=Cc2ccccc2OC1)Nc1cc(C(=O)OC)cc(C)c1 C(=O)(CCCC(C)(C)C#N)NC(CN(C(c1nc(C)c(C(F)F)cc1)=O)C)C C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2nc(CC)oc2)=O)CC1)CC C1(NC(C(C)(C)NC(C)=O)=O)CN(C(=O)NC2CCN(C)CC2)C2CCCC2O1 c1(C(N(C2C3CN(C(C(CC)C(C)C)=O)CC32)C)=O)c[nH]c2cccc(F)c12 N1(C(C2CCN(C(CC)=O)O2)=O)c2ccccc2CC1C N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(C)C1 c1(OC)ccc(CC(C)C(N2CCC(O)(CNC(=O)C(C)=CC3CC3)C2)=O)cc1 Cc1c(CNC(C2CCN(C(c3nnn(C)c3N)=O)C2C)=O)cccc1O c1(C(=O)NC2(F)CC=CCC2)ccccc1-n1cc(CC(CO)CO)nn1 c1(-c2cccc(C(N(c3ccccn3)CCCC)=O)c2)nnc2n1CCC2 c1(OC)ncc(Cl)cc1C(C(=O)NC1CCCC1)N(CCC#N)C c1(N)oc2ccccc2c1CO.c1(C(C)(C)C)ccccc1C(N1CCCC1CO)=O C(=O)(C1CN(N2CCC=C(Cl)C2)Cc2c1ccc(C)c2F)OC C1(CNC(C(C)(C2CCOCC2)OC)=O)C2CN(C(c3ccc(F)cn3)=O)CC12 C1(CNC(c2c(C(C)C)nns2)=O)COCCN(C(c2nncn2C)=O)C1 C1(C(=O)N(CCCOCc2ccco2)CCOC)CSC(Cc2ccco2)C(=O)N1 c1(C(N2CC3(C(CNC(CCCC)=O)CC3)C2)=O)ccc2c(c1)nc(O)n2CC C(=O)(C(C(C)O)N(C)C)N1C(CC(=O)NCc2nc(C)[nH]n2)CCC1 C1(C(N)=O)CN(C(c2cnc(C3CC3)s2)=O)CCC1NC(C1(C2CCCO2)CC1)=O Cc1cc(Br)c(C(=O)NCC2CN(C(=O)C3=CCSC3)C3CC23)s1 C1(CCOC)CC(N=c2cc(NCCc3ccccc3C)nc(C(C)C)[nH]2)C1 Cc1ccn(C(C)CC(=O)N(CC(O)CN(C)C(c2c[nH]cc2C)=O)C)n1 c1(C(=O)NC(CN(C(c2c(NC)cncc2)=O)C)C)nc2cc(O)ccc2[nH]1 c1(OC)cc(NC2CC(NC(=O)Cn3nc(C)oc3=O)C23CCC3)nc(OC)n1 C12(NC(C3CCCC3)=O)CC(CNC(c3cnc(C4CCCO4)s3)=O)(C1)C2 c1(C(=O)NCC2(O)CC(NC(C(C)NC(=O)NC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C c1(NC(CCC2(C)N(C(CC3N(C)CCC3)=O)CCC2)=O)cccc2cncn12 CCC(C(=O)N1CCC(CCNC(=O)C#CC2(C(F)(F)F)CC2)CC1)C(C)C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(=O)NCCCNC(=O)CCCc1cncs1 N1(C(C(C=C)(C)C)=O)CCC2C(NC(c3ccccc3OCCC)=O)C2CC1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(=O)C(C)=C(C)CC)C(C)C1 C(C(O)CN=c1[nH]cncc1I)NC(Cc1ccc(NC(C)=O)cc1)=O n1(CC(=O)N(CCOCCNC(C2CCC(C)C2)=O)C)ncc2ccccc12 c1(CC(N2C(CCNC(CN3CC(C)(C)C3)=O)COCC2)=O)ccc(F)cc1F C(=O)(N=c1nc2c(I)cccn2[nH]1)N1C(c2cc(CC)no2)CCCC1 c1(C(N(C2CCN(C(=O)C(C)(C)c3cncs3)C2)C)=O)cc2n(c1)CCCC2 C(C)(C(C(C)C)NC(=O)CCc1cccc(O)c1)NC(CCOCCC)=O N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CC(NC(C2CCCC2)=O)C(S(C)(=O)=O)C1 C1(NC(C(C)SC)=O)CCCC1(C)NC(=O)CN(CC(C)(C)C)C N1(C(C(c2cccs2)N(c2nnnn2C)CCOC)=O)CCC(=C(F)F)CC1 c1(N2CCCC(C(=O)NCc3cn(CCC)nc3)C2)cc(C)ncc1C#N N1(C(Cc2ccc(C)cc2)=O)CC2CC1CCC2NC(=O)CC1CC2CC2C1 CC(C)C(C)(O)C(=O)NC1CN(C(c2cc(C#N)cs2)=O)CC1n1ccnn1 c1(C(N2CC(F)(c3ccccn3)C2)=O)sc(F)cc1Cl N1(C(Cn2c(C(C)C)nnn2)=O)CCC2CC2(NC(c2cn(C)cn2)=O)CC1 c1(CNC(c2c(CCNC(C3C(C)(C)C3)=O)n[nH]c2)=O)ccc(F)nc1F C1(C(=O)OC)C2CCCC2CN1Cc1coc(C#N)c1 C(C(CO)(CO)NC(=O)COCC1CCCO1)N(C(=O)COC(F)F)C CCC(COC)C(=O)NC1CCC1NC(=O)Cc1sc(S)nc1C CCCCC(CC(=O)NC1(c2ncccn2)CC1)NC(=O)CC1CC2C=CC1C2 n12ccc(cc1=O)C(=O)NCC2.c1(C(n2cccc2)(C)C)ncnn1CCCl CN1CCC(CC(N2CCC(C)(NC(c3ccc(C(F)F)nc3)=O)C2)=O)C1=O c1(C(=O)NC(CCOC)C)ccccc1NC(c1cccc(C)c1)=O N1(C(CC(C)CNC(C2CCN2C(C)(C)C)=O)=O)CCC2(CC1)CSC2 C1(C(=O)NC2CC(C)(NC(C(C(C)C)n3ccnc3)=O)C2)CN2CCCC2CO1 C(=O)(CC(O)CC(C)(C)C)NCC1(F)CCN(C(C(CCC#C)O)=O)CC1 CC1CN(C(C2CN(C3CCCCC3)C2)=O)CC1NC(=O)C#CC(=O)N(C)C c1(C(=O)NCC(CNC(C(c2cccnc2)C)=O)C)ccc2c(c1)N(C)CCO2 C1(c2ccc(F)cc2)(C(=O)NCCCNC(=O)CN2CC3CC3C2)CCCCC1 C1(C#N)(CC)CCN(C(C2C=CCCN2C(C2CC3CC3C2)=O)=O)CC1 N1(C(CCCN(C)C(C2CCCN2C2CC2)=O)=O)CCN(CC(N)=O)CC1 C1(NC(CNC(CCC)=O)=O)COCCC1NC(=O)COC1CCCC1O C1(NC(C(CC)NC(C)=O)=O)CC2C1CCN2C(c1ccco1)=O N1(C(C(CN(C(C2C(=C)C2)=O)C)(C)C)=O)CC2CC(C)C2C1 N1(CC)CC(NC(=O)CCC2CC(NC(=O)Cc3cc[nH]c3)C2)CCC1=O c1(NC(C(=O)N(CC)Cc2sccc2Br)=O)cccc2c1CN(C1CC1)C2=O N1(C(C2C(C)(C)C2)=O)CCCC(C)(NC(c2ccc[nH]2)=O)C1 C(C(CC(C)C)C(=O)NCC(C)(F)CNC(C1CC(=O)C12CCC2)=O)OC c1(C(N2CCC(C(=O)NCc3cc(C)cc(F)c3)C2)=O)cc(F)c(Cl)cc1C C1(C(=O)N(C(C)CNC(=O)CSc2cscn2)CC)(OCC)CCOC1 C=CCCCCCC(=O)NC1CC(F)(F)CC1NC(=O)C(C)CSC c1(C(=O)NCCCCC(C)NC(C2CC(C)OC2C)=O)nnc2ccccc2n1 C=CC(C)(CC)C(=O)N1CCC(C)(CCNC(c2coc(C(C)C)n2)=O)C1 N1(C(C(CC)n2cncn2)=O)CCCN(C(c2cc(C)c(C)nc2C)=O)C(C)C1 c1(C(N2CCC(C)(CNC(C(CC)C#N)=O)C2)=O)cc(Br)cc2scnc12 C1(CCCC)C(=O)N(C)CCN1C(=O)NC1CCOC12CCOC2 C1(C(=O)NC(CC)CSC)(C(C)C)CCN(C(=O)C=Cc2ccoc2)C1 c1(CCNC(C=Cc2ccc(OCCCC)cc2)=O)ccc2c(c1)CCN2 CC1(C)CCC(C(=O)NCC(=O)NCC(=O)NCCC(Cl)Cl)CO1 N1(C(C(CC(CC)CC)F)=O)Cc2n[nH]cc2C1C(=O)N1CCCC1CC(N)=O CCC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NC1(C)CSC1 c1(-c2scc(NCC(C)F)n2)ccc2c(c1)CCCO2 c1(-c2cn(C3CCCN(C(=O)NCCC=C)C3)nn2)cc(C)cc(Br)c1 Nc1ccc2c(NC3CCC(=O)N4CCCC34)nccc2c1 C1(OC)CN(C(=O)CCOCCNC(c2ccccc2)=O)CC(C)(O)C1 C(=O)(C(CC(C)C)C(C)C)NCC1(OC)CCN(C(=O)CCc2ccn(C)n2)C1 c1(C(=O)NCCC2(NC(CCc3n(C)ccc3)=O)CCC2)cnn(C)c1C(F)F C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)NCC(CO)NC(CN(C)CC)=O c1(C(=O)NCCOCCN(C(c2c(CC)con2)=O)C)cc(Br)ccc1C C(=O)(CCCCCC#N)N1CC(C)OC(CCNC(=O)C(=O)NC2CC2)C1 Cc1ccc(C(N2CCC(CN(c3ccc(CO)cc3Cl)C)C2)=O)cc1[N+](=O)[O-] CC1=C(C)CC(C)(NC(=O)C(CO)NC(=O)CCc2ccccn2)CC1 Cc1[nH]c2ncnc(NCc3nncn3-c3ccccc3)c2c1C C=C1CCN(C(c2c[nH]nc2OC)=O)C(C(=O)NCC(C)C(F)F)C1 C(C(C)(CC(C)C)NC(=O)CCc1cncn1C)NC(COCCCC(C)C)=O C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1 C(=O)(CCCCCS(N)(=O)=O)N1CC2=C(CN(C(C=Cc3n(C)ccc3)=O)C2)C1 C(C(=O)N1CCN(C(=O)C(C)OCC2CC2)CC1)(C(C)C)n1ccc(C)c1 CCCS(=O)(=O)CC(=O)N1CCN(C)CC1CNC(=O)CSCC(N)=O C1(N(C(CC(=O)OCC)=O)CC)CCCN(C(C2CC(c3ccccc3)C2)=O)C1 c1(CNc2nc(COC)nc(N3CCCC(C)(OC)C3)c2)cc(C#N)ccc1Br N1(C(C2N(C)C(=O)NC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1CCO CC1CN(C(C2(C)CSC2)=O)CCC1NC(c1cc(OCC(F)F)ccn1)=O N1(C(c2c(COC)cco2)=O)CCC(NC(C2(C)COC2)=O)C(C)C1 N1(C(CCn2c(C)ccc2C)=O)C2CCC1CN(C(c1cnn(C)c1Cl)=O)CC2 N1(C(COc2cc(C)on2)=O)CC2(C1)CN(C(=O)CC(C)C(C)(C)C)CCO2 C1(C(=O)NCC(O)CCOC)(CC)CN(C(=O)CCc2ccoc2)C1 n1(C2CCN(C(=O)NCC3C(C)COCC3)CC2)cnc2ccccc2c1=O c1(OC(C)C(N2CCC(C)(NC(C3(C)CC3C)=O)C2)=O)ccc(F)cc1Cl C1(C(N2C(C(N3CC(SC(F)F)C3)=O)CSC2)=O)CC2CCCCC12 c1(NC(C2(C)N(C(c3c(Cl)ncc(OC)c3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I c1(C(N2CCC(O)(CNC(=O)C3=CCCCC3)C2)=O)cc(Cl)cc2ccccc12 C1(n2cc(C(C=C)(C)O)nn2)CN(C(C2(C)COCCO2)=O)CC1O CCCC(C(=O)NCCOCC1CC1)NC(=O)CC1CCCN1C CC1(CNC(c2cc(C3CCCCC3)[nH]n2)=O)CCN(C(C2CCCCO2)=O)C1 c1(CC(=O)NCC2C(NC(C(C)OC3CCCC3)=O)C2)ccc(F)cc1[N+](=O)[O-] N1(C(C2N(C(=O)NC)CCC2)=O)CC2(CC(NC(=O)CCC(C)C)CO2)C1 c1(C(N2CCN(C(CCC(C)OC)=O)C(CF)C2)=O)ccc(Cl)c(C)c1Cl c1(N(C)CC2CCCN(C(C(COC)O)=O)C2)nc(C(F)F)nc(=N)[nH]1 c1(C(=O)NCCC(CNC(C2CCC(C)(C)OC2)=O)O)cc2cccnc2[nH]1 C(CNC(c1cc(F)ccc1OC)=O)(C(C)C(C)C)NC(c1ccn(CC)n1)=O C1(CC)C(NC(=O)CSC(F)(F)F)CCN1C(C1CC(C)N(C)C1)=O c1(C(=O)NC2CCC(CNC(C3CCC(CC)O3)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(c2c(C)cno2)=O)CCC(NCC2CCCCC2C)C(C)C1 c1(NC(C(CC)Br)=O)ccc2c(C(=O)Nc3ccc4nc(C)oc4c3)ncn2c1 C(=O)(C#CC1(C)CC1)N(CCCCCNC(=O)COCC1CCC1)C c1(CCCC(=O)NCC(C)NC(=O)Cc2ccnn2C)ccc(Br)cn1 c1(N2CCC(OCCNC(C3CCCOC3)=O)C2)nccc(-n2ccnc2)n1 N1(C(c2n(C)c(O)nc2)=O)CC2CC(NC(c3csc(C(C)(F)F)n3)=O)CC1C2 N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(CO)oc2C)=O)C(CO)C1 N1(C(Cc2ccc(SC)cc2)=O)CCN(C(=O)C(F)=CC2CC2)C(C)C1 C1(C)(C(=O)NCCN(C(c2cnc(C3CCOC3)s2)=O)CC)CC(C(C)C)=NO1 N1(C(CC(=O)OC)=O)C(C)CC2CN(C(=O)CCc3cnc(C4CC4)o3)CC12 N1(C(C(C)(C)C(F)F)=O)CCC2(CCC(NC(=O)C3=CCOC3)CC2)CC1 C(CN=c1[nH]c(N2CCOCC(C)(F)C2)nc2c1CSC2)c1c(C)cccc1 CC1(C)C(CC(=O)NCc2cc(C(=O)NCc3csc(O)n3)cs2)CC1O C1(C(=O)NC23CN(C(C4CC(OCC)C4)=O)C(C2)C3)CCCC(C)CC1 CC(C)(C)C(C)(C)C(=O)NC1CN(C(c2cccc(N)n2)=O)CC1O C1(CC(=O)N(C)CC2CCCOC2)C2CCCC2N1C(=O)C(C)(C)CF c1(C(C(=O)NCCOC2CN(C(CCSCC(C)C)=O)C2)C)cccc(Cl)c1 CC(CCC(=O)NCC=CCNC(c1ccncc1C(F)F)=O)S(C)(=O)=O c1(CC(=O)N(C(C(C)N(C(Cc2c(CC)con2)=O)C)=O)CC)cccnc1O Cc1cc(C#N)sc1C(N1CCC(N(C)C(C2CCC(C)(C)OC2)=O)C1)=O N1(C(CC=C)=O)CCOCC1SC.N12CCOC(C1)CC2=O Cc1cccc(C(N2CCCC2CCCNC(c2cnc(N(C)C)nc2)=O)=O)n1 CCC(C)C(O)C(C)C(=O)N1CCC(F)CC1C(=O)NCCn1ncccc1=O C(=O)(C1CCCn2ccnc21)N1C(CNC(CC(CCC)C)=O)CCC1 c1(CC(=O)N(C2CCC(NC(c3ccncc3F)=O)C2)C)cnn(C)c1C(F)F N1(C(C(CC)n2cncn2)=O)CCC(CCC(N2C(C)CC2(C)C)=O)CC1 c1(C(=O)NC(CCNC(CC2CCCN(C(C)C)C2)=O)C)occ2c1CCOC2 CCC(C(C)(F)F)NC(=O)CC1CCCC1NC(c1cc(OC)nn1C)=O N1(C(c2ccnc(CO)c2)=O)CCC(CC(F)(F)F)C(NCCC2CCCC2)C1 N#CCCCCC(=O)N1CC(NC(c2cccc(C3CC3)n2)=O)C1 c1(C(=O)NCC2(NC(c3ccc(O)cc3O)=O)COC2)n[nH]c2cccc(F)c12 C=CC1(CC(=O)NC2CCCC(NC(=O)Cc3ccc(C)cc3)C2)CCCCC1 C=C=C(C)CC(=O)NC(C)CN(C(=O)CCCc1ccc(Cl)cc1)C Cc1cc(S(=O)(=O)NC2CCC(F)(F)C2)c(C)cc1-c1sccc1C C=CCCCCCC(=O)NCC1(F)CC2CCC(C1)N2C(=O)Cc1ccco1 c1(C(=O)OCC)ccc(NCCc2n[nH]cc2C)cc1O c1(C(N2CC(O)CC(NC(c3scnc3Cl)=O)C2)=O)ccc2ccsc2c1 c1(C(=O)NC2CCC(CNC(CCCS(N)(=O)=O)=O)C2)cnc2ccccc2c1 c1(CC(=O)NCC(C)(C2CC2)NC(C23CC(OC)C2C3)=O)cnccc1Cl c1(CC)cnn(CNC(=O)C(C)(C)C2CCN(C(=O)CCOC3CCCC3)C2)c1 C12(CNC(C3=NOC(C)C3)=O)CCCC1N(C(=O)CC1(C)CC1)CCC2 c1(CC(=O)NCC(CN(C(c2cnn(CCC)c2C)=O)C)O)noc(C)c1C#N c1(-c2nc(C3C(C)CN3C(=O)CC(C)O)on2)ccc(N(C)C)c(F)c1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CC(F)F)C2(CCOC2)C1 C1(N(C(C=Cc2occ(C(=O)OC)c2)=O)C)CCCN(C(=O)C(C)C(C)O)CC1 c1(OCCCC)ccc(C(=O)N(CCNC(=O)C(O)c2ccsc2)CC)cc1 N1(c2[nH]c(=NCCn3c(C)nnc3)[nH]c(=N)n2)CC(C)(C)C12CCOCC2 C#Cc1ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC(OC(C)C)C2)nc1 N1(C(C=C(C)C)=O)CC2CCCCC2(CNC(=O)Cc2nc(=N)[nH][nH]2)C1 C1(NC(C(CCC)=CCC)=O)CN(C(c2cnn(C)c2)=O)C2(CCOCC2)C1 C1(c2cn(C3CCCC(C(C)(C)C)CC3)nn2)CCC2(CC1)OCCO2 c1(CNC2CCC(C(=O)Nc3c(CC)nccn3)CC2)cc(C)c(F)c(F)c1 c1(CC(N2CCCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc2cnccc2c1 N1(C(c2c(C)oc(Br)c2)=O)CC2CC(NC(c3ncncc3Cl)=O)CC2C1 C=C(CNC(=O)C(C)CNC(=O)CCCCC=CC)c1ccccc1 c1(C(N(CC(CNC(C(C)OCCC=C)=O)(C)C)C)=O)cccn(C)c1=O c1(C(N(C2CN(C(CNC(C(CC)C)=O)=O)C2)C)=O)cnc2c(c1)NC(=O)CS2 C(=O)(C1CC(C)Nc2ccccc21)NC(CNC(CCN(CCC)C)=O)C1CC1 Cc1cc(=NC(=O)C(=O)NCC2(NN(C(=O)C(C)C3CCC3)C)CC2)[nH]o1 C(=O)(CC(C)C(C)C)NC(CNC(c1c(C(=O)OC)nccn1)=O)C C1(CN=[N+]=[N-])COCCN1C(c1ccc(CNC(c2ccc(O)cn2)=O)cc1)=O N1(C(Cc2ccc(C)s2)=O)CCC(NC(C2C3CNC(=O)C23)=O)C(O)C1 Cc1ccc(CN2C(C(N3CCN(C(=O)C4CC4)CC3)=O)CC3CC23)cc1O C(C(C)(C(=O)N1CCC(OC(C)C)CC1)NC(c1cnc(O)o1)=O)SC CC1CN(C(=O)NCCCC2CCOC2=O)c2ccc(Br)cc2O1 CCCCC(C(=O)NCCCN1CCC1)NC(=O)CC1C(=O)NN=C1C c1(OCCC)ccc(C(=O)NCCCN(C(C2CC2Cl)=O)CC)cc1CC c1(C(=O)NCCC(C)N(C(=O)C2=CCCC2(C)C)C)cc2sccc2n1C c1(OC)cc(C(=O)NC(C)C(CO)NC(c2ccc(=N)[nH]c2Cl)=O)ccc1Cl c1(CN2CC(NC(c3c(C(F)(F)F)cccc3Cl)=O)C(F)C2)c(O)cccc1O Cc1ccc(S(N)(=O)=O)cc1NC(C1CC(C)CCC1C(C)C)=O C(C(CNC(N1CCC(O)C1c1ccc(Br)cc1)=O)C(F)(F)C(F)(F)F)OC C(=O)(C1CN(C(=O)N(C)CC2COC2)Cc2n[nH]cc21)OC O=S(=O)(c1ccc(NC2C3CCCOC23)c(F)c1)N1CCCC(F)CC1 C1(c2nnnn2C)(NCc2nnn(CC)n2)CCCN(C2CCCC2)C1 CC(C)CC(C)(CNC(=O)N(C)CC1C2CC1N(C(=O)OC(C)(C)C)C2)CC c1(NC)cc(C(N2CC(OC)CC(NC(=O)CC3CCOCC3)C2)=O)cc(Cl)n1 Cc1ccc(C(=O)NCCCC(C)(C)NC(=O)CN2CCN(C)C(=O)C2)nc1C C(CCCCC(=O)N(C)CC1CCCN1C(C1CC2CC1CO2)=O)SC c1(CSCCNC(=O)NCC(C#C)O)ccc2ccccc2c1 N1(C(C(C)C)=O)CCC(C)(C)C(CNC(=O)CC(C)c2cnn(C)c2)C1 C1(CNC(c2c(Cl)cnc(C)n2)=O)CC2(CO1)CN(C(=O)CCC1CC1(C)C)C2 C1(CC(=O)NC(c2cn(Cc3ccc(Cl)cc3)nn2)CCC)CC2C=CC1C2 C(CC(C)CCNC(c1c[nH]cc1C(=O)Nc1ccccc1)=O)NC(C(C)C)=O Cc1cc(CNC(C2SCCS2)=O)oc1C(N1CCC1C(=O)N(C)C)=O C(=O)(CCCCCOC)N(C1CCN(C(=O)COCC)CC1)CCC N1(C(C2N(CCC)CCCC2)=O)CC(NC(c2ccn(CC)n2)=O)C(C2CC2)C1 N1(C(C2(C)CCCC2)=O)CCCC(C(=O)NCCN2CCNC2=O)C1 c1(CCC(=O)NC(CCNC(C(CCSC)OC)=O)(C)C)ccc(F)cc1Cl c1(OC)cc(CN(C)C(C2CC2c2ccc(C(C)(C)C)cc2)=O)ccc1C c1(C(=O)NCC2(C)CCN(C(C(C=C)O)=O)C2)cc(S(N)(=O)=O)c(C)cc1C Cc1cc(C(=O)NC(C)(CNC(=O)CC2CC3C=CC2CC3)CO)cc(N)c1 N1(C(CSC)=O)CCCC2(CNC(C3CCC(C(N)=O)CC3)=O)CCCC12 C(C(=O)N=S(=O)(c1ccccc1F)C(F)(F)F)c1cccc(OC)c1 N1(C(=O)NCCc2cccc(Br)c2F)CCC2CS(=O)(=O)CC2C1 C(=O)(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(C)C(C)n1cncn1 c1(OC)nc(C(=O)NCC2(C)CCC(NC(c3cc(Br)no3)=O)C2)ncc1F CCC(CC(=O)NC1CON(CC)C1=O)NC(=O)C(c1ccccc1)F C(=O)(C(C)(C)CC(C)(C)C)N1CC(CC)(NC(c2cncc(-n3ccnc3)n2)=O)C1 c1(OC)c(C(=O)NCC2CCO2)cccc1Br.N12CCCC1(C)C2=O c1(CC(N2CCCC2CC(N2CCCC2C(F)(F)F)=O)=O)ccnc(F)c1 c1(CC(=O)N(C2CCCN(C(C(C)OCCC#C)=O)C2)C)ncc(F)cc1F c1(-c2c(C(=O)Nc3ccc4ncoc4c3)nccc2)cccc2cncn12 N1(c2nc(C(C)C)nc(N3CCC(c4ccco4)CC3)c2)CC2CC(O)CC2C1 C1(C(N2CCCC(Cc3ccc(F)cc3)C2)=O)CCn2cnnc2C1 C12(NC(C3(SC)CC3)=O)CCC(n3cc(C(C)(C)N(C)C)nn3)(CC1)C2 N1(C(CCS(=O)(=O)NC)=O)CCC2C(C1)CN2C(=O)C(C1CCCCC1)O N1(C(CNC(N)=O)=O)CCC2(CC1)CC2(CO)CNC(c1ccc2c(c1)CC2)=O C(N=c1[nH]c(N(C)CC2CCCC2O)nc2c1SCC2)c1c(C)cn(C)n1 CCCCCC(O)C(=O)N1CCN(C(c2ccn(CC)n2)=O)CC1CCCC c1(C(N2CCC(OC)(CNC(C3CCCC3O)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCCCCCN(C(=O)C(F)C2CCOC2)C)nccc2ncccc12 C1(NC(C(=O)N(CCC(=O)OC)C(C)C)=O)CC2CCCCCC2C1 c1(C(=O)NCC2CCN(C(C(CC)CCOC)=O)C2(C)C)c(F)cc(Cl)cc1F C1(CC(=O)N(C)CCOCCNC(c2cc(C3CC3)on2)=O)CCC(=O)NC1=O C1(C(=O)NC2CC(NC(c3c(N(C)C)nccc3)=O)C2)C2CC3CC(C2)CC1C3 c1(C(N2CC(NC(C3CC34CC4)=O)CC23CCC3)=O)cncc2cc(Cl)ccc12 c1(C(=O)NC2(CN3CCN(C(=O)C(O)C(F)F)CC3)CC2)cncc2c1CCC2 c1(CC(=O)N(C(C)=O)C(C2CC(O)C2)C2CCCO2)nc(Cl)cs1 C1(C(N(CCCC2CCCC2)C)=O)CCC(n2cc(CC3CCOCC3)nn2)C1 C=CC(C)CC.C(=O)(C(C)N(CC(F)(F)F)CC)OCC(F)F C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC1CC(NC(C2CC2(F)Cl)=O)C1 C1(CNC(C(COC)C)=O)CC(NC(c2cc(N3CCCC3)ncn2)=O)C(O)C1 C#CCCCCC(=O)N1CCC(C(C)C(=O)NC2CC23CCCC3)CC1 CC1CCN(C(c2cnc(Cl)s2)=O)C1C(=O)NC(C)Cc1nc[nH]n1 N1(C(=O)CCc2ccncc2)CC(F)CC1CNC(C12CCCCC1C2)=O C1(CNC(CN(C(=O)CCCOC(C)C)CCC)=O)C=CCCC1 CC1=CCN(c2cccc(NC(=O)C(C)COc3ccccc3)n2)CC1 C1(O)(C(C)(C)NC(CCN(CC=C)C(C2C[SH](CC)C2)=O)=O)CCCC1 Cc1cc(C(=O)NCC2CCCN2C(=O)C(F)F)n(C2CCC2)n1 N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(c1cc(Cl)ncc1Cl)=O C(=O)(CCCC(=O)NC1CCOC1C(=O)NCc1ncc[nH]1)N(C)C Cc1ncccc1C(N1CCC(C)C1C(=O)NC(CCO)C(C)C)=O c1(CNC(c2cnns2)=O)ccc(N2CCC(O)C2)cc1 c1(C(CC)(C)C)ccc(C(N2CCN(CC3C4(CC4)C34CC4)CC2)=O)cc1 N1(CC)C2CCC1CC(NC1(c3cn(-c4sc(C)cc4Cl)nn3)CCCC1)C2 c1(NC(Cc2c(C)occ2)=O)cccc(NC(=O)C(c2cccc(Br)c2)C)c1 C(=O)(CCC(CF)CF)NC1CCCC(C(N2CC(C)C(C(N)=O)C2)=O)CC1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CN(C(c1cc3c([nH]1)CCOC3)=O)C2 S(C(=S)N1CCCC1)CC(=O)NC1CCN(c2cn(C)nn2)C1 c1(C(=O)NCCN(C(C(COCC)(C)C)=O)C2CC2)cnc2cc[nH]c2c1 C(c1ccc(C)nc1)=CC(=O)NC(CC=C)CNC(c1ccc(C2CC2)nc1)=O c1(N2C3C(NC(C=CCCC)=O)(CCC3)CC2)c(F)cc(C#N)cc1[N+](=O)[O-] Cc1nc(NCCSc2ccccc2)cc(=NCCN2CCCC2)[nH]1 C1(NC(C(c2cccc(C)c2)F)=O)CC2CC1N(C(c1[nH]nnc1C)=O)C2 Cc1cc(Cl)cc(N)c1C(N1CCC(CC(C)NC(=O)C(=O)N(C)C)CC1)=O c1(NCC2(C)CCC(NC(C=CC(CC)C)=O)CC2)cc(C)c([N+](=O)[O-])cc1Br C(=O)(C1=CCC(F)(F)CC1)N1CCC(OC)(CNC(C2(C)CCCS2)=O)C1 n1(CC)nc(C)cc1C(=O)NC1(CC(=O)NC2CCCC2(C)CO)CCC1 c1(OC)cc(C(=O)NC23CC(C2)N(C(=O)CC(C)c2ccco2)C3)c(F)cc1N C=CCCCCCCCC(=O)NCC(CC=C)NC(=O)CC12CC(C1)C2 c1(C(N2CC(NC(C(CC)NC)=O)C(C)C2)=O)ccc(N2CCOCC2)c(Br)c1 N1(C(c2c3n(nc2)C(C)CO3)=O)CCOC2(CCN(C(C3(C)CC3Br)=O)CC2)C1 CCC(C)(CO)C(=O)NCC(C)N(C)C(c1cnc(=N)[nH]c1)=O c1(C(N2CC=C(CNC(c3c(C)nccc3)=O)CC2)=O)cccc2cc[nH]c12 C1(C(=O)NCc2cc(C)c(F)cc2)CCN(C(=O)C(O)CCC(C)C)C(C)(C)C1 C1(CC)CN(C(c2cnc(C(C)(F)F)s2)=O)CCN1C(c1cncn(C)c1=O)=O CCCC(CCCNC(c1sc(N(C)C)nc1Cl)=O)NC(=O)COCCOCC N1(C(C(C)OCCOC)=O)C2CC1CN(C(c1ccc(O)cc1OC)=O)C2 c1(CC)ccc(C=CC(=O)NCC2(NC(=O)C(C3CCCCC3)OC)CC2)cc1 Cc1cc(C(=O)NCc2n[nH]cc2C(=O)NC2(C)CC2C)no1 CCCC(CCC)C(=O)N(C)CCN(C(=O)C(c1ccncc1)C1CCCC1)C c1(C(N2CCC(c3cccc(Cl)c3)C2)=O)cc2cccc(O)c2[nH]1 C(C(CC(F)(F)F)NC(=O)C(C1CCCCC1)F)NC(c1cncc(O)c1)=O CCCCCCC(=O)N1CCCCC(N(C)C(c2cnc(OCC)cn2)=O)C1 N1(C(c2c(C)nco2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CC(F)(F)F)C1 c1(OCC(=O)NC2CCN(Cc3cnc(COC)s3)C2)ccc2c(c1)OCO2 C1(C(N(C)Cc2cccc(CNC(C3CC(F)C3)=O)c2)=O)CC2C(C1)C2(F)F CC1CCCCC1(CNC(C1CC2(C1)CC(O)C2)=O)NC(=O)COC(F)(F)F C(=O)(CS(=O)(=O)C(C)C)N1CC(CC)C(NC(=O)C=Cc2ccccn2)C1 C1(C)(CCNC(C(COC)N(C)C)=O)CCN(C(c2c[nH]nc2F)=O)C1 C(=O)(C1CCc2nccn21)NC(C(=O)NC(c1ccc(C)cc1)C)c1cccs1 c1(CNC(CNS(NC)(=O)=O)=O)n[nH]c2c1CN(C(C1(C)COC(=O)C1)=O)CC2 C1(NC(c2cn(CC=C)nn2)=O)(CO)CCN(C(=O)C(C)NC(C)(C)C)CC1 C(=O)(C1=CC(O)C(NC(C2(CCOC)CC2)=O)C1)N1CC(O)(CC=C)C1 c1(SC)ccc(Cl)c(C(N2CCC(CNC(=O)C(CO)NC(=O)C(C)C)C2)=O)c1 N1(C(CCOCC#C)=O)CC2CC1C2NC(C1CC(CCCCC)C1)=O Cc1cc(NC(=O)CC2C3CN(C(c4c[nH]c(=N)c(C)c4)=O)CC23)c(C)cc1F C1(CC)CN(C(c2ncnc(O)c2Cl)=O)CCN1C(=O)C(C(C)C)n1cnnc1 C1(NC(c2c(OCC)cccc2)=O)CN(C(=O)C=C(CC)CC)CCC1CO C1(C(=O)NCC2(COC)CN(C(=O)C=CC3CCCO3)C2)CC(=O)NC(=O)N1 CN1CCC(NCCC2COCCN2)CC1c1ccc(Br)cc1 C1(C(N(CCNC(c2csc(C(C)(C)C)n2)C)CC)C)CC2CCC1C2 N1(C(=O)NCc2nccc(OC)c2)CC2CCCCN2CC1C c1(NC)cnc(C(=O)NCC(O)CN(C(=O)C=Cc2ccc(C(N)=O)o2)C)cn1 C(=O)(C1=COCCO1)N1CC(CNC(c2c(C)nc(CCCC)s2)=O)C(O)C1 Cc1n[nH]c(C)c1CC(N1CC(NC(c2cc(Br)ccn2)=O)C(O)C1)=O O(NC(=O)C(CCC(C)C)NC(c1ccc(C)s1)=O)CC(=O)OCC c1(OC)cc(Cl)c(Cl)cc1C(=O)N(C(C)CCNC(C1CCCC(=O)O1)=O)C N1(C(C2CC(NC(c3cc(=O)cco3)=O)C2)=O)CCCC2(CCNC2=O)C1 c1(C(N2CC(N(C(CSCCC)=O)C)C3(C2)CC3)=O)cc2cccc(C)c2o1 N1(C(C2C(C)C2)=O)CC2(CC(NC(c3cc(-c4cn(C)nn4)on3)=O)CO2)C1 c1(C(N(C)CCNC(=O)C=Cc2ccccn2)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)NC2CCN(C(Cc3c(C)n[nH]c3)=O)CC2C)cc2c(nn1)CCC2 CCCC(C)CC(=O)N1CC2(CC2)CC1CNC(=O)CCn1ccnc1 c1(C(=O)Nc2ccc(C)nc2I)cc(-c2ccccc2F)cc2cc[nH]c12 N1(C(c2c(C)onc2)=O)CCN(C(=O)COc2ccc(Cl)cc2)CC(C)(C)C1 C1(CNC(CCNS(CC)(=O)=O)=O)CN(C(c2cc3[nH]ccc3s2)=O)CC1(C)C c1(-c2cc(NC(CN(C3CCOCC3)C)CO)no2)ccc(F)cc1F N1(C(CC(=O)NCC#C)=O)CCN(C(C2CCOC(CCC)C2)=O)CC12CCC2 C1(CNC(c2c(C)cc(F)s2)=O)CC(NC(=O)Cc2cc[nH]n2)C12CCC2 c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCCC2)ccc(OC)cc1C CC1(C)C(NC(c2cc(Cl)no2)=O)CC1CNC(c1ccccc1SCCO)=O N1(C(c2ccc(C)cc2O)=O)CCC2CCC(NC(=O)CCC3CCCO3)C1C2 Cc1nc2ccnn2c(C)c1C(=O)NCC(CNC(c1cncs1)=O)CO C1(c2n(CCCOC)nnn2)(NCC(c2ccc(F)c(F)c2)C)CCCN(C)C1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CC(F)CN(C(=O)CCN2CCCC2=O)C1 C(CCCCC(=O)N1CC(OCCC(N2CCOC(C3(C)CC3)C2)=O)C1)OCC c1(C(N2CC(NC(c3c(SC)cccc3)=O)C(C)C2)=O)cc(C)cnc1F N1(C(c2ccc(F)c(C(F)(F)F)c2)=O)CCC(C2CCN(C(C3CCC3)=O)C2)C1 C1(c2cn(CCCNC(C3(COCC)CC3)=O)nn2)CCCC(=O)C1 C1(C(=O)NC(C(=O)OC)C(C)C)CC(C)CN(C(C2CS(=O)(=O)C2)=O)C1 c1(C(C(=O)NCc2nnn(C)n2)N(CCOCC=C)C)ccc2c(n1)OCCO2 C12(NC(CCC=C)=O)CCCC1CN(C(c1cnnc(C3CC3)c1)=O)C2 N1(C(CCC)=O)CCCC(N(C(=O)C(F)=CC2CC2)CC2(COC)CC2)C1 C1(NCC2C(NC(C)=O)CCC2)C2CCCC1N(C(=O)CC(C)(C)n1cnnn1)C2 C1(CNC(=O)NC2CCC(N3CCCC3)CC2)CCCC2C1C2(F)F CC1(C)CCC(C(=O)NC2CCSCC2)(NC(=O)Cc2cc(C3CC3)no2)C1 CC1Cc2c[nH]nc2CC1NC(=O)COC(c1ccc(C(N)=O)cc1[N+](=O)[O-])=O C1(C)(CNC(c2ccnc(C)n2)=O)CCN(C(=O)CCC2CCCCN2C)CC1 N1(C(CS(CCOC)(=O)=O)=O)CCC2CN(C(c3ccc(C(N)=O)o3)=O)CC2C1 c1(N2C(NCC(CNC(CSC)=O)O)CC2)nnc(C(C)(C)C)s1 CC1(C)CN(C(=O)CC2=CCN(C(C3CC(C4CC4)C3)=O)C2)CCCO1 CCC(CC(=O)N1CC2(CCN(C(C3CCC3(C)C)=O)C2)C1)C(F)F N1(C(C(C)=CC2CC2)=O)CCC2C(NC(c3ccc(OC(F)F)nc3)=O)CC12 C1(OCC)CC(C(=O)N(C(C)CN(C)C(C2(C(F)F)CCC2)=O)C)C1 N1(C(c2cnc(CC)nc2O)=O)C2CCCC1CN(C(C1CCCOC1)=O)C2 c1(C(N2CCC(CCCCNC(CCCOCC)=O)CC2)=O)cc(O)nc(O)n1 c1(CC(=O)NC2CN(C(CN(C3CC3)CC)=O)CC(O)C2)n[nH]c2c1CCCC2 O(NC(=O)CCOCCCO)CC(=O)N(CC(F)OC)CCO C1(C(=O)NCCC2CCN(C)C2)(NC(CC2C(C)CC2)=O)CC(F)(F)C1 N1(C(C2CCC(C)S2)=O)CCCC2(C1)CN(C(=O)C(F)(F)c1ccncc1)C2 C1(CC)(NC(=O)CC2CCOCC2(C)C)CCCN(C(=O)Cc2c[nH]nc2C)C1 C=CC(C)(CCOC)C(=O)NCCN(C(C1(C2CCCO2)CC1)=O)CC C1(NC(c2cc(C)cc(Cl)c2)=O)CCN(C(C2CCCSC2)=O)C12CCCC2 C#Cc1ccc(OC)c(C(N2CCC(C)C(NC(=O)Cn3ccc(C)n3)C2)=O)c1 CC(C)CCCCCC(=O)N1CCC1CC(=O)NCc1conc1C(C)C c1(CCC(N2C(CN(C(C(F)=CC)=O)CC)CCC2)=O)ccc(O)nn1 c1(C(N2CCC(C3N(C(c4c(C)cncc4)=O)CCC3)C2)=O)ccc(Br)cc1F C1(C(N(CCN=[N+]=[N-])C)=O)CC(NC(=O)CCN2CCCCC2)CCO1 c1(C(=O)NCCN(C(c2sccc2C#N)=O)CC)ncc(C)nc1OC N1(C(C(CC(C)C)C)=O)CC(C(=O)N(C2CCOCC2)C2CC2)C2(CCC2)C1 N1(C(C(CC)C(=O)OC)=O)CC2(C=C(C(=O)N(c3ccsc3)C)CO2)C1 C1(N(CC(C)N(CC(=O)NCC(C)C)C)C)CCN(c2ccccc2Cl)C1=O C1(C(N2CCC(CC=C)(NC(=O)CNS(N)(=O)=O)C2)=O)COC(C)(C)CO1 c1(CC)ccc(C(N2C3CCC2CN(C(=O)C(C)NC(N)=O)C3)=O)cc1C#N N1(C(c2nc(CC)sc2)=O)CCC(C)(C)C1CC(=O)NCC1=NOC(C)C1 CC1(CNC(=O)COCCN(C)C)CCCN1C(=O)Cn1nccn1 c1(C(N2CCN(S(Cc3nc(C)sc3)(=O)=O)CC2)=O)ccc(OC(C)C)c(Br)c1 Cc1nc(CNC(c2n[nH]c(C)c2Cl)=O)oc1C(=O)NCC1(C)CNC(=O)O1 c1(N2CCCC(NC(C(CCSC)O)=O)C2C)cc(C#N)nc(C)n1 N1(C(CC2CCN(Cc3ncc(C)cc3F)CC2)=O)CCc2cc(F)ccc2C1 C1(CNC(c2cnn(CC)n2)=O)CCC(NC(=O)CCCc2n[nH]c(=N)s2)CC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCC(NC(=O)CC(=O)N(C)C)C(O)C1 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(=O)C(c1ccccc1)C c1(N(C(C(=O)NC(C)CNC(=O)CC2CC2C2CC2)C)C)nccn2cnnc12 C1(C(C(=O)NCCNC(=O)CCC2CC2CC2CC2)N(C)C)CCCCC1 N1(C(c2cc(F)cc(F)c2)=O)CC2CCCCC2(CNC(C2CC(O)C2)=O)C1 c1(-c2cc(C)c(=N)[nH]c2)cccc2c(C(=O)NCc3noc(C)n3)[nH]nc12 N1(C(=O)CCCc2ccccc2)CCN(C(=O)CC2CC3CC2C3)C(CCO)C1 c1(C(=O)NCCCCN(C2CCC(F)(F)CC2)C)nc(F)ccc1F c1(C(N2C3C(NC(C(CC)C)=O)C(C3)C2C)=O)ccnc2[nH]c(C)nc12 Cc1nn(C)c(S(=O)(=O)NC(C)Cc2cccs2)c1C(F)F Cc1cc(OCC(=O)NC2C=CC(CNC(C3C=CCCC3)=O)C2)ccc1Cl c1(C(C)=O)ncc(CCC(=O)NCCN(c2ccccc2)C(=O)CSS(C)(=O)=O)o1 c1(-n2c(C(C3CC4CC4C3)NCCCO)nnn2)ccc2c(c1)OCO2 C1(C#N)(C(=O)NC(C2CC2NC(c2cc(F)ccc2F)=O)C)CC12CCCC2 CC(CC(=O)NCCCN(C)C(c1csc(C(F)(F)F)n1)=O)c1cccnc1 c1(C(=O)NCCNC(C2N(C)C(=O)CC2)=O)cc(Cl)cc(Br)c1 N1(C(C=CC=CCC)=O)CC(NC(C2(N(C)C)CCCC2)=O)C2CC12.N1CCCC1 c1(C(N2CCCC(O)(CNS(CCC)(=O)=O)C2)=O)ccc(OC)c(S(N)(=O)=O)c1 C1(NC(C(CC)(C)CO)=O)CN(C(c2ccc(F)c(Cl)c2)=O)C2(CCOCC2)C1 O=S(=O)(c1ccc(Nc2ccnc3ncnn23)cc1)NCC1CC1 C1(CN(C)C(C2(C)CC2(F)F)=O)CCCN(C(=O)CCF)C1 Cc1cc(C#N)sc1C(=O)NC1CCCCC1NC(C1CC12CC2)=O C12=NC=CC(=NCCCCCN1)N2.CCCS(=O)(=O)NCCCN(C)C1CC1 C(=O)(CC(C)CC(C)C)NCC(CC=C)NC(c1cc2n(n1)CCO2)=O c1(C(N2CCN(C(c3c[nH]c(=N)s3)=O)C3C2C3)=O)cncc2nc[nH]c12 c1(OC)cccc2c1OCCC2N=c1[nH]c(=N)[nH]c(=NC(C)CC2CCC2)[nH]1 c1(CC)cn2c(n1)CCC(C(=O)NCCC(C)NC(c1c(C)cnn1C)=O)C2 c1(OC)ccc2c(C)c(C(N3CCC(n4ccnn4)C3)=O)oc2c1 c1(CNC(=O)NC(C)C)cccc(C(=O)NCC2CC3CCC3C2)c1 Cc1cccc(C)c1C(=O)NC(C)Cn1cc(-c2cc(F)cc(Cl)c2)nn1 C=C(C)CC(Cc1ccccc1)NC(C1CC1C1CC1C(c1ccccc1)=O)=O N1(C(c2ccc(C#C)cc2)=O)C(C)CC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 C(c1cocn1)=CC(=O)NCC(CNC(=O)C(C)C#N)OC C(CCCCN=[N+]=[N-])NC(C1(CO)CCN(C(CC(C)CN(C)C)=O)C1)=O C1(O)(C(=O)NC2CC3CN(C(CCC(=O)NC)=O)CC32)CCC(C)(C)CC1 c1(C(=O)NC(C2CCN(C(C3CCOCC3)=O)C2)C)cc2cccnc2[nH]1 S(=O)(=O)(c1ccc(NCC)c(Br)c1)NCC(C(C)(C)C)OCCN1CCCOCC1 c1(C(=O)NC2(C(N)=O)CCC2)coc(CNC(=O)CC(C2CCC2)C2CCC2)c1 C1(C(=O)NCC(n2ccnc2)C)COCCN(C(=O)CC2CCC(=O)NC2)C1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC3CC3C2)=O)(OC)C1 Cc1cc(C)c(C(=O)NCCCCCN(C)C(C2CN3CCC2C3)=O)cn1 c1(CCC)ccc(C(=O)NCC2CC2NC(=O)CNC(=O)CC(C)(C)C)cc1 C1(CNC(c2n(CC)ncn2)=O)C2CN(C(=O)C(Cc3ccccc3)CC)CC12 N1(C(C2(F)CN(C(c3nccc(CC)c3)=O)C2)=O)CC(C#N)C2(CCC2)C1 Cc1nc(C2CC2)ncc1C(=O)NC(C)CNC(c1cnn(C(C)(C)C)c1)=O C1(C(=O)OCC)CCCC(C(=O)NC2CC(NC(c3ncccc3SC)=O)C2)C1 C1(CN(C)CC)CCN(N2CCC(C3CCCO3)CC2)C1 N1(C(C2CC(C)(O)C2)=O)CCC2(NC(=O)Cn3nnc(C4CC4)n3)CCCCCC12 N1(C(c2c(C)cccn2)=O)CC2(CCN(C(C3CC(C)CC(C)(C)C3)=O)C2)C1 c1(C(N(CC(O)CNC(C2CCCC23CC3)=O)C)=O)cc2nccc(Cl)c2s1 c1(C(=O)NCC(CNC(C2(C)N(C(C)=O)CCC2)=O)(C)O)ccc2nnnn2c1 C1(NC(=O)CC2(C(F)(F)F)CC2)CCN(Cc2cnn(-c3ccccc3)c2)C1 C1(C(C)C(=O)NC(C)(C)C)CCN(Cc2c[nH]c(Br)c2)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CN(C(C2C=C(C)CS2)=O)C)COCC1 c1(C(=O)NC2(CNC(C34CCC3C4)=O)CC2)cccc(C2CC2(F)F)c1 c1(OC)cc(F)cc(S(=O)(=O)NCC2C=CCCCC2)c1 C(=O)(C(C(C)(C)C)n1cc(C2CCCCC2O)nn1)NCC1(C)CNC(=O)O1 c1(C(=O)NC2(CC=C)CN(C(c3cc(C)co3)=O)C2)cccnc1S C1(NC(COc2cc(C)on2)=O)CC2CCC1(NC(c1cc(F)cc(Cl)c1)=O)C2 C(=O)(CS(=O)(=O)CC(=O)N(C1CN(C(C2CCCC2)=O)CC1(C)C)C)OC N1(C(CCCC=C)=O)CCC(F)CC1C(N1CC(C(CC)CC)C1)=O c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(C)(C)CN(C)C)C3)nc1 C1(c2nnnn2CC2CCCO2)(Nc2cc(SC)nn2C)CC2(COC(C)C2)C1 N1(C(C2CCC(C)(C)CC2)=O)Cc2nccn2CC(NC(=O)C=C2CCCC2)C1 c1(C(=O)NCC#CC(=O)NCC2(CC)CCCO2)cc2n(n1)CCO2 CCC(C)(C(F)(F)F)NC(=O)CC1C(NC(c2cnoc2C)=O)CC1O c1(C(N2CC3C(NC(c4cc(C)n(C)n4)=O)C3C2)=O)ccc2ocnc2c1 C1(ONC(c2ccc(C)n2C)=O)CC(C(=O)N(C)C)C12CCC2 c1(CC(N2CCCCC2c2cccc(Cl)c2)=O)ccc(F)c(Cl)c1 N1(C(c2c(OCC)ccs2)=O)CC(NC(c2nc(C)nn2C)=O)C(O)C1 N1(C(c2c(N)ccc(C)c2)=O)CCC2CC(NC(C3CC34CC4)=O)CCC2C1 C(=O)(CC(=O)Nc1nccs1)NCCC(C)N(C)C(C1CCC=CO1)=O c1(CC(C)C(=O)NCC(CO)NC(=O)CCOCC(F)(F)F)ccc(Cl)cc1 C1(O)(CCNC(C2CC(OCC)C2)=O)CCN(C(C2OCCC2C)=O)CC1 C1(C(=O)NCC23CC(NC(C4CC(=O)N4)=O)(C2)C3)C2C3CCC(C3)C12 N1(C(C=C(CC)CC)=O)CCC(CC)C1NC(N1CCC(CC(C)C)C1)=O N1(C(Cn2c(CCC)ncc2)=O)CC(NC(=O)C(C)(C)C)CC(F)C1 N1(C(c2c(C)nccn2)=O)CC(C)(C)OCC1CNC(C1CSCCS1)=O c1(OC)ccnc(CNC(=O)CC2CCCC2NC(C2(C)CC2(F)F)=O)c1 C1(OCCOCC)CCCN(C(C2(C)CNC(=O)N2)=O)CC1 C1(CC)(CC)CC(C(=O)NC2CC(C(F)C(=O)Nc3cnsc3)C2)C1 c1(C2(C(=O)O)CC2)ccc(C2CC2(C2CCCCCC2)C(=O)OC)cn1 N1(C(CC2(C)CC2(F)Cl)=O)CCN(CC(=O)NCC(N2CCCC2)=O)CC1 C1(C)(C(N(CCC#C)C)=O)CCN(C(=O)C=CC2(C)COC2)C1 C1(CNC(C(C2CCCC2)NC(COCCSC)=O)=O)CC2CCCC2C1 c1(C(=O)NCC(CCOC)NC(=O)CN(C2CCC2)C)c(C)csc1Cl C=CCCCCC(=O)NCCC1(NC(=O)CC2(O)CCOC2)CCC1 CC1CN(C(c2ncc(Br)cn2)=O)CCCN1C(c1cnc(O)s1)=O C1(N(c2ccc(-c3nc(C)on3)cc2)C(=O)CN(C)C)CCNCCC1C C(=O)(CCCC(C)(F)F)NCC1(OC)CN(C(C(COC)C)=O)C1 C1(CC(=O)NCC(NOCC)=O)CN(C(c2cc(C)[nH]n2)=O)C(C)(C)C1 c1(OC)ccc2c(C(=O)NC3CCN(C(=O)CC(C)OC)C3C)n[nH]c2c1 C1(NC(CCCCC#C)=O)CCCC12CCN(C(c1cnc(CC)s1)=O)CC2 C=C(Cl)CC(C(=O)NCC1C(C)C1C)NC(=O)CNC(=O)NC C1(CC)CC(CC(N2CCC2CNC(c2cscn2)=O)=O)CCO1 C1(CN(c2n(CC)c(CC(C)C)nn2)C)CN(Cc2cc(C)cs2)C(CC)CO1 c1(C(=O)NC2CC(CNC(C3C(C(=O)OC)C3)=O)C2)ccc(S(N)(=O)=O)cc1Cl c1(C(N2CC(NC(C(CC)N(CC)CC)=O)(CC)C2)=O)cc(F)c(F)cc1O N1(C(c2ncn(CC)c2)=O)CCCC(NC(C2(COC)CCC(=O)N2)=O)C1C C1(CC)CCCC(NC(C2(CC)CN(C(c3n[nH]cc3CC)=O)C2)=O)CC1 C1(NC(CCN(C)CC)=O)CCC(O)CN(C(C2(C)CCN(C)C2)=O)C1 C1(CNC(=NCC)NCC(=O)NC2CCCCC2)CCC2(CCCCC2)O1 Cc1sc(CNC(c2nnnn2C(C)C)CC2CCCS2(=O)=O)nc1C(C)C C(=O)(C(=O)CC(C)C)NCC1(C(=O)NCC2C3COCC23)CC(=C)C1 c1(OC)ccc2nc(C(=O)NCC3CC(OC)CN3C(c3cnco3)=O)cn2n1 C1(NC(C2(C)CCSCC2)=O)CN(C(=O)Cc2cn[nH]c2)CC2(CCOCC2)C1 c1(OC)cc(NC(c2cn(CC(F)F)cn2)=O)ccc1-n1cccn1 C1(C(N2CC(CC(C)NC(c3c(C)nns3)=O)C2)=O)CCc2nnnn2CC1 C1(CC)CCC(C(=O)NCC2C=CC(NC(=O)CSc3ccccn3)C2)O1 C1(NC(CC2(C=C)CCCCC2)=O)CC1C1CCN(C(C2(O)CCSC2)=O)CC1 C1(CCC)(NC(c2cn(CCCC)nn2)=O)CCCN(C(=O)C(C)(CC)CC)C1 N1(C(CCCCOC)=O)CC2CCC1C(NC(c1ncccc1Cl)=O)C2 c1(NC(C(CCCOC)C)=O)ccc2[nH]c3c(c2c1)CCCC3C C1(CNC(C2CC3CCC2O3)=O)CN(C(c2c[nH]nc2C2CCC2)=O)CCCO1 N1(C(c2ccc(CC)c(N)c2)=O)CCCC2CN(C(=O)C(C)N3CCC3)CC12 C1(C(=O)NCC(C#C)OC)C2CC2CN1C(=O)CCc1ccccc1 c1(C(=O)NCCCC(C)NC(C2C(F)(C(=O)OC)C2)=O)cc(C(F)(F)F)cn1C c1(CC(=O)NC(CCCCNC(c2ccc(OC)s2)=O)C)cccc(F)c1Cl N(C(=NCCCC1CC1)N1CCC(C(=O)N(C)C)C1)CC(c1ccccc1)O C(c1ccncc1)=CC(=O)NCC1(F)CC(NC(c2ccoc2C(F)(F)F)=O)C1 C1(NC(c2[nH]c(=NC)sc2)=O)CC2CC(NC(=O)C(F)C(C)C)CC2C1 c1(C(=O)NC2CCC(CNC(CCC)=O)CC2)cc2scnc2[nH]1 c1(C(=O)NCC(C)N(C(=O)C=Cc2cncn2C)CC)ccc(Cl)cc1F Cc1ncc(CCC(=O)NC(CNC(c2ccsc2Cl)=O)C2CCC2)s1 CC1(C)CN(CC(=O)NCCC2(N3CC3=O)CCC2)C1.N1(CC2CC2)CCCC1 C(C(C)C(C)(C)C)N(C(C(CC)N(C)C(c1ccc(COC)o1)=O)=O)C c1(C(=O)NC(C(C)NC(c2cn(CCC)nc2)=O)C)ccc(OC(C)C)cc1 N1(CC)CCN(CC(=O)NCC2(OC)CN(C(=O)C=C(Cl)Cl)C2)C(=O)C1=O N1(C(C2(CSC)CC2)=O)CCC(C2CCN(C(c3c(C)ncn3C)=O)CC2)CC1 c1(C(=O)NCCCNC(C(c2ccc(Cl)cc2)OC)=O)cccc(Cl)c1N CC1CC=C(C(=O)NCC(=O)N(CC(C)C(F)(F)F)C)CC1 C1(CNC(c2cccc(SCC)c2)=O)CC2CCCC2N1C(C1CC(CC)=NO1)=O C#CC1(C(N2CC3CCCC2C3)=O)CCN(C(C2CN3CCC2C3)=O)CC1 C(=O)(CCC(=O)N(CCCCCCNC(=O)C(F)(F)C1CCCCC1)C)NC C1(NC(CCc2cnc(C)o2)=O)CN(C(C2(C#N)CC2)=O)Cc2nccn2C1 c1(C(=O)OC)ccnnc1NCCN(C)C(C1(C(F)(F)F)CCC1)=O.C1C(=O)N1 C1(CNC(CC2CC(C)C2)=O)CC2(CCN(C(C3CCC(N(C)C)CC3)=O)C2)CO1 C(=O)(C#CC1(CC)COC1)NC(CC)CN(C(=O)Cc1nncn1C)CC C(=O)(C(C)S(N)(=O)=O)NCCn1cc(C(=O)NCC(NOC)=O)nc1 C1(CNC(c2c(C)cn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C12CC2 C12(CNC(c3n(CCC)ccc3)=O)CC1CN(C(=O)Cc1cc(COC)on1)C2 CC1C(=O)CC1C(=O)N(C)CC1CCN(C(=O)CCOC2CCCC2)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CCC(CCNC(=O)Cn2cccn2)C1 c1(CC(=O)NCC2(C(N(C)Cc3cnn[nH]3)=O)CCC2)ccc(Cl)cn1 C(C(CNC(C1(C)CCCCO1)=O)C(F)(F)F)NC(CC(=O)OCCC(C)C)=O C12(CNC(c3cc(C)no3)=O)CCCC1N(C(=O)CN1CC3C=CC1C3)CCC2 c1(C(=O)NCC2CC(C)N(C(c3cnn(C)c3Cl)=O)C2)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C2CCCO2)(C)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O Cc1sc(C(=O)NC2CC(NC(=O)C(C)Cn3ccnc3)CC2O)nc1O C1(C(=O)NC2C(CNC(C3(F)CC3)=O)CC2)CCC2(CCCC2)CC1 c1(C(=O)NCCCC2(NC(C(C)OC3CCCCC3)=O)CC2)cc(Cl)cn1C O=C1CNc2ncc(C(=O)Nc3csnc3OC(F)F)cc2N1 C1(NC(CC2C(CNC(C3CC(C)(C)C3)=O)C2)=O)CCC2CCCC1O2 c1(C(=O)NC2CCC(NC(=O)CCN3CCCCC3)C2)ccnc2nccnc12 N1(C(C(c2c(C)cc(F)cc2)O)=O)C2CCC1CN(C(c1cccc(=O)o1)=O)C2 C=CCC(C(=O)NC(C1CCCN1C(c1cnc(O)n1C)=O)(C)C)C(C)C C(CCCC(=O)N1CC(F)(F)CC1C(=O)NCCc1cn(C)nn1)(OC)OC C1(C(=O)O)CC2(CCC(CNC(C3CCCC3N3CCCC3=O)=O)O2)C1 C=CC(C)CCNC(=O)C(C)N(C(=O)CC1(CC)CCC1)C1CC1 CC1CN(C(c2cc(F)ccc2O)=O)CCN1C(=O)CC1CC=CC1 C1(CNC(C=CC=CCC)=O)C2CN(C(c3cnn(C)c3C)=O)CC12 n1(CC)cc(-c2cn(CC(C)NC(c3ncccn3)=O)nn2)cn1 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)n3)CC(O)C2)=O)ccc(Br)c(F)c1F N1(C(CC2CCN(C(C(C=C)C)=O)C2)=O)CCC(C)C(O)C1 Cc1nc(N2CCC(CC(=O)CCN3CC(C)OCC3C)C2)ccc1C#N CC(CN(C)C)NC(=O)NCCOCCN(C(C=CC(=O)N)=O)C.C(C)(C)C c1(C(C(C)C)N(C)C)cn(C2CC(C(=O)NC(C)C(C)n3ccnc3)C2)nn1 C1(NC(=O)C2=CCCC2)CN(C(c2ccn3ccnc3c2)=O)CC1C1CC1 O=C1CC(c2cn(CC(c3ccc(Cl)cc3O)N3CCOCC3)nn2)NC(=O)N1 C1(NC(Cc2c(C)noc2C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 C(CCCC(=O)NCCCN(C(=O)C=C1CCOCC1)CCO)OCCC=C C(CCC(c1ccccc1)NCCCOC(F)F)NC(=O)NC1CCCC1 Nc1cc(CC(=O)NCC2CCC2NC(=O)COC2CC2)c(Br)cc1[N+](=O)[O-] N1(C(c2cc(C)ncn2)=O)CC(C2CCCN(C(=O)CCC3CCC(=O)N3)C2)C1 N1(C(CC(=O)N(C)C)=O)CCCN(C(c2cccc3c2CCO3)=O)C(CO)C1 CC(C)CC(F)C(=O)N(C1CCN(C(C2CCCC2)=O)CC1)C C1(C(N2CCN(C(c3c(OC)ccnc3)=O)CC2CO)=O)CCc2cncn2C1 c1(-c2cn(CCN(C(c3cc(CC)sc3)=O)C)nn2)c(C)nsc1N c1(C(=O)NCC2(C)CCN(C(CC(CC)SC)=O)C2)cc(Br)c(O)nc1C c1(OC)cnc(C(=O)NC2CCN(Cc3ccc(C(=O)O)cc3O)C2)c(F)c1 C1(NC(C(C)SCC)=O)CC2(C1)CC2NC(c1coc(C(F)F)n1)=O C1(C(=O)NC2C(NC(c3nc(COC)oc3)=O)CCC2)CC(O)CN1C C1(O)(C(C)NC(CSCCCC)=O)CN(C(C2CCCC2c2ccccc2)=O)C1 c1(C(=O)NC(C(=O)NC(C(=O)OCC)C)CC2CC2)nccnc1C C1(C(C)C)C(C(=O)O)CCN1C(=O)CC1(c2ccccc2)CCCO1 N1(C(c2ncc(C)c(Br)c2)=O)CCOC2(CCCN(C(=O)CCCCBr)C2)C1 C1(CC)CN(C(=O)CCOCC(F)(F)C(F)F)CCC1N(CC)CC c1(OCCN(C)C)ccccc1C(=O)NCC(C1CCC1)NC(c1cn[nH]c1)=O C1(CC)CN(C(=O)C(F)(F)CO)CCC1CNC(C1CC1C1CCCO1)=O C1(CNC(C(C)N(C(C)C)C)=O)CN(C(=O)CCC(=O)OC(C)(C)C)CCCO1 C(=O)(C(C)(C)C)NC(CCCN(CCOC)C(C1CC1C(=O)OC(C)(C)C)=O)=O N1(S(CC(C)C)(=O)=O)CC2CC1CN2Cc1c(Cl)cncc1Cl C(=O)(C1=CCS(=O)(=O)C1)NC1(C2CN(C(c3cc(C)ns3)=O)C2)CC1 C1(C)(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCCCC2)CCCCC1(F)F N1(C(C(c2ccc(C)o2)C)=O)CCOCC(CNC(c2ncoc2C)=O)C1 N1(C(C2(OC)CCCC2)=O)CCC2(CC1)CN(C(C1CC1C)=O)C2C(C)C CC1(C)CCCC(O)(C(=O)NCC2CCC(NC(C3(CO)CCCC3)=O)CC2)C1 C1(C(C(C)C)NC(c2cnc(C)s2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 C1(CC)C(NC(=O)CC(O)CN(C)C)CCCN1C(C1CCOCO1)=O C1(NC(CC2CCN(C(CCCCCC)=O)C2)=O)C2CCC(C2)C1(C)C c1(CC)c[nH]c(C(=O)NCC2CC(CNC(c3cc(CN(C)C)c[nH]3)=O)CO2)c1 Cc1c(CN2CCCC(CCNC(C3CCC(=O)N3)=O)C2)cnn1C c1(C(=O)NCCN(C2CCCCCC2)C(C2C(C)(Br)C2)=O)cccc2nsnc12 C12(NC(C(C3CCOCC3)OC)=O)CCCC1CN(C(c1cnc(C3CC3)[nH]1)=O)C2 c1(C(N(CC(C)N(C(C(C)NC(COC)=O)=O)C)C)=O)cnc2[nH]c(=N)sc2c1 C1(OC)CC(NC(=O)CCF)C1.C12C=CCN1C2=O.C(C)(C)(C)OC(=O)NC C12(NC(c3cncs3)=O)COCCC1CN(C(C13CCC(CO)(CC1)CC3)=O)C2 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCC(C)(CCO)C2)=O)C1 Cn1cc(CC(O)C(=O)N2CC(CCNC(c3ccsc3Br)=O)C2)cn1 C1(=CC(=O)N(C)CCN(C)C(c2cn(CCCF)nn2)=O)CCN(C)CC1 C(=O)(C(C)(O)C(C)(O)C(=O)N1CC2C=CC2C1)OC C1(NC(CCc2ccn(C)c2)=O)CC2(C1)CC(NC(=O)CC1C=CCC1)C2 C1(NC(c2n(C)c(S)nn2)=O)CCC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C2CCN(C(=O)C(O)C(C)C)C2)C)n1 c1(C(N2C(C)CC(NC(c3ccc(C)c(C)n3)=O)C2)=O)cc(N)c(Cl)c(O)c1 N1(CC(N2CCN(C(C(CC)(C)C#N)=O)CC2)=O)CC(=O)Nc2ccccc21 CC1(C)CN(C(C23CSCC2C3)=O)CC1NC(c1cc(N)ccn1)=O Cc1c[nH]c(=NCCCC2CCN(C(=O)CC3C(=O)N(C)N=C3C)C2)nc1O CC1CCC(CC(=O)NCC(C)NC(=O)Cn2nnc(=N)[nH]2)C1 c1(C(=O)NCCC2CCN(C(C3N(C)C(=O)CC3)=O)C2)nc2c(s1)COCC2 N1(C(C=CC2C(C)C2(Cl)Cl)=O)CCC2(CCN(C(C3CCS(=O)(=O)C3)=O)CC2)C1 C(=O)(CC(C(C)C)NC(=O)CCCC(=O)N(C)C)OC.C12CCN1C2=O c1(C2C(C(=O)NCC(CCNC(CCCN(C(C)C)C)=O)O)C2)ccccc1Cl C=C1CC2(C1)CC(C(N1CCOCC1CCNC(c1c(C)nn(C)c1Cl)=O)=O)C2 C1(C(N2CC3CC2(c2ccnn2C)C3)C)CC2(C1)CC2F C1(C(N2CCC(NC(=O)Cn3cnnn3)(CF)C2)=O)Cc2cc(F)ccc2O1 C(CN=c1cc(C)nc(N(C)Cc2cc(Br)cs2)[nH]1)N1CC(CC)OCC1 N1(C(CC(C)SC)=O)CC(CNC(C2CC(=C3CC3)C2)=O)C2(CC2)C1 c1(NC(CC(C)C)=O)ccccc1C(=O)NCC1CC1NC(=O)CC C(C)(CC(=O)N1CCC(NC(=O)C(F)n2cccn2)CC1)(C1CCC1)N(C)C S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)NC(CN(C(=O)CCOC)CC)C c1(NCC2(N(C)C)CCOCC2)[nH]c(=NCCNC(N)=O)nc2c1ncn2C C1(CNC(CCOC(C)C)=O)CCC2(CCC2)CN1C(C1CCCCN1N=O)=O c1(C(=O)NCC2N(C(C3CCC(C)O3)=O)CC(C)(C)C2)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2(F)C(C)C2)=O)CCCCC(CNC(=O)Cc2ccc(F)cc2F)C1 C#Cc1ccc(C(N2CCCC2CNC(c2occc2C(C)C)=O)=O)c(OC)c1 Cc1cc(C(N2CCC(NC(=O)C3CC3)C(O)C2)=O)c(C)n1C1CCCCC1 c1(C(=O)NC(C)CCN(C)C(C2CC(=C3CC3)C2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(C)NC(C(c1cc(C)c(Cl)nc1)(F)F)=O)C C1(N(C(c2ccc(-c3ccc(F)c(F)c3)s2)=O)CC)CCCN(C(=O)C(N)=O)CC1 Cc1ccc(C(=O)NC(C)CC2CCN(C(C3(CO)CCC3)=O)CC2)nc1O N#CCCCC(=O)NCC1CC1NC(c1cnn(CCN2CCOCC2)c1)=O C1(N(C(=O)Nc2cccc(C(=O)O)c2)CC2CCOC2)CC2CCC(C1)S2 N1(CC)C(=O)CCC1C(=O)NCCCCCN(C)C(C1(COC)CC(F)(F)C1)=O Cc1cn(C)nc1CNC(=O)C(C)C(C)NC(c1ccc(C(N)=O)o1)=O N1(C(C2CC=CCO2)=O)CCC2C(CCCN2C(=O)CCOc2cccnc2)C1 C(C)(C)(C(=O)NCc1ccccc1)NC(=O)NCC.C12CCCN1CNC(=O)C2 Cc1cc(N)cc(C(N2CCN(C(=O)CCC3OCCO3)CC2CO)=O)c1F C(=O)(C1=CNC2=NCCC2=C1)N(CCNC(=O)CC1(N2CCCC2)CC1)C1CC1 c1(C(=O)NCC(C2CCCC2)NC(C(CC)=CC)=O)cnc(C#N)s1 c1(C(N2C3C(NC(=O)COCC4CCC4)C(CC3)C2)=O)ccc2sncc2c1 C(CCCCC(=O)N1CC(C(=O)NC2CN(C)C(C)(C)C2)C(F)C1)OC c1(C(=O)NCCCN(C(C(C2CCCOC2)OC)=O)CCO)c[nH]nc1Cl C(CC(C)CC)(C(=O)N(CC(C)(C)OC)C)NC(C(CCC)OC)=O C1(O)(CC(N2CCOC(CNC(C3CC4C=CC3C4)=O)C2)=O)CCCCCC1 Cc1cc(-c2cn(CCOCCN(CC(N)=O)C3CC3)nn2)cc(F)c1 c1(CC(C)C)cc(C(=O)NC2CC23CC(NC(C2(C)CCCS2)=O)C3)cc(O)n1 C1(CNC(CC(C(=C)C)OCC)=O)CCCC2CN(C(=O)CC3(CO)CC3)CC12 C(=O)(C(C)C(C)C(C)(C)C)N1C2CC(NC(CSc3ccc(CC)nc3)=O)(C2)C1 Cc1ccc(CCCC(N2CC(C)CCC2CNC(=O)CSC(C)C)=O)cc1C C1(CC(=O)N(CC(=O)N(CCCO)C2CC2)CCCO)(COC)CC1 Cc1noc(CCC(=O)N(CC(=O)NC(c2ncc(C)o2)C)C(C)C)n1 C1(NC(c2c(CC)c[nH]c2)=O)(COC)CCCN(C(=O)C(c2cnn(C)c2)C)C1 C(CCCCC(=O)N(CCCNC(=O)C(C)c1ccco1)C(C)C)NC(=O)OC c1(OC)ccc(C(=O)NCC2CC(NC(C3CC(OC(F)F)C3)=O)C2)o1 C1(C(=O)OCC)CCC(NC(=O)C(c2ccsc2Cl)N2CCOCC2)C1 C(N=c1[nH]c(=NCCCOC2CC2)[nH]c2cc[nH]c12)C1(C)CCCCC1O N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CC(C1)CN(C(=O)C1=CCC1)C2 C1(OC)CN(C(=O)C(c2ccccc2)O)CC1CCN1CCCC1.C1(=O)CO1 c1(Nc2c(C(N=S(C)(C)=O)=O)cccc2)cc2c(cc1F)NCCC2 C1(C(=O)NCC(C(C)(C)C)NC(CSCC=C)=O)CC(C(C)(C)C)=NO1 C12(NC(CC(C)(C)C3CC3)=O)CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2 Cc1cc(Cl)c(C(=O)NCC(C2CCC2)NC(=O)C(C)(C)N2CCOCC2)cn1 CCCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(C(C)C)SC C1(C(C)CNC(=O)NC(C)C(=O)NC2CCC2)CCCCC1 N1(C(C(C(C)(C)C)C2CC2)=O)CCC2CN(C(=O)CCc3cc(Cl)cs3)CC2C1 c1(C(=O)NCCNC(C(C(C)C)OCC(C)C)=O)cccc2nonc12 C1(CN(C(c2[nH]cc(C)c2)=O)C)CCCC(NC(c2sccc2C#N)=O)C1 N1(C(C(C(CC)C)O)=O)CCC(C2(NC(=O)CCN(C)CC)CCC2)CC1 N1(c2nc(C(F)(F)F)cc(C)n2)CCC2(CCN(C(=O)CCc3ccon3)C2)C1 c1(OC)cc(C(=O)N(C)CC2(CNC(C3CC3(F)Cl)=O)CC2)ccn1 C(c1ccc([N+](=O)[O-])s1)=CC(N1CCC(N(C(=O)CC2CCC2)CCO)CC1)=O c1(-c2ccc(OC)cc2)n[nH]c(=NC(=O)N(C)Cc2nnc(C)o2)s1 N1(C(CNC(N)=O)=O)CCC2(CC(C(=O)N3CC4CCC3C4)=NO2)C1 C12(C(N(CCN(C(C3(O)COC3)=O)CC)CC)=O)CCN(CC1)CC2 n1(CCN(C)C)nccc1C(=O)NCC1(O)CN(C(c2cc(Br)no2)=O)C1 C1(CNC(c2ccc(C3CC3)cc2)=O)CC(O)CN1C(c1ncc(Br)cn1)=O C(=O)(C(C)(C)C1=CCSCC1)NCCCN(C(=O)COCC1CCOC1)CC c1(C(=O)NCC2(O)CN(C(C(CCC(C)C)O)=O)C2)cnc2c(c1)NCC(=O)N2 C(N=c1[nH]c2c(c(=NCCCS(C)=O)[nH]1)CSC2)C1(OC)CCC(C)(C)CC1 Cc1cccnc1-c1cn(C2CN(C(C3(N4CCCC4)CCC3)=O)C2)nn1 C12(C(N(CC(CN(C(c3c(C(C)C)cco3)=O)C)O)C)=O)CCC(CC1)C(C)O2 CC1CN(C(=O)C(CC(N)=O)NC(=O)OC(C)(C)C)Cc2ccccc21 C(=O)(C1=CC2C=CC(C1)C2)NC(CN(C(=O)CCCC(F)(F)F)CC)C Cc1ccc(Cl)c(-n2cc(CCNC(CCN3CC(O)CC(F)C3)=O)nn2)c1N C1(O)(CNC(CSCCCC)=O)CN(C(c2[nH]nnc2CC)=O)C1 c1(C(=O)NCCC2CCN(C(CC=C=C)=O)C2)nc2c(Br)cncc2[nH]1 N1(C(Cn2c(CCC)ncc2)=O)CC2C(CNC(c3conc3C3CC3)=O)C2C1 C(=O)(CC(C)(O)C(F)(F)F)N1C2CCC(CNC(CCC=C)=O)(C2)C1 O(N(C(=O)C1CC(CCNC(=O)CC(O)CN(C)C)C1)C(C)C)CC N1(C(c2cc(Br)nn2C)C(=O)NC)c2ccccc2CC1Cc1ccccc1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CC(NC(=O)Cc2cccc(C(N)=O)c2)C1 Cc1nn(C2CC2)c(Cl)c1C(=O)NC(C)C(CO)NC(=O)CC(=O)OC(C)(C)C C12(C(=O)NCC=CCNC(c3c(C(=O)OC)n(C)nc3)=O)CCN(C1)S(=O)(=O)C2 Cc1ccc2c(C(=O)NCC(C)(CO)NC(=O)C3=NOC(C)C3)ccnc2c1 c1(NC(C(C(C)C)Oc2ccc(Cl)cc2F)=O)nc2c(F)cccc2n1C N1(C(C23CC(C)C2C3)=O)CC(NC(=O)CN(C2CCCC2)C)CC(C)C1 c1(C(N2C(C)(C(=O)O)CCCC2)=O)cc2n(n1)C(C(F)(F)F)CC(C)N2 N1(C(C(C)(Cl)Cl)=O)CC(CNC(c2sccc2-n2cnnn2)=O)C(O)C1 CCCCC(CC)CCC(=O)NCC1CC(C)N(C(=O)CSC(C)C)C1 CC(C)CC(=O)NC(C1CN(C(=O)CCN2CCC2)C1)C N1(C(C2C(C)(C)CO2)=O)CC2CCC1CN2C(=O)CCC(=O)c1cccnc1 c1(CC)cc(C(=O)NCCC2CC(NC(=O)C(C)(C)C3CCOCC3)C2)ncn1 C(=O)(CC(C)(C)C(=O)N1CC(C(C(=O)NCc2cnccc2Cl)OC)C1)OC c1(OC)ccc(S(=O)(=O)NC(C)CCCCN2CCCC2)c(F)n1 C1(NC(c2c(C)nc(C)s2)=O)CCCCCC1C(=O)N(C1CC(O)C1N)CCOC C=CCCC(F)(F)C(=O)N1CC(COC)(NC(=O)Cc2ccn(C(C)C)n2)C1 c1(C(N2CC3CC(NC(c4nc(Cl)cs4)=O)C3C2)=O)cccc2ncoc12 c1(CC(N2C(CCCNC(c3cc(C)ncc3)=O)CCC2)=O)ccc(O)c(Cl)c1 c1(C(=O)NC2CCCCC2CNC(C2CC23CCCC3)=O)csc([N+](=O)[O-])c1 N1(C(C2C(OC)CC2)=O)CC(NC(c2ccccc2CO)=O)C(C2CC2)C1 CC12CC(C(=O)NCC3CCC(NC(c4cc(O)ncn4)=O)C3)(C1)C1(CCC1)O2 c1(CNC(=O)N(C2CC2)Cc2ccccc2)cc2ccccc2s1 Cc1ncc(CCC(N2CCCC(N(C)C(C3COC(=O)N3)=O)C2)=O)c(O)n1 c1(C(=O)NCc2nnc(CN(C)CCO)o2)cccc2c1nnn2C N1(C(C(C)OCC)=O)CCC(C(=O)NOc2ccc(CC)cc2)C12CC2 c1(CN(C(c2ccn(CCC)c2)C(=O)NCCC)CC=C)ccc(Cl)cc1 C1(NC(Cc2nnc(C)o2)=O)COC2(CCCN(C(c3cccnc3O)=O)C2)C1 N1(C(CCC=C=C)=O)CC2(C1)CN(C(=O)CCCOCCOCC)CC2CO c1(C(=O)NC(C)C(CO)NC(=O)CC2CCOC2=O)cc(Cl)cn1C N1(C(CN(C(C)C)C(C2COCCC2C)=O)=O)CCN(C2CC2)CC1 c1(OCC)ccc(Cn2c(C3(NC)CC4(CSC4)C3)nnn2)cc1OCC C(=O)(CCCCNC(C)=O)N1CC(C(N)=O)(CNC(c2ccc(CC)o2)=O)C1 CC(CC(=O)NCC(CO)C1CCC1)C(C)(C)NC(c1cnccn1)=O c1(C(=O)N(C(C2CCCCN2C(=O)C2=CCC2)C)CC)cn(C)c2ncccc12 CC(C)CC(C)(O)C(=O)Nc1cccc(NC(C2CC(=O)N(O)C2)=O)c1 c1(C(=O)NCC(CNC(c2nccnc2C)=O)OC)ccc(C(C)C)c(C)c1 c1(NC(C2N(C(c3c(C)ocn3)=O)CCC2)=O)ccccc1C(C)(C)C C1(NC(c2ccc(C)nn2)=O)CCC(C)N(C(C2CCC(C)(C)O2)=O)C1 C(C(C(C)C(C)C)NC(c1cc(O)nn1C)=O)NC(COCCC=C)=O C=C1CCC(CNC(=O)NC(C2CCCO2)C2CC2)CC1.c12ccccc1S2 C(=O)(C(CNC(c1cc2occc2[nH]1)=O)CCC)NC(C=C)C c1(NC(=O)NC(c2ccno2)C)coc(C2CCCN2c2ccncn2)n1 CS(=O)(=O)c1cccc(C(=O)NC23CC(NC(C4CC5CC4CC5O)=O)(C2)C3)c1 c1(OC)cc(C)c(C(N2CCC(O)C(NC(=O)CC(C)NC(N)=O)C2)=O)c(F)c1 c1(COC)cc(C(=O)N(CC(C)CNC(C2CCCC2(F)F)=O)C)n(C)c1 CCCCCC(F)C(=O)NCC(C)CNC(C1(CC(C)C)CC1)=O Cc1nc2cnn(C)c2cc1C(N1CCC(N(C)C(c2cscn2)=O)C(C)C1)=O N1(C(=O)CC2CC3CCC2O3)CCN(C(=O)Cc2nc[nH]n2)C(C2CC2)C1 C(=O)(C(C)C(C)C)N(C(C(=O)NC(c1ccnn1C)CC)C)C C(N=c1[nH]c2c(c(=NCc3ncc(C)[nH]3)[nH]1)COC2)c1c(CCC)nns1 C1(CNC(C(C=C)(C)C)=O)CC2(CCC2)CN1C(C1CCC(=O)NC1)=O Cc1c(Cl)c(C(=O)NCC(C)(CO)NC(c2csc(C(C)=O)c2)=O)nn1C N1(C(CC=CCNC(C2(C)CCC(=O)NC2)=O)=O)CC2CCC(O)C2C1 c1(C(=O)NCC2(NC(Cc3ccc(C)o3)=O)CCC2)cnc2n1CC(C)CC2 c1(NC(C2C(NC(CC(C(=O)OC)(C)C)=O)C2)=O)cc(C)c2cc[nH]c2c1 C(=O)(C1CCCc2c[nH]nc21)N1C2CC(NC(c3cccc[n+]3[O-])=O)(C2)C1 C1(NC(=O)C=Cc2ccncn2)CC(O)CN(C(c2cscc2C(F)F)=O)C1 Cc1cccc(Br)c1C(C(=O)N(CCCC(F)(F)F)C)NC(=O)C1=CCOCC1 N1(C(C=C(C)Cl)=O)CCN(C2CCC(NC(c3csnn3)=O)C2)CC1 N1(C(CCCCC)=O)CC2CCCC(C1)N2C(=O)CSCc1csc(=N)[nH]1 N1(C(C=NOC)=O)CC2CC(C)C(C1)N2C(C1CC1OC(C)(C)C)=O c1(CC)cccc(C(=O)N(CC(O)CNC(=O)C(F)n2cccn2)C)n1 CC1(NC(c2ccc(Cl)c(O)c2)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1 C1(C(=O)NC(CC(=O)OC)C)CCN(C(c2cccc(CO)c2)=O)C12CCC2 C1(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)CCC2C1C2(F)F Cc1ccc(-c2csc(CC(=O)NC(c3ccccc3)CN)n2)cc1 Cc1ncccc1CC(N1CCCC(CCC(=O)NC(C(C)C)C2CCC2)C1)=O c1(OCCN(C)C)ccc(NCC(Cc2ccncc2)CO)cc1 N1(C(C2C(=C)CC2)=O)CCC2CCC(C1)N2C(=O)C=C1CCCCC1(C)C c1(CC(=O)N(C2CCN(C(=O)Cc3cnccc3Cl)C2)CC)ccc(C)cc1C C1(N(C(C(C)S(N)(=O)=O)=O)C)CCN(C(c2cc(C3CC3)ccn2)=O)CC12CC2 C#CC1(C(=O)N(C)CC2CCCS2)CCN(C(=O)CC2CCC(C)(C)O2)C1 c1(NC(C)=O)c(C(=O)N(CCCNC(=O)Cc2cnc(C)[nH]2)C)cccc1C c1(OCC(N2CC(COC)N(C(C)=O)CC2)=O)cccc2c1CNC2=O C1(CN(C(=O)NC(C2CC(=C)C2)C(=O)OC)Cc2ccccc2)CC(C)CO1 N(C1CCc2c(Br)ccc(Cl)c21)C(=O)Nc1c(C(C)C)ccc(C(N)=O)c1 N1(C(c2c(CC)occ2)=O)CCCC(NC(C2CCN(c3ccncc3)C2)=O)C1 c1(OC)ccc(CCC(=O)NC(C)CCNC(=O)C(C)c2ccon2)cn1 c1(CC(=O)NCC(N2CCCCC2)C)ccnn1C C1(NC(C2(C(N(C)C)=O)CC2)=O)CCN(C(C2CC3CCC2C3)=O)CC1(C)C c1(C(N2CCC(OC)(CNC(=O)CSC)CC2)=O)sc2[nH]cnc(=O)c2c1C N1(C(C(=Cc2cc(C)ns2)C)=O)CCc2nc[nH]c2C1c1ccncc1 C1(C(N2C(C(C)NC(=O)CCc3ccccn3)CCC2)=O)COC(C)(C)CO1 c1(CC)cc(C)ccc1NC(=O)C(F)C1CC(NC(c2c[nH]nc2C)=O)C1 N1(C(C(CCC)N(C)C)=O)CCCC(CCNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(c2c(C)nsc2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC12CCC2 CC1CN(C(=O)C(C)(C)C2CCCO2)CCN1C(=O)CSCC(N1CCOCC1)=O C(=O)(C(C)(C)CC(F)(F)F)N.Cc1cc(C(=O)NC2CCCC2C)nn1C(C)C C1(N(C(C(C)=C2CC2)=O)C)CCC(NC(=O)Cc2cc(C)cs2)C1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CN(C(c3cnns3)=O)CC2O)c1 c1(OC)cc(Br)ccc1Cc1cn(C(C2CN(C(=O)COC3CCC3)C2)C)nn1 c1(OC)ccncc1C(=O)NCC#CC(=O)N(CC(O)CF)C C1(CN(C(C(COC)O)=O)C)CCC(CNC(C2CC2C(F)(F)F)=O)CC1.C(C)C C1(C)(OC)CC(NC(=O)CC2CCCC(NC(=O)C(O)CN(C)C)C2)C1(C)C c1(C(=O)NC2CCN(CC(=O)N(CCCC)CC)C2)nc(Cl)sc1Cl N1(C(C(CC)N(C)C)=O)CC(OC)C(NC(=O)CSc2cccc(F)c2)C1 C1(NC(c2c(C)nsc2)=O)CC(C2CCN(C(=O)Cc3cccc(Cl)c3)C2)C1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(c3cnc(C4CC4)o3)=O)C2)nn1 CCCC(CCC)CC(=O)NCC(CO)NC(C1CCC1C(=O)OC)=O CC1CCCCN1NC(=O)C1(c2c(Cl)cccc2Cl)CC1 C1(C(=O)NC(C)Cc2ccsc2)CCCCCN1C(=O)CSC(F)F Cc1cncc(NC(C2(CNC(C3(C)CCSCC3)=O)CC2)=O)c1 C(C)(C)(CC(F)C(=O)N(C1CCN(C)C1)C)NC(c1c(CC)cncc1)=O C1(C(N2CC3C(NC(=O)OCC)C3C2)=O)CC2CCCCC2N1C(c1ccco1)=O C12(NC(c3c(C)nc(NC4CC4)s3)=O)CCCC1N(C(=O)C(C)O)CCC2 C(=O)(C#CC1CCCO1)NC1CCN(C(c2ccnc(C)c2C)=O)CC1 C=CCC(C)(CNC(C1CC(O)CN1C(=O)CCOCCCOC)=O)CO C1(NC(C(Cc2ccc(C)cc2)C)=O)CCSC12CN(C(=O)C(C)CN(C)C)C2 CCCC(CC)CC(=O)NCC1(C)CCN(C(=O)CSc2ccccn2)CC1 c1(SC)cnn(-c2ccccc2)c1NC(=O)NC(C(C)(C)C)c1cnn(C)c1 C(=O)(CC(C)(C)C(F)F)N1CCN(CC(=O)NC(C(C)O)C)CC1 C1(C)(CNC(=O)Nc2sc(C(=O)OC)c(C)n2)CCC(C)C1(C)C C1(N2C(C#C)CCC2)C(=O)NN2CC(CC1C)C2.C1(C(=O)OC)CCOCC1 CCCCCC(O)C(=O)N1CCCC(CCNC(c2c(C3CC3)cnn2C)=O)C1 CCC(CC)CC(=O)N(CCSC)CC.C12CCN(CC1O)C2=O N1(C(C(C)(C)OC)=O)CCC2CC2(NC(c2cc(Cl)ccc2Cl)=O)CC1 C#CCCC(=O)NCCCCNC(=O)C(C)(C)NC(=O)Nc1ccccc1 c1(C(C)C)cc(C(=O)NCC2CC(NC(c3sc(C#N)cc3Cl)=O)C2)cc(O)n1 C(=O)(CCCCCNC(N)=O)N(CCNC(C1(C)CC=CCC1)=O)CCO N1(C(c2[nH]c(=N)sc2)=O)CCCC(NC(=O)C(O)Cc2cnc[nH]2)CC1 C1(CNC(C(C=C)(C)O)=O)CN(C(c2ncoc2CC)=O)C2(CCC2)C1 c1(CC(=O)NC(C(N2CCC(COCC)C2)=O)(C)C2CCC2)ccc(F)cc1 C12(C(=O)NC(CNC(CNC(CCNC(C)=O)=O)=O)C3CC3)CC(C1)C(C)(C)O2 C#CCC(C)C(=O)NCC1CC1CNC(=O)CSCC(c1ccncc1)=O C1(C(N(C(C)C(=O)NCC2SCCS2)C)=O)CCCN1C=O c1(C(=O)NCC2(C(C)NC(=O)CC(C)N(C)C)CC2)cnc(Cl)c(N)c1 C1(C(N(Cc2cn(CCC=C)nn2)O)=O)CC2(C1)C(C(=O)OC(C)(C)C)C2(F)F N#Cc1ccccc1N1CCCC(NC(=O)NC2CSC2)C1 Cc1cc(C(=O)NCC=CCNC(C23CC(CO2)C3)=O)oc1Br C1(=CC(=O)NCCSCC(=O)NCCC2CCSC2)CCOCC1 C1(NC(C(C)CC2CC2)=O)CC12CCN(C(c1cc(C3CC3)on1)=O)C2 c1(CC(N2CC3(C(NC(C(C)C)=O)CCS3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(c2cscc2F)=O)CCCCN1C(c1conc1C1CC1)=O c1(CC(=O)NC23C(CN(C(c4c(C)ccs4)=O)C2)C3)ccc2n[nH]cc2c1 N1(C(c2n(C)cnc2)=O)CC2(CCCN(C(C3CC3c3ccccc3Cl)=O)C2)C1 N1(C(c2cc(C)c(C)s2)=O)CC2COCC2(C(=O)NC2C(=O)OCC2(C)C)C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)C1(C)C c1(C(=O)NCC2(CN(C(C3CCC(CC)C3)=O)C)CC2)cnc(OC)c(C)n1 C1(CNC(=O)COCCO)CCCN(C(=O)CN2CC3CC3C2)C1 c1(OCC(=O)N(C(C)C)CCNC(c2cncc(O)c2)=O)cc(Cl)cc(Cl)c1 C=CCC(C)(O)C(=O)N1CCN(C(C23CCCC2C3(F)F)=O)CC1 N1(C(Cc2n(C)ccc2)=O)C(CC(=O)NCCn2cnccc2=O)C2CCCC12 Cc1ccncc1CC(=O)NCC1(O)CCN(C(c2ccon2)=O)C1 CC(C)CCC(O)C(=O)NC(C1CCCN1C(=O)Cc1ccc(F)cc1F)(C)C c1(Cn2cc(C(C)NC(C3CCC(SCC)CC3)=O)nn2)ccc2c(c1)CCO2 C1(C2CCCN(C(=O)C(O)C3CC3)C2)(NC(c2n(C)c(C(F)(F)F)cn2)=O)CC1 c1(C(=O)NC2C(CNC(C3(O)CC(C)(C)C3)=O)CCC2)ncc(Cl)cc1Cl CC(CS(C)(=O)=O)C(=O)N1CCC(CCNC(c2cncc(C(N)=O)c2)=O)CC1 N1(C(C2C(C)CCS2)=O)CCN(C(c2ccc3[nH]ccc3n2)=O)CC12CC2 c1(C(C(=O)NCCCF)N(CCCC)C)ccc(OCCOC)cc1 C12(C(N(CC)CC3CCCN3C(=O)CSC(C)C)=O)CCCC1C2(F)F C(=O)(C(C)C(O)CC)N1CC(CNC(c2ccc(C(=O)OCC)cc2)=O)OCC1 c1(CC(=O)NC2(C)CN(C(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)cc(F)c1 C12(C(N3C(C(=O)NC)CC3)=O)CCCC1CCN2C(=O)C(n1cc(C)cn1)C N1(C(c2cc(C#N)[nH]c2)=O)CC2CCN(C(=O)CCc3cccc(F)c3F)CC12 N1(C(c2c(C)oc(Br)c2)=O)CCC(O)(CNC(=O)C=C2CCC(C)C2)CC1 C1(O)(C(=O)NC2C(NC(C(=O)NCC)=O)CCC2)CCCC(C)(C)C1 C1(C(=O)NC(C)CCCNC(=O)CCN2CCOCC2)NC(=O)OC1C C(C(C(=O)NC1CC=CC1)NC(=O)CC1CC=CC1)OC(C)C C1(NC(c2cc(OC)ncc2)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1C C=CCC(CC)C(=O)N1CCCCC1CN(C)C(C1CN(C(C)C)C1)=O C1(C2=CCOCC2)(CNc2cc(N3CCCC(c4cc(O)n[nH]4)C3)ncn2)CC1 N1(C(C2NCCN(C(c3c(OC)ccs3)=O)C2)=O)CC(O)C(O)C(O)C1CO c1(C(=O)Nc2ncc(Cl)cc2I)csc2c1CCN(C(c1ccc(Br)cc1)=O)C2 CC1(CNC(C2CCN(c3nncs3)C2)=O)CN(C(c2cnc(O)s2)=O)CCO1 C(CC(C(=O)N1CCOCC1CCC)NC(C1C=CC=CC=C1)=O)=CC N1(C(c2c(C)con2)=O)CCN(C(c2cc(Br)cnc2O)=O)C2CC12 C(=O)(C(F)C(=O)N(C(C)C(=O)NC1C=CC(C(=O)OC)C1)C1CC1)OCC c1(N2CCC(OC)(OC)C2)ccc(S(=O)(=O)NCc2ccn(C(F)F)n2)cc1Cl C(=O)(C1=CCC(C)(C)CC1)NC1CC(C)N(C(c2cc(Cl)cnc2O)=O)CC1 C1(C(N2C(C)(C(=O)OC)CC2)=O)CCCC(NC(=O)CCc2cnco2)CC1 C#CC1(OC)CCN(CCCNC2CC2c2cc(Br)ccc2F)CC1 C1(CCC)CN(C(c2ncoc2C(C)C)=O)CCN1C(C1CC1(F)F)=O N1(C(C(CC)CCOC)=O)CCC2CC(NC(C3CCSC3)=O)CCC2C1 Cn1ncc2c1CN(C(c1csc(NC(c3ccc(O)cc3)=O)n1)=O)CC2 C1(C(N2CCC(C3N(C(=O)OC(C)(C)C)CCCC3)CC2)=O)C2CC(F)(F)CC12 C(=O)(C(C)(C)c1cnsc1)N(CC(O)CNC(=O)C1CC1)C N1(C(c2nc(C#C)sc2)=O)CCCC2(C1)CN(C(=O)CC1(OCC)CC1)CCO2 N1(C(C2CC(C#C)(O)C2)=O)CCC(CCNC(C2(COC)CC2)=O)C(F)(F)CC1 C1(NC(=O)Cc2cc(Cl)ccc2O)CC12CCN(C(C1(Cl)CC1(F)F)=O)CC2 C1(NC(CCC#C)=O)CCCCCC1NC(=O)COc1ccc(F)cc1Br Cc1c(C(N2CC(O)CC2C(N2CCC3(CCOC3)C2)=O)=O)ccc2c1OCO2 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CC(CS(C)(=O)=O)C2)ccc1F C(N=c1nc2c(ncn2C)c(NC(C)Cn2ccnc2)[nH]1)c1cc(C)ns1 CN1CCOC(CNC(C2OCCC2NC(c2nc[nH]n2)=O)=O)C1 CCCCCCCC(=O)N1CC=CC1CNC(c1cc(C)c(F)cn1)=O CCC(C(=O)NC(C(=O)N1CCC1C(C)(C)O)c1ccco1)C(F)(F)F CCCCC(CCC)NC(C1(NC(=O)CN(C)C(=O)OC)CCN(C)C1)=O C(=O)(C(C)(C)CCCF)N1CC(C(NOC)=O)C(CNC)C1 C(CC(C(C)(C)C)NC(=O)Cc1ccc(Cl)cc1)N(C)C(C1CCNC1=O)=O c1(C(=O)NCCCCC(CO)NC(C(C2CC2)OCC)=O)sc([N+](=O)[O-])cc1Cl CC(C)(C)CC(CO)CN=c1[nH]c(=NCCC2CCC2)[nH]c2c1SCC2 N1(C(C(CC)O)=O)CC2CCOC2(CNC(c2c(C(F)(F)F)cccc2F)=O)C1 c1(NC(COC(C)(C)CNC(=O)CN2CCCC2=O)=O)ccc(CCO)cc1 C1(NC(C2CCC(CCC)CC2)=O)CCN(C(c2ncccc2F)=O)CC1F C1(NC(C2CC(=C)C2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)CC12CCC2 CC1(C)COCC1CNC(=O)Cn1cc(CCc2ccc(C(F)(F)F)cc2)nn1 C(C)(C1=NOC2COCC12)NC(=O)NC(C)C(=O)OC(c1ccc(Cl)cc1)C C(=O)(C(CC)(CC)CC)N1CC(CCC)C(C(=O)NC2CCOC2CC)C1 n1(CCC)ncc(C(=O)N(CCNC(=O)C(=O)NC2CC2)CC)c1Cl C1(NC(C2CC(C)(O)C2)=O)CC(CNC(c2cc(F)n[nH]2)=O)C12CCC2 C1(NC(CN(CCOC)C)=O)CC2CCC1CN2C(=O)CCc1cccc(O)n1 C#CCCCC(=O)NCC(C1CC1)NC(=O)Cc1conc1C C1(NC(C2CCC(O)CC2)=O)CC2CC(C1)N(C(c1ccc3sncc3c1)=O)C2 c1(C(N2CCC(NC(C(C(C)C)CO)=O)(CO)CC2)=O)cccc2cncn12 c1(C(=O)NC(C(C)NC(=O)Cc2cc(Br)cs2)C)ccc(Cl)cc1N C12(NC(C3CC(C)(C)C3)=O)CC(C1)N(C(=O)C(=O)NCc1ccc(F)cc1)C2 S(=O)(=O)(c1cnccc1N1CCC(O)CC1)NCC1CCN(C(CC)CC)C1 CC(c1cnn(C)c1)=CC(N1CC(NC(=O)CNS(=O)(=O)C2CC2)CC1C)=O C1(NC(C2(OC)CCSC2)=O)CN(C(C2SCC=C2C)=O)CC1(C)C n1(CC)cnc2c(NC(C)C)[nH]c(=NCCNC(C)(C)COC)nc12 c1(C(N2CCC(COC)(NC(c3csc(C(F)F)n3)=O)C2)=O)cc(C)cnc1C CC(C1CCCc2ccccc21)NC(C1CC1CF)=O c1(N2CCCC(CNC(c3c(C)ncn3C)C3CCC3)C2)nc2ccccc2[nH]1 N1(C(CNC(=O)OC)=O)CC(OC)C(C(=O)NC(CC2CC2)CO)C1 C1(C(=O)NC(C)(C)CNC(N)=O)C2CCCC2CN1C(=O)C=CC1CCOC1 C(C)(C(C(=O)NCc1nccnc1C)NC(=O)CC1CC2CCC1O2)OC N1(C(CNC(CC)=O)=O)CC(C)N(C(c2nc(OC)cc(C)n2)=O)CC1C C1(CCC)CN(C(=O)CC2CC(F)C2)CCN1C(c1cc(COC)cs1)=O N1(C(CCC2(CCC#C)N=N2)=O)CC2CCC2(CCNC(=O)CCCCSC)C1 C1(Nc2ccc(Cl)c(C3CCCN3CC=CC)c2)Cc2cccnc2NC1=O C(C1CCCN1C)=CC(=O)NC(C1CN(C(c2coc(C(F)F)n2)=O)CCO1)C Cc1cc(C(F)(F)F)nc(NC2(CNC(=O)C(C)C3CCCO3)CCC2)n1 c1(C(=O)OC)ccc(Br)c(C(=O)NCCCCc2cccc(Cl)n2)c1 C1(NC(C2(C)CC(C)C2)=O)CC2(C1)CC(CNC(=O)Cc1cncn1C)C2 Cc1oc(C(=O)Nc2ccc(C(n3cc(C(C)O)nn3)C#N)cc2)cc1Br Cc1ccc(C(=O)N(C)Cc2cn(Cc3ccc(Cl)cn3)nn2)c2c1NCCC2 CC(F)(F)CCCC(=O)NCCN1CCN(C(=O)C(C)(C)C2(O)CCC2)CC1 c1(C(=O)NC(CCCC)CNC(=O)C(C)O)c(Cl)nc2sc(C)cn12 c1(C(=O)NC(C2CN(C(=O)C(C)n3cccn3)C2)C)nccc2cc[nH]c12 CC1C(NC(C2CCCC3(CC3)C2)=O)C(C)CCN1C(=O)CCc1cn(C)nn1 C1(NC(C(C)NC(N)=O)=O)CCC12CN(C(=O)CN1CCN(C)C(=O)C1)C2 N1(C(CN(C(=O)CC2CCCCO2)C)=O)Cc2ccc(O)cc2C1 C(c1ccc(F)cc1F)=CC(N1CC2C(NC(C3N(C)CCOC3)=O)(C2)C1)=O CCC(C)C(O)CC(=O)NC(C)C=CC(=O)N(CC(F)(F)CC)C C1(C)(CNC(=NCCC)NCCOC2CCOC2)CCC(F)(F)CC1 c1(OC)cc(F)c(C(=O)NC2CCC(NC(=O)CC34COCC(C3)C4)C2)c(F)c1 n1(C(C(=O)NCCNC(CC2C(C)(C)OCC2)=O)(C)C)cc([N+](=O)[O-])cn1 c1(C(CC)NC(=O)CC2CCCO2)cc(-c2cc(OC)ccc2OC)ccc1F C1(NC(c2cncc(CC)c2)=O)CCN(C(c2cocn2)=O)CC12CCC2 O=C1NCC2(CN(C(=O)CC=CCNC(c3cc[n+]([O-])cc3)=O)C2)N1 c1(CC(N2CC(O)CC(NC(c3cc(C)c(C)s3)=O)C2)=O)ccccc1[N+](=O)[O-] c1(NC(=O)NCc2c(C)ccs2)cc([N+](=O)[O-])ccc1F C1(C(=O)NCc2ccncn2)CCC(C2CC2)N1C(c1ccnc(O)c1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)cc(C)cc2c1OCC2 Cc1ccnc2nc(C(=O)NC(C)C(C3CCCCC3)NC(=O)C(N)=O)nn12 C1(CNC(=O)C(Cl)=CCl)CCN(C(c2cnc(-c3ccco3)s2)=O)C12CCC2 C1(C(N2C(C)(C)CC(c3cn(CCC(F)(F)Cl)nn3)C2)=O)CNc2ccnn2C1 C(=O)(CCCCC(C)=O)NC1CN(C(C(CC)CC)=O)CC1(F)F N1(C(CC2(c3nn[nH]n3)CCC2)=O)CCC2(C=C(C(=O)OC(C)(C)C)C2)C1 n1(CCc2onc(C3CCC(=O)NC3=O)n2)ncc(=O)c2ccccc12 c1(C(=O)NCC2CCC(NC(c3csc(Cl)n3)=O)C2)cnc(O)c2ccccc12 C(=O)(C1CCCc2ccccc21)N1CC(NC(c2nn[nH]c2Cl)=O)CC2(C1)CC2 CC1C(C(=O)NCCCn2nccn2)CCCN1C(=O)C(C)n1cccn1 c1(CCC)cccc(CC(=O)NC2(CO)CN(C(=O)COCCN(C)C)C2)c1 c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)CC2CC(N(C)C)C2)cc1F CC1CN(C(C2CCCCN2N=O)=O)CCCN1C(C1CC(S(C)(=O)=O)C1)=O c1(CC(=O)NC(C(=O)NC(C=C)(C)C)C2CCC2)cccnc1C c1(CC(=O)NCC2(O)CC(NC(c3ccnc(O)c3)=O)C2)nc2c([nH]1)CCCC2 Cc1cc(=NC(=O)C(C2CCCO2)NC(C2SCCS2)=O)[nH]n1C(C)C CC1C(C(=O)NCC2(CN(C)C(c3cnn(C(C)(C)C)c3)=O)CC2)CCN1C c1(C(=O)NC2C(OC)CN(C(c3cc(C(N)=O)no3)=O)C2)nccn2nccc12 c1(C(=O)OCC)[nH]c2ccc(Oc3cn(C)nc3C)cc2c1C c1(C(=O)NC2CN(C(CN(CCOC)C)=O)C(C)(C)C2)ncc(OC)nc1OC c1(C(=O)NCC2N(C(C(C)N3CCC3)=O)CCCC2C)ccnc2nccnc12 c1(OC)c(C(N2CC3CC3(NC(=O)Cn3ccc(C4CC4)n3)C2)=O)csc1Cl N1(C(C2CCCO2)=O)CCN(CCCNC(C2CC2(c2ccccc2)F)=O)CC1 c1(C(=O)NCC2C3CN(C(C(CC4CC4)OC)=O)CC32)ccc(Cl)cc1F C(CCC(=O)N(C(C)C(=O)N(C)C(c1ncccn1)C)C)OC(C)C C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(=O)COCCOCCO)CC1C Cc1cc(C)c(C(=O)NC2CC(NC(C3CCC(C(F)F)CC3)=O)C2)cn1 n1(CC)nc(C2CC2)cc1C(=O)NCC(C)(CO)NC(=O)CCC1CCCOC1 C1(C(N2C(CC(=O)NC(c3ccncc3)C)CCC2)=O)CCCN1C=O C1(NC(CC(C)(C)OC)=O)C(C)(C)C(NC(=O)C(CCO)N(C)C)C1(C)C N1(C(CC2CN(C)C2)=O)CCC2CCCN(C(c3cnsn3)=O)C2C1 Cc1ccc2c(c1)CC(C(=O)NC1CN(C(=O)C(C)(C)CN(C)C)CC13CC3)S2 C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(CCCC)NC(C1CC1(C)C(F)F)=O CCC(C)C(O)C(=O)NC1CC2CC1N(C(c1cnc(C)s1)=O)C2 C1(CC)C(NC(=O)C(C)CC(N)=O)CCCN1C(=O)CC1CC(C)(C)CO1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(COCC)C)=O C1(NC2CN(C(CNS(C)(=O)=O)=O)C2)CCN(C(c2cccnc2)=O)CC1 c1(C(N(C(C)CNC(=O)COCC2CCOCC2)C)=O)cncc2nnn(C)c12 c1(C(=O)NC2(C)CC(NC(C3CCC(C)(CC)O3)=O)C2)cc([N+](=O)[O-])cn1C c1(NC(c2onc(C3(NC(C)=O)CC4(CC4)C3)n2)=O)ccc2c(c1)OCC(=O)N2 C1(C(=O)NCC=CCNC(CN(S(CC)(=O)=O)C)=O)CC(=O)N(OC)C1 N1(CC(=O)NC)CCC2(CCCN(C(c3cnn(C4CC4)c3)=O)C2)C1 N1(C(C2=CC(O)C(NC(C3(C)CCSCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 C=C(C)C(CC(=O)NCCCC1(CNC(=O)C(CC)OC)CCCC1)OCC C=CCCCC(C(=O)NCc1c[nH]nc1C1CC1)NC(C1CC(C2CC2)=NO1)=O c1(C(N2CC(C(C)NC(=O)CC3CC=CCC3)OCC2)=O)ccc2ncsc2c1 C(C(=O)NCC(C)C(C)O)(C(C)(C)O)NC(c1c(C)oc(CO)c1)=O c1(C(=O)NC2CC(C)N(C(c3cnsn3)=O)C2)cc(=O)cc(Cl)[nH]1 CC(C)C(CCC(=O)NCc1nnn(C)n1)NC(=O)C(C)(C)CCC#N C1(NC(=O)C(=O)NC)CCC2(CCN(C(C3CCSC3=O)=O)C2)C1.C12(CC1)CS2 C1(c2nnc(-c3cc(C#N)c[nH]3)o2)(C2CCCO2)CCN(C(=O)CSSC)CC1.CO c1(CCC(=O)N(CCCNC(CC=C)=O)CC)cccc(C(=O)OC)c1 C1(CC=C)(C(=O)NC2CN(C(=O)Cn3nccn3)CC2C(F)F)CCOCC1 N1(C(CC2C(C)CCC2)=O)CC2CCN(C(C34CCOC(C)(C3)C4)=O)C2C1 c1(COC)nc(C)c(C(=O)NCC2CN(C(=O)C(C)SCc3ccccc3)C2)s1 C12(C(=O)NC3CN(C(C4=C(C)CCCC4)=O)CC3C)CC3CC(CC(C3)C1)C2 CC(C)CC(O)C(=O)NCC1CC(CNC(=O)Cc2cccc(C(C)C)c2)C1 C1(C(=O)NC2CCC(C)CC2)CCN(C(C2C3CCCC23)=O)CCC1CO C1(C(=O)NC(C)(CO)C2CCC2)C2CCN(C(=O)CC3CSCCO3)CC12 N1(C(CC=CC)=O)CCC(NC(c2ccc(NC(=O)NC(C)C)cc2)=O)CC1C c1(N(C)C(=O)NCC2OCCC2F)ccccc1F c1(C(N2CCC(N(C(CCCC=C)=O)C)C2)=O)ccc(Br)c(OC)n1 c1(C(=O)NCc2cc(C)nc(C)n2)ccc([N+](=O)[O-])c(C)c1 C(=O)(C1=NNC(C(F)(F)F)C1)NC(CC=C)CNC(C1(OCC)CCSCC1)=O c1(C(=O)NC23CC(CNC(c4ccoc4)=O)(C2)C3)cc2c(F)cc(F)cc2o1 n1(C2CC2)nc(C(=O)NC2CCCC(NC(=O)OC(C)(C)C)C2)cc1C1CCC1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCCN(C)C)CC1O C(=O)(CCC(C)(C)NC(C1C(C)(C)C1(F)F)=O)NC(c1ccccc1)C C#CC1(C(=O)N(C)Cc2ccc(F)cc2)CCN(C(=O)C(C)Cn2cccn2)C1 c1(C(=O)NC2(C)CC(NC(C3(c4ccccc4)CC3)=O)C2)ccc(C2CC2)c(F)c1 N1(C(C2C(C3C(C)C3)C2)=O)CC2CC1CN(C(=O)CN(C)C(c1cccs1)=O)C2 C12COCCN(C1)C(=O)C2.C1(C(C)(C)C)CN(C(c2ccc(CO)o2)=O)CCO1 N1(NC(=O)CCc2cccs2)CCCS(=O)(=O)CC1.c12cn(nn1)CCCC2 N1(C(c2cc(CC)on2)=O)CC(C)C(NC(c2cnn(CCO)c2N)=O)C(C)C1 CN1C(=O)C(c2nnc(-c3ccn(C)n3)o2)Cc2ccccc21 c1(NC(C(=O)OC)C)nc(COc2ccccc2)n[nH]1 C(=O)(CC(C(F)F)NC(C12CCC(C1)OC2C)=O)NCC(C1CCC1)OCC CC(C)CC(C(=O)NC1CC2(C1)CC2C(=O)N(C)CC1CCCS1)C(N)=O c1(CC(=O)NC2CC3CN(C(COCC(=O)OC)=O)C2C3)ccc2nonc2c1 c1(NC(CC2CC3(CN(C(C(C)=CCC)=O)C3)C2)=O)ccc2ncccc2c1 C12(C(=O)NCC3N(C(C4CCOC4)=O)CCC3)COCC1CS(=O)(=O)C2 CCCCC(C)CCC(=O)N1CC=CC1(C)C(N1CCCC(C(C)(C)O)C1)=O C(C(C)C(F)C(=O)NOCc1cccc(C)n1)NC(Cn1ccc(C)c1)=O N1(C(CC2N(C(CC(C)C(F)F)=O)CC2)=O)CCC(F)(F)C(O)C1 N1(Cc2c(OC)nccc2)CCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C(F)C1 C1(CNC(C2CCCC(O)C2)=O)CN(C(c2ncoc2C(F)F)=O)CC1C(F)(F)F N1(C(=O)NCCC)CC(O)CC1c1ccccc1 C(C(=O)NOC1CC1)OCCN(C(C(C)C1CCCC1)=O)C c1(C(=O)OCC)cc(C(=O)NC2CN(C(=O)Cc3ccccc3)CC2F)n(C)c1 c1(NCC2(F)CC(NC(C(C)=C3CC3)=O)C2)ncnc2cccc(C)c12 n1(CCC(=O)N(CCCOC)C(C)C)c(=O)oc2cc(I)ccc12 Cc1noc(CCC(=O)OCC(=O)NCc2ccco2)n1 C1(NC(C(C)OCCC(C)C)=O)CC2CCC1CN2C(=O)C(C)CC(F)(F)F N1(CC(OC)OC)CCCC(CNC(=O)CSCc2ccccc2)C1 CC1=NC(Cl)=CC2=NCCN1N2.c1nc(C2CCCS2)no1 c1(NC(C(CNC(CC2C(C)(C)CCO2)=O)CC2CC2)=O)cccc2c1CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC1CC(C)(NC(=O)CC2(O)COC(C)(C)C2)C1 C1(CCOC)CN(C(=O)C=C=C(C)C)CCN1C(=O)C(C1CCOCC1)F Brc1ccc(C=CCCCN2CCN(C3CCCC3)CC2)cc1 c1(C(C)C(N2CC3CC2C3NC(=O)CCc2cnccn2)=O)ccc(Cl)c(Cl)c1 C1(CNC(C2C(C)OCCC2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 c1(N2CC(CC=C)(NC(=O)C=CS(C)(=O)=O)C2)cncc(C#N)n1 C=CCC(CNC(=O)CCCN(C)C)C(=O)N1CC=CC1(C)COC N1(C(C2(COC)CC=CC2)=O)CCCC(N(C)C(C2(C3CCCO3)CC2)=O)CC1 c1(C(N2CCC(CC)C2CNC(C2CCCCC2O)=O)=O)cccc(F)c1C c1(C(=O)NC2(CNC(c3ccn(C)c3)=O)CCCC2)cn2ccsc2n1 C1(NC(CCC(=O)NC)=O)COCCN(C(C2CC(C)=NO2)=O)C1 C1(C(=O)NCC2CCC(CNC(C3CC(OC)C3)=O)CC2)CC2COCC2C1 c1(C(=O)NC2CC3(C(NC(c4c(N)nccn4)=O)C3)C2)cc(F)cc(F)c1 c1(C(N2C(C3(NC(C(CC#C)(C)C)=O)CC3)CCCC2)=O)cc(F)c(C)cc1F CC(CC(C)(F)F)C(=O)NCC1(C)CCN(C(=O)CCc2cnc(O)[nH]2)CC1 C1(NC(C=C(CCN(C)C)Cl)=O)(CO)CCN(C(=O)C(O)CC2CCCC2)C1 C12(C(=O)NCC(CN(C(C3C(C)CCC3)=O)C)(C)C)CC3CC(C1)CC(C)(C3)C2 CN1CCCCC12CCN(C(c1cccc(NC(C3CCCCC3)=O)c1)=O)CC2 c1(CNC(CCN(C2CCCOC2)CCCCC)=O)ccc(OCC)nc1F c1(OC)nccnc1C(=O)NCC(C)CC(=O)NC(C12CCC(CO1)C2)C C1(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CC2CC(F)C2)C1(C)C C(=O)(CCCCCO)NC1CCC(CNC(CCNC(COC)=O)=O)C1 c1(N2CCCC(CO)CC2)nc2cc[nH]c2c(=NCc2c(F)cc(F)cc2F)[nH]1 N#Cc1ccc(NCCCNC(=O)Cc2nc(F)c(F)cc2F)c([N+](=O)[O-])c1 c1(NCC)ccc(-c2nc(C(=O)Nc3ncco3)ccc2F)cc1[N+](=O)[O-] N1(C(Cc2ccn(C)n2)=O)CCC(C2CCCN(C(=O)C(C)(C)C)CC2)CC1 c1(C(N2CCC(F)(CNC(CCC=C(C)C)=O)C2)=O)cc(F)cc2cccnc12 CS(=O)(=O)C1CSCCN1CCCCOc1ccc(Cl)cc1 N1(C(c2cnc(C3CC3)s2)C(=O)NC2CC2)CCOc2cc([N+](=O)[O-])ccc2C1 C1(F)(C(N(C)C)=O)CCN(C(c2cccc(-c3cccc(CO)c3)c2)=O)C1 c1(C(C(=O)NC(C)C)N(CC)CC2CCOC2)cccc2c1COCC2 CCC(COC)C(=O)NCC(CO)NC(=O)CC1(NC(C)=O)CCCCC1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1C2CCN(C(C(c3cn(C)nc3)=O)=O)C21 N1(C(C(C(C)OC)NC(c2cnn(C3CC3)c2)=O)=O)CCCC(CCF)C1 CCCCC(CC)C(=O)NCC1(C)CCN(C(=O)C(C)(C)C2CC2)C1 N1(CC)CCOCC1C(=O)NCCC(O)C(=O)NCCn1cnccc1=O c1(C(=O)NCCCCCNC(C(COC)(C)OC)=O)cnc2nc(C)oc2c1 c1(-c2c(OC)cccc2)nc(=NC2CC(NC(=O)C3=CC4(CCOC4)C3)C2)s[nH]1 C1(c2ccccc2)(N(C(c2cn(C)nn2)=O)CC)CCN(C(=O)C(C)C#N)CC1 c1(CC)nccnc1C(=O)NCC(c1ccccc1)NC(=O)C(F)CC N1(C(c2cc(COC)no2)C(=O)NCCCF)CCNC(=O)CC12CCC2 Cc1cccc(N2CCC(OC(=O)CC3CC(C)OC3C)C2=O)c1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCC(NC(=O)CCC2CCCCC2)C1 C1(CN=[N+]=[N-])CCCN(C(C2CCCCN2C(=O)C=CC2CCCC2)=O)C1 CN1CC(C)(C(N2CC(C)(NC(c3ccc(Cl)c(F)c3F)=O)C2)=O)CCC1=O CON(CCCO)C(=O)C1(NC(=O)COCC(C)(C)C)CC1(C)C c1(C(N2C(C)(C(=O)OC)CC2)=O)[nH]c(C)c(C(=O)NCCCn2ccnc2)c1C N1(C(c2c(CC)con2)=O)CCC(C)N(C(c2conc2C)=O)CC1 Cc1cn2c(C(=O)NCCC3COCCN3C(c3cnn(C)c3C)=O)cnc2s1 N1(C(Cn2c(C)cc(C)n2)=O)CCCC12CCN(C(C1CCCN1C(C)C)=O)C2 C1(NC(C(=O)Nc2ccc(N(C)C)nc2)=O)CCC2(CC1)OCc1ccccc12 Cc1cc(C(=O)NCC2(CNC(C3CCS(=O)(=O)C3(C)C)=O)CC2)c(N)c(F)c1 N1(C(C=CC=CC)=O)CC(C(=O)Nc2ccc(C(F)(F)F)nc2)CC(F)C1 c1(C(=O)NC2CCC2CNC(=O)C(O)c2ccsc2)ccccc1N1CCCC1 N1(C(C(CCCC=C)NC(=O)C(C)CC(=O)OC)=O)CCc2oc(C)nc2C1 Cn1cc(C(=O)NCC(CNC(c2cccn2C2CCCC2)=O)CO)nn1 c1(C(N2CCOCC(C)(CN)C2)=O)ccc2cccc([N+](=O)[O-])c2n1 N1(C(C2C(C=C)CC2)=O)CCCC(CCNC(=O)CN(CCOC)CC)C1 C(=O)(CCCCCC#N)NCC1(Cn2cc(C(CC)OC)nn2)CCOCC1 C1(C(=O)NCCCCSC)N(C(C2CCC(F)(F)C2)=O)CCC1(C)C CC1(C)CC(Nc2ccc([N+](=O)[O-])cc2)CN(C(c2ccc3scnc3c2)=O)C1 N1(C(=O)NCCn2cc(-c3ccc(Cl)s3)nn2)CCOC(C(F)(F)F)CC1 N1(C(C(CC(=O)OC(C)(C)C)NC(=O)C2CC2)=O)CC(NC(N)=O)C2CCCC12 C(=O)(CCC(=O)N1CCC(C(C)NC(=O)Cn2cnnn2)C1)Nc1nnc(C)s1 c1(CC)ccc(F)cc1NC(C12CC(CO)(CN1C(C1CN(C3COC3)C1)=O)C2)=O c1(C(=O)NCC(CC)NC(C2(C#N)CC3CC3C2)=O)c(F)ccc(C)c1F c1(C(c2n(CCCC)nnn2)(C)NC23CC=CC(C2)OC3)c(F)cccc1F c1(NC(=O)OCC)nnc(S(=O)(=O)N2CCN(C(c3nc(C)c(C)o3)=O)CC2)s1 CCC(CC)C(C(=O)N1CC(NC(c2nc(O)c(C)s2)=O)C(C)(C)C1)OC c1(C(C(C)NC(C(CC)O)=O)OC)cccc(Br)c1 c12ccc(C)cc1CC1CN(C1)C2=O.C12(NC(C3(SC)CC3)=O)CC(C)(CO1)C2 C(C(C(C)(C)C)NC(C1NC(=O)CC1C)=O)NC(C1C(C)(C(C)C)C1)=O CCCCC(CC)CCCN(C)C(=O)NC(c1cccs1)CN1CCOCC1 N1(C(C2CCCN(CC(C)=CC)C2)=O)CCCN(Cc2ccc(F)nc2F)CC1 c1(C(C)C)ccc(C(N2CC(N(C(=O)Cc3nc[nH]n3)C)C2)=O)cc1Br c1(C(N2C(C(=O)NCCc3n(C)cnc3)C=CC2)=O)cccc(CO)c1 N1(C(C(C)(CO)OC)=O)CCOCC(C)(CNC(=O)C=Cc2ccnn2C)C1 c1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)occ2c1CCC2 c1(C(N2CC(NC(=O)CCc3nc(O)n[nH]3)C2)=O)cc2c(o1)CCCNC2=O c1(C(=O)NCCOCCNC(CC(=O)NCC#C)=O)ccc(C(F)F)cc1 N1(C(C2CC(CC)(CC)C2)=O)CCC(CNC(c2cc(Cl)ccc2N)=O)CC1C c1(C(N(C(C(C)C)C2CCC2)Cc2nnnn2C2CC2)=O)cccc(SC)c1.CO c1(C2(C(=O)NCC(C)N(C(=O)COC3CC3)C)CCCC2)ccc([N+](=O)[O-])cc1 C1(C(N(C(C)CCNC(c2cnc(S)[nH]2)=O)C)=O)CC2(C1)CC(O)C2 C1(CC(=O)N(C)CC2CCCN(C(=O)CCS(C)=O)C2)CC2CCC(C1)C2 C(CC(=O)NN1CCCC1C(=O)NCC1CCN(C(C)C)C1)OC(C)C C(=O)(C(CC(C)C)NC(=O)CC(C)N(C)C(c1cc(F)n(C)n1)=O)NC c1(C(=O)NC(C)CCCCNC(c2cc(Br)no2)=O)cccn2cnnc12 C(=O)(CC(CC)CCC)NCC(CNC(c1cnc(CCCC)s1)=O)C N1(C(C(C2CC2)OCC)=O)CCCN(C(=O)C(C)C(C)C)CCNC1 CCC(CC1CCCC1)C(=O)NCC1CC1NC(c1ccnc(OCCO)c1)=O c1(C(=O)NCC2C(NC(c3cc(OC)nn3C)=O)COC2)cnc2n1CCS2 CCC(CC)C(C(=O)NCC1CCN1C(c1sccc1C#N)=O)OC N1(C(N2C(C)C(N3CCOCC3)CC2)=O)CCC(S(=O)(=O)c2ccccc2)C1 C1(CC)CCCCC1C(N1CCC(C(C)(C)C)(CNC(=O)C(C)CSC)C1)=O C(CC(CNC(=O)CC1CNC(=O)C1)NC(=O)Cc1csc(C(C)C)n1)OC N1(C(c2c(Nc3c(Br)cnc(C)n3)cccn2)=O)CCC2COCC2C1 N1(C(C2=CC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)Cc1cnc2cccnn12 C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 CCCCCCCC(=O)N(C)CC1CCCCN1C(C1CC(=O)CCO1)=O c1(OCC)ccc2c(c1)CC(C(=O)NCC#CCNC(=O)C(C)(CC)OC)CO2 C1(C(=O)NCC(c2ccccc2)(C)C)CCC(Cn2ccnc2)C1 c1(C(=O)NC2(CNC(c3cc(CC)[nH]n3)=O)CCCCC2)ccc2nn[nH]c2c1 c1(C(C(=O)NC)N(C(CC(=O)OCC)C2CCCCC2)C)ccc2ncsc2c1 C(=O)(C#CC1CCCOC1)N1C(CNC(C2(CCCC)CC2)=O)COCC1 N1(C(CCc2n(C)ccc2)=O)CC(O)CCC1C(=O)NCC1OC(=O)CC1(C)C N1(C(C(COC)O)=O)CCn2ncc(CNC(c3cc(Cl)ccc3Cl)=O)c2C1 C1(C(=O)NC(C2CN(C(=O)Cc3ccc(CO)cc3)C2)C)CCCC(C(N)=O)C1 CC1(C)CC1(C#N)CNC(C1(n2cc(Br)nn2)CC1)=O C1(C(N2CCC(F)(CNC(CP(C)(C)=O)=O)C2)=O)CCCCC12OCCO2 c1(CCC)cc(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)n(C)n1 O=C1NC(C(=O)NC2(CCO)CN(C(c3sccc3F)=O)C2)Cc2n[nH]cc21 CCC(CCO)C(C)NC(=O)NC1C2CCOC2C1(C)C O=C(C1=CCCCCC1)N1CC(C(=O)NCc2ccoc2)C2(CCC2)C1 N1(C(C2C(C)CCCC2)=O)CCC(C)C(CNC(C2CCC3CC3C2)=O)C1 c1(C(N2C(C)(C(N(C3CCCCC3)CC)=O)CCC2)=O)cccc(Br)c1O c1(C(N(CCNC(C2CC(C)(F)C2)=O)CC)=O)ccc(NC)c(F)c1 c1(OC)ccc(Br)c(CN2CC(CNC(=O)CCc3ccccc3)C2)c1F c1(NC(CC2(NC(CNC(CCNC(=O)NC)=O)=O)CC2)=O)cnc(C)cn1 O=C(CC1CCOc2ccccc21)NCC1(c2ccccc2)CC1(F)F C1(CC)CCC(C(=O)NC(C)C=CC(=O)NCC2(C3CC3)CC2)O1 CN1C2CCC1CN(CCNC(=O)CC1CC3CC1C1CC31)CC2 CC1=CCN(C(C2(NC(=O)CC3CCCC3C)CC(F)(F)C2)=O)CC1 C1(NC(C(C)Sc2ccc(Cl)cc2)=O)CCOC(C)(C)C1 c1(C(=O)NCCC(=C)CNC(c2ccc(C)n2C)=O)c(Cl)cc(C#N)cc1Cl N1(C(=O)Cc2cnsc2)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)cc1F)C2 N1(C(c2cn(CC=C)nn2)=O)CCC(NC(c2sccc2F)=O)C12CC2 c1(NC)cnc(Cl)cc1C(N1CC2CC1C2NC(=O)COc1ccc(O)cc1)=O c1(NCC(S(=O)(=O)NC)C)ncccc1S(=O)(=O)N(C)Cc1csc(C2CC2)n1 C1(CC)CCCN(C(C2CC(O)CN2C)=O)C1C(=O)N(C)CC1CCN(C)C1 N1(C(C)Cc2ccccc2)CCN(Cc2cc(C(C)(C)O)on2)CC1 C(=O)(C1CCCc2c1ncn2C)N1CC(CNC(CCOC)=O)CC12CCC2 c1(C(=O)NCC2(F)CC(NC(C(=O)NCCNC(C)=O)=O)C2)cnc(O)c(F)c1 O=C1NC2(CCN(C(c3cc(O)cc(F)c3)=O)CC2)Nc2ccccc21 c1(OC)ccc2[nH]c(=O)c(C(=O)NCCc3cc(C)sc3C)cc2c1 c1(NC2CC(F)(CNC(=O)Cn3ccc([N+](=O)[O-])n3)C2)ncnc2c1CCO2 C1(CNC(=O)CCn2cccc2)CCC2(CCC2)C1NC(=O)C(Cl)=CCl C1(NC(CCOCC(C)C)=O)C=CCC(C(=O)N(CCCC(O)CO)C)C1 n1(CC(=O)NCC2CC(C(=O)NCCC(C=C)C)C2)cnc(C#N)n1 CC(CCCNC(=O)CCN(C)CCO)NC(=O)CC1CCSC1 N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(=O)Nc1cccc(Br)c1)=O N1(C(C(CC)C(C)C)=O)CCC2(CC1)CC(NC(C1CC1(C)Br)=O)C2 C1(C#N)(C(N2CC(C)(NC(Cc3c(C)cnn3C)=O)C2)=O)CCOCC1 c1(CC)ccc(C(=O)NC2CC(NC(c3nc(C)ncc3Br)=O)C2)c(OC)c1 O=C(C(Cc1cccc(Cl)c1)CCCCCO)OCc1noc(-c2ccsc2)n1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)N(CC(=O)O)C1CCC1 N1(C(c2c(CC)c[nH]n2)=O)CCOCC(NC(c2oc(C3CCC3)nc2C)=O)C1 C(=O)(C(C)C(C)NC(=O)CCOC)N(CC=C)C c1(C(=O)NCC(CCC)NC(=O)CC2OCCC2(C)C)cc(C(C)C)nn1C C1(CCNC(=O)C(C)N(C)CC2CCCC2)(OC)CN(C(=O)CC2CCCO2)C1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCN(C(C(CC)c2cccnc2)=O)CC1 C1(NC(C(C)OC2CCOC2)=O)CC(NC(=O)C(C)Cc2ccncc2)CC1O c1(C(=O)NC(=O)OCC=C)ccc(C2(F)COC2)cc1 c1(C(N(C)CC2N(C(CCCC)=O)CCC2)=O)c(F)ccc(C)c1Cl N1(C(C(CC(=C)Cl)NC(C2CCC(C)CC2)=O)=O)CCC2(CCC(O)C2)C1 C1(NC(c2c(CNC(C(C)CC#N)=O)nccc2)=O)CC12CCCCCC2 N1(C(C2(OC)CCOCC2)=O)CCOCC(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1ccc(Br)c(C(N2C3CCC(C(=O)NC(C)(C)C)C2CC3)=O)c1F c1(C(C)(C)C)ccc(Br)cc1NC(C1C=CCN1C(=O)Nc1cccnc1)=O Cc1nc(O)ccc1C(=O)NC(C)(C)CN(C(=O)CC1C=NN(C)C1=O)C c1(N2CC(COC)OCC2)nc(=NC(C)CCO)[nH]c2c1ncn2CC Cc1cc(C(=O)NC2(C3CCN(C(=O)C(C)N(C)C)C3)CC2)c(Cl)cc1Cl C(N=C(NC(CC)CC)NC1CCN(S(=O)(=O)C(F)F)C1)c1nc(CC)oc1 CCC(C)CCCCC(=O)N1CCCC(Cc2cn(Cc3cnns3)nn2)C1 CCC(CCOC)C(=O)N1CC(n2cc(C(C)(C)C(=O)OC(C)(C)C)nn2)CO1 c1(CNC(C2CCN(C(=O)Cc3cncnc3O)C2)=O)ccc(Cl)cn1 N1(C(c2cn(C)c(O)n2)=O)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC12 CC1CN(C(c2cccc(Cn3cc(COCCO)nn3)c2)=O)CC(C)(C)C1 N1(C(C2(N(C(C3(C(CC)=O)CC3)=O)C3CC3)CC(O)C2)=O)CCCC(C)(C)C1C C1(C(=O)NCC23CCCC2C3)CN(C(C2CC3(CC3)CO2)=O)C2(CCC2)C1 c1(C(N(C2CCC2)CC)=O)cnc2c(c1)CCN(Cc1cnc(OC)c(Cl)c1)C2 c1(CC)ncccc1C(=O)NC1(CCCC)CC1.C1C(=O)NCCO1 c1(C(N2C3CC(CNC(c4c[nH]c(=O)o4)=O)C(C3)C2)=O)n[nH]c2ccc(F)cc12 N1(C(CN2CCN(CC)CC2)=O)CCN(C(c2cc(OC)cc(F)c2)=O)C(C)C1 c1(C(=O)NCC(C2CCCCC2)NC(=O)CCF)sccc1Cl N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(=O)CN2CCCCC2=O)C2CCCC12 Cc1nccn1CC(=O)N(C)CCNC(=O)Cc1nncn1C C(=O)(C(CNC(=O)CCc1cn[nH]c1)N(C)C)NC(C1CCOCC1)C#C NS(=O)(=O)C1(C(=O)NC2CCN(C(=O)CCCCc3cnc[nH]3)CC2)CCC1 c1(C(=O)NC2CC(NC(c3nc(C(C)(C)C)oc3)=O)C2)ncc(Br)cc1N Cc1cc(C)n2nc(C(=O)N(C)Cc3cn(CC4CCCCC4O)nn3)nc2n1 c1(C(N(C2CCCN(c3ccccn3)C2)C)=O)n[nH]c2cccnc12 c1(C(=O)NCC2CC(NC(=O)CC3CC3(Cl)Cl)C2)cccc2c1CCO2 c1(C(N2CCCC(NC(CC(C(C)C)O)=O)CC2)=O)cnc2ccnn2c1 C1(=O)CCCCCC(c2nnnn2C)N1.C(C1CCCc2n[nH]cc21)c1n(C)nnn1 N1(C(CCc2cccc(OC)n2)=O)CC2CC(NC(=O)Cn3cccn3)CC1C2 C#Cc1ccnc(CN(C(=O)C(CN2CCCC2)c2ccccc2)C)c1 Cc1cc(CNC(C2C=CCS2)=O)oc1C(N1CCC(c2ncc[nH]2)C1)=O C12(CNC(CC3CCN(C)C3=O)=O)CCCC(CN(C(=O)Cc3cnns3)C1)C2 C1(CNC(c2cc(C)on2)=O)CN(C(c2ccc(S(N)(=O)=O)o2)=O)CCC1(C)C CCCC(C)(O)C(=O)N1CCC(C)(CNC(c2cc(F)ccc2C(C)C)=O)C1 C=Cc1cc(C(=O)N(C2CCCCN(C(=O)C3=CCCCC3C)C2)C)cc(F)c1 CC(C)CC(C(=O)C(=O)CC1CC2(CC2)C1)NC(N)=O.C1(C(=O)NCCNC)CC1C CC(C)C(O)CC(=O)NC(C)CC(=O)N(C)CCn1cncn1 C1(C(=O)OC)C(C)OCCN1C(c1cccc(-c2cc(F)ccc2F)c1)=O C12(CNC(N3CCCCC3)C)CCC(CC1)N2C(=O)OC(C)(C)C CCC(C)(F)C(=O)N1CCC(NC(=O)Cn2cc(-c3ccccc3)nn2)C1 C1(CC(C)NC(CC(=C)C)=O)CC2CCC(C1)N2C(=O)CSc1ccc(C)cc1 Cc1[nH]c2cccnc2c1CNC1CCN(CCC(C)C)CC1 N1(C(C=Cc2c(C)nccc2)=O)CCC2(CC1)CN(C(C1CC3(CCC3)C1)=O)C2 N1(C(C(C2CCCOC2)OC)=O)CC(F)(F)CC1Cn1cc(Cc2cccs2)nn1 C(=O)(CCCCCN(C(=O)CC1(OCC)CC1)C)N1C(CCC)CCC1 Cc1cc(C(=O)NC2CN(C(C3CCCSC3)=O)C(C)(C)C2)c(O)nc1C C1(NC(C2C(CN(C)C)C2)=O)COCCC1NC(c1ccc(F)cc1)=O C12(C(=O)NC(C)(CNC(c3cnco3)=O)C3CCC3)CC(CC(F)(F)F)(C1)C2 c1(C(=O)Nc2ccc(-c3cccc(O)c3)cn2)c[nH]c2cc(Cl)ccc12 c1(C(N2C3(CNC(C4CCC5CC45)=O)CCC2CC3)=O)ccc2c(c1)CCCS2 c1(NCc2c(CNC(=O)Nc3ccc(Br)cc3)[nH]nn2)ccc(C(F)(F)F)cc1Cl c1(CNC(CC(CC)CN(C)C)=O)cc2n(n1)CCN(C(=O)COCCOC)C2 C=CC(C)(CC)C(=O)NC1CCN(C(c2cnn(C)c2C(C)(F)F)=O)C1 C1(C)(C(=O)NCC(CNC(=O)C(c2cnccc2C)(C)C)OC)CC2CC2C1 N12c3ccccc3CC1OC2=O.N1(C(C)(C)C)CCC(O)C(Cn2ccnc2)C1 C(C(C)(C)CNC(c1cnc(-c2ccco2)s1)=O)NC(C(=O)NCC)=O C(CC(C)(C)C(=O)NCC(CO)NC(c1cccc(-c2nc(=O)o[nH]2)c1)=O)OC N1(C(c2n(CC)ccn2)=O)CC(=O)N2CCCC2C1 C12(CNC(c3c(C)cnn3C)=O)CCC(CC1)N(C(=O)C(CN(C)C)N(C)C)C2 N1C2C(=O)NCCCN2CC1=O.N1(C(C)C)CCCC(c2cccc(F)c2)C1 S1(=O)(=O)c2ccc(s2)CN(C)C(=O)C2CN1CCC2O.c1noc(C)n1.CO C(=O)(N(C)OC(F)F)C1CC(NC)C1.c1(CC2CC(CC=O)C2)ccccc1 CC1CC(CNC(C2(C(F)F)CCCO2)=O)CCN1C(c1ccc(Cl)nc1N)=O N1(C(Cc2c(C)ccs2)=O)CCC(F)CC1C(=O)NCc1cccc(F)c1 C1(NC(N2CCCC(COc3cnccn3)C2)=O)CCCC1(F)F N1(C(C=CC=CCC)=O)CC2(CCCC2NC(C2Cc3nnc(C)n3C2)=O)C1 C1(CC=C)(NC(=O)C=CC2CC2)CN(C(c2cnccn2)=O)C1 c1(C(=O)NC(CC)C(c2cc(Cl)ccc2Cl)O)ccc(-c2ccco2)nc1O N1(C(CN(C(=O)C(C)CC#N)CC)=O)CCCOC(C(C)C)C1 c1(C(=O)NCCCC(CCO)C(=O)O)cccc2cc(F)ccc12 C(=O)(C(C)CC(C)C(C)=O)NC(COCC)C(=O)NCc1coc(C)c1 c1(C(=O)NCC2CCCCN2C(C2CC2F)=O)cccc2c1NCCNC2=O C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(=O)Cc2ccccc2O)C1(C)C c1(CCNC(C2NCCC(CC)C2)=O)cc(Cl)c(OC)cc1Cl C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)CC2CNC(=O)C2)CC1(C)C N1(C(CN(C2CCSC2)C)=O)C2CCC1CC(NC(c1ccccc1S(C)=O)=O)C2 C1(N(CCC)C(C2CC3CC(C2)C3)=O)CCN(C(=O)C(C)SC(C)C)O1 C(=O)(C(F)C(F)(F)F)N1C(CNC(C(C=C)C)=O)CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(CC(C=C)(C)C)=O)C1 N1(C(C(N)=O)=O)CCC(F)(F)C(CNC(=O)Cc2cc(C(F)(F)F)cc(Cl)n2)C1 N(C1CCCc2ccoc21)C(C(CN(C)C)NC(c1ccc(C#C)nc1)=O)=O O=C(C1=CCCOCC1)NC1CC(NC(c2ccc3c[nH]nc3c2)=O)C12CCC2 c1(C(=O)NCCN(C(c2cc(CCCCC)[nH]n2)=O)CC2CC2)nc(C)oc1OC N1(C(C2(O)CCC(C)CC2)=O)CCCC(C2CC2NC(C2CC2(C)Br)=O)C1 Cc1nnc2c(C(=O)NC3COCC3NC(C3CCOC(C)(C)C3)=O)cccn12 c1(C(=O)NC2CN(C(=O)Nc3ccc(C)cc3)CC2F)ccc([N+](=O)[O-])cc1F c1(OC)c(C(=O)NC2C3CC2N(C(c2ccc(C4CC4)cc2)=O)C3)cccc1Cl Cc1ccccc1C(C)(C)C(=O)NC(C)CN(C)C(C1CCN(C)C1)=O N1(C(COCCCC(C)C)=O)CCOC2CCN(C(c3cccc(=O)o3)=O)CC12 c1(OC2CCN(C(c3cn(CC)nc3)C(=O)NCCC#N)C2)c(F)cccc1F Cc1cn2c(CC(N3CCOC(C(=O)NC4(c5cnn[nH]5)CC4)C3)=O)csc2n1 C(=O)(C(C)(C)CNc1cc(C)sc1C)NC(C(CO)SC)C C(CO)(C(C)(C)CO)NC(C(CSC)(C)NC(c1cncnc1C)=O)=O CCC(CC)CCCC(=O)NCC1CCC(C(=O)NOCc2ccncc2F)O1 N1(C(C(C(CC)C)c2ccccc2)=O)CC2CCN(C(C3(CF)CC3)=O)CC2C1 c1(C(=O)NC(CC)CNC(=O)CCC#N)ccc(C2CCC(=O)N2)cc1 CC(C)C(O)C(C)C(=O)NC1CC(C(=O)NCC(F)(F)C(F)F)CC1O CCCCS(=O)(=O)CC(=O)NC1CC12CC(NC(=O)CNC(=O)NC)C2 C1(NC(C(c2cnn(C)c2)NC(CCN(C)CC)=O)=O)CC=C(C)CC1 C(=O)(CCCCCc1nn[nH]n1)NC1CCN(CCOC)C1 c1(C(=O)NC2CC(C)(CNC(c3nscc3Br)=O)C2)coc(C#N)c1 c1(CCC(=O)Nc2ccc(-c3cnc(C4CC4)nc3)nc2)ccc2c(c1)OCO2 CC1CCC(NC(C2CCCC(O)C2)=O)N(C(=O)CC2CCN(CCF)CC2)C1 c1(C(=O)NCCN(CCC)C(C2(C)CCC(C)(C)CC2)=O)cnc2ncccn12 CC1CN(C(=O)CCc2cscn2)CC1CNC(c1cccc(C2CC2)c1)=O CC(CC(=O)OCC1(Oc2ccccc2)CC1)CC(F)(F)F c1(N(C)CC2(C)CCCO2)nc(=N)[nH]c(=NC2CC2c2ccn(C)n2)[nH]1 c1(CCNC(C2(CC)CC2)=O)cncc(C(=O)NCC2=NOC(C)C2)c1 C1(NC(C2N(C)CCCC2)=O)CN(C(=O)C(C)(C)O)Cc2ccnn2C1 C1(NC(C2C(c3c(C)c(Br)ccc3)C2)=O)CCC2(CC1)CNC(=O)C2 N1(C(C2N(C)C(=O)OC2)=O)CCC(C)(C)C1CC(=O)NCC1CC12CCCCC2 N1(C(CN2CCC(C(C)=O)CC2)=O)CCC(NC(C2CC2C2CC2)=O)C(C)(C)C1 C1(CC(N2CC(C(C(=O)N(CC(=O)NC(C)(C)C)C)O)C2)=O)CC(C2CC2)C1 c1(-c2cccc(OC)c2C)ccc2cc(C(N3CCC(C)C3)=O)cn2c1 C1(C(N2CC3C(CNC(c4c(OC)c[nH]n4)=O)(C3)C2)=O)CS(=O)(=O)CCO1 C1(NC(CSCC#C)=O)CN(C(=O)CCSc2ccccn2)C2CCCC12 c1(CC)ccc2ccccc2c1CNC(=O)Cc1ccc(O)cn1 N1(C(C2=CC(C)(C)C2)=O)CCC2(CC2)CC1C(=O)NC(Cc1ccco1)CO CCCC(O)(CCC)CC(=O)NC1(C)CCN(C(c2conc2COC)=O)C1 Cc1nc(O)ccc1C(N1CCCC(N(C)C(C2CC3(CCC3O)C2)=O)C1)=O C1(C(N2C(CCNC(c3c(C(C)(C)C)ocn3)=O)CCC2)=O)CC2(C1)CC2(F)F C1(NC(C2C3CCCC23)=O)CCN(C(=O)Cc2ccco2)C12CCC2 c1(OC)c(C(=O)NC(C)CC2CN(C(=O)CC(O)C(C)C)C2)cccc1Cl n1(CC)cnc2c(NCC3(Cl)CC3(F)F)[nH]c(=NCCCc3cccnc3)nc12 O(P(C)(=O)CNC(C1CC(C)CN1C(=O)CCC1CCOC1)=O)CC N1(C(CCC(C)C)=O)Cc2ccccc2C(NC(C2CCC=CCCC2)=O)C1 N1(c2cc(NCCCOCCOC)nc(C)n2)CCc2ncnc(C)c2C1 n1(C(C)C)nncc1C(=O)NCC1CCN(C(=O)C=CC2CCCC2)C1 C(=O)(CC(O)CC(C)(C)C)N1CC2C(CNC(c3n[nH]c(CC)c3Cl)=O)(C2)C1 C1(C(=O)Nc2c(CC)cccc2)CCN(C(=O)CCCCCNC(C)=O)C(C)C1 N1(C(C2N(CCC)CCC2)=O)C2CCC1C(CNC(c1ccncc1F)=O)C2 CCC(C)(C)C(O)C(=O)NCc1cc[nH]c1C(=O)N(C)CC12CCC(CC1)C2 CC1CN=C(NCCF)NCc2ccc(cc2)O1.c1(NS(C)(=O)=O)ncccc1F CC1CN(C(C2CN(C(c3cccnn3)=O)CC2C)=O)CC(C2CC2)O1 N1(C(C2CC(OC)C2)=O)CCCCC1CN(C(=O)CCCOC)C C(CC(C)C(=O)NC12CC(C(N3CCSCC3C)=O)(C1)C2)=CCC c1(CNC(C(CCC)CC2CCCC2)=O)cc(F)c(C(=O)O)c(F)c1 C(CNC(C1CCN(C(=O)C(C)C)CC1)=O)(C(C)C(C)C)NC(CCOCC)=O c1(C(=O)NC(CNC(COC)=O)C(C)C)ccc(O)cc1F C(=O)(CCCCCN(C(=O)C=CC1CCOCC1)C)NC(C=C)C(F)(F)F c1(C(N2C(CNC(C=CC(=O)OCCCC)=O)CCC2)=O)cccc(C#N)c1 S(=O)(=O)(c1cccc(Cl)c1F)N1CC(OC)C(NC(C2CCCCO2)=O)CC1 N1(CC)CCC(NC(C2CCN(C(=O)CCc3nc(C)no3)CC2)=O)C1=O C1(C(N2CC(CC(=O)OC)C2)=O)CCCC1CNC(C1CCSC1)=O Cc1c(CC(=O)NC(C)C(C)NC(c2ncn(C)n2)=O)ncn1C N1(C(c2c(C)scn2)=O)CCCCC(CNC(c2ccc(=N)[nH]n2)=O)C1 n12cc(nn1)NC(=O)C2.C1(C(CC(N)=O)NC(CC2CN(C)C2)=O)CCCCC1 C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C)n(C)c1)=O)CC c1(COCC)cccc(OCCOCc2[nH]cnc2C)c1 CCC(CC)C(F)C(=O)N(C1(CC(=O)N(C2COCC2(C)C)C)CC1)C N1(C(C2C(NCc3c(Br)ccc(C#N)c3)C2)=O)CCc2cc(F)ccc2C1 CC(CC(=O)NCC1CCC(F)(CNC(C2(C#N)CC2)=O)CC1)CC(C)(C)C CN1CC2CCC(C1)N2C(c1c(O)ccc(F)c1F)C(=O)OC1CCCCC1 C1(CC)(NC(c2ccoc2C)=O)CCN(C(c2cccc(N)c2N)=O)CC1 N1(C(c2cc(C)ns2)=O)CC(NC(c2ccc3scnc3c2)=O)CC12CCOC2 N1(C(C(CC=C)CNC(C2CC2OC(C)=O)=O)=O)CCC(C)(O)C(O)C1 C12(NC(CC(C(C)C)OCC)=O)CC3CCC(C1C2)N3C(c1ccc(Cl)s1)=O Cc1ccc(N(C)C(C2CCN(C(c3cnc(O)o3)=O)C23CC3)=O)cc1F C12(C(N3CCC(=CCNC(c4c(C)nco4)=O)CC3)=O)CCC(C)(CC1)OC2 N12CCOC(C1)C(=O)N1CC3C(C3C1)CC2=O.C12(CC)CCCC1C2 c1(C(=O)NC(C(=O)NCCOCCC)Cn2cccn2)cncnc1C C1(NC(C23N(C(c4cccc(C)c4O)=O)CC(C2)C3)=O)CCN2CCCC2C1 N1(C(COCC)=O)CC2CCC1C(NC(c1ccc(OC(C)C)cc1Cl)=O)C2 C(N=c1[nH]cnc(Cl)c1C#N)C1(O)CN(C(c2n(C)nc(C(F)(F)F)n2)=O)C1 CP(C)(=O)c1cccc(NC(=O)C(=O)NC2CC3CCC2CC3)c1 N1(C(C(C)CC(F)(F)F)=O)CCC2CN(C(c3cc(O)cc(O)n3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CC2COCCO2)C)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)CC(F)(F)CCC1(C)C N1(C2(NC(=O)CO)CC(NC(C3N(N=O)CCCC3)=O)C2)CCCCCCC1=O N1(C(CC(c2ccc(OC)cc2)N)=O)CCC(O)C(NC(=O)CCCC(N)=O)C1 N1(C(C(=O)NCCCC)C)CCCC(NC(c2cc3occc3s2)=O)CC1 Cc1nc(-c2ccccc2)sc1C(=O)NC(C)CNC(=O)COc1cnn(C)c1 c1(C(=O)NCCC(C)N(C(COCC=C)=O)C)cnc(OCC)c(C)c1 CC(CC(=O)N1CC(CNC(c2ccc(C3CC3)nc2O)=O)CC1C)C(F)(F)F C(=O)(C(C(C)(C)C)OC)N(C)Cc1c(CNC(C2C(CCC)C2)=O)cccc1 c1(NC(CNC(C2C(CCC)CCC2)=O)=O)cn(CC)nc1C#N C(=O)(CCCc1cc[nH]n1)NCC(CNC(CN(C1CCC1)C)=O)O C1(NC(c2coc(Br)n2)=O)CC2(CCCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 c1(C2C(C(=O)N(CCOCCO)CCOCCO)C2)ccccc1F C1(O)(C(C(=O)NC(c2nc[nH]n2)C)NC(C2CCS2(=O)=O)=O)CCCCC1 c1(C(=O)NCc2cccc(CNC(c3ccc(F)nc3)=O)c2)cc(O)ccc1Cl Cc1ccc(OCC(=O)NCC23CCC(C2)N(C(C2OCCO2)=O)C3)cc1C C(=O)(C(CC(C)C)NC(=O)C=CCC(C)(C)SC)N1C(CC)CCCC1 N1(C(CC2ON=C(CC)C2)=O)CCCC(C(=O)NC2CCC(C)(O)CC2)CC1 c1(C(=O)NCCOCCNC(C(C(C)C)n2cnnn2)=O)cnc2[nH]c(O)nc2c1 N1(C(CCC=C)=O)CCC(C2(O)CCN(C(C34CC(CN3C3CC3)C4)=O)C2)CC1 N1(C(CC(C)SC)=O)CC2(C1)CN(C(c1ccn3c(C)cnc3c1)=O)CC2CO C1(OCC)COCCC1NC1CCC(NC(=O)OC(C)(C)C)C1 C1(NC(C=Cc2ccc(C3C(C)C3)o2)=O)CCN(C(=O)CO)CC1(C)C C(CC(C)(C)F)NC(CNC(C(C)n1cncn1)=O)=O C1(CCOC)(NC(=O)CC(=O)N(C)C)CCN(C(C2CCCSC2)=O)CC1 C1(CC(N2C(COC)COCC2)=O)CCCN(C(C2SCCS2)=O)CC1 N1(C(CCCCC)=O)CCN(C(c2c(C)nsc2NC(C)=O)=O)CC1CC Cc1nn(Cc2sccc2Br)c2sc(C(=O)N(C)Cc3ccccc3)cc12 c1(C(=O)OC)ccc(C(=O)NC(C)CCCNC(c2cc(Br)no2)=O)[nH]1 Cc1nsc2ncc(C(N3CC(NC(=O)CC(F)F)CCC3C)=O)cc12 C1(NC(C2(COC)CC2)=O)CCCN(C(c2cnn(CCO)c2N)=O)CC1 CCC(C)C(CC(=O)NCC1CCC2(CC2)C1)NC(c1csc(C)n1)=O N1(C(COCCC=C)=O)CC2CC(C(N3CCCC(CC(C)C)C3)=O)(C2)C1 C(=O)(C(F)CC(C)(C)C)NC(c1cnn(C)c1)C(=O)NCc1occ(C)n1 c1(C(=O)NCCN(C(c2c(CCC)nsc2N)=O)C)ccc2scnc2c1 C(=O)(CCC(C)(C)C#N)NCc1c(C(N2CC(C)S(=O)CC2)=O)n[nH]c1 N1(C(c2c(C)onc2)=O)CC2(CCCC(CNC(C3CC(=O)NC3(C)C)=O)O2)C1 c1(CCN2CCC(CNC(c3ncsc3Br)=O)C2)cccc(F)c1 C1(CCC)CN(C(=O)C(C2CCCCC2)O)CC1C(N1C(C)CC1(C)C)=O C1(c2cn(CC)nc2)CN(C(CN2CCC(c3n[nH]cc3CO)C2)=O)CCO1 C(c1ccc([N+](=O)[O-])cc1)=CCNC(C1CC1(F)C(=O)O)=O NS(=O)(=O)CCCC(=O)NC(C1CCCC1)CNC(=O)CCCCC1CC1 C1(C)(C(=O)NC(C)CCNC(=O)CC2CSC2)CCCCC1 c1(CCNC(=O)NCCCC(C(C)C)C)cccc2ncccc12 c1(OC)ccc(C(=O)NCCC(O)C(=O)NCC2(O)CN(C)C2)nn1 C(=O)(C#CC1CC1)N(CC)CC1CCCN1C(C1CCC(c2cc[nH]n2)O1)=O N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CCC(=O)N2)=O)C(COC)C1 C#CCC(CC(F)F)C(=O)NCCC1(O)CCN(C(=O)C(OC)OC)C1 N(C(=NCc1ccc(Br)cc1OC)N1CC=C(F)C1)C(CC)C Cc1csc2ncnc(N3CCC(O)CC3C(=O)Nc3ccccc3)c12 O=C1CCOC(COC(=O)CCc2ccc(C(F)(F)F)cc2)C1 c1(C(=O)OC)cccc(Cl)c1S(=O)(=O)NC1CN(Cc2sccc2OC)CC1F Cc1cccc(Cl)c1C(=O)NC1CN(C(C23CC(C)(CO2)C3)=O)CCC1C c1(C(=O)NCC2CN(C(C(CCOC)OC)=O)C(C)C2)nc(Cl)ccc1F c1(C(=O)NC2CCN(C(c3cnc(Cl)nc3)=O)CC2F)c(O)cc(O)cc1O CCCCC(C)(F)C(=O)NCCCC(C)NC(=O)Cc1nc(C)sc1C N1(C(c2ncn(C(C)C)n2)=O)CCC2(CC(NC(C34CSCC3C4)=O)C2)C1 c1(OC)ccc(F)c(C(N2C3CN(Cc4c(C)noc4C)CC23)=O)c1F c1(CC)cc(CC(N2CC(C(N3CC=C(C)C3)=O)(COC)C2)=O)on1 n1(CC(N2C(CNC(C3C(C)C3(F)F)=O)CCC2)=O)nnc2ccccc2c1=O c1(C(=O)NCC(CC=C)NC(=O)C(C2CCCN(C)C2)(C)C)cnc(NC)cn1 N1(C(c2c(OC)cc(C#N)cc2)=O)CC2C3CCC(C2C1)N(C(C1CCSC1)=O)C3 NC(=O)CCCCC(=O)N1CCCCCC(NC(c2nccc3ccsc23)=O)C1 C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(CC)CSC N1(C(COCC(C)(C)C)=O)CC2CC(NC(=O)CC3CNC(=O)C3)CC(C2)C1 c1(CN(C(=O)C(C)CN(C(=O)CN2CCNC2=O)C)CC)ccncc1 c1(CCC(=O)N(C)CC2(NC(C3CC(CC)OCC3)=O)CC2)cccc(F)c1Cl Cc1cnccc1C(C)C(=O)NC(C)CNC(=O)CCC1CCC1 CCC1=C(C(=O)NC(C)C(c2ccccc2)NC(=O)CN(C)CC)CCCO1 c1(C(N(CCC(=O)NC2(CC#C)CC2)C)=O)cc[nH]c(=N)n1 Cc1c(C(N2CCN(C(=O)CC3CCN(C(C)C)CC3)C3CC23)=O)cccc1F C1(C(CNC(C2CC=CC2)=O)NC(c2ccn(C3CC3)n2)=O)CCCCCC1 N1(C(CCNC(=O)OC)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 CN1CC(O)CC1(C)C(N1CC(C)(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1)=O N1(C(c2c(C)c[nH]n2)=O)C2CCC1CC(NC(c1ccc(CN(C)C)cc1)=O)C2 c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccccc1O C1(C(N(CCC(C)NC(=O)CCC2CNC(=O)N2)C)=O)CN2CCCN1CC2 c1(C(C)=O)nc(C(N2CCC(C)C(CNC(C3CCC(C)O3)=O)C2)=O)cc(O)n1 N1(C(CCOCCOCC)=O)CCC(C(=O)NC2(C#N)CC2)C1 C1(CCCC)CN(C(=O)CSC(F)F)CCN1C(=O)CCCCSC c1(CCC(=O)NC2CC3CC2N(c2ccncn2)C3)ccc(F)c(F)c1 C=CCCCCCC(=O)NC(C)(C(=O)NC(c1ccn(C)n1)C)C1CCC1 c1(OC)ccc2ncccc2c1C(N1CCCC(CCNC(=O)CC(C)O)C1)=O C1(NC(=O)C=Cc2cn[nH]c2)CCCCCN(C(C2CC(F)C2)=O)C1 C1(N)CC(CNC(=O)C=CC(=O)N)C1(C)C.C1(CC)CN(CC(=O)C2CC2)C1 c1(C(N(C(CNC(CC2(OC)CCCC2)=O)C)C)=O)ccccc1CC#N c1(NC2CC(=O)NCC2)ccc(S(=O)(=O)NCc2nc(Cl)cs2)cc1F c1(C(=O)NC2(C(=O)NCCCN3CCOC3=O)CSC2)conc1C1CC1 c1(CNC2C(C(N3CC(O)C(F)C3)=O)CCC2)c(F)ccc([N+](=O)[O-])c1F c1(-c2cn(CCN(C)C)nc2)ccc(C(=O)Nc2cc(CO)no2)c2[nH]ccc12 c1(OC)cc(C(N2CC(CCCCNC(=O)CSC3CC3)C2)=O)cc(N)c1N c1(C(N2CC3C(CNC(C(C)OCCC#C)=O)(C3)C2)=O)c(CC)nn(C)c1CC C(c1cnn(C)c1)=C(C(=O)NC1C(CNC(C(C)=C2CCC2)=O)C1)C C(=O)(C1=NN(CCO)C(=O)CC1)NC1C(C)CN(C(=O)CC2OCCC2C)C1 c1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CCCC2)cc2cnccc2[nH]1 C1(C(=O)NC(C)C(F)(F)F)CC12CN(C(C1(C(F)(F)F)CCC1)=O)C2 C1(NC(=O)CCOC2CN(C(c3cn(CC#C)nc3)=O)C2)CC1C1CCCC1 N1(C(c2ncn(CC)c2)=O)CC(NC(c2ccc(Br)cc2)=O)CC1(C)CC c1(C(=O)NCC2OCCN(C(CSCCN(C)C)=O)C2)ccc2nc(S)oc2c1 C1(CC)CC(C(=O)NCC(C)N(C(=O)Cc2c(C)noc2Cl)C)CCC1=O Cc1cnc(NC2CCCOC2C2CCN(C(=O)C3CC3)CC2)nc1S(C)(=O)=O C1(O)(CN(C(C(C)NC(C2CCCC2)=O)=O)C)CN(C(C2CC(F)(F)C2)=O)C1 O=C(C1=CCC(F)(F)CC1)NC1(CNC(C2CCS2(=O)=O)=O)CC1 C1(C(=O)NCCC2CC(C(=O)NCc3nc(CC)oc3)C2)OCC2CCCC12 c1(C(=O)NC2(C)CC(NC(C(C)OCCCC)=O)C2)cc(CC)c(C)s1 N1(C(CCC2C(C)C2)=O)CC=C(CC(=O)N2CCC(C)(C(N)=O)C2)CC1 CC1(C)CN(C(C2(C(F)(F)F)CC3(CCC3)C2)=O)CC2(CC3CCC2C3)O1 C1(CNC(C(=O)N(C)CC2N(CC)CCC2)=O)CCC(N(C)C)CC1 C1(CC(C)NC(=O)CC2(CNC(C3CCCS3)=O)CC2)CCOC1 C1(C(=O)NC2(C(=O)NC3(C)CCSC3)CC(CO)C2)Cc2nccn2C1 CC(C)(C)C(C)(C)C(=O)NCCC(O)C(=O)Nc1ccc(Cl)cc1Cl c1(CCC(=O)N(CCN(C)Cc2ccc(COC)o2)C)ccc(OC)cc1Br C1(CCOC)(C(=O)NCC2(CCNC(=O)C=CC(=O)N(C)C)CC2)CCC1 C1(C)(C(N(C)CCOCCNC(c2[nH]ccc2C2CC2)=O)=O)COC(=O)C1 N1(CCN(C(CC(CCC)C)=O)CC)CCC(F)(F)C(C#N)C1 Cc1c(C(N2CC(F)(CNC(C3CCOC3)=O)C2)=O)sc2cc(F)ccc12 C1(NC(C(C(C)C)NC(=O)Cc2cn[nH]c2)=O)CCC2(CC1)N=N2 C1(CC(=O)NC(CNC(c2ncc(C)cc2C)=O)CO)CC(C)(C)OC(C)(C)C1 C1(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C(C)C2)Cc2ccccc2N1 CC(C)(C(=O)NCC(O)CNC(C1CCCN(S(=O)(=O)C(F)F)C1)=O)C(N)=O N1(C(C(CC)Br)=O)CCc2ccc(C(N3CC(C)CC3CO)=O)cc2C1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)CC(C)C(C)=O)Nc1c(CC)noc1 C1(CNC(C(CO)NC(C2C(C)(C(F)F)C2)=O)=O)NC(=O)CC1(C)C Cn1ccc2ccnc(C(=O)NC3(C)CC(NC(c4cnc[nH]4)=O)C3)c12 c1(OC)ccc(C)cc1CC(=O)NC1CC(O)CN(C(c2csc(C)c2)=O)C1 C(=O)(C(CCCCNC)N(C(CCC)C(=O)NC)C)NCCC C1(C(=O)NCC(CNC(c2n(CCCC)ncc2)=O)CO)CN(C(C)C)CCO1 c1(OC)cc(C)cc(C(N2C3CCC2C(NC(c2cc(F)c[nH]2)=O)C3)=O)c1O N(C1CCc2cccnc21)C(C12N(C(CC(C=C)(C)C)=O)CCC1C2)=O Cc1cccc(F)c1C(N1CCC(NC(C2CCC2(F)F)=O)CC1)=O C1(C(N)=O)C=CCCN1C(=O)CCC1CCCN1C(=O)CC=Cc1ccccc1 c1(C(=O)NCCOCCCNC(CC(C)CF)=O)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NCCOC2CCN(C(C3(O)CC(O)C3)=O)C2)cc(F)c(F)cc1F N1(c2nc(SC)nc(C)c2)CC(C2CCCN(C(c3cc(O)nc(Cl)c3)=O)C2)C1 Cn1nc(Br)nc1-n1nc(-c2nc[nH]n2)nc1CSC1(C)CCC1 C(=O)(CC(C)F)N(C1CCN(C(=O)CCSC)C1)CC N1(C(c2c(C(C)C)occ2)=O)CC(C(=O)NC(c2nccc(O)n2)C)C(C)(C)C1 C1(C2CCC2)(C(N(C)CC2CCN(C(c3cncs3)=O)C2)=O)CC1(F)F C(=O)(C(CC)CC(C)C)NCC(CNC(COCCCC)=O)OC c1(OC)cc(C(N2CC(c3nncs3)C2)=O)cnc1C(F)(F)F c1(CC(=O)NC(C(C)(C)C)CNC(c2cc(C3CC3)no2)=O)cc(O)nnc1O N1(C(C(C)SC)=O)CCC2(CCN(C(=O)CN3CCCC3)C2)C1 CCC(CC)CCCC(=O)N1CCC1C(=O)NCC(C)(F)C(C)(C)F c1(CC(C(=O)NCC(C(C)C)NC(C2CN(C)C2)=O)C)cnc2ccccc2c1 C1(NC(C(CC)C#N)=O)CC2(CCCCN2C(=O)C(c2ccccc2)F)C1 C1(NC(C(C)C)=O)CCN(CCNC(=O)C(c2ccnn2C2CCCC2)C)CC1 C1(NC(=O)C2=COCCC2)CC2CCC(C1)N2C(C12COCC(C1)OC2)=O C1(CNC(CCC(=O)NCC)=O)CC2CCC1N2C(C1(O)CN2CCC1CC2)=O c1(N2CCC(NC(c3c(C)noc3C3CC3)=O)C2)ncccc1S(C)(=O)=O N1(C(C(C)OCCOCC)=O)CCCC(O)(CN(C(=O)C2=NOC(CC)C2)C)C1 N#Cc1ccc2cc(C(N3CCN(C(c4cncs4)=O)C4CC34)=O)ccc2c1 C1(C(N2CCC(CCNc3c(C#N)c(Cl)ns3)CC2)=O)Cc2cccnc2C1 c1(N2C(C)CCC(NC(c3ccn(CC)n3)=O)C2)ccc([N+](=O)[O-])cc1Br N1(C(C(COC)(C)C)=O)CC2(CCCN(C(=O)CS(=O)(=O)CC(=O)OC)C2)C1 Cc1cccnc1C=CC(N1CCC2CCC12CNC(=O)CCCCC1CC1)=O Cc1ccc(CN(C(=O)C(CCN(C)C)NC(C2CC(O)C2)=O)C)nc1 N1(C(C(C)NC(COC)=O)=O)CC(C(=O)NCC2C(C)C2(F)F)C(C(C)C)C1 C12(CNC(c3scc(C)c3C)=O)CCC(C1)N(C(=O)C(C1CCC1)C1CCC1)C2 C=CC1(C(=O)NC2CCN(C(=O)C(=O)CCc3ccccc3)C(C)C2)CCOCC1 C1(C(N2CCN(C(c3cnn(C)n3)=O)C(CO)C2)=O)CCCCCC1(F)F C1(C)(NC(c2nc(C(C)C)sc2)=O)CCN(CCO)CC1 Cc1cc(C)c(C(=O)NCC2CCC(C)(C)CN2C(c2oncc2C)=O)c(=O)o1 c1(C(=O)NC(CNC(C(CC)C)=O)(C)CC)ccc2c(c1)CCO2 c1(NC(C2N(C(CCC=C)=O)CCSC2)=O)ccc(C2CC2)c(C#N)c1 C1(SCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)CCC2)CCS(=O)(=O)C1 N1(CC(=O)N(CCC(=O)N(C)Cc2cccs2)CC)CCCNC1=O CCCC1CNC(=O)C(C)CN(C)C1=O.C(c1cc[nH]n1)=CC c1(NN2CC(C)(C(=O)NCc3sc(Br)nc3Br)C2)c(Cl)cc(C#N)cc1Cl C=CC1(C(N2CCC(CNC(C3(C)CCCC3O)=O)CC2)=O)CCOCC1 CCCCC(CC)CC(=O)NCc1ccc(C(C)NC(c2ccncn2)=O)cc1 c1(NC(c2c(NC(C(C(C)C)O)=O)nccc2)=O)ccc2c(c1)n(C)c(=O)n2C c1(CC)ccc(O)c(C(=O)NCCCCC(C)NC(c2ocnc2C)=O)c1 N1(C(C(CC=C)C)=O)CC(CNC(=O)Cc2cnns2)CC12CCC2 c1(C(N2CC(N(C(C3CCC(OC)C3)=O)C)C2)=O)nc(C)c(C)[nH]c1=O CCN=C(NCCCCNC1(C(C)C)CCCC1)NCc1ccccc1F c1(C(=O)NCC(C(C)C)NC(=O)CCCS(C)(=O)=O)nnc(O)c2c1CCCC2 C1(C)(C(=O)NCC2C(N(C)C)CN(C(COCC)=O)C2)CC2(CCC2)C1 Cc1ccc(O)c(CNC(=O)C(CO)NC(c2ccc(C(C)C)o2)=O)n1 n1(CC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)co2)=O)ccc(=O)n(C)c1=O C1(OC)CN(C(C2CC2C2(C)COC2)=O)CCC1NC(C1CCC1(F)F)=O c1(CNC(C(=O)NCC2(C(C)(C)C)CCNC2)=O)cncc2c1CCC2 C(CN=c1[nH]nc(C(N)=O)s1)C1N(C(CCC(=C)Cl)=O)CCCC1C CC(C)C1=NOC(C(N2CCC(CF)(NC(=O)CCCc3cccnc3)C2)=O)C1 C(=O)(C#CC1CCCOC1)N1CCCC2(NC(CCCC)=O)C(C1)C2 N#Cc1ncc(CC2CC2)nc1N1CCC(C(N)=O)CC1 C1(NC(c2nc(CCC)oc2)=O)CN(C(c2cn(CC)nc2C)=O)CCC1C C1(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC12CCN(C(=O)CO)CC2 Cc1[nH]nc(C(=O)NCC2CC2NC(=O)CCC(=O)c2cccc(Cl)c2)c1O c1(OC)ccc(C(C)=CC(N2CCCC(NC(=O)COC3CC=CC3)C2)=O)cc1 CCCCC(CC(=O)NC1(CO)CCCCCC1)NC(c1sccc1C)=O N1(C(C2(F)CN(S(=O)(=O)CCCl)C2)=O)CCc2c(F)ccc(F)c2C1 c1(C(=O)NC2CCN(S(C)(=O)=O)C2)cc(OC(F)F)ccn1 C1(CNC(=O)Cc2cc[nH]c2)COCCN1C(=O)CC1CC=CC1 Cc1cc(CO)oc1C(=O)NC(CNC(=O)C(O)CCc1ccccc1)CO C=CCC(C(=O)N(C)CC1(C#N)CCC1)NC(=O)CCN1CCOCC1 CC1(C)Cc2cccc(C(N3CC4CC4(NC(C4CNC(=O)C4)=O)C3)=O)c2C1 c1(CC(=O)NCCC2CCCN2C(c2sncc2Cl)=O)ccc(CO)cc1 C1(COC(c2c(SCC)cccn2)=O)CC2C(C1)C2(F)F C#Cc1ccc(C(=O)NCC(CCC)C(=O)N2CCCC(C)C2CO)cc1 C(CC(C(C)(C)C)NC(=O)C1=CC(C)(C)C1)N(C(C(CC)n1cncn1)=O)C c1(C(N2CCC(C(C)NC(CN(C(COC)=O)C)=O)C2)=O)ncc(Cl)nc1Cl Cc1cn2nc(C(N3CCN(C(=O)C(O)C(F)(F)F)CC3)=O)cc(C)c2n1 N1(C(c2ccc(CC)[nH]2)=O)C2CCCC1CC(NC(c1c[nH]ccc1=O)=O)C2 C1(NC(c2ncn(CCNC(CC(C)C#N)=O)c2)=O)CC2CCC(C1)N2C C(=O)(C(C)CCCc1ccccc1)NCC(CC(C)C)NC(c1cscc1Cl)=O N1(C(CNS(C)(=O)=O)=O)CC2CC1CC2NC(c1cc(Cl)ccc1O)=O C(=O)(C(=O)C(C)(C)C)NC(C)CCCCNC(c1cccc(C2(O)COC2)c1)=O CC1(C)C(CNC(=O)C=CCN2CCC2)CCN1C(c1cc(O)nc(O)c1)=O n1(CC(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)nc(C)n(C)c1=O N1(C(C(C)=CC)=O)CCC(NC(=O)Cc2cccc(OC(C)C)c2)C12CC2 c1(C(N2CCN(C(C=CC)=O)C(C)C2C)=O)cccc([N+](=O)[O-])c1OC CN1CC(C(=O)N(C)CCOCCNC(=O)CCCN2CCCCC2)CC1=O C1(C(=O)NC(C2CSC2)C)CCOCCN1C(=O)Cc1nc(=N)[nH][nH]1 Nc1c(C(N2CCC=C(CNC(=O)CC3CC=CCC3)C2)=O)cnc2ccnn12 c1(C(=O)NC2(CCNC(C(CCSC)O)=O)CC2)cc2c(nc1N)CCCC2 Cc1cccc2nc(NC(c3ccc4c(c3)CC4)C3CC3)sc12 C(=O)(C(F)(CNC(c1ccn(COC)n1)=O)C(C)C)NC(C1CCOCC1)CC c1(C(=O)NCC2C(NC(CCCC=C)=O)C2)ccc(C(F)(F)F)c(O)c1 C1(CCCC)CN(C(=O)C(C2CCC2)OC)CCN1C(C1CC1C(F)F)=O c1(C(=O)NCC2N(C(c3ccc(OC)o3)=O)CC2)c(OC)cncc1Br C1(C(=O)NCC2C(C)CCCN2C(c2cnc(Cl)cn2)=O)CCc2nncn2C1 N1(C(c2cc(F)ccc2F)C(=O)NCCCSCC)CCC2(CC1)CNC(=O)C2 N1(C(c2nccc(C)c2)=O)CCCC(O)(CN(C(=O)CCC(C)(F)F)C)C1 c1(C(=O)NCC(C)N(C(CC2CCC(C)O2)=O)C)cc2c(=O)[nH]ccn2n1 c1(CNC(C2CCN(C3CC3)C2)=O)ccc(C(=O)NCCOC2CC2(F)F)s1 c1(C(N2C3CC(NC(=O)OC(C)(C)C)C2CC3)=O)c(F)ccc(O)c1F c1(C(=O)NCCC2OCCN(C(C(CC)(F)F)=O)C2)c(N)cccc1[N+](=O)[O-] c1(C(N2CC(N(C(Cc3c(C)nsc3)=O)C)C2)=O)[nH]c2ccccc2c1Cl C#CCCCCC(=O)NC(C1CCCCC1)C(=O)NCC1CC(C)=NO1 c1(CCC(=O)NCCC(C)N(C)C(c2cc(C(F)F)n(C)n2)=O)cncc(F)c1 c1(C(=O)NCC2C(C)(C)C(=O)C2)ccc(F)c(F)c1F C#CC1CN(C(C2CC(O)C(F)C2)=O)CCN1C(=O)CCCSC(C)(C)C c1(C(C(=O)NCCCOC)N(c2ccc(C)cc2)C)ccc(F)c(I)c1 N1(C(c2c(C(=O)OC)con2)=O)CC(NC(C2CCN2S(C)(=O)=O)=O)C(C)(C)C1 N(C1CC2(CCCC2)c2ccccc21)c1n(C)c(Cl)nc1Cl N1(C(C(C)(CC2CCC2)OC)=O)CC2CC(NC(=O)CC3C=CCCC3)C(C2)C1 Cc1cc(Cl)cnc1C(N1CC(C)CC1C(N1CCS(=O)CC1)=O)=O c1(N(C(CNC(C2(SC)CC2)=O)C)C)nc(C#N)ncc1Cl CCC(C(=O)N1CCCC1CC(=O)NCc1ocnc1C)C(F)(F)F C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1C(NC(CN(C)CC)=O)CC1 N1(C(CCC(C)OC)=O)CC(NC(c2cn(C)c(O)n2)=O)CC12CCCC2 CCCCC(C(=O)NC)NC(=O)C(O)CCCNC(=O)CC(C)CC C1(NC(COCCCC#C)=O)CCCC(CN(C(=O)CSCC2CCCO2)C)C1 N1(C(C)=O)CC(O)CC1C(N1CC(CCNC(c2coc(C(F)F)c2)=O)C1)=O c1(C(N(CCN(C(=O)CCN2CCCCC2=O)CC)CC)=O)nn(C)c(N)c1C n1(CCC(C)C)nc(-c2ccc(F)cc2)nc1CC1COC(C)(C)C1 C(=O)(C1=CCCOCC1)N1CC=CC(C(=O)NCc2nc(C3CC3)n[nH]2)C1 c1(C(=O)NC(CC(C)C)CNC(C2CC(O)CN2C)=O)ccc(Br)c(O)n1 CCC(CCCC(=O)NOCCC(C)O)Nc1cccc(C)n1 C1(CNC(C=C(C)Cl)=O)CCN(c2ncnc(Cl)c2[N+](=O)[O-])CCC1(F)F c1(CN2CCC(NC(=O)C(c3ccccc3)C3CC3)CC2)cc(Cl)nc(Cl)c1 C1(C(N2CC(N(C(=O)CCc3cccnc3Cl)C)C2)=O)CC2C(C1)C2(F)F C1(NC(C(CC)SC)=O)CCCCN(C(=O)C(c2ccc(F)cc2C)(F)F)C1 C1(C(=O)NC(c2c[nH]ccc2=O)C)(CC)CCCN(C(=O)CCCC(OC)OC)C1 c1(C(=O)NC23CC(CNC(=O)CSc4cccnc4)(C2)C3)onc2ccccc12 c1(N(CC(=O)O)CC)cnc(OC2CCOCC2)nc1.C12CN(C1)C2=O N1(CCC(N2C(CNC(C(C)CC3CCCC3)=O)CC2)=O)CCCCC1C N1(CC(=O)NC2C=CCN(C(COC(CC)C)=O)C2)CCSC(C)(C)C1 c1(C(N2C(C3(NC(CCSCCC)=O)CC3)CCCC2)=O)cnc2ccoc2c1 c1(C(=O)NCCC(C)N(C(c2ccn(CC(C)C)n2)=O)C)ccccc1S(C)=O C1(=CC(=O)NCCC2CCC(NC(=O)C(O)C3CCCC3)C2)CN2CCC1CC2 Cc1ccc(C(C)(C)C(=O)NCC=CCNC(=O)CC2CCCC(O)C2)cc1 C(=O)(C(F)C(C)(F)F)NC1CC(C(=O)NC(C2CNC(=O)N2)C)C1 N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(c2ccc(OC)o2)=O)CCN(C(C2CCN(C)C(C)C2)=O)CC(C)(F)C1 C1(C(NOCC)=O)C(CC)CCN1C(=O)C(C)Oc1ccc(C)cc1 CC1CCN(C(=O)CN(C23CC2CN(C(c2c[nH]nc2C(C)(C)C)=O)C3)C)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(C1(O)CCN(C(=O)C(C)(C)CCC#N)C1)C CC1(CNC(C23CCC(CC2)CC3)=O)CCCN(C(C2CCCN2C2CC2)=O)C1 c1(C(N(CC(CN(C)C(c2csc(C#N)c2)=O)O)C)=O)ccsc1S(N)(=O)=O O=C(CC(C(F)(F)F)NC(C1CCC2(CCC2)C1)=O)NC1CC(O)C1 c1(CNC(=O)NC(c2c(C)noc2C)CC)cc(C)c(OC(F)F)c(C)c1 C1(CC(N2C(CC(=O)N(C3CC4CC4C3)C)CC2)=O)CC=CCN1C C(=O)(CCCC(C)(C)CC)NCC1CCC(C(=O)NC2C(OCC)C2C)C1 C(=O)(C(C)(C)CCCNC(C1CCC(C)(C)OC1)=O)N(C)Cc1ncc[nH]1 c1(C(=O)NC(CCOC)CNC(=O)COc2cnc(Cl)cn2)ccnc(Cl)c1O C1(CC(=O)NCC2(C)CCN(C(c3ncc(Cl)cc3F)=O)C2)CN2CCN1CC2 C(=O)(C(F)(F)C(F)(F)F)N1CCC(C)(CNC(c2c(O)ccc(C)c2)=O)C1 c1(C2C(C(=O)NCC3CC(CNC(CCCC#C)=O)OC3)C2)cc(O)ccc1C N1(C(C2C3CN(C(c4cc(C)nc(C)n4)=O)C2C3)=O)CCn2ncc(O)c2C1 c1(C(=O)NC2CC(O)CN(C(=O)Cc3csnn3)C2)ccc2ccccc2c1 C12(NC(CN(CCC)C)=O)CCCN(C(=O)CSc3ccc(OC)cc3)CC1C2 C(=O)(C(C)CNC(=O)NC(C1CC2(CC2)C1)C(=O)OC(C)(C)C)OC C1(NC(C2CCN(C)CC2)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1N=[N+]=[N-] c1(C(N2CC(NC(CN3CCN(C)CC3)=O)C(O)C2)=O)sccc1S(C)(=O)=O C1(O)(C(=O)OC)CCN(C(c2nnc(C)n2C)C(=O)NC2CCCCC2C)CC1 CC1=C(C(=O)N2CCC(CCC(=O)NCc3noc(C(C)C)n3)CC2)CCC1 C1(NC(CSCC#C)=O)(CNC(=O)C(C)CS(C)=O)CCC(F)(F)CC1 C1(C(=O)OC)CCN(C(=O)CCc2ccc(Br)nc2)CC1O C1(C(=O)NCCN(C(=O)C(n2ccc(C3CC3)n2)C)C(C)C)CCOC1=O CC1CC(C(=O)NC2C3CCN(C(=O)Cn4cnnn4)C23)=NO1 c1(C(=O)OCC(=O)N(C(C2CCCC2)CC)CC)ccc(C)n(C)c1=O C(CCC(C)CC(=O)N1CC(NC(=O)C(C)(C)C(C)C)C(C2CC2)C1)=C(C)C C(=O)(N1CCCc2nccn21)C12N(C(Cc3n(C)cnc3)=O)CCC1CCC2 c1(C(N2CCC(N(C(c3nnc(C)s3)=O)C)C2)=O)cc2cnccc2[nH]1 C(CC1CO1)OC.c12cnn(c1)C2.C1(N(C)C)CC(CNC(=O)OC(C)(C)C)C1 N1(C(c2nc(C)oc2)=O)C2CCC1CN(C(=O)CN1CCCCC(O)C1=O)CC2 c1(C(N2CC(F)CC(C(=O)NCC3CCS(=O)(=O)C3)C2)=O)ccc(I)c(F)c1F Cc1nccc(C(=O)NC(CNC(=O)Cc2c[nH]nc2C)C2CCC2)n1 Cc1nc2sccn2c1C(N1CC2CCC1C(CNC(C1CCC(C)C1)=O)C2)=O Cn1cc(NC(c2ncc(CNC3CCNC(=O)C3)s2)=O)nc1C(=O)O C1(C(N(C2CCN(C(c3cn(C)nc3C)=O)C2)CCC)=O)CC(C)CC(C)(C)C1 C(=O)(N=c1nc(O)c2ccccc2s1)NCCc1c(F)ccc(C)c1 c1(C(=O)NCC2N(C(c3cc(C)nnc3)=O)CCCC2C)cc(F)c(F)cc1F CCC(CC)(C(C)C)NC(C1CC(O)(CNC(=O)C(=O)C(C)(C)C)C1)=O c1(C(N2CCC(O)(CNC(C(C)C3CCC3)=O)C2)=O)cnc(O)c(Br)c1 N1(C(Cc2c(C)ccs2)=O)CC2CCC2(CNC(C2CCS2(=O)=O)=O)C1 C(=O)(CC(=O)NCC1CC1NC(C1(C(C)C)CCC1)=O)NCC N1(C(C(CN(C)C)(F)F)=O)C2CCC1CC(NC(=O)CCCc1ccsc1)C2 C1(NC(CCc2[nH]c(=N)sc2)=O)CCN(C(=O)C(C2CCCCC2)O)CC1CO N1(C(=O)C#CC2CC2)CCCC(F)(CNC(=O)C(c2ccccc2Cl)O)C1 N1(C(CCC=C)=O)CC(NC(c2cnc(C)cn2)=O)C(C#N)C1 Cc1cc(CNC(c2cc(Cl)ccn2)c2nnnn2CCCF)c(C)o1 Cc1ccc(NC(=O)C(=O)NCC2CC(C)N(C(c3cnsn3)=O)C2)cc1C N1(C(CCCCN(C)C)=O)CCC(NC(c2cn(C(F)F)cn2)=O)C12CCC2 c1(C(N2CCC(COCc3cn(C4CCCC4)nn3)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C2(O)CCN(C)CC2)(C(=O)NC2CCN(C(C(CC)(C)CC)=O)CC2F)CC1 CCC(C(=O)NC1CCCN1C(=O)CC1CCC(C2CC2)O1)NC(N)=O CCCC(CNC(=O)C1=CCCC1)C(=O)NCc1[nH]ccc(=O)c1O N1(C(C=C(CCC)C)=O)CCN(C(C2(N(C)C)CCCC2)=O)C(CF)C1 S(=O)(=O)(c1ccc(N2CCCC3(CCCO3)CC2)c(Br)c1)NCC=C CCCC(C)(O)C(=O)NC(C)CCC(N1CC2CCC(C1)O2)=O CCC(CC(F)(F)F)C(=O)N1CC(NC(=O)CC2(CCOC)CCCC2)C(C)C1 C1(NC(C2CSC2)=O)CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1F C1(C(N(C)Cc2ncn(C)n2)=O)CC(N=[N+]=[N-])CN1C(=O)C1=CCCCC1 c1(OC)ccc(OCC(=O)N(C2CCCN(C(C3C=CCC3)=O)C2)C)cc1 O=C(C(O)CC(F)(F)F)NC1CCN(C(c2ccnnc2SC2CCCC2)=O)C1 c1(OC)ncc(CONC(C(=O)NCCc2ccccc2)=O)cn1 C1(CNC(C2C(C)CC(=O)NC2)=O)CC2(CCC2)CN1C(C1(NC(N)=O)CC1)=O N1(Cc2ccc(C)c(C)c2)Cc2ccccc2C1C(=O)Nc1cc(Br)cnc1Cl N1(CC2C(OC)CCC2)CCC(=O)N(CC(C(F)F)c2ccccc2)C1=O C=CC(C)N=C(NC1CC2(C1)CC(F)(F)C2)N1CCc2cc(Cl)cc(Cl)c2C1 c1(NCC2(O)CCN(C(C3(CC(C)C)CCC3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] CC1CCC=C1C(=O)N1CCC(O)(CNC(=O)COc2ccccc2Cl)C1 c1(C(N2CCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)ccc2nccn2c1 C1(NC(C(C)C2CC2)=O)CCCOC12CCN(C(C1CC(C)(F)C1)=O)CC2 C(C(C)C(=O)NC1(C)CC1(C)C)NC(COCCC)=O N1(C(c2cnsc2Br)=O)CCC(c2cn(CC3CC3C(F)(F)F)nn2)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(C(N2CCCN(C(C3CC3(Cl)Cl)=O)CCC2)=O)cc(=O)n2nccc2[nH]1 c1(C(CNC(N2CCCC(=C)C2)=O)C(F)(F)F)c[nH]c2ccccc12 c1(C(=O)NC2C3OCC(NC(c4c(CC)ncs4)=O)(C3)C2)cc2c(s1)CCCCC2 Cc1ccc(C(=O)N(C2CCC(CNC(=O)C(=O)NC3CC3)CC2)C)c(O)c1C CC1CN(C(=O)C=CC(F)(F)F)CCC1CNC(c1cccc(Cl)c1O)=O N1(C(C2C(C)C2)=O)CCCC2(C1)CN(Cc1cc(C(=O)O)cc(Br)c1)C2 c1(-n2cc(SCC3(C)CCCCO3)nn2)cc(F)cnc1Br c1(OC)ccc(N(CCC#N)C(=O)CN(c2c(C)cnn2C(C)C)C)cc1 CN1CCN(C(c2cncc(Cl)c2)=O)C(CNC(=O)C(F)(F)C2(O)CCC2)C1 c1(CC)cc(C(N2CC(F)(CNC(c3noc(C)c3Br)=O)C2)=O)c(C)o1 C(=O)(C(C)(C)c1ncco1)NCC1(CNC(C=CC(C)(C)SC)=O)CCC1 c1(CC(=O)NCC(CNC(C(C)OCCN(C)C)=O)C)cc(F)ccc1Cl C1(Cc2cn(CC(C)NC(=O)CCCc3cccs3)nn2)CCCCN1C C(CC(Cc1ccccc1)NC(=O)C(C)C#N)NC(C=C(CC)C)=O c1(N(CCOC)C)nc(NCC2CCCC2)cc(NCCN(C)CCO)n1 c1(C(N2CC(C)C(NC(CNC(C)=O)=O)C(C)C2)=O)ccc2cccnc2c1 CC(CC(=O)NC1CN(C(C2(C#N)CC3CCC2CC3)=O)CC1O)CC(C)(C)C C(C)(C)(CCCC(=O)NC1CC(C)(C(=O)NC)C1)NC(CNC(C(CC)C)=O)=O CN=c1cc(CNC(c2ccccc2CCC(C)C)=O)cc[nH]1 c1(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)cnn2c1OCC(F)C2 c1(C(=O)NC(C)CCCCNC(C2CC3CCC2CC3)=O)ccnc2[nH]cnc12 C1(N(C)C)CCN(CCNC(N2CCC(CC(C)(C)C)C2)=O)CC1 c1(C(=O)NCC2CC(F)(CNC(c3cc(COC)on3)=O)C2)cn(C)ccc1=O C1(NC(c2cccc(-c3cnco3)c2)=O)CCCCN(C(C2(Cl)CC2(F)F)=O)C1 CC1(C(=O)NCC(CO)NC(c2cscc2Br)=O)COCCO1 C=CC(C)(CCOC)C(=O)NCC(C1CC1)NC(=O)COc1ccc(C)c(C)c1 N1(C(CS)=O)CCC(OC(COC)O)CC1.C1(C(N(C2CCSC2)C)=O)CCCO1 c1(C(C)C)cc(C(=O)Nc2ccnc(CF)n2)n(-c2ccccn2)n1.C1(=O)CO1 c1(C(=O)N)ccccc1OCCN(CC(C)NC(=O)CCC1CC1(F)F)CC C12(CCNC(Cc3c(NC(=O)OC(C)(C)C)cccc3)=O)CCC(C1)C(=O)N2 CC(C)CC(C(=O)NCC1(CNC(=O)CN2CCCCCC2=O)CCC1)C(N)=O C1(NC(c2c(C)ocn2)=O)CN(C(=O)CCn2c(C)n[nH]c2=O)CCC1C N1(C(C(C)SC)=O)CCN(C(c2ccnc(OC3CC3)c2)=O)CC1C(C)C Cc1ccnnc1C(=O)NC(C)CCCCNC(C1CC(=O)N(C(C)(C)C)C1)=O N1(C(C(C)C(F)F)=O)CC2CCN(C(=O)CCCc3ccc(F)c(F)c3)C2C1 CC(CC(F)F)C(=O)NC1CC(NC(c2ncc(Br)cc2O)=O)C1 C(=O)(CC(C(C)OC)NC(=O)CCC(N)=O)NCCC(=O)NCC c1(OC)cc(F)c(C(=O)NC(C)CN(C)C(C2Cc3nncn3C2)=O)c(F)c1 CC(C)CC(C)CC(=O)N1CCOCCC1C(=O)N(C)Cc1cn(C)nn1 N1(C(C2(COC)CC=CC2)=O)CCC2(NC(c3c(OC)cccc3Cl)=O)CC2C1 C(=O)(C(CCNC(=O)C(C)(C)c1cnsc1)N(C)C)NC(CC=C)CNC(C)=O c1(NC2CCC3CN(C(CC(C)n4ccnc4)=O)CC32)ncnc2c1CCCC2 C=CCC(C)C(=O)NC(c1ccccc1)CNC(c1sccc1C1CC1)=O N1(C(C2C(CC)C2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 CC1CC2(CC(C(N3CCN(C(=O)CCCC4CCCC4)C(CO)C3)=O)C2)C1 c1(N(C(c2cccc(-c3c(C)cc(C(N)=O)s3)c2)=O)C(C)C)c[nH]cc(Br)c1=O c1(C(CC)C)cc(C(=O)NCCC2(NC(c3sccc3SC)=O)CC2)on1 c1(OC)csc(C(=O)N(C)CC2(NC(C3CCSCC3)=O)CC2)c1OC C(C(C)(O)C(=O)NCC1CCC1C(=O)NCC1(CO)CC12CCC2)OC c1(N2CC(O)(CCNC(C3C(C)CC(=O)NC3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(C(C(C)C2CC2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl N1(C(c2c(C)ocn2)=O)CCCN(C(C2CCC3C2C3(F)F)=O)CCC1 C1(NC(=O)CCF)CN(C(c2ccc3n[nH]cc3c2Cl)=O)Cc2nccn2C1 CCC(F)(F)C(=O)NC(CO)C(C)NC(=O)CCN1CCCC(C(N)=O)C1 c1(C(CNC(CN(C2CCC2)C(C2C(=C)C2C(=O)OC)=O)=O)O)ccncc1 C1(CNC(COCC(C)C)=O)CC(C)N(C(=O)CCOC(C)=O)C1.c1ccccc1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1CC2NC(C1CCC(C)C1)=O C(=O)(C1CCCc2nnn(C)c21)NC(C1CCCC1)CNC(CCCC#C)=O c1(NCC2ON=C(CC)C2)cc(N2CC=C(Br)CC2)nc(C(C)C)n1 C(C(CN=c1[nH]c2ccc(O)cc2s1)C(F)(F)F)NC(C(C(CC)C)OC)=O C1(CNC(C2(F)CN(C(CCc3cn(C)nn3)=O)C2)=O)CNC(=O)CO1 C=CC(C)CC(=O)NC1CCCN(C(c2ccc(CCC(F)(F)F)cc2)=O)C1 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2CC(NC(c3ccc[nH]3)=O)C1C2 c1(C(=O)NCC#CCNC(C(c2cccc(OC)c2)C)=O)ccc2c(c1)CCN2 N1(C(COCC(=C)C)=O)CC(NC(c2ccc(N(C)C)cc2)=O)CC(C)C1 C(=O)(C1=CCc2ccccc21)NCC1CCCC(NC(C(C(C)(F)F)(C)C)=O)C1 Cc1ncc(Br)c(C(=O)N(C(C)CCNC(=O)COCC2CCC2)C)n1 N1(C(C)=O)CCCCC1CNCc1ccc(CNC)cc1 C1(C(=O)Nc2cnc(C)nc2)C2CCC(C2)N1C(=O)C(O)CC(N)=O CC1(C)CCCN(C(=O)CC2CCCC(=O)N2)C1C(=O)NCCOC1CCCC1 c1(CC(=O)NC(C)CCNC(C2CCCN2C)=O)ccnnc1O CCCCCC(O)CC(=O)NOCC(N1CCC2(CCSCC2)CC1)=O N1(C(C2ON=C(CC)C2)=O)CC(NC(c2cc(O)ccc2O)=O)CC(C)(C)C1 C=CCN=c1[nH]cc(C(=O)N(C(C)CNC(C2CN(C)C2)=O)C)s1 C1(CNC(CC=C)=O)CN(C(c2cnn[nH]2)=O)CCC1C(F)(F)F C1(C(=O)NC2CCN(c3ncn(C)c(=O)c3)CC2F)CC2(CCCC2)CO1 CC(CNC(c1cocn1)=O)C(F)C(=O)N(C1CCC1)C C(=O)(C(C(CC)CC)OC)N1CCCC(CC=C)(NC(=O)CCc2nc[nH]n2)C1 C=CC(CC)CC(=O)N1CC(C(N2CCC3C(C(N)=O)C3C2)=O)(CC)C1 c1(C(N2CCCC(C)C2C)C(=O)NC(C(=O)OC)C)cc(C)ccc1OC c1(C(=O)NC(C)(C)CNC(c2ccccc2CC#N)=O)cncc2sccc12 N1(C(c2cc(OC)no2)=O)CCCC(C(=O)NCC(n2cccn2)C)C1 c1(C(=O)NCC(C2CC2)NC(Cn2cc(C(C)=O)nn2)=O)c(C)nsc1C c1(C(N2CCC(NC(=O)C=CCF)CC2)=O)cnc2nc(O)nc(O)c2c1 C(=O)(C(C)(C)CCC(=O)N1CCC(NC(C2C3COCC23)=O)CC1)OC CCC(CC(=O)NCCCCCCN(C)C(c1cn(C)cn1)=O)C(F)F c1(C(N(C2CCN(C(CC3CC(C)C3)=O)C2)C)=O)cc(=O)c2ccncc2o1 CC(CC(N)=O)C(=O)N1CCCN(C(C2(C(F)F)CCCO2)=O)CC1 c1(C(=O)NCCNC(C2(Cc3ccccc3)CCCO2)=O)cc(O)cc(O)n1 c1(CCC)onc(C)c1C(=O)NCCC(C)NC(C1CCOC1=O)=O N1(N2C(CC=C)(C=O)CCC2)CC23CCC2(COC3)C1.C(=O)CC(C)SC Cc1ccc(CCNC(=O)CC2(NC(C3CC(C4CC4)C3)=O)CCCCC2)nc1 c1(C(N2CCC(C(C)(C)NC(C3CNC(=O)N3)=O)C2)=O)cc2cc(Cl)sc2[nH]1 Cc1cc(C(N2CCC(C)(CNC(=O)C(C)C3CCOC3)CC2)=O)ccc1Cl C1(c2n(C)ncc2)CN(C(=O)C(F)n2cccn2)CCN1C(=O)Cn1cccn1 CCC(CNC(=O)CCCOC)(CC)NC(=O)C(C)C(C)O C(=O)(CS(=O)(=O)CC(F)(F)F)N(C1CCCN(C(C(CCC)OCC)=O)C1)C Cc1cc(-n2cc(C(=O)NC(CCO)C(C)C)nn2)cc(C)c1 N1(C(c2nnn(CC)c2C)=O)CCC(C2CCN(C(C3CCCC3O)=O)CC2)C1 c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)CC3CC3(C)C)CC3CC3)cc2n1 N1(C(C2CCCN(CCCN)C2)C)CCCCCC1=O.c1(C)cn(CC#N)nn1 C1(CN(C(=O)CCCNC(c2ccoc2)=O)C)CN(C(=O)CN(C)C)CC12CC2 C1(CC(NOC(CC)CC)=O)CCCCN1C(=O)CC1CC1CC C1(CC=C)(NC(=O)CCCn2cncn2)CCN(C(=O)C(C)(C)CSC)C1 c1(C(N(C)CC2(NC(C(C(C)O)C)=O)CC2)=O)c(F)cncc1Br NC1(C(N2CC(OC(=N)O)C2)=O)CC2CCC(C2)C1 C(=O)(CCC(C)(C)C(=O)N1CC(NC(=O)CC(C)(C(F)F)N(C)C)C1)OC Cc1cn2c(n1)CN(C(c1csc(CNC(c3cc(O)n(C)n3)=O)c1)=O)CC2 C1(C(N(CC(CNC(c2nccc(C)c2N)=O)(C)C)C)=O)CCn2nnnc2C1 C1(CC(N2CCC2C(=O)CC(=O)OC(C)(C)C)=O)SC(=Nc2ccccc2)NC1=O C(C(O)CCCCCCCCCCO)N1OCC2(C(=O)NC(=O)N2)OCC1 Cc1nn(-c2ccccc2)cc1-c1nc(CC2CC2)nn1CC1CCCO1 C12(C(=O)NC(C)Cc3ccccn3)CCCC1CCN2C(C1CCC(=O)O1)=O O=C(C1CCc2c[nH]nc21)NCC1(O)CCCN(C(=O)C2=CCCC2)CC1 C1(C)(CC)CCN(C(=NCCN2CCC(C)CC2)NC(C)COC)C1 N1(C(c2ccc(CC)o2)=O)CCC(CNC(c2ccn(C(C)C)n2)=O)(COC)C1 CCC(=O)CCC(=O)NOCC(N1CCCC12CCOC2)=O N1(C(C2(CC)CCC2)=O)CC(NC(=O)CC2CCCCCO2)C(C2CC2)C1 c12nc(c(C)s1)CN(CCN(C)C)C(=O)C2OC.C(=O)(C(C)OC)OCC CC1(C(=O)NCC2(F)CC(NC(=O)Cc3cccs3)C2)CCNC1=O CCC(C(=O)N1CCN(C(c2ccccc2I)=O)CC1)C(C)O C12(CNC(CC(=C)C)=O)CCCCC1N(C(c1cc(OC)cc(Cl)c1O)=O)CC2 N1(C(C=C(CCC)C)=O)CC(NC(=O)CC2COC(=O)N2)CC(C)(C)C1 c1(CC(=O)NCC(C)CNC(C2(C)CCCNC2=O)=O)cccc(Cl)c1Cl N1(C(C2(C=C)CC2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C(F)C1 c1(NC(C2C(NC(=O)OC(C)(C)C)C2)=O)cc(Cl)c([N+](=O)[O-])cc1O Cc1nc(NC(c2ccc(F)cc2Cl)C)cc(N2CCCC(OCC3CC3)C2)n1 C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(=O)Cc1csc(-c2nc[nH]n2)n1)C c1(C(=O)NCC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)cccnc1N1CCCC1 c1(C(=O)NCCC(C)N(C(=O)C#CC2CCCO2)C)ccc2cnnc(O)c2c1 Cc1cccc(C(N2CC(NC(c3nccc(Cl)c3C)=O)C3(CC3)C2)=O)c1C#N C1(C(=O)NCCCc2cnccn2)CC2(CC2)CN1C(c1ccc(F)c(O)c1)=O C12(CC)CC1CN(C(c1cc(CNC(=O)C=CCN3CCCC3)on1)=O)C2 C(CC(C)C(=O)NCCN(CC(C)O)C(=O)Cc1cnsc1)=CC c1(CN(C)C)ccc(OCC(=O)NC2CCC2c2ccc(F)cc2)cc1 C1(O)(CN(C(C(=O)NCCOC)=O)C2CC2)CCN(C(=O)C=CC2CCC2)C1 N1(C(c2ccc(SC)s2)=O)CCC2CN(C(=O)CCCC3CCCC(=O)N3)CC12 C1(C(=O)NC(C(=O)NC(CCC=C)C)Cc2ccoc2)CC2CC(=O)C1C2 C=C1CC(C(=O)NCc2ccc(Cl)s2)N(C(c2ccnc(F)c2)=O)C1 CC(C)(C#N)CC(C)(c1nnnn1C1CCCC1)NC1C2COCC12 C1(CC)C2CC1N(Cc1cn(-c3ccc(Nc4nscc4C(=O)O)cc3)nn1)C2 Cc1nc2cccc(C(=O)N(C3CN(C(=O)C=Cc4ccsc4)C3)C)c2s1 c1(OCCC)ccc(Cl)cc1NC(c1csc(Cl)c1)c1nnnn1C1CCC1 C(=O)(C1=Cc2ccccc2C1O)NC1C2C(C)N(C(c3cc(C)c(C)o3)=O)C1C2 N1(C(=O)Nc2cc3c(cc2Br)OCO3)CCC=C(c2cccnc2)C1 N1(C(CSc2n(C)nnn2)=O)CCN(C(=O)C(F)C(F)(F)F)CC1C1CC1 CCC(C)(C)CCNC(=O)CC=CCNC(C1COCC1C(N)=O)=O CCC1=NOC(CC(N2CCC(NC(=O)CCN3CCCCCC3)C2C)=O)C1 C1(C)(CC)C=C(C(=O)N2CCC(C)C(NC(=O)CCc3cncc(F)c3)C2)C1 C(C1=NOC2(CCC2)C1)NC(C(CNC(=O)Cc1cccnc1)N(C)C)=O Cc1c(C(N2CCCC(NC(c3cnc(C#N)s3)=O)C2)=O)cncc1Br C1(NC(COCC)=O)CC2CC(NC(c3scc4c3CCCC4)=O)CC2C1 C(=O)(CCC(=O)c1ccc(Cl)cc1)NCC(CNC(CC(C)C1CC1)=O)(C)O CCCCCCC(C)NC(=O)C(CCC)c1nn[nH]n1 c1(CC(C)NC(C(C)C)=O)ccc(CNC(c2scnc2C(C)C)=O)cc1 C1(CNC(C(COC)(C)O)=O)CN(C(=O)C(F)=C(C)C2CC2)CC12CCC2 N1(C(c2n(CC)cnn2)=O)CC2(C1)CN(C(C1CC13CCCC3)=O)C2 CC1(NC(=O)CC2CNCCN2)CCC(O)CC1 CCC(C)(C)CCN=c1[nH]c(=NC(C)c2ncccc2Cl)[nH]c2cccnc12 C=CCCC(C(=O)NCC(C)(C)C1CCC1)NC(C1CC2(CCC2O)C1)=O N1(C(C(Br)=C(C)C)=O)CCC(C2CCN(C(=O)C3=C(Cl)CCOC3)C2)C1 CC(C)(C)C(O)CNC(C1(CNC(c2nocc2Cl)=O)CCCC1)=O CCC(C)(CO)C(=O)N1CC(CCNC(c2ccc(-n3cccn3)cc2)=O)C1 C(=O)(C1Cc2ccccc21)NCC1C(NC(Cn2cc(C(C)(C)C)nn2)=O)CC1 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(c1ccc(C)c(F)c1)=O C(C)(C(=O)NCCCCN(C(=O)COC1CCOC1)C)OCC=C c1(NC(C2N(C(CN3C(C)CCC3)=O)CCCC2)=O)cn(C)nc1C#N C1(NC(CN(C(C(C)C)=O)C)=O)CC(F)CN(C(c2ccc(Cl)cc2)=O)C1 C(=O)(C(F)CC1CCCCC1)N(CC(C)NC(=O)CCNC(=O)C1CC1)CC C1(CNC(c2ccc(Cl)s2)=O)C2CN(C(C3CCCC(F)C3)=O)CC12 C1(CCO)CCCCCN1Cc1nc(Cl)cs1 C1(CNC(C2CC(CC)C2)=O)CC(F)(F)CN1C(c1cc(OC)no1)=O c1(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] NC1CC(CC(N2CCN(C(C3CCCCN3)C)CC2)=O)C(O)C1 C1(O)(CC)CCN(C(=O)C(CCNC(c2c[nH]c(C#N)c2)=O)OC)C1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)N(C)C)C2)ccc(C(C)C)c(C)c1 Cn1nnc(C=CC(=O)NC2CCCC(NC(c3csc(Cl)c3)=O)C2)n1 C1(C(=O)NC2CC2)OCCC1C(=O)N(CCCO)CCOCCCO CCCCCC(O)CC(=O)N1CCN(C)C(CNC(c2occ(C)c2C)=O)C1 C1(C(N(CCCNC(C2CCCC23CCC3)=O)CCO)=O)CC2(CCO1)CC2 N1(C(c2ccc[nH]2)=O)CCC2(CCOCC2C(N2CC(F)C2)=O)CC1 N1(C(c2cnc(C)s2)=O)CCC(C)(C)C1CNC(c1n[nH]cc1C(C)C)=O c1(CSC)ccnc(C(=O)N(CCCN(C)C(c2cnn(CCN(C)C)c2)=O)C)c1 N1(C(C(C=C)C)=O)CCN(CC(=O)NCCn2cc(C(C)O)nn2)C(=O)C1 C1(COC)(NC(c2nc(Cl)cs2)=O)CCN(C(c2c(C)csc2Cl)=O)C1 c1(C(=O)OCC)cc(C(=O)CNCC(=O)N(CCCC2CC2)CC)on1 Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCN(c2ccnc(C3CC3)n2)C1 c1(OCC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(O)C(F)F)cc1 CC1OCCC1CC(=O)NC(Cc1ccoc1)C(=O)NC(CC1CCCC1)CO c1(C(=O)NCC2N(C(C(CCC)C(C)C)=O)CC2)nccn2nc(C)cc12 c1(CC)onc(C)c1C(=O)NC(C)CC1CN(C(C2CCN2CC)=O)C1 c1(C(=O)NCC2CC(NC(c3cnc(NC4CC4)s3)=O)C2)ccc2c(n1)NCC2 C12(C(=O)NCC(C)N(C)C)CCC(CC1NC(c1cn(C)nn1)=O)C2 N#Cc1cc(F)c(C(N2CCSC(C(=O)NCC3CCC(O)CC3)C2)=O)c(Cl)c1 CCCCC(O)C(=O)N1CCC(CC(COC)NC(C2CC=CCC2)=O)CC1 CCC1=NOC(C(=O)NC(C)CN(C(c2cnn(C(C)C)c2)=O)CC)C1 n1(CC(=O)NCC(CO)NC(c2nnc(C3CC3)s2)=O)nnc(=O)[nH]1 n1(CC=C)ncc2c(O)nc(=NCC3CCN3C(=O)CC(C)(C)O)[nH]c12 C1(C(=O)NC(CC)C(=O)OC)CC(F)(F)CN1C(C1CCC(C(=O)OC)C1)=O N1(C(c2cocn2)=O)CC(C(=O)NCCOCC(F)(F)F)C(C2CC2)C1 c1(C(=O)NC(C)C(C)(C)NC(C2CCC(=O)O2)=O)ncnc2c1OCCO2 c1(OC)ncc(C(N2C(C(=O)NCCn3cc(C)cn3)CC3CC23)=O)cn1 C12(NC(c3occ(C)c3C)=O)CCC1CN(C(=O)CCN1CCN(C)CC1)C2 c1(NC(N2C(c3onc(-c4c(OC)cccc4)n3)CCC2)=O)c(F)cccc1Cl c1(C(N(C)CC2CCCN2C(=O)COCCF)=O)cccc(OC(F)(F)F)c1 N1(C(CC(=O)NC(=N)N)=O)CCCC(c2ncon2)C1 O=C1COC(c2ccc(NC3CC4CCCCCCC34)cc2)=NN1 C1(NC(C(=O)OC)CC2OCCO2)CCC(P(C)(C)=O)C1 CCC(CC)CC(F)C(=O)NOC(CC(C)C)C(=O)NCC1CC(OC)C1(C)C C(=O)(CCCCCCCC1CC1)NC(CCCNC(C1(CC)CCCC1)=O)C c1(-n2c(CCCc3cc(C)no3)nc(-c3cc[nH]n3)n2)ccc(F)cc1C C(CC(C)C)(C(=O)N1CC(CCNC(c2nnc(Cl)cc2N)=O)(OC)C1)OC N1(C(C2CCC(NC(C(C)OC(C)=O)=O)C2)=O)CCc2ncncc2C1 c1(COCC=CC(=O)NC2CN(C(c3sccc3Cl)=O)C2)ccccc1 Cc1cc(=NCCC2CCCC23CC3)[nH]c(=NCc2ncc(C)o2)[nH]1 c1(OC)cc[n+]([O-])c(C(=O)NC2CC(N(C)C(C3CCCCC(=O)N3)=O)C2)c1 C(=O)(CCCC(C)(C)C)NCCCN(C(=O)CCc1cncn1C)CC CCC(CC)CCC(=O)NCC(C)C(F)C(=O)N(CCOCCO)CC N1(C(c2c(C)ncs2)=O)CCCC(C)C1CCNC(c1sccc1OC(F)F)=O CC1(C)CN(c2cc(C(F)F)ncn2)CCC1NC(C1CCC(=O)N1)=O CC(CN(C)C)CC(=O)N1CCC(F)(CNC(=O)Cc2cc(Cl)sc2Cl)C1 c1(C(=O)O)ccc(C=NOC2CCCN(CC(F)(F)F)C2)cc1F CC1Oc2ccc(C(=O)N(C3CCCN(C(=O)CN(C)C)CC3)C)cc2C1C C1(NC(Cc2c(OC)ccc(Br)c2)=O)CCCC2CN(C(C3CCCO3)=O)CC12 N1(C(C(C(C)O)N(C)C)=O)CCCC(N(C)C(c2cc(C3CCC3)[nH]n2)=O)CC1 N1(C(c2cccc(CCC)c2)=O)CCC(NC(=O)CSCc2cscn2)C(C)C1 C1(C(=O)NCc2c(C(=O)NCC3CCC(C)C3)c[nH]n2)CC2(CC(=O)C2)C1 [N-]=[N+]=NC1CCN(C(=O)Cc2ccnc(C(F)(F)F)c2)CC1 Cc1cnc(C(=O)NCCCC2(NC(C3CCOC3C(F)(F)F)=O)CC2)c(C)c1 c1(C(=O)NCCCN(C(CC(C)C2CCCO2)=O)C2CC2)cc2ncccc2o1 c1(C(=O)NCC2CC(O)CN2C(C2CCCC2)=O)ccn2ncnc2c1 c1(NC(C(C)Oc2cccc(F)c2F)=O)nc2c(s1)CC1(CCCCC1)CC2 C1(NC(CN2C(C)CCC2)=O)CN(C(=O)CCc2cc(Cl)sc2Cl)CCC1F C1(NC(=O)CSc2nc[nH]n2)C2CC3C(C2NC(C(C(=O)OC)C)C)C13 N1(C(C(C)C)=O)CC2(CCN(C(C3CSc4ccccc4O3)=O)CC2)CC1C C1(CNC(C(C=C)C)=O)C(C2CC2)CCN1C(=O)Cc1ccc(OC)nc1 c1(C(=O)NCC(C(=O)NCCC2CCN(C)C2=O)OC)cnc(N)cn1 c1(C(N(CCC(C)NC(CCCCCC)=O)C)=O)cccc2sncc12 CC(C)CC(F)C(=O)NC1CC(NC(C2(c3cccc(F)c3F)CC2)=O)C1 Cc1cc(-c2nc(CC3(C(F)(F)F)CC3)n(Cc3cnccc3Cl)n2)ccc1F N1(C(C(CCNC(=O)C=Cc2ccoc2)OC)=O)CCC2(CCC2)CC1 C=CCC(CC=C)C(=O)NCC#CC(=O)N(CC(CC)OC)C CCC(C)C(C(=O)N1CC(NC(C2CC2c2ccccc2Cl)=O)C(C)C1)N(C)C C1(COC)CC(CNC(c2c[nH]c(=N)s2)=O)N(C(=O)C(C)n2cccn2)C1 CC(CCCNC(C12COCC1C2)=O)NC(=O)CSS(C)(=O)=O N1(C(COCC#C)=O)CCC(NC(=O)CCCC2CC2C)C1 C1(C(N(CC(CN(C(CC=C)=O)C)O)C)=O)Cc2ccc(Br)cc2C(=O)O1 c1(CC)c(C(=O)NCC2CC2NC(c2ccoc2C)=O)cnn1-c1ccc(C)cc1 CCC(CC(=O)NCCC(C)NC(C1(C)CCCO1)=O)C1CCC1 C(=O)(N=c1cc[nH]c2ccc(Br)cc12)c1ccc(-c2cc(C#N)c(F)cc2)nn1 CCC(C)(C)C(O)C(=O)N1CCCC1C(C)NC(=O)CC(C)(C)COC CCCCC(=O)NCC1CCC1C(=O)NC(CCC)C1CC1 C(=O)(C1CCCc2cncn21)NC(CCCNC(c1c(C)cncc1)=O)C C1(N(C(=O)CCC2CCCO2)CC)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(CC(C)O)cn(CC(=O)NC2(CC(C)(C)C)CC2)nn1.C1CCC(=O)N1 Cc1ccnnc1C(=O)NC(C)C(c1ccccc1)NC(=O)C(C)N1CCCC1 CN1CCCCC1CCC(=O)NC1CCOCC1NC(c1cnsn1)=O C1(C)(CNC(c2c(CC)n[nH]c2)=O)CCC(NC(=O)CCc2nncn2C)C1 C1(NC(Cc2cc(OC)ncc2)=O)CN(C(c2ccc(C)s2)=O)CCC12CCC2 c1(C(C)NC(CCN(C(c2cnc(CC)s2)=O)CC)=O)[nH]c(C)nc1C Cc1c(NCCOC2CCCC2)ncnc1NCC1CC(C)OC(C)C1 c1(SCC)nccnc1C(=O)NCC12COC(CNC(=O)CC(F)(F)F)(C1)C2 C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(=O)COC2CCCCC2)CC1(C)C c1(C(=O)NC2(CO)CCN(C(C3CC(C#C)(O)C3)=O)C2)cc(F)c(O)c(F)c1 CCCC(CCC)CC(=O)N1CCOCC1CN(C)C(c1c[nH]cc(F)c1=O)=O Cc1nsc2ncc(C(=O)NCC(C3CCCC3)NC(=O)CC(O)C(C)C)cc12 c1(C(=O)NCCNC(C(C(C)SC)O)=O)ccc2nc(C(F)F)[nH]c2c1 CCC(CC)(C(=O)N1CCCC(NC(=O)CN2CCP(C)(=O)CC2)C1)OC C(C#N)(c1nc2ccccc2s1)=CCNC1Cc2c(nc(C)o2)CC1 CC1CN(C(=O)C(c2cn(C)nn2)NC(C2C=CCS2)=O)CC1CO C1(NC(C)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1.c12cn(nn1)CC2 c1(CC(=O)N(CC(C)NC(C2ON=C(CC)C2)=O)CC)csc2ccc(C)cc12 C(=O)(CC(C)NC(C1CCN(CCCO)C1)=O)OC c1(C(=O)NC(C)C=CC(=O)NC2CC(C(N)=O)C2)ccc(N)c(F)n1 c1(CC)cc(C(=O)N(CC(C)(C)NC(C2CC(SC)C2)=O)C)cc(O)n1 C1(CC(=O)NCCC(=O)OC(C)C)C2CN(C(c3cncn3C)=O)CC12 c1(NC(CC2CC(=O)OC2)=O)nc2c(s1)CC(C(=O)O)CC2 Cc1ccc2cc(C(=O)NCC3CC3NC(c3cccc(N)c3C)=O)[nH]c2c1 CC(C)CCC(=O)N(CC(C)NC(c1cnn(C(C)C)c1C1CCCC1)=O)C C1(C(=O)NCC2N(C(CC3(C=C)CCCCC3)=O)CCC2)CC2(CCCCC2)C1 C(=O)(CCCCCCCCCO)NC1CC(C)N(C(C2CC2F)=O)CC1 CCC(C)(C)CC(=O)NC12CCN(C(c3csc(-c4ccccc4)c3)=O)CC1C2 C1(OC)CN(C(=O)C=Cc2ccccc2)CC1NC(c1cccc(C)c1)=O Cc1c(CNC(=O)Nc2nnn(C)c2C(F)(F)F)cccc1O N1(C(CCSCCCC)=O)CCOC(C(C)NC(c2cc(COC)oc2C)=O)C1 C(=O)(C(C(C)C)Sc1cccs1)NC(C1(NC(c2c(C)cco2)=O)CC1)C N1(C(C2(C#C)CCCC2)=O)CCCC(F)(CNC(=O)CN(C(=O)C(C)C)C)C1 c1(C(=O)NCCCOCCN(C)C(c2cnc(S)nc2)=O)cc(F)cc(N)c1F Cc1ccnc(C(=O)NCC2(F)CCN(C(C3SCCS3)=O)C2)c1F C(=O)(C#CC1CCCCC1)N1C(CNC(=O)Cc2ccno2)CC(COC)C1 C#Cc1cc(F)c(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(F)c1 N1(c2[nH]c(=NCC3CC=CC3)cc(C)n2)CCc2c(ccc(Cl)c2F)C1 c1(OC)ccc(SC(C)C(N2CCC(NC(=O)C=CC3CCC3)C2)=O)cc1 N1(C(c2c(NC(c3ccc(O)cc3)=O)cccn2)=O)CCCC12CCCC2 C1(NC(c2c(I)ccnc2Cl)=O)CN(C(=O)Cc2ccc(Br)cc2F)CC1(F)F C=CC(C)(C)CCNC(=O)C(C)(CSC)NC(=O)C=C1CCC1 Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NC(CCO)C(C)(C)O)cc1O Cc1noc(C(F)F)c1C(=O)NC1CCCN(C(=O)CC2CCCN2C)C1 c1(C(N2CC3(CN(C(C4CC4C4CCCC4)=O)C3)C2)=O)sc2sccc2c1Cl c1(OC)cc(F)ccc1NC(=O)C(=O)NC1CCN(OCC)CC1 c1(C(=O)NC2(CCCNC(C(n3ccc(C)n3)C)=O)CC2)cc(C)c(Cl)s1 Cc1nn(CC(N2CCCCC2CN(C)C(C23CCC2CC3)=O)=O)cc1Cl c1(C2C(C(=O)NCCC(C)(C)NC(=O)C(F)C3CC3)C2)cccc2ccccc12 C(N=c1ccnc(NC2CCCC2C(C)C)[nH]1)c1ccc(NC(C)C)cc1 C1(c2ccccc2)(NC(C(COC)C)=O)CCN(C(c2cnsc2C)=O)C1 c1(OCC)ncc(C(=O)NC2(CNC(=O)CCc3cc[nH]n3)CCCC2)cn1 C(C)(N=c1[nH]nc(Cc2ccco2)o1)C1OCCN(C(CCC)=O)C1 C(=O)(C(CCC)S(N)(=O)=O)NCCC(=C)CNC(C1CCC(C)(C)C1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(=O)CCCCN(C)C C(CC(=O)C1=C(c2ccccc2)OCCC1)N(C)Cc1ccc(C#N)cc1O C#Cc1ccc(C)c(NC(C2C(C)CCN2C(C2CC3(CSC3)C2)=O)=O)c1 c1(C(NS(N(CC)CC)(=O)=O)C(=O)OC)cc(F)c(F)c(F)c1 Cc1nc2cccc(C(N3CCCC3C(C)NC(C3COCCO3)=O)=O)c2[nH]1 N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)C2=CS(=O)(=O)CCC2)C2CCCC2C1 N1(C(C#CC(C)(C)O)=O)CC2(CCC2)CC1CNC(=O)CCCn1cncn1 Cc1c[nH]nc1C(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnn(C)c1)C C#Cc1ccc(C)c(NC(=O)C(CC)NC(=O)CSCCC#N)c1 c1(C(=O)NCC2N(C(C=CC(=O)OCC)=O)CC2)c(C)c(C)cc(C)c1C C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(N2CCN(C(C)=O)CC2)=O)CC1(C)C N1(C(C23CC(OC)C2C3)=O)C2CCC1CN(C(c1cc(Cl)cnc1C)=O)C2 Cc1cnc(C=CC(N2CC(C(C)NC(=O)C=C3CCC(C)C3)C2)=O)[nH]1 Cc1c(C(=O)NCCCNC(=O)C(C)CC(N)=O)sc2[nH]cnc(=S)c12 C1(NC(c2ccn(CC)n2)=O)C2CC3CN(C(c4[nH]nc(OC)c4Cl)=O)C1C3C2 CCC(C)C(C)C(=O)N1CCCC(c2n[nH]c(CNC(=O)CCC(F)(F)F)n2)C1 c1(-c2cn(CC(CCNC(C3C(F)(F)C34CC4)=O)F)nn2)cccc(F)c1F Cc1cc(C(N2CCC(C3(C)N=N3)C2)C(=O)NCCC2(C)CC2)c(C)o1 CC1(C)CN(C(=O)CCC2CCCCN2C(=O)C#CC2CCC2)CCS1 c1(C(=O)NC2CC(CNC(C3(CC#C)CCOC3)=O)C2)cccc(N(C)C)c1 c1(C(C(=O)NC2C(CNC(C(C)=C(C)C)=O)C2)(F)F)ccc(C)cc1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 N#CC1(C(N2CC(CC(F)C(=O)NCC3(C4CCC4)CC3)C2)=O)CC2CC2C1 CC1(CNC(C2(C)CCCO2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC2C1CCN2C(c1cc[n+]([O-])cc1)=O CC1(C)CC(CNC(=O)Cc2c(F)cccc2Cl)N(C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NC2(CC=C)CN(C(c3ccsc3SC)=O)C2)n[nH]c2c1CCSC2 N(C(=NCCSc1ncc[nH]c1=O)NCC1CCCO1)C(CC)C N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)C(CO)C1 C12(C(N(OCC(=O)OC)C)=O)CC(C)(CN1C(C1CCC(=O)CC1C)=O)C2 c1(OCC(=O)OC)ccc(NC(=O)C(C(C)C)c2cc(C)no2)c2ccccc12 C1(=CCNC(c2scnc2Cl)=O)CCN(c2nc(Cc3ccccc3)ns2)CC1 CC(O)C(C(=O)NC1(C)CN(C(=O)CC(=O)NC2CC2)C1)NC(=O)C(C)(C)C CCCC(C#N)C(=O)NC1CC2(C1)CN(C(C1(NS(C)(=O)=O)CCCC1)=O)C2 C(CCC(O)C(=O)NCc1cccc(CO)c1)NC(c1cc[nH]c1)=O c1(C(CC)=O)cc(NC(=O)C(OC)OC)ccc1Cl.N12CCCC(C1CC)C2=O N1(C(C2CCN(C(c3cn(CC(C)C)nc3)=O)CC2)=O)CC(C)CCC1CO c1(C(CC)C)ccc(C(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)cc1 c1(CC(=O)N(CCNC(CC2(C)CC2(F)Cl)=O)CC2CC2)ccc2nn[nH]c2c1 N1(C(=O)CCc2c(Cl)cncc2Cl)CC2CCCC(C1)N2C(C1CCCO1)=O N1(C(C(SC)SC)=O)CCC(NC(=O)C(C)CC2CCCC2)C1C c1(C(N2CCCC(C)(CNC(C(CC)(C)CO)=O)C2)=O)cc2c(cn1)OCCC2 C1(C(=O)NC2CCN(C(=O)C(F)F)C(C3CCOCC3)C2)CC2CCC(C1)C2O N1(C(C2CCC(C)O2)=O)CC2(CC2)CC1CC(=O)NC1CCC2(C(C)C)CC12 C#Cc1ccccc1CN1CCC(C(=O)Nc2ccnc(-c3cccs3)c2)CC1 CCCC(CC)CCC(=O)N1CC2(CNC(=O)COC)CCC1C2 Cc1nc(NCCC2CCC2)cc(=NC(C)c2cnccc2C)[nH]1 N1(C(C(N2CCC(C)C2)=O)=O)CC2(CCCC(CNC(=O)C3=CCCC3)O2)C1 Cc1cc(C(N2CC(N3CC(NC(c4occc4C)=O)CC3=O)C2)=O)ccc1Cl c1(C(=O)NCC23CC2CN(C(=O)CC2CCCCO2)C3)cc(Cl)cc(Cl)c1O C(CN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1)OCC(c1ccccc1)C Cc1cc(NC(c2ccncc2Cl)c2nnnn2C(C)(C)C)ccc1F N1(C(c2ccnn2CCF)=O)CC2CCC1CN2C(C1CCn2nncc2C1)=O Cc1c(CNC(C)CC(C)(C)O)c(C(F)(F)F)nc2[nH]nc(O)c12 c1(-c2nn(CCOC(C)C)c(Cc3cccc(Cl)c3Cl)n2)cccc2scnc12 CCC(CCC(=O)NC(c1cscn1)CO)NC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC(CC)CNC(c2ccc(OC(C)(C)C)cc2)=O)ccc(F)cc1C N12CC(CC1(C)C)C2=O.C(CCCCCSC)n1cc(-c2cn(CC)nc2)nn1 C=CC(C)(O)CC(=O)NCC1CC(NC(=O)CCNS(C)(=O)=O)C1 CC1CC(CNC(C2CCC23CCC3)=O)CCN1C(c1ccco1)=O C1(C(C)NC(=O)C=CC(=O)N(C)C)CN(C(=O)CSC2CCOC2=O)CCO1 c1(C(N2CCC(N(C(=O)Cc3cnccc3Cl)C)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C(CC)c2ccccc2)=O)CC2CCOC2(CNC(=O)CC2CCC2C)C1 CC1CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)CN1C(c1cocn1)=O C1(NC(COCCOCC#C)=O)CCCCC12CCN(C(c1cnc[nH]1)=O)C2 N1(C(CC(CC)(F)F)=O)CC2CCN(C(C3Cc4nc(C)cn4C3)=O)CCC2C1 CCC(O)C(C)C(=O)N1CC2CC(C1)C2NC(=O)CCCCCN(C)C c1(C(=O)NC(C)CCNC(c2cnn(C)c2F)=O)ccc(N)cc1[N+](=O)[O-] CC(C1Cc2ccccc21)Nc1ccccc1OC(F)(F)Cl CCCC(CCC)=CC(=O)NCC1C(C)CCN1C(c1cnoc1)=O N1(C(CC2C(NC(C(CC=C)OC)=O)CC2O)=O)CCN(C)CC1CCO c1(OC)ccc(C(F)(F)C(=O)NCC2CCN(C(c3cc(C)co3)=O)C2)nc1 CCCCCC(O)C(=O)N1CCCC1C(C)NC(c1cccc2ccoc12)=O N1(C(C2(OC)CC(C)C2)=O)CCOCC(NC(c2ccn(C3CC3)n2)=O)C1 c1(NC(=O)NC(C(C)OC)Cc2ccc(C#N)cc2)ccc2ccccc2c1 c1(C(=O)NC2CC(O)C2)cc2[nH]ccc2cc1-c1cc(CO)ccn1 O=C(CCSCc1cc(Cl)ccc1Cl)N(O)Cc1cn(-c2cccnc2)nn1 CCN=C(NCC12CC(CC(F)F)(C1)C2)N1CC2CC=CCC2C1 C1(NC(c2cccc(Cl)c2)=O)CC2CCC(C1)N2C(=O)CCn1cncn1 CCCCC(CNC(C1CC(C)(C)CO1)=O)NC(=O)Cn1cc(CO)nn1 c1(OC)ccc(S(=O)(=O)N2CCc3c(ncn3C)C2C)cc1-c1cccc(F)c1 C1(CC(=O)N(CC(C)N(C(COCCOCC)=O)C)C)CCCCO1 C(c1ccc(Cl)cc1F)=CC(=O)N(CCNC(C1Cc2nncn2C1)=O)C1CC1 C1(N(C(c2scc(CC)c2)=O)CC)CCCN(C(C2C(C)C2C)=O)CC1 C1(C(=O)NC2CC2CNC(=O)Cc2cncc(F)c2)(OC)CCSCC1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC1CCCC(NC(=O)CSC(C)(C)C)C1 c1(C(=O)NCCC2N(C(C(CO)NC(N)=O)=O)CCCC2)nccc2n[nH]cc12 c1(C(=O)NC(CC)(C)CNC(=O)C(C2CC2)SC)cc2c(o1)CCCC2 N1(C(C=CC(C)C)=O)CCC2(CC1)CN(c1ncc3[nH]ccc3n1)CCO2 c1(CC)n[nH]c(CC)c1CC(=O)NC1CCN(C(=O)COC2CCCCC2)C1 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1(NC(=O)C(O)C2CCC2)C(C)CCCC1 c1(N(C)CC=CC=C2CCCC2)nc(=NCCSC(F)F)[nH]c2cc[nH]c12 N1(c2c(OC)cc(OC)c(Br)c2)C(=O)NC2(CC(C(C)(C)C)C2)C1=O O=S(=O)(c1c[nH]ccc1=NCCC(F)(F)F)NCc1ccccc1 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cnn3c2OCCC3)=O)CC(O)C1 C1(NC(Cc2cccc(CC)c2)=O)CCN(C(c2ocnc2C)=O)CC1C CC1=C(C(=O)NC2CCC(N(C)C(C3CC3C3CC3)=O)CC2)CCS1(=O)=O C1(C2CCN(C(C3(C)CC4CCC3C4)=O)C2)(NC(C(C)C2CC2)=O)CC1 Cc1cc(C(N2CCCC2CNC(C2CCCC(F)C2)=O)=O)c2c(c1)CCCN2 N1(C(CCOCC)=O)CC(N=c2[nH]ccn3nnnc23)C(C)(C)C1 c1(CC)nc(C)ncc1C(=O)NC1CN(C(c2c[nH]cc2C(C)C)=O)CC12CC2 C1(NC(c2cc(C)nc(O)c2)=O)CCCOC12CCN(c1nnco1)CC2 CCCC(C)(C)CC(=O)NC1CC(NC(C2(F)CCCN(C)C2)=O)C(O)C1 c1(C(=O)NC(C)CN(C)C(C2CCC(C)(C)OC2)=O)cc(Cl)c(Cl)cc1N c1(OC)ccc2c(=NCCC(N)=O)[nH]c(=NC3CC(CCF)C3)[nH]c2c1 CCCC(C)(O)C(=O)NCCOC1CCN(c2ncncc2I)C1 C#CC1(O)CCN(C(C2CCN(C(c3c[nH]nc3CCC)=O)C2C)=O)C1 c1(CC)nn(-c2ccccc2)cc1C(N1CCC(NC(=O)COCC)C1CC)=O C1(C(=O)NCC(F)(F)C(N)=O)(CNC(CC=CC)=O)CC12CCC2 Cc1ccc(C(N2CC(F)(F)CC2CCNC(C2CCN(C)C2=O)=O)=O)c(N)n1 c1(C(N(c2nc(C)c(F)cn2)C2CCNCC2F)=O)ccc2cccnc2c1 c1(CCC(=O)NCCC(C)NC(=O)C(C)NS(C)(=O)=O)nnc(-c2ccco2)o1 c1(C(N2CCC(N(C(c3cnn(CCC)c3C)=O)C)C2)=O)cnc(O)n(C)c1=O Cc1nn(C)c(C(F)F)c1C(=O)NC(CNC(C1(CO)CCCO1)=O)CC(C)C C1(NC(C2(C)CCOCC2)=O)Cc2ccccc2C1NC(c1cc[n+]([O-])cc1)=O c1(C(N2CCC(NC(COCCCC)=O)C(C)C2)=O)c(F)cc(C)cc1Cl C1(CNC(C2(C=C)CCC2)=O)C(C2CC2)CCN1C(=O)C(O)C(C)(C)CC C1(C(=O)OCC(=O)Nc2cc(Br)ccc2F)CC2(CCOC2)C1 Cc1sc2ncn(CCCC(=O)N(C(C)CNC(C3CC3C)=O)C)c(=O)c2c1C c1(C(=O)NC(CCN(C(C(C)OCCC=C)=O)C)C)cc(C(C)C)nc(O)c1 N1(C(CNC(C=C)=O)=O)CC(CNC(c2ccc(F)c(C)n2)=O)C2(CC2)C1 Cc1cc(CN2CCOCC2C(=O)Nc2ccc(Cl)cc2I)cc(C#N)c1 CCCC(C#N)C(=O)NC(C1CCN(C(=O)C=CCF)CC1)(C)C c1(C(N(CCN(C(C)C)C(C2C3COCC23)=O)C)=O)cc(C#N)ccc1Br C(=O)(C(C)S(C)(=O)=O)N1CC(OC)C(NC(c2cc(-c3ccoc3)[nH]n2)=O)C1 c1(C(=O)NCCC(CNC(c2cc3ccccn3n2)=O)O)ccc2nc[nH]c2c1 C1(CNC(=O)CCn2ccnn2)CCCC1C(=O)NCCCN1CCCC1 Cc1cc(N2CC3C(C2)C3(C)C)ncc1S(=O)(=O)NC1CC(C)n2ccnc21 O=CN1CCCC1C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CC(CO)C1 C(CNC(=O)CCCc1ncco1)(C(=O)NCCCC(F)F)N(C)C N1(C(C2C(CC(C)(C)C)C2)=O)CC2CCC(C1)N2C(C1(C2CCCO2)CC1)=O Cn1c(C(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cnc1[N+](=O)[O-] CC(C)C(C(=O)NC1C2CCC1CC2)C(C)NC(=O)CCc1cnn(C)c1 Cc1cc(=O)c(C(N2CCC(CN(C(=O)CSc3nncn3C)C)CC2)=O)c[nH]1 c1(OC)nc(Cl)ccc1C(=O)NC1CCCN(C(c2ccc(CO)nc2)=O)CC1 c1(COC)nc(CC(=O)NC2CC(CNC(=O)Cc3ccnn3C(C)C)C2)cs1 N1(C(C)C)CC2CC1CN(Cc1nscc1-c1nc(-c3cccc(Cl)c3)no1)C2 C1(F)(CNC(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2ccn(C)c2)=O)C1 CC1=C(C(=O)NCC2(O)CCN(C(C3C(C)(C)OC3(C)C)=O)C2)C(C)(C)CCC1 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(=O)C(=O)Nc2ncc[nH]2)C1C1CC1 c1(C(c2n(CC=C)c(N3CC(OCC)CC(F)C3)nn2)O)ccc2c(c1)COC2 C1(C(=O)N(C2(CO)CC2)C)(CC)CCCN(C(=O)CCN=[N+]=[N-])C1 c1(C(=O)NC2CCC(NC(C=NOC)=O)CC2)ccc2ccccc2c1 Cc1ccc(C(N2CC3C(CNC(c4cnc(Cl)s4)=O)C3C2)=O)c(F)c1F N1(C(c2c(NC)cncc2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(C(=O)NC(CCCC)(C)CO)CCN(C(=O)C(C)C(CC)CC)O1 C1(C(=O)OCC)(C(=O)NC2CCCC2NC(c2ccc(OC)s2)=O)CCCCC1 Cc1cn2c(CCC(N3CC4CC3(CNC(C3CCC(F)C3)=O)C4)=O)csc2n1 N1(c2nc(N3CC4CC3CS4=O)cc(C)n2)CC2(CCOCC2)CC1CO N1(C(C(=O)Nc2ncc[nH]2)=O)CC2CC1C2NC(c1ccccn1)=O c1(C(=O)NC(C2N(C(c3occ(C)c3)=O)CCCC2)C)c(C)nn(C)c1F N1(C(C(C(C)C)NC=O)=O)C(C(N2CC(N(C)C3CC3)C2)=O)C2CCCC12 N1(C(C2C(C)(C)C2)=O)CCC(N(C(=O)Cn2nccn2)CCO)C1 C1(NC(c2ccc(CC)o2)=O)CN(C(=O)Cn2cc(F)ccc2=O)CCC1F C12(C(=O)NC(CNC(c3c(C)cccc3)=O)CO)OCCCC1C2(F)F c1(OC)cc(N)ccc1C(=O)NC1CCC(CNC(C2CC=CCC2)=O)CC1 c1(-c2c(OC(N3CCN(C(C)=O)CC3)=O)cccc2)nccc(C(F)(F)F)n1 c1(C(=O)NCCC(C)OC(C)(C)C)ccc(NC(=O)C(F)=C2CCCC2)nc1 c1(C(N2C(C)CNC(=O)C2)=O)cc(O)nc2c1CN(C(C1CC1F)=O)CC2 Cn1cc(C(N2CCC(Oc3ccccn3)C2)CC2CCCC2)nn1 c1(C(N2CC(CC)(NC(c3ccncc3OC)=O)C2)=O)ccc2nccnc2n1 CC1NC(=O)OC12CN(C(=O)CC(C(F)(F)F)NC(=O)CC(Cl)Cl)C2 c1(C(=O)NC2CCC(NC(C3(C#C)CCC3)=O)C2)cc(Cl)c(Cl)s1 C1(CNC(C(C)OCCN(C)C)=O)N(C(C2CCC(=O)N2C)=O)CCCC1(C)C Cc1c(N)cc(C(N2CC3CC(NC(c4ncn(C)n4)=O)C3C2)=O)cc1N Cc1nn2c(C(=O)NCCNC(=O)Cc3cccc(Cl)c3Cl)c(C)nc2s1 c1(C(=O)NCCC2(NC(C(C3CCC(=O)N3)C)=O)CC2)ccc(Br)c(O)n1 C(C(CCC)C(=O)N1CC=CC1CF)NC(CC1C(CC)C1)=O c1(C(N(C(CNC(Cc2c(C)cnn2C)=O)C)C)=O)cc(F)cnc1O c1(CCC(=O)NC(C2CCCC2)CNC(c2ccoc2Cl)=O)cc(Cl)cs1 N1(C(C2(C)CNC(=O)C2)=O)CCC(O)C(NC(c2cccc(C3CC3)c2)=O)C1 N1(CCN(CCN(CC=C)C)C)CC(=O)N(CC2CCC3(CCC3)O2)C1=O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)Cc2cncn2C)C(C)C1 C#CC1(C(N2CCCOC(CC)C2)=O)CCN(C(=O)C=CC2CCCN2C)C1 C1(NC(C2(OCC)CCC2)=O)CN(C(C2CCOCC2(C)C)=O)CC2(CCC2)C1 Cc1ccc(C(=O)N(C)CC2(O)CCCN(C(c3ccccn3)=O)C2)nc1O c1(COC)nc(C)cc(=NC2CN(C(=O)CCn3cccnc3=O)CC2C)[nH]1 C1(C(N2CCC(F)(CNC(Cc3cncc(C)c3)=O)C2)=O)CC2(C1)CC(C)C2 N1(C(C(c2ccccc2)NC(c2ncn(CC)c2)=O)=O)CCOC(C)CC1 N1(C(Cn2c(=N)nn[nH]2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 N1(C(C2(C=C)CCC2)=O)CCCCC2(CCN(C(=O)Cc3cnns3)C2)C1 C(C(CO)(CO)NC(=O)C(C1CC1)OCC)N(C(CCCOCC)=O)C N1(C(C2(N(C)C)CCCC2)=O)CC2(C1)C(NC(=O)CN(C)C1CC1)CCS2(=O)=O C12(N(c3cnn(C)c3)C(N3CCC(C(C)O)C3)=O)CCCC1C2(F)F N1(C(CCCC(=O)NC(C)C)=O)CCC(NC(c2cn[nH]c2)=O)C(CO)CC1 c1(C(=O)NC(C(C)(C)NC(c2cn(CCOC)nc2C)=O)C)cc(O)nc(O)n1 N1(C(C2(CCOCC)CCC2)=O)CC(NC(=O)C(F)(F)COC)CC(O)C1 CC1(O)CCN(C(=O)C(O)C2CN(C(C3CC4CCC3CC4)=O)C2)CC1O C12(C(=O)NCC(CNC(c3cncc4nc[nH]c34)=O)O)C(=O)C3CCC1C2C3 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(c2ncoc2C2CC2)=O)C12CC2 C(=O)(CCC(C)(F)F)N1CCC(C(N(CC(C)C)C)=O)(CF)C1 c1(CC(N2CCC(O)(CN(C(C(C)NC3CC3)=O)C)C2)=O)cnn2c1CCCC2 n1(CC)nc(C)cc1C(=O)OC(c1nc(-c2ccccc2C)no1)COC N1(C(C2C(COC)C2)=O)CCN(C(c2cccc(C)c2Cl)=O)C(c2cn[nH]c2)C1 c1(C(N2CC(CC(C)NC(c3cc(Cl)on3)=O)C2)=O)sccc1CC#N C1(F)(C(N(C2(COC)CC2)C)=O)CCCN(C(C2(C)CCCCO2)=O)C1 c1(OC(C(=O)NC2CCN(C(CC(=O)OCC)=O)C2)(C)C)cc(Cl)ccc1F c1(C(C(=O)NCC2(C)CCN(C(CC3CC(C)C3)=O)C2)C)ccc2c(c1)OCO2 C(=O)(CC1=CCOCC1)N(C)CC1(CNC(c2ccn(C3CCC3)n2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1C(C)(C(=O)NC(C)CCC2CCCC2)C=CC1 CC1=C(C(=O)N2C(C(=O)Nc3cnc(CO)nc3C)CC2C)CCCO1 N1(C(C=CCCC)=O)CC(NC(=O)Cc2cnn(C)c2)CC12CCCC2 CCCC(CNC(=O)C=Cc1ccoc1)C(=O)NCc1ncc(CC)o1 c1(SC)nc(C(N2CC=CC2CNC(c2coc(C)n2)=O)=O)c2ccccn12 c1(OC)cc(I)c(Cl)cc1NC(=O)NC1(c2ccc(C(F)(F)F)cc2)CCCC1 N1(C(c2c(C)cc(Br)cc2)=O)CCc2c(C(N3CCCCC3C)=O)cccc2C1 c1(CC(N2CCC(NC(C3CCC(C)S3)=O)CC2)=O)ccc(S(N)(=O)=O)s1 Cc1cc(=NC(=O)C2CC(C)CN2C(c2cccc(Br)n2)=O)[nH]c(C)c1C#N N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)N2CCC(C)C(CO)C2)CC1 C12(CNC(=O)C3=CCCC3)CCC(Nc3ccnc(CO)n3)(CC1)CO2 c1(OC)ccc(CN=C(NCC(C)C#N)NCc2nnc(SC)s2)cc1 C1(CNC(CP(C)(C)=O)=O)CN(C(=O)CC2CCCCCCC2)CCCO1 N1(C(c2cc(C(=O)OC)on2)=O)C2CCC(C2)C1CNC(c1ccc([N+](=O)[O-])o1)=O c1(C(N2CC(C(=O)Nc3cc(OC)cc(C)c3)NCC2)=O)cc(Cl)c(O)cc1F c1(C(NC=O)C2CC2)cn(CC2CCCN2C(C2C=CCS2)=O)nn1 Cc1ccc2c(=NCCc3cccnc3C)[nH]c(=NC(C)C3CCCO3)[nH]c2c1 CC(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccoc2C)=O)CC1C)=O N1(C(CC(C)OC)=O)C2CCC(C2)C1C(=O)N(C)Cc1ccns1 c1(OCC)ccc(C(F)(F)F)cc1NC(=O)Nc1ccnn1C1CCOCC1 CN1CCCC1C(=O)NC(C)(CNC(C1CCSC1)=O)C1CC1 c1(C(=O)NC2CCC(C)(NC(C3(CC)CCC3)=O)CC2)c(OC)ccc(Cl)c1C C1(NC(CNC=O)=O)CCN(C2CCN(C(C3CC(F)(CO)C3)=O)CC2)CC1 CC1=C(C(=O)NC2CCN(C(C3CCCN3C)=O)C2)CCC1 N1(C(C)=O)CCCC1C(=O)NC1(C2CCCN2C(=O)C=CC(C)(C)C)CC1 C(=O)(C#CC1(C)CCCO1)NCC1C(NC(CC2CC(=C)C2)=O)COC1 c1(C(C)C)c(NC(C2(NC(=O)C(C)N3CCCC3)CCCC2)=O)cnn1C CCCCCC(CC)C(=O)N1CCCCC(NC(=O)Cc2c(C)cccc2C)C1 C=C=CC(C)C(=O)N1CC(OCCNC(=O)CC2CN(C)C2)C1 C(C1=CCN(C(=O)CCC2CC2)CC1)NC(C(c1ccccc1)NC(C)=O)=O N1(C(c2cc(Cl)ccc2O)=O)CCOC2(C1)CN(C(C1(C(F)F)CC1(F)F)=O)C2 Cc1cnc(C=CC(=O)NC2COCC2CNC(=O)CC2CSCCS2)[nH]1 CC(C)CC(C(=O)NC1COCCOC1)NC(=O)CC(C)N(C)C c1(C(N2CCC(C(N(CCCC(=O)OC)C)=O)CC2C)=O)cccn2nccc12 N1(C(c2n(CC)nnc2)=O)CCCC(C)(C(N2CC(C)(F)C2)=O)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(c2cncc(OC)n2)=O)C(C2CC2)C1 c1(C(=O)NCC(CNC(C2N(C(C)=O)CCOC2)=O)F)cn2c(n1)SCC2 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(c3n[nH]c(C)c3F)=O)C2)C1 C(CC)(CC)(CCNC(c1ccc(C(C)=O)cc1)=O)NC(C(CC=C)C)=O C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(NC(C(C)c2cccs2)=O)CC1 Cc1nn(C)c2c(NCCN3CCCC3C)nc(N3CC4C(C3)C4(C)C)nc12 c1(C(=O)NC2C(NC(C(COC)OC)=O)CCCC2)cccc2c1NCCC2 N1(C(CCC=C)=O)CCC(CNC(c2ccccc2SC(C)C)=O)C12CC2 N1(C(C(C)Cc2ccnn2C)=O)CCSCC1CCNC(c1cnsc1)=O C(=O)(C(C)(C)CCC#N)N1CC(C(C)NC(=O)CN2CCSCC2)OCC1 C1(NC(=O)NC(CN(CCCC)C)(C)C)CCCC(O)C1 C(CCO)(CC(C)C)NC(C1(NC(c2c(OC)nn(C)c2)=O)CC(O)C1)=O C1(C2CCCN(C(c3ccc(N)c(C)c3)=O)C2)(NC(C(CC)C(C)O)=O)CC1 CCC(O)C(C)(C)C(=O)NCC1CCN(C(c2c(C)ncn2O)=O)CC1(F)F C1(CNC(C2CCC(COC)C2)=O)CCN(C(=O)C=Cc2ccc(C)o2)C1(C)C N1(C(CNC(C2C(C)C2)=O)=O)CC=CC(NC(c2ccc(CC(N)=O)cc2)=O)C1 C1(C(=O)NC(C(=O)OCC)CC2CC2)CC2CC2N1C(=O)COCC(C)C c1(C(N2C(C)(CNC(C(C(C)C)OCC)=O)CCC2)=O)cc(=O)n2ccsc2n1 C1(c2cn(C3(COCCO)CC3)nn2)(NC(C2CCC=CCC2)=O)CCCOC1 c1(-c2cccc(CNC(c3ccco3)=O)c2)ccc(C(=O)OCCCC)nc1C C(C)(CCCC(=O)O)NCc1n(-c2c(OC)cccc2)ncc1 N1(C(C)=O)CCCC(N(CC(C(F)(F)F)N2CCCC2)C(=O)C(=O)OC(N)=O)CC1 C(=O)(CCC(C)CN(C)C)NCC1CN(C(CCCOC(C)=O)=O)CC1C c1(C(N(C(C)C)C)=O)cn2c(n1)CN(Cc1cc(F)c(Cl)nc1Cl)CC2 N1(C(c2n(CCC)ncc2)=O)CCCCC1CCNC(=O)C(C)C1CCCC1 C1(CC(N2CC=CC(NC(=O)Cc3cnn(C)c3)C2)=O)(OC)CCCCC1 c1(C(=O)NCCCc2cn(Cc3ccc(Cl)cc3)nn2)cn2cc(Cl)ccc2n1 c1(C(N2CCC(NC(COC(C)=O)=O)C2)=O)ccc2ncnc(O)c2c1 C(CCC(N)=O)(C(=O)NC1CCN(C(c2cc(F)c(Br)cc2C)=O)CC1F)OC c1(C(=O)NCC2(C)CC(NC(C3CCC(CC)CC3)=O)C2)nc(C)c(C)nc1C c1(C(=O)NC(CCCC)CNC(C2(C)COCCO2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCCC2CC(NC(CSCCC(C)C)=O)C2)cn2c(n1)CCC(C)C2 c1(C(C(=O)NCC(=C)C)N(c2ccccc2)CCCC)cncc2ccccc12 c1(C(=O)NC2C(OC)CN(C(c3ccc(C#N)o3)=O)C2)cc(F)c(F)cc1Cl N1(C(C(C(=C)C)(C)C)=O)CC2CC(C(=O)NCc3ncnn3C3CC3)CC2C1 n1(CN(C)C)ccc(=NC(c2csc(Cl)c2Br)c2nnnn2CC2CCOC2)[nH]1 Cn1ccc2ccnc(C(=O)NCC3CCCN(C(C4(C)CC=CC4)=O)C3)c12 N1(C(C=CC)=O)CCN(C(c2cc(-c3ccccc3C)on2)=O)C2CCCCC12 N1(C(c2c(C)snn2)=O)CC(CC(=O)N(C(C)CO)C2CC2)C2(CC2)C1 N1(CC)CCOC(C(=O)NCC=CCNC(=O)CCc2ncc[nH]2)C1 C(CNC(C1CCN(c2ccccc2F)C1)=O)(C(F)(F)F)OC C1(F)(CNC(C2CCSC2)=O)CN(C(=O)CCc2nc(-c3ccccc3)no2)C1 c1(CNC2CC(NC(=O)Nc3c(C)cccc3C(N)=O)C2)c(Br)cc(F)cc1Br CC1CCN(CCC(N2CC3C(CNC(C4CC(Cl)(Cl)C4)=O)C3C2)=O)CC1 C1(NC(c2scnc2C2CC2)=O)CCOCC1NC(c1ncccc1F)=O c1(CC(=O)NCC(C)(O)CNC(C2CCSC2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)NC(CC)CN(C)C(C2(N(C)C)CCCC2)=O)CCCC12CC2 Cc1ccc2c(N3CCC4(CC3)CC(NC(=O)C(O)C(C)C)C4)ncnc2c1 c1(CC(=O)NCCCOCCNC(C2COC(=O)O2)=O)ccsc1Br C12(C(=O)NC)CCC(Cn3ncc(C(=O)NCC4C(C)=NNC4=O)c3)(CC1)OC2 c1(CC)c(C(=O)NC2(CF)CCCC2)cnn1CC.C1(O)CCCC1 C1(C(N(CCN(C(=O)CC2C=CCCC2)C)C)=O)Cc2ccccc2O1 C1(C(N2CCC(C)C2(C)C)=O)COc2cccc(F)c2O1 c1(C(N(C(C)CNC(C2CC2(C)C)=O)CC)=O)cnc(C(F)(F)F)s1 c1(C2CCN(C(C(CCCC)NC)=O)CC2)nc2ccccc2[nH]1 N(C(=NCCOC(F)F)NCC1(C#N)CC1)C(C1CCOCC1)C C(=O)(C1=C(CC)OCCC1)NCCCN(C(C1(C#N)CCCOC1)=O)CC c1(C(N2CCC(CCOC)C2)=O)[nH]c(Cl)c(Cl)c1Br C1(NC(C(C)(C)CF)=O)COC2(CCN(C(C3CC3c3cccnc3)=O)CC2)C1 Cc1csc2ncc(C(=O)NCCCN(C(=O)C=Cc3ccoc3)C)n12 c1(C(N2CC(C)N(C(=O)C(=Cc3cccn3C)F)CC2)=O)cnc2cc[nH]c2c1 C1(C(N2CC(NC(CCc3ccc(C)s3)=O)C(O)C2)=O)CC12CCCCCC2 C1(NC(CNC(CNC(C=C(C)C(C)C)=O)=O)=O)CN(C)C2(CCC2)C1 c1(C(N2C(C(=O)Nc3c(C)cc(F)nc3)C3CCC2C3)=O)cc2cccnc2[nH]1 c1(OCCC(=O)NC2(CN(C(=O)C(C)(O)C3CCOC3)C)CC2)ccc(Cl)cc1 n1(C(C)C)cc(C(=O)NCCCN(C2CCCC2)C(c2ccon2)=O)cn1 C1(C(=O)NC(CNC(CCC=CCC=C)=O)C(C)C)C2CCC1CC2 c1(C(N(CCC(C(C)C)NC(C2CC(O)(CC#C)C2)=O)C)=O)csc2nccn12 c1(CC(=O)NC2(CN(C(C3C(OC)CC3)=O)C)CC2)n[nH]c2ccccc12 N(C1CCc2cccnc21)C(C1N(C(c2ccc(OCC)cc2I)=O)CC1)=O C1(NC(CC2CC(COC)C2)=O)CN(C(c2cc3n(n2)CCO3)=O)CC12CC2 C=CC1COCCN1C(C12CC1CCN2C(c1cc[nH]c1)=O)=O c1(CNC2C(NC(C3CCN(C(C)=O)CC3)=O)CCCC2)c(F)ccc(F)c1O N1(C(C2CCC(=O)C2)=O)CCCN(C(C2OCC3COCCC23)=O)CCC1 C1(O)(CNC(c2cc(Br)ncc2Br)=O)CCCN(C(c2cnnc(O)c2)=O)C1 Cc1ccc(CNC(c2cc(CNC(=O)CCOC3CCCC3)cs2)=O)cc1C n1(CCCC(=O)N(CC)CC2CCCN2C(=O)CCCSC)nc(C)cc1C CC1CCC(C2CCC2)CN1C(=O)C(N1CC(C)(Cc2ccccc2)C1)=O C1(C(=O)NC(COC)C(=O)N(C)Cc2nncs2)C2CC3C(C2=O)C13 C(=O)(C(=O)N=S(C)(C)=O)NCC1(C)CCCN(C(CSc2n(C)cnn2)=O)C1 c1(CN2CCCC(NC(c3cccc(Cl)c3Cl)=O)C2)cc(F)c(Br)cc1[N+](=O)[O-] CCC(C)(C)C(=O)N1CC(NC(=O)CCc2ncco2)C(c2cncn2C)C1 c1(C(N2CC(CNC(=O)OCc3ccccc3)C2)=O)cc(F)cc(F)c1F CC1Cc2ccccc2C1NC(c1cc(Oc2ccc(F)cc2)cs1)=O C(=O)(C(C)CCCC(C)=O)NC(COCC)C(N1CCCC2(C=CCO2)C1)=O c1(NC(c2cc(OC)ncc2-c2ccncc2OC)=O)cc(F)c2cc[nH]c2c1 C(=O)(C(C(C)C)n1cccc1)NCC(CC)NC(c1cc(Cl)ccn1)=O CC(F)(F)CCC(=O)NCCOCCC(=O)NCc1ncnn1C1CC1 N1(CC(=O)NCCCCCC)CCC(NC(c2csnn2)=O)C(C)(C)C1 c1(C(C)C)ccc(C(=O)NCC2CC(O)CN2C(=O)CC2CCCCC2O)nc1 CCCCCCC(CC)C(=O)NC1CCCC1(C)NC(=O)C=Cc1ccsc1 Cc1cc2c(cc1C)OC(C(=O)NC1CC(O)CN(C(=O)CCP(C)(C)=O)C1)C2 N1(C(c2c(O)cccc2Cl)=O)CCCC2C1CCN2Cc1cc(O)cc(F)c1 C1(C(N2CCC(CC=C)C2)=O)CN(C(=O)CC2(O)CCCCC2)CCO1 c1(NCCc2c(OC)nccc2)[nH]c(=NCCn2cc(C)cn2)nc2sccc12 C1(NC(c2ccc(OC)c(Br)c2)=O)CC2CC1CN(C(=O)CNC=O)C2 N1(C(c2nc(NC(C)=O)sc2)=O)CC(CNC(C2(N(C)C)CCC2)=O)CC1C C(=O)(CS(=O)(=O)c1ccccc1C)NCC1CC2(CN(C(C(F)=C(C)C)=O)C2)C1 O=C(C(Cc1ccccc1)C(F)(F)F)NC1CC2OCCC12 C1(NC(C(=O)N(C)Cc2ccc(OC)cc2)=O)CC2(CCCCO2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccc(CN(C)C)o2)=O)C2CCCCC12 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(=O)CCC(N)=O)CC12CCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(=O)CCC(F)F)COCC1 C1(CNC(CCCNC(C)=O)=O)CN(C(c2ccnc(N(C)C)c2)=O)CCN1C C1(CO)CC(N=c2nc3sccc3c(NCCc3ccc(C)c([N+](=O)[O-])c3)[nH]2)C1 c1(N2C(CCNC(C3CCC(OC)CC3)=O)CCC2)nc(Cl)nc2c1ncn2C Cc1cc(-c2nc(C(=O)NCc3ccc(C(C)C)cc3)ccc2F)cnc1O N1(C(C2C(CC)C2)=O)CC(NC(C2CNC(=O)N2)=O)C2CCCCC12 CS(=O)(=O)c1cccc(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)c1 N1(C(C(CCC)O)=O)CC2CCC(CNC(=O)Cn3cccnc3=O)(C2)C1 C#CCCCC(C)C(=O)NCC(C)N(C(=O)CCCN1C(=O)CN(C)C1=O)C Cc1cc(C(=O)NC(CNC(=O)COCc2nnc(S)n2C)C2CC2)c(C)s1 N1(CCC)C(=O)CCC1C(N1CC(NC(c2cnn(CC)c2CC)=O)C(C)C1)=O CN1CC(C(=O)NCCCC2CCN(C(C3CC(O)(C(F)F)C3)=O)CC2)CC1=O Cc1ccc(F)c(C(=O)NC(C)CCCNC(C2CC2C(C)C)=O)c1F c1(C(N(CCCCNC(=O)CC2OCCC2(C)C)C)=O)cccn2[nH]c(=N)nc12 C1(C2(O)CN(C(=O)CCCC(F)F)C2)(CNC(c2c[nH]c(=N)o2)=O)CC1 c1(C(N2CC(OC)(CNC(C3CCCC(C)CC3)=O)C2)=O)cc(Cl)c(Cl)cc1N CC1CCCC=C1C(=O)NC1(CN(C(=O)C2=CCCCCC2)C)CC1 C1(CCC=C)CCCCN1C(=O)CCCN(C(=O)COCC(=O)NC)C(C)C N1(C(C2CCC(C(N)=O)O2)=O)CC2CCN(C(c3n[nH]cc3Cl)=O)C(C2)C1 C=CCC(C(=O)NC(C(N1CCC(OCCO)C1)=O)c1cccs1)C(C)C C1(CNC(C(C)(c2ccccc2)OC)=O)C(C)CCCN1C(c1conc1C)=O N1(c2nnc(C)o2)CCCC1C1CCCCN1C(=O)CC1(N(C)C)CCCCC1 CC1(F)CCC(NC(CC2CCCCC2)CO)CC1 C1(NC(=O)CC2(CNC(C3CC=CC3)=O)CC2)CC(Cl)(Cl)C1 c1(C(c2n(C(C)C)nnn2)NC2CC2c2cccc(Br)c2)cc2ccncc2s1 C=CCCCCCC(=O)NCC1CC2(CCC2)CN1C(=O)CC(F)(F)F c1(C(=O)NCC2C(C)CN(C(C3CCNC3=O)=O)C2)cc(Br)c(C#N)s1 c1(C(=O)NCC2(F)CC(NC(CS(CC)(=O)=O)=O)C2)cc2ccc(F)cc2o1 c1(CC)oncc1C(=O)NCC(CO)NC(c1ccc(-c2ccco2)s1)=O N1(C(c2cnc(C)s2)=O)CCOC(CCNC(C2CCCC2(C)C)=O)C1 C12(NC(c3sc4cccnc4c3Cl)=O)CCCCC1CN(C(=O)C=CCO)C2 C(CC(=O)NCCN(CCO)C1CC1)NS(C)(=O)=O.C1CC1F C1(NC(c2n(C=C)ncc2)=O)(CC)CCOC(C(F)(F)F)C1.C1(CC(C)C)C(=O)N1 C12(C(=O)Nc3cc(C)c(NC(C4CC(O)CN4C)=O)cc3)CCC(CC1)C2(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CC(C)(NC(c2c(Cl)cccc2[N+](=O)[O-])=O)C1 C1(NC(c2cscn2)=O)CCN(C(c2ccns2)=O)CC1O N1(C(C(C)=C2CC2)=O)CCC(CNc2nccc(CO)n2)C(F)(F)CC1 C1(C(N(CCC(=O)NCC2(C)CC3CC3C2)CC2CC2)=O)CC2(CCC2)CO1 N1(C(C2CN(C(CN(C)C(N)=O)=O)CC2F)=O)CCC12CCC(O)CC2 C1(C(=O)NC(COC(C)=O)CO)C2CC1N(C(C1CCCSC1C)=O)C2 C1(CCC(C)C)C(=O)NC(=O)NC2CCN1C2.C1(C)CC(=O)N1.C=CCOC C(CCCCCOC(C)C(=O)OC)NC(=O)CNCCOC.NCC.CCCC c1(C(=O)NCC2C3CN(Cc4c(OC)ccnc4)CC32)nccc2ccccc12 c1(C(=O)NCC2=CCN(C(C3CCC(C)(C)CO3)=O)CC2)cnc2n1CCOC2 C1CCCC(=O)N(c2ccccc2)C(=O)C2CC2C(=O)N1C.C(C(C)(C)C)SC N1(C(c2cc(C)nn2C)=O)CC2CC(CNC(=O)Cc3ccc(Cl)c(F)c3)C2C1 C(=O)(C1CCCc2nncn21)N1CCN(C(CNC(C(C)CC(N)=O)=O)=O)CC1 c1(C(N2CCC(CN(CCC)C)C2)=O)c(C)nn(CC(F)F)c1C Cc1cc(F)c(CNC(c2conc2-c2ccccc2)=O)nc1Cl C1(CCC)CN(C(c2nc(C)nn2C)=O)CCN1C(=O)Cc1c[nH]ccc1=O c1(C(=O)O)cc(S(=O)(=O)N2CC3(CN(C(C4C5COCC45)=O)C3)C2)ccc1Cl CC1CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1CNC(C1(C)CCOC(C)C1)=O C1(CNC(CCS(=O)(=O)N(C)C)=O)CCC2(CN(C(C3CCOCC3)=O)C2)O1 Cc1cnc(Cl)[nH]c1=NCCCCNC(C1CCC(NC(=O)OC(C)(C)C)CC1)=O C1(NC(C(C)CC#N)=O)CN(C(=O)CC2CCC2)C2(CCC2)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnn(C)n3)=O)C2)=O)cc(F)c1 C=CCCC(F)(F)C(=O)NC1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C1 c1(C(=O)NC(CN(C(C2CC2F)=O)CC)C)ccc2c(n1)OCC(=O)N2 c1(C(=O)NC(CCNC(c2ccc(OC)cc2C)=O)(C)C)cc2c(ncn2C)[nH]1 C1(CC)(CC)CC(NC(=O)CC(c2ccc(F)cc2)C)CN1C(c1cnco1)=O C1(C(N(C)Cc2ccc(CC)o2)=O)(CNC(c2cnc(Cl)s2)=O)CC12CCC2 C(C)(CC1=CCCCC1)NC(C(CC)NC(=O)CCc1nccs1)=O C1(CC)CC(C)CN(C(=O)Nc2ccc(Br)cc2SC)C1 N1(C(CCN=[N+]=[N-])=O)CC2(CCNC(C34CCCC3C4)=O)CCC1CC2 N1(C(C(CCC)F)=O)CCC(NC(c2ccc(OC)cc2F)=O)C(CO)C1 c1(OC)cc(C)cc(C(=O)NC2CCCCCN(C(=O)C(F)=CC3CC3)C2)c1C C1(C(=O)OC)CCN(C(C2(CNC(c3cc[nH]n3)=O)CC=CC2)=O)C1C N(C1CN(C(=O)COCCSC)Cc2ccccc21)C(CC(C=C)CC)=O C1(=O)C(=O)NCCCC2(CC2)N1.CC1CC1NC(=O)CC1(N(C(C)C)C)CC1 c1(C(N2CC(C(=O)Nc3nc(SC)nc(O)c3)NCC2)=O)cc(Cl)cc(Br)c1O c1(C(=O)OCc2cc(C(=O)OCC)n(C)n2)c(C)nn(CCOC)c1C C1(CNC(C=CCOC)=O)CCC2(CN(C(c3ccc(C(C)=O)cc3)=O)C2)O1 c1(C(N2CCCC(CNC(CCCCOC)=O)C2)=O)nn2c(c1C)CCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CC)CCNC(=O)C(C#N)CC N1(C(C(=Cc2ccco2)C)=O)CCN(C(=O)Cc2csnn2)C2CCCC2(C)C1 C1(C(=O)OCC)CCCC(C(=O)N(CCNC(c2csc(C)c2C)=O)C(C)C)C1 C1(CNC(C2CC3CCCC23)=O)CC2CCC1N2C(C1CC1(F)F)=O c1(-c2n(-c3c(OC)cccc3)nc(C)n2)ccc(=O)n(CC(F)(F)F)c1 Cc1ccc(C(=O)NCC2CC3CN(C(C4CC4(C)C)=O)CC23)cc1F C1(O)(C(=O)NCC2C(CNC(C(COC(C)=O)C)=O)C2)CN2CCC1CC2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(=O)C(C(C)(C)C)N(C)C)CC2C1 C(=O)(C1=NOC2(CCC2)C1)NC1(C)CCN(C(C2CC(C)SCC2)=O)CC1 C1(CNC(c2cnc(C)s2)=O)COCC2(CCN(C(=O)C(N)=O)C2)O1 C12(Nc3cc(C)ncn3)CCCN(C(c3c(C)cc(F)cc3C)=O)CC1C2 N1(C(CNC(C)=O)=O)CC2CCN(C(=O)C(=Cc3ccccn3)C)CC2C1 c1(OC)ncccc1C(=O)C(=O)NCCNC(c1nocc1-c1ccccc1)=O Cc1nc(CO)ncc1C(=O)NC1(C)CCCN(C(=O)C(c2cnccn2)C)C1 c1(CN2CCCC(C(=O)Nc3nnc(Br)s3)CC2)ccc(F)c(Br)c1F N1(C(c2cn(C)nc2Cl)=O)CCC(NC(c2ccc(F)cc2O)=O)C(CO)C1 Cc1cc(C)c(-c2nc(Cc3ccccc3F)no2)cn1 c1(CC)cc(C(=O)NCCCN(C(c2ncnc(C)c2C)=O)C2CC2)cc(F)c1 O=C1CC(CC(=O)NC23CC(NC(C4CCCCC4(F)F)=O)(C2)C3)=NN1 C=C1CC2CC1CN2C(=O)C(C)(CSC)NC(=O)CC1CCC(C)(C)O1 c1(OCc2cn(Cc3cc(SC)nn3C)nn2)ccccc1C#N C(=O)(C1=NOC2(CCC2)C1)N1CCC(COC)(CNC(=O)C2CC2)CC1 C(=O)(C(C)CC(N)=O)NC(C1(O)CN(C(CC2(OC)CC2)=O)C1)C C(C(N=c1[nH]nc(C#N)s1)C1CCC1)NC(C1C(c2ccccc2)(C)C1)=O c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)(C)C)C2)=O)ccc(CC)cc1 Cn1cc(C#CCNC(=O)NC2(c3cccc(Br)c3)CCC2)cn1 c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)C(C)C)ccc(C#N)c(F)c1 c1(C(N(C(C)CNC(c2ccnc(C3CC3)n2)=O)C)=O)ccc(S(C)=O)cc1 C1(NC(CC(=O)NCC)=O)CCCN(C(C2CCSCC2)=O)CC1 N1(C(C2CCC(=O)N2)=O)CCOC(CCNC(c2cccc(C(F)(F)F)n2)=O)C1 c1(C(N2C(C(C)C)C(NC(C3CCC(C)O3)=O)CC2)=O)ccn2nnnc2c1 Cc1c(C(=O)NCC2CCC2NC(=O)CCCc2ccccn2)cncc1N C12(C(=O)Oc3nc(C)sc3C)CCC(CC1)N2C(=O)OC(C)(C)C N1(C(CC(C(C)C)C)=O)CCC(CNC(c2cncc(C(F)F)c2)=O)C(F)(F)C1 c1(C(=O)NCCn2ncc(C(=O)NCCC3ON=C(C)C3)c2)ncc(C)cc1C C1(C(N(C)CC2CCCN(C(COCC#C)=O)C2)=O)CN2CCN1CC2 C1(Cn2ncc(Cl)c2)CN(N2CCC(CN3CCCCC3)CC2)C1 c1(C(=O)NCCC(C(C)C)NC(CC(=O)OCC)=O)cc(OC)c(OC)c(Cl)c1 S(=O)(=O)(c1cc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=CCSC2)c(C)o1)NC C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2scnc2C(F)(F)F)=O)CC1F Cc1ccc(N)cc1C(=O)NCC(F)CNC(c1coc(C(F)F)c1)=O C12(C(=O)NC(CC)CNC(c3ncc(N(C)C)cn3)=O)CC1COC2(C)C N1(C(CCC(C)(C)NC(Cc2cnc(C)s2)=O)=O)Cc2n[nH]cc2C1CO C1(C(=O)NC2(CCNC(=O)CCCC3CCCCC3)CCC2)COC2(CCC2)C1 CC1CC(C(=O)NCC2CCCCC2NC(C2CCOC(C(C)C)C2)=O)=NO1 C1(NC(C(C)S(N)(=O)=O)=O)CCN(C(c2n[nH]cc2Br)=O)CC1(C)C CCCCC(O)CC(=O)N(C1CCCN(C(=O)CCc2ccc(C)c(C)c2)C1)C c1(-n2c(C(c3c(COC)ocn3)NCCCCF)nnn2)c(C)cccc1C N1(C(CC(CC=C)(C)C)=O)CC2CC(C)N(C(C3CCCN3C3CC3)=O)C2C1 CCCC(CCCNC(c1ccc(CC(C)(C)C)cc1)=O)NC(=O)C=CC=C(C)C N1(C(CCOCC)=O)CCN(C(=O)CC2OC(C)(C)OC2=O)CC1C1CCCC1 CC1CN(C(c2coc(Cl)n2)=O)CC1NC(c1cnc(OC2CCOCC2)cn1)=O c1(N(C)CCc2ccccc2)nnc(-c2cnc(C3CC3)[nH]2)n1CC(=O)N(C)C N1(C(C(C(C)C)n2cnnn2)=O)CCN(C(c2cc(=O)n(C)o2)=O)C(C)C1 C1(C(N2CC(N(C(=O)CSC3CCOCC3)C)C2)=O)CCC2(CCC2)O1 CON1CCC(C(=O)NC2CC(O)C2CC(=O)NCC2CC=CC2)CC1 C1(O)(CN(C(C=CCOC)=O)C)CCCN(C(c2cc(C(F)(F)F)ns2)=O)C1 CC(C)C(C)C(C)CC(=O)NC1CCCC1CNc1ncccc1S(C)(=O)=O N1(C(CNC(CN(C(CNC(=O)NC)=O)C2CCC2)=O)=O)CCCC1CF CN1CCCN(C(=O)C(C(C)(C)C)NC(c2ccc[nH]2)=O)CC1 C1(CC)(CC)CC(NC(c2cc(O)n(C)n2)=O)CN1C(=O)CSC1CCOC1=O C1(C(=O)NCCCCC(CO)NC(CC=CC=C)=O)CCc2ncccc2C1 C(CN=c1[nH]ncnc1I)(N(C(C(C(CC)O)C)=O)C)C1CC1 CC(C)C(F)(CNC(=O)CCC(CF)CF)C(=O)N(C(C)CC(=O)OC)C C=CCCC(F)(F)C(=O)N(CCCCCNC(c1cc(Cl)cs1)=O)C N1(c2nnc(CSC)n2CC2CCOC2)CCc2c(ccnc2Cl)C1 Cn1cnc2nc(NC3CC(F)(CNC(=O)Cc4ccc(F)cn4)C3)ncc12 N1(C(C(CC)Sc2ccccc2)=O)CC2CC(C)N(C(=O)CSC(F)F)C2C1 c1(C(N2CC(NC(=O)C=CC3CCCC3)C(F)C2)=O)cc(Cl)c(Cl)cn1 N1(C(C2=C(C)OCC2)=O)CC2(CCCC2NC(C2CS(=O)C2)=O)C1 C(=O)(C1=C(Cl)CCC(C)C1)NCC#CCNC(c1c(C)oc(Cl)n1)=O C(c1ccc(Cl)cc1F)=CC(=O)NC(C(C)C)C(=O)N1C(C)C1C c1(C(=O)NCC2CC(OC)CN2C(c2ccc(O)nn2)=O)csc(=NC2CC2)[nH]1 N1(C(C2C(Br)(C(=O)OCC)C2)=O)CC(C)(c2cn(Cc3csc(C)n3)nn2)C1 C12(C(=O)NC(C)(CNC(c3ccoc3C3CC3)=O)CO)CCCC1CC(=O)C2 c1(NC2C(C)CN(C(C3Cc4cscc4C3)=O)CC2C)ccc2c(n1)CCC2=O c1(SCC)ccc([N+](=O)[O-])cc1C(N1CC(Nc2ccoc2)C(C)C1)=O Cc1ccc(OC)cc1.c12nc(cs1)C(=O)NC1(CCCC1)CNC(=O)COC2=O CC1CCCC(C(=O)NCc2ncccc2C(F)(F)F)O1 CCC(CC(=O)NC1(CCCOC)CCCCC1)NC(=O)C(C)SC c1(C(=O)NCC(C)(CO)NC(c2ccnc(O)c2)=O)cc2n(c1)CCCNC2=O C(=O)(C(C(C)C)NC(=O)NC1(c2ccc(OC)cc2)CC1)OCC N1(C(CCC(=O)OC)=O)CCCC(O)(CN(C(=O)CN(C)S(=O)(=O)N(C)C)C)C1 C12(CNC(c3csnn3)=O)CCCC1CN(C(=O)Cc1cccc(O)c1)C2 c1(CC(N2CCN(C(c3c(C)ccc(O)c3)=O)C(C)C2)=O)cccc2c1OCO2 C1(N(CC(=O)NC2CCCNC2)C)CCN(CC(F)F)CC1 c1(C(N2C(C)C(NC(=O)Cc3ccoc3)CC2)=O)coc2c1NC(=O)CCC2 Cc1nc2ccnn2c(C)c1C(=O)NCC1COCCN1C(=O)C(C)NC(N)=O C1(CC)CN(C(c2ccccc2Br)C(=O)NC2CCC2)CC(C)O1 N1(C(CN(C)CC)=O)CC(NC(C23CC(CC)(CO2)C3)=O)C(F)C1 N1(C(c2c(CNC(C3CC4(CC4)CO3)=O)cco2)=O)C2COCC1C2 c1(SCC(=O)NC2CN(C(c3nc(C(C)C)oc3)=O)C2)nc2ccccc2[nH]1 c1(C(=O)OC)ccc(Br)cc1C(N1CCC(CN=c2ccnc[nH]2)CC1)=O C1(C(C)C)CN(C(C2COCC2C(N)=O)=O)CC1C(N1CC(SC(F)F)C1)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CO)NC(C1CCSC1)=O C(=O)(N1CCCc2nncn21)C1CC(CNC(c2cccc(C#N)c2)=O)OC1 N1(C(c2ccn(CC)n2)=O)CCN(C(=O)CCC=C2CCC2)CC1 N#Cc1nccc2cc(NC(C3CN(c4ccccn4)C3)=O)ccc12 C(=O)(CC(F)(F)C(C)C)NCCN(C(=O)CCN1CCCC(C(=O)OC)C1)CC C(C(C)(C)CC(=O)NC1(CCCCNC(=O)COc2cccc(C#N)c2)CC1)OC C1(C(=O)NC(C)CC2CCCCC2)CC2(CCN1C(=O)C(C)C(F)(F)F)CC2 N1(C(C2NCCC23CC3)=O)Cc2ccccc2CC12CCC2 N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1C(=O)Nc1csnc1OC N1(C(c2cccc(CC)c2)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)C(C)C1 C=CC(C)(CCOC)C(=O)NCC(CCNC(c1cc(C(C)(C)C)no1)=O)OC C(CCN=C(NC(c1cccs1)=O)NC1CC(=O)N(CCC(F)(F)F)C1)=CC=C c1(C(N(C)CCNC(C2CCC3CC3CC2)=O)=O)ccc2sc(=N)[nH]c2c1 Nc1cc(C(=O)NC2CCC2C(=O)NC2CC(CO)(CO)C2)cc(F)c1 Cc1ncncc1NC1(c2nnnn2CC(F)F)CC2CC2C1 N1(C(C(CCC=C)(C)C)=O)CC2COCCC2(NC(C2CCCNC2=O)=O)C1 C1(C)(C(=O)NCC(CC)NC(c2c[nH]nc2-c2cccnc2)=O)CC=CCC1 C1(OC)(CO)CN(C(=O)CN(C)C(C2(CO)CCOC2)=O)C1 c1(C(C)C)ccc(C(C)CC(=O)N(C)CCNC(=O)C=CC2CCCN2C)cc1 c1(CC)c(C(=O)NC2CCCCC2NC(=O)CC2CCCCN2CC)nnn1C Cc1nc(C(=O)N(C(C)(C)CC(=O)N2CC(F)(C#N)C2)C)sc1C C1(S(N)(=O)=O)(C(=O)NC2C(CNC(C(C)OCCC(C)C)=O)COC2)CC1 N1(C(C(CC)CC)=O)CC2CN(C)CCC2(CO)C1 c1(CC)cc(C(=O)NCCOC(C)(C)CNC(c2cscc2F)=O)ccc1C c1(C(N2C(C)CC(NC(C(CC)CC3CCCCC3)=O)C2)=O)c[nH]c(=N)cc1C C1(NC(C2(F)CCOC2)=O)CC2(C1)CC(CN=c1nc(C3CCOCC3)[nH]s1)C2 c1(C(CN)O)ccccc1Br.CC(C(CO)c1ccccc1)c1ccccc1 Cc1cc(Cl)ccc1C(N1CC(N(C(=O)C2=COCCO2)C)C(O)C1)=O C1(OCC)CC2(C1)CC2C(N1CC(CC(C)NC(=O)C(C)(F)F)C1)=O Cc1ccc2c(c1)C(NC1CCCCN1C(c1ccoc1)=O)CCCO2 c1(C(CC2CC2)NC(c2nnnn2C(C)C)CCOC)ccc(Br)cc1 c1(CC(=O)NC(C2CCN(C(C(C)OCCOC)=O)C2)(C)C)ccncc1Cl c1(C(N2CCSCC2C(N2CCC(OC(F)F)CC2)=O)=O)ccc(Br)c(Cl)c1F N1(C(C2CC(C)(CC)C2)=O)CC2CCN(C(=O)C(C)(F)F)C2C1C C#CC(CNC(=O)C(CC=CC)NC(=O)C(C)N(C)C(C)=O)CC(C)(C)C C1(C)(C(=O)NCCSCc2ccc(C)cc2)CCCN(c2cc(C#N)ncn2)C1 CC(CCCNC(=O)C(C)(F)c1ccccc1)NC(C1(O)CCCC1)=O CCC(C)CCC(O)CC(=O)N(CCN(CC)CC)CCOCC1CC1 N1(c2ccc(C(C)=O)cn2)C2CCC1CN(C(=O)CCc1cnn[nH]1)C2 c1(C(=O)NC(C)CNC(=O)CC2CCCC2C)cn2c(n1)CCC2 C(N=c1cc(NCCCn2cnnc2)nc[nH]1)c1c(C)sc(Br)n1 c1(C(N(CCNC(CC=CC(=O)OCCO)=O)C2CC2)=O)ccnc(OC(F)F)c1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)CC1CCC3(CC1)CC3)C2 C1(CC(C)OC(C)=O)CCN(C(=O)NC2CC(O)C(O)C2)CC1 CC1CC2(CC2)CN1C(c1cc(CNC(c2cncs2)=O)on1)=O c1(C(N2CC(CCNC(C(C)C3CC3)=O)OCC2)=O)cc2n(n1)CCC2 C(C)(CCC(=O)NCC(C)NC(=O)C(C)Cc1ccncc1)OCC C(C)(N=c1[nH]n(C)c(C(F)(F)F)c1[N+](=O)[O-])C1CCC(NC(C(C)N(C)C)=O)C1 C(=O)(C1=C(Cl)CCC1)NC1C(C)CN(C(C2CC(=O)N(C3CCCCC3)C2)=O)C1 N1(C(CN2CCC(OC)C2)=O)CCCCC(CNC(c2nnn(C)n2)=O)C1 Cc1c(N)cc(C(N2CCC(NC(C3CCS(=O)(=O)N3)=O)C(C)C2)=O)cc1N C1(NC(C2(CSC)CCC2)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 c1(C(N(C2CCCC(NC(c3c(C#C)c[nH]n3)=O)C2)C)=O)cccn2nccc12 Cc1sccc1C(=O)NCC(C)(C)OCC(=O)NOCCCC1CC1 c1(C(=O)NCCOCCNC(C(CSC)O)=O)cc(C2OCCO2)ccc1O C1(NC(CCCCC)=O)C2CC3CC(C2)CC1(CNC(=O)C(F)CC)C3 C1(NC(c2c(CC)cco2)=O)CN(C(c2ccc3oncc3c2)=O)C2(CCC2)C1 N1(C(C(COC)O)=O)CCC2(CCCN2C(=O)C(C)c2ccco2)CC1 N1(C(C(C2(O)CCC2)NC(c2oc(CC)c(C)c2)=O)=O)CCC2(CNC(=O)N2)C1 C1(C)(CNC(Cc2ncc(C)o2)=O)CCCN(C(c2cnc(O)s2)=O)C1 C1(OCC)CC2(C1)CC2C(=O)NCC(O)CNC(=O)Cc1cn(C)cn1 c1(SCC)ccc(C(=O)N(C)CCN(C(C2CCC(C(C)C)C2)=O)C(C)C)cn1 CC1CN(C(=O)C=Cc2ncco2)CC1NC(=O)C(c1ccc(Br)cc1)(C)C C(C(=O)NC1(CNC(=O)Nc2cccc(C)c2)COC1)(C(C)C)SC C12COCCN1C(=O)NCC2.c1(CSCC)ccc(C2CC2C)o1 N#CC1CCCCC1NC(=O)Nc1ccc(OCC(F)F)cc1 C(CNC(C1CC2CC2N1C(=O)CCC(C)N(C)C)=O)(C(C)(C)C)OC C(=O)(CCC1=NNC(=O)CC1)NC1C(CC)CN(C(C23CC(F)(C2)C3)=O)CC1 C=C=CC(C)C(=O)N1CCC(CC(=O)N(CC(C)CC)C)C1 N1(C(C2(C#C)CCCC2)=O)CC(C2CN(C(C3CCC([N+](=O)[O-])CC3)=O)C2)C1 CC(C)C(C(=O)NCC1CCN(C(=O)CCC(F)F)C1(C)C)C(C)C C(CNC(=O)CCOCC1CCC1)(CCNC(c1nonc1C)=O)OC C1(N(C)C)CN(C(C2CC(NC(=O)CCC(N)=O)C2(C)C)=O)CC1O C1(CNC(CCC=C)=O)(COC)CCCN1C(c1c(C)cnn1C)=O c1(CNC(=O)NCC2N(C(=O)OC(C)(C)C)CC2)c[nH]nc1F.c12cc([nH]n1)C2 c1(CN2CCN(C(c3cccc(=O)n3O)=O)CC2)ccc(Cl)cc1[N+](=O)[O-] C(CCCC(=O)NC(C)CCCNC(C12CCCC1(C(N)=O)C2)=O)N(C(C)=O)C C(=O)(CC(C)CCC(=O)NCC(C)CNC(C1(C)CC=CC1)=O)OC C=CC1(C(=O)NCCCCCNC(=O)Cc2cccn2C)CCC1 Cc1cc(C(=O)NCCCCNC(=O)CC2CCCC2O)ns1 C1(NC(=O)CC2C=CCC2)CC2CC(NC(c3csc4nnsc34)=O)C1C2 c1(C(N2CCC(C(=O)NCc3n(C)ncc3)C(O)C2)=O)c(F)ccc(Cl)c1Br c1(C(C)N(c2nccc(Oc3ccccc3)n2)C)cccc(N2CCNC2)c1 C(=O)(C(CCC1CC1)NC(=O)CCn1cnc(=N)[nH]1)NCCSCCCC C(=O)(CCC(CC)OC)NCCN(CCOC)C(C1CCC(N(C)C)CC1)=O N1(CCC#C)CC2CCN(C(c3csc(C(F)(F)F)n3)=O)C2C1 CC1(C)CCCCC1NC(CCC(F)(F)F)c1ccccc1 c1(CNCc2ccc(OC)cn2)ccnc2cc[nH]c12 N1(C(C(C(C)C)OC)=O)CC23CCCC2(C1)CN(C(c1cccnc1S)=O)C3 CC(C)CC(O)C(=O)N1CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C(CO)C1 C(=O)(C(C)(C(F)F)c1ccccc1)N(CC(C)NC(c1n(C(C)C)cnc1)=O)C c1(C(=O)NCc2cccnc2N2CCCCC2)cc2c(cn1)OCCC2 CC1CCN(C(c2cnccn2)=O)CCN1C(C1CC2(C1)CC(O)C2)=O c1(CN(C(=O)CN(C(=O)Cc2ccco2)C2CC2)CC=C)ccncc1Cl c1(CC(N2CCC(CCNC(COC(C)(C)C)=O)C2)=O)cccc(S(C)(=O)=O)c1 C1(C(N2CC(NC(C)=O)(CO)C2)=O)CN(C(=O)CCCCN(C)C)CC12CCC2 CC1(C(=O)NCC2(CNC(c3cc(C#N)no3)=O)CC23CCC3)CCOCC1 CC1CCN(C(=O)CC2CCC2C(F)(F)F)CC1CC(=O)N(C)CC1(O)CCC1 N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3CC(NS(C)(=O)=O)C3)=O)CC2C1 N1(C(CSCCC(C)C)=O)CCC2C(C(=O)NCC3CCC(C)(C)CO3)C2C1 C(=O)(C=C1SCC(=O)N1C)NC(C(C)C)CNC(C1CN(S(N)(=O)=O)C1)=O CC1C(NC(c2cc(Cl)ccc2Cl)=O)CC2CCC1N2C(C1(CO)COC1)=O c1(C(N2CC(C)(NC(c3ccc(C)[nH]3)=O)C2)=O)cccc2c1OCC2C CON1CCC(C(=O)NCCN(C)C(c2nocc2CC(C)C)=O)CC1 N1(C(Cc2n(C)cnc2)=O)CC(C(=O)NCc2csnn2)C(F)(F)C1 c1(C(N2CC3(N(C(c4ccc(C=C)cc4)=O)CC3)C2)=O)cc2c(cc1C)OCO2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(C2CCCOCC2)=O)CCCC1 C(=O)(C(O)CC(N)=O)NC1(C2N(C(c3c(OC)cccc3)=O)CCC2)CC1 c1(CC)cccc2ccc(C(N3CC(NC(=O)C(O)C(C)C)C3)=O)nc12 S(=O)(=O)(c1cccc(CC(=O)NCCc2nc3c(s2)COCC3)c1)NC C1(CC(=O)NCC(CNC(=O)CNc2ccc(Cl)cc2)O)CC(=O)NC(=O)C1 C1(C(NOCC2(C=C)CCC2)=O)(CC)CCCN1C(=O)OC(C)(C)C c1(C(=O)NCC2CN(C(C(c3cccc(C)c3)C)=O)C2)ccc2c(c1)C(C)CO2 n1(CC)ncnc1CSc1nc(CO)n[nH]1 CC(C)S(=O)(=O)C(C)C(=O)NCC(C)N(C(c1ncsc1Br)=O)C1CC1 N1(C(c2cc(C#N)on2)=O)CCC(NC(=O)CSCC2CCCO2)C(F)(F)CC1 c1(C(N2CC(C)C(NC(=O)CC3C=NN(C)C3=O)C2)=O)cc2c(s1)CC(C)(C)C2 C1(NCCCCn2cc(-c3ccn(C)n3)nn2)CCCCN1C1CCCC1 c1(C(N2CCC(N(C(Cc3c(C)con3)=O)C)C(C)C2)=O)ccc2cncn2c1 c1(NCc2cc(Sc3cccc(NC(=O)C4CC4)n3)ncc2)nccc2occc12 N1(C(C(C)Cn2ccnc2)=O)CC2=C(C1)CN(C(=O)CN1CCOCC1=O)C2 c1(OC)cnc(F)c(C(N2CC(C)(C)CC2CNC(=O)CC2CCCC2C)=O)c1 c1(C(=O)NCCN(CCCN(C)C)C(=O)Cc2cccnc2)onc2c1CCCC2 Cc1c(F)ccc(C(N2CCCC(N(C(=O)CC3CSCCS3)C)CC2)=O)c1N c1(C(=O)NCC2CC(CNC(c3cscn3)=O)C2)cccnn1 N1(C(C2C3(CN(C(c4ccc(CC(C)C)cc4)=O)C3)C2)=O)CCn2cccc2C1 c1(C(=O)NC(C)CCCCNC(C2CCSCC2)=O)cnc2c(F)cccc2c1 c1(C(=O)OC)nccc2c1CCCN2C(=O)C(CC(F)F)C1CCC1 c1(CC(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(O)nc1O c1(C(=O)NCCCN(C(=O)C(F)(F)C2CC2)C2CC2)cc(C(F)(F)F)ncn1 C1(C(N(CC)OC)=O)CN(C(=O)CNC=O)CC12CCC2 C1(NC(C2(CCC)CC2)=O)CCC(CNC(C2CC2Cl)=O)CC1 CC1CCCC1(C)NC(C1CCC(NC(=O)C(C)NC=O)CC1)=O C1(C(=O)NCCC2CSCCN2C(c2ccn(C3CC3)n2)=O)Cc2nccn2C1 c1(CNC(=O)NC2C(CN(CCC)CCO)C2)cc(F)cc(F)c1Br Cc1ccc(C2CC2C(=O)NCCCN(C)C(C2CCO2)=O)cc1C N1(CCn2cc(C(N(C)C)=O)nn2)CCCN(CC(C2CCCO2)=O)CC1 c1(C(=O)NC2(CCCNC(C3CCCO3)=O)CC2)cc(F)cs1 c1(C(=O)NC2CC(CNC(C(CSC)O)=O)CC2O)cncc2c1CCC2 C=CCC(C(=O)N1CCC(C)C1CNC(c1cc(COC)nc(O)c1)=O)C(C)C c1(N(C)C)ccc(N(C2CC3CC2CN3)C(=O)CCN2CCOCC2)cc1C#N CC#CCCCCNC(=O)C(C)N(C(c1cc(CCC)on1)=O)C1CC1 N1(C(c2cccc(F)c2)CCCC)CCCC(C(=O)OCC)C1CC C1(NC(C2C(CC)CN(C(=O)CC=C(C)C)C2)=O)CCOC12CCCC2 C1(CCC)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCN1C(C1CC12CC2)=O C12(NC(CSCC#C)=O)CCCN(C(=O)CN3CCCCCC3=O)CC1C2 c1(CNC(c2cc(C)on2)=O)cc(C(=O)NC2CCCC2CF)ccn1 Cc1ccccc1S(=O)(=O)CC(=O)NC(C1CCSCC1)=O.C12(CF)CCN1C2 Cc1cc(C(=O)NCc2ccccc2C)cc(C)c1.C12(CCC(C)(C)C1)C(=O)N2 c1(CC(=O)NCCC2N(C(CC(C)(C)OC)=O)CC(OC)C2)ccc(F)c(F)c1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CC(NC(=O)Cc2csc(C(C)C)n2)C2CC12 c1(CNC(CC(CCC)CC)=O)nn(C)c2c1CN(C(c1csc(C)n1)=O)CC2 C1(NC(Cc2ccc(OC)c(F)c2)=O)CN(C(C2CC23CC3)=O)C2(CCCC2)C1 c1(C(=O)NCC2N(C(C(CCC)CC)=O)CC=C2)ccc(F)c2c1OCC2 C1(CC)(CC)CC(NC(c2cc(N)cnc2C)=O)CN1C(c1nnn(C)c1C)=O N1(C(CC2(C)CCN2C(c2ncccc2F)=O)=O)CCC(F)(F)C(O)C1 C(=O)(C1=CCc2ccccc21)NCCCCCN(C)C(c1cncnc1)=O c1(C(N(C(C)CN(C)C(C2CCCN2C=O)=O)C)=O)cc(F)ccc1O c1(OC)cccc(C(=O)N(CC(N2CC(CO)C2(C)C)=O)CC(C)C)c1 N1(C(C2CCN(C(CC(C)F)=O)C2(C)C)=O)Cc2cccc(F)c2C1 C1(C(N(CC(C)N(C)C(c2cncc(CO)c2)=O)C)=O)COc2ccccc2C1 C(C(C)C(=O)NCC12CC(NC(=O)C(C)N(CC(F)(F)F)C)(C1)C2)OCC c1(C(=O)NCC(=C)CCNC(C2CC2(C)CC)=O)cn(C)c(=O)c2c1CCCC2 c1(C(=O)NC2(CF)CCN(C(C3(C#N)CC34CCC4)=O)C2)cccc2c1CCO2 CC(C)C(CC(=O)NC1(CCO)CCC1)NC(C1CC(F)C(=O)N1)=O C(=O)(CC(CC)OC)NCC(C)(C1CC1)NC(c1cnc(CCCC)s1)=O N1(C(COCC(C)C)=O)CC(F)CC1CNC(c1csc(-c2cnc[nH]2)n1)=O c1(OC(c2ccc(NC(=O)OC(C)(C)C)o2)=O)cnn(S(C)(=O)=O)c1 C(=O)(C1CCCc2sc(=N)[nH]c21)N1CCNCC1.C(=O)(C(O)CC(N)=O)N(C)C S(=O)(=O)(c1ccc2c(c1)CC(C(=O)O)C2)N1CCC2(CNC(=O)OC2)C1 C1(C(=O)NCCOCCC)C2CN(C(C)CC3COCCO3)CC12 N1(C(c2cnc3n2CCC3)C(=O)NC2(C)CC2)CCSC2COCCC12 C(C)(C)(CCCCNC(=O)CN1CCCCC1)NC(C1C(C=C)OCC1)=O Cc1cc(CN2CCC(F)(CNS(=O)(=O)c3cccs3)CC2)c(O)c(Br)c1 C1(C(=O)OCC)CCCC(C(=O)NC2(CCNC(C3CC4(CCC4)C3)=O)CC2)C1 c1(C(=O)NC(C(=O)OCC=C)Cc2ccccc2)ccc(CC(F)(F)F)cc1F N1(C(c2cc(OCC)ns2)=O)CCN(C(=O)C(C)OC)C(c2cn[nH]c2)C1 C1(C(N2CC3(CC(NC(COCC(=O)OC)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 c1(SC)cccnc1NC(c1ccc(Nc2cc(C(F)(F)F)ncn2)nc1)=O C1(CC(N2CC(F)(CO)C2)=O)C2CCCC2N1C(=O)CSc1nc[nH]n1 Cc1cc(C(N2CCC2CNC(=O)CC(O)C(C)(C)C)=O)c(F)cc1F N1(CC(=O)NCC(CNC(C2(C(F)F)CCCC2)=O)CO)CC(=O)NC1=O C1(C(=O)NC(Cc2ncn(C(C)C)c2)C(=O)O)CCS(=O)(=O)CN1 N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2c1cn(CC2(OC)CC=CC2)nn1 N1(C(C=CCN(C(=O)CCC2(C)CC2)C)=O)CC2(CC2)C1 C1(O)(CN(C)C(C2CC(O)CN2C)=O)CCCN(C(=O)CNC=O)C1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC2(NC(=O)Cn3cnnn3)CC2C1 Cc1cc(CNC(C2CC2C(C)NC(=O)CCOCC(F)F)=O)cc(F)c1 C(C(CC1CC1)CO)NC(CN(C(=O)Cc1ccnn1C)CC)=O C(N=c1[nH]c(=NCCN(C)C(C)C)[nH]c2c1SCC2)C1CCCC(CC)C1 CCCCC(CC)CC(=O)NC(C1(NC(=O)CC2(C)CC2)CC1)C S(=O)(=O)(c1cccc(NC(=O)CN2CCC(C3CC3)C2)c1)NCC c1(C(N(CCNC(c2cc(C)c[nH]2)=O)CC)=O)cc2ccccc2cc1C C12(NC(CCC=CC)=O)CCOCC1CN(C(C1(C#N)CCN(C)CC1)=O)C2 CC(CCC(=O)NCC1(C)CCC(=O)N1)NC(=O)CCCOC(C)(C)C N1(C(C2CN(CC)C(=O)C2)=O)CCCC2C1CCN2C(c1ccncc1)=O c1(C(N2C(CNC(c3c(O)ncc(CC)c3)=O)CC2)=O)cccc2c1CC(=O)N2 Cc1cccc2c1CC(C(=O)NC1COCC1NC(c1cc(C(C)C)[nH]n1)=O)O2 N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(-n4cccn4)c3)=O)CC1C2 O=C(CCCCCCCCCCNC(C1CC1COCC1CC1)=O)NCC1CC1 C(CC(C(F)(F)F)N1CCOCC1)NC(=O)C(=O)Nc1cccc(C2CC2(F)F)c1 c1(CC)nn[nH]c1C(=O)NCC(CCOC)NC(c1cnnn1C(C)C)=O c1(C(N2C(C(=O)NCCC(=O)OC)CSC2)=O)c(C)ccnc1C N1(C(CCC#C)=O)C2CCC1C(CNC(c1cncc(OC(F)F)c1)=O)C2 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CC(NC(CN(S(C)(=O)=O)C)=O)C1 CCCC(O)C(CO)NC(=O)CCC1CCCN(C(=O)Cc2ncccc2F)C1 Cc1nc(N2CCCC(CNC(=O)Cc3ccc(O)nc3)C2)c2c(C)csc2n1 N1(C(C(C2CC(NC(=O)COC3CCC3)C2)F)=O)CCCC2(CC2)C1 CC1(C)CC(NCc2cncn2-c2ccc(F)cc2)CS1 N1(C(C2CC(CC(=O)OC)C2)=O)CC(C)(NC(=O)C=CC2CCOC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NCC(CCNC(C=C(COC)C)=O)(C)C C1(NC(C2(OC)CC2)=O)CC2CC(NC(=O)Cc3ccnc(Cl)c3F)CC12 C1(OCC(=O)NCCC2CC(NC(c3nn[nH]c3Cl)=O)C2)CCOCC1 c1(CC(=O)N(C(C)C(=O)NCC(c2ccco2)O)CC)cc(C)on1 N1(C(C(C)NC(=O)C2CC2)=O)C2CCC1CC(N(C)C(c1ccns1)=O)C2 Cc1cc(S(C)(=O)=O)cc(C(=O)NCC2CC2CNC(c2nocc2Cl)=O)c1C c1(C(C(=O)NCCC(=C)CNC(C2(n3cncn3)CC2)=O)(C)O)cccc(F)c1 N1(C(C2(CC)COC2)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(NC(COc2ccc(C)cc2C)=O)CC1 C1(C(N2C(c3nc(C)on3)CCC2)=O)CCCN(C(c2cnc[nH]c2=N)=O)CC1 c1(C(N2CC(C)(NC(c3onc(CC)n3)=O)C2)=O)cc(C#N)c[nH]1 C1(CNC(CCC2(C)CC2)=O)CN(C(=O)C(C)C(C)(F)F)CCC12CCOCC2 C(CO)(CCCCNC(C1CCC(O)CC1)=O)NC(c1coc(Br)c1)=O c1(CC(=O)NC(CCN(C(C=C(C)C)=O)C)C)cn(C)c2ccccc12 C1(C(N2CCC(CNC(C(N3CCC(O)CC3)C)=O)C2)=O)CCC2(CCC2)CC1 C1(CC)CN(C(C23CCC(CO2)C3)=O)CCN1C(c1ccc(CCO)cc1)=O c1(C(N2CC3N(c4nc(SC)cc(CC)n4)C3C2)=O)ccc([N+](=O)[O-])cc1C C1(C(=O)OC)CN(C(=O)NCc2cccc(C(=O)N(C)C)c2)CCS(=O)(=O)C1 N1(C(c2n(C=C)nnc2)=O)CCOCC1(C)C CC1=C(C)CN(C(C2(CNC(C34CCCC3C4)=O)CC2)=O)CC1 c1(C(N2CC(NC(C34CC(C3)S(=O)(=O)C4)=O)C(F)C2)=O)ccc(Cl)c(Cl)c1 CC(C)(C)C#CCCNC(C1CC(O)CN1C(=O)Cc1cnns1)=O C1(NC(c2cnn(C)n2)=O)CCC(F)(CNC(C2CCCN2S(C)(=O)=O)=O)C1 c1(C(=O)NCC=CC)cc2c(cnn2C)nc1C Cc1cnc(N2CC(=C(F)CNC(=O)CCC3CCCO3)C2)nc1 c1(CNC(=O)NC2CCN(CC(=O)OCC)CC2)cnc(C#N)c(Cl)c1 n1(CCC)ncc(C(=O)NCC2CCCC(NC(C3(SC)CC3)=O)C2)c1Cl c1(C(=O)NC2CC(NC(C(CCCC)CC)=O)C2)ccnc2c(C(N)=O)cnn12 c1(CN2CCC(N(C(c3cc(C)nn3C(F)F)=O)C)C2)ccc(F)c(C#N)c1 c1(C(N2CC(O)(CN(C(CCCNC(=O)OC)=O)C)C2)=O)nnccc1C c1(C(=O)NC(C(C)C)C(=O)NC2CC=CC2)ccc(=O)n(C)c1 c1(CCC(=O)NCC2(F)CC(NC(CC3(OC)CCC3)=O)C2)ccc(SC)cc1 C(=O)(CC(=O)NCC(C)(C)OCC(=O)NCCCC1CCOC1)N(C)C N1(C(c2ccn(CC)n2)=O)CCC2(CNC(=O)CNC(=O)C3CC3)CCCCC12 c1(C(CNC(=O)C(F)(F)Oc2ccccc2)NC(CSCC)=O)ccnc(Cl)c1 c1(C(N2CCC3C(C(N4C(C#C)CC4)=O)C3C2)=O)ccc2cc[nH]c2c1 C1(C(=O)NCCC2(NC(C3CC(CC(=O)OC)C3)=O)CC2)CCCOCC1 N1(C(C2(NC(=O)OC(C)(C)C)CCSCC2)=O)CCC(C(C)(C)C)n2nccc21 N1(C(C)=O)CC2(CCC2)CCC1CNC(c1csnn1)=O CCC(C)CC(C(=O)NCC12CCC(CC1O)C2)NC(=O)CC1CC(N(C)C)C1 CCCC(C(=O)NCCN(C1CCCCC1)C1CC1)N(C)C(C1C(C)(C)C1(F)F)=O CCCCC(CNC(C1(C(C)C)CCCO1)=O)NC(=O)C(COC)COC C(CCCCC(=O)NC1CCCN(C(=O)COCCCF)C1)OC C(CCCCCC1CC1)NC(CC1(NC(C2N(CCC)CCC2)=O)CCC1)=O CC(C(C)(O)C(=O)N1CCC(NC(=O)C(C)(C)C2CCCC2)C1)c1ccccc1 c1(C2(C(=O)OCC(c3cccc(Br)c3F)C)CCC2)cc(Cl)ccc1F N1(C(CC(=O)NCC#C)=O)CC2CCCC(NC(=O)C(C#N)C(C)C)C2C1 N1(C(CC2(C)CCN(C(C(C=CC)O)=O)C2)=O)CCc2nc[nH]c2C1 N1(C(C2(NC(c3cnc(C)nc3C)=O)CCSC2)=O)C2CCC1CC(F)C2 C(=O)(C(C(C)NC(c1cc2cccnc2[nH]1)=O)C(C)C)NCC(CSC)OC c1(C(N2CCCC(N3CCCCC3)C2)C(=O)NCCC)ccc2c(c1)CCCO2 Cc1ccc(CC(N2CC(CNC(c3cscc3F)=O)C3(CC3)C2)=O)cc1F O=C(C1=CCCCC1)NC1(C(N2CCC(C3CCCO3)C2)=O)CC1 c1(C(=O)NCC(C)CNC(C2CSCCS2)=O)cc(CC2CCC2)c[nH]1 CC(=O)C(C)(C)CC(=O)NC(C1(O)CCCCC1)C(=O)Nc1ccc(C)c(CO)c1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CCC(C1)N2C(C1CCO1)=O c1(N(C(CCNC(CCNC(=O)OCC)=O)=O)C)cc(OC)n(C)n1 CC1CN(C(c2cc(CNC(=O)CCCC3CCCO3)on2)=O)CCN(C)C1 C(=O)(C(COC)COC)NCCC1(C(N(CC#C)CCF)=O)CCCC1 C1(OC)CCCC(CNC(=O)CN2CCN(C(=O)CC(C)O)CC2)C1 c1(OC)ccc(C(=O)NC2CCN(C(=O)CN3CCCCC3C)C23CC3)c(Cl)c1 c1(C(=O)NCC(CNC(CC(C=C)C)=O)F)ccc(OC)c2occc12 c1(C(=O)OC)ncccc1CCC(=O)NCC1CN(C(C2CC3CCC2C3)=O)C1 c1(C(N(CCCNC(C2(C)CCOC(C)C2)=O)CC)=O)ccc2cnc(C)n2c1 C1(C(=O)N(CCC(C)NC(=O)Cc2cncs2)C)(OC)CCC(C)(C)CC1 C(CCCC(C)NC(C1(c2cccc(F)c2)CC1)=O)NC(C(C)SCCCC)=O C1(CC(=O)NCCOC2CN(C(C(COC)C)=O)C2)Cc2ccccc2O1 C1(NC(COCC(=O)NC)=O)CC2(C1)CN(C(c1[nH]c(C3CC3)nc1C)=O)C2 O=C1NC(c2ccc(CNCC3CC3)o2)CO1.C12CCC(N1)COC2=O C1(C(=O)NC(C(C2CC2)OC)C)CN(C(=O)C(SC)SC)CCO1 c1(OC)ccc(C(=O)NCCC(C)N(c2snc(C)c2C#N)C)c(Cl)n1 N1(C(C(CC)(C)COC)=O)CC(NC(=O)C=Cc2cccs2)C2(CCC2)C1 c1(C(N2CC3C(NC(CCC=CCC=C)=O)(C3)C2)=O)cccc2[nH]cc(Cl)c12 S(=O)(=O)(c1cccc(C#N)c1)NC(c1c(Cl)cc(F)cc1Br)=O.CC12CN(C1)C2 N1(C(C(c2cc(F)cc(F)c2)C)=O)CCC(F)C(NC(C2(NC(N)=O)CC2)=O)C1 N1(C(CSC(C)C)=O)CCN(C(c2ccc(O)nn2)=O)CC1 c1(OCC(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc(C)c(Cl)c(C)c1 c1(C(N2CC(F)(CNC(CCCCOC)=O)C2)=O)nn(C)c2ccccc12 c1(CCC)onc(C)c1C(=O)NC(C1CCCC1)CNC(c1sc(=N)[nH]c1C)=O N1(C(c2ccc(C#C)nc2)=O)CCC2(CCC2)C(NC(=O)CCNS(C)(=O)=O)C1 C(C(=O)O)(C1CC1)(C1CC1)NC(C(n1cc(C2CC(F)(F)C2)nn1)C)=O Cc1nsc(C(=O)NC2CCC(NC(=O)C=Cc3ccc(C(N)=O)o3)C2)c1N c1(C(N2CC(C)N(C(=O)C=Cc3ncco3)CC2)=O)cncc2[nH]ccc12 C(=O)(C(F)(F)C(O)C(C)C)NCCCCCCN(C(C(n1ccc(C)n1)C)=O)C C1(OC)CC(NC(c2ccnnc2O)=O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 Cc1cn2nc(C(N3CC(NC(=O)CCC4(C)CC4)C4(CC4)C3)=O)cc2c(=O)[nH]1 c1(C(=O)NCC(C)(C)NC(C(C)P(C)(C)=O)=O)cccc2c1COCC2 C1(NC(c2cc(COC)sc2)=O)CCCN(C(c2cccn2C(C)C)=O)CCC1 N1(C(c2c(C)cn(C)n2)=O)CC2CC(NC(=O)Cc3cccc(C)c3Cl)C2C1 N1(CC)CCOCC1CC(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC1CC1CC1 N1(C(C2C(C(=O)OC)C2)=O)CCOCC1CNC(c1cc(C)ns1)=O N1(C(C(c2cn(CC)nc2)=O)=O)CC(C)(C)C1CNC(=O)CC1CC12CC2 C1(NC(C(C)NC(N)=O)=O)CN(C(c2csc3cccnc23)=O)C2(CCCC2)C1 N1(C(Cc2c(C)occ2)=O)CCCC(NC(c2cc(C(F)(F)F)ccn2)=O)C1C C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2nccc(C)c2O)=O)CC1)C c1(C(=O)OC)cccc(C(N2CCCC2CCNC(C23CCCCC2C3)=O)=O)n1 CC(N=[N+]=[N-])C(=O)N(CC(=O)NOCCCO)C1CC(C#N)C1 c1(C(=O)OC)c(C)cc(C)nc1N(C1CCN(C(=O)C(C)(F)F)CC12CC2)C C(=O)(C1=NNC(=O)C1)NCC(C)N(C)C(C1CCOC1)=O n1(COCC)nnc(C(=O)Oc2ccc(SCC(F)(F)F)cc2)c1N N1(C(C(COCC)N=[N+]=[N-])=O)CC2(CCC2)CC1C(=O)NCC1CCC(=O)O1 N1(C(=O)OCC)CCC(Nc2cnc(C(F)(F)F)cc2C)C(C)C1 c1(C(N(CC(CNC(C(COC)C)=O)O)C)=O)noc2c1CCc1sccc1-2 c1(C(c2nnnn2C)NC(c2cc(Cl)cc(Cl)c2F)C)ccccc1[N+](=O)[O-] N1(C(c2c(CC)nn[nH]2)=O)C2COCC1CC(NC(c1cc(C)[nH]n1)=O)C2 N1(C(C2(CCCC)CCC2)=O)CCC(NC(=O)CCC2CCCN2C)C(C)C1 N1(C(C(C2CCC2)OC)=O)CC(CNC(c2cc(C)cs2)=O)C(F)(CO)C1 c1(C(c2nnnn2Cc2ccco2)NCCNC(C)=O)c(F)cc(F)c(Br)c1F C1(C(=O)NCC2(NC(c3ccc(C)cc3F)=O)CC(OC)C2)CC2(C1)CC(C)C2 Cc1ccc(C=CC(=O)NC(C)(CNC(C2CC2C(C)C)=O)CO)cc1 C=C(C)C(C)(C)C(=O)NC1CCOCC1NC(C1SCC=C1C)=O C1(C(=O)NC2CC(C(=O)NCC(C)C(F)F)C2)CC(=O)C12CCC2 c1(C(=O)NCC2N(C(c3ccc(C(C)(C)C)[nH]3)=O)CCC2)cc2[nH]ccc2s1 N1(C2CCCN(C)C2)CCN(C(=NCCF)NCC2CCC(=O)NC2)CC1 c1(OC)ccc(F)c(C(N2CCC(NC(c3sccc3OC)=O)C(F)C2)=O)c1 CCS(=O)CC(=O)NC1C=CCN(C(=O)CNC(=O)NCC2CCCC2)C1 C1(NC(C=CC(CC)C)=O)CCN(C(c2cccc(Cl)c2N)=O)C1(C)C N1(C(CC(=C=C)C)=O)CCN(C)CC1CNC(=O)C(C)OCc1ccc(C)cc1 C1(CC)(NC(c2cc(C)nc(O)c2)=O)CCCN(C(C2CCCOCC2)=O)C1 N(C1c2ccccc2CCC1OC)Cc1ccc(C(=O)Oc2c(N)cccc2)o1 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(c3ccc(N(C)C)cn3)=O)C2)C1 c1(C(N2CCN(C(C(C(CC)O)C)=O)C(C)C2)=O)cccc2nc[nH]c12 N1(C(CNC(C)=O)=O)CCC(C2CCCN(C(C)C(=O)NC(C)C)C2)CC1 Cc1ccc(C(C)C(=O)N(C(C)CCNC(=O)C=C2CCOCC2)C)s1 N1(C(C2(C(C)C)COC2)=O)CC2CCCC2(C(=O)NC2CNC(=O)C2)C1 C12(C(=O)OC)CCCN1C2=O.C1(NCc2nnc(CO)s2)(NC(C)=O)CCCC1 C1(NC(=O)CCc2ccncc2Br)CCN(C(=O)C=Cc2cnc[nH]2)CC1O CCCCC(C(=O)NCC1CCN(CC)C1)NC(=O)CC(CC)C1CCC1 C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)C)NC(=O)CNC=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NCC1(O)CC(CNC(C(CC)N(C)C)=O)C1 c1(SC)cn(C)nc1CNC(=O)CC(CC1CC1)NC(=O)C(N)=O c1(OC)ccc(CNCC2CCC(C(=O)NCc3ccc(Br)cc3Cl)CC2)cc1Br c1(NC(C(C2CC(NC(CC(C)O)=O)C2)F)=O)cccc2c1OCC2 CC1(C)CN(C(=O)C=C2CCCC2)CC(CNC(=O)CN2CCS(=O)CC2)O1 c1(OCCC(=O)NC(CN(CCCO)CC)C)ccncc1 CCC(CC(=O)NCC1(CF)CCC1)NC(c1cn(C)nc1C)=O N1(C(C(=O)NC(c2c(O)cc(C)c(Cl)c2)C)=O)CCc2ccc(C#N)cc2C1 c1(NC(C2CN(Cc3cc(Cl)cnc3Br)CCO2)=O)ncc(F)cc1Br C1(NC(C=C(C)C(C)C)=O)CCC(C)(CNC(c2ccc(F)cc2)=O)C1 CCC(C)(C)CC(=O)NCC=CCNC(c1cc(C(F)(F)F)cs1)=O CC1CN(C(C2(C)CC(C#N)C2)=O)CCC1C(=O)NC1CC2CCCC2C1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(c3cccc4nccn34)=O)C2C1 C1(CC(N2CC(COC)(CNC(c3cc(C(C)C)no3)=O)C2)=O)CCOC1(C)C C1(C(=O)OC)(OC)CCCN(C(=O)C(c2cccc(Cl)c2F)NC(C)=O)C1 N1(C(CC2(C#N)CCCCC2)=O)CCC2(CCC(NC(c3cn[nH]c3)=O)CC2)CC1 c1(NC(C2OCCN(C(c3n(CC)ccc3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(CC)C(F)(F)F)=O)CCN(C(c2cc3n(n2)CCCO3)=O)C2(CCC2)C1 C=CC(C)(CC)C(=O)NCC12CC(C1)C(NC(=O)CC1(O)CCCC1)CO2 C1(N(C(CCC2N(C)CCC2)=O)C)CN(C(=O)CS(C)(=O)=O)CCC1O C1(NC(c2n(CC(C)C)ncc2)=O)CC(C)CN(C(c2cncn2C2CC2)=O)C1 c1(C(N2CCOCC(CNC(c3nc(C)oc3)=O)C2)=O)cc([N+](=O)[O-])nn1C CC1CN(C(=O)COCC2CCCO2)CCC1CNC(c1ccnc(Cl)c1)=O C1(CNC(c2c(C(C)C)n(C)nc2)=O)(NC(=O)Cn2cnnc2)CCCCC1C Nc1cnc(Br)c(C(=O)NCCNC(C2CCCS(=O)(=O)N2)=O)c1 CC1C(NC(=O)COc2cccc(F)n2)CCCN1C(=O)CCCC1CC1 c1(CC(=O)NCCC2CC(OC)CN2C(=O)CC=C(C)C)csc2sc(C)cc12 C1(CC(=O)NC(C(CO)NC(C2(CCC)CC(=O)C2)=O)C)CC(C)(C)CO1 n1(CC(N2CCC(C(C)(C)NC(C3(F)CC=CC3)=O)C2)=O)ncc2ccccc12 C12(C(=O)NC(C(CCC)C)C)CCC(CC1)N(C(c1cc(C)n(C)c1)=O)C2 C(=O)(CC(C)n1cccc1)N(CCNC(CN(CCC)C)=O)C C1(C(=O)NCCC(C)N(C)C(C2COCCN2C)=O)CC2C=CC1C2 c1(-c2occc2)cccc(-c2cnc(N3CCC(CN4CCCC4)C3)nc2)c1 c1(-c2c(C(=O)Nc3c(C)ncc(C#N)c3)ncnc2)cccc([N+](=O)[O-])c1O Cc1ccc(C2(C(=O)NCCCC(C)NC(c3nc(C)oc3C)=O)CC2)cn1 O=S(=O)(c1cccc(=NC2CCSCC2)[nH]1)NCc1ccc(Br)cc1F c1(C(CC)(C)C)ccc(C(=O)NC2(CO)CN(C(=O)C(C)c3cccs3)C2)cc1 c1(CCCC)nc(C)c(CC(=O)NC2CN(C(C3CC(C)(O)C3)=O)CC2O)s1 C(=O)(CCCC(F)(F)CO)NC(CCNC(C1CCN(C(CCC)=O)C1)=O)C C(=O)(C(O)C(F)(F)F)NC(C(=O)NCC1(C)CCOCC1)CCC1CCC1 c1(OC)c(NC(=O)C=C2CCN(Cc3c(F)cc(O)cc3F)CC2)cc(Cl)cc1Cl Cc1nc2n(n1)CC(CNC(N1CC(c3ccc(F)cc3)OC(C)C1)=O)CC2 c1(N2CCC(c3c(OC)ccc(F)c3)C2)c(Br)cnc2ccc([N+](=O)[O-])cc12 Cc1nc(O)[nH]c1C(=O)NC1(CNC(C2CCCC2n2cccc2)=O)CCOC1 c1(CC)c[nH]nc1C(=O)NC1CC(OCC(=O)NC2CCC(CO)C2)C1 CC1CCC(CNC(=O)CCc2cscn2)N(C(=O)C(C2CC2)C2CC2)C1 C(C(C)(C)C(F)(F)F)N(C(c1ccn(C(C)C)n1)C(=O)NCC)CC S(=O)(=O)(c1ccc(N(CC(F)Cl)C)c(Cl)c1)NCCC(=O)NC C12(CNC(N3CCC(C(C(N)=O)F)CC3)=O)CC(C#N)(CO1)C2 C1(NC(COC)=O)CCCC(C(=O)Nc2ccc(CCF)cc2)CC1.C1CO1 c1(C(N(CC(C)CNC(C2(CF)CCOCC2)=O)C)=O)cccc(F)c1F Cn1cc(C(=O)NC2CCCCC2NC(c2cncn2C(F)(F)F)=O)c(O)n1 C1(NC(CC(c2ccc(C)cc2)(C)C)=O)CCN(C(=O)C(C)(O)C2CC2)CC1F C1(CCNC(=O)CSc2n[nH]c(O)n2)CCCCN1C(=O)CC(F)(F)F N1(C(=O)NC2CC(CC)C2)CCC(C)(CSC)CC1 N1(C(C2N(C(C(n3c(C)ncc3)C)=O)CCC2C)=O)C2CCC1COC2 C1(CC)(NC(c2nnn3c2CCC3)=O)CCCN(C(=O)CCOC2CC2)C1 N1(c2c(C#N)c(O)cs2)CCCC2(CNC(=O)CSc3nncs3)CCCC12 N1(C(CCN(C)CCO)=O)CCCC(F)(C(=O)NCC2CCC(O)CC2)C1 c1(OCCC)ccccc1C(=O)NC(CC)C(C)NC(c1ccc(CO)cc1)=O C1(C(=O)NCC2C(C)CC2)CNC(=O)CN1C(c1ccncc1N)=O c1(C(=O)NC(c2cccs2)C)c[nH]c2ccc(-c3scc4c3OCCO4)cc12 N1(C(C(C)C#N)=O)CC(CNC(=O)C=Cc2cc[nH]n2)CC(C)(C)C1 CC(C)C(O)CONC(C1C(C)CN1C(=O)C(C)N1CCCC1)=O C12(C(=O)NCc3[nH]nc(N(C)C)n3)CC1CCN2C(C1CC(O)C(F)C1)=O CS(=O)c1ccccc1CC(N1CCC2(NC(c3ccncc3)=O)CCCC12)=O c1(CC)ccccc1CC(N1CCC(C(C)NC(c2ccc(CC)nc2)=O)C1)=O C1(C(=O)OCC)COCCC1NC(=O)Nc1cc(Cl)ccn1 C1(NC(c2c(C)ccs2)=O)CN(C(=O)C=CC(C)C)C2(CCOC2)C1 CCC(C(=O)NCCCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)NC(C)=O CCC(C)C(O)C(=O)NCC1CN(C(=O)CCCn2ccccc2=O)C(C)(C)C1 c1(CN2CC(C(=O)Nc3c(OC)cc(O)cc3)OCC2)n[nH]c2ccc(Cl)cc12 C1(O)(CNC(=O)CC2(O)CCC2)CCN(C(c2cnnc(Cl)c2)=O)C1 N1(C(c2ccc(Cl)s2)=O)CCC2CN(c3cc4ncnn4cn3)CCC12 C(N=c1[nH]cnc(Cl)c1F)C1CCC(NC(c2c(C)nc(CC)o2)=O)CC1 C=C(Cl)C(C)(C)C(=O)NCC1CN(C)CCN1C(c1nnn(CC)c1CCC)=O c1(CC(=O)NCC(C)N(C(=O)COC2CCCC2)CC)cc(F)cc(F)c1 C1(C(N(C(C)CNC(=O)Cn2ccnn2)CC)=O)Cc2cc(F)ccc2C(=O)O1 C#CC1(O)CC(C(=O)NC2CCN(C(=O)C(C=C)c3ccccc3)C2C)C1 c1(C(C(=O)NCCOCCCN(C(C2C(C=C)C2)=O)C)CC)c(C)noc1C c1(C(=O)NC2(C)CCN(c3snc(CC)n3)C2)cccc2c1OCCCO2 C1(CC)CC(CC(=O)NCCC(C)(C)CNC(=O)Cc2ccsc2)CCO1 C1(NC(COCC#C)=O)CCC2CCN(C(C3CCCCN3CC)=O)C12 N1(Cc2c(F)ccc(C)c2Cl)CC(C)Cc2cccc(O)c21 CCCCC(CNC(C1(C)CCCOC1)=O)NC(=O)C(C)CCc1ccccc1 c1(OC)cccc(NCC(=O)N(C)CC2CCCCC2)c1Cl c1(C(=O)OC)cc2cc(NC(=O)NCCOCc3cccs3)cnc2[nH]1 CC1CCC(C(N2CC(F)(CNC(C34CC(F)(C3)C4)=O)C2)=O)C1 c1(C(N2CCC(NC(c3nc(C)[nH]c3C(F)(F)F)=O)C2C)=O)cnc(O)cc1C C=Cn1ncc(C(N2CCC(CC(=O)NC3CON(CC)C3=O)C2)=O)c1N C1(CCNC(COC(C)(C)C)=O)CN(C(C2(C)CC=CCC2)=O)CCS1(=O)=O N12CCC(CC1)OCC(=O)N1CCCC1C2=O.C1(N(C(C)=O)C2CC2)CCOC1 c1(CNC(=NCC(C)C)NCC2(CC(N)=O)CC2)ccc2c(c1)C(=O)NCC2 c1(C(=O)NC2CC(C)(NC(C(CC)c3ccccc3)=O)C2)nnn(C(C)C)c1C c1(C(N2CC(CC3C(=O)NC(=O)N3)C2)=O)ccc2c(n1)CCCC2 N1(C(=O)CO)CCCC1CC1CC(Cn2cc(CCCO)nn2)C1 N12CCCC1C1CCCN1C(=O)C2=O.c1(CC)ccc(I)c(I)c1 CC1CCN(C(=O)CCc2nncn2C)C(C(=O)NCC2(F)CCOC2)C1 Cc1cc(CN2CC3C(C(=O)NCCCN4CCOCC4)C3C2)c2cc[nH]c2c1 c1(C(=O)NC(C(=O)NC2C(C)CCC2C)Cc2ccoc2)cn(C)ccc1=O C(C(C(=O)NCC#CC1CC1)NC(c1cc[nH]c1)=O)OCC c1(OC)ccc(-c2cnccc2C(=O)NCCCS(=O)(=O)N(C)C)cc1F C1(C(C)C(N2CC=CCC2)=O)CCCN(C(=O)CC2COCC2(C)C)C1 C(=O)(CCCCC#N)N1CCC(C2N(C(Cc3cnc(C)s3)=O)CCCC2)C1 N#Cc1cscc1C(=O)NC1(CNC(=O)CCOc2ccccc2Cl)CC1 C(=O)(C#CC1(C)COC1)NCCC(C(C)(C)C)N(C(=O)CCc1nncs1)C C1(C(=O)NCCC23CC(CO2)C3)CCCCCCN1C(=O)Cc1cn[nH]c1 CC(CN(C)C)C(=O)NC1CC(C)(NC(=O)CC(=O)N(C)C)C1 CCC(CC(=O)N1CCCC1C(=O)NCc1cc(OC)ncn1)C1CCC1 CC1(C(=O)NCC2CC2CNC(=O)C2=NNC(=O)C2)CCS(=O)(=O)CC1 c1(C(C(=O)NC(C)CCNC(=O)CN2CCCCC2)C)ccc(F)cc1 CCCCC(C)C(=O)N(CC(=O)Nc1cncc(F)c1)C(C)C c1(C(N(CCN(C(CCC(=C)Cl)=O)C(C)C)C)=O)nsc2ccc(C)cc12 C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CCNCC2)CO1 Cc1cc(CNC(=O)CCN(CCCO)C(=O)CC2COCC(C)O2)oc1C C1(C(N2CCCC(CC=C)C2)=O)CCC2CCC1N2C(c1cn2c(n1)CCC2)=O Cc1oc(C)c(C(=O)NCC(C2CC2)NC(C2CCCN2C(=O)C2CC2)=O)c1C N1(C(C(C)OCC=C)=O)CC(NC(=O)C(C)(C)c2ccns2)CC2(CC2)C1 c1(C(=O)NC2(c3ccno3)CCOCC2)ccc(Oc2ccccc2)c(Cl)c1 C1(CNC(C(CC)(C)O)=O)(CO)CCCN(C(c2ccc(C)cn2)=O)C1 C12(CCCC1)C(=O)N2.C1(C(=O)OC)CC(C(=O)NCCc2ccsc2)C1 Cc1cc(N2CC(C)OC(C)C2)ncc1S(=O)(=O)N(C)C(c1cccnc1)C C1(NC(Cc2cc(C(C)C)no2)=O)CN(C(=O)CN2CCNC2=O)CC1O CC(C)(CCNC(C1CCC(=O)C1)=O)C(=O)NCC(C)(O)C1(C)CC1 c1(C(=O)NC2CC3CC(NC(=O)CC4CC=CCC4)C2C3)cc2sccc2cn1 CC1CCCN(C(c2ncc(F)cn2)=O)C1CCNC(c1cc(O)nn1C)=O C1(C(N2CCCC(C)C2)=O)CN(C(c2ccnc(CO)c2)=O)CC(C)(C)C1 CC1CN(C(=O)Cn2cccn2)CC(C)N(C(=O)CCn2ccnc2C(C)C)C1 CCC(C)CCCCC(=O)NC(C)CN(C(c1ccc(P(C)(C)=O)cn1)=O)CC Cc1nn(CC(=O)NCC2CC(NC(C3CS(=O)(=O)C3)=O)C23CCC3)c(C)c1C N1(C(C)=O)CC(N(C(c2cnc(O)cc2C)=O)Cc2ccccn2)CC(O)C1 Cn1c(CN2CC3CCCC(C2)N3Cc2ccccc2)nc2cc(Cl)ccc12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 C1(C(=O)NCCCNC(C(COC)OC)=O)CCCCC1c1nc(S)n[nH]1 c1(C(=O)NCC2N(C(C3CCC(OC)CC3)=O)CCC2)cnc2n1CCC2 c1(-c2cn(CC3N(C(C4C=CCC4)=O)CC=C3)nn2)ccc2ccccc2c1 C=C(Br)CCC(=O)N1CC(NC(=O)C(C)NCCCC)C(F)C1 c1(CC)nn(C)c(C(=O)NCC(C)NC(c2ccn(C)c(=O)c2)=O)c1Cl N1(C(Cc2nccc(OCC)n2)=O)CCC(NC(=O)C(CCO)N(C)C)C1(C)C Cc1nc(C(=O)NCCC(O)CNC(C2(O)CCSCC2)=O)c(C)o1 c1(NC(C2(CNC(c3cc(OCC)no3)=O)CCC2)=O)nn(C)cc1C C1(C(N2CCC(CNC(C3CC(SC)C3)=O)C2)=O)CCCC(C)(C)C1 C(=O)(C1CC(=O)c2ccccc21)NC(CNC(C(C)OCC(C)C)=O)C c1(CCCNC(N2C(CC(=O)NC3CCC3)CCCC2)=O)cc(F)c(F)cc1F c1(CCC(=O)NCCC(C)NC(C2(C(C)C)COC2)=O)ccc(N)nc1 N1(C(C(C)SCCCC)=O)CC2(CC(NC(=O)C(C)OCCN(C)C)C2)C1 C(=O)(C(C)(CC)CCC)NCC(CCNC(CC=C=C)=O)O c1(C(N2C(C(=O)NC(c3c(OC)cccc3)C)CCC2)=O)ncc(F)cc1C C1(C)(NC(C)=O)CCN(C(C2(CNC(C3C4COCC34)=O)CC2)=O)C1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(C(=O)Nc1ccc(Cl)cc1C#N)CO2 Cn1cc(Cl)cc1CC(=O)NC1C2CC(NC(C3CC(C)(F)C3)=O)CC12 C1(CC=C)(C(=O)OC(C)(C)C)CCCN(CC(=O)N2CCC2)C1 Cc1c(C(N2CC(NC(C34CC(CCO3)C4)=O)C2)=O)sc2ccc(Cl)cc12 c1(C(N(C2CCN(C(c3cc(C(F)F)cs3)=O)C2)CCC)=O)cn(C)cc1C N1(C(c2c(C)scn2)=O)CCC2CN(C(=O)CCC3CCCCN3C)CCC12 C12(CNC(CC3C(C)CCC3)=O)CCC(CN(C(c3ccn(C)c(=O)c3)=O)C1)C2 C1(C(N2CC(CC(C)NC(c3c(C)n(CCO)nc3)=O)C2)=O)CCC(N=[N+]=[N-])C1 CC1CCc2nc(N3CCC4OCCC4C3)[nH]c(=NC3CCC3)c2C1 c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2n[nH]cc2cc1Cl CC(C)C(C(=O)N(CC(C)(C)C#N)C)C(C)NC(=O)CCCn1cccc1 C(=O)CC(C)(CN)C(F)(F)F.C#CCC(C(C)(C)C)c1nc(C(N)C2CC2)no1 C1(CNC(Cc2nc(C)oc2)=O)CCC(F)(NC(c2nn(C(F)F)cc2Cl)=O)C1 c1(OCCCC)cccc(C(=O)NCC(COC)NC(=O)C=C(Cl)Cl)c1 N1(C=O)CC(S(C)=O)C1.C1(CNC(=O)OC(C)(C)C)(CO)CC1(F)F C(=O)(CCC(C)SC)N1CCC(CCC(N2C(C(=O)OC)C=CC2)=O)C1 CC(C)CC(CNC(=O)CC1CCCOC1)NC(=O)C(C)CO c1(C(=O)NC2C(C(N3CC(OC)(CO)C3)=O)CC2)ccc(Cl)cn1 CC12CCC(CNCC3(C(=O)O)CC(F)(F)C3)(CC1)CO2 CC1(C)C(CNC(=O)C(F)F)CCN1C(C1Cc2nncn2C1)=O c1(NC(CC)(CNC(=O)CC2CC3(CCC3)C2)CC)ccc([N+](=O)[O-])cc1C CCC(C)CCC(O)CC(=O)N(CCCCCCNC(=O)C1=CCCS1)C C1(CNC(C2(OC)CCC2)=O)CCCCN(C(C23CCC2C3)=O)C1 Cc1cc(F)ccc1C(O)C(=O)NCCCC1(NC(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)NCC2CN(C(C(C)C)=O)C(C)(C)C2)ccc2c(c1)C=CS2(=O)=O CC1(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)CC2O)CCCCO1 C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC=C)C(C)C C=C(Cl)CCC(=O)N1CCC(CCNC(=O)C(C2CCC2)OC)CC1 C1(C(N2CCC(C3CC3)(NC(=O)CSC(F)F)C2)=O)CCC2(CC1)CC(O)C2 c1(OC)ccc(Cl)cc1S(=O)(=O)NC1CN(c2nccc(C(C)C)n2)CC1F CC(C)CC(CN=c1cc(C(C)(C)C)nc(Cl)[nH]1)NC(C1C=C1C)=O CC1C(NC(c2cccc(F)c2)=O)CC2CCC1N2C(=O)Cn1ccnn1 C1(C(N(C2CCN(C(C3(F)CCOC3C)=O)C2)CC)=O)CCC(N=[N+]=[N-])C1 N1(C(C(CSC)O)=O)CCC2CC2(C(=O)NC(c2nc(C)cs2)C)CC1 C#CCCC(=O)NCc1cn(CC(C)NC(=O)C(C)OCOC)nn1 Cc1c(NC(c2cccc(F)c2)CF)cccc1NC(C(=O)OC(C)C)=O Cc1cc(C)c(C(=O)NCCCN(C(C2CC2c2ccc(F)nc2)=O)CC)cn1 N1(C(CCNS(C)(=O)=O)=O)CCC(C(F)CNC(c2cccnc2O)=O)CC1 C(=O)(CCCCCCC(C)C)NCC(CO)NC(CCCC(=C)C)=O c1(C(N2CC(CNC(C(CN(C)C)O)=O)OCC2)=O)nnc2ccccn12 n1(CCC(=O)NCC2C(NC(C=C(CC)C)=O)CC2)ncc2c1CCCC2 N12CCC(CC1C)OCCC(O)C2.C(C)(C)(C)OC C(C)(C(=O)NC1CC(NC(=O)CC2(O)CCC2)C1)OC(C)=O c1(C(N(CCC(C(C)C)NC(C2CC3C=CC2O3)=O)C)=O)ccn2ccnc2n1 CCCCCC(O)C(=O)N1CC(C)(C)CC1CC(=O)NCCNC(=O)C(C)(C)C C1(C(=O)NCC(c2ccc(F)cc2)NC(COCCCOC)=O)CCCC(=O)N1 S(=O)(=O)(c1cc(F)ccc1C#N)NC1CCN(C(CC)CC)C1 c1(C(=O)NC2(CCNC(C(C(C)OC)O)=O)CCC2)cccc2nccn12 C1(N(C)CC2(C(=O)OC)C=CCC2)CCN(C(=O)OC(C)(C)C)CC1(C)C C1(C(=O)NC(CCNC(c2ccc(C(CC)(C)C)cc2)=O)C)CCCCS1(=O)=O c1(C(=O)OCC(C(C)C2CCOC2)=O)cccc2oc(C(C)C)nc12 CCC(CC(F)(F)F)NC(=O)NNC(c1cc(F)cc(F)c1)=O CN1C(=NC(=O)c2ccn(C3CCCCC3)n2)NC(=O)C1O CCCC(CNC(=O)Cc1ccns1)C(=O)NC(C)(C)CC(N)=O C1(CNC(C2(OC(C)C)CCC2)=O)CCCCN(C(c2cccc(CF)c2)=O)C1 N1(C(C(c2ccnn2C)C)=O)C2CCC1CC(N(C)C(C1CCCCC1)=O)C2 C1(NC(C(c2ccccc2)OC)=O)CN(C(C2CC(F)C2)=O)C2(CCC2)C1 c1(C(N(CCNC(CC2(CC)CCCC2)=O)CCOC)=O)cc2cnccc2[nH]1 CCC(C)C(C(=O)NCC(C)(C)OCC(=O)NCc1ccc(OC)nc1)OC Cc1cc(C2CCC2)ncc1C(N1CCCN(C(C2(NC(N)=O)CC2)=O)CC1)=O C1(C)(NC(C(C)Cn2ccnc2)=O)CCCC1NC(c1cc[nH]c1C1CCC1)=O C(=O)(CC(C)(O)C1CC1)NCCN(C(C1CCC(C)CC1)=O)CC N(C1CCCc2ccoc21)C(C1(NC(c2ncn(C(C)C)n2)=O)CC(CO)C1)=O c1(C(C(=O)NC(CCNC(c2c(CC)n(CC)nc2)=O)C)O)cc(F)cc(F)c1 c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN2C(C2(C3CC3)CC=CC2)=O)n1 S(=O)(=O)(CC(=O)NCC1C(C)CCN1c1ncc(O)cn1)NC Cc1nc(Cl)c(NC(C2CN(C(c3ccc[n+]([O-])c3)=O)CCN2)=O)c(Cl)n1 CC(F)(F)C(C)(C)C(=O)NCC1CCC1NC(c1ccc(-c2cc[nH]n2)cc1)=O N1(C(c2c(OC)scc2)=O)CCC(C(F)(F)F)C(CNC(=O)C(F)=C(C)C)C1 C(=O)(CC(CNC(C1CC2CCCCC12)=O)C(F)F)OC N1(C(C(CC(C)C)O)=O)CCN(C(=O)CCc2cccc(C#N)c2)CCC1C CC(C)(C)C(CO)C(=O)NCC1CC(NC(=O)Cc2ccc(F)c(Cl)c2F)C1 C(CS(=O)(=O)CC(=O)N1CCC1CNC(=O)C(N1CCCCCC1)C)OC N1(CCC#N)C(C)(C)CCCC1(C)C.c1(OC)ccc(Cl)cc1C(O)CN C1(NC(c2cnc(CC(C)C)s2)=O)CCCC(NC(C2(F)CCCCC2)=O)CC1 O=C1NCCC1C(=O)NC(C1CCCCC1)C(=O)NCCOCC1CC1 N1(C(CC2N(C(c3cc(C)ncn3)=O)CCC2)=O)CCC(C)C(CO)C1 C(c1ccc(F)c(F)c1)=CC(=O)N(C(C)(C)C)CC.n12cc(nn1)CNC(=O)C2 c1(NC)ccncc1C(=O)NCC1CCCN1Cc1ccc(C(=O)O)s1 CC12CCC(C(=O)N(O)Cc3cn(C4CCC4=Cc4cccnc4)nn3)(CC1)OC2 c1(OC)ccc(OC(=O)C(C2CC=CCC2)NC(C2CC(=O)CCO2)=O)cc1 C1(C(N(CCCNC(C2C(C=C)C2)=O)CCO)=O)CCCN1Cc1ccccc1 C(CCCCCN=c1[nH]nc(-c2ccccc2)o1)N(C(C(C(CC)C)OC)=O)C C1(C(=O)NCCN(C)C(C2CCOC2C(F)(F)F)=O)CC2OC(=O)OC2C1 C1(CS(=O)(=O)NC)CCN(CC2CC(=C)C2)CC1C c1(C(=O)NC2CCN(C(Cn3ncc(CC)c3)=O)C(C)C2)cnc2[nH]ncc2c1 C1(C(C)NC(C2(C(F)(F)F)CCC2)=O)CN(C(c2nn(C)cc2N)=O)CCO1 CC(C(=O)NCC1(O)CC(C(=O)NCC2SCCS2)C1)S(C)(=O)=O C1(OC)CC(CCNC(c2cn(C)cn2)=O)N(C(=O)CSc2ccncc2)C1 Cc1cccc(Br)c1CN1CC(CC(=O)NCCCOCc2nccn2C)C1 c1(NC(=O)C2=CCC2)cccc(NC(C2C3CCCOC23)=O)c1 C1(O)(CN(C(c2ccc(Cl)cc2C)=O)CC)CCN(C)CC1 N1(C(CSCC)=O)CCC2(CCC(CNC(c3ocnc3C)=O)OC2)CC1 C=CC1(C(N2CCC(OC3CC3)C2)=O)CCN(C(C2CC23CCC3)=O)CC1 c1(C(=O)NC2CC3CN(C(C4CCC(C)CC4)=O)C2C3)ncc(P(C)(C)=O)cn1 C=CCC(C(=O)NCCC1(NC(=O)C(O)C(C)C)CC1)C(C)C C(=O)(CC1OCc2ccccc21)N(C)CC1(CNC(CCC=C)=O)CC1 C1(NC(=O)NC(C)(C)C)CCC2(C1)CC2C(=O)OC CN1CCOCC1C(N1CC(C)(CNC(=O)Cc2ccccc2C(F)(F)F)C1)=O Cc1cnn(C(C)C(=O)NCC2CC2NC(C2CC2c2ccc(Cl)s2)=O)c1 c1(C(N2CCC(C3CC3)(NC(C=CC=CCC)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(CNC(c2cccc(OCC)c2)=O)cc2n(n1)CCN(C(=O)C(C)CC#N)C2 c1(C(N(CCC(=O)NC2CCC2CO)C(C)C)=O)ncc2ccccn12 Clc1ccc(-c2cc(C3CCN3Cc3ccsc3)on2)cc1 C(CNC(c1csc2cncn12)=O)(CC(F)(F)F)NC(CC(C=C)C)=O C1(NC(C2(C)CCCOC2)=O)CC2CC1N(C(c1c[nH]nc1C1CC1)=O)C2 C1(NC(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(=O)CCSc1ccccn1 C(=O)(C1=CCC2CCC1N2C(c1cncc(Cl)c1)=O)N(CC(CC)O)C C1(C)(CC(=O)NCC(CC=C)NC(=O)Cc2cnccn2)CCCCC1 C(=O)(NNC(=O)CCCN)NC(c1ncc(CC)s1)C c1(C(N2CC(O)(CNC(c3nc(CC)oc3)=O)C2)=O)n[nH]c2cc(OC)ccc12 C1(C(N(C)Cc2ccc(CC)o2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C(C)(C(C(=O)NC(C)(C)CC=CC(=O)NCC1COCCN1C)N(C)C)OC n1(CCC(=O)NC(CC)CC(=O)NC2(C3CC3)CCCO2)c(O)nnc1O C1(C(N(C(CNC(c2ncc(CC)nc2)=O)C)CC)=O)CCc2cnnn2C1 C1(NC(C(C2CC(F)(F)C2)OC)=O)CCCN(C(C2OC(C)CC2C)=O)CC1 C1(OC)CC(CCNC(c2csc(O)n2)=O)N(C(=O)CCOCC2CCCO2)C1 C=C(C)CC(C(=O)N(CC(C)(C)CNC(C1CCC1C(=O)OC)=O)C)NC(C)=O C1(NC(c2c(CNC(c3nsnc3O)=O)occ2)=O)(CO)CC(F)(F)C1 N1(C(c2c(-n3ccc(C)n3)cccc2)=O)CC2(CC2)c2ncccc21 CN1C(=O)CC(NC(N2CCN(C(=O)CCCC#N)CC2)=O)C1c1cnn(C)c1 N1(C(=O)CN2CCN(C(c3cccs3)=O)CC2)CC2CCC(C1)C2O N1(CC(=C)C)CCc2cc(OC)c(F)cc2C1 N1(C(C(C)(C)C2CCOCC2)=O)CCCC(CNC(=O)CN2CC3C=CC2C3)C1 C1(CNC(=O)CN2CC3CC3C2)CCC(C(N2CCC3CC23)=O)CC1 C(=O)(C(Cc1ccccc1)C1CC1)N1CC(OCCOC)C1 N1(C(C(CC)SC)=O)CCN(CCCNC(C2CCCN2C=O)=O)CC1 C1(CC)(CC)CC(O)CN1C(c1ccn(CCNC(=O)C(C)(Cl)Cl)c1)=O C1(C(=O)NC2CC(CNC(COCC(=C)C)=O)C2)CCCCC(C)(C)C1 c1(C(=O)NCCC(F)Cn2cc(CCCO)nn2)cnc(O)c2ccsc12 N1(C(C(CCC)(C)O)=O)CCC2(CC1)CC2CNC(c1ccnnc1O)=O C1(C(=O)NCC(C2N(C(COCC(C)C)=O)CCC2)(C)C)C(F)(F)C12CC2 c1(C(=O)NC2C(CNC(C3(C(C)C)CC3)=O)C2)cc2ccc(F)cc2nc1O Cc1cc2ccc1CC1OCCN(C1)C(=O)N2.C1(CN(C)C)CC(F)(F)C1 C1(C(=O)NC2C(C)CCC2)CC2OCCC2N(C(=O)Cc2ccsc2)C1 c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)CC3(C2)CC3)=O)ccc2c(cnn2C)c1 CC1CC(NC(C2C3COCC23)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 c1(C(=O)NCCC2OCCN(C(C3ON=C(CC)C3)=O)C2)cnn2c1OCCC2 CC1CC(NC(C2(O)CCSC2)=O)CN(C(c2cnn(C(C)(C)C)c2)=O)C1 N1(C(c2ccc(Cl)[nH]2)=O)CCC2OCCN(C(=O)CCc3cnoc3)C2C1 c1(C(=O)NC(CNC(C2CC3(C2)CC(F)C3)=O)CO)cc2cccc(Cl)c2s1 C(c1ccoc1)=CC(C)(C)NC(=O)NC12CC(CO1)C2 C12(C(N3C(CN(C)C)C=CC3)=O)CCC(CN(C(=O)CCC3CCCC3)C1)C2 c1(C(N2CCC(C(=O)NCCC3CC(F)C3)O2)=O)cccc2[nH]ncc12 C1(C(=O)NC2CC(C(=O)NC(c3cccnc3F)C)CC2O)CC2(CC2)CN1C N1(C(C(CSC)(C)C)=O)CC2(CC(CNC(=O)Cc3cc(F)ccc3C)C2)C1 C(CC(C(=O)NCC(C)C1CC1)NC(c1ccc(OC)o1)=O)OCC C(CCN(C(=O)CCc1ccccc1)C)(C(C)(C)C)NC(CSCC#C)=O N1(C(CSCCN(C)C)=O)CCC2(NC(=O)C=Cc3ccsc3)CCCCC12 c1(NC(CNC(CNC(c2c(CCC)[nH]cc2)=O)=O)=O)cncc([N+](=O)[O-])c1 c1(C2C(C(N3CC(F)(c4ccccc4)C3)=O)C2)cccc(C(F)(F)F)c1 Cc1cccc(CC(=O)NCC2(O)CC(NC(=O)C(c3ccccc3)F)C2)c1 O=S(=O)(c1c[nH]ccc1=NCC1CC2(CCCCC2)CO1)N1CCCCC1CF c1(CCCC)ccc(Oc2ccc(N(S(C)(=O)=O)Cc3nncn3C)cc2)cc1 c1(CC(=O)NC2CN(C(C3COCCO3)=O)CC23CC3)cc(Br)cnc1F C1(CCC)(NC(=O)CNC=O)CCN(C(c2cn(C)nc2C)=O)CC1 C1(C(=O)NC2C(CC(=O)N(C(CC(C)C)C)C)CCC2)COCCN1C C1(NC(c2ccc(C(C)=O)o2)=O)CCC(O)CN(C(c2nccc(C)n2)=O)C1 c1(C2(C(N(C(CNC(c3cc(C)[nH]n3)=O)C3CC3)C)=O)CC2)cccc(Cl)c1 c1(C2N(C(C3C(NC(CC(=O)OCC)=O)CCC3)=O)CCC2)ccccc1F.C(=O)OC Cc1cc(Cl)ccc1C(=O)NCCC1CCCN1C(c1cnc(S)n1C)=O C1(CNCCC(CC)CC)CCC2C(CC1)C2(F)F n1(CC(C)C)[nH]c(CC(=O)NCC2(NC(=O)Cc3cnc[nH]3)CC2)cc1=O N1(C(CC2CN(C(Cn3c(C)ccn3)=O)CC23CC3)=O)CC2(COC(C)C2)C1 CCCCC(CC(=O)N(CC(C)(O)C1CC1)C)NC(C1CC2CC(=O)C1O2)=O c1(CCC(=O)N(C2(NC(CN(C(=O)OC)C)=O)CC2)C)ccc(Cl)cc1F CC(C)(O)C(F)C(=O)N1CC2CC1C2NC(=O)CC1=CCCC1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(C2(C(F)F)CCCC2)=O)CC(C)(C)C1 c1(OC)c(C(N2CC(F)CC2C(=O)Nc2cc(C)c(F)cn2)=O)cccc1Br N1(c2ncnc(C(C)(C)C)n2)CC2CC(NC(=O)C(O)C(C)(C)C)CC2C1 C1(CCC)(NC(=O)C(C)CO)CCN(C(c2cccc(F)c2SC)=O)CC1 C12(NC(CC(=O)OC)=O)CCCC1CN(C(c1nccc3occc13)=O)C2 C1(C(=O)NCC(C)(C2CC2)NC(COCC=C)=O)CCC(C(N)=O)CC1 c1(C(=O)NC2CC(C(C(=O)NCCC=CC)F)C2)cc(OC)n[nH]1 C(=O)(CS(=O)Cc1cccc(Br)c1)N(CC=C)CCOC N1(C(c2ncc(C)cc2C)=O)CCC(NC(c2cnn3ccsc23)=O)C12CCC2 N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(C(=O)NC2C3C=CC(C3)C2CO)C1 c1(NC(C23C(CN(Cc4c(O)ccc(OC)c4)C2)C3)=O)cccc(C#N)c1F CN1C(=O)CSC1=CC(=O)NCC1(F)CCC(C(=O)NNC(=O)NC2CC2)C1 C1(COC)(NC(=O)C(C)C2CCC2)CCN(C(=O)Cc2ccc(Cl)cc2C)CC1 N1(C(c2cc3c(Cl)cccn3n2)=O)CCC2OCCN(C(C3CC(F)C3)=O)C2C1 C1(C(=O)NCC(c2ccccc2)CNC(CCCOC)=O)(OC)CS(=O)(=O)C1 C1(CC(=O)N(CCC(C)NC(CC2(OC)CC2)=O)C)CCCCN1C c1(C(=O)NC2(COC)CN(C(C3CCCCC3(C)C)=O)C2)ccc(C#N)cc1C CC1(NC(c2cc(=O)cc[nH]2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 C(=O)(CC(C(C)C)c1ccccc1)NCC(CNC(C1C(C)(C(C)C)C1)=O)O CCC(CC(C)C)C(=O)N1CCC2(C1)CN(C(c1ccc(O)c(N)c1)=O)C2 c1(C(N2C(CNC(C(C(C)(C)C)(C)C)=O)CC2)=O)cccc2c1C(=O)NC2 C1(C)(C(=O)NCCC(C)NC(=O)C=NO)CCCN1C.c12ccc(cc1)[nH]c2=O c1(CNC(C2(CCC=C)CN(C(=O)C(C)CCC)C2)=O)cncc(C#N)c1 C1(C(N2CC(CNC(C(C(=O)OCC)F)=O)C(C)C2)=O)CCOCC1(C)C N1(C(c2c(C)nc(C)o2)=O)CC2C=CC1C(C(=O)NC1CN(C(N)=O)C1)C2 C(=O)(CC(C)C(F)(F)F)NCC1(C)C(C)CN(C(c2c(NC)nccc2)=O)C1 CCC(C)C(O)C(C)C(=O)N1CC(CC(NCP(C)(C)=O)=O)(OC)C1 c1(NC(C2CCOCC2)C=C)nccc(N(C)CC2CCN(C)CC2)n1 N1(CC)CCCC(C2CN(c3ncc(NC(=O)CCCCCO)cn3)C2)C1 CC1(C)CC(NC(=O)Cc2cc[nH]c(=N)c2)CN(C(c2ccc(Cl)s2)=O)C1 c1(C(=O)NC2CN(C(C3(C=C)CCCC3)=O)C2)cc(N(C)C)ccc1F Cc1c(C(N2CC3CC(NC(c4ccncc4O)=O)C3C2)=O)cnc2ncnn12 Cc1cc(=NC2CCN(C(c3noc4c3CCCC4)=O)CC2)[nH]cc1C#N c1(OC)nc(Cl)ccc1C(=O)N(CCC(C(C)C)NC(=O)CC(O)C(C)C)C c1(OC)cccc(CNC(C2CSCCN2C(=O)COC2CCC2)=O)c1F N1(C(C(C)CO)=O)CCC(CNC(=O)CC2CC(F)(F)C2)C(F)(F)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(C(CCOC)C)=O)c(C)cc(C)oc1=O Fc1nc(F)c(F)cc1-c1nc(COC2CCC2)nn1CCCc1ccccc1 C1(CNC(C2CC(C#C)(O)C2)=O)CC12CCN(C(=O)C=C(C)Cl)CC2 CC1(C)CN(C(=O)C(CNC(C2(C)C=CCC2)=O)CC2CC2)CCS1 N1(C(C2C(C=C)C2)=O)CCCC12CCC(NC(=O)C=C(C)CCC)CC2 Cc1cccc(F)c1C(N1CCCC(CCCCNC(c2cnn[nH]2)=O)C1)=O C1(CNC(C(COC)NC(C)=O)=O)CCC2(CN(C(c3ccnn3C)=O)C2)O1 Cc1ccc(CCC(N2CC3CN(C(c4cncn4C)=O)C3C2)=O)c(C)c1 C1(NC(=O)CSC(F)(F)F)CCCC12CN(C(=O)Cn1cc3ccccc3n1)C2 n1(CC(C)C)nccc1CNC(C)(C(C)C)c1nnnn1C1(C)CC1.C1CN1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCC(O)(C(C)CNC(=O)CCN(C)CC)C1 C(=O)(CCC(C)NC(=O)CCc1ccc(C)o1)N1C(C(=O)OC)C=CC1 C(=O)(CS(=O)(=O)Cc1cccs1)NCC(CC)NC(=O)CCCC1CCC1 n1(CC(=O)NC2(C)CN(C(C(CC)(C)C#N)=O)C2)cc(C(N)=O)c(O)nc1=O N1(C(CCCOCC=C)=O)CCCCC1CN(C(=O)CCCCF)C c1(C(N(C(C)CNC(c2ncnc(C)c2C)=O)CC)=O)cc(N)cc([N+](=O)[O-])c1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(CCNC(C(CCC#C)O)=O)CC1 c1(C(C)N(C)Cc2cccc(O)c2)nc2c(s1)CCCC2 c1(C(=O)NC2(C(=O)NC(C)C(F)(F)F)CCCC2)cc(F)ccc1F c1(C(C(N2CCC(NC(C3C4CC4C4CC34)=O)CC2)=O)=O)ccc(Cl)cc1O Cc1cnc(C(=O)NCC2(CCNC(=O)CC34CCC(CC3)C4)CC2)cc1Cl c1(CCC(=O)NC2CCCC23CC3)ccccc1-n1cc(CCCCO)nn1 c1(C(=O)NCC(CC=C)NC(C2CC(=C3CC3)C2)=O)cccc(OC2CCC2)c1 C1(CNC(C2C(=O)NCC2)=O)(NC(=O)CC2CCC(C(F)(F)F)O2)CCCCC1 CC1CN(C(=O)CC2CCCCC2NC(=O)C(C)CC(F)(F)F)c2ccccc21 c1(C2C(C3N(C(C(C)N(C(=O)CCF)C)=O)CCCC3)C2)cccc(F)c1 c1(C(N2C(COC)CN(C(=O)CN(C)C(C)=O)CC2)=O)nc2c(s1)COCC2 c1(C(C)NC(N2CCC(C(N3CC4CC4C3)=O)C2C(=O)O)=O)ccc(Cl)cc1 c1(C(=O)NC(CC)CN(C)C(C2(C)CNC(=O)C2)=O)cccc(C)c1C#N CCCC(CCC)=CC(=O)NC1(CF)CCN(C(=O)C(C)(C)N2CCCCC2)C1 C(=O)(CCCCCCC)NCC1(C(=O)NCCCC)CCCO1 C(=O)(CCC(C)C)NCC1N(C(C2N=C(C)SC2)=O)CC1 Cc1cc(C(N2CC(C(O)C(=O)NC3CCC4(CCC4)C3)C2)=O)cnc1O Cc1ccc2c(c1C(=O)NC1CCCC1NC(=O)C(C)c1cc[nH]n1)CCCN2 C(=O)(CCCN(C(=O)CC1C=CCCC1)C)N(C1C(C)CC1)C C1(CC(=O)O)CC(CC(=O)NCc2cccc(OCc3ccccc3)n2)CCO1 Cc1noc2cc(C(=O)NC3CCC34CN(C(=O)CN3CCCC3=O)C4)ccc12 Cc1cc(C(N2CCCC2CNC(=O)CN2CCCCC2C)=O)ncc1C(N)=O c1(C(=O)NCC(CCNC(C(C=CCCC)O)=O)O)sc(C)c(C)c1C N1(C(C2C(OC)CCCC2)=O)CCC(CNC(c2cnc(Cl)[nH]2)=O)C(C)C1 N1(C(CC(C)O)=O)CC(C)(C)CC1CNC(=O)CCCCN(C)C c1(NC2C(c3ccc(C)cc3)CCC2)ccncc1S(=O)(=O)NCc1cncs1 C1(C2CCN(C(=O)C=Cc3ccc[nH]3)C2)(NC(CCCNC(N)=O)=O)CC1 C1(NC(c2cnc(C)[nH]2)=O)(CO)CCCN(C(C2CCCN(CC(F)F)C2)=O)C1 C(=O)(CS(=O)(=O)CCO)N1C(C(C)NC(C(C(C)(C)C)NC(C)=O)=O)CCC1 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C)(COC)CC(NC(=O)CC=C(C)C)C1 C(=O)(C1=CC2(CCN(C(c3csc(C#N)c3)=O)C2)C1)N1CC2C(C)(CSC2)C1 n1(C(N(CCN(C(=O)CCOC2CCCC2)CC)CC)=O)nc(C)c(C)c1C N1(C(C2(CCC=C)CCCC2)=O)CC(CNC(=O)C(C)CC)C(C)C1 CC1CCC2(CC2)N(C(C2CCC(C)(C)N(C(=O)CC3COCCO3)C2)=O)C1 C12(CNC(=O)Cc3cnc[nH]3)CCC1CN(C(c1ccc(C3CCC3)nc1)=O)C2 Cc1cc(C(=O)NCC2CC2CNC(C2(C)CC2Br)=O)nn1-c1ccccc1 N1(C(CCC#C)=O)CCN(C(c2nc(C)ccc2F)=O)C(C)CC1C N1(C(C2(COC)CCCO2)=O)CC(CNC(c2cc(O)nc(O)n2)=O)C(F)(F)C1 c1(C(N2CC(NC(C(CCCC)O)=O)(CO)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(CN(C(=O)OC)C)=O)CC2CCN(C(=O)C=Cc3ccc(F)cc3)CC2C1 c1(CC(N2CCN(Cc3cc(O)ncc3Br)C3CC23)=O)ccc(Br)cc1I C1(NC(C2CCS(=O)(=O)C2)=O)CC2CCC(C1)N2C(=O)CCC1CCCC(O)C1 c1(C(N2CC(NC(C(c3cn(C)nc3C(F)F)C)=O)C(O)C2)=O)ccc(Cl)nc1N C#Cc1ccc(OC)c(C(=O)NC(C)(CNC(=O)Cc2ccc(F)cc2)CC)c1 Cc1ccc(C2(C(=O)NC3CCN(c4nc(C)cs4)CC3)CC2)c(Cl)c1 Cc1cccc(C)c1CC(N1CC(C)(C)CC1CNC(=O)C(c1cccnc1)O)=O C=C(C)CCCC(=O)NCC1CCC(NC(=O)CCCC2CCCO2)C1 C1(CNC(Cc2c(C)con2)=O)CC(C(=O)NCCC2(C)CCCO2)=NO1 C1(O)(C(C)NC(C(C)=C2CC2)=O)CCN(C(C2CCC(=O)N2C)=O)CC1 C=CCCCCCCCC(=O)NCC(O)CCNC(=O)Cc1ccccc1OC CCC(CCC(=O)NC(CNC(C1CCC(=O)N1)=O)C1CC1)OC CC1(C(=O)OC2CC3(CCC3)C2)CC2C=CC1C2.C1CC(=O)CNCCO1 C1(C(=O)N(C)OC)(CC)CCCN(C(=O)Cc2ccc(OC)cc2)C1 C(C(C)N=c1[nH]c2ccccc2cc1C#N)(C1CCCCC1)NC(C(C=C)O)=O O=C(CCCC(=O)NCC1CC(C(N2C3CCCC2CC3)=O)C1)C1CC1 C(=O)(C(C)CC1CCC1)N(CCC(=O)NCC1CC12CC2)CC=C c1(CC(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCCCC2)cn2ccccc2n1 c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cnc2cccnc2c1 C(C)(N=c1[nH]c2ccc(Br)cc2o1)CN(C(COc1ccc(OCC)cc1)=O)C c1(C(=O)NCC2N(C(c3ccc(C)o3)=O)CC=C2)cc(C)c(F)c(C)c1 C1(C(=O)NC(C)CO)CN(C)CCN1C(=O)CCS(C)(=O)=O c1(CC(=O)NC2CN(C(=O)OC(C)(C)C)CCC2c2nn[nH]n2)cc(F)ncc1Br c1(C(=O)NC(C(N2CC(C#C)C2)=O)C)cncc(F)c1 CC1(C)CC(NC(c2conc2-c2ccccc2)=O)CN1C(=O)CNC(N)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)C2=COCC2)CC1c1ccccc1 C(=O)(C1=CCCOCC1)NCCC1C(C)CN(C(=O)CC2(C)CCOCC2)C1 N(C(=NCc1ccc(NC)cc1)N1CCC(C(=O)NC)C1)C(C=C)C N1(C(C2N(C)CCC2)=O)CCCC(NC(=O)C(F)(F)c2csc(Cl)n2)CC1 c1(OC)cccc2[nH]c(-c3cccnc3C(=O)NC3CCNC3=O)cc12 Cc1cc(CNC(=O)CN(CC(C)C)C(C2CCCC(=O)CC2)=O)cnc1C c1(CN2CCCC(C(=O)NCC3N(CCC)CCCC3)C2)c(OC)cccc1F N1C2CCC1CN(C(c1cnc(Cl)cn1)=O)CC2.Cc1coc(C2CCCCC2)c1 N1(C(c2c(C)nccn2)=O)CC(NC(=O)C(c2ccc(Cl)c(Cl)c2)C)C(C)(C)C1 C(=O)(CC1=CCCC1)NC1C(NC(CCC=CCC=C)=O)CCC1 N1(C(C2C(COC)(COC)C2)=O)CCC(C2(NC(=O)CC3COCCO3)CC2)C1 c1(CN2CC(C)C2)ccccc1NC(C1CN(C(=O)COC2CCCCC2C)C1)=O c1(C(=O)NC(CC)CNC(=O)CCCNC(=O)C(C)(C)C)cc(O)cc(Br)c1 C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 c1(CC(C)NC(=O)NC(c2ccccc2)C2CC2)cn(C)c2ccc(F)cc12 C(=O)(CCCCC#N)NC(c1ccc(C)cc1)CNC(C1(Cl)CC12CCC2)=O C=CC(C)(O)C(=O)NC1CCOC1C(=O)NC1CCNC(=O)C1 C1(C)(C(=O)NCC(CN(C(CCC=C=C)=O)C)C)CCC(=O)NC1 CC(C)CC(C)(O)C(=O)N1CCC(F)(C(=O)NC2CC(CCO)C2)C1 c1(C(N2CCC(NC(c3cnc(CCC)s3)=O)CC2)=O)cnn2c1CN(C)CC2 N1(C(C(C)C(C)(C)C)=O)CC2(CCN(C(=O)CCC3NC(=O)NC3=O)CC2)C1 Cc1cnncc1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCC1CC1 CN(C)S(=O)(=O)N1CC2CC2C1=NC(O)COCc1ccccc1 CCC(CC)C(C(=O)NC1(COC)CCN(C(c2ccc(OC)s2)=O)CC1)OC CC1=C(C(=O)NC2CN(C(c3onc(C)c3C)=O)CC2O)CCS1(=O)=O N1(C(C(C)OCC)=O)CC(CNC(c2csc(C(F)F)n2)=O)C(O)C1 CC(O)C(C(=O)NC1CC(OCC(=O)NC2COCCC2O)C1)OC C(=O)(C(C)(C)C(C)(C)C)NC1CC(N(C(C23CCC(OC)C2CC3)=O)C)C1 c1(C(=O)NC2C(CNC(CCCN(C)C)=O)C2)nc(Br)n2c1COCC2 C(C)(C)(CCC(=O)NC1CCCC(OC)C1)NC(C(COC)COC)=O C1(CNc2ccc(C(=O)OC)cc2C)CN2CCCN1CC2 N1(C(C(N2CCC(O)CC2)C)=O)CC2CC(C1)CN(C(c1csnn1)=O)C2 C=CCC(CC=C)C(=O)NCC(c1cccc(C)c1)NC(c1cc(OC)cs1)=O Cc1ccnc(O)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 C1(C)(CN(C)C(c2ccc(CC#N)cc2)=O)CCCC1NC(c1ccoc1Cl)=O C1(NC(=O)C(=Cc2c[nH]cn2)F)CCOCC1NC(=O)CC1CCCC12CC2 c1(C(N(CCNC(C(C)N2CCC2)=O)C)=O)ccc(=O)n2c1CCCC2 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC(C1CC1)NC(C(COC)(C)C)=O Cc1cnc(Cl)c(CN2CCSC(C(=O)Nc3ccccc3CO)C2)c1 C1(COC)CC(CNC(c2cc(C3CC3)sn2)=O)N(C(C2CCOCC2)=O)C1 CCC(C)(C#N)C(=O)NCCC1CN(C(c2nccn2C)=O)CCCO1 C1(NC(CCCOC)=O)CC(CNC(c2ccc(C)nn2)=O)C1(C)C c1(C(N2CC(F)CC(C(=O)Nc3cc(O)n[nH]3)C2)=O)ccc(F)c(F)c1O C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(C2(CCO)CC2)=O)CC2(CC2)C1 c1(OC)ccc(C(CNC(=O)C=CC2CC2)NC(C2OCCCO2)=O)cc1 N1(C(CC(C)(C)n2cc(CNn3ccnc3)nn2)=O)CCn2nc(CO)cc2C1 N1(C(C(C(CC)(C)C)=O)=O)CC2CCCC(NC(c3ccno3)=O)C2C1 C1(CC)(CC)CN(C(C2(NC(c3ccncc3F)=O)CCCC2)=O)CCO1 C1(C(N2CC3C(N(C(=O)C=C4CCSCC4)C)C3C2)=O)CCN(CCO)C(=O)C1 Cc1cc(C(=O)NC2CC(CNC(C3CCC(C)(C)CC3)=O)C2(C)C)nc(C)c1 N1(C(CC2CC(=O)OC2)=O)CCC2(CC1)CC(NC(c1occc1Br)=O)C2 C=C(C)C(CC(=O)NCC1CCCN(C(=O)CCC2CCC(C)O2)CC1)OCC C1(NC(c2n(C)nnc2)=O)C2CCN(C(c3cccc(O)n3)=O)CC12 c1(OC)cccc2c(C(N3CCCC(NC(=O)CCC(F)(F)F)C3)=O)c(C)[nH]c12 C1(NC(CN(C)C)=O)CN(C(=O)CC2OCCCC2(C)C)C2(CCC2)C1 C1(C2C(=O)N2)CCc2c(nnn2C)C1.C(=O)(CC(C)C)N1CC(N(C)C)(SC)C1 c1(C(=O)OCC)cnn2c1N(C(c1ccnc(N(C)C)c1)=O)C(C)CC2 CCS(=O)(=O)c1ccc(-c2ccnc(C(N3CCOC(CO)C3)=O)c2)cn1 C(=O)(C(O)C(CCC)NC(=O)C(C)C(O)C(C)C)N(CC(=C)C)CC#C C1(OC)Cc2cc(F)ccc2N(Cc2c(F)ccc(C(=O)N(C)C)c2Cl)C1 N1(C(COCC=C)=O)CCC2(CC1)CC(NC(c1cccc(C)c1)=O)CCO2 C(C#CC(=O)NC(C1CCCN(C(c2cccnn2)=O)C1)C)(OCC)OCC C1(CC(=O)NCCc2cn(CCNC)nn2)CCCN(c2ccc(OC)cc2)C1 c1(C(=O)NC2CCCC(NC(c3ccns3)=O)CC2)cccc2c1CCC2 N1(C(C2(C)N(C(c3c(C)nsc3)=O)CC=C2)=O)CCCN(C)C(=O)C1 c1(C(=O)NC2CCN(CCO)C23CCOCC3)nn(C)c2ccc(F)cc12 N1(C2C(NC(c3cccs3)=O)COC2)CCN(C(=O)C2=CSCS2)CC1 Cc1nc(C(N2CCC(CO)(NC(c3cncc(N)c3)=O)C2)=O)cn1C c1(C(=O)NCCC2N(C(c3c(C)snn3)=O)CCC2)nc2sccn2c1C c1(OC)cc(F)c(C(=O)NCCNC(c2ccc(CO)c(Cl)c2)=O)cc1Br c1(C(C)C)ncsc1C(=O)NC(C)CN(C(=O)C(C)Oc1ccccn1)C C1(CC)C(C(=O)NC2(C(=O)N(C)CCc3ncon3)CCOCC2)CCN1C C1(NC(C(C)(C)CCC#N)=O)CN(C(=O)CC(O)C2CCCC2)CC2(CCC2)C1 N1(C(COCC(=C)C)=O)CC2(C1)CN(C(=O)CCN1CCCC1=O)C2 Cc1cc2c(C(N3CC(CNC(c4ccc(C)s4)=O)CCC3C)=O)cccc2o1 c1(CNC(CCCCC)=O)nnc2n1CCN(C(C1(n3cccn3)CC1)=O)C2 C1(C)(CNC(CC(c2ccc(C)cc2)C)=O)CCCN(C(C2CNC(=O)N2)=O)C1 c1(C(=O)NCC=CCNC(C2(C)CCN(C)CC2)=O)ccn2c1CCCC2 C(c1cccnc1)=C(C)C(=O)NC(C1CCCN1C(=O)Cc1cnn(C)c1)C C1(C)(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1 CC1(CCNC(=O)CCF)CCN(C(=O)C(O)c2ccsc2)CC1 c1(SC)ccc(CNC(=O)Cn2cc(C(=O)OC(C)(C)C)nn2)cn1 c1(CC(=O)NCCN(C(COCC)=O)CC(C)O)cnn2c1OCCC2 C1(NC(C2CCCC(C)C2)=O)(CO)CCCN(C(=O)C#CC(=O)N(C)C)C1 c1(C(C)C)ncc(C(=O)NC(C2CCCCO2)C2CC2)[nH]1 n1(CC(=O)NC2CC(C)N(c3ncc(C#N)cc3Br)C2)cc2ncccc2n1 c1(C(=O)NC2(CCC)CCCN(C(C(C=CC)O)=O)C2)ccc(Cl)c(Cl)c1N N1(C(CCN(C2CCCCC2)C)=O)CC(NC(c2cccnc2O)=O)CC2(CC2)C1 Cc1nc(SCC(=O)NCCC(O)CNC(C2C(C)C2C)=O)n[nH]1 C(C1CN(C(C2(C)CCC2)=O)CC1C(N1CC(F)(CC)C1)=O)=CC N1(C(CC(=O)NCC)=O)CCC(NC(=O)CCn2ccc(O)nc2=O)C(O)C1 C(CCC(C)C)(C(=O)N1CCC(C(C)OC)CC1)NC(C(CCCOC)C)=O N1(C(c2c(C)cccc2F)=O)CCOC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C1 c1(OC)cc(CN(CCCS(N)(=O)=O)C(=O)CNC2CCCO2)nc(C)c1 Cc1ccc(C2CCN(C(CCCc3nc(-c4ccncc4)cs3)=O)C2)c(C)c1 C1(C)(NC(C=C(C)C(F)F)=O)CCC(NC(c2cccc(C3CCC3)c2)=O)CC1 CC1CN(C(C2(C)CCCCC2)=O)CCN1C(c1cscc1Br)=O C1(CC#C)(C(=O)NCC(C)(C2CC2)NC(=O)Cc2c(C)noc2Cl)CCOCC1 CC1CN(C(=O)C(N2CC3CCC2(C(F)(F)F)C3)=O)CC(C)(C)C1 C12(NC(C=CC=CCC)=O)CC3CCC(C1C2)N3C(=O)Cn1nc(C)cc1C C(=O)(C#CC1CCOCC1)NC(C=CC(=O)NC1CCC(OC)C1)C c1(C(=O)NC(CCNC(C2C(COC)C2)=O)(C)C)c[nH]c2ccc(Cl)cc12 c1(C(C(=O)NCC2CN(C(c3c(C)nns3)=O)C2)C)ccc(Br)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CCN(C(=O)CCc2ncccn2)CC1 C1(CC(=O)NC(C2CC(NC(=O)CN(C)S(N)(=O)=O)C2)C)CCC(=O)N1C N1(C(c2cn(C)nc2)=O)CCC(C(C)(C)CNC(c2ncoc2C2CC2)=O)CC1 c1(SCC(=O)NCCCNC(c2cc3scnc3[nH]2)=O)ccc2c(c1)CCC2 C1(NCCCOC(C2(C(=O)NCCCCN(C)OC)CC2C)=O)CC(=O)N(C)C1 c1(C(=O)NCC(CN(C(c2ccc(C)c(Cl)c2)=O)C)C)c(C)sc2ccccc12 C1(CC=C)(NC(=O)CC2CC2C)CC2CCC(C1)N2C(c1cc(C(C)(C)C)on1)=O N1(C(C(C)CO)=O)CC(CNC(=O)C=C2CCOCC2)CC1(C)C c1(OC)cccc(F)c1C(=O)NCCCCNC(=O)C=Cc1ncc(C)[nH]1 Cc1cccc(C2(NCc3cc(C)[nH]c3C(=O)O)CCC2)c1 c1(CC)cc(N)cc([N+](=O)[O-])c1.C12CCC(O)(CC1)C(=O)N(CC(=O)C1CC1C)C2 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(CC(F)F)C1 C1(C(=O)NCCCN(C(=O)C(C)=C2CCCC2)CC)CCCN1c1nccs1 S(=O)(=O)(c1ccc(NC2CCC(F)(F)CC2)c(F)c1)N1CC(C)OC(C)C1 c1(C(N2CC(C(=O)NC)C(c3ccc(C)cc3)C2)=O)cnc(OC)c(F)c1 Cn1ccnc1C(=O)NC1CC(O)(C(=O)NCCOCc2ccccc2)C1 N1(c2nc(C)cc(C)n2)CCN(N2CCc3cc(F)ccc3C2)CC1 c1(CC)oc(C)cc1C(N1CCC(C(=O)Nc2cccc(F)c2)(CF)C1)=O c1(C(=O)NCC(CNC(c2ccc3n[nH]cc3c2)=O)F)nccc2ncncc12 c1(C(=O)NCC2CN(C(C(CCC)(C)O)=O)CC2C)ccc2c[nH]nc2c1 C(=O)(CCS(=O)(=O)c1ccccc1)Nc1ccc(OCC)c(OC)c1 c1(C(=O)NC2C(C)N(C(=O)C(O)CCS(C)=O)CC2)cccc2c1NCC2 CC1ON=C(C(=O)NC2C3CC(NC(C4C5COCC45)=O)CC23)C1C c1(NC(C(C)C)CNC(=O)Cc2cc[nH]n2)cc(-c2cccs2)ncn1 C(=O)(C1COc2ccccc21)N(C1CCN(C(C2(CN(C)C)CC2)=O)C1)CCC N1(C(CCSc2ccc(C)cc2)=O)CCN(C(=O)C(O)C(C)(C)C)CC12CCC2 N1(C(CSCCC)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(C2CCC2)C1 c1(C(N2CCC(N(C(C=CC(C)C)=O)CC3CC3)C2)=O)cc(N)ccc1Br N1(C(CC2C(=O)OCC2)=O)CCC(N(C(c2cnn[nH]2)=O)CC2CC2)CC1 N1(C(C2=CCC(NC(c3ccoc3)=O)C2)=O)CCCC(C2CC2)CC1 CCN=c1[nH]cnc2cc(C(=O)NCC(C)NC(=O)C=Cc3cccs3)ccc12 C#CCCC(C(=O)NCCc1ncc[nH]1)NC(c1cc(O)cc(F)c1)=O C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC=CCNC(C(CC(N)=O)O)=O c1(C(C)C)nc(NCCN2CCOCC2)cc(N2CCC(CF)CC2)n1 N1(C(C(C(C)C)O)=O)CC(CNC(c2cc(C(F)F)ccc2F)=O)C(C)(C)C1 c1(C(=O)NCC2CCCN(C(C3CC(=C)C3)=O)C2)ccc(Cl)c(C)c1 CS(=O)CCC(=O)NCC1CCCCC1NC(=O)CC1(CO)CCCC1 c1(CSCC)cc(C(N2CCC(N(C)C(c3cnn(C(F)F)c3)=O)C2)=O)no1 C1(NC(C2N(C)CCCC2)=O)CC2(CCCCN2C(=O)CC2(CO)CC2)C1 Cc1ccc(CC(=O)NC(C)CCCNC(c2ccc(Cl)nc2O)=O)cc1Cl C1(CNC(C2(C)CNC(=O)C2)=O)CN(C(=O)C#CC2CC2)CC2(CCC2)O1 C1(C(N(CC(CNC(C=C(C)C(C)C)=O)C)C)=O)CC2C=CC1CCC2 C12(NC(=O)COC3CC3)CC1CN(C(=O)CCc1cncs1)C2 C1(NC(c2sccc2F)=O)CCN(C(=O)C(F)n2ccnc2)CC12CCC2 C1(NC(C=CC)=O)C(C)(C)C(NC(c2ccc(-c3nc(C)cs3)cc2)=O)C1(C)C N1(C(C=CC(=O)NC2CCOCC2)=O)CC(CC(=O)NOCC2CC2)C2(CC2)C1 C1(NC(CCCCOC)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 N1(C(CCc2cc(C)n(C)n2)=O)CCOCC(C)(CNC(=O)CC2(O)CCC2)C1 N1(C(Cc2ncc(C)[nH]2)=O)C2CCCC1CN(C(c1ccc(N)cc1Br)=O)C2 Cc1ncc(NC(=O)COCCNC(c2ncccc2O)=O)c(C)c1C CC1CC(C(=O)N(C2CCN(C(C3CCC3)=O)CC2)Cc2ccccc2)C1(C)C C1(C(=O)NCC)CCN(C(c2ccncc2F)C(=O)NCCCF)CC1 c1(CNC2CCCC(COC)C2)c(C)n(C)c2ccccc12 Cc1cccc2c1CCOC2C(=O)NCC(CNC(=O)C1CC1)C(F)(F)F c1(OC)cnc(F)cc1C(=O)NC1CS(=O)(=O)CC1NC(=O)C(=O)N(C)C c1(C(=O)NCCC2(C(F)(F)F)CC2)ccccc1C(F)(F)C(F)(F)F C#CC1(O)CCCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)C1 C(=O)(C(C)(C)CC(F)F)NCCC1(C)CCN(C(c2scc(C)c2C)=O)C1 c1(OC)cc(F)ccc1CN1CC=CC1C(=O)Nc1ccc(C(C)(F)F)cc1 C1(NC(C(N(C(=O)CC2OCCCO2)C)C2CC2)=O)COC2(CCC2)C1 C1(CNC(=O)NC2(C#C)CCOC2)CCC2C(CCN2C)C1 c1(N2CCC(C(=O)OC(C)(C)C)(COC)C2)nccc2ccc(N)cc12 N1(C(C(C(C)C2CCCCC2)O)=O)CC2(C1)CN(C(=O)C=CCn1cncn1)C2 O(NC(=O)C(C1CN(C(=O)C(F)F)C1)OC)CC#C c1(C(N2CCC(CC(C)NC(C(CC)(C)C)=O)CC2)=O)ccc(F)c(F)c1C N1(C(c2c(C)[nH]cc2)=O)CC(CNC(c2cc(=O)cc[nH]2)=O)CC(C)(C)C1 CC(C)(CC(=O)NCC1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(F)(F)C1)C1CC1 N1(C(c2c(CC)c[nH]c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(O)C1 C1(C(=O)NCCCCNC(C(CC)n2cncn2)=O)(CO)CCCCC1 N1(C(c2ccn(CC)c2C)=O)CC2(CNC(C3(CC)CCCC3)=O)CCC1CC2 C(=O)(Nn1cnnc1C)C1N(C)CCN(C(C(C(C)C)OC)=O)C1 N1(C(C2(CCOC)CCC2)=O)CC(C2(NC(=O)CCCc3ccc(C)s3)CC2)C1 C1(N(C(CN(CCC#C)C)=O)CCO)CCN(C(=O)C(C)C=C=C)CC1 S(=O)(=O)(c1c[nH]c(=NCC(C)C(C)(F)F)cc1C)NC(C(CC)C)CO C1(NC(c2n(C)cnc2)=O)CC(CNC(c2cc(O)ncn2)=O)C12CCC2 Cc1ccnnc1C(=O)NC1CN(C(c2cc[nH]n2)=O)CC1CC(C)(C)C C12(CNC(CCC=C)=O)CC1CN(C(=O)C(C1CCOCC1)OC)C2 c1(OCC=C)cc(Cl)ccc1C(=O)NCC(C)N(C)C(c1cncs1)=O c1(CCC(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)ccc(CO)cc1 C1(C(=O)NCCC(C)NC(C2CS(=O)(=O)C2)=O)CCS(=O)(=O)C(C)C1 c1(C(N2CCC(CCNC(c3ccnc(S)c3)=O)C2)=O)ccc2cnoc2c1 N1(C(C2OCC(C)(C)C2)=O)CC(C(N2CCC(CO)C(O)C2)=O)C(C)(C)C1 CC(O)C(C)C(=O)N1CC(CCCCNC(=O)C(=Cc2cccnc2)F)C1 CCCCC(C)C(=O)N(C)CC1CN(C(c2cccc(F)n2)=O)CCO1 CC1=C(C(=O)NC(C(=O)NCC2CCCCN2C(C)C)C2CCC2)CC1 N(S(=O)(=O)N(C)C)CC(N1C(C2CCN(C(CCN(C)CCO)=O)C2)CCC1)=O C(=O)(C(C)(Cc1ccccc1)C(C)C)NCC(CNC(CN(C1CC1)CC)=O)O C(CCC(=O)NCC(C)C(=O)NC1CC1)N(C(C(OC)OC)=O)C c1(C(=O)NCC(C)OC)ccc2c(n1)CN(C(=O)C1=NOC(C)C1)CC2 c1(C(=O)NC(CNC(CC2C(C)(C)C2)=O)CO)cc(Cl)cc(Cl)c1O C1(N(C(C(c2cnn(C)c2)NC(CC=CC)=O)=O)CCO)CCCCC1 C1(NC(CSCCC)=O)CCC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCCC(C2CN(C(=O)COCP(C)(C)=O)C2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC(C)(CO)C1.c12ccoc1C(=O)NC2 CC1CCN(C(=O)C#CC(C)(C)C)CC1CNC(c1cnn2c1CCC2)=O C(C(CC(C)C)NC(c1cnnc(O)c1)=O)NC(Cc1cnc(C)[nH]1)=O C(=O)(C(C)(C1(C)CC1)OC)NC(C(=O)NCCC(=O)OCC)C1CCCO1 c1(CC)ccc(C(=O)NCC(C)(F)CNC(c2n[nH]c(C3CC3)n2)=O)o1 S(=O)(=O)(c1ccc(N2CCC(CC3CC3)C2)c(Cl)c1)NC(CSC)C c1(OC)cc(C(=O)N(CC(C)O)CCNC(c2cc(C(C)C)nn2C)=O)ncn1 c1(C(N2CCOCC(NC(CCC(=C)C)=O)C2)=O)cc(O)cc([N+](=O)[O-])c1 CS(=O)(=O)CCC(=O)N1CCC(OCCCNC(C2OCC3CCCC23)=O)CC1 c1(CC(=O)N(CCCCCCNC(=O)Cn2nnc(=N)[nH]2)C)ncn2c1CCC2 c1(C(=O)NC2CN(C(c3c[nH]c(=NCC)s3)=O)CC(F)C2)cccc2c1CCC2 C12(NC(=O)CCc3cccnc3Cl)CCC1CN(C(c1cn3ccnc3s1)=O)C2 N1(C(C(C)CCN(C)C)=O)CCC(c2cn(-n3cnccc3=O)nn2)CC1C N1(C(C2(C)CC2c2ccccc2)=O)CCCCCC(NC(C2CC(O)C2)=O)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(O)CCN1C(C1CCCO1)=O N1(C(c2c[nH]c(=NCC)s2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)CCC(O)C1 C=CC1(C(N2CCCC2C2(C(=O)NCC(O)CN(C)C)CC2)=O)CCOCC1 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)CC1(F)F N1(C(C(C)N(C)C)=O)CCC(NC(c2ccccc2F)=O)C1c1ccccc1 C1(N(C)C)CCC(c2cn(C3CCCCC3NC(c3nc(I)cs3)=O)nn2)CC1 Cc1ccc(N)c(C)c1C(=O)NC1CN(C(c2cc3c(s2)CCCC3)=O)CC1C c1(C(N(CCCN(C)Cc2c(OC)ncc(Br)c2)C)=O)ccnc2ccccc12 c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(=O)CN(C)C)c1OC C(C(C)(C)CCNC(=O)Cc1ccco1)NC(C(C)OCCC#C)=O Cc1c(CNC(=O)CC23CCC2CN(C(c2cc(Cl)no2)=O)C3)cccc1F Cc1ccc(C(CO)NC(=O)NC(C2CCC3(CCC3)O2)C2CC2)c(F)c1 c1(C(=O)NCC(CNC(=O)C(O)C(C)C)OC)cncc(F)c1C(F)(F)F c1(NC2CN(C(Cc3nnc(C)o3)=O)CC2O)ncnc2ccccc12 N1(C(CC(COC)C)=O)CCC(N(C(=O)CCc2cccc(O)n2)C)C2(CC2)C1 c1(C(N2CC(CCNC(C(CC)=CC)=O)OC(C)C2)=O)cc(CC)c(=O)n(C)c1 N1(C(C=C(C)C(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)CCc2nncn2C1 CCCCC(O)C(=O)NCC(C)(Cn1cccn1)NC(=O)CCC(=O)N(C)C CCC(C)(CCO)NC(=O)C(CO)NC(=O)CC1CC(F)(F)C1 n1(C(COC)C)nc(-c2ccncc2)nc1-c1ccnn1Cc1ccccc1 c1(CC(C)C)n[nH]c(=NC(CNC(c2ccc(F)nc2)=O)C(C)C)s1 N#CC1CN(Cc2ccc(SC(F)(F)F)cc2)CCN1C(c1cc([N+](=O)[O-])cs1)=O c1(CCC)c(NCC2CCCC3CC23)nnn1CC c1(C(N2CCC(CC(=O)NC3CCC(C#N)CC3)C2)=O)c(O)cccc1[N+](=O)[O-] C1(NC(CC2(C)CCN(C(CC3CCN(C)C3=O)=O)C2)=O)CCn2cnnc2C1 C12(C(=O)NCCC3(C)CCN3)CCOCC1C2(F)F C1(C(=O)NCCN2CCN(C(C(C(=C)C)(C)C)=O)CC2)C2CCCCCCC12 c1(C(N2CCC(COC)(NC(=O)C=CSC)C2)=O)c(C)nn(C)c1F C1(COC)(OC)CCCCC1.C1CCCNC(=O)C(C2CCCO2)OCC(=O)N1 Cc1cncc(C(=O)NC(CNC(=O)Cc2cc(C)on2)C2CCC2)c1 C(=O)(C(C(=O)N1CCC(CN(C(=O)C(F)CC2CCOC2)C)CC1)OC)OC C1(C(N(CC(=O)NCCCN(C)C)CC)=O)CCC(=O)C1 n1(CC)nc(C(=O)NCC(C)(O)CNC(=O)C(C(C)C)n2ccnc2)c(C)n1 N1(C(C(C(=O)OC)N)=O)Cc2ccccc2C(C)(C)C1.CCCC1=CCCCC1 C1(C(=O)NC2C(NC(c3c(C)nsc3)=O)COC2)C2CCCCC12 C(C(C(=O)N(C)CCN(C)C)NC(c1nccs1)=O)OC(C)C CCC(CN=c1cc(NC(c2ccoc2)C)nc[nH]1)N1CCCC1 Cc1ccc(OCC(N2CCC(c3c(Cl)cccc3Cl)C2)=O)c(F)c1C N#CC1(NCC(O)CN2CCOCC2)CCOC1 CC1CN(C(C23C(=O)C4CC2C3C4)=O)CCC1CNC(=O)CC1NC(=O)NC1=O C12CC(C)CN1C2=O.C1(CC)CCC(NC(=O)CC2CCSC2)CC1 C(=O)(C(C)C(C)(F)F)NC(C)CN(C(=O)Cc1ccnc(C(F)(F)F)c1)C O=C(N=c1cc(Cl)cn[nH]1)C1CSCCN1C(c1cccc2[nH]ncc12)=O CC1CCC(CNC(=O)CC=CC(C)(C)C)CN1C(=O)C(=O)C(C)(C)C c1(C(=O)OCc2cc(C(C)C)nn2C)ccc2c(cnn2C(F)F)c1 c1(COC)nc(N2CCCC(CNC(=O)CC3CC(F)C3)CC2)cc(C)n1 O=S(=O)(c1c[nH]ccc1=NCc1c(F)cccc1Cl)N1CCC(C23CC(C2)C3)CC1 CN1CC(C(=O)NCC2CCN(C(C3CCNC3=O)=O)C2)C(C(F)(F)F)C1 c1(C(N2CCN(CC(O)C3CC3)CC2)C(=O)NCCC#N)c[nH]c2ncccc12 Cc1cc(C(=O)NC2CCC(NC(=O)CC3CC=CCN3C)C2)c(C)n1C(C)C Cc1cc(C(=O)NC2CCC(C)N(C(c3oc(Br)nc3C)=O)C2)cc(O)c1 c1(C(C)C)ccc(C(=O)N(CCCN(C)C(C2(c3ccccc3)CC2C)=O)C)s1 C(=O)(C(N)CCC1CCCCC1)NC(CC(=O)NC)C C1(N(C(Cn2c(C)nnn2)=O)C)CN(C(C2CC2Br)=O)CC1(C)C Cc1ccc(C(=O)Nc2ccc(NC(c3cccc(=O)n3C)=O)cc2F)c(C)c1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2csc(C)c2)=O)C(C(C)C)C1 C1(C)(NC(C2CCN(C(CCCCCOC)=O)C2)=O)CN2CCC1CC2 C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC(COC)CO)C1(C)C CC1(C)Cc2cc(C(=O)NCc3ccc(N4CCCC4)nc3)ccc2O1 c1(C(N2C(C)CCN(C(c3cc(C)nn3C)=O)CC2)=O)nn2c(c1C)OCCC2 n1(CCC(=O)N(C(c2ccc(C)c(F)c2)C(=O)OC)C2CC2)cc(Br)ccc1=O c1(C(N2CCN(C(C(CCC#C)O)=O)CC2C2CC2)=O)occ2c1CCCC2 C=C(C)CCN=c1cc[nH]cc1S(=O)(=O)N1CC(C)SC(C)C1 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)OC)c(F)cncc1Cl c1(C(=O)NC(c2ccccc2)C(C)C)cccnc1OC(=O)C1CC1 N(C1CCc2ccc(Cl)cc21)C(C1CC2(C1)CN(C(=O)CCN1CCCC1)C2)=O Cc1nnc(CNC(=O)CN(C2CC(C#N)C2)C(=O)C(F)C2CCCC2)o1 c1(C2(C)C(C(=O)NC3C(C(C)(C)C)CCC3)C2)ccc(F)cc1F CC1=CCC(C(N2CC3CC2(CNC(=O)C(O)C(C)C)C3)=O)CC1 c1(C(N2C(C(N3CCN(COC)C(=O)C3)=O)CC(=C)C2)=O)cccc2nonc12 CC1CN(C(=O)CC2CC2(C)C)CCCN1C(=O)Cn1cc(S(C)(=O)=O)cn1 c1(C(=O)NCc2nnc(COC)o2)cccc(S(=O)(=O)N2CCCC2C(=O)O)c1 C1(CNC(Cc2cc(C)no2)=O)CCCCN1C(c1ccnnc1)=O CCCC(C)CC(=O)N1CCCCC1CN(C(=O)C(=O)C(C)(C)C)C CCC(C)(O)C(=O)NCCN1CCN(C(=O)Cc2ccc(Cl)s2)CC1 CCS(=O)(=O)c1ccccc1C(=O)NC1CC2CCC1N2C(C1CCN(C)C1)=O N1(C(CC2C(C)CCC2)=O)CCC2CN(C(c3csnc3Cl)=O)C2C1 C1(CNC(C(C)CN(C)C)=O)CC(O)CN1C(=O)CNC(=O)CCCCO c1(C(N2CCC3(C(=O)Nc4cc(C)on4)C(C2)C3)=O)cc(C#N)ccc1Cl C(CC(C(=O)NCCc1ncn(C)n1)NC(=O)C=C(C1CC1)C1CC1)OC CCCC(C)CC(=O)NCC(C)CNC(=O)C(F)CC1CCCC1 n1(CC)cc(Cl)c(C(=O)NC(CO)C(C)NC(=O)CCCOC(C)=O)n1 N1(C(c2cnn(CCCl)c2)C(=O)NCCOCC)CC(C)CCC1CCO C1(OC)CN(C(=O)C(=O)Nc2ccccc2CC2CCOC2)CC2CC12 N1(C(CN(C(=O)OC)C)=O)CC2(CNC(=O)Cc3ccc(Cl)cc3)CC(F)(C1)C2 c1(C(=O)NC2CC(n3cc(-c4n(CC)ncc4)nn3)C2)cc(Cl)c(Cl)c(Cl)c1 C(=O)(C(C)CC(F)(F)F)N1CCN(C2CCN(C(CC(C)C)=O)C2)CC1 C1(C(=O)NC23COC(CNC(C4CC=CC4)=O)(C2)C3)(OC)CS(=O)(=O)C1 C1(CC(N2C(CNC(C3(C4CC4)CC3)=O)CC(OC)C2)=O)SC2=NCCN2C1=O N1(C(CC)=O)CCC2(CC1)CC2NC(c1ccnc(C2CCCC2)n1)=O C1(C(=O)N(C(C)C(=O)NC(C(=O)NCC2CC2)C)C2CC2)(COC)CCCCO1 c1(C(=O)NCCN(C(=O)CC2(C#N)CC2)CC)cccc(C2CC2(F)F)c1 C(=O)(C(Cc1cccnn1)NC(=O)NCCOC1CCOC1)OCC N1(C(C=CC)=O)CCN(C(=O)C(C)NC=O)CC1CS(C)(=O)=O O=C(C1=NOCC1)N1CCC(NC(C23CCC(C2)C3)=O)C1C(C)(C)C c1(N(C)C)cc(-c2ccc(CN3CCCC(F)C3)s2)ncn1 N1(C(C(C)OC2CCOC2)=O)CC=C(CC(=O)N2CC3CC(C2)C3(C)C)CC1 c1(C(=O)NCC2(F)CC(CNC(CN(CC(C)(C)C)CC)=O)C2)nnc(S)n1C CN1CCC2CCC(C1)N2C(c1coc(CNC(=O)CNC(=O)CN(C)C)n1)=O c1(C(=O)NC2CCCN(C(C(C)(O)C3CC3)=O)C2)c(F)cc(N)cc1F C1(NC(CC(CC)CC)=O)CCN(C(c2cnc(C)c(N)c2)=O)CCC1CO c1(C2N(c3n(Cc4c(C)nco4)nnn3)CC2)ccc(F)cc1.N12CCCC1C2 N1(C(C2(CC#C)CCC2)=O)CC2C(NC(=O)C(C#N)(CC)CC)CS(=O)(=O)C2C1 N1(c2c(C)c(N3CCN(C)CC3CO)ncn2)CCNC(=O)CCCC1 N1(C(C=CCCC)=O)CCCC(NC(=O)CC2CCCC2)C(F)C1 c1(C(N2CCN(C(=O)C=CCl)CC2)C(=O)NCCOCC)ccnc(Cl)c1F C#CCCCCCCC(=O)N1CCCCC1CNC(C1CCC2CC12)=O C(C)(C)(CCCC(=O)NCC1(O)CC=CC1)NC(C(C)C1CCCO1)=O C1(CNC(C(CC)N2CCCC2=O)=O)CN(C(C23COCC(C2)C3)=O)CC1N(C)C Cc1cc(C(=O)NCC2CCC2NC(C2COCCO2)=O)c(N)c(C)c1 CSC=CC(=O)NCCCN(C(C1COCC1c1ccccc1)=O)C1CC1 Clc1ccc2c(c1)C(NCc1cn(C3CCCC3)nn1)CCCO2 CN1CCC=C(CNC(=O)CC2CC(NC(=O)Cc3ccc(O)nc3)C2(C)C)C1 N1(CC#CC)CCN(C(=O)C(c2ccnn2C)NC(=O)CN2CCCCC2=O)CC1 Cc1ccc2c(C)c(C(=O)NC3Cc4cccnc4C3)[nH]c2c1 CCCCCC(C)(C)C(=O)NCc1cc(C)c(C(=O)NCCn2cnnc2C)o1 C1(C(=O)NCC2CC3CCC3C2)(CNC(=O)Cc2cc[nH]n2)CC12CCC2 C(=O)(CCC(C)(C)C)N1CC(C)C(NC(=O)CSCC(F)(F)F)C1 N1(C(c2cc(C(N)=O)c[nH]2)=O)CCC2CC12C(=O)NCc1ccncc1Cl Cc1ncncc1C(=O)N(CCCN(C(=O)C(CO)c1ccccc1)C)C c1(C(C2CC=CCC2)NC2(CC=C)COC2)nnnn1-c1ccccc1 c1(C(=O)NC(CC(C)Nc2nccc(SC)n2)C)ccc2cnsc2c1 CCC(CC(=O)NC(C)CN(C(=O)CN1CCCCC1=O)C)CC(F)(F)F N1(C(C2(CCF)CN(C(=O)CN(C)C)C2)=O)CCN(C2CCC2)CC1.CS CC(C)CC(C)(C)C(=O)N(CC(=O)NCCC1CCN(C)C1=O)C N1(C(C=CCC)=O)CCCN(C(=O)CC2CC2C2CC2)CC1C Clc1cccc(CCC2CCCN2Cc2cnccn2)c1 CCCC(C(=O)N1CCC(CNC(=O)Cc2ccc(CO)cc2)(OC)C1)C(C)C C1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)C2CC2)CCC(NC(C)=O)CC1 N1(C(=O)C=C2CCCC2)CCC(CCNC(C2CN(C3CCOCC3)C2)=O)CC1 C1(CCOC)(NC(c2cn(CC)nc2)=O)CCN(C(=O)Cc2cnns2)C1 CCCCC(CNC(c1ccn(-c2ccncc2)n1)=O)NC(=O)C(C(C)C)SC c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cc(F)c(Cl)nc1Cl c1(C(N(CCCNC(CCc2ncc(C)[nH]2)=O)C)=O)ccccc1OCC(C)C CC1CC(NC(=O)C(C)(C)N2CCCCC2)CCN1C(=O)CSCc1ncc[nH]1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C(=O)NCC2(C3CC3)CC2)CC1(C)C CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C1CC1)NC(=O)CCn1cncn1 c1(C(N2CC(C)CC(NC(CCOCC)=O)C2)=O)cc2c(s1)CCC2=O C1(C(=O)NCCCc2cn(CCCSCC(C)C)nn2)CCc2cnn(C)c2C1 c1(CCCCN(C)C)nc(-c2ccnc(N(C)C)c2)nn1CCCCO c1(C(=O)OC)cc(N2CCCC2CCCNC(C2CC23CCCC3)=O)ncn1 c1(C(=O)NCC(CC)NC(C2CC2C)=O)nn(C)nc1Br Cc1cc(C(=O)NCC2CCCN2C(=O)Cc2cccc(Br)c2)c(C)cn1 Cc1cc(Br)sc1C(N1CCC(NC(=O)C=CC(=O)NC(C)C)C1)=O C(=O)(CC1=CCOCC1)NC(CCCNC(c1c(C)coc1C1CC1)=O)C N1(C(Cn2cc(COCC(OCC)OCC)nn2)=O)CCCN2CCCC2C1 CC(C)CC(C)CC(=O)N1CCCCC1C1(NC(=O)C(C)(C)C2CCC2)CC1 c1(C(N2CC(NC(=O)COCC3CCCOC3)C(O)C2)=O)cc2c(s1)CCSC2 N1(C(=O)COC2CCCNCC2)CCC12CCCOC2 c1(C(=O)NC2(COC)CCN(C(=O)C(C)OCCC(C)C)C2)cnc(O)cc1C C1(C(=O)NC(C)C(C)NC(c2cccc(CC3CCCC3)c2)=O)C2CC3C(C2)C13 C1(CNC(c2sc(CCC)c(CC)c2)=O)CCN(C(=O)C(C#N)C2CC2)C12CC2 Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)CC2CC(F)C2)c2nccn2c1 C1(NC(CC2ON=C(CC)C2)=O)CC(NC(=O)Cc2[nH]cnc2C)C12CCC2 C12(C(N3CC(C(=O)NCCC4CCCN(C)C4)(SC)C3)=O)C(=O)C3CC1C2C3 CCC(CC)(CCNC(c1cccc(CO)n1)=O)NC(C1CCC(C)(CC)O1)=O Cc1ccc(Br)c(S(=O)(=O)C(=O)NCCNC(Cc2c(F)cccc2F)CO)c1 N1(C(C(C2CC2)NC(CCOCCCOC)=O)=O)CC2CCC(C1)C2C#N CC1CC(C(=O)NCc2cccc(Cl)c2)CN(C(=O)C(O)Cc2ccc(O)cc2)C1 C=CCC(CC(=O)Nc1cc(CC)ccc1C)NC(=O)C(COC)OC C(=O)(CN=c1ccc(Cl)n[nH]1)NC(C)CCCCNC(C12CC(C1)C(C)(C)O2)=O c1(C(=O)NC(CNC(C2C(=C)C2)=O)C2CC2)cc(C(F)(F)F)[nH]c1C c1(CNC(CC)=O)ccc2c(c1)CCCC2NC(C1CCc2nc[nH]c2C1)=O CCC(C)CC(=O)C(=O)N1CCC(CNC(C2CCCS(=O)(=O)C2)=O)C(O)C1 c1(C(=O)OC)cc(C(C)NC2(CNC(c3ccncc3)=O)CC2)nn1C c1(C(=O)NCC2CCCC(NC(c3ccc(SC)o3)=O)C2)c(Cl)cncc1Cl CC(O)CCCCCC(=O)NCC1CC2(CO1)CN(C(=O)COC(F)F)C2 C12(C(=O)NCCOC(C)=O)CC(CN(C(=O)CC3CCCCN3C)C1)C2 C1(C(=O)NCCCCC=C)(NC(=O)CSC)CCC(C)(C)C1 c1(C(=O)NC2(C)CC(NC(C(C(C)O)(F)F)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC(C)O1)NCCCCCC#C O=C(CCC(CF)CF)NC1(C(=O)NCC2CC23CCOC3)CC(O)C1 C1(CCC)CC(C(=O)NCc2cc(C3CCN(C(C)C)CC3)no2)CCO1 Fc1ccc(C(Cc2ccc(Cl)cc2)NC2(C(CNC(F)(F)F)(F)F)CCCC2)cc1 CC12CN(C(C3CCO3)=O)CC1(C)CN(C(c1ccc3oc(O)nc3n1)=O)C2 CS(=O)(=O)c1ccsc1C(=O)OCC1C[Si]2(CCCC2)CN1 C(=O)(CC(C)CC(=O)N1CCC(C(N2CCc3n[nH]cc3C2)=O)O1)OC c1(C(=O)NCC(C)(O)CNC(C2CC(F)C2)=O)ccc2c(c1)NC(=O)CCS2 O=C1COc2ccc(-c3cscc3CCCNCc3ccc(Cl)cc3Br)cc2N1 C(=O)(CCCC(=O)NC(C)(CSC)C(=O)NC(c1ncc[nH]1)CO)OC N1(C(CNC(C(CC)CC)=O)=O)CCN(C(=O)C2=COCCO2)C(COC)C1 c1(CC)ccc(C(=O)NCC(O)CNC(=O)CNC(=O)COc2ccccc2)s1 c1(OC)ccc(OCCC(=O)NC2(CN=c3[nH]nco3)CCCC2)cc1 c1(CNC(C2N(CC#C)CCC2)=O)ccccc1CNC(=O)CCCc1ccsc1 C1(C#N)(C(=O)NCCN(C(c2n(CCC)nc(C)c2)=O)CC)CC12CCCC2 Cc1cc(Br)ccc1-n1cc(C2CC(NC(=O)CC34CCC(C)(C3)OC4)C2)nn1 Cc1cccc(CCNC(c2ccn(CCNC(=O)Cn3nccc3C)c2)=O)n1 c1(OC)cccc(C(=O)NCC2CC2NC(=O)CCc2cnco2)c1O C1(O)(CCNC(=O)CC2CCOC2=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1CC2(CC(C(=O)NC3(CCNC(=O)CCCF)CCOCC3)C2)C1 CC1CC=C(C(=O)NC2CC=C(C(=O)N(CC(C)C(F)(F)F)C)C2)CC1 c1(OC)cccc(Cl)c1CC(=O)NC1CCC1NC(C1(C)CCC(OC)CC1)=O c1(CCC)ccc(C(=O)NCC2CC(CNC(=O)C=CCO)CO2)[nH]1 C(=O)(C#CC1CCOCC1)N1CC2=C(CN(C(C3C(C)NC(=O)CC3)=O)C2)C1 C1(CNC(c2ncc(NCC)nc2)=O)C(C)CCCN1C(C1(CF)CCC1)=O C(=O)(CC(C)C(=O)NCCNC(=O)C(C)(C)SC1CC1)OCC c1(C(=O)NC2(C)CN(C(c3cc(C(F)(F)F)ns3)=O)C2)cnc2ccccn12 C1(NC(C(CC)C)=O)CCN(C(c2nc(-c3ccccc3C)oc2C)=O)C1C N1(C(C2(C)CC2Br)=O)CCC2(NC(c3cncc(-n4cccn4)n3)=O)CCCC12 C12(NC(C=Cc3c(C)ccs3)=O)CCN(C(=O)C(c3ccccc3)F)CC1C2 c1(C(C)OC)ncc(C(=O)NC(C)(C)CNC(C2CC3(C2)CN(C)C3)=O)c(C)n1 Nc1ccc(F)c(F)c1C(N1CCN(C(C2CCCS2)=O)C(C2CC2)C1)=O N1(C(c2cnc(C)o2)=O)CCC2(CC2)CC1C(=O)Nc1conc1C N1(C(=O)OC(C)(C)C)CCC2(CCC(C(N3CCOCC34CC4)=O)CC2)CC1 N1(C(C(CC)O)=O)CCN(C(C2CCCC(CF)C2)=O)C(c2ncc[nH]2)C1 CN1CCC(NC(=O)Cc2csc(S)n2)C12CCCN(C(C1CS(=O)(=O)C1)=O)C2 C(CC(C(C)C)NC(=O)CC1(C#N)CCC1)NC(C(CC)n1ccnc1)=O CON(CCC(=O)N1CCSC(C)(C)C1)C(=O)c1ccc2c(c1)CC2 N1(C(CC2CCC(=O)O2)=O)CC2CCC1C(CNC(c1snnc1C1CC1)=O)C2 C12(C(COC)NC(C3CC3C(F)(F)F)=O)C3C(=O)C4C5CC(C14)C2C35 C1(NC(C(C)(C)O)=O)CN(c2nccc(-c3ccccc3F)n2)CC1(F)F C1(NC(C2(CC)CN(C(c3cc4ccccn4n3)=O)C2)=O)CN(C)CCN(C)C1 C(CC(C(C)(C)C)NC(C1COC1)=O)N(C(=O)C=Cc1cnc(C(C)(C)C)s1)C N1(C(C2(C(F)F)CC(=C)C2)=O)CC(NC(c2cc(F)ccc2O)=O)CC(O)C1 c1(C(N2CCC(O)(CNC(CN(C)C)=O)C2)=O)n[nH]c2c1COC2 C1(C(N2CCC(NC(CCC=C=C)=O)(CO)C2)=O)CCC2(CC1)CC2 Cc1ncnc(C(=O)NCC(C2CCN(C(C3C(C)(C)C3(F)F)=O)CC2)O)c1C CC(C)(CC(=O)N1CCCC(C)(NC(=O)COCCO)C1)CC(F)F N1(C(CC(CNC(c2nn(CC)c(C)c2)=O)(C)C)=O)CCC2CCN(C)CC12 CCC(C)CC(C(=O)NCCC(C)(C)COC)NC(=O)C1=C(Cl)CCC1 N1(C(c2c(CC)ncs2)=O)CCC12CN(Cc1c(Br)cnn1C)C2 CCC(CC(=O)N1CC(NC(c2csc(C(C)=O)c2)=O)C2(CC2)C1)C(C)(C)C C1(NC(COCCC)=O)CCS(=O)(=O)C12CN(C(=O)C(=C1CCCCC1)F)C2 Cc1ncc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CCC(C)(C)C)C1 c1(C(=O)NC2C(CNC(CC(C)F)=O)CC2)nc2ccccc2[nH]1 N1(C(CCN(C(CC)CC)C)=O)CC(NC(=O)CCNC(C)=O)C(N=[N+]=[N-])C1 c1(CNC(Cc2cc(CC)no2)=O)nc(C(=O)NCc2cncc(Cl)c2)c(C)o1 C(CC(C)C)(C(=O)NCC(F)CNC(c1cccc(F)c1Cl)=O)NC(C)=O C(C)(C)(C(C)NC(c1cn(C2CCCC2)nn1)=O)NC(C(C)O)=O c1(C(=O)NC2CC(NC(CC3CC(SC)C3)=O)C2)ccc(NC2COC2)cc1 c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)C(C2CCC(=O)N2)C)o1 C1(NC2(c3n(CC(=C)C)nnn3)COC2)CC(C(=O)OC)C12CCC2 C1(Cc2cn(CCC=C)nn2)CN(C(=O)C(C)CC2CCC2)CCO1 c1(OC)ccc(OC)c(C(N2CCC(CCNC(=O)CN3CC=CC3)C2)=O)c1N c1(C(=O)NC2CCCC(CC(=O)NCc3ccnc(F)c3)C2)c(O)cccc1F C(CN=c1[nH]cnc2c(Br)cccc12)OCCNC(C1(CC#C)CCCCO1)=O c1(N2C(C)C(NC(c3cc(Cl)c[nH]3)=O)CCC2)nc2c(cc1C#N)C(=O)CCC2 Cc1cc(C(N2CCC2C(N2CCC(Oc3ccccc3)CC2)=O)=O)cc(Br)c1 N1(C(C(C)NC(N)=O)=O)CCC2(CCN(CCNc3cn4c(n3)CCCC4)C2)C1 N(C1CCCn2ccnc21)C(c1c(CNC(C(CO)OC)=O)nccc1)=O CC1CC(C(=O)O)CN(Cc2ccc(OC(CO)C3(C)CC3)cc2)C1 c1(-c2nc(C)c(NCc3ncccc3C(F)(F)F)s2)c(F)cc(F)c(O)c1F c1(CNC(c2c(OC)csc2)=O)ccnc(Br)c1 C1(CNC(c2ccc[nH]2)=O)C2CN(C(c3ccc(Br)o3)=O)CC12 C(=O)(CC(C)(C)CC(=O)OC)N(C(CNC(c1ccc(C#C)cc1F)=O)C)C CC(F)(F)CCC(=O)NC1CS(=O)(=O)CC1NC(=O)CNC(C1CCC1)=O c1(OCC)ncc(C(=O)NCC2CC(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 Cc1cc(C(=O)NCC(C)NC(C2CC2c2ccccc2)=O)nnc1C C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)C(C)(C)C(F)(F)F)C1)OC CC1(CNC(=O)CCN(CCO)C(C2CCCCC2O)=O)CC2(CCC2)C1 CC(C)C(C(=O)NCC(C)(O)CNC(c1cncc(Cl)c1)=O)NC(=O)C(F)(F)F CCCCC(O)C(=O)NCC1CCN(C(=O)Cc2ccsc2)C1C C1(NC(=O)CCC2CC(F)(F)C2)CC2CC(C1)N(C(C13CCCC(C1)OC3)=O)C2 CN1CCN(c2cccc(C(=O)OCC3(CNC4CC4)CC3)n2)CC1 Cc1c(C(N2CCCC(C)(CNC(=O)C(C)OC3CCCC3)C2)=O)nn(C)c1N N1(C(c2ccc(C)n2C)=O)CCCC1C1CCCN1C(=O)CNC(N)=O c1(C(=O)NCC(CC)NC(c2cnc(C(F)F)s2)=O)coc(Cl)c1 Cc1noc(Cl)c1CCC(=O)NC(C)CC1CN(C(c2cnn(C(C)C)c2)=O)C1 C(C1=CCCN(C(=O)CC2CCCC3CC23)C1)N(C(C1CC(OC)C1)=O)C1CC1 c1(NS(CC)(=O)=O)ccc(-c2ccnc(CC(=O)NCC3CCSCC3)c2)cc1 Cn1cc(Cl)cc1C(=O)NCC(N1CCN(C(c2csc(C(F)F)c2)=O)CC1)=O c1(-c2cccc(C#C)c2)ccc2[nH]cc(C(=O)Nc3ccc(OC)c(F)c3)c2c1 Cc1cc(C(=O)NC(C)CC2CN(C(=O)CCN3CCC(F)C3)C2)cn(C)c1=O c1(C(=O)NCCC(C(=O)N(CCCCC)CCO)O)ccc2cc[nH]c2c1 CC1CN2CCN1CC2C(=O)NCC(C)(O)CNC(c1cnn(C)n1)=O C1(NC(Cc2ccc(C)o2)=O)CCCC(NC(c2cnn(CCF)c2)=O)C1 c1(C(=O)NC2C(NC(=O)Cc3cscn3)CCCC2)cc2cccnn2c1 CCC1=C(C(=O)NC(CC(=O)NCC(c2ccsc2)O)C(F)(F)F)CCCO1 N1(C(C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)CCC1CCCCCC1 C1(C(=O)NC2CN(C(=O)C(C)(C)COC(C)C)CC2C)(OC)CCC(F)(F)CC1 Cc1cnn(C)c1NC(C1CCCC(C(=O)NCc2nc(C(=O)N(C)C)no2)C1)=O C1(CCNC(C(C2CCOC2)OCC)=O)CCN(C(=O)Cc2ncc(C)s2)CC1 N1(C(c2cc(CC)no2)=O)CC(CNC(=O)C=NOC)C(F)(F)C1 CC1CC(CNC(c2nn(C)cc2Br)=O)CN1C(c1sccc1F)=O c1(N(C(CCNC(c2cc(OCC)ncc2)=O)C)C)nc2c(cc1C#N)CCC2 Cc1nc(O)[nH]c1C(=O)NCCCCNC(c1ccc(C2CC2)cn1)=O c1(C(N2CC3C(NC)C3C2)=O)cccnc1OC(C)C(F)(F)F C1(C(=O)NCCOCCCNC(C2CC(C)(C(C)(C)C)C2)=O)CC2CC(=O)C1O2 CC1CCN(C(=O)Cc2cccnc2Cl)CCN1C(=O)C(O)Cn1cncn1 c1(C(C)C(=O)N(C2CC2)Cc2nc(C(F)(F)F)n[nH]2)cccc(C#N)c1 CC1CN(C(C2(C(=O)NCC3CC3)CCO2)=O)CCN1C(=O)CC1CC12CC2 C=CC1OCCC1C(N1CCC1CC(=O)NC(CC)CCOC)=O C(C(C)(C)CC(=O)NC1CCC(C)(CNC(=O)C2=NOCC2)C1)N(C)C C12(NC(=O)Cc3cccc(C4CC4)c3)CCN(C(c3cocn3)=O)CC1C2 c1(C(=O)NC2CCCN(C(C3CC(=O)NC3)=O)C2)ccnc(O)c1F c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CCC2)=O)cc(N)cc(O)n1 c1(C(C)C)cc(C(=O)NC2CCC(C)N(C(=O)C(=O)NC3CCCC3)C2)ccc1O CCC(CC(=O)NC(CNC(C1NC(=O)CC1C)=O)CC)C(C)C C1(C2CCN(C(c3cn(C(F)(F)CO)nn3)=O)CC2)(NC(CC(CC)O)=O)CC1 C1(C#N)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)O)CC2(CC2)C1 C1(NC(C(C)NC(CC)(C)C)=O)CCN(C(c2cncc(Cl)c2)=O)C1C(C)C c1(COCC(N2C3CC(NC(CCCCC)=O)C(C3)C2)=O)ccc2c(c1)OCO2 CC(C)C(O)CC(=O)NCC(CNC(=O)CSCC(N)=O)CO c1(-c2n(CC)ccn2)ccc(F)cc1-c1cccc(C2(CO)CC2)c1F C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(C)CCC(NC(C(C=C=C)C)=O)CC1 N1(C(c2c(C)ccc(OC)c2)=O)CC2CCN(C(=O)C(C)n3cccn3)CC2C1 c1(C(N2CCN(C(=O)COCC3CC3)CC2CC2CC2)=O)ccc2occc2c1 C1(CC=C)(NC(C2CCCCN2CC)=O)CCN(C(=O)C(Br)=C(C)C)C1 C1(C)(CC)CC(NC(C2CC(O)C2)=O)CN1C(c1ccc(N(C)C)cc1)=O c1(CN(CC(C(C)C)O)C)ccncc1OCc1ccccc1 Cc1cc(Br)cc(C(N2CC(N(C)C(c3ncoc3C(C)C)=O)C2)=O)c1C c1(C(N2CCC(CC(N3CCCC(C(=O)OC)C3)=O)CC2)=O)c(I)ccnc1Cl CC1(C)CC(CNC(=O)CC2(O)CCOCC2)CN1C(C12CC(F)C1C2)=O C(CCC(F)(F)F)NC(C=C(C)CNC(C1(N(C)C)CCCC1C)=O)=O Cc1ccc(CC(=O)NC(C2CCN(C(=O)C(c3ccccc3)=O)C2)C)c(Cl)c1 Cc1ccc(F)c(O)c1C(=O)NCc1cn(-c2nc3ccccc3s2)nn1 CC(C)CCC(=O)NCC1CC1C1CC1.C12(CCC1)C(=O)N2C1CC1 C1(C(=O)NC2(CF)CCN(c3nc(CC)cc(CC)n3)C2)CC12CCOC(C)C2 CC1CN(CCCOC2CCCCO2)C=C1C#N C1(C(=O)Nc2c(-c3ncn(C)n3)cccc2)CCOCC12CCC2 n1(CC(C)N(C)C)ccc(=NC(=O)CC(Cl)S(C)(=O)=O)[nH]1 C1(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2)CCC(N(C)C)CC1 CCC(CC(=O)NCCc1ccsc1)N(C(=O)CC1CCCC2CC12)C N12CC(C)OC3(CCN(C3)CC(=O)N(C)CC1=O)C2.c1(NC(C)=O)ccccc1 C=C(F)C1(CC(=O)NCc2cc(C(=O)NCC3COCCO3)no2)CCC1 C1(C(=O)NCC2N(C(c3c(C)nc(C(C)C)o3)=O)CC(F)C2)CCCC(F)(F)C1 N1(C(CC(C)(C)SC)=O)CCOCC(NC(=O)C(O)c2cnc[nH]2)C1 c1(C(=O)NC2CCN(C(CC(CC)OC)=O)C2C)cc2c(Cl)cncc2o1 C1(CC(=O)NCC2(N3CCCC3)CC2)C(NC(=O)CCC2CCCOC2)CC1O c1(CN2C(c3ccc(C)c(C)c3)CCC2)ncn2ccccc12 CS(=O)(=O)c1sccc1C(=O)NCC1(NC(=O)CC2CCOC2=O)CCC1 Nc1c(Cl)cnc(C(=O)NC(Cc2nn[nH]n2)C(F)(F)F)c1Cl N1(Cc2ccc(OCC=C)cc2)CCC(O)C(C(=O)Nc2cnncc2Br)C1 c1(C(N2CCC(NC(c3c(C)nc(CO)s3)=O)C(F)C2)=O)cnc2cc[nH]c2c1 N1(C(CCN(C(=O)CCc2ccccn2)CC)=O)CCCC2NC(=O)CC12 CCCCCCCCCCCC(=O)NC1CC2C1CCN2C(=O)CCCOCC c1(C(N2CCC(NC(COC(CC)(C)C)=O)C(CO)C2)=O)c2c(nn1C)CCC2 Cc1ccc(C=CC(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)O)c(C)c1 CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(C(c2ccc(C(N)=O)s2)=O)CC1 CCCC(CNC(=O)C(C1CCCCC1)C)C(=O)NC1CC1c1ncc(C)o1 c1(CC(N2C(CC(=O)NCC3(C(=O)NC)CCOC3)CC2)=O)ccc(NC)cc1 CC1CN(C(=O)Cn2nnc(C3CC3)n2)CC1Nc1ncccn1 C(=O)(C1=CCCCO1)NCc1occ(C(=O)NC2CC(CC(N)=O)C2)n1 Cc1ncnc(O)c1C(N1CCCN(C(C2COC(C)C2C)=O)CC1)=O C(=O)(CCC(N)=O)N(C(CNC(CN(C(C)=O)C)=O)C)C.C(C=O)N C1(NC(C(C2CCCO2)NC(=O)Cc2ccc(O)nc2)=O)CC2CC3C(C2)C13 CCCC(C#N)C(=O)NC(C)(CO)C(=O)N(C(C(N)=O)C1CC1)C N1(C(C2(C)N(C(c3ncc(C)c(Br)c3)=O)CC2)=O)Cc2cccc([N+](=O)[O-])c2C1 C1(CNC(=O)CCSCc2ccccc2)COCCN1C(=O)Cc1cscn1 C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(=O)C(C)(O)C1CCC1)C2 C(CN=c1[nH]c(=NCCCN2CCCCCC2)[nH]c2c1SCC2)(C(C)(C)C)OC Cc1c(CCNC(C2CCN(C(c3ccoc3)=O)C2C)=O)cnn1C N1(C(C2C(C)C2)=O)CCOCC1CNCc1ccc(F)nc1 C#CCC(C)(C)C(=O)N1CC(OCCC(=O)NC2(C(=O)OC)CC2)C1 N1(C(c2c(C)cnn2COC)C(=O)NCCCC)CCC2CCCC12C(=O)OC C1(NC(COCCOCC)=O)CCCC(N(C)C(c2cccc(F)c2)=O)C1 c1(CC(=O)NC(C2CN(Cc3ccc(OC)cc3)C2)C)ccc(F)cc1F c1(OC(C)C)cncc(C(=O)NC2CCCCC2N(C(=O)C(C)CO)C)c1 c1(OCC)nn(C)cc1N(CC(C)OCC)CC(c1ccc(NC(C)=O)cn1)=O C=CCCC(F)(F)C(=O)NCC(CC(C)C)C(=O)NCCc1cocn1 C1(CNC(C(C)NC(=O)NC)=O)CN(C)CCN1C(C1CC1C(C)O)=O N1(C(c2cnc(OC)c(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(N=[N+]=[N-])C1 C1(NC(C(C2CC(F)(F)C2)OC)=O)CN(C(c2ccc(Cl)s2)=O)C(C)(C)C1 C1(NC(c2ccc(C)s2)=O)CCC(C)N(Cc2snnc2C)C1 N1(C(CCOCCCOC)=O)CCC(C)N(C(C2CC(C)(F)C2)=O)CC1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(NC(C3CC3C3CCCC3)=O)CCCC12 C1(CNC(c2ccc(C)cn2)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC12CCC2 N1(C(c2ccc(C#N)c(O)c2)=O)CC2(CC1CNC(c1ccc[nH]1)=O)CC2(F)F c1(CC)ccc(CNC(=O)C(CCSC)NC(=O)CCC2CCOC2)nc1 c1(C(=O)NCC2C(C)CCN2C(c2ccccc2Cl)=O)cc2ccnn2cn1 c1(C(N(C)Cc2nc(O)n[nH]2)=O)cc(Br)cc(Cl)c1O C#Cc1cnn(C)c1C(=O)NCc1c[nH]nc1C(=O)NCCC1CC1C C1(CNC(=O)Cc2cc[nH]n2)C2CN(C(=O)CC=Cc3ccccc3)CC12 CCC(C)C(C)C(=O)NCCN(C)C(C1(c2cccc(Cl)c2F)CC1)=O C1(NC(c2cn(CCN(C)C)nc2)=O)CC2CC(NC(=O)C(C)(C)C)C2C1 N1(C(=O)CO)CCC(n2cc(COc3cncc(Br)c3)nn2)CC1 CON1CCC(C(=O)NC2CCCCC2N(C(=O)CC2CC(SC)C2)C)CC1 N(C1c2cccc(F)c2OC1C)C(c1cc(-c2ccc(OC)cc2)ncn1)=O N1(C(c2n[nH]c(C)n2)C(=O)Nc2ccc(OC)cc2)CCCN(C(C)CO)CC1 N1(C(CC)=O)C2CC=C(C(=O)N(C3CCC3O)C)C1CC2 CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)C(c2ccc(F)cc2)O)C1 c1(C(=O)NCC(CC)NC(c2c(C(F)(F)F)n[nH]c2C)=O)cncc(SC)c1 c1(NC(N2CCC(c3ncon3)C2)=O)nccc2cc[nH]c12 C(C1CCCCC1)=CC(=O)NC1(C(=O)NCC(O)C(F)F)CSC1 Cc1cc(NC(=O)CN2CC(C)C2)ccc1NC(=O)COCCOCCO C1(CNC(C2(n3cc(CC(C(C)C)O)nn3)CC2)=O)CCCC2CCCCC12 CCCC(C#N)C(=O)NC1(CNC(c2ccc(-c3sccc3C)s2)=O)CC1 C12(OCC)CCC(NC(=O)NC3(F)CCCN(C(=O)C(C)C)C3)(CC1)CC2 c1(C(=O)NC(C2CN(C(CC)=O)C2)C)cnn(-c2cccc(C(C)C)c2)c1C C(C)(CC(=O)NC1(CCCC(=O)NCC2(O)CC=CC2)CCC1)NC(C)=O c1(SCC(=O)N=c2nc[nH]n2CCO)cccc(S(=O)(=O)C(F)(F)F)c1 c1(C(N2C(C)CCN(C(C3CCCOC3)=O)CC2)=O)cnn2c(N)ccnc12 c1(CN(C(c2cnn(C)c2C)C(=O)NCC=C)C)ccc(Cl)c(Cl)c1Cl c1(C(=O)NC2CCN(C(c3ccc(SC)s3)=O)C2)cccc(O)c1[N+](=O)[O-] C=CCC(C(=O)Nc1ncc(C(=O)OC)s1)NC1CN(CC)C(=O)O1 CC(C)C(C(=O)NC1CC(=O)N(C(C)C)C1)NC(c1ccncc1Cl)=O c1(NC(C=CC(C)NC(C2(SC)CC2)=O)=O)cc(C#N)ccc1O c1(C(N2CCC3CN(C(C(C(CC)C)OC)=O)C3C2)=O)cc2ccccc2cn1 c1(C(=O)NCC(CN(C(c2cc(C)sn2)=O)C)(C)C)cc(C)n(C2CC2)n1 C1(NCc2scc(C(=O)NC(COC)C)n2)CCCC(C)C1 c1(NC(C2CC(O)CN2c2ccncn2)=O)n[nH]c2ccccc12 Fc1ccc(N=c2scc(-c3ccc(Cl)s3)n2Cc2cccc(Cl)c2F)cc1Cl N1(C(CCCOC(C(C)C)=O)=O)CCC2C1CCCN2C(C1C=CCCC1)=O c1(C(=O)NCCNC(=O)Cc2cnc[nH]2)cc(C(F)(F)F)c[nH]1 N1(CC(=O)NCC2CN(C(C3CCC=CCC3)=O)CCCO2)CCCCCC1=O c1(CCC(=O)NC(C2CS(=O)(=O)C2)CC)ccc(N)c(F)c1.N12CCOC(C1)C2=O c1(-c2scc(C(=O)OC)c2)ccnc(-c2ccnn2C2COC2)c1 Cc1ccc(C)c(CN2CCC(C(N3CCCC3CO)=O)C(O)C2)c1O C1(NC(c2c(C)csn2)=O)CCCC(C(=O)NCc2c(C)cnn2C)CC1 N1(C(c2c(C)nsc2N)=O)CCC(C2CC2)(NC(=O)CN2CCCC2C)C1 C(=O)(CCN=C(NC1C(C)C1(F)F)N1CCCC(C)C1)NC(C)=O CC1(C)CN(C(=O)CC23COCC(C2)C3)CC1NC(c1ccc(Cl)c(O)c1)=O N1(C(Cc2cn(C)nn2)=O)CC2(CCC2)CC1CNC(=O)CC1NC(=O)NC1=O c1(COC2(C#N)CC(NC(c3cccc(OC)c3)=O)C2)ccnc(Cl)c1F c1(CC(=O)NCCOCCNC(CCC(=O)OC)=O)ccc2[nH]ccc2c1 C1(C(N2CCC(CC(C)NC(=O)Cc3csnn3)CC2)=O)CC(=O)C12CCCC2 Cc1nnc(CCCC(=O)NC2CCN(C(C3CN(C(C)C)CCO3)=O)C2)n1C c1(NC2CC(C)n3c2ncn3)cc(Br)ccc1S(=O)(=O)N1CC2CSCC(C2)C1 c1(NCC2N(C(C3CC3C3CCCC3)=O)CCCC2)ncnc2c1CCC2 C=CC(C)(C)CC(=O)N(C1CCN(C(c2cn(C)nc2Cl)=O)CC1)CC c1(N(C2CCOCC2)C(CN2CCC(CC)C2)=O)ccc(C)c(OC(F)F)c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)n2ccnc2)ccc(C#N)c(F)c1 C1(C(=O)NCCCN(C(CCCC=C)=O)CCO)(COC)CCCNS1(=O)=O CC#CCC(C(=O)NCCCC(O)CO)NC(C1CC(C)(C)CCO1)=O CC1CC(C)N(C(=O)CNC(=O)CC(F)(F)F)CCN1C(=O)C=Cc1cncs1 C1(C(N(C)CC2OCCN(C(C(COC)(C)C)=O)C2)=O)C(C)OC(C)C1C CC1CCCCC1NC(=NCc1cccc(C2CC2)c1)NCC12CC(C1)C(C)O2 S(=O)(=O)(c1ccccc1)N(C(C(=O)OC)C)C(C1CC(O)C1)=O c1(N2CCC(NC(c3c(CCC)n[nH]c3)=O)C(F)C2)ncnc2ccc(Cl)cc12 c1(C(N2CC(CC(C)NC(c3nn(C)cc3Br)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(N2CC3CN(C(CCS(C)=O)=O)CC3C2)=O)cn2ccc(CO)cc2n1 CC1(C(=O)Nc2cc(CO)ccn2)CCN(C(c2c[nH]ccc2=N)=O)C1 c1(OC)ccc(C=CC(N2CC3CC2CN3C(=O)C(C)(C)F)=O)c(OC)c1 CC(C)(C)CC(O)CC(=O)NCCC(O)C(=O)Nc1ccc(F)c(CO)c1 C1(n2cc(-c3n(C)c(S)nn3)nn2)CC2(CCCCC2)CO1 CC(C)C(C)CNC(C1CCCN1C(=O)C=CC1CCC1)=O C1(C(=O)NCC(CNC(CN(c2ccccc2)C)=O)(C)C)CCC2(CCC2)O1 Cn1nc(C(=O)NCCC2CCN(C(=O)CC(C)(C)O)C2)cc1C(C)(C)C C(=O)(C1=COCCO1)NC1(CC=C)CCN(C(c2cc(C(F)F)no2)=O)C1 N1(C(c2ccc(N(C)C)cc2)=O)CC(CNC(=O)Cn2ncnn2)C2(CC2)C1 CC1CCc2ccccc2N1CCC(=O)NC(CNC(=O)Cc1ccsn1)CO C1(c2nnnn2C2CC(F)(F)C2)(CCN(CC(F)(F)F)CCCC)CCC(C)(C#N)C1 C(CCC)(C(=O)N1CC(CNC(=O)CC2CCN(C(C)C)CC2)(OC)C1)=CCC C#CCC(CC#C)C(=O)NC(CN(C(=O)C=C1CCOCC1)CC)CC Cn1ccc(CC(=O)NC2CC(NC(c3csc(-c4nc[nH]n4)n3)=O)C2)c1 C12(CNC(=O)CC3CSC3)CCCCC1N(c1ccc([N+](=O)[O-])cn1)CC2 CCC(CCC(=O)N(CCCNC(=O)C=C1CCOCC1)CC)OC CC1CCCC(C(N2CC(CO)(NC(=O)CC(C)c3ccccc3)C2)=O)CC1 c1(OC)[nH]c(=NCC2CCCCN2C(c2ccc(F)cn2)=O)ccc1[N+](=O)[O-] C1(NC(c2c(C)sc(C(F)(F)F)n2)=O)C2CCC1N(C(=O)C(CO)N(C)C)C2 c1(OC)cnc(C(=O)NC2CCCCC2N2CCOCC2)c(F)c1 CCCC(Cc1ccccc1)C(=O)N1CC2CC2(CNC(=O)COCC(C)C)C1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)C(n3ccc(C)n3)C#N)C2)=O)o1)NC CC(CCC(=O)NC12CCN(CC1)C2)NC(C1CC(=C2CCC2)C1)=O c1(N(CC(C)(C)C)CC(C)O)nc(N2CCCN(C(N)=O)CC2)c2sccc2n1 C(C)(CCN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1cc(SC)oc1)=O N1(C(c2c(CC)cns2)=O)CCCC(C)(C)C1CNC(c1ccc(O)cn1)=O Cc1cc(C(=O)NCC(O)CN(C)C(C23CSCC2C3)=O)cc(O)n1 N1(C(CC(C)OC)=O)CCC(CF)(NC(c2cc(C)cnn2)=O)C1 C1(NC(=O)CCOCC2CC2)CCN(C(C2(C3CCC3)CC2)=O)CC12CCC2 c1(OC)cnnc(C(N2CCC(NC(=O)CN(C)C3CC3)C2C2CC2)=O)c1 c1(C(N2CC(NC(c3c(O)cccc3F)=O)CC(C)C2)=O)ccn2ccccc12 N1(C(C2CCC(N(C)C)C2)=O)CCCC(C2OCCO2)C1 c1(OC)cc(C)c2cc(C(N3CCCC3c3ccccc3OC)=O)[nH]c2c1 C(=O)(CC(C(F)(F)F)NC(=O)OC(C)(C)C)N(C1(C)CC(NC(=O)C2CC2)C1)C C1(NC(c2scc(C)c2Cl)=O)CCC2CC1CN2C(c1ccc(C#N)[nH]1)=O c1(C(=O)NCCN(C(=O)CCS(=O)(=O)N(C)C)CC)cn(CC)c2ccccc12 CCC(C)N(OC)C(=O)C(F)C1(O)CN(C(=O)Cc2ccccc2OC)C1 c1(C(=O)NCCCCCN(C)C(C2CCOC2(C)C)=O)ccc2cnn(C)c2c1 C=CCC(CC)C(=O)N1CCCC1C(C)(C)CNC(c1ccccc1)=O C1(c2n(C(C)(C)C)cnc2)CCCN(CCc2ccns2)C1 c1(N(C)Cc2cc3cc(OC)ccc3n2C)c(SC)oc2ccccc2c1=O.CN CCCCC(F)C(=O)NCCC1CSCCN1C(=O)Cn1cnc(=N)[nH]1 c1(-c2[nH]cc(C)n2)ccc(NC(=O)C(N2CC(c3ccc(Cl)cc3)(O)C2)=O)cc1 c1(C(N2C(C)CC(NC(c3c(CC)n[nH]c3)=O)C2)=O)cc(C)cc(Br)c1F c1(C(=O)NC2CC(NC(C3(C(N(C)C)=O)CC3)=O)C2)cc(O)nc2ncn(C)c12 N1(C(C2C(C)CCOC2)=O)CCC(C(=O)NCCC2CCCC3CC23)C(C)(C)C1 C1(C(N(CCO)CC)=O)(OC)CCN(CC(=O)NCc2n[nH]c(=N)s2)CC1 C1(NC(C(CCC2CC2)NC(C=CC(CC)C)=O)=O)CCn2nccc2C1 c1(OC)ccc(O)cc1C(=O)NC(CN(C)C)C(N1CCC(OC)C1C)=O C1(CN(C(C=C(CC)CC)=O)CC)CCCN1C(=O)C=CSCc1ccco1 N1(C(C(CC)C#N)=O)CC(OC)CC(NC(C2(c3ccn(C)n3)CC2)=O)C1 C1(CNC(c2cc(Cl)cs2)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CC12CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(CN(C(=O)Cc2cn(C)nn2)CC)C1 c1(OC(c2ncc(C(N3CC(OC4(C)COC4)C3)=O)o2)C)cccc(F)c1 c1(C(N2CCC(CC)C2C(=O)Nn2ccnn2)=O)cc2cccnc2[nH]1 Cc1ccc(C(N2CC=CCC2C(N2CCCC(CC3CC3)C2)=O)=O)cc1F C(=O)(C(O)CC(F)(F)F)NC(CC=C)CNC(=O)C=Cc1ccccc1OCC c1(SCC(N2CC3C(NC(C=NOC)=O)C3C2)=O)nnc2ccccn12 c1(OC)ccc(C(=O)NCCCN(C)C(c2cocc2C)=O)nn1 c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(C2CSC2)=O)C(C2CC2)C1 C1(C(=O)NCC(CC(F)(F)F)NC(c2cn(C)nc2)=O)CCC(N=[N+]=[N-])CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CC(=O)NCC=CCNC(CN2CCC(OC)C2)=O)CCC(=O)NC1=O c1(C(N2CC(NC(CCOC(C)C)=O)C(O)C2)=O)ccc(F)c(O)c1F C1(NC(c2c(C)[nH]nc2Cl)=O)CC2CC1N(C(c1cc(Cl)ccn1)=O)C2 N1(C(C(CCSC)OC)=O)CC(CNC(=O)C=Cc2ccc(C)cc2)CC1(C)C N1(C(C2C(NC(C3CCCO3)=O)C2)=O)CCOC(C2CC2)C1 Cn1ccc2nc(N3CC(CO)(NC(c4ccncn4)=O)C3)ncc12 CC1COCCC1N(C)C(c1cn(CCNC(=O)CCOCC(F)F)cn1)=O CC(C)CC(C)CC(=O)NCC=CC(N1CCN(C)CC1)=O N1(C(CC(C=C)(C)O)=O)CCC(C(N2CCC(CN(C)CC)C2)=O)C(C)(C)C1 C(=O)(C(Cc1ccncn1)NC(=O)OC(C)(C)C)NC(C)CF c1(C(CO)NC(C2NCC(=O)NC2)=O)c(F)cccc1Cl c1(CNC2(C(=O)OC)CCN(c3ccnc(Cl)n3)CC2)noc2c1COCC2 CCC(CC(=O)N(C)CCN(C(=O)C(C)COC)C)C(C)C c1(C(=O)NCC2CCC(NC(c3c(C)n(C)cc3)=O)C2)cc2n(c1)CCCC2 CCC(C)(CNC(c1cnn(C2CC2)c1)=O)C(=O)N1CC2CC1CS2 c1(C(N2CCC3C(NC(C(C)OCC=C)=O)C32)=O)ccnc2c1cnn2C c1(CN2CC3C(Nc4cnn(C)c4C(F)(F)F)C3C2)cccc(C(F)(F)F)c1F c1(SC)ccc(C(=O)N(CC(C)NC(c2nocc2Cl)=O)C)cc1[N+](=O)[O-] n1(CC)nnc(C(N2CCCC2C(C)(C)NC(=O)CC2CC(F)(F)C2)=O)c1C C(CC(=O)NCc1conc1C)(C(F)F)NC(CCc1cnc(C)o1)=O c1(C(=O)NCC2CN(C(CCC3CCC(C)O3)=O)C2)cnc2ccccn2c1=O Cc1nnc(NCC2CCN(C(=O)Cc3cnoc3)C2)c(C#N)c1C C1(CNC(C=C(C)C(C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1C CCC(CC(=O)N(CCC(C)NC(=O)CCc1cccnc1)C)SC c1(NC(CC)(C)Cc2ccccc2F)cc(CN(C)C)cc(C(F)(F)F)c1 CC1CC2CN(C(=O)C(O)c3ccsc3)CC2N1C(=O)CC1CC2CC2C1 N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)C(=O)NCC(C)(C)OC Cc1cc(C(N2CCSCC2CCNC(C2CC2C(F)F)=O)=O)sc1C C1(C)(CO)CN=C2NC(=NC3=C2COCC3)N2CCN3C(=O)N(C1=O)CC23.CO C(=O)(CCC1=NNC(=O)CC1)NC1C(C)CN(C(C2CC(OC(F)F)C2)=O)CC1 N1(C(Cc2c(CC)n[nH]c2CC)=O)CC2(CC(NC(c3csc(C)n3)=O)CO2)C1 N1(C(C2(OCC)CCCC2)=O)CCOC(C(C)NC(c2cncc(F)c2)=O)C1 C1(C(=O)NCc2ncco2)CCCCN1C(C1CCCN1C1CC1)=O C1(C(=O)OC)CC2C(CCC(C)N2CCOC2CCC2)O1 CC1=NN(C)C(=O)C1CC(N1CCN(C(c2[nH]cnc2C)=O)C(C2CCC2)C1)=O N1(C(CC(=O)NCC#C)=O)CCCC(NC(c2cncc(C)n2)=O)C1CC c1(CCC)ccc(S(=O)(=O)NC2CCC(C(=O)Nc3cc(O)ccc3Br)C2)cc1 C1(C(=O)NCC=CCC(=O)N(CC(C)OC)C)CCCC(=O)C1 c1(C(N(CC(CO)(CO)NC(=O)C=Cc2cnc[nH]2)C)=O)csc([N+](=O)[O-])c1 CC1(CNC(c2ncnn2C2CCC2)=O)CC(F)(F)CN1C(C12CC(C1)C2)=O N1(C(CCC=C(C)C)=O)CCN(C)C(CNC(c2ccncc2)=O)C1 c1(CN(C(=O)C(C)(C2CCC2)NC(c2ccc(O)cc2)=O)C)cccc(F)n1 C1(C2CCCNC2)(C(=O)OCC(=O)NC2CC2)CC1 C1(C)(CNC(CCN(C(CCOC)=O)C2CC2)=O)C=CCCC1 C1(NC(C(C(C)C)OC)=O)CC2(CCCCN2C(=O)C(CSC)OC)C1 c1(C(=O)NC2CCC(N(C)C(c3cccs3)=O)C2)cccc(NS(C)(=O)=O)c1 C1(C(N2C(CO)CC(NC(C(CCCC)NC(N)=O)=O)C2)=O)Cc2nnc(C)n2C1 Cc1ccc(F)c(CNC(c2c(I)cnn2C)c2nnnn2C2CCCC2)c1Cl Cc1cc(C(=O)NC2(C(=O)NC(c3ccns3)C)CCCC2)ncn1 C(=O)(CC(C(=O)N1CCC(NC(=O)CC(C)OC)C1C)N(C)C)OC c1(OCC)cccc(OCC)c1C(N1CCN(C(c2ccsc2)=O)CC1)=O C1(NC(COc2ccc(C(CC)C)cc2)=O)CCCCN(C(=O)CC(F)F)C1 CCC(C)(C#N)C(=O)NCC(C)CNC(c1nc(C)ccc1Br)=O c1(C(=O)NC(CNC(C(Cc2c(C)noc2C)C)=O)C)ccc(F)c2occc12 CN=c1[nH]c(=NCc2cncnc2)[nH]c(=NCCCN2CCCN(C)CC2)[nH]1 c12cc(on1)NC2=O.C(=O)(C(C1CCC1)OC)NC.C=CC(C1CC1)C1CC1 N1(C(Cc2nc(C)oc2)=O)CCCN(C(=O)CCc2ncccc2C)CC1C c1(CC(=O)N(C)CC2(CNC(C(C(CC)O)C)=O)CC2)c(C)nc2ccccn12 CC(C)CCCC(=O)N1CCC(NC(c2cn(C(C)C)nn2)=O)C1 CCC1=NOC(C(=O)NC(CNC(=O)C(c2cncn2C)=O)CC(C)C)C1 Cc1nn(CCO)c(C)c1C(=O)NCC(C)CN(C)C(C1COC(=O)C1)=O Cc1cc(C(=O)NC2CC(F)(CNC(c3cc(C(C)C)on3)=O)C2)c(N)cc1F N1(C(C2C(C)(COC)C2)=O)CC(C2CN(C(c3ccc(Cl)c(OC)c3)=O)C2)C1 C1(C(N2CCC(NC(c3sccc3Cl)=O)C2)=O)CCCCC12CCC2 C1(C(=O)NC23CC(CNC(c4cnccc4Cl)=O)(C2)C3)CCCC1C1CC1 c1(NC(N(CC(c2ccccc2)CC)CC)=O)nc2ccc(I)cc2s1 C=CCN=C(NCC(=O)N(CC)CC)NCC1(C)CCCCC1 c1(CC(CNC(c2cc(-c3cccs3)ns2)=O)CO)ccccc1F C(=O)(CC1=CCCCC1)NCC(N(C(C(C(COC)C)C)=O)C)C1CC1 N1(C(CCOCC)=O)CC(C)C(C)(CNC(c2c(N)cccc2Cl)=O)C1 c1(NC(COc2c(C)cccc2)C)ccc(S(=O)(=O)NCC(O)C2CC2)c(Cl)c1 c1(NC(=O)NC(C)CC#N)cc(NC2CCCC2C(C)(C)C)ccn1 N1(C(c2n(C=C)ncc2)=O)CCC2(NC(=O)C=C3CCSCC3)CCCC12 c1(C(=O)NC(CNC(CCSCC)=O)(C)CO)cncc(F)c1 c1(C(=O)NC2C3N(C(C=CC=CC)=O)C(CC3)C2)cc(Br)cc([N+](=O)[O-])c1 N1(C(c2n(CCOC)ncc2)C(=O)NCC2CCCO2)CCc2ncc(C)n2CC1 c1(C(N2CCC(OCCNC(=O)Cc3cncs3)C2)=O)cncc(C(F)F)c1 c1(C(=O)NC2C(C)(CN(C(=O)C(C)(F)F)C)CCC2)cc(O)c2cnn(C)c2c1 N1(C(=O)Oc2ccccc2Cl)CCCc2[nH]c3ccc(F)cc3c2C1 Cc1ccc(O)c(NC(=O)CC2CN(C(=O)C(O)CNC(N)=O)CC2C)c1 c1(OCC)cncc(NC(C2CCCN2C(c2ncccc2Cl)=O)=O)c1 C(=O)(C(CNC(C1(C)CC(C)(C)C1)=O)C(C)C)Nc1c(CC)nsc1 C1(C(=O)NCCN(CCCN(C)C)C(=O)Cc2cnccn2)CCC2CCC1O2 C1(C)(C(N2CCCC(CC(=O)NC(C(=O)OC)COC(C)C)C2)=O)CC2(CCC2)C1 Cc1nc(CCNC(C2(NC(=O)CCc3ccsc3)CCOCC2)=O)c(C)o1 C(=O)(C1=C(c2ccccc2)SCCO1)N1C2CC(NC(=O)CC(F)(F)F)C(C2)C1 CC(C)(CC#N)C(=O)NCC1(F)CCC(NC(=O)COCc2ccccc2Cl)C1 N1(C(CNC(=O)OC)=O)CCN(C(=O)CN2CCCC(C)C2)CC(O)C1 C12(C(=O)OCC)COC(CN(CCCc3nnc(C)o3)C)(C1)C2 CCCCCCC(C)(CC)C(=O)NC(CNC(C1(C(N)=O)CCC1)=O)CC CC1Cc2cccc(C(=O)Nc3cccc(C4SCCCS4)c3)c2O1 N1(C(C2(C)COC(=O)C2)=O)CCCC(C)(C)C1CNC(=O)Cc1csc(S)n1 c1(C(C(=O)NCCCN(CCCC)CCCC)N)cccnc1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C=COCC)=O)(CO)C1 c1(CN(C(C2CCOCC2)C(=O)NCCOC2CC2)CC)ccc(N(C)C)cc1 N1(C(C(CCC)=CCC)=O)CCC(C)(C)C1C(=O)NCCC(C)(C)OCC C(=O)(C#CC1CCCOC1)NC(C)(C)CNC(=O)C(C)(C)C(C)(C)C C1(C2CC2)(C(=O)OCC(COC)OC)CCN(C(=O)OC(C)(C)C)C1 N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCC(CCNC(C2CC(=O)N(C)C2)=O)CC1 Nc1ccnc(C(N2CCC(F)(CNC(c3cncn3C3CC3)=O)C2)=O)c1 c1(CC(C)NCc2cn(CCCCCO)nn2)ccc(O)cc1 C1(C(N2CCC(C)(NC(c3sc(C)c(O)n3)=O)C2)=O)CC1C1CCCCC1 c1(CC)nc(=N)[nH]cc1C(=O)NC(CNC(=O)C1=COCCC1)CC(F)(F)F c1(C(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=CCC2)C(=O)NCCCF)CCCC2(CC(O)C2)C1 N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(c1oc(C)nc1C)=O CC1(C)CN(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)CCO1 CCCC(CC)CC(=O)NC(C)CCNC(=O)CCSc1ccccc1F c1(CNC(c2cc3ncccc3[nH]2)=O)cccc2ccccc12 C1(C(N2C(C(N(C)Cc3cccc(F)c3)=O)CSC2)=O)C2CC3C(C2)C13 C1(C(=O)NCC(CNC(CSC(C)(C)C)=O)(C)F)CCC(C2CC2)C1 CCC(CC(=O)N1CCCC(C)(CNC(c2snc(C)c2N)=O)C1)C(C)(C)C Cc1c(NC(=O)C(CCC2(C#N)CC2)N(C2CC(F)(F)C2)C2CC2)cccc1Cl C(=O)(C(O)CC(C)(C)C)NC1CCC(C(=O)NCc2nn(CC)nc2C)C1 C(=O)(C1=NN2CCCN=C2N1)N1C(CCNC(C=CC2C(C)C2(Cl)Cl)=O)CCC1 c1(C(=O)NCCC(C)NC(=O)C(C)(C)c2ccnn2C)cc(Cl)c(Br)[nH]1 C1(NC(CN2CCN(CC)CC2)=O)CC(F)CN(C(c2cncs2)=O)C1 N1(C(C(C)=CC)=O)CC2CCCC(N(C(=O)CSCc3ccc(Cl)cc3)C)C2C1 C1(NC(C(c2ccco2)NC(C2CC3(CCC3=O)C2)=O)=O)CCCCCCC1O c1(C(=O)NCC(CO)NC(c2ccn(C)n2)=O)ccc2cc(O)ccc2c1 c1(C(C)C)cc(C(=O)NC2CN(C(C3(O)CCC3)=O)C2)cc(F)c1 C(=O)(C(CC)C(=O)N)NCCCN(CC)CC.C12CC(C1)NC2=O.N(C)(CC)CC c1(C(N2CCC(CC(=O)NCC3(C)OCCO3)C2)=O)ccnc(Br)c1F CCC(CC(=O)NC(C)(C)CN(C(=O)CCCCN(C)C(C)=O)C)C1CC1 C(c1ccc(-c2ccccc2)s1)=CC(C)N(C(C(CC)C1CCC(=O)N1)=O)CC c1(CC)ccc(C(=O)NCCOC2CN(C(c3cnsc3)=O)C2)nc1 c1(C(=O)NC(C2CN(C(=O)CC3CCC(C)(C)C3)C2)C)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C3(CN(C(c4c(C)ncn4O)=O)C3)CC2)=O)cc(C#N)c(N)cc1O CC(C)CC(O)C(=O)NC1(C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(C2OCCC(=O)C2)=O)CCC(NC(=O)C=Cc2ccco2)C(F)C1 c1(NC)cc(N2CCCC(C)(C(=O)NCCC(N)COC)C2)nc(=N)[nH]1 CC1(CNC(C2CC2F)=O)CN(C(=O)C(c2ccc(F)cn2)(F)F)CCO1 c1(C(N2CC(O)(C(C)NC(C3C4CCC34)=O)C2)=O)ccccc1Br c1(OCC)cccc(NC(=O)C(=O)N(C2CCSC2)Cc2ccco2)c1 C(=O)(CCCC(=O)NC)NCC1N(C(C(CCC)F)=O)CC(O)C1 N1(C(c2nc(OC)oc2)=O)CCOCC1CNC(=O)CCc1nc(C2CC2)no1 Cc1cc(NC(=O)CC2CN(C(c3cc(Br)ccc3Cl)=O)C2)ncc1F C1(CNC(C(c2cccc(Cl)c2)C)=O)CCC(NC(=O)C(F)(F)CO)CC1 N1(C(C(CC)SCC)=O)CCCCC12CN(C(=O)CN(c1c(C)noc1C)C)C2.C(CO)O N1(C(CC(CNC(C(CC(C)C)OC)=O)C)=O)CCCC(C)(C#N)C1 C(C(C)(C)CNC(C1CCC1(C)C)=O)N(C(=O)COCc1ncnn1C)CC Cc1sc(C(=O)NC2CCN(C(c3ccoc3Cl)=O)C2C)nc1Br CCC(C)(C(=O)N1CCN(CC2CCCN(C(C3CC=CC3)=O)C2)CC1)C(F)F N1(C(c2c(F)ccc(C#C)c2)=O)CC2CN(C(=O)C=Cc3ccco3)CC2(C)C1 C1(C(N2CCC(N(C)C(c3nccnc3Cl)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(CNC(Cn3ncc(C)c3)=O)CC(F)(F)C2)=O)cccc2nccn12 c1(C(=O)NC23CN(C(CCC(C)C)=O)C(CC2)CC3)c[nH]c2cc(F)ccc12 Cc1cn(C)cc1C(N1CC(NC(=O)CC2CSC2)CC1C)=O C(CCC(C)C(=O)N1CCN(C(c2nc(C)ccc2C)=O)CC1C(C)(C)C)OC CN1CCC(C)(C(N2CC(NC(=O)C(Cl)=CCl)C(F)C2)=O)C1 N1(CCN(c2ccccc2)C)CCC(NC(c2csc(O)n2)=O)CC1 c1(OC)ncc(Br)cc1NC(C1CC1C(=O)Nc1cccc(C2CC2)n1)=O N1(C(C(C(=O)OCC)OC)=O)CCOCC(NC(=O)CCC2CC(F)(F)C2)C1 c1(-c2cn(C)nn2)ccc(N)c(F)c1.C1(C(N2C(CC=O)CC2)=O)(CC)CCC1 CCCCCCCC(=O)NC(C)(CNC(c1ccnc(O)c1F)=O)CC C=C(C)CCCC(=O)NC1(C)CN(C(c2ccc(OC)cc2C(F)F)=O)C1 N1(C(CNC(C2CC(C)C2)=O)=O)CCCC2CN(Cc3ncnn3C)CC12 c1(SCCCC(=O)NC2(c3nn[nH]n3)CC(O)(SC)C2)nc2ccccc2s1 c1(C(=O)NC(C(C)NC(C2CN(C)CCO2)=O)C)cc(C(F)(F)F)cnc1O N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(c3occ(C)c3C)=O)C2)C1 C(C)(C)(CC(=O)Nc1ccc(C(C)=O)cn1)N(C(CSC)=O)C c1(CC)c(C(=O)NC2CC(CNC(c3c(C)coc3C3CC3)=O)C2)cccc1C c1(C(N2CCC(NC(c3c(C)nccc3)=O)CC2C)=O)cc2ccccc2cn1 CN1CC(O)CC1C(N1CC(CCCCNC(=O)C(c2cccnc2)O)C1)=O CC(C)CCCCC(=O)N(C1C2CN(C(=O)C=CC3CCCCC3)CC12)C C1(C(C)CNC(c2c[nH]nc2C(C)(F)F)=O)CCN(C(=O)CCS(C)=O)CC1 N1(C(C(C)NC=O)=O)CC2CC1CN2C(c1ccoc1CN1CCCC(O)C1)=O N1(C(C2(COCC)CCC2)=O)CC2OCCN(C(=O)C(C)CSC)C2C1 NS(=O)(=O)c1ccsc1C(=O)NC1CC(NC(C2CCO2)=O)C1 c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(=O)CN2CCC2C)C)C)c(F)c1 c1(CC(=O)NC2(CO)CCN(C(=O)CC3CC(C4CC4)C3)C2)cccc(F)c1Cl C1(NC2CC=CC(C(N3CC=CCC3c3cccnc3)=O)C2)CC2C(C1)C2(F)F Cc1ccc(C(C)C)cc1OCC(=O)NCC1CCC1NC(c1ccc[nH]1)=O N1(C(C(CC)C(=O)OC)=O)CCC2(CCC2)C(NC(c2nc(C)ncc2Cl)=O)C1 N1(C(=O)CCc2cnccn2)CCC2(CC1)CN(C(c1nncs1)=O)CC2CO N1(C(c2c(CC)c(C(N)=O)c(C)[nH]2)=O)CC2(CCCCN(C(=O)C3=CCC3)C2)C1 C=CC(CC)CC(=O)N1CCC2C(C(=O)NCCC3COCCO3)C2C1 C(=O)(C1=C(Cl)CCCC1)NCC1C(C)CN(C(=O)CCc2cc[nH]n2)CC1 c1(C(=O)NC(CNC(c2n(CCC)ccc2)=O)C2CCC2)cccc(N)c1O Cc1ncc(C(N2CC(NC(c3ccc(Cl)cc3)=O)CCC2C)=O)cc1Cl c1(C(C(=O)NCC2CCN2C(=O)CNC(=O)C(F)(F)F)C2CC2)cccc(Cl)c1 S(=O)(=O)(c1c[nH]c(=NCC2COCO2)cc1C)NCc1c(SC)cccc1C n1(CCNc2cc(C#N)ncc2)cc(CO)cc(CC#N)c1=O N1(C(c2occ(C)c2C)=O)CCN(C(C2CCN(C)C2)=O)CC1C1CC1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(=O)CCNC(=O)C(C)(C)C)sc1C C1(=O)CCCCOCCC2(CC2)CN1.C#CC1(C(=O)NC(C)(C)C)CC1.C1CO1 c1(OC)c(Cl)ccc(C(N2CCC(F)C(NC(=O)CSC(C)=O)C2)=O)c1F N1(C(=O)Nc2cc(-c3ccc(OC)cc3)nn2C)CC(N(C)C)CC1(C)C c1(CC)ncnc(NC2CCCC(NC(c3c(C)nsc3NC)=O)C2)c1F c1(OC)cccc2c(C(N3CCC(N(C(=O)C(C)=C4CC4)CCO)C3)=O)coc12 C1(C(=O)NC2CC(C)C2)CCN(C(=O)C2=COCC2)CC1(C)C c1(C(=O)NC2C(C)CN(C(=O)Cc3csnn3)CC2)cccc2c1ccn2C C1(C(C)C(=O)NC2(CF)CN(C(=O)CCc3cn[nH]c3)C2)CCC(=O)N1C CC1(C)C2CCC1(CC(=O)NC1CCCC(NC(c3cc(F)n[nH]3)=O)C1)CC2 N1(C(Cc2cc(OC)ncc2)=O)CCN(C(C2CC(N(C)C)CCO2)=O)CC1C C1(CS(=O)(=O)N(C)C)(C(C)C)CCOCC1.N12CC(C(C)C1)C2=O C(CC(C)C(=O)N1CCC(CN(C(=O)CC(C)CF)C)CC1)=CCC N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CSC)CC1CC C1(OC)(CNC(C2C(C)C2C)=O)CCN(C(c2sccc2C(C)C)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(c2cncc(C(C)C)c2)=O)C(C)C1 O=C(C(F)C(F)(F)F)N1CC2(C(N3CC4CC3(C(F)F)C4)=O)CCC1C2 c1(NC(C2(F)CCN(C(=O)Cn3cc(Cl)cn3)C2)=O)cc(Br)cnc1[N+](=O)[O-] C1(CC=C)(NC(c2coc(Cl)n2)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 C1(NC(COC2(C)CCCC2)=O)CCC2CN(C(=O)C#CC3CC3)CC2C1 C1(NC(c2cc3ccccn3c2)=O)CCCCC12CCN(C(=O)CCCF)C2 N1(C(CC2C(C)=NNC2=O)=O)CC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 c1(C(N2CCC(OCCNC(=O)C(F)OC(F)(F)F)C2)=O)cc2ccccc2o1 Cc1cc(C(=O)NC2CCCC(N(C(=O)CC3CCOCC3)C)C2)ncc1F c1(C(=O)NCc2occ(C(=O)NCC(CC)C3CCC3)n2)cc(OC)cnn1 C(=O)(C1=C(F)CN(C(=O)CC(C)(C)CC(F)F)CC1)NCCCCCC(C)C C1(CNC(C2(C)CC2F)=O)(NC(=O)CC2CC3(CCC3)C2)CCOCC1 C1(CCNC(C(COCC)C)=O)CC(OC)CN1C(c1cccn1CC)=O c1(C(C(N2C(C(=O)NC)CCC2)=O)NCc2cn(CC)cn2)c(C)cccc1Br CC(C)(C(=O)NCC1CCC(NC(=O)CC2CC2)C1)C1CCOC1 c1(OC)cccc(CN2C(C(=O)NC(C3CCC3)C)CC3CC23)c1O c1(C(N2CC(CCC)C(OC)C2)=O)nn(-c2ccccc2)c(=O)nc1O c1(C(=O)NC(C)(C)CNC(c2coc(Cl)c2)=O)ccc2c(c1)CC(C)(C)C2 C1(OC)CN(C(c2nn(C)nc2Br)=O)CC1NC(c1ccc(C)cn1)=O C1(OC)CCN(C(C2CN(C(c3ccc(O)nc3)=O)CC2F)=O)C1C C1(C(=O)NC)C2CN(C(=O)CNC(=O)C(=O)NC)CC12 c1(NCC)cc(Cl)ccc1C(=O)NC1CCC1CNC(C1CN2CCC1CC2)=O n1(CCC(N2CCC(N(CC(=O)OC)C)C2)=O)sc2ccccc2c1=O c1(N2CCOCC(NC(C34CCCC3C4(F)F)=O)C2)nc2ncc(Cl)cc2s1 C1(C)(C(N(CC(O)CNC(=O)COC2CCC2)C)=O)CC(C2CC2)=NO1 CC12CCCCC1CN2c1ncc(C(F)(F)F)cc1Br c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)ccc(F)c(Cl)c1F C(=O)(C#CC(=O)N(C1CN(C(c2ccc(C(F)(F)F)o2)=O)CC1F)C)N(C)C C1(c2n(C)ccn2)CN(C(C2CC2c2ccsc2)=O)CC1NC(C1(O)COC1)=O CC(C)CCC(O)C(=O)N1CCN(C(c2cccc(F)c2)=O)C(c2ncc[nH]2)C1 C(=O)(C(C(=O)N1CC(C)C(C)(CNC(=O)COC2CC2)C1)C(C)(C)C)OC(C)(C)C Cc1cccc(C(=O)OC(C)(C)C)c1Cl.N12CC(C(C)C1)C(=O)NCCOC2=O c1(C(N(CC(C)CNC(=O)CCC(C)N(C)C)C)=O)cc(C#N)ccc1Cl N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(C2CC(C)(O)C2)=O)C2CS(=O)(=O)CC12 C1(C(N(CC)CC2CC=CCC2)=O)CCCN(Cc2noc(CC(C)C)n2)C1 C1(C(N(CCOC)CCO)=O)CCC(CNC(C2CCCCC2C)=O)CC1 c1(C(=O)NCCOCCCNC(Cc2c(C)occ2)=O)c[nH]ccc1=N C1(C(=O)NCC(C)F)CN(C(=O)CCC2CCCC2)CC1F Cc1ccnc(C(N2CCC(Cc3cccnc3)C2)C(=O)NC2CCOC2)c1Br c1(CCC(=O)NCC2(CCNC(CSC)=O)CC2)cncnc1 Cc1[nH]cc(C(=O)NC2CN(C(c3cc(C#N)c[nH]3)=O)CC2C)c(=O)c1Br C1(C(N2CC(C)(NC(C(CCCC)O)=O)C2)=O)CC(=O)CC12CCC2 N1(C(C2CC23CCCC3)=O)CC2CCN(C(=O)C(c3ccc(C(F)F)cc3)F)C2C1 C1(C(=O)NC(C(C)NC(c2n(CC)cnn2)=O)(C)C)CN(C(C)=O)CCO1 CC(C)(CCNC(=O)C(F)C1CCCC1)C(=O)NOCCCCC1CC1 c1(CN(C(=O)CC2CCCCO2)C)ccccc1CNC(=O)C(CO)S(C)(=O)=O n1(CCCOC)nnnc1C(c1ccn(CC(F)(F)F)n1)NCC1CC1(C)C c1(C(=O)NCc2c(CC)n[nH]c2)cccc(OC(C)(C)C)c1 CCC(O)C(C)C(=O)N1CCCC1CCCNC(=O)CCc1ccccc1 CC(C)CC(C(=O)NC1CCCC(NC(=O)CCc2nncs2)C1)N(C)C c1(C(=O)NCC(CC=C)NC(=O)CC(C)c2ccco2)c([N+](=O)[O-])cnn1CC c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2C)c(Cl)cncc1Cl CCCC(C(=O)N(C)CCOCCNC(=O)C=C(Cl)Cl)C(C)C N1(C(C(CC)Sc2ccccc2)=O)CCC(C)(NC(c2nn(C)cc2N)=O)C1 c1(OC)ccc(C(C)C(N2CC(NC(=O)CC#N)C(C)(C)C2)=O)c(C)c1 c1(OC)cc(C(C(=O)NC2CC2)N(C2CCS(=O)(=O)C2)C2CC2)ccc1Cl c1(C(N2CC(CNC(C3(SC)CCC3)=O)N(C)CC2)=O)ccn2nccc2c1 N1(c2c(C(=O)OC)cccn2)CC(NC(c2n[nH]c(C)c2Cl)=O)C(C)(C)C1 C123COC(C1)(C2)NC(=O)C(C)NCC1CN(C1)C(=O)C3.S(C)(=O)(=O)N(C)C C(=O)(C(CC(F)F)NC(c1ncoc1C)=O)NCc1scc(C)n1 C1(ONC(c2ccc(CN(C)C(C3CCC(=O)NC3)=O)cn2)=O)CCCCC1(C)C c1(-c2nnc(COC3CCN(S(C)(=O)=O)C3)o2)cccc(Cl)c1 C12(NC(C(CC)SC)=O)CCCN(C(c3ncc(Cl)nc3Cl)=O)CC1C2 C(=O)(C#CC1CCCCC1)NCCOCCC(N1CCC(C)(CO)C1)=O c1(CNC2CCC(C(=O)Nc3c(OC)nc(Br)cn3)CC2)cc(Cl)cc(Br)c1O C1(CNC(c2cccc(C(C)C)c2)=O)CCN(C(=O)Cc2cncn2C)C1(C)C C1(NC(C(C(CC)C)N(C)C)=O)CC2(CCCCN2C(=O)C(C)=C(C)C)C1 Cc1ccnc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(C)CC2CCCC2)C1 C1(C(N2CC=CC2)=O)CCCCN(C(C2(C)CCCS2)=O)C1 N1(Cc2cc(C(C)=O)c(O)cc2)CC2CCN(C(=O)Cc3ccc(Br)cc3)C2C1 C(=O)(CCCC(C)(C)C)NCC1(F)CCCN(C(C(C)OCC2CC2)=O)C1 C1(CS(=O)(=O)N(c2cccnc2Cl)C)CCOC1(C)C C1(N(C)C(c2ccc(F)o2)=O)CCCC(NC(C2(C(N)=O)CC2)=O)C1 c1(CNCc2ccc(-c3ccc(COC)c(OC)c3)o2)c[nH]c2ncc(Cl)cc12 Cc1nc2c(s1)CCCC2C(=O)N1CC2(CCCC(c3ccccc3CO)O2)C1 C1(NC(C(=O)NCC)=O)CN(C(C2(c3ccc(OC)cc3)CC(O)C2)=O)CC1(C)C S(=O)(=O)(CC(C)c1ccccc1)N1C(C(NOCC=C)=O)CC1 c1(OCC(N2CC(CCNC(C(C)(C)n3ccnn3)=O)C2)=O)nc(O)nc(O)n1 C=C1CCN(C(c2ccc(C3CCCC3)cc2)C(=O)NCCOCC)CC1 N1(C(c2c(C)coc2)=O)CC2CCC(C1)N(C(c1csnc1Cl)=O)C2 CCCC(O)CC(=O)N1CC2CC2(CNC(c2ccc(C)cc2Cl)=O)C1 CC1CC=C(C(=O)NC2C=CCN(C(c3cccc(F)c3C3CC3)=O)C2)CC1 c1(C(=O)NC2(C)CCN(C(C3C(C)C3(F)F)=O)C2)ncc(C(F)(F)F)cc1N C1(NC(C(C)=CC2CC2)=O)CC2(C1)CC2NC(c1cc(CS(C)(=O)=O)on1)=O C(c1ccccc1Cl)=CC(=O)NC(C)CC(C)NC(=O)C(C)n1cnnn1 c1(C(=O)OC)ccc2c(c1)CN(C(=O)NC(c1ccc(C)nc1)C)CC2 C1(OC)CCN(C(=O)C2=CCN(C(=O)CCCC(=O)OC(C)(C)C)C2)CC1C c1(C(=O)NC2C(CNC(c3cn(C4CC4)nn3)=O)C2)cc(F)cc(Br)c1O Cc1ccnn1CC(=O)N(CCC(=O)NCCCn1cncn1)C1CC1 CCC1=NOC(C(=O)NCC2CN(C(=O)CC(C)CN(C)C)C2)C1 CON1CC(C(=O)NCCN(CCOCCO)C(c2ccccc2C)=O)CC1=O c1(OCCOC)cccc(C2CC2OCC=CCl)c1 N1(C(C=C(CC)CC)=O)CC2(CCC2)CC1CNC(c1nnn2c1CSCC2)=O c1(CC)cnccc1CNC(=O)NCC(C)COc1ccccc1C c1(CCC(=O)NCCCN(C(C(CC)O)=O)C)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)NCCCNC(=O)C=Cc2ccc(Cl)s2)cc2cccn2c(O)n1 C1(NC(C2C(C)CCO2)=O)CN(C(=O)CCCCN2CCOCC2)CC1F c1(C(N(CC(C)NC(c2cnn(C)c2)=O)CC)=O)cc(C(C)(C)C)n(C)c1C N1(C(c2c(CC)scc2)=O)CC2COCCC2(NC(c2csc3nnsc23)=O)C1 C(=O)(CCCCCN(C(=O)COC(CCCOC(C)C)=O)CC=C)OCCC(C)C C1(C(C)(C)C)(C(N2CC(NC(=O)CCc3ccsn3)C2)=O)CCCCC1 O=C(C1=CCOC1)NC1CC1NC(C1(c2ccsc2)CC1)=O Cc1ccncc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)s1)=O c1(OC)cc(C(N2CCCC(NC(=O)C(C)C(C)C)C2)=O)cc(Cl)n1 C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(c1ccnnc1S)=O)CCO2 c1(NC(C2CCCC2)C)nc(N2CCC(F)(CO)CC2)nc2scnc12 Cc1cccc(C=CC(=O)NC2CCN(C(=O)Cn3cc(C(F)(F)F)cn3)C2)c1 c1(OC)ccc2c(c1)CC(C(=O)NCC(CO)NC(=O)CC(F)(F)Cl)O2 c1(OC)ccc(N(C)C(C23CC2CN(C)S3(=O)=O)=O)c(OC)c1 CCC(COC)C(=O)N1CCCC1(C)C(=O)NCc1ncn(C2CC2)n1 Cc1[nH]c(C)c(C(=O)NC(C)CCNC(=O)CC2NC(=O)NC2=O)c1C O=C1Cc2cc(C(N3CCCCC3CNC(C3CC34CC(O)C4)=O)=O)ccc2N1 N1(C(C(C(C)(C)C)O)=O)CC=C(CC(=O)NC2CC3(COCCO3)C2)CC1 C(=O)(N=c1nc[nH]n2cc(Br)cc12)c1c(C)nc(CN)nc1C N1(C(=O)COCCF)CC2(CCCCN2C(c2scnc2C(F)(F)F)=O)C1 C1(CNC(C(C)=C2CC2)=O)CC2COCC2N1C(=O)Cc1ccccc1Cl N1(C(C(N2CC(NC(C(C(CC)(C)C)O)=O)C2)=O)C)C(=O)c2ccccc2C1=O Cc1csc(C)c1C(=O)NCc1cc[nH]c1C(=O)NCc1ccccc1O C1(O)(CN(C)C(c2cccs2)=O)CN(C(c2cn(C3CCC3)nn2)=O)C1 Cc1c(C(=O)N=c2nn[nH]n2CC(C)C)cc(C(F)(F)F)cc1[N+](=O)[O-] O=C(CC1CCc2ccc(O)cc21)NC1(Cc2ccccc2)CCCC1 CC1(O)CC(CNC(=O)CCC2CCN(C(=O)CC3CCOC3=O)C2)C1 C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(=O)COCCF)C)C1 N1(C(C2CC2(Cl)Cl)=O)CCCC(n2cc(C(c3cccnc3)O)nn2)C1 N1(C(CC=C)=O)CC(NC(c2ccc(=O)n(CCOC)n2)=O)CC12CCOC2 C1(C(N(C)Cc2nnnn2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 CC1CCCN(C(=O)C(=O)NC(C)CCNC(=O)CCOCC2CCC2)C1 c1(C(C)(C)C)ocnc1C(=O)NC1CCC1CNC(=O)CC1CC2(CC2)C1 C(=O)(C(F)C(C)C(F)(F)F)NC(C)CCNC(=O)CC(C(F)F)n1ccnc1 CC1(C)CC(C(=O)NCC23CC2CN(C(C2CCCO2)=O)C3)CC(C)(C)S1(=O)=O CC1=C(CNC(=O)NCc2cccc3c2CCCC3)C(C)(C)CCC1 N1(C(c2cccc(NCC)c2)=O)CC(C)(C)CC1CNC(=O)C(CC)OC N1(CC(=O)NCCCC(C)NC(=O)Cc2nc[nH]n2)CCn2nccc21 Cn1ccc2ccc(C(=O)NCC3C4CN(Cc5cccnc5Cl)CC34)cc12 CC1(C)CC(NC(c2ccc(C#N)cc2)=O)CN1C(=O)C=CI C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCCC(C)NC(c1ccn(C(F)F)n1)=O c1(NC(C2CCC(C)N2Cc2cnc(Cl)s2)=O)cccc2c1C(=O)CC2 C12(NC(c3c(CC)nc[nH]3)=O)CCOCC1CN(C(C1CC(OC)C1)=O)C2 c1(CC)cccnc1C(=O)NCC1(NC(=O)CC2C=CCC2)CCCC1 Cc1sc(S(=O)(=O)NC(c2ccc(OC(C)C)nc2)=O)cc1[N+](=O)[O-] C=CCC(CO)NC(C12CC(NC(=O)CCC3CCC(C)O3)(C1)C2)=O c1(C(=O)NC(CNC(CS(CC)=O)=O)C(C)(C)C)cnn2c(N)cc(C)nc12 c1(C(=O)NCCOCCC(=O)N(C)CC2(C)CCC2)cccc(=O)o1 CC(C)CC(C(=O)N1CCCC(N(C)C(c2coc(C(F)F)c2)=O)CC1)N(C)C C=CCCC(C(=O)NCC1CC1C(N)=O)NC(C1CCCC(C(=O)OC)C1)=O c1(CN=C(NC2CCCN(C(C(C)C)=O)C2)NC2CC2)cc(Cl)ccc1Cl c1(CC(N2CC(NC(C3(CCF)CCC3)=O)C(O)C2)=O)noc2ccccc12 C1(C)(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)CC(C2CC2)=NO1 N1(C(Cc2c(C)nc(SCC)s2)=O)CCN(C(=O)COc2cnn(C)c2)C(C)C1 C1(CC(=O)N(CC(CC)NC(=O)Cc2cc(C)sc2C)C)CCCC2(CC2)C1 N1(C(C2C(C)(C)OCC2)=O)CCOCC(NC(=O)C(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1CNc2ccccc21)NCCCNC(C1Cc2n(C)nnc2CC1)=O c1(OCCC(=O)NC(C)CN(C)C(c2ccc(C(C)(C)C)s2)=O)ccc(Cl)cc1 C1(C(=O)NC(C)CC2CN(C(=O)CSCCC#N)C2)C=CC=CC=C1 O(NC(=O)C(C1(C)CC1)NC(C1CCO1)=O)C(CC)CC C#Cc1cccc(CN(C2CN(C(=O)OC(C)(C)C)CCC2F)C=O)c1 N1(C(CC(C)SC)=O)CC2(CCCC2)C1C(N1CCC(CO)C(C)C1)=O C(=O)(CC(C)(C)CNC(=O)CC1CCCOC1)N1CCN(CC(C)C)CC1 Cc1nn(C)cc1-c1cn(CC(O)CCC2CCC(=O)NC2)nn1 C1(C(N(C(CC)C(=O)OC)C)=O)C=CCN(C(=O)CCc2nc(C)no2)C1 Cc1nc(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)c(C)o1 Cc1cnc2n1CCC(C(=O)NCC13CC(NC(=O)CSCCC)(CCO1)C3)C2 C=CC1(C(=O)N(CCC(=O)OCC)C)CCN(C(C2C=CCS2)=O)C1 S(=O)(=O)(c1ccc(NC2CN(C)C2)cc1Cl)NC1C(CC)CN(C)C1 Cc1cccc(NC(C2CC23CCN(C(c2ccccc2Br)=O)C3)=O)c1[N+](=O)[O-] Cc1cc(C(=O)N(C)CC2(NC(C3CNC(=O)CC3C)=O)CC2)c2c(c1)CCO2 c1(CC(N2CC(N(C(=O)CC34CCCC3C4)C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(c1n[nH]cc1Cl)=O CC(C)(F)C(C)(F)C(=O)NCC1CN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(C(N(CCCNC(=O)C(C)(F)CC2CCCC2)C)=O)cc(Cl)c(F)cc1F c1(CC(CNC(=O)C(C2CC2)N(C)C)NC(=O)CNC(=O)C2CC2)ccccc1 c1(CC(=O)N(CCCNC(=O)CC2CC23CC3)CCO)ccccc1O c1(C(N(CC)CC2CCN(C(c3ncoc3C)=O)CC2)=O)cccc(=S)n1O c1(COCCOCCC#C)noc(-c2ccn(CC(=O)O)n2)n1 N1(C(CCCOCCC)=O)CCC12CN(C(=O)CC1COCC(C)(C)O1)C2 CC(CC(Cl)Cl)NC(c1sccc1-c1nn[nH]n1)=O C(=O)(C(F)(F)CCn1cccn1)NC(CC(C)NC(C(C1CC1)OC)=O)C n1(CCNCCC(c2nn[nH]n2)NC(c2cc(C)oc2C)=O)cnc2ccccc12 C#CCCCCCC(=O)NCC(C1CCCC1)NC(=O)CC1COCC(C)(C)O1 CC(C(C)(C)C)NC(=O)CN(C(=O)CC1CCC1)C1CCC1 c1(C(C)C(=O)NC2CCCC(NC(C34CC(CO3)C4)=O)C2)c(F)cccc1F Nc1ccc(C=O)nc1N.N1(N2C(C(=O)OCC)CCCC2)CCS(=O)(=O)CC1 Cc1ccc2c(C(=O)NC3CCCN(C(c4nnccc4C)=O)C3C)coc2c1 N1(C(=O)CCOCC2CC2)CCC(NC(C2(F)CCCCC2)=O)C(F)C1 CC1=CCC(C)(C(=O)NC(C2CN(C(=O)C(C)N3CCC3)C2)C)CC1 CC1COCC(CC(N2CC(=O)CC2C(=O)NOCCOCCO)=O)O1 C(c1cnn(C)c1C)=CC(=O)NC1C(NC(c2scc(C)c2C)=O)CCC1 CC1(CNC(=O)C=CCO)CCC(NC(C23CCC(CC2)C3)=O)C1 C(C1=NOC2CN(C(=O)C3=CCCOCC3)CC12)NC(c1cc(C)nc(O)c1)=O n1(CC(=O)NC(C(=O)NCC(F)(F)Cl)C2CC2)cccn1 N1(C(c2ccc(Cl)c(Cl)c2)C(=O)NCC=C)CCCC(C2CCCC2)C1 C(=O)(CC(CNC(=O)CC1CCOC1C)C1CCC1)NCC(c1ccsc1)C N1(C(C(CC)C(C)O)=O)CCCN(C(c2cc(C)cs2)=O)CCC1 N1(c2nc(OCC)c(C)cn2)C2CCC1CC(NC(=O)CCCC(N)=O)C2 C#CCC(O)C(=O)NC1CCC(CC=CC(=O)NCCC2(OC)CCC2)C1 C(=O)(C(C)(O)C(C)(C)C)NC1CCN(C(c2cnc(CCCC)s2)=O)CC1 CCCCC(O)C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cnccn2)cn1 c1(C(=O)NC(C2C(C(=O)Nc3cnc(C)nc3)C2)C)c[nH]c(=N)c(C)c1 C=C(Cl)CCC(=O)NCc1ncccc1CNC(c1cccnn1)=O c1(C(c2n(C3(C)CC3)nnn2)NCCc2ccsc2)cnn2c1CCC2 c1(C(N2CC(C(=O)NCCNC(C(C)C#N)=O)C2)=O)cn(C)c(=O)n(C)c1=O c1(C(N(CCOCCNC(CS(C(C)C)(=O)=O)=O)C)=O)ccc2oc(=O)oc2c1 C1(NC(C2N(C)CCC2)=O)CN(C(=O)CCn2cnc([N+](=O)[O-])c2)CC12CC2 C1(CCCC)CCCN(C(C2C(C)CN2C(=O)CCC)=O)C1 CC(C)(CNC(c1ccc(Br)cc1)=O)CCNC(=O)Cc1cocn1 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CNC(c3snc(O)c3Cl)=O)c12 N(C(=NCCF)NCC(c1ccccc1)N1CCCC1)C(C)C1CC1 C(=O)(C(=O)C(C)(C)C)N(C)CC1CCN(C(c2c(CC)ncs2)=O)C1 c1(OC)ccc(F)cc1C(=O)NC1CC(NC(c2cn(C)nc2C2CCC2)=O)C1 C1(C(C(=O)Nc2cn(CCC)nc2)C)CCCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2C(NC(=O)CN(CCO)CCO)CCOC2)ccc2ccccc2n1 c1(C(N(CCN(C)CCO)C(C2CC3CC3C2)=O)=O)ccc(-c2cnn(C)c2)cc1 CC(C(=O)NCc1cc(C(N2CC(C)OCC2C)=O)co1)C(C)(C)C c1(OC)c(NC(C2(C)CCN2C(c2cc(OC)ccc2Cl)=O)=O)cccc1C#N N1(c2n(CC(C)C)c(-c3cscc3F)nn2)CC2CCC1C(CO)C2 N1(C(c2c(C)snc2)=O)CCCCC1C(C)NC(c1csc(-c2nc[nH]n2)n1)=O C12(NC(CS(CC)=O)=O)CCC(CNC(=O)CC3OCCO3)(CC1)OC2 CCCN=C(NCc1nnc(CO)s1)NCC(c1ccncc1)O C(CC(F)(F)F)(c1ccccc1)SCC(=O)Nc1ccc(Br)s1 c1(-c2n(-c3cccc(CC)c3)nc(CCN(C)C)n2)n[nH]c2c1COCC2 N1(CC(=O)NC(C)C(=O)NC2(CN(C)C)CCCC2)CCC(O)CC1 CC1CN(C(c2ccc(Cl)nc2N)=O)CCN1C(c1ccc(C(F)F)c(F)c1)=O C=CCCCCCC(=O)NCCCN(C(c1ncc(C(=O)OC)s1)=O)CC Cn1nnc2cc(C(N3CC(O)CC3C(=O)NCC3CCC3)=O)ccc12 N1(C(C2CC(C)SCC2)=O)CCC(C(=O)N2CC3(COC(=O)C3)C2)=C(F)C1 C(N=c1[nH]cnc2[nH]ccc12)C1CC(NC(=O)C2=CC3CCCCCC23)C1 Cc1ccc(C(N2CC(NC(C3CNC(=O)C3)=O)C3(CCC3)C2)=O)c(N)c1Cl C1(C(=O)NC(C)C(C)(C)NC(c2ccc(O)c(C(N)=O)c2)=O)CC2(CCC2O)C1 c1(C(=O)NCC(CC)NC(c2cccc(CO)n2)=O)cc(NS(C)=O)ccc1F C(=O)(C1CCCc2scnc21)N(C)CC1CN(C(=O)Cn2nnc(=O)[nH]2)CCO1 N1(C(c2cccc(F)n2)C(=O)Nc2ccc(OC)cc2C)CCS(=O)CC(C)C1 N1(C(C23C(CN(C(C(C4CC4)OCC)=O)C2)C3)=O)CCn2nc(C)cc2C1 C(C(C(=O)Nc1cccn2ncnc12)C(C)(C)C)NC(CCC#C)=O N1(C(C(Cc2ccc(C)cc2)C)=O)CCC2CCC(NC(=O)CC3CC3)C12 C=CCC(CC(C)C)C(=O)NC1CN(C(c2cc[n+]([O-])cc2)=O)C2(CCCC2)C1 Cc1cc2cccc(C(N3CCCC(O)(CN=c4[nH]nc(O)s4)C3)=O)c2s1 C(=O)(CCCSC)N(C1CCN(C(=O)CC(O)C2CC2)C1)CC#C N1(C(C(C)(C)C#N)=O)CC2CCC1C(NC(=O)CC1CC(=O)NC1=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)NC1CC(CNC(c2c(C)cnn2C)=O)C1 c1(C(=O)OC)cc2ccccn2c1CN(c1ccn(C(C)C)n1)CC1CCCO1 CCC(C(=O)NCCNC(C1CCCC1O)=O)NC(=O)COC1CCCOC1 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1OCC(CNC(C#CC2(C)CC2)=O)C1 N1(C(C(C)C2CC2)=O)CC(N=[N+]=[N-])CC1C(N1CCC2CC12)=O Cc1nc(SCC(=O)NC(c2ccc[n+]([O-])c2)C)c(C#N)c(C)c1C N1(C(C(C)OCC#C)=O)CCCC2(C1)CN(C(=O)Cc1cccc3c1CCC3)C2 c1(C(=O)NCC(CC)NC(c2csc(C3CCCO3)n2)=O)cccc([N+](=O)[O-])c1 c1(OC)nccnc1NC(=O)CC1CCCN1C(=O)COCCSC C1(NC(CC(C)C(F)(F)F)=O)CN(C(=O)CN2CC3CC3C2)CCC12CCOCC2 CCC(CCCC(=O)NCC=CC(C)(C)C)NC(=O)C(F)C(C)(F)F N1(C(C)=O)CC(CNc2ccnn2NC(=O)C(C)(O)Cc2ccccc2)C(C)C1 c1(Sc2nccc(C)n2)ccc(C(F)(F)F)cc1S(=O)(=O)NCCN(C)C C(=O)(CCCOC(C)C)N(CCC(=O)NC(C(=O)NCCC)C)CC.C1CC1 c1(C(N2C(C(=O)NCCOCCC)CCC2)=O)cccc2c(Cl)cccc12 c1(C(=O)NC(CN(C(=O)C(c2cnccn2)C)CC)C)c[nH]c2c(F)cccc12 CC#CCCCC(=O)N1CC(OC2CCN(C(=O)C(C)(C(C)C)OC)CC2)C1 CCCC(O)CC(=O)N1CCC(CN(C)C(C2(C#N)CC3CC3C2)=O)CC1 C1(CNC(C(CN(C)C)NC(Cc2c(CC)con2)=O)=O)COCC1(C)C N1(C(Cn2ccc(C)n2)=O)CC2C(CNC(=O)CC(O)C3CCCC3)C2C1 C(=O)(C(O)CC(C)(C)C)N1CC2C(CNC(C3N(C)CCCC3)=O)(C2)C1 c1(C(=O)NCC2(NC(c3csc(Cl)c3)=O)CCC2)cnc(C2CCOCC2)nc1 c1(C(=O)NC(CC2CN(C(c3c(C)nns3)=O)C2)C)nnn(C2CC2)c1C(F)F N1(C(c2c(N(C)C)ccnc2)=O)CC(C2CN(C(C3CC(N(C)C)C3)=O)C2)C1 c1(N(CC(C2CCOC2)O)C)cc(Br)ccc1S(=O)(=O)NC12CCC(CC1)CC2 C1(C(N2CC(N(C)C(C3CC(CF)C3)=O)C2)=O)CCCCCS1(=O)=O c1(C(=O)NC(c2ccc(Br)cc2)C#C)ccnc2ccc(Cl)cc12 C(=O)(C(CCC1CC1)NC(C1CC12CC2)=O)NC1CC(NCC(N)=O)C1 c1(SC)cn(-c2ncc(CN3CCCC3)s2)nn1.N12CCC1C2=O N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C2CC2)(NC(=O)Nc2ccsc2)C1 C1(CCNC(c2c(C)nsc2)=O)CN(C(C2CC3CC2C3)=O)CCO1 N1(C(C2(CCC=C)CC2)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C2(CCC2)C1 c1(C(=O)NCC(CNC(C(COC)(C)OC)=O)(C)F)cccc2cn(C)nc12 N1(C(C(C)(C)C2CCN(C(c3ccnc(O)c3F)=O)C2)=O)CCC2(C1)CC2(F)F C1(C(=O)NC(C(CC)C)CN(C)C)CCN(C(=O)Cn2ncnn2)C(C)(C)C1 Cc1ncc(C(=O)NCC(C2CCC2)NC(=O)Cc2cccc(O)c2)n1C(F)F c1(C(N(C(CNC(C(C)OCCC=C)=O)C)CC)=O)cn(-c2ccccc2)cn1 C(=O)(C1CCCc2nncn21)NCCCCCNC(=O)C(F)C(F)(F)F c1(C(=O)NCC(CN(C)C(C2CCC([N+](=O)[O-])CC2)=O)O)n[nH]c2cccnc12 C(=O)(CCC(C)(C)F)N1CC(OC2CCN(C(C3C(C=C)C3)=O)CC2)C1 C(C(=O)NCc1cnco1)(C(C)(C)O)NC(CNC(CC)=O)=O C(=O)(C(CNC(=O)CC1(O)CCCC1)CC1CCCC1)NCC(C(C)O)C c1(C(=O)NCC(C)NC(C(CC)N(C)C)=O)cnn(-c2ccccc2)c1Cl N1(C(c2c(C)nco2)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)C(F)(F)C1 N1(C(COC)=O)CCCC1(C)CNC(c1ncoc1-c1ccc(F)cc1)=O C1(NC(CCN(CC)CC)=O)CC(O)CN(C(c2nc(OC)cc(OC)n2)=O)C1 C1(C(N2CCC(NC(CC(=C)C)=O)C2c2ccccc2)=O)CC(C2CC2)=NO1 c1(C(N(CC)CC2CC2)C)cc(OC)c(Br)cn1 n1(NC(c2ccc(F)cc2F)CC(N)=O)ncc2c(O)ncnc12 CCC(CC(=O)NCCOCCCN(C(=O)CCNc1ccccn1)C)C1CC1 CN1CCN(C(C2CCCC2NCc2ccc(Cl)nn2)=O)C(CO)C1 n1(CC)nc(SCC(=O)OCCNC(C)C)c(Br)n1 C1(NC(c2nc(C)oc2)=O)CC(F)CN(C(c2cnn(C3CCC3)c2C)=O)C1 N1(C(=O)NC2C(CC)CCN2C(=O)CC(C)C(F)F)CCN(C)CC(C)C1 N1(C(C2CCCN(CC)C2)=O)CCC(C2(NC(c3ncc[nH]c3=O)=O)CC2)CC1 C1(C(=O)NCCOC(C)=O)CCCCCC1NC(C12CCCC1C2(F)F)=O N1(C(C2CC(OCC)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1C c1(NC(CCN(C(COC)=O)CC2CCCC2)=O)n[nH]c2ccccc12 c1(C(=O)NCC(N(C(CC=C)=O)C)C2CC2)c[nH]c2nccc(Cl)c12 N1(C(C2C(C)(C(C)C)C2)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC(C)C1 CC1(CNC(=O)CC(O)CNC(c2nc[nH]n2)=O)CCCC(=O)N1 Cc1cc(C)c(C(=O)NC2CCCN(C(c3c[nH]cc3Br)=O)C2)c(O)c1 N1(C(C2=C(C)CCC2)=O)CC2OCC(NC(=O)C(CCO)N(C)C)C2C1 CC1c2cccnc2CCN1C(=O)NC1CCN(c2ccnc(Cl)n2)CC1 C1(OC)(OC)CCC1C(=O)NCC1CCC1NC(C1CCN(C)C1)=O C1(CC)COCCN(C(=O)C(O)C2CN(C(C3CC4CCC(C3)O4)=O)C2)C1 c1(C(N2C(C)CC(CNC(c3cncc(N)n3)=O)C2)=O)coc2ccc(Cl)cc12 C1(CNC(C(C)OCC(C)C)=O)CN(C)CCN1C(c1cn2c(n1)CCC2)=O C(=O)(CCC(N)=O)NCCOCCCNC(C1(CC#C)CCCC1)=O c1(C(=O)NC(C)CNC(C2CCN2C2CCCC2)=O)cnc(O)n(C2CC2)c1=O C1(C(CO)NC(c2ccccn2)=O)CCN(C(=O)C(F)n2ccnc2)CC1 O=C(CCCCCF)NC1CCCC(C(N2CCC3(CCC3)C2)=O)CC1 N1(C(C=NOC)=O)CC2CCN(C(c3cccc(F)c3Cl)=O)C2C1 C#CCCCC(C)C(=O)N1CC=CCC1C(N1CCC(CN(C)C)C1)=O C(=O)(C(O)Cc1ccccn1)N(C1CC(NC(=O)C=CC(=O)NC2CC2)C1)C C1(NC(c2c(OCC)c(F)ccc2)=O)CN(C(c2cnccn2)=O)CC12CCC2 C(CCC(C)(C)C(=O)NCC1(C)CC2(CC2)C1)NC(CC1C(C)CCO1)=O C=CC(C(=O)N1CC(O)(C(F)C(=O)NC(CC)C2CC2)C1)OC CC(C)CCCCCC(=O)N1CCC(C)C(NC(=O)CCSc2ccccn2)C1 C1(C(=O)NC(C2CCN(C(CCn3c(C)ncc3)=O)C2)(C)C)CCCC(=O)N1C C1(C#N)(CNC(C2C(NC(C(C3CCC3)OCC)=O)CCCC2)=O)CC(C)(C)C1 c1(C(=O)NCCCN(C)C(C2CCC3CCCCN23)=O)ccc(S(N)(=O)=O)s1 c1(C(N2C(CNC(c3cc(COC)cn3C)=O)CCC2)=O)cn2cccnc2n1 c1(OC)ccc2cc(CC(N3CCCC(C(=O)NC4CCOC4)C3)=O)ccc2c1 N1(C(C2C(COC)C2)=O)CCC(C)(NC(c2sc(C3CCCO3)nc2C)=O)CC1 Cn1ccc(C(C)(C)C(=O)NCC(C)(C)CNC(c2ccc(Cl)o2)=O)n1 C=C(C)C(CC(=O)N(CCC(=O)NC1CCCCC1(C)C)C1CC1)OCC c1(OC)cc(CN2CCC(NC(c3ccc(OC)c(I)c3)=O)CC2)ccc1O C1(CNC(c2cc(CNC(CNC(C3C(C)C3)=O)=O)sc2)=O)CCC2(CC1)CC2 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(F)s3)=O)C2)nc1C C1(CCNC(c2c(C)onc2)=O)CCN(C(=O)CCCCC(C)C)CCC1(F)F c1(C(=O)NCC(CNC(c2cccc(OC(C)C)n2)=O)C)nc2c(s1)CCCC2 C(=O)(CCP(C)(C)=O)N1CC(C)C(CCNC(c2sccc2CO)=O)C1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC(CNC(=O)COC(C)C)CC1C N1(C(C2C(CC)N(C(C3CCCC4CC34)=O)CC2)=O)CC(N(C)C)C2(CC2)C1 CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2cn[nH]c2)CCC1 c1(C(=O)NCCOCCCC#C)c(CNC(C2(C)CCC(C)C2)=O)cnn1C c1(C(=O)NCCCOC2CCN(C(CC(C)F)=O)CC2)cnc2sccn12 C(C(CC(C)C)NC(C1(C)CCN(C)C1)=O)NC(COCC)=O CCCC(C#N)C(=O)NC1C2CC3C1C3C2C(=O)N(C1CS(=O)(=O)C1(C)C)C C1(c2ccccc2)(NC(CCOC)=O)CCN(C(c2c[nH]cc(C)c2=O)=O)CC1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc([N+](=O)[O-])ccc1N(C)C CC(C)S(=O)(=O)C(C)C(=O)NC1COC2C(NC(=O)C(O)C(F)(F)F)COC12 C(C(CNC(=O)C=Cc1cn[nH]c1)C(F)(F)F)NC(c1c(C#N)csc1)=O N1(C(CC2CN(C(C)=O)C2)=O)CCCC(F)(C(=O)NC(C)(C)CCCF)C1 C#Cc1ccnc(C(=O)NCC2(NC(=O)C=Cc3nccs3)CCCCC2C)c1 C#CCCCC(C)C(=O)N1CCCC(F)(CNC(C)=O)C1 c1(C(N(CCN(C(C=C(C)C(C)C)=O)C)C)=O)cc(F)cc(C)c1N N1(C(C2(CC)CCN(C(=O)CCc3ccncc3)C2)=O)CC2CSCC2(C)C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C(NC(c2ccnn2C)=O)C1 N1(CCCC)CCOCC1C(=O)NCCCC(C)NC(c1cnoc1C(C)C)=O c12cn(nn1)C2.N1(C(=O)NCC2CC(CN)C2)CCCC1CC(N)=O C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 c1(C(N2CCC(C)(N)C2)=O)ccc(F)c(F)c1.Cc1ccccc1CC1(C)CC1 Cc1nccc(CNC(C2(CNC(=O)CCCF)CC(C)(C)C2)=O)n1 N1(C(C2N(C(c3c(O)ccc(C)c3)=O)C3C(C2)C3)=O)CC2CCCC(C1)N2C C1(C(=O)NC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)CCC(C)(F)CC1 C(=O)(C(C)CC(C)C(C)=O)NCc1c(C(=O)NCC(CCCC)O)n(C)nn1 C1(NC(CN(C(C(C)C)=O)C)=O)CCCC(CNC(=O)C(=Cc2cccs2)C)C1 c1(CC)oc(C(N2CCCC2c2ccc(OC)cc2)=O)cc1C(=O)OC N#Cc1c(F)c(NCC2CCCN2CC(F)F)nc(F)c1F CC(O)CCCC(=O)N1CC(N(C(=O)Cc2cccc(O)c2F)C)C1 C1(COC)(CNC(C2CC3(CC3)CO2)=O)CCCN1C(=O)C=Cc1cc(C)no1 CCC(C)(C)CC(=O)N(C(C)CNC(C12COC(C1)C2)=O)C N1(C(C(CC=C)OC)=O)CCCN(C(c2cccn3ccnc23)=O)C(C)C1 N1(C(C(CC(C)C)OC)=O)CCC2CCCC(C1)N2C(c1cncnc1C)=O N1(C(c2ccc(OC)cn2)=O)CCC2(CC1)COC(CNC(=O)CS(C)(=O)=O)C2 c1(N(C(CC(=O)OCC)(C)C)C)cc(C)nc(S(C)(=O)=O)n1 c1(-c2cc(O)ncc2)nncc2ccoc12 N#Cc1cc(NC2CC(F)CN(C(c3cc(C4CC4)on3)=O)C2)ncn1 C12(NC(CC(=O)NCC#C)=O)CCCC1N(C(c1ccc(Br)cn1)=O)CC2 C=C(C)C(C)(C)C(=O)NCC1CC(C(F)(F)F)CN1C(C1COCCO1)=O Cc1cc(Br)cc(S(=O)(=O)NC2CC3CC2CN3C(c2ccncc2)=O)c1 N1(C(CCS(C)=O)=O)CCC(NC(=O)Cn2ncc3ncccc23)C12CCC2 C(=O)(CCCCN(C)C)NCC(CO)NC(C(c1ccccc1Cl)OC)=O C(CC(C)(C)C)(C(=O)N(CCCCCC(=O)N(C1CCC1)C)C)OC C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)N(CCNC(=O)C(C)CC#N)CC C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)CC1)=O)Nc1c(OC)ccc(C)c1 CCCCCC(O)C(=O)NC(CNC(=O)C(c1cnn(C)c1)C)(CC)CC N1(C(CCC(C)C#N)=O)CCC2C(C1)CN2C(=O)CCc1ccc(Cl)c(Cl)c1 Cc1cc2occ(C(=O)NC3CCCC3NC(C3CCNC(=O)C3)=O)c2cc1C N1(C(C2C(C)C2)=O)CC2CN(C(c3nc(C4CC4)ncc3Cl)=O)CCC12 N1(CC(C)(O)C2(NCCC=CC)CC2)CCCC(C(N)=O)C1 C1(N(C(C(=O)NCCOC)C2CC2)CCC)CCCC1 C1(CNC(c2ccc(OCCO)cc2)=O)(NC(C2CC2(F)Cl)=O)CCCCCC1 c1(N2CCN(CNc3cc4c(nc3)C(=O)NC4)CC2)ncnc2cccc(F)c12 Cc1c(C(N2CCC(NC(=O)CC3CCC3)C(CO)CC2)=O)nn2ccccc12 C1(C(N2C(CC=C)(C(=O)NC34CCN(CC3)C4)CCC2)=O)CC2(CCO1)CC2 C(C(C)(CC(C)C)NC(=O)C(O)Cc1cccc(Cl)c1)NC(CCC=CC)=O C1(C)(C(=O)NC(C)CCCNC(c2c[nH]ccc2=N)=O)Cc2ccccc2C1 N1(C(CC=CCCCCC)=O)CC2CCC(CNC(c3cscc3C)=O)C2C1 C1(C(=O)NC2CCC(N(C(CC3CCN(C)C3)=O)C)CC2)CN(CP(C)(C)=O)C1 CC(C)CC(C(=O)NCC1CSC1)NC(=O)C1=CCCC1 c1(C(=O)NC(C(C)(C)C)c2cccs2)ccc(-n2cccn2)c(F)c1 CC1CC1C1CC1C(=O)NC1CN(C(=O)Cn2ccc(=N)[nH]2)CC1C c1(C(=O)NCC2CC(NC(C(C)OCOC)=O)C2)coc2cc(F)cc(F)c12 CN1CC(C)(C(=O)NCC(C)(C)NC(C2C(C(F)F)C2(C)C)=O)CCC1=O C(=O)(CC(C(C)C)NC(=O)Cc1ccoc1)NC(CCC)CCC C1(C(=O)NCCN(CCCC)C)COCC1NC(=O)CNC(C)=O C1(C2CCN(C(C3CNc4ccnn4C3)=O)C2)(NC(C2CCCC(O)C2)=O)CC1 c1(C(N(CCCNC(=O)C(F)CC2CCC2)CC)=O)[nH]c2c(C)cccc2c1C c1(CC)[nH]ccc1C(N1CC(CNC(=O)C(C)c2ccco2)(OC)C1)=O C1(NC(c2ccc(CO)cc2F)=O)CCN(C(=O)Cn2cccn2)CCC1(F)F c1(C(=O)NCC2C(NC(C3(C)C(CC)CCC3)=O)CCC2)cc(C)ccc1C c1(N(c2ccc(C(C)C)cc2)C(C)=O)ccc(C#N)cn1.c12c(csc1C)NC2 c1(CNC(CCN(CC#C)C(C2CCCS2)=O)=O)nn(C)cc1CO c1(C(=O)NCC2C(CNC(CCC=CC)=O)C2)cn(C)nc1COC n1(CCC(=O)NC2CC2NC(=O)C(C2CCCCC2)O)nc2ccccn2c1=O CC#CCC(C(=O)NC(C)C(=O)NCC)NC(c1cn(C)nc1CC)=O Cc1cc(C)c(C(N2C3CC2CN(Cc2ccc(Cl)cn2)C3)=O)cc1C N1(C(CCc2onc(CC)n2)=O)CCCN(C(c2coc3c2COC3)=O)CC1C C1(NC(c2ccc(CO)cc2F)=O)CC2CCC1N2C(=O)CC1CCCCCC1 c1(-c2n(C)ncc2CNC(=O)NC2(C)COCCC2C(=O)O)cc(O)nc(O)n1 C1(NC(C2C(C(C)C)CCC2)=O)CN(C(=O)C=CCOC(C)(C)C)CC(C)(C)C1 N1(C(C(C(C)CNC(=O)Cn2nnc(C3CC3)n2)F)=O)CC=C(C(C)(C)C)CC1 CC(C)C(C(=O)NCCOCCNC(=O)C(C)c1cccs1)c1cccc(Cl)c1 C1(CNC(=O)C=Cc2cccnc2)CCCCCN1C(C1(F)CCOC1)=O N1(C(CCC(C)O)=O)CCCC12CCN(C(c1cc3ncccc3s1)=O)C2 CCC(C)CCCC(=O)NCC1(CC(=O)NCC(O)C(C)C)CC1 C12(NC(Cc3c(C)cco3)=O)CCN(C(c3cnn(CCO)c3N)=O)CC1C2 N1(C(C=C=C(C)C)=O)C2CCC(C2)C1CNC(C1CC(C)(O)C1)=O C1(NC(CC2(C=C)CC2)=O)CCC(C)N(C(=O)CN2CCOC2=O)C1 c1(C(=O)NCC(C)C(=O)NC2CCCCC2C#N)c[nH]nc1[N+](=O)[O-] c1(OC)ccc2cc(C(=O)NCC(F)CNC(C3CCN(C)C3=O)=O)ccc2n1 CC1(C2CN(C(=O)CC3COCCN3C(c3ccsc3C#N)=O)CCO2)N=N1 c1(C(N2CC(NC(c3ccc(NC)cn3)=O)C(C)C2)=O)c[nH]cc(C)c1=O c1(C(N2CC(C)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 Cc1cccn2nc(C(N3CCCC(C)(NC(c4ncncc4Cl)=O)C3)=O)cc12 c1(CNC2C(C(N3CCOCC3CO)=O)C2)cnc2ccccc2n1 c1(CC)cc(F)ccc1C(N1CCC(O)C(NC(c2cscc2OC)=O)C1)=O CC1Cn2nc(C(N3CCCC(N(C)C(C4CC=CC4)=O)CC3)=O)cc2C(=O)N1 CN1CCN(C(=O)CCCN=[N+]=[N-])CC1CNC(=O)C(C1(O)CCCCC1)(F)F c1(C(N2CC=C(CNC(=O)C=C(Cl)Cl)CC2)=O)ccc2c(n1)COCC2 c1(NC(=O)CC2CN(C(C3CC3C(=O)O)=O)C2)nnc(Br)s1 c1(C(N2CC(O)(CN(C(C=C(CC)C)=O)C)C2)=O)cncnc1C C(=O)(C1CCCc2scnc21)NCCCNC(C1N(C)S(=O)(=O)CC1)=O CCC(CC(=O)NCCCOCCC(=O)NCC(=O)NC(C)C)SC c1(C(=O)OC)c(NC(c2sc(NC(=O)CCCCN)nc2C)=O)sc(C)c1C N1(C(CNC(CC)=O)=O)CC=C(C(=O)NCC2CCOC(CC)C2)C1 N1(C(c2n(C)cc(Cl)c2)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C(C(N)=O)C1 C(=O)(C1=CCCCO1)NS(N)(=O)=O.O=C1CC2CC2C1.N12CCOC(C1)CC2=O c1(-n2c(C(C(C)C)NC(c3ccco3)CC)nnn2)ccccc1OC CC(c1ccccc1)=CC(=O)NC1CCC1CNC(=O)C(C)(C)C Oc1nc(-c2ccc(OCC3CCCCO3)c(F)c2)cc2nccn12 N1(C(C2(c3cccc(C)c3)CC2)=O)CC(CNC(C23CC2C3)=O)C2(CC2)C1 C1(NC(C(C=C)O)=O)CN(C(c2cnn(-c3ccncc3)c2)=O)C2CCCCC12 N1(C(C(CN(C(c2nn(CC)c(C)c2)=O)C)(C)C)=O)CCS(=O)CC1C C1(CNC(C(C)N(C(C2(F)CCOC2)=O)C2CC2)=O)CCCCCCC1 n1(C(C)C)ncc(C(=O)NCC2(NC(=O)C(c3ccc(Cl)s3)C)CCOC2)c1N N(C(=NCCC(C(F)(F)F)N1CCOCC1)NCc1cccs1)CCC(CC)C c1(C(N2CCC(C)(NC(CN3C(=O)CC(C)(C)O3)=O)C2)=O)cn2ncccc2n1 C1(C(=O)NC2CCC(NC(C3CC=CCO3)=O)C2)(OC)CCCCCC1 N1(C(c2cc(COC)on2)=O)CC2(CC2)CC1CNC(c1c(F)cccc1F)=O C1(CCNC(C(=O)NCC)=O)CCCN(C(=O)CCCOc2cccc(Cl)c2)C1 C(=O)(C1=C(C)CCCC1)NC12CC(NC(c3ccc(OC)c(N)c3)=O)(C1)C2 C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCC1)NC(c1cc(C)n(C2CC2)n1)=O N1(C(CCOC)=O)CC(C)C(NC(=O)CC2OCCCC2(C)C)C(C)C1 C1(CNC(COC(C)=O)=O)CCCC1C(=O)NCc1noc(C)n1 c1(OC)ccc(F)cc1S(=O)(=O)N1CC(CC(=O)Nc2c(Br)c(C)nn2C)C1 c1(C(=O)NC2(CO)CCCN(C(C(CC=C)C)=O)C2)cc(F)c(C(C)C)cc1F C=C(C)CCCC=O.CCC(C)(C)N Cc1csc(C)c1C(=O)NC1CC1CNC(=O)Cc1coc(C2CC2)n1 CN1CC(C(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)CCC1=O C1(OCCCC)CCC(C)N(N2CCn3ncc(S(C)(=O)=O)c3C2)C1 N1(C(C2(CC)CCCC2)=O)CC(OC)CC(NC(=O)C(C(C)(C)C)SC)C1 C1(OC)CC2CC(NC(C3(C(C)C)CCN(C(=O)C(O)CCSC)C3)=O)CC12 C1(O)(CNC(c2ccc(O)cc2)=O)CCCN(c2nccc(Br)n2)C1 c1(C(=O)NC2CCCN(C(C(C)P(C)(C)=O)=O)C2C)nc2ccccn2c1F C(C1CC(C)(C)Oc2ccccc21)NC(=NCC)NCCS(=O)(=O)CC1CCC1 CN1CC(NC(C2(C)C=CCN2C(c2nonc2N)=O)=O)C2(CC2)C1=O C1(N(CCCCOCC=C)C)CCN(C(=O)CNC(=O)CCCC)CC1 CC(C)C(C(=O)N1CC(CNC(c2ccoc2)=O)C(O)C1)c1ccccc1 c1(C(=O)NC2CC(CNC(=O)C3=CCOC3)C2)cn2c(n1)COCC2 N1(C(C2COCC(C)O2)=O)CC2CC1CN2C(=O)Cn1cccc(O)c1=O N1(C(C(C)=CC=C)=O)CC=CC(C(=O)NC(C2CCC2)C2CC2)C1 c1(C(=O)NC(CN(C(C2CN(S(CC)(=O)=O)C2)=O)C)CC)cccnc1 N1(C(C(CNC(=O)OC(C)(C)C)(C)C)=O)CC(NC(C2CC(O)C2)=O)C(C)(C)C1 CC(C)C(CO)C(=O)NC1CC(CNC(C2(O)CCOCC2)=O)C1 Cc1cccc(C)c1C(=O)NCC1CCCCN1C(c1cc(O)nn1C)=O C(C(=O)N1CCC(C)(NC(c2cnn(CCO)c2)=O)CC1)(C(C)(C)C)N(C)C C1(NC(Cc2c(C)con2)=O)(CO)CCCN(C(c2ccc(O)c(Cl)n2)=O)C1 C#CCCCCCCC(=O)N1CCN(C(=O)C#CC2CCCOC2)C(C(C)C)C1 Cc1c(C(N2CC=CC2C(=O)N(C)CC2CCC2)=O)ccn1C c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C)ccsc1Br c1(C(=O)NCC2CN(C(C3CC3F)=O)CCCO2)cc2n(n1)CCCO2 c1(C(N2CC(CC(C(=O)NCCC3(C)CCCO3)F)C2)=O)ccc2c(c1)CCC2 N1(C(C(CSC)(C)C)=O)CC2OCC(NC(C3COCCN3C)=O)C2C1 c1(NC(C2N(C(CCSC)=O)CC=C2)=O)cccc(-c2cncnc2)c1 C1(CC)CCN(C(=O)C(C)C#N)C1CNC(=O)Cc1cc(C)nn1C N#Cc1cccc(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCN2)=O)c1Cl c1(C(=O)OC2CC2)sccc1OC(F)F.C12CCC1NC(=O)N2 c1(C(N2C3CN(C(=O)CCOCC(F)(F)F)C(C3)C2)=O)cccc2nccnc12 O=C(C1=NOC2COCC12)NC1C=CCN(C(c2ccncc2F)=O)C1 CC(c1ccco1)=CC(=O)Oc1ccc(-c2nnc(Br)o2)cc1 C(=O)(C(C)CC(C)C(C)=O)NC(C(N1CCC(OCC#C)CC1)=O)c1ccco1 C1(C(=O)NC(C(=O)N(C)CC2CCSCC2)Cc2ccoc2)C(C)(C)C1(C)C CCCC(C)C(=O)NCCCN(C(=O)CC1CCCCC1C)C(C)C C=CC(C)C(=O)NCCN(C(=O)CC1CC(F)C1)C c1(OC(C)C(N2CCCC(COC(=O)C(N)=O)C2)=O)cccc(N)c1 S(=O)(=O)(c1ccc(F)cc1)N1C(CC(=O)Nc2cc(N3CC3)cc(Cl)n2)CCC1 N1(C(C(N2CC(C)C2)C)=O)CCC(C(=O)NCC(C)(O)C2(C)CC2)C(C)(C)C1 n1(CC)cc(C(=O)NCCCCN(C)C(c2coc(C)c2)=O)c(C)n1 c1(CC)cc(C(=O)NCC(=O)NCC(=O)NCc2cscn2)no1 N1(C(c2ccc(SC)o2)=O)CC2(CCCCN2C(c2nccn2C)=O)C1 C1(O)(C(C)NC(C(C=CCCC)O)=O)CCN(C(=O)CCc2cn[nH]c2)C1 c1(CC)ccnc(C(=O)NCC2CCCC(CNC(c3nnsc3C)=O)C2)c1 CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NCC1(C)CC1(C)C C1(C(=O)N(C)C)(NC(c2cscn2)=O)CC1(C)C.C12(CC1)N(C)C2=O c1(C(=O)NCC2N(C(CC=CC)=O)CCC2C2CC2)ncn2cc(Cl)ccc12 c1(CC)c(Cl)nc(C)[nH]c1=NCCCN(C(=O)C(C)(C)c1cncnc1)C1CC1 C=CCCCC(C(=O)NCCC(C)(O)CC)NC(c1cc(C)c(C)s1)=O C12(C(=O)NC(CNC(C(C(C)C)O)=O)C3CCC3)CCC(=O)N1CCS2 C1(NC(C2(CC)CCOCC2)=O)CCN(c2nc(C3CC3)ns2)C(C)C1 N1(C(C2(C)CC2(F)F)=O)CC(CNC(=O)C=CCN2CCC2)C2(CC2)C1 C1(CNC(CCOCCCOC)=O)CN(C(c2cc(C)nn2C)=O)CCO1 c1(C(=O)NC(CNC(COCCOCCOC)=O)C2CCC2)sc(=N)[nH]c1C C1(CC)CN(C(C2CCC3(CC2)CC3)=O)CCN1C(c1ccc(O)c(C)c1)=O C12(NC(c3cnn(CC)n3)=O)CCCC1N(C(=O)C=Cc1ccccn1)CC2 C1(O)(C(=O)NC2C(NC(C3CC(CC)(CC)C3)=O)CCC2)CCC(C)(C)CC1 C=C(C)CCCC(=O)N(C)C(c1cn(CC2(F)CCOC2)nn1)C CC(CC(=O)NC1(C)CC(NC(c2cn(CC3CCC3)nn2)=O)C1)C1CCCO1 c1(SC)c(C(=O)NCC(c2ccccc2)NC(=O)Cc2csc(Cl)c2)cnn1C C1(CNC(C2CC(C(=O)OC)C2)=O)CN(C)CCN1C(=O)CC1CCC(=O)NC1 C(=O)(CC(C)CC(=O)NC1CC(N(C(=O)CC(F)(F)Cl)C)C1)OC C(=O)(CC1=CCOCC1)NC(CC#C)(C)C(=O)N1CCSCC1CO Cc1c(Cl)ccnc1C(=O)NCC(C(C)(C)C)NC(C1(C)CC(C)(C)C1)=O N1(C(C2(S(C)(=O)=O)CC2)=O)CCN(C(C2CCn3cncc3C2)=O)C2CCCC12 c1(C(=O)NCC(C(C)(C)C)NC(C2CCC3CC2CO3)=O)ncn2c1CCC2 N1(C(CCCC2(C)NC(=O)NC2=O)=O)CC2(CCC(NC(C3CC3F)=O)CC2)C1 c1(C(N2CC(NC(=O)CCCC(F)(F)F)(CO)C2)=O)ccc2c(=O)cc[nH]c2c1 N1(C(C=CCCC(C)C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C2CCC2)C1 Cc1cc(C(=O)NC2CCCN(C(C3CCC3CF)=O)C2)cc(=O)n1C c1(NCC2CCN(C)CC2)ccc(S(=O)(=O)NCCCCC(F)F)cc1C#N N1(C(COC(C)=O)=O)CCCC(C(C)NC(c2sc(F)cc2Br)=O)C1 c1(N2CCC(F)(C(=O)OC)C2)ncnc2c1cnn2C(C)(C)C Cc1cc2ncn(-c3nnc(C4CC4)s3)c2cc1C C#CCCCC(C)C(=O)N1CCC1(C)CC(=O)NCC1CC(N(C)C)C1 C(=O)(C(CO)NC(=O)CCOCCNC(=O)CC1CN(C(C)=O)C1)NCC C(=O)(NNC(=O)c1cccnc1-c1ccncc1)N1C(C2CC(=O)NC2)CCC1 C12CCC(C)CC1C(=O)N2.n1(C(C)C)cnc(-c2nn[nH]n2)n1 C1(CNC(CCc2onc(CCC)n2)=O)CC(F)CN1C(C1CCOC1CC)=O C1(CC=C)(NC(c2cnc(C)s2)=O)CCN(C(C2CC(CC(C)C)C2)=O)C1 N1(C(Cc2nc(C(C)OC)sc2)=O)CC(C)C(C)(CO)C1 N1(CC(=O)N(CC(CNC(c2cnc(C)s2)=O)C)C)C(=O)NC(C)(C2CC2)C1=O C(=O)(CCCCC(=O)N(CCCNC(C1(OC(C)C)CCC1)=O)CCO)OC C1(CCC)C(=O)NCCN1C(=O)C=CCC(C)(C)NC(c1coc(CO)c1)=O c1(NC(C2CC=CCC2)C)ccc(S(=O)(=O)NCCn2cnnn2)cc1Br C1(C(CO)NC(c2scc(OC)c2)=O)CCN(C(C2CCCOC2C)=O)CC1 C#CCCCC(C)C(=O)NCC1CN(C(=O)C(C)OC(C)(C)C)CC1(F)F c1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CCC2)=O)ccc(SC(F)(F)F)cc1 C(CCNC(=O)CC(C)(F)F)(C(=O)NCC1COCC(C)O1)OC Cc1cc(C(c2nnnn2C2COC2)NCCc2ccnn2C)ccc1Cl N1(C(C(C=C)(F)F)=O)CC(O)(C2(CNC(=O)CN3CCC(OC)C3)CC2)C1 C1(C(=O)NC2(CO)CN(C(C(C)(C)C3CCC3)=O)C2)CCCC2(CCCCC2)C1 Cc1scnc1C(=O)N(C)CCOCCNC(c1cnn(-c2ccccc2)c1)=O N1(C(CCCSC)=O)CC(CNC(=O)CN2CC3C=CC2C3)C(C)C1 CC(C)C(C#N)C(=O)N1CCOCC(NC(=O)CCCOc2cccnc2)C1 N1(C(C2CC(C)(F)C2)=O)CC(NC(c2ccc(C(N)=O)o2)=O)C(n2cccn2)C1 c1(C(=O)NCC(CCCC)NC(=O)COC2CCC2)cc2c(cnn2C)nc1C N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2(COC)CC2)CC(C)(F)C1 C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(C1CCC(F)(F)CC1)=O c1(C(=O)NCC(C(C)(C)C)NC(C=CS(C)=O)=O)cnc2c(c1)OCC(=O)N2 C1(C(N2CCC(O)CC(C)C2)=O)(NC(=O)OC(C)(C)C)CC2(CCCCC2)C1 C1(CNC(C2C(CNC(c3c(C)ocn3)=O)CCC2)=O)CCC(CO)CC1 N1(C(C#CC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CCCc1cccnc1)C2 CC(C)C(O)C(C)C(=O)NCC=CCC(=O)NCC1(F)CCOCC1 c1(C(=O)NC(C2CN(C(C3CC(C)(F)C3)=O)C2)C)cscc1-c1ccccc1 c1(CNC(C(=O)N(C2CCOCC2)CCCC)=O)cnc(-c2ccccc2)s1 c1(C(c2noc(C(C)(C)C)n2)C)nnc(CCCc2cccn2C)o1 C12(CCNC(C=CCN(C)CC)=O)CCC1CN(C(=O)C(C)(C)n1cncn1)C2 c1(CSC)cc(C(=O)NCC(C)CN(C)C(C2(C#N)CC23CCC3)=O)ccc1F c1(C(=O)NCC(C2CCC2)NC(c2cc(F)cc(F)c2)=O)ccccc1[N+](=O)[O-] N1(C(C2CCOCC2C(=O)NOCc2ccccn2)=O)CCc2sccc2C1 N1(C(CC(CNC(C=C(C)c2ccccc2)=O)C)=O)CC2(C1)CC(C)(O)C2 N1(C(C)=O)CCCC(C2CN(C(c3cc(C)c(Br)cc3Cl)=O)C2)C1 C1(C(=O)NCC(=O)NCC#C)(OC)CCN(C(C2CN(C)CCO2)=O)C1 S(=O)(=O)(c1cccc(OC(F)(F)F)c1)N1CC(NC(C(C(C)C)O)=O)C(F)CC1 N1(C(COC(C)C)=O)CCCC1c1nc(C(=O)NC(C)Cc2cnccn2)cs1 N1(C(C2CCCCN2CC(F)F)=O)CCC(F)(F)CC1c1ccco1 c1(CNC2C(C(=O)NCc3onc(C)n3)C2)cc(Br)ccc1C#N C(=O)(C(CC)C(=O)NCCC(C)N(C)C(c1ccc(CCF)cc1)=O)OCC C(C(C(=O)SCC)NC(c1cccn1C(C)C)=O)SCC.c12cc(n[nH]1)NC2 C(=O)(CN=C(NCC(C)(C)C(F)(F)F)NC1COCC1F)NC(C)C C1(CCNC(c2nnn(CC)c2C)=O)CCN(C(c2ccccc2F)=O)C(C)C1 N1(C(c2cnc(SC)s2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)C(O)C1 Cc1ccn2cc(CCNC(=O)C(C(C)C)NS(N)(=O)=O)nc2n1 C(=O)(CCCn1cc(NC(=O)NCc2ccnn2C2CCC2)cn1)NC C1(NC(=O)CCCn2cccn2)CC2CCC1CN2C(C1C=CCCC1)=O N1(CC2(OC(C)C)CCC2)CC(=O)N(Cc2ccc(Cl)cc2Br)C1=O Cc1cc(F)ncc1-c1cn(C2CC(C(N3CC(c4nncs4)C3)=O)C2)nn1 C1(C(=O)NCC(Cc2c(C)nc[nH]2)O)CCN(C(C2CCC2)=O)CC1C C12(C(=O)NCC(C)(C)NC(c3c(CC)c(C)ccc3)=O)CCCCCC1OCC2 c1(C(N(C2CN(C(CC3(C=C)CCC3)=O)C2)C)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(CN2CCC(CNC(=O)CCC(F)(F)F)CC2)ccc2ccsc2c1 C(=O)(NNc1ccc(S(=O)(=O)C(F)(F)F)cc1)NC(c1nc(CC)[nH]n1)C N1(C(C2=NOC(C)C2)=O)CC2CC(NC(c3cccc(CC#N)c3)=O)C(C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)N(C(c2ccn(C3CCC3)n2)=O)CC1 C1(N(C(CCC(C)C)c2ccc(Cl)cc2)C2CC2)COC2(CCC2)C1 CS(=O)CCC(O)C(=O)NCC1(F)CC(CNC(=O)C=CBr)C1 C1(NC(C2CC23CCC3)=O)CCC2(CC1)CN(C(=O)CN1CC3CC3C1)CCO2 C(=O)(C(C)C(F)F)N(CCOCCC(=O)NCC=CCCOC)C c1(C(N2CCCC(CCNC(CC=CC)=O)CC2)=O)ccc(OC)c(OC)c1Cl N1(C(C2(C#N)CC=CC2)=O)CC(C(=O)NC2C3CCCC23)C2(CCC2)C1 N(C1CC(C(=O)O)c2ccccc21)C(CN1CCN(C)CC1CO)=O c1(C(=O)NC(Cc2cncs2)CO)cc(C2CCCCC2)cc(Cl)c1O N1(C(C(CCN(C)C)O)=O)CCC(CC(=O)NCC2CCCC2CF)C1(C)C Cc1cc(Cl)cc(C(N2CCN(C(=O)CC34COC(C)(C3)C4)CC2C)=O)c1O C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C=CCOC)=O)C(F)(F)F C12(C(=O)NC)CCC(Nc3cccc(-c4cn(CC5C(C)C5)nn4)c3)(CC1)CC2 N1(C(C(C)c2cc[nH]n2)=O)CCC(C(F)C(=O)NCCNC(=O)N(C)C)C1(C)C c1(CNC(CCN(CC#C)C(C2CCC(C)(CC)O2)=O)=O)ccc(Cl)cc1 CC12CC(C(=O)NCC3CC(CNC(=O)Cn4cc(CO)nn4)C3)(C1)C(C)(C)O2 C1(CNC(CCC(=O)OCC)=O)CC2CCC1N(C(=O)C(C)SC(F)(F)F)C2 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCS3)=O)C2)ccc(Br)c(F)c1 c1(CCC(=O)NCc2cn(CCNC(=O)CO)nn2)nc2ccccc2s1 c1(OC)cc(C)cc(C(=O)NCC2COCCN2C(c2sccc2C#N)=O)c1C N1(C(CC2CCCC(=O)N2)=O)CC(C(=O)NCC2(CO)CCCO2)C(F)(F)C1 c1(CC)cc(CC(=O)NCC2CC(O)CN2C(=O)C=C(C)C(C)(C)C)n(C)n1 C1(C(N2Cc3ccccc3C2)=O)C2CC(CC2F)N1C(c1cnnc(O)c1)=O C(=O)(C(F)C(F)(F)F)N1CC(C)(NC(C2CC(C)(F)C2)=O)C1 N(C1c2cc(C)ccc2CC1C)C(=O)NCc1nnc(COC)s1 C(=O)(CC(C)CCC(=O)NC1(C)CN(C(C2CCS(=O)(=O)N2)=O)C1)OC N1(C(CSSC)=O)CCC2(CCCCN(C(=O)CSC(F)F)C2)C1 C=CC(C)C(C)C(=O)NCCN(C1CCCC1)C(=O)C=Cc1sccc1C c1(C(=O)NC2CCC(C)(NC(c3ccc(C)s3)=O)CC2)c[nH]c2cccc(C)c12 N1(C(c2nc(C)oc2C)=O)CC2CCC1C1CN(C(c3ccc(O)nn3)=O)CC21 c1(C(N(CC(CC)NC(c2nnsc2N)=O)C)=O)cc(OC)n[nH]1 C1(C)(C(=O)NCCc2c(C(=O)NCc3c(CC)n[nH]c3)c[nH]n2)CCCOC1 CC(C)C(C)C(=O)NCC1CCC(CNC(=O)C(C)Sc2nncn2C)CC1 N#CC12CC(C(=O)NCC(c3ccccc3)NC(c3cnn(CCO)c3)=O)(C1)C2 c1(OC)ccnc(N(C2CNCC2C#N)Cc2ccc(OC(C)C(=O)O)cc2)n1 CC1CCC(CC(N2CCCC2CN(C(=O)Cn2cccnc2=O)C2CC2)=O)CC1 c1(CNc2c(C)c(NC3CCC(C)CC3C)ncn2)n[nH]c2c1CCCC2 N1(C(COCC(C)C)=O)CCC2C1CCCN2C(=O)CN(C)C(C)C n1(CC(=O)NC2CCC(CNC(C3OCC(C)(C)C3)=O)C2)cnc([N+](=O)[O-])c1 c1(C(=O)NCCCCC(C)NC(C(F)=CC)=O)c(F)cc(Cl)cc1F N1(C(CCCC(CC)CC)=O)CC(=O)NC2CN(C(C3CCS3(=O)=O)=O)CCC12 N1(C(Cc2cc(C)nn2C)=O)CCC(NC(=O)C=CC2CCOCC2)C12CC2 CC(C)(C)CC(O)CC(=O)NCC(O)CNC(c1ccc(NC=O)cc1)=O C1(CC2(C(N(C)C(=O)NC)=O)CC2(F)F)CCCN1C(=O)COC1CCC1 C(C(C)(C(C)C)NC(=O)CC(C)N(C)C)NC(c1cnc(CC(C)C)s1)=O S(=O)(=O)(c1cccc(Br)c1F)N1CCC2CN(C(C=C(C)C)=O)CC2C1 c1(C(=O)NCC(C)CNC(C2C3CCC23)=O)nc(-c2ccco2)n2ccccc12 c1(C(N(C2CCN(C(CN(CCC)C)=O)CC2)CC)=O)cc2ccccn2c1 C1(CC(=O)N(C)Cc2ccco2)CC2(C1)CN(C(c1ccnc(N(C)C)c1)=O)C2 N1(C(c2c(CC)nns2)=O)CCC(CNC(=O)C(C)(C)C)(OC)C1 c1(NC(C2CCCCC2)C(=O)NC(C)C)ccc(N2CCCCC2)cc1 C1(C(N2CCC(NC(c3cccnc3S)=O)C(F)C2)=O)Cc2cccnc2C1 N1(C(c2ccc(C)o2)=O)CCCC2(C1)CN(C(c1ccc(CO)cc1)=O)CCO2 c1(C(N2CCN(C(CCOCC#C)=O)CC23CC3)=O)c[nH]c2ccc(O)cc12 C(=O)(CCCOC)NCCCN(C(C(=O)N(CC)CC)C)C.C1CCN1C C(C(=O)N1CC(O)CC1C(=O)NCC1CN(C(=O)OC(C)(C)C)C1)(C(C)C)OC CC(O)CC(=O)NCC(O)CCNC(=O)CC1CCSC1 c1(CC(=O)OC)ccc(NC(C2CSCCN2C(=O)C=Cc2ccsc2)=O)cc1 c1(OC)c(C(=O)NCC2CC(NC(=O)C3CC3)C(O)C2)sc(S(N)(=O)=O)c1OC c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C)C)nccc2ccccc12 CCC(C)(CNC(c1cccc(F)c1Br)CO)C(C)O CN1CCCCN(C(=O)C(C2(C)CC2)NC(C2CC23CCC3)=O)CC1 c1(NCc2scc(C)n2)cnc(F)cc1C(=O)Nc1cccc(F)c1Br C(c1ccccc1)=C(OC)C(=O)N(C(C)CNC(=O)CCCN(C)C(C)C)C C1(C(=O)NCC(CC)NC(C2CC3(CSC3)C2)=O)CC(c2ccccc2)=NO1 c1(C(=O)NCC2CC(F)(CNC(C(CC)SC)=O)C2)cn2cc(C)nc2s1 CC(C)CC(CNC(C1C2CCC1(c1ccc(C(F)F)cc1)C2)=O)N(C)C N1(C(CCCSC)=O)CCN(C(C2C3COCC23)=O)CC1C C1(C(=O)NC(C#C)C(C)C)(NC(=O)Cc2cncc(C)c2)CCOCC1 C1(CC=C)(NC(=O)CCC(F)F)CCN(C(c2cc(COC)no2)=O)C1 C(=O)(C1CCCc2ccnn21)NCC(CNC(CN(CCC)C)=O)(C)OC C#CCC(C(=O)N(CCC(=O)NC1(CO)CCSC1)C1CC1)C1CC1 C(=O)(CC(F)(F)F)NC(C1(O)CN(C(=O)C(C2CCOCC2)O)C1)C N1(CCNC(C23CC(n4cc(Cn5cccc5)nn4)C2C3)=O)C(=O)CCC1=O N1(C(CCC2CC(NC(CC(CC=C)(C)C)=O)C2)=O)CCC2(CC=CCO2)C1 C1(N(c2nc(SCC)c(Cc3ccccc3Cl)s2)C(C)=O)C2CCOC2C1(C)C C(CCCCC(=O)NC1CCN(C(c2cc(C)ccc2Cl)=O)CC1CO)=CC CC(C(=O)NC1(C)CCN(C(C2(F)CCC(F)(F)CC2)=O)C1)C1=CCCC1 CCCC(O)(CCC)CC(=O)N1CCCC1Cc1ccc(F)cc1 c1(NC(CC2N(Cc3cc(C)nn3C)CCC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1ccc(NCCCC2CCC2)c(F)c1)NCC(C(C)O)(C)C CC1=C(C(=O)N2CCC(O)(c3cn(Cc4ncon4)nn3)CC2)CCCO1 N1(C(C(C)OCC#C)=O)CCC(C)CC1CNC(=O)CCCOCC C1(NC(C2C(OC)(OC)CC2)=O)CC2(C1)CC1(CC(NC(=O)C3=CCC3)C1)C2 C1(CNC(C(C)Sc2ccc(Cl)cc2)=O)(CF)CC12CCOCC2 C1(CCNC(=O)CC2(O)CCC2)CCN(C(c2nnc(O)cc2O)=O)CC1(F)F c1(-c2c(C(N3CC(C)OC(C)C3)=O)sc3c2CCC3)ccc2nc(O)[nH]c2c1 c1(CNC(C(C2CC2)CC)=O)cccc(NC(=O)C=C(C)C)c1 C(CC(=O)N1CCC(N2CCC2)C1)(C(F)F)NC(C=NOC)=O C(=O)(C(O)CCC(C)C)NC1CCN(C(C(CC)=CC)=O)C1C(C)C C1(NC(=O)CCC2CC2)CC2CN(C(c3cccc(CO)n3)=O)CC2C1 C(=O)(CCCCC#Cc1ccccc1)NC(CNC(C(C=C)(C)CC)=O)C1CC1 C12(NC(CCCOC)=O)COCCC1CN(C(c1cnn3ccn(C)c13)=O)C2 c1(NC(C2N(Cc3cc(C)c(F)cc3)CC2)=O)cc([N+](=O)[O-])cnc1C N1(C(c2n(C)ncc2)=O)CCCC(NC(c2ccnc(C3CC3)n2)=O)CC1 C1(NC(Cc2nc(=N)[nH][nH]2)=O)CC2CCC(C1)N2C(=O)CC1CC1C(F)(F)F N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C(C)(C)C1 C(CNC(C1(C)CCCS1)=O)(CC(C)C)NC(c1c(CC)non1)=O CC1C(C(=O)NC(C)(CN(C)C)C2CC2)CC1(F)F C(C(COC)CC(=O)NCC1CC1C(=O)NCc1ncccc1OC)OC C1(C(=O)NC(C2CN(C(c3nonc3N)=O)CCO2)C)COC2COCC12 C#CCC(C)(C(=O)NC1CCN(OC)CC1)NC(C1CCCC1CC)=O C#CC(C)(C)C(=O)N1CCC(NC(=O)CNC(C)=O)C1 c1(CS(N2CCC3(C(C(=O)NC4(CO)CC4)C3)C2)(=O)=O)cc2ccccc2[nH]1 C1(C(N(C(C(=O)NCC(n2cccn2)C)C)C)=O)CN2CCC1C2 Cc1ccc(C(C)C)c(OCC(=O)NC(C)CN(C(=O)C=Cc2ccoc2)C)c1 N1(CCc2cn(C3CC(C(=O)NCC4(C)CC4(Cl)Cl)C3)nn2)CCC(O)CC1 c1(C(N2C(C(=O)Nc3cccc(CF)c3)CC(C)C2)=O)ccc(Br)cc1I C(=O)(C1CCCn2ccnc21)N1CCOCC(NC(C(NOC)=O)=O)C1 N1(C(Cc2cc(COC)on2)=O)CCC(C)(CNC(c2ccn(C(F)F)n2)=O)C1 c1(C(N(C2CCCN(C(C3CCS(=O)CC3)=O)C2)C)=O)c[nH]c2nc(Cl)ccc12 c1(C(=O)OCC)ncc(F)cc1NC(=O)Nc1cccc(NS(=O)(=O)C(C)C)c1 c1(C(=O)NCC2(CO)CCN(C(c3c(CC)ncs3)=O)C2)c(F)cc(O)cc1F N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3cc[nH]c(=N)c3Cl)=O)C2C1 Cc1cc(C(=O)NC(CNC(C2CCCC2(F)F)=O)C(C)C)c(N)c(F)c1 C#CC1CCCC(CNC(=O)C(CC2CCCC2)NC(c2cc(Cl)ns2)=O)C1 c1(N2CCC(c3cccc(OC(F)(F)F)c3)(F)C2)c(Cl)cnc2[nH]nnc12 N1(C(c2c(N)non2)=O)CC2(C1)CN(C(=O)CC1CC1(Br)Br)C2 N1(C(COCCC=C)=O)CCN(C(c2cocn2)=O)C(C)C1C CC1(C(=O)NCC(=O)Nc2ccccc2O)CC12CCN(C(=O)C1CC1)CC2 CCCC(O)C(=O)NCC(C1CC1)NC(c1[nH]ccc1-c1ccccc1)=O C=CCC(C(=O)NC(c1cnn(C)c1)C(=O)N1CC(CC)C1)OC Cc1cc(C)c(C(=O)CN2CC3CC2C3C(=O)N(C)C)[nH]1 N1(C(CC2N(C(C3=NOC(C)C3)=O)CC2)=O)CCCC(F)(F)CC1 c1(CN(C(c2cccc(CO)c2)C(=O)NCCCCCC)C)cc(Br)ccc1F C(=O)(CC1=Cc2ccccc2C1)NCC(CCC)NC(c1scnc1Cl)=O C(=O)(C(C)CC(N)=O)NCC1C(C)CCN1C(c1cc(CN(C)C)c[nH]1)=O C1(CC(=O)N(CC(=O)NC(CC=C)CO)CCOC)CCCC(=O)C1 Cc1cc(C(=O)NC(C)CCCC(=O)N(C)CC2CCCCCC2)cc(O)n1 C(=O)(C(C)(C)C(=O)NCCN1CCN(C(C2(C)CC2(F)Cl)=O)CC1)OCC C(c1ccc(F)c(Cl)c1)=CC(N1C(C)(CCN(C)CCO)CC1)=O.C(C)(C)(C)OC(=O)O C(=O)(CC(CN(C)C)C(F)(F)F)NCC(C)(C)OCCNC(C(CCCC)C)=O C1(c2cccc(F)c2)(NC(=O)NC(c2cccnc2)C2CCOCC2)CCOCC1 C1(C(N(C)CCOCCN(C)C(C2(C)CCC(=O)N2)=O)=O)CCC(C)(F)CC1 Cc1cc(C)n(CCCC(=O)NC(C)CCNC(c2cc(Br)c(C)o2)=O)n1 c1(C(N(C(C(=O)N(CCCSC(F)F)CCO)C2CC2)C)=O)cnc[nH]c1=N Cc1cc(C(N2CC(OCCC(=O)NCC3(O)CCN(C)C3)C2)=O)nn1C c1(C(=O)NCC(C)CNC(c2c[nH]nc2C(C)(F)F)=O)cc(Cl)ccn1 N1(C(COCCC=C)=O)CCN(C)CC1CNC(=O)CNC(=O)CCC c1(C(N2CC(COC)(NC(=O)CC=C(C)C)C2)=O)cccn2c(C)nnc12 N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C)CC1CNC(=O)C(F)C(C)C C1(CNC(COCCOCC#C)=O)COCCN1C(=O)C(C)SC CCC(C)C(O)CC(=O)NC(C1(C(=O)NC2CCCN(C(C)C)C2)CC1)C c1(C(=O)NC(C(C)NC(C2ON=C(C)C2)=O)(C)C)cc(OC(F)F)cc(F)c1 C(C)(CC(F)(F)F)NC(c1n(CC=C)nnn1)c1ccncc1 C1(C(=O)OC)OC(C(=O)OCCCc2nocc2C)CC1C C(=O)(CCC1=NNC(=O)CC1)NC1C(NC(CNC(=O)OCC=C)=O)COCC1 C(CCC(C)CC(=O)N1CCC(=CC(=O)NCC(C)C)CC1)=C(C)C c1(C(N2CC(NC(=O)CC3CCOC3)C(F)C2)=O)cc2c(cn1)OCCC2 c1(CN2CC(C(=O)OC)C(c3cn(C)cn3)C2)cc(C)c(I)cc1C Cc1cc(Cl)ncc1NC(C1COC(CNC(c2cc[nH]c2)=O)C1)=O C1(NC(COC2CCN(C(CCCOC(C)=O)=O)C2)=O)CCCSCC1 C1(C(N(CC(C)O)C)=O)CN(C(=O)C(F)C(C)(F)F)CC12CC2 Cc1nn(C)cc1NC(=O)C(c1ccccc1)NC(=O)Cc1ccoc1 C(=O)(CS(=O)(=O)CC(=O)N(C)CC1(O)CN(C(C2COCC(C)(C)O2)=O)C1)OC N1(C(C(CC=C)OC)=O)CC(NC(C2CC(=O)N(C)C2)=O)C2(CCCC2)C1 C1(C(C)(C)C)(CNC(CCC2C(C)(C)C2)=O)CCN(C(=O)CCn2cccn2)C1 Cc1ncnc(C)c1C(=O)NCC12CC(NC(c3snc(O)c3Cl)=O)(CO1)C2 C#CCC(C(=O)NC(c1cnn(C(C)C)c1)C)NC(C)=O C1(CNC(CC=CCC)=O)C(O)C(O)CN1C(c1sc(C)cc1Br)=O C(C(=O)NNc1nc2ccccc2s1)c1ccc2c(c1)OC(C)C2 C(CCC(=O)NC(C)Cn1cc(CC(C)O)nn1)OCC=C c1(COC(=O)CC23CCCC2C3)ccc(C(F)(F)F)cc1F.C12CC(C1)NC2=O c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(C1CC(C(F)F)C1)=O C(=O)(C(CCC)NC(=O)CC1CCC(C)(C)O1)NCCOCCC=C c1(C(C(=O)NCC(CC)NC(C2CCC3CC3CC2)=O)C)ccc(F)cc1F c1(NCCC2(OC)CCC2)ccc(S(=O)(=O)NCc2nc(C)ccc2Br)c(Cl)c1 c1(C(=O)NCCC(C)NC(C2(O)CC(F)(F)C2)=O)ncc[nH]c1=O C(=O)(C1(C)CCc2ccccc21)Nc1c(C)cc(NC(c2nocc2Cl)=O)cc1 Cc1cc(C(=O)NC(C)CCC(=O)NCCCCN2CCC2)ccc1O N1(C(=O)C(C2CC2)C2CC2)CC2(C1)CN(C(C1CC1(F)F)=O)C2 Cc1ncccc1CNC(=O)CCN(C(=O)CCCN(C)C(C)C)CCO C1(C(=O)NCC(C(C)C)NC(=O)CCc2cnccn2)CCn2c(O)nnc2C1 N1(C(c2c(C)cccc2)=O)CCN(C)CC1CNC(C1CCC(C)C(C)C1)=O c1(CC)nc(C)c(C(=O)NC2(CO)CN(C(c3cc(Cl)c(Cl)s3)=O)C2)o1 N1(C(=O)OC(C)(C)C)C=COCC1C(=O)OCCCCC1CCCO1 CC(C)(C)CCCC(=O)NC1CC(NC(C2CCOC(=O)N2)=O)C1 C1(NC(c2ccc(NC)cn2)=O)CN(C(c2cn[nH]c2)=O)C(C)(COC)C1 CCCC(C)(CCC)C(=O)N(C)CC1(O)CCN(C(C2CC2c2cccs2)=O)C1 C(=O)(C(C)(C)CCC(=O)OC)N1CCCC(CNC(CCSCCCC)=O)C1 N1(C(c2c(C)scc2)=O)CCC(C2CCCN(C(C3Cc4cscc4C3)=O)C2)C1 c1(C(N2C(C)CC(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(CNC(C(=O)Nc2ccc(CCC)cc2)=O)cccc(F)c1F CCCC(C(=O)N1CCOCC(NC(c2cnc(OC)c(C)c2)=O)C1)C(C)C CCCCCCCC(=O)NCC(CC1CC1)C(=O)Nc1cc(C)cc(C)c1 C1(F)(C(=O)NCC(COCC)O)CCN(C(c2occc2CC)=O)C1 CCC(CNC(=O)CC1CN(C)C1)(CC)NC(=O)Cc1ncn(C)c1C C1(O)(CCNC(c2nc(C#C)sc2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C(N2CC(O)(C(C(=O)NCC(C)(C)C#N)F)C2)=O)CC(=O)C12CCC2 CCCCC(CC)C(=O)N1CCCN(C(c2cnc(OC)s2)=O)CC1 CC(CCNC(=O)CCC1CCCCN1C(=O)Cc1ccn(C)c1)C(F)F C(C(F)(C(=O)N1CCN(C(=O)CC)CC1)C(C)C)NC(C1(CCCC)CC1)=O C(=O)(C1=CC2CCCC12)N(CCCCN(C(=O)CCCn1ccnc1)C)C n1(CC(=O)NC2CC(C)(CNC(C3CCN(CC)CC3)=O)C2)cccc(O)c1=O c1(OC)cccc2c(C(=O)NCC(C)N(C3(CS(C)(=O)=O)CC3)C)n[nH]c12 c1(C(=O)NCCCC(C)NC(C2CCOC(=O)N2)=O)ccc2c(n1)CCC2 c1(C(N2C(CNC(CC3(C(=C)F)CCC3)=O)C=CC2)=O)ccc(OC)c(OC)c1 c1(C(N2CCC(n3cc(CCCC=C)nn3)C(O)C2)=O)cccc2occc12 c1(COC)csc(CNC(c2ncoc2-c2ccccc2)=O)c1 CN(CCCC(=O)NC(C1CCOC1)CNC(c1n[nH]c2c1COCC2)=O)N=O C1(C(=O)NCC(CC#C)(C)C)CCCCCN1C(=O)CCc1cnc(C)o1 Cc1sc(O)nc1C(=O)NC(C)CN(C)C(c1cncc(-n2cccn2)n1)=O c1(C(N2CCC(Cl)=C(Cl)C2)C(=O)NCCCCCC)nnc2n1CCCCC2 c1(CC)cc(OC)ccc1C(N1CCCC1C(C)NC(=O)C1=CCC1)=O CC1CN(C(=O)CNC(C2CC2C)=O)CCC1C(=O)O CC1(C)CCCCC1C(=O)NC1CC(C(=O)NOCC2CCC2)C1 c1(C(=O)OC)ccccc1NNC(=O)C=CCC1CCCC1 N1(C(CC(CC)(C)C)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(=O)C2=COCCO2)CCCC12CCN(C(C1(Br)CC1(F)F)=O)C2 c1(C(=O)NCCC2C(C)CCCN2C(=O)CCCC2CC2)ccc(C#N)cc1F C1(C(=O)NCCS(=O)(=O)NC)CCCN(C(=O)CCCC2CC2)CC1 CC(=O)CCN=C(NCCN(C(C)(C)C)CCO)NC1Cc2ccccc21 c1(C(=O)O)cccc(C2(F)CC2C(=O)NC(c2cccc(F)c2)C(F)F)c1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCCC(NC(=O)CCOCCC)C(F)C1 c1(OCCOC)c(CC(=O)NCC(C)N(C(=O)C(C)CC2CC2)C)cccc1Cl N1(C(C2C(C#N)C2)=O)Cc2ccnn2CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC(NC(c2cnsc2)=O)CC(C)(C)C1 c1(-n2c(C)ncc2)ncccc1C(=O)OCC(C)C.C12(CCOC1)C(=O)N2 c1(C2C(C(=O)NCCS(=O)Nc3ccc(F)c(F)c3F)C2)ccc(F)c(F)c1F C(=O)(CS(=O)(=O)CC(C)C)NC1CN(C(CC2N(CC)CCC2)=O)C1 C(CC1CCCO1)(C(F)(F)F)NC(N1CCC1COCC1CC1)=O C#Cc1ccc(C(=O)NC2CC(CNC(c3coc(C)c3)=O)C2(C)C)cn1 N1(C(c2c(SC)n(C)nc2)=O)CC2OCC(NC(=O)CCC3CCCCC3)C2C1 c1(C(=O)NC(CC)CNC(C2(C)CCOC(C)C2)=O)cc(C)c(OC)c(C)c1 C1(NC(=O)OC(C)(C)C)CN(C(c2cc3c(F)cccc3[nH]2)=O)C2(CCCC2)C1 C1(C)(C(=O)NCC2CCCC(NC(CN(C(C)=O)C)=O)C2)CC2CCC1O2 C1(CNC(=O)NCC2(C(C)(F)F)CCC2)C2CC3C(C2)C13 CS(=O)(=O)C(CNC(=O)CC1CNC(=O)C1)CNC(=O)COCCC(F)(F)F c1(CCC(=O)NC(C(=O)NCC(C=C)O)c2cccs2)cc(C)[nH]n1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(C2OCC2(C)C)=O)C(C2CC2)C1 N1(C(C(c2cn(CC)nc2)=O)=O)CCN(C(c2cccnc2C)=O)CC(CO)C1 C1(OC)CC(C(=O)NC2CCC2NC(C2CCN2C(C)(C)C)=O)CC1NC(C)=O C(C(C)C(=O)N1CCC(CCNC(c2cc(C(F)(F)C(F)(F)F)on2)=O)C1)SC CON1CC(C(N2CCC(C)(CNC(=O)CCSc3ccccc3)C2)=O)CC1=O CCCCC(C)C(=O)NCC(C)(C)CN(C(c1cn(C)c(C)n1)=O)CC CCC(C)(CCNC(c1sccc1F)=O)NC(c1c[nH]c(C(N)=O)c1)=O C1(CN(C(CC(C)OC)=O)C)CN(C(c2cc(N(C)C)ccn2)=O)CCO1 c1(COC)ccc(C(=O)NC(C)C(C)NC(C2(CC(=O)OC)CC2)=O)s1 N1(C(C(=O)NC2CCCN(S(C)(=O)=O)C2)=O)CCCC2NCCC12.C1(=O)CN1C N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 N1(C(C(=O)NC(c2csc(C)n2)CC)=O)CC2(CC(CO)CO2)C1 C1(NC(c2cc(CNC(C3CCN(C4COC4)C3)=O)[nH]n2)=O)CCCC(CO)C1 c1(OC)c(Cl)cc(C(=O)N(CC(C)N(C)C(c2cnc(C)cn2)=O)C)cc1Cl CCC(CCCC(=O)N1CCSC(C)CC1)NC(=O)Cc1n[nH]c(C)n1 N1(C(C=C(CC)CC)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C(C)C1 c1(C(N2CC(NC(c3c(C)ncn3O)=O)C(C)C2)=O)cc(F)ccc1S(C)(=O)=O N1(C(C2CCC(C)CC2)C(=O)NC2CC2)CC=CCC2(CCOCC2)C1 N1(C(=O)OC(C)(C)C)CCC(C(=O)NCCC2CN(C(c3nn[nH]c3Cl)=O)C2)C1 C=CCCCC(C(=O)NCC(O)CC(C)C)NC(=O)C(c1cccn1C)=O N1(C(c2c(C)nccn2)=O)CCCCCC1CNC(=O)CCC(C)(C)C N1(C(C(C2CN(C(CCCNC(=O)OC)=O)C2)O)=O)CCC(O)C(F)C1 C(=O)(N1CCC(C(=O)N(C)CCO)O1)C1ON=C(C)C1 C1(C(C)N(CC(=O)Nc2ccc3occc3c2)C2CC2)COc2ccccc2O1 c1(C(=O)NC2CC(CCNC(C3(C)CC=CCO3)=O)C2)cncc(S(C)(=O)=O)c1 c1(NC(C)=O)cnc(C)c(C(N2CC(C)C(NC(C3CCCO3)=O)C2C)=O)c1 Cc1cc(F)ncc1CNC(=O)CC1CC2(CC2)CN1C(=O)CSCCC#N C1(C(=O)NCC2CC2)(NC(C(C)OC(C)(C)C)=O)CCSC1 C(=O)(CCC(=O)NC(C1CCN(C(c2ccncc2NC)=O)C1)C)NCCC C1(OC)(CNC(=O)C(C(C)C)OCC(C)C)CCN(C(=O)CC2(C#N)CC2)C1 N1(C(C2N(C(C(C)SCCCC)=O)CC(=O)C2)=O)CCC2(CCCO2)C1 CCC(CCC(=O)N(CCC(N)=O)C)NC(c1cccc(C)c1)=O C1(OC)(CNC(=O)C(C)CN2CCCC2)CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NC(C#N)C(N)=O)cc2cc(-c3ccn4cnnc4c3)ccc2o1 CC(C)C(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC1CC(O)C(O)C1 CC1CCC(=CC(=O)NCC2C3CN(C(c4ncoc4Br)=O)CC23)CC1 c1(C(=O)NCC2CC(CNC(CN(S(CC)(=O)=O)C)=O)OC2)occ(C)c1C N1(C(C(CCC)N(C)C)=O)CCN(C)CC1CNC(=O)C(F)CC1CCCCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(CC(F)F)N(C(=O)COCC(F)F)C C#Cc1cnc(C(=O)NCC2CC(F)CN2C(=O)CC2CNC(=O)O2)c(C)c1 c1(C(C)C)nnc(CN(CCCNC(=O)CCOCC(F)F)C(C)C)s1 CC1C(=O)N(C)CCN1C(=O)CCC1(C)CN(C(=O)CC2CCC(C)(C)C2)C1 NC1(C(=O)NCC2(Cl)CC23CCC3)CC2(CCOCC2)C1 N1(C(C=CC)=O)CC(NC(=O)C=CC2CCOCC2)CC(O)C1 CC(C)C(C(=O)N1CCCC(C(C)NC(C2SCCS2)=O)C1)c1cccnc1 Cc1oc(C(=O)NC(C)(CNC(=O)C(C)CO)CO)cc1Br CC1CN(C(C2CC23CC(O)C3)=O)CC1(C)CNC(c1ccc(F)cc1)=O N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1C(=O)N(CC(O)C1CC1)C N1(C(C(C)=C(C)C)=O)CC=CC1CNC(=O)CCc1nc(-c2ccco2)no1 n1(C2C(C)C2)c(N2CCCC(C(=O)NC3CC3)C2)nnc1-c1ccc(Cl)nc1 c1(-c2n(C)nc(-c3ccc(C(C)(C)C)cc3)n2)cnn2ccc(O)nc12 C1(C(NOC(COC)C(C)C)=O)CC2CC1CN(C(=O)CS(=O)(=O)C(C)C)C2 Cc1nc(NCCCc2nc3ccccc3[nH]2)cc(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C2CC(NC(C3CN(C(=O)NC)C3)=O)C2(C)C)=O)CC(COC)C2(CC2)C1 c1(NC(C)=O)cc(C(N2C(C(=O)NCC3(O)CCC3)CC3CC23)=O)ccc1F Cc1cc(O)ccc1CNC(=O)C(C)N(C)C(c1cc[nH]c1)=O c1(C(=O)NCc2nccc(C(=O)NC(CCC)CCO)c2)cc(N)cc(F)c1 c1(C(N2CC(CNC(C=C(CC)C)=O)C(C)C2)=O)cc(N)c(OC)cc1OC C1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C2)NC(=O)CC1C(F)(F)F N1(C(CCCC)=O)CC(NC(C23COC(CS(C)(=O)=O)(C2)C3)=O)CC1C CC(C)C(O)C(=O)NCCOC1CCN(C(=O)CC2CC(N(C)C)C2)CC1 C1(C)(C(=O)NC(C2(O)CCN(C(=O)Cc3ccon3)C2)C)CCSCC1 Cc1nn(C)c(Cl)c1CC(=O)NC(CNC(C1CCC(O)C1)=O)C1CCC1 C1(CNC(C2N(C(c3n(C=C)nnc3)=O)CC3CC32)=O)CC2(CCC2)CO1 CC(C)CC(C(=O)NCCc1nncs1)NC(C1C2CCCC12)=O CC1CCCN(C(=O)C2=NOC(C)C2)C1CNC(c1ccc(N)c(Cl)c1)=O C1(NC(CCC2COC(C)(C)O2)=O)COCCN(C(C2CC(CC3CC3)C2)=O)C1 Cc1cn2c(n1)C(C(=O)Nc1nccc3ncccc13)CCC2 c1(N2CC=CC(NC(c3c(C)nc(O)nc3C)=O)C2)nc(Cl)nc2sccc12 N1(C(c2nnn(CC)c2C)=O)CC(F)(F)CC1CNC(=O)CS(=O)(=O)CC C1(C(=O)NCc2cnn(CC)c2C)CC2CC1CN(C(=O)CC(F)(F)F)C2 C(=O)(C(C)(CC)CCC(C)C)NC1CC2(CC(CNC(C(C=C)O)=O)C2)C1 c1(C(N2CCN(C(C(C(CC)C)OC)=O)CC(O)C2)=O)nc2nccc(C)n2n1 C1(C(=O)NCC2(C)N=C(C)SC2)CCN(C(C2(C)CCCCO2)=O)CC1C c1(OC)ccccc1C=CC(=O)NC(C)CCCCNC(C1CCCOCC1)=O c1(C(N2CCC(C)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)COC2 c1(C(N2CC(CNC(CSC(C)C)=O)C3C2C3)=O)cc(Cl)cc(Cl)c1N C1(NC(c2nnc(C(C)(C)C)s2)=O)CCC2CCN(C(C3CSCCS3)=O)C1C2 C(=O)(C(=O)N=S(C)(C)=O)NCC1(NC(C(NOC)=O)=O)CCCCC1C c1(C(=O)NC(C2CCCCN2C(=O)C(=O)NC2CC2)C)cnc(=NCCF)[nH]c1 C(=O)(CC(CC)C(C)C)NC(CCCCNC(C=CCOC)=O)(C)C C1(C(=O)NCC2(CNC(CC=C(C)C)=O)CCCCC2)CC(=O)CC12CCC2 CCC(C)C(C(=O)N1CCC(C)C(NC(C2CCNC2=O)=O)C1)NC(C)=O Cc1nc(C(=O)NCC(C)(CO)NC(c2ccc([N+](=O)[O-])[nH]2)=O)ccc1[N+](=O)[O-] c1(CCC(=O)NCCC(C)NC(c2cccc(C3(C)CC3)c2)=O)cncc(F)c1 C1(C(=O)NC2(CO)CN(C(CCNC3(C)CC3)=O)C2)CCCCC12CC2(F)F c1(C(N2C(CNC(Cc3ccc(C)nc3)=O)CC2)=O)c[nH]c2nccc-2c1 Cc1nn(C)c(C(=O)NC(CNC(=O)Cc2cnn(C)n2)CC(C)C)c1Cl C(=O)(C1CCCc2ncnn21)NC(C(C)C)CNC(c1cnc(F)c(Cl)c1)=O N(C(=NCC(C)C)NCc1ncccc1Cl)CC(NOCC)=O c1(C(=O)NC2C(CC)CN(C(=O)C(Cl)=CCl)CC2)cc2cc(OC)ccc2[nH]1 Cc1cccc2c(C(=O)NCCCCC(C)NC(=O)CC3CCSC3)n[nH]c12 c1(C(=O)NCC2(CN(C)C(C3CC3(C)Br)=O)CC2)nnc(O)cc1O C1(F)(CNC(=O)Cc2ccc(F)cc2)CCN(C(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)NCCNC(C(C)OCCC#C)=O)cc(S(C)(=O)=O)c(NCC)cc1C CC1CN2CCCC2CN1C(c1ccc2c(c1)CCC2)C(=O)NC1CCCCC1 C1(C(C)C(=O)NCCCC2CCCC2O)CCN(C(c2cc(O)ncn2)=O)CC1 S(=O)(=O)(CC1=NOCC1)NC(c1nnc(CC(C)C)s1)C N1(C(C2CC(=O)NC2)=O)CC(C2(NC(c3cnc(CO)nc3O)=O)CC2)C1 n1(CCC2(c3n(C)ccn3)CC2)nc(-c2cccc(F)c2)nc1C1CCCO1 c1(CCNC(c2n(CCOCC)nnn2)CC2CCOC2)cccc(C)n1 Cc1cc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCCO3)C2)s1 C(=O)(CS(N)(=O)=O)NC(C1CN(C(=O)CCc2cccc(O)c2)CCO1)C c1(C(N(C(C)C)CCN(C)C(C2CC2F)=O)=O)cnc2c(F)cccc2c1 C1(C(=O)NC(c2ccccc2F)CNC(c2cnns2)=O)CCCNC1=O c1(C(C)=O)ccc(C(N2CC3(CCC3NC(=O)CC(C)CN(C)C)C2)=O)c(C)c1 c1(C(N(C2CCCC(NC(C3CCC=CCC3)=O)C2)C)=O)cc2n(n1)CCO2 c1(C(N2CC(CNC(C=C(C)C)=O)C(C)C2)=O)ccn2nccc2n1 N1(CCC(=O)OC2COCC2Oc2ccccc2)C(=O)C2CCCCC2C1=O c1(OCCC)cccc(C(N2CCOC(CNC(=O)C(O)C3CC3)C2)=O)c1 c1(C(=O)NCC(CN(C(c2[nH]cc(CC)c2)=O)C)C)cc(C)c2occc2c1 C(=O)(C1CN(C(=O)CN(C)C(N)=O)Cc2nnn(COCC(C)(C)OC)c21)OC c1(C(=O)NC23CC(NC(C(C(C)C)SCC)=O)(C2)C3)noc2c(F)cccc12 C1(NC(=O)CCc2cnn[nH]2)CC2CN(C(C3(F)CC=CC3)=O)CC2C1 C12(C(N3CCC(N4CCC(NC(C5CCCC5)=O)CC4)C3)=O)CCC(CC1)OC2 c1(N(C)CCC2CCCCC2)nc2cccnc2c(=NC2CC2C(C)(C)C)[nH]1 C=CCC(C(=O)N(C1CCCN(C(c2csnc2OC)=O)C1)C)OC N1(C(c2cncc(C(C)(C)C)c2)C(=O)NCC)CC(CO)C2(CC2)C1 CCC(CC(=O)NCc1cc(C(N2CCCCC2C(C)CC)=O)on1)CC(C)C c1(C(N2CC(C)C(NC(=O)CCc3ccn(C)c3)C2)=O)csc2nnsc12 Cc1cc(CNCC2CC3(CCC3O)C2)nnc1C N1(C(CC(C)F)=O)CCC2(CC1)C(N(C(=O)C(N)=O)C)CS2(=O)=O C1(Cn2cc(C3CN(C(C(C)CCO)=O)C3)nn2)CCCCCCC1 N1(C(C2(COC)CCCO2)=O)CC(NC(=O)C(Cl)=CCl)C(n2cccn2)C1 C12(NC(N3CCC(c4cc(C(C)C)[nH]n4)C(C)C3)=O)CCCC(C)(C1)OC2 c1(C(=O)NC2CC(NC(CSCC=C)=O)C2)sc(CC)nc1C c1(CCC(N2CCCC(O)(CNC(=O)C(F)(F)C3CC3)C2)=O)cc(F)cc(F)c1 C1(CC(=O)Nc2nc(C(C)C)on2)CCCN(C(=O)NCCCN(C)C)C1 C1(CN(c2cc(OC)cc(OC)c2)C)CCC2(CCNCC2)CO1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCC3(O)CCC3)CC2)ccc2ocnc2c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC3CN(C(=O)CCCN(C)C)CC3C2)nn1C N1(C(CN(C)C(=O)C2CC2)=O)CCN(C(=O)C(F)C2CCC2)CC1 N1(CC(=O)NCCc2c(OC)ccc(Cl)c2)CCCCC2CCCCC12 C(=O)(C#CC1CCOCC1)N1C(CNC(COCC(=O)N(CCOC)CC)=O)CC1 C(=O)(C(C)(O)CNC(c1cccc(OC(C)(C)C)c1)=O)OC c1(C(N(CC(C)CNC(=O)CCC2CC2(F)F)C)=O)cc(N)c2ccccc2n1 C1(CC(N2CC(O)(CN(C(CC3CC(OCC)C3)=O)C)C2)=O)CC(=O)NC1=O CCCC(C(=O)NCC1(C)CCCN1C(C1CC(N2CC(O)C2)C1)=O)OC C=CCCN=C(NCc1cc(O)ccc1Cl)NCC1CCCC(C(=O)OC)O1 c1(C(=O)NCC(CCNC(C2C(C)CCC2)=O)(C)C)cc2c(s1)C(C)(C)CCC2 C1(NC(C(CCC)N(C)C)=O)CCOC12CCN(c1ncc(C)c(O)n1)CC2 c1(C(=O)NCC2(C(=O)NC3(C)CC3)CC(=C)C2)ccc(OC)cc1.C(C)(C)O N1(C(C(=O)NCC)=O)CCOC(CCNC(=O)Cc2cncn2C2CC2)C1 Cc1ccc2[nH]nc(C(=O)NCCC3CN(C(=O)CC(C)P(C)(C)=O)C3)c2c1 Cc1c(C(=O)NC2CCN(C(=O)C(O)CN(C)C)C2)cc([N+](=O)[O-])cc1[N+](=O)[O-] CCCCCCCCC(=O)N(C1CCN(C(=O)CC23COC(C)(C2)C3)CC1C)C C(=O)(CC(C)(C)N(C)C)N(CCC(=O)NC(CCC=C)C)C O=C1CCc2cc(-c3cnn4c3CN(Cc3cc(Br)cnc3F)CC4)ccc2N1 c1(C(N2CC(CNC(c3cc(CCOC)on3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(CC(C)(C)C2CC2)=O)CCC(C2=NOCC2)C1.C1CC(=O)NCCS1 N(C(=NCC(F)(F)F)NC(C1COCCOC1)=O)C1CC(NCC(C)(C)O)C1 c1(N2CCC(Cc3n(C)ncc3)C2)cc(C#N)ccc1Br C(=O)(C(O)CC(N)=O)NC(CSC)(C)C(=O)NCc1csc(C)n1 C1(NC(C=C(CC)C)=O)CC2CCC1CN(C(c1ncn(C)c1C)=O)C2 C(C(O)CC(=O)N1CC(C)(C#N)C1)NC(Cn1ccc(C)n1)=O c1(OC)cc(C)c(C(N2CCCN(C(=O)C=C(C)C(C)C)C(C)C2)=O)cc1Cl C1(C(N2C(CC(=O)NCC3(C)ON=C(C)C3)CCC2)=O)NC(=O)OC1(C)C c1(C(N2CCN(C(c3ccc(C)cc3)=O)CC2)=O)ccc(C(C)(F)F)nc1O C(c1scnc1C)=CC(=O)NCC(CNC(C=CCOCCOC)=O)CO C(=O)(C(C)(C)S(C)(=O)=O)NCCN(CCCN(C)C)C(c1cccc2c1OCC2)=O C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(=O)CC(O)C1CCCC1)C2 C1(NC(CCCC(=C)C)=O)CCCCN(C(c2cc(O)ccc2Cl)=O)CC1 C1(C(N(CC(CN(C(C(C)Oc2cccnc2)=O)C)O)C)=O)CCC2CC2CC1 c1(CC(=O)N(C2C3CN(C(C4COC4)=O)CC23)C)ccc(F)c(Cl)c1 CC1CN(C(=O)C=C2CCN(C)C2)CCN(C(C2CC(=O)C23CCC3)=O)C1 C(N=c1[nH]c2c(c(=NC3CSC3)[nH]1)CSC2)c1sc2ccc(N)c(Cl)c2n1 Cc1nc(C(N2CCC(NC(=O)Cn3ncccc3=O)C(C)C2)=O)ccc1C#N C(=O)(CCCCCCN=[N+]=[N-])NCC1CCN(c2cc(C)ncn2)C1C C1(F)(CNC(C(C)(C)C)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCOC1CCCC1)NC(c1n(CC)ccn1)C C#CC1CN(C(C2CCN(C(=O)C(C)OCC3CC3)CC2)=O)CCN1C CC1(C)CC=C(C(=O)N2CC(CNC(=O)CNc3ccccc3Br)C2)CC1 C#CCC(CC(=O)N1CCC(C(N)=O)C1)NC(c1oc(C)nc1C)=O N1(C(C(=O)NC(C)C)=O)CC2(C=C(C(=O)NC3CCCC(O)C3)CO2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(N(C(=O)C=Cc2ccsc2)C)C(F)C1 c1(C(=O)OCC)sc(N(C(=O)C(n2ccc(C)n2)C)C(C)C)nc1C1CC1 Cc1ccc(C2(C(=O)NCC(F)CNC(=O)C(F)(F)CO)CCC2)c(C)c1 C(=O)(C(C)(O)CNC(C1CCC(C(=O)NC2CCS(=O)(=O)C2)CC1)=O)OC CCC(C)CC(C(=O)O)c1nc(-c2ncccc2Br)no1 N1(C(c2c(N)c(F)ncc2)=O)CC2CCN(C(=O)C3=C(Cl)CCOC3)CC2C1 CC1(C)CCCC(CNC(=NCCC2CCN2C2CCOCC2)NC2CCC2)O1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(C=C(C)c2ccco2)=O)C12CC2 CCCC(C#N)C(=O)NC(C)CN(C(=O)CCc1nnc(-c2ccsc2)o1)C c1(C(N2CC(CC)N(C(c3csc(=NC)[nH]3)=O)CC2)=O)cc(C)c(=O)n(C)c1 c1(C(N(C2CCN(C(c3n(CC)ncc3)=O)CC2)C)=O)c[nH]c2cccc(F)c12 N1(C(COCCCC(C)C)=O)CCC2CC2(C(=O)NC2(C)CCCC2)CC1 C(C)(C(=O)NC1CC(CCNC(=O)CCC2(C)CC2)C1)OCCCC CCC(CC)(CCNC(C1(CCOC)CC1)=O)NC(c1ccnc(OC)c1)=O C(=O)(C(C)CO)N(C(C)CNC(=O)CCN(c1ccncc1)C)CC C1(N2CCCC(C(=O)OC)CC2)(CCC)CN(C(C2(C)CCN(C)C2)=O)CCC1O N1(C(c2cnc(CNC(Cc3n(C)ncc3)=O)nc2)=O)CC(C2CCCC2)C1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)CC(C)(F)F)CC12CCC2 C12(C(N(C)CC3CCN(C(C4CN5CCN4CC5)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 Cc1nnc2n1CC(C(N)=O)N(CCC(=O)N(C)Cc1ccncc1)C2 C1(C(N2CC(SC)C(NC(C3CCOC3)=O)C2)=O)CCN(CP(C)(C)=O)CC1 N1(C(C2(CCC)CC2)=O)CCC(C)C(CNC(c2cccc(OCCF)c2)=O)C1 C(=O)(C1=C(c2ccccc2)CCCC1)NCCCCN(C(=O)CC#N)C c1(C(C)C)cccnc1C(=O)NC1CCCCC1CNC(=O)C(O)C1CCCC1 C1(CNC(C(C)C2CCC2)=O)CN(C)CCN1C(=O)CC1CCC(C)(C)CC1 C1(CNC(CNS(NC)(=O)=O)=O)C2CCC(C2)N1C(C1(OC)CCOCC1)=O c1(C(N2CCOCC2)=O)cc(S(=O)(=O)Nc2cccnc2O)ccc1Cl C1(NC(CC=CC=C)=O)CCC12CN(C(c1ccc(OC)c(C)c1)=O)C2 N1(C(c2nc(C)[nH]n2)=O)CC2CCN(C(=O)Cn3ccc(C(F)(F)F)n3)CC2C1 C=CCC(CC(C)C)C(=O)N1CCC=CC1C(=O)NC1CSC1 N1(C(COCC(=C)C)=O)CCC(C2CCN(C(c3cc(CC)[nH]n3)=O)CC2)CC1 c1(C(=O)NC2CC(C)(CNC(C#CC(C)C)=O)C2)cc(=O)c2ccccc2o1 C#Cc1c[nH]nc1C(=O)NC(C)Cc1ccc(CNC(=O)C(CCC)OC)cc1 Cc1cc(CNC(c2cccc(C)n2)c2nnnn2C2CCCCC2)cc(Cl)n1 C1(CC#C)CCN(C(C2(CNC(=O)CNc3ccccn3)CCC2)=O)C1 N1(C(C(CC)F)=O)CCCC(CCCCNC(=O)C(=O)NCCOC)C1 c1(-c2scc(C)n2)nc(CCN2CCCC2)n(CCC(F)(F)F)n1 CN1CCCC(C(=O)NCC2(NC(=O)CCOC3CC3)CCCC2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)N(CCNC(C1C2CC2C2CC12)=O)CC1CC1 S(=O)(=O)(c1c[nH]c(=NCCn2cnnn2)cc1C)NCCCc1cccc(C)c1 C1(N(Cc2c(C)[nH]c(-c3ccccc3)c2)C2CC2)CCC2(CCCCC2)CC1 c1(CNC(C2N(C(c3nccc(OC)c3)=O)CCOC2)=O)ccc(Br)nc1Br C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1CC(C)CN1Cc1cccc(I)c1O c1(C(N(CCCNC(C(CSC)O)=O)C)=O)c(C)c(Br)n(C)c1C Cc1nn(C)c(C)c1C(=O)NCC1(F)CN(C(=O)COC2CCOC2)C1 N1(C(C=C(CC)CC)=O)CCC(NC(=O)C(CSC)OC)C(CO)C1 C1(C(=O)Nc2c(C)nsc2)C2CN(C(=O)CC3CCN(C)CC3)CC12 N1(C(CCSc2n(C)nnn2)=O)CC2(COC(CNC(=O)CS(N)(=O)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)cns3)=O)C2C)=O)ccnc2c(F)cccc12 C1(CNC(C2C(NC(c3n(CC)nc(C)c3)=O)CC=CC2)=O)CN(C)CCN1C CC(O)C(F)(F)C(=O)NCC1CN(C(=O)C(N)=O)CCCO1 N1(C(c2cn(CC(=O)OCC)nn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 c1(C(=O)OC)cc(C(=O)NC(C2CCN(C(c3cn[nH]c3)=O)C2)C)c(C)o1 c1(NCCN2C(=O)CC(OC)C2)nc2c(c(=NCCC(C)N3CCC3)[nH]1)CCC2 S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)NC1CN(C(C(CC)C)=O)CC1C Cc1cnc2cc(-c3nc(Cc4ccccc4F)nn3CC3CC3C)ccn12 CC1CC(C(N2CC(N(C(=O)C(F)(F)c3cnn(C)c3)C)C2)=O)CC(C)O1 c1(CNC(c2nc(COC)sc2)c2nnnn2CC2CC2)cc(C)nn1C Cn1nccc1CNC(=O)CCC1CC(NC(=O)C=CC(=O)N(C)C)C1 c1(NC(c2ccc(C)s2)C)nccc(=NCC(F)C2CCC2)[nH]1 c1(-c2cn(CC(N3C(CC)CC3)=O)nn2)cccc(Cc2cc(CO)on2)c1Cl C=CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CN2CCN(C3CC3)C2=O)C1 Cn1ncc(C(N2CC(NC(=O)COCc3nc[nH]n3)C2)=O)n1 C1(C(N2CCC(NC(CCc3cc(C)on3)=O)CC2C)=O)CCCC2C1C2(F)F c1(C(=O)NCC(C)N(C(CC2(CCC#C)OCCO2)=O)C)cccnc1C1CC1 C1(C(=O)NC2CC(CCC(=O)Nc3c(C)noc3C(C)C)C2)NC(=O)OC1(C)C C1(C(=O)NC(CNC(c2c(O)nc(C)c(C)n2)=O)CO)CCc2cnn(C)c2C1 c1(N2CCC(CC=C)(NC(=O)CSC(F)F)CC2)ncnc2c(OC)cccc12 C1(C2(Nc3nc(CC)oc3)CC2)CCCCN1C(C1(C(F)(F)F)CC=CC1)=O Cc1nc(CCC(=O)NCC2(O)CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)oc1C c1(CNC(NCCOCC=C)=NC)cccc(C)c1Cc1ccccn1 FC1COc2ccccc2C1NCC1CC2(CC2)C1 c1(CN(C(CN2CCC(C)(OC)C2)=O)C)ccc(C(F)(F)F)cc1C C1(CCNC(CCOC)=O)(C(=O)NCC2(N(C)C)CCCC2)CCCC1 C1(CCNC(C(C)C)=O)CC(F)(F)CN1C(=O)C=Cc1ccnn1C C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(c2cc(C3CCOCC3)no2)=O)C1 C1(NC(c2n(CCC)nnn2)c2ccncc2)CC(=O)N(CCOCC)C1 C(=O)(C(C)(C)C(C)(F)F)N1C(CNC(CNC(CCC)=O)=O)CCC1 c1(C(N2C(CCCNC(C3CCC4CC34)=O)CCC2)=O)cnc2[nH]ccc2n1 c1(C(C)=O)c(N(C)Cc2cncc(C(F)(F)F)c2)ccnc1Cl S(=O)(=O)(CCC(=O)NCC1(C)CCC(NC(=O)Cn2cnnc2O)C1)NC C(=O)(C(C)(C)CC(=O)OCC)N1CCC(CCOC)(NC(=O)C=C(Cl)Cl)C1 c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(C)C2)=O)cc(Cl)nc(Cl)c1 c1(OC)ccc2nccc(C(=O)NC3(CO)CCN(C(c4cscn4)=O)C3)c2n1 C1(NC(CCP(C)(C)=O)=O)CCSC12CN(C(=O)CCc1ccc(N)cn1)C2 c1(CC(=O)NC2CC(C)(NC(=O)CC(=O)N3CCOCC3)C2)cc(F)ccc1Cl Cc1cc(C(=O)NCC2(C)CN(C(=O)C(N)=O)C(C)(C)C2)c2c(O)nn(C)c2n1 c1(OC)ccc(O)cc1C(=O)NC(C)(C)C(C)NC(C1CCN(C2CC2)CC1)=O c1(C(N(C2CCN(C(CC=CC=C)=O)CC2C)C)=O)ccn2cc(C)nc2c1 c1(C(N2CCCC(n3cc(CCC(C)=O)nn3)C2)=O)sc2ncccc2c1Cl Cc1cnccc1C(C)C(=O)NCC1(O)CCN(C(C2CC2C(=O)NCCO)=O)C1 C1(C(=O)NCC2C(NC(c3c(CCC)n[nH]c3)=O)C2)CCOC2(CCC2)C1 CC(C)CC(O)CC(=O)NC1CCCCC1C(=O)NC1CCCC1(C)C C=CC1CN(C(=O)C(C)OC(C)(C)C)CC1NC(c1cccc(C)c1Cl)=O N1(C(CC(C)SC)=O)CCN(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)CC2)CC1 C1(C(=O)O)(NC(c2c(NC)ccc(F)c2)=O)CCc2c(F)cccc21 C1(C(N2CC(C)(NC(C3CCN(C(CC)=O)C3)=O)C2)=O)CCCC(N(C)CC)C1 C1(NC(C2(NC(C(CC3CCC3)NC(C)=O)=O)CCSC2)=O)C2CCC(C2)C1CO N1(C(C(C)O)=O)CCC(C2(NC(c3c[nH]c4nccc-4c3)=O)CC2)C1 C1(OC)CC(C(=O)NC2CC(CNC(c3coc(C(C)C)n3)=O)C(O)C2)C1(C)C N(C1CCSc2ccc(Cl)cc21)C(C(c1cccc(OC)c1)C)=O c1(C(=O)NC2CCN(C(COCCCOC)=O)CC2OC)ccc2sccc2c1 C=Cn1ncc(C(=O)NCC(C)C(=O)NC(CCC)C2CCCC2)c1N c1(OC)ccc(C(=O)NCCCCNC(=O)CCCSc2ccccc2)s1 CC1CCCC=C1C(=O)N1CCCC1(C)CNC(C1CCCN1C)=O CC1CC(NC(=O)Cc2cncs2)CCN1C(=O)C(C)N(C)C C1(CC(C)C)COCC1(c1nnnn1CCCF)NCc1ccccn1 CC(CC(=O)NC1(CCNC(=O)C(Cl)=CCl)CCC1)C(C)(C)C Cc1cc(C(=O)NC(C2CCN(C(c3cn(C)nc3Cl)=O)C2)C)cnn1 Nc1c(C(N2CC3CC3(CNC(C3CC4C=CC3O4)=O)C2)=O)cc(Cl)cc1Cl C1(C(=O)NCCc2c(OC)cccc2)CCN(S(=O)(=O)N2CCCCC2C)CC1 C1(C(=O)NCCCOCCCNC(c2c(C)c[nH]c2)=O)CCN(C)S1(=O)=O C1(C(=O)NC(C(=O)N(C2(C#C)CC2)C)CCF)CN2CCC1CC2 N(C1CCCc2c(OC)cccc21)C1(c2n(CC)nnn2)CCC1CS(N)(=O)=O c1(C(N2CC(C)C(C)(C(=O)NC3CC(F)(F)C3)C2)=O)ccc2c(c1)COC2(C)C c1(C(=O)NC2C(C)CN(C(=O)CS(N)(=O)=O)C2)cccc(N)c1Br c1(OC)cccc2c1OCC(C(N1CCN(C(=O)CC#N)CC1C(C)(C)C)=O)C2 C(=O)(C1=NOC2(CCC2)C1)NCC1(C)CCC(NC(c2ccc(Br)o2)=O)C1 Cc1cc(C)n2ncc(C(=O)NC3CCN(C(=O)CCOC(C)C)CC3F)c2n1 Cc1nsc(N)c1C(N1CCC(O)(C(C)NC(C2CCSCC2)=O)C1)=O N1(C(c2c(CC)nn[nH]2)=O)CCC(CNC(=O)C(C2CC(F)(F)C2)O)C(F)(F)C1 C1(C)(CNC(CSCC)=O)CCN(C(c2cc(-c3ccccc3)sn2)=O)C1 C1(c2nnnn2CCCF)(NCc2c(C)ccnc2)CCCC(C2CC2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCC(C(C)NC(C(C(C)C)CN(C)C)=O)CC1 C1(COC)CCN(C(=NCCC(C)(C)S(C)(=O)=O)NC2CCC2)C1 c1(C(N2CCCC(=C)C2)C(=O)NC)cc2n(n1)CC(C)(C)CO2 C1(C(=O)NC2CC(CC(=O)N(C)CC3CC3(F)F)C2)(OC)CCCCC1 C1(NC(C2C(=C)CC2)=O)CC2CCC1CN(C(c1scnc1C)=O)C2 CC1CN(C(c2ncn3ccccc23)=O)C(C)CN1C(=O)CN(CC(C)(C)C)C C1(CNC(C(c2ccc(Cl)cc2)C)=O)C(C)CCCN1C(C1CCCC1O)=O c1(C(C2CCCO2)NC(=O)NCCOc2cccnc2)ccc(F)cc1 C(=O)(C(C)C(C)NC(C1(C)CCN(C(=O)Cn2cnc(=N)[nH]2)C1)=O)OC Cc1cc(C#N)cc(C)c1COCC(=O)NCC(C)(CO)CC(=O)O C(=O)(C1=CCC(NC(=O)CC(O)C2CCCC2)C1)NC(CC#C)CC C1(N=c2ccn(CCCO)[nH]2)(c2n(CCC(=O)OCC)nnn2)CSC1C Cc1ccc(C(=O)NCC2COC(CNC(=O)C#CC3(C)COC3)C2)c(=O)n1C CCC(C)C(C)C(=O)N(C)CCNC(c1ccc(CN2CCS(=O)CC2)cc1)=O c1(C(N2C(C)C(NC(=O)C=C3CCN(C)C3)CCC2)=O)cccc2c1CNC2=O C1(C(N2CC(OCCNC(=O)CCn3ccnn3)C2)=O)CC(O)C(F)C1 C1(CNC(Cn2ncc(CC)c2)=O)CC(C)(C)CN1C(=O)C(C)SC C1(C(=O)NC(c2nc(C)on2)C)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(=O)NCC(CC)NC(=O)C(O)P(C)(C)=O)ccc(O)c(C(=O)OC)c1 N1(C(CC(=O)OC)=O)CCC(C=CC(=O)NC2CCC3(CC2)N=N3)CC1 N1(C(C(F)=CCC)=O)CC2CCC(C1)N2C(=O)CC12CCCN1CCC2 C1(CNC(c2c(C)con2)=O)CCN(C(=O)C(F)(F)Sc2cnn(C)c2)CC1C c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)C2=CCCCC2C)c(C)c1 Cc1ccc(OC(C)C(=O)NCC2(F)CCC(NC(=O)CN(C)C(N)=O)C2)cc1 C12(C(N3CCC(CN(C(C=CC)=O)C)C3)=O)CCC(CC)(CC1)OC2 CCC(CC)(C(=O)N(C)CCN(C)C(C1CC1C)=O)c1ccc(Cl)cc1 C1(C(N2CC(C(C)NC(c3ccc(C(F)F)o3)=O)C2)=O)CC(=O)CC12CCC2 c1(CN(C(=O)CCN(CC(C)(C)C)C)C)cncn1C.C12(CCC1)C(=O)NOC2 C1(CC(=O)NCC2(NC(Cc3ncn(C)c3)=O)CCOC2)CCCS(=O)(=O)C1 Cc1cccc(Br)c1C(C(=O)NC1CC1(C)CO)NC(c1cc(C(N)=O)[nH]n1)=O CCC(C)(C#N)C(=O)N1CC(CN(C(=O)C=Cc2nc(C)c(C)[nH]2)C)C1 N1(C(c2nnc(C)s2)=O)CCCC(C)C1CCNC(c1cc(C2CCC2)no1)=O CC(C)(C)C(CCO)NC(c1c[nH]nc1C1CCNC1)=O c1(C(N(CCNC(c2c(F)cc(Cl)cc2F)=O)CC)=O)cccc2ncn(C)c12 CCC(C)CCCC(=O)N(CCC(=O)NC(C)CN(C)C(C)C)CC C1(NC(C2N(C)CCOC2)=O)CN(C(C2CCC3CCCCN23)=O)CC2(CC2)C1 c1(NC(C(Cn2ccnn2)NC(C(C)S(N)(=O)=O)=O)=O)cnc2[nH]cnc2c1 c1(C(C(=O)N(CCN(C(C(F)=CC)=O)C)C)NC(=O)COC)ccccc1 C1(NC(N2CCn3c(cnc3C(F)(F)F)C2)=O)CCOC12CCS(=O)(=O)CC2 c1(CC)cc(N)c(C(=O)NC2CN(C(=O)C(O)C(F)(F)F)C(C)(C)C2)c(F)c1 Cc1cccn2ncc(C(=O)NCCCNC(C34CCC3CC4)=O)c12 c1(CCC(=O)NC(COC)CC(=O)N(C)CC)cnc2ccccn12 N1(CC)CC(C)N(C(c2c(CNC(=O)CSC(F)F)nnn2C)=O)CC1C C=CC1CN(C(=O)CCc2ncc[nH]2)CC1NC(=O)CCCNC(N)=O c1(C(N2CC(N(C(C(CC)N(CC)CC)=O)C)C2)=O)ccc(OC)c2ccsc12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(N(C)Cc2ccccn2)=O)CC(O)CC1 C1(CN(C(=O)CC2CCCCC2)CC)CCN(C(C2COCOC2)=O)CC1 C1(CNC(c2c(CNC(c3c(C)cn(C)c3)=O)c[nH]n2)=O)CC2CCC1CC2 c1(CC(=O)NC2CCC(C)C2)ccc(CNCC2(N(C)C)CC2)cc1 C=CC(C)(C)CC(=O)NCC(c1ccccc1)N(C(=O)CSC(C)C)C C(=O)(C1=C(C(C)F)N(CC)C(=O)NC1c1ccc(OC2CCSC2)cc1O)OC c1(C(=O)NCCCN(C(=O)C(C)(F)CC2CCCC2)CC)coc2c1COC2 c1(CCC(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)C2)ccc(Cl)cc1 CC(C)CC(C(=O)NCCCC1CCCN1C(=O)CCCF)c1ccccc1 N(C1CN(C(C2CCCCCC2)=O)CCc2ccccc21)C(C(=O)NC1CC1)=O c1(C(N2C(CN(C(COC(CC)C)=O)C)CCC2)=O)cc2ncccc2o1 c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCCN(C)C(C1CN(C)CCO1)=O c1(SC)cnn(C)c1C(=O)NC1(C)CN(C(=O)C(c2ncccc2F)(F)F)C1 C1(NC(c2c(C)csc2)=O)CCCCC1C(N1CCC1(C)C(=O)OC)=O N1(CC=C)CC2COCC2(CN(C(=O)C(N)=O)Cc2cccnc2)C1 c1(NC(C(C2CCC(C)(C)CC2)C)=O)ccc2c(c1)S(=O)(=O)CC(=O)N2 C12(NC(CSC)=O)CCC1CN(C(=O)CC1(N(C)C)CCCC1)C2 c1(C(=O)NC2C(NC(C(C)CC(F)(F)F)=O)CCCC2)cc2c(s1)CC(C)(C)C2 Cc1ccnc(C(C)NC(=O)CCN(C(C2CN(C3CCC3)C2)=O)C(C)C)n1 CCC(C)C(O)C(C)C(=O)N1CC(O)CC1C(=O)NCCCc1ncc[nH]1 N1(C(c2c(C)nn(Cc3ccccc3)c2)=O)CC2(CC(CNC(=O)C(F)F)C2)C1 C1(C(F)(F)F)(C(N(CC(C)NC(c2coc(C3CC3)n2)=O)C)=O)CCN(C)C1 c1(CC(=O)NC2(COC)CN(C(CCCOCCC)=O)C2)cccc(Cl)c1Cl N1(C(C(CC)OC(C)C)=O)CC2CC1(CNC(=O)CCCOc1ccccc1)C2 N1(C(C(F)=CCC)=O)CC2CCC1C2NC(=O)CC1CCCCC1(C)C c1(SCC(=O)NC2C3CN(C(N4CCC(O)CC4)=O)CC23)cc(F)c(Cl)cc1F N1(C(c2ccc(N(C)C)cc2)=O)CC2CC(NC(=O)CSCC(N)=O)C2C1 N1(C(CC(CC)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CC=CC12CCOCC2 N1(C(C2(CC#C)CCCC2)=O)CC2(C(=O)Nc3ccccc3O)CC1CO2 c1(OC)ncccc1C(=O)N(CCNc1ccc(F)cc1)C(c1cc[nH]n1)=O c1(OCc2ccc(C(=O)NC3CCCCC3)o2)ccc(F)c(F)c1 CC(C)CCCCC(=O)N(C1CC(NC(=O)COCC2CCCO2)C1)C c1(C(=O)NCC2CC(C)(C)N(C(=O)C(F)C(F)(F)F)C2)cnc2c(c1)CCOC2 c1(CC)nnc2c(C(N3CC(N(C(C4CC5C=CC4C5)=O)CC)C3)=O)cccn12 Cc1cc2cccnc2nc1C(=O)NCC(CO)NC(=O)CC1C=CCC1 CCCC(CCC)CC(=O)NCC1CC(NC(C2CCN(C)CC2)=O)CCO1 CN=c1[nH]c(=NCc2cnc(C)[nH]2)[nH]c(=NC(C)Cc2nc3ccccc3s2)[nH]1 C(=O)(C(F)(F)CCN(C1CCOC1(C)C)C(C)=O)N1C(C(=O)OC(C)C)CCC1 c1(C(=O)NCC2N(C(c3ncc(C)nc3)=O)CC(O)C2)cnc([N+](=O)[O-])cc1C c1(CN2CCOCC(NC(c3c(C)ncn3C)=O)C2)c(Cl)ccc(Cl)c1Cl c1(C(=O)NC2C(CNC(C3(CC#C)CCC3)=O)CCC2)ccc(N)c(C(C)=O)c1 C1(CNC(c2ncc(C)nc2)=O)C(C)CCCN1C(c1n[nH]cc1C)=O c1(NC(C2N(c3nc(C)nc4c3c[nH]n4)CCC2)=O)cccn2nc(C)nc12 n1(C(C)C(=O)NC2CCCC2NC(c2cc(O)cs2)=O)cnc2ccccc12 C(=O)(CC1=CCN(C(=O)CC(C)(C)CN(C)C)CC1)N(CC)Cc1occc1C C1(C(=O)NC(c2nccn2C)CC)(CNC(c2cncn2C)=O)CC12CCC2 C(=O)(CC1=CCCCC1)Nc1cc(C)c(NC(=O)CC(O)CN(C)C)cc1 c1(CCC(=O)NCC(C2CCCC2)NC(C(CCC)C)=O)ccc(F)cc1F C(=O)(CC(C)(C)C#N)N1C(C(N2CCC2CC(C)(C)C)=O)(COC)C=CC1 C1(NC(c2ccnc(C)n2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C(C)C1 N1(C(CN(CC#C)C(c2cc(C)co2)=O)=O)C2C=CCC1CC2 S(=O)(=O)(c1ccc(Br)cc1NC1CCN2CCCC12)NCC(CSC)OC C(CC(O)C(=O)NC1(CF)CCCC1)NC(C(C)C1C(C)C1)=O C(C)(CO)(C(=O)NCCS(C)(=O)=O)NC(CSC)=O c1(OC)nsc(OC)c1C(=O)NCCOC(C)(C)CNC(=O)Cc1csnn1 c1(C(N2CCC(CC(=O)Nc3cncnc3)C2)=O)c(F)cncc1Br C(=O)(C(=O)N=S(C)(C)=O)N1CCCC(NC(C(CC)n2cncn2)=O)CC1 c1(N2CCC(=O)NC(=O)C2)nc(NCC2CC23CCCCC3)c2ncsc2n1 c1(C(=O)NCC2C(NC(C(C=C)(C)O)=O)CC2)cc2cc(Cl)ccc2[nH]1 N1(C(C=CC(C)C)=O)CC(NC(c2cnc(-c3cccnc3)s2)=O)C2CC12 c1(C(C(=O)N(C)CC2CN(C(=O)C3=CSCS3)CCO2)(C)C)ccc(F)c(Cl)c1 C1(CC(=O)NCc2cccnc2F)COCCN1C(C1CCCC(O)C1)=O C1(NC(C2CCN(C(C=C(CC)CC)=O)C2C)=O)CN(C)C(=O)C12CC2 C1(NC(C=CSC)=O)CC2(CCN(C(=O)CC3CC4(CCCC4)CO3)CC2)C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CCCC2(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)ccc(F)c(F)c1F N1(C(c2snc(C)c2N)=O)CC2(CC(C(N3CCC(CC(F)F)C3)=O)CO2)C1 c1(C(c2nnnn2CCOC2CCSCC2)CSC)ccc(F)cc1C(F)(F)F C(C(CC)CC(CC)CC)NC(c1n(CC=C)nnn1)c1ncc[nH]1 Cc1cc(N)c(C(=O)NC23CCN(C(C4(O)CCC4)=O)CC2C3)cc1C N1(CC)CC(C(=O)NC2CCCCC2N(C(=O)CCc2ccco2)C)CC1=O c1(C(=O)NC(CC(C)NC(c2[nH]cc(C(=O)OC)c2)=O)C)c(F)cc(C)cc1Cl C1(C(=O)NCCN(C(C2CC2C2CCC2)=O)CC)CCCCC1(C)C c1(C(C)(C)C)cc(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCCF)on1 n1(CC(N2CCN(C(c3nccc(C)c3)=O)CC2)=O)cnc2c1CCCC2 C1(C(N2C(COC)(CNC(=O)CC34CC(C3)C4)CCC2)=O)CCCCN1N=O c1(C(=O)NCC(C(C)C(C)C)NC(C2(CCC)CC2)=O)cnc2n(c1=O)CCS2 S(=O)(=O)(c1c(C)o[nH]c1=N)NCc1c(C)cn(CC)n1 N1(C(N2C(CC=C)(CC=C)CCCC2)=O)CC23CCCC2(C1)CN(C)C3 c1(CNC(C23N(C(c4c(OC)nccc4)=O)CCC2C3)=O)nc(C)ccc1O OC1CCCC(N=c2[nH]c(=NCc3ccc(Cl)o3)[nH]c3c2CCC3)C1 Cc1cccc(CCNC(C23CC2CN(C(C2(CO)CCOC2)=O)C3)=O)n1 c1(OC)cc(C(=O)NCCCC(C)NC(=O)CNC(C)=O)cc(N)c1OC c1(C(=O)NC(c2ccccc2)C2CN(CC3(n4cccn4)CC3)C2)cc(O)ncn1 c1(-n2cc(C3N(C(c4cc(C)ncn4)=O)CCCC3)nn2)ccc(Cl)cc1Cl C#CC1CCCN(C(=NCCCC)NCCSc2cccc(OC)c2)C1 C=CCCCCCC(=O)NC1CC2CCC1N2C(=O)CCc1nc(O)n[nH]1 c1(NCCC(=O)NC2(CC)CC2)ccccc1.C12CN(C1)CC(=O)N2 C(=O)(C1=CC2CCCC12)NCCOC1CN(C(c2nccc(C)c2)=O)C1 c1(C(C)C)ccccc1C(=O)N(C1CN(C(C2CC2c2ccco2)=O)C1)C C(=O)(CCCCCN=[N+]=[N-])NC1(C)CN(C(C2(OC)CCSC2)=O)C1 C(=O)(C(CCN(C)C)NC(=O)CC=C(Cl)Cl)NCCN(CCCF)C c1(C(N2CCC(NC(Cc3cn(CC)nc3C)=O)(CF)C2)=O)cc(C)nc(O)c1 C1(C(=O)Nc2c(CC)nsc2)CN(C)CCN1C(c1cc(C2CC2)on1)=O c1(N2CCC(S(=O)(=O)NCC)C2)nc(=NCc2ncoc2C)[nH]c2ncn(C)c12 N1(C(C2CC2CC)=O)CCN(C(=O)CC2(OCC)CCC2)CC(C)C1 C1(C(N(C)CC2(O)CCN(C(c3ncc(C)nc3)=O)C2)=O)CC1C1CCCCC1 Cc1nc(CCCNC(=O)CC2CCN(C(=O)Cc3sccc3C)C2)n[nH]1 Cc1cc(C(C)(C)C)ccc1C(=O)NCCCCCNC(=O)Cc1ccno1 N1(CC(CC)(O)C(F)(F)F)CCCC2CCCN(C)C12 C(=O)(C(C)(C)C(=O)N(C)C)N1C(COC)CC1.C12CC(C(O)C1)NC2=O N1(C(C2CN(C)C2)=O)CCCC(C(=O)N(C)Cc2nccn2C)C1 c1(C(=O)NCC(C)NC(=O)C(C)C(C)O)cccc2c1CCOC2 C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1CCCC1)CNC(C(C)OCC#C)=O c1(Cc2nnnn2C2CCC2)ccccc1Br.C(CCO)CCSC c1(SC)cccc(CC(=O)NCCC(C(C)C)NC(=O)C2=COCC2)c1 C1(N(C(C(=O)NCCOC)C(C)C2CC2)C)CC2CC3CC(C2)CC1C3 c1(CC(C)C)cn(C2CN(C(=O)CC3CC(NS(C)(=O)=O)C3)C2)nn1 N1(C(CC2N(C(C(C(C)C)OC)=O)CC2)=O)CCC(O)(C(N)=O)CC1 Cn1nc(C(F)(F)F)cc1CC(=O)NCC(CO)NC(c1cc(CCO)on1)=O c1(SCC)ccccc1CC(N)=O.N12CCN(CC1)C1CN(C1)OC2=O N1(C(c2scc(OC)c2)=O)CCC(C#N)(NC(C2CC=CCC2)=O)C1 c1(C(C)C)ocnc1C(=O)NCC1(O)CC(NC(=O)CCc2ccon2)C1 c1(OC)cccc(CCC(=O)NC(C)(C)CF)c1 N#Cc1ccc(F)c(-c2cccnc2C(N2CCCC(Br)C2)=O)c1 C1(NC(CSCCC)=O)CN(C(c2ccc(N)cc2Cl)=O)CCC1CO N1(C(c2c(COCC)ocn2)C(=O)NC2COC2)CCCSCC1C C1(NC(c2ncccc2F)=O)CN(C(C2CC3CCC(C2)C3)=O)CC12CCCC2 c1(NC(C2CC(c3cccc(F)c3)C2)=O)nnc2n1CCNC2 C1(CC)CCCCC1NC(=NC)NC1CCN(c2cccc(N(C)C)c2)C1 c1(C(=O)NC(C2CCN(C(c3ncc(OC)nc3)=O)C2)C)cccc(C#N)c1 C1(NC(C2(C)CCCN(C(C3CCN(C)C3=O)=O)C2)=O)COC2(CCOC2)C1 C12(CC(C)(CBr)C1)c1nnnn1CCN2.CC(C)CCCN1CCOCC1 Cc1nncn1NC(=O)C(C)C1CCN(C(=O)C(N)=O)C1 C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC(C)C)CC2)CC2(CCC2O)C1 c1(CC(=O)NCC2N(C(COCCCC)=O)CCC2C)c(Cl)cccc1Cl CC1CC2CC(C(=O)N(C)Cc3cc(C(F)(F)F)ccc3Cl)(C2)O1 C#Cc1ccc(C(=O)NCC(O)CCNC(=O)Cc2cc(C)ccc2O)cc1C c1(CC)oc(C(=O)NCC2CCN(C(=O)C(C)Oc3ccccc3)C2)cc1C c1(C(N2CC(C)(NC(C(C)OCc3ccccn3)=O)C2)=O)cc(F)c(O)c(F)c1 CC1(C)CC(CNC(C2CCCCNC2=O)=O)N(C(C2(C)CCOC2)=O)C1 c1(OC(C)C(=O)N(C(C)CNC(=O)Cn2nnc(C#N)n2)C)ccc(Cl)cc1Cl Nc1c(C(=O)NC2CCC(NC(c3ccnc4[nH]ncc34)=O)C2)cc(F)cc1F c1(C(N2CC(N(C(CCNC(=O)NC)=O)CCO)C2)=O)ccc(C(C)=O)cc1F C(CC1=CCN(C(c2cc(Br)cc(F)c2F)=O)CC1)NC(C(C(C)O)C)=O C1(C(=O)NCC2C(NC(=O)CCCC(F)(F)F)CC2)CCc2nnc(O)cc2C1 C1(CC)CC(C)CN(C(CCC2(C#N)CC2)C(=O)NC2CC2)C1 Cc1nc2cc(CNC3CC3C(=O)Nc3nc(Br)cnc3Cl)ccc2s1 C1(CC(=O)OC)CCC(NC(=O)NCCOC(C)C)CC1 c1(C(N2CC(O)(CNC(c3c(CC)non3)=O)C2)=O)c(N)cc(C)cc1F C1(C(=O)NCc2c(F)ccc(C)n2)N(C(=O)CC(C)C(C)C)CCCC1(C)C C1(C2CC2)(CNC(C2C(CC)OCC2)=O)CCN(C(=O)Cc2ccncc2Cl)C1 C1(C(=O)NC2CCC(NC(CCC=C=C)=O)CC2)CNC(=O)C(C)(C)C1 CN1C(=O)CCC1CC(=O)NCC(C)(C)NC(=O)CCN1CCCCC1=O C12(C(=O)NCC(C(=O)NC(C(C)(C)OC)C)C)CCC(C1)C2(C)C c1(OC(CC)C)ccc(C(=O)N(C2CC(NC(c3ncccc3Cl)=O)C2)C)cc1 c1(CNC(C(CCF)NC(C2C(C)=CCS2)=O)=O)cccc(F)c1C C1(NC(C(C)N2CCC2)=O)CN(C(c2ccnc(C(F)(F)F)c2)=O)C(C)(C)C1 c1(NC(c2n(C(CC)C)nnn2)c2ccno2)ccc(OC)c([N+](=O)[O-])c1 O=S(=O)(c1ccc(O)cc1)N1CC2(CN(Cc3ncc(-c4ccccc4)[nH]3)C2)C1 c1(C(C)CC(=O)NCC(O)COC(F)(F)F)cccc2ccccc12 c1(CCC)nnc(S)n1CC(=O)NCC(CC)NC(=O)C(C)Cn1ccnc1 C1(NC(NC(CC)CC)=NCCSC(F)(F)F)COc2c(C)cccc2C1 C12(CNC(C(C)(C3CCC3)NC(=O)COCCCF)=O)CCC(CC1O)C2 c1(OC)cc(N2CCC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)ncn1 Cc1ccc(C(=O)NC(C)C(N2CC(NC(c3sccc3F)=O)C(C)C2)=O)cc1 CCCCCCN=c1ccn2nccc2[nH]1.C(=O)CC1CC1 C1(CNC(CC(C)(C)OC)=O)CC2CCC1N(C(C1CC=CCC1C)=O)C2 C1(CC(=O)NCC(C2CC2)NC(c2cccc(C(F)(F)F)c2)=O)CCC2CC2C1 C1(C(N(CCNC(c2cc(C3CCOCC3)on2)=O)CC)=O)(CC)CCNC1=O c1(C(N2CC(C)(C(F)F)OCC2)=O)nccn2c(Br)ccc12 C(=O)(C1=NOC(C)C1)N1CC2C(C(N(C)Cc3n(CC)cnn3)=O)C2C1 CN1CCC(CC(=O)NCC2CC(NC(c3ccco3)=O)C2)C1=O Cc1ccn(C(C)C(=O)NCC(O)CNC(C)(C)C)n1 Cc1cc(Br)cc(F)c1C(=O)NC1CCN(C(=O)C(O)P(C)(C)=O)C1C S(=O)(=O)(c1cc(C2OCCO2)cs1)NC(CC(=O)OC)CC1CC1 N1(C(=O)CC2CNCCO2)CCC(CCF)(C(=O)O)CC1 c1(NC(c2cc(-c3ccc(C#C)cc3)[nH]n2)=O)c(C)cc(F)cc1[N+](=O)[O-] c1(NCC(C(CC)CC)O)ccc(S(=O)(=O)NCC(C)SC)cn1 C1(NC(c2ccc(C(CC)C)cc2)=O)CC2CN(C(=O)CC3CC3C)CC2C1 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(C)cc(N)c1 C(=O)(CCCC(=O)N1CC(NC(=O)Cc2ccccc2)C2CC12)OCC N1(C(c2c(C)onc2)=O)CCC2CN(C(=O)C=Cc3cccc(F)c3F)CC2C1 N(C1CCc2cc(OC3CCC3)ccc21)C(=O)C=Cc1ccc2c(c1)OCO2.C N1(C(C(C)Oc2ccccc2)=O)C2CCCC1CN(C(c1ccsc1C#N)=O)C2 N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2C=CCCC2)=O)C(CCO)C1 C#CCC(CC(F)F)NC(=O)CC1CCC(NC(c2ccc(CC)[nH]2)=O)C1 C1(CC)CCN(C(=O)C(C)N2CC(C)C2)C1C(=O)NC(CO)C(F)(F)F CC1(C)CN(C(c2n[nH]cc2F)=O)CCC1NC(=O)CC1CCC(C)CO1 c1(C(=O)NC2CC(NC(C3CC(C)SCC3)=O)C2)ccc(S(=O)(=O)CF)cc1 C1(N(C)C(c2coc(O)n2)=O)CCN(C(=O)CCCc2ccc(CO)cc2)CC1 CCC(CC)CC(F)C(=O)NC1CC(=O)N(C2CN(C(=O)CCc3cnc[nH]3)C2)C1 N1(C(CNc2n(C)c(=O)n(C)c(=O)c2C#N)=O)CCOc2c(F)cccc2C1 n1(CC)c(C)cc(C(=O)NC(C(C)NC(=O)CCS(N)(=O)=O)C(C)C)c1C C(=O)(C1=CCCOCC1)NCC1(C)CCCN(C(c2cnn(NCC)c2C)=O)C1 C(=O)(C1=COCCC1)N1C(C)CC(CNC(c2ccc(OC(C)(C)C)cn2)=O)C1 N1(C(COC)=O)CC2CCC2(CCNC(=O)CCP(C)(C)=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC(CC)CNC(=O)CC(C)CN(C)C C12(NC(c3cnc(SC)s3)=O)CCCC1N(C(=O)C=Cc1ccn(C)c1)CCC2 C(C)(C(C(=O)NCc1ccsc1C)C(C)C)NC(C(C1CC1)SC)=O c1(CNC2CCCC(c3[nH]nc(C(=O)O)n3)C2)csc2cc(Br)ccc12 N1(C(C(C)(C)OC(C)C)=O)CCCN(C(c2scnc2C2CC2)=O)C(C)C1 C1(NC(C(C)c2ccsc2)=O)CCCC12CCN(C(=O)C=C(Cl)Cl)CC2 C1(CNC(C(C2CCOC2)OC)=O)CN(C(=O)CC(C)C(C)C)CC(C)(C)O1 C1(C(=O)NCC(C2CC2)NC(=O)C=CCN2CCOCC2)CCC(F)(F)C1 N1(C(=O)OC)CCC(NC(C2CC2CNC(=O)CC2(O)CCCC2)=O)C1 C(=O)(C(C)(CNC(c1cc(F)ccc1F)=O)CC)NC(CC)CN(C)C N1(C(C(ONC(c2cc(SCCC)[nH]n2)=O)C)=O)CCc2nccnc2C1 CCC(C)CC(=O)NCC(C1CC1)N(C(=O)CCC(=O)N(C)C(C)C)C N1(C(c2c(C)c[nH]n2)=O)CCOCC(NC(=O)CC2(C#N)CCCCC2)C1 C1(OCC)CCCCC1NCCO.c12cnn(c1)CCNC(=O)C1CC1NC2=O c1(C(=O)NC23C(n4cc(CC(C)(C)O)nn4)CC(CC2)C3)cnc2ncccn12 C(C(=O)N1CCC(C(N2CCN(C)CC2C)=O)O1)c1cccc(C)c1 c1(N(CCC2CCN(C(c3c(C)cns3)=O)CC2)C)cc(=O)n2ccccc2n1 C1(C(=O)NCCCCNC(c2n(C)nc(C(C)(C)C)c2)=O)CC2CCC(C1)O2 c1(C(=O)NCC2(F)CC(NC(CCC)=O)C2)ccc2c(c1)OCCCO2 C1(OC)CCC12CC(C(=O)NC1(CCNC(=O)C=C(C)C(F)F)CCC1)C2 CC(C)(CC(=O)NCC1CC1NC(C1CNC(=O)N1)=O)C(F)(F)F Cc1cc(C(=O)OCc2ccn(C3CCCC3)n2)nn1C(C)(C)C N1(C(C2(CC#C)CCOC2)=O)CC2(NC(=O)CCc3cc(OC)no3)CC1C2 c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C(C)C)cccc(C2OCCO2)c1 N1(C(CCC2CCN(C(c3c(C)nn[nH]3)=O)C2)=O)CCC2(CNC(=O)O2)C1 c1(C2CCCN(C(C3CCN(C4CCC(N)C4)CC3)=O)C2)nc2ccccc2s1 Nc1c(C(=O)NC2(CNC(C3SC4C=CC3C4)=O)CCC2)cccc1[N+](=O)[O-] c1(C(=O)OC)cnc(Cl)nc1N1CCC(NC(C23CCCN(CC2)C3)=O)C(F)C1 N1(C(C(CCC)NC(=O)C(C)C2(O)CCC2)=O)CC(C)C(C)(CO)C1 CC(C)C(C)C(CNC(=O)COCc1nc[nH]n1)NC(=O)C(C)(C)C C(=O)(CCCN=[N+]=[N-])NC1CC(F)(CNC(CC2N(C)CCC2)=O)C1 c1(C(=O)NCC2CCN(C(CCN(CC)CC)=O)CC2)cccn2cncc12 C1(NC(C(C2CCC2)OCC)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 C1(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(c1cc(N(C)C)ccn1)=O c1(C(N2CCC(C(=O)Nc3nnc(C)o3)C2)=O)cccc(C(F)(F)F)n1 C1(C(N2CCCCC(NC(Cc3nc(C)sc3)=O)C2)=O)CCc2ncncc2C1 c1(C(=O)NC(C2C(C(=O)NCc3nc(COC)on3)C2)C)nc(O)sc1C N1(C(c2c(C)nc(C3CCC3)o2)=O)CCC(F)(CNC(C2(F)CCCC2)=O)CC1 c1(-c2n(C(CC)C)nc(-c3ccc(Cl)cc3)n2)ccc(C)nc1Br N1(C(C2CCC(NC(c3c(C)cc(F)s3)=O)CC2)=O)CCC2(C1)CN(C)C2 c1(C2CCN(C(COc3c(C)cccc3)=O)CC2)cccc2c1OCCO2 N1(C(CC(CC)NC(c2cnn(C)c2Cl)=O)=O)CC(C)(C)OC(C)(C)C1 c1(OC)cc(Br)c(Cl)cc1C(N1CC2(CCCN2c2ncc3[nH]ncc3n2)C1)=O CCC(CNC(c1ccccc1)=O)(CC)C(=O)Nc1ccc2nonc2c1 c1(CN(C(CC(C)N(C)C)=O)Cc2ccsc2)ccc(Br)cc1 N1(C(C2CC(C)C2)=O)CCN(c2ncc(Br)c(O)n2)C(c2nccn2C)C1 c1(N(CCCN(C(C(F)OC)=O)C)C)nccc(-c2ccccc2F)n1 c1(NC(C2CCCN(C)C2=O)=O)ccc2c(c1)CCC2(C)C c1(C(=O)NC(C)CNC(c2ncnc3sccc23)=O)cnc(O)c2ncccc12 C(=O)(CCCC(C)O)N1C(CNC(COc2cccc(C(C)=O)c2)=O)CCC1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CC3OCCC3(C)C)CC2)c(C)c1 N1(C(C(C2CCCN(C(C3CC3C3CC3)=O)C2)C)=O)C2CCC1COC2 c1(OC)ccc2nc(C)c(C(=O)NC(C)CCF)n2n1 C(N=c1[nH]c(N2CCN(C(=O)NC)CC2)nc(=NC)[nH]1)C1N(CCC)CCCC1 C1(C(=O)NC(COC(C)=O)C)CCN(C(=O)CC2(C)CCOCC2)C1C(C)C CN1CCC(CC(N2CCOC(CNC(=O)Cc3cn(C)nc3Cl)C2)=O)C1=O c1(C(=O)NCC(CO)NC(C(C(C)C)C)=O)ccc2c(c1)CCCCN2 c1(C(=O)NC2CC(CC)C23CCC3)c(OC)c(Cl)cc([N+](=O)[O-])c1Cl N1(C(COC2CC(NC(CCC(C(C)C)=O)=O)C2)=O)CCCC2CN(C)CC12 Cc1cc(O)nc(C)c1C(=O)NC1CN(C(=O)CC(C)(C)CN(C)C)C(C)(C)C1 C1(NC(=O)C(c2ccc(F)cc2)O)CN(C(=O)COCCCF)C2(CCCC2)C1 C(CNC(c1cscc1C)=O)(CCOC)NC(COCCCC)=O c1(CN(C)CCOCCN(C(=O)CCCC2CCCC2)C)cc2n(n1)CCCC2 C1(CCNC(c2ccc(C3CC3)s2)=O)CC(F)(F)CN1C(C1C2CCCOC12)=O N1(C(CCn2ccc(C)n2)=O)CCN(C(=O)C(F)F)C(C)C1 c1(OCC(=O)NC(C(C)C)(C)CNC(C2(C)CNC(=O)C2)=O)cccc(F)c1F O(NC(=O)CCOCCCN(C1CC1)C(C)C)CCOCCOC c1(OC)ncc(C(N2CCCC(CCNC(C)=O)C2)C(=O)NC(C)CC)cn1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C3CCCO3)C3CC3)C2)ncn1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)cc2sc(F)cc2[nH]1 c1(C(C)NCCC2CCCO2)ccc(I)cc1 c1(C(N(CC(c2ccccc2)C)C2CC2c2ccsc2)=O)ncc(F)cn1 c1(CNC(Cc2ccc(C)s2)=O)ccccc1CNC(C1C=CCC1)=O C(=O)(C(C)C(F)(F)F)N(CC1CCN(C(c2cnc(CC)s2)=O)CC1)CC C=C(C)C(CC(=O)NC(COC)C(=O)Nc1cccc(CO)c1)OCC C1(NC(C2C(C)C2)=O)CN(C(C2CC2C(F)(F)F)=O)CC1O c1(C(=O)NCCCN2CCN(C(C3(C)CC3(F)Cl)=O)CC2)cccc(N)c1O c1(CN(C(=O)C(C)c2ccsn2)CC(C)C)cn(CC(=O)O)nn1 c1(C(=O)OC)nc(N2CC3CC2CN(C(=O)COC(F)F)C3)c(F)c(Cl)n1 C1(NC(C(=O)NCC)=O)CN(C(=O)Cn2nnnc2C)CC12CCOCC2 N1(CCN)CCc2cc(CN3CC(NC(c4cc(CO)on4)=O)C(O)C3)ccc21 n1(CC)nc(C)cc1C(N1CCCC1C(=O)NCc1nn[nH]n1)=O CCC(C)(C)C(C)CC(=O)N1CCC(F)(CNC(=O)CCC2CCCCO2)CC1 Cc1cc(COC(c2cc(N3CCNC3=O)ccc2C)=O)nc(C)c1.C1C(=O)O1 c1(CC)ccc(C(=O)NCC2CC(C)N(C(=O)C3=CCCCC3)C2)c(O)c1 CCC(CC(F)F)C(=O)NCC1CN(C(=O)CSS(C)(=O)=O)CCC1C c1(C(N2CCC(N(C(C3CC(CC)OCC3)=O)C)CC2)=O)nccc2occc12 Cn1cc(Cl)cc1C(=O)NC1CCN(C(c2c[nH]nc2Cl)=O)CC1 c1(C(N)=O)ccc(C(=O)NCCNc2ccc(C=O)cn2)cc1.c1(S)ccccc1 C1(=O)CC(CC)N1.C1(CNC(=O)NCCC(=O)OCC)COC(CC)C1 CN1CCN(C(=O)Cc2cscn2)C(CNC(=O)COC2CCCOC2)C1 c1(CCCNC(c2n(CCCC)nnn2)(C)CC2CCCC2)ccccc1Cl C1(NC(C2(OCC)CCC2)=O)CN(C(c2cc(C)n(C)c2)=O)CC1N=[N+]=[N-] C(C)(C)(C(=O)NCC(C)NC(=O)CC=CC(C)(C)C)OCCC CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC(C)NC(c1cc2n(c1)CCCC2)=O C1(C(C(=O)N(C(C)CNC(=O)C=Cc2c[nH]cn2)CC)=O)CCCCC1 C(C(C)(C)CC(=O)N(CC(=O)N(C)C)C)NC(CCCNC(=O)OC)=O CC(C(F)C(=O)NC1CCN(c2ncnc(Cl)c2Br)CCC1CO)C(F)(F)F c1(OCC)ncc(C(=O)NCC(N2CCOC(CC(C)C)C2)=O)cc1F c1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)cnn(CCC)c1Cl c1(C(=O)NC2CC3CN(C(CCC(=C)C)=O)CC2C3)ccc2c(n1)CCC(C)C2 C(CCCCC(=O)NCC1CC12CCOC2)N(C(c1n(C(C)C)ccc1)=O)C N1(Cc2c(C)cc(F)cc2)CCC2CC(C(=O)NCC(O)CO)C2C1 c1(Cc2nnc(CN(CCc3ccc(OC)cc3)C)n2C)nc2ccccc2s1 c1(C(N2CC(NC(CC(CC)CN(C)C)=O)(CO)C2)=O)cc2ncc(C)cn2n1 c1(C(=O)NC2CCCOC2)n[nH]c2cccc(-c3ccc4[nH]ccc4c3)c12 N1(CCc2cn(CC)nc2)CCC(NC(=O)Cn2cc(Cl)cn2)CC1C N1(C(c2cn(CC)nc2)=O)CC2CCCCC2(CNC(c2cncc(C)c2)=O)C1 Cc1cccc(-n2cc(C(C)(O)C(=O)O)nn2)c1Br.c1(C)cc[nH]c1C1CCC1 C(=O)(C(C)(F)C(C)(C)F)NC(C(C)C)C(=O)NC1(C)CCCCCC1 N1(C(=O)CCc2ccccc2N2CCCS2(=O)=O)CCN2CCOCC2C1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(C(=O)NC2(CNC(C(C)(C3CC3)OC)=O)CC2)ccc2c(c1)CC2 C1(c2ccc(CC)o2)CCCCCN1C(=O)Cc1cscc1Br CCC(C)C(O)C(C)C(=O)NCCc1cc(C(N2CC(C)CCC23CC3)=O)no1 C(=O)(C(C)C(C)c1ccc(F)cc1)N1CC(CC=C)(NC(=O)CCOCC)C1 CC1C=C(C(=O)N(C(C)CCNC(c2csc(C3CCCCC3)n2)=O)C)CC1 C1(CC)CN(C(c2ccnn2CC(F)(F)F)=O)CCC1NC(=O)COCCCF CC(CN(C)C)C(=O)NCCSCc1cn(C2CCCC2)nn1 CC(C)C(C)(C(N)=O)NC(=O)C(C)NC(=O)CNC=O C1(C(N(CCC(C)NC(=O)C2=CCCSC2)C)=O)CCC2C(C1)C2(F)F N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(C2CC(C3CC3)C2)=O)C2(CCC2)C1 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)Cc2cncnc2)CC12CC2 c1(NCC(=O)COC2CCCCC2)ncc(O)cn1.C12CN(CCO1)C2 c1(N2CC(C)C(NC(C3CC34CCOCC4)=O)C2)nc2ncc(Cl)cc2s1 N12CC3(CCOCC3)C1c1cn(nn1)C(C)(C)CC2=O.CC(C(=O)O)C1CC1 C1(CN(C(C2(CC#C)CCC2)=O)C)COCCN1C(c1ccnc(CC)n1)=O C(CN=[N+]=[N-])(C(=O)NCC(C)(C)C1CC1)NC(Cc1c(C)n[nH]c1)=O c1(C(N2CC(N(C)C(c3cccc(F)c3N)=O)C(F)C2)=O)cc2cccnc2s1 CC1CC(NC(C2CCCO2)=O)CCN1C(c1ccc(C(F)(F)F)c(O)c1)=O C(C)(C(=O)N1CCCCO1)OCCNC(COC(CC)CC)=O N1(SCNC(CC(C)c2ccco2)=O)CCC(C)N(CCSc2cccc(Cl)c2)CC1 C1(C(=O)NC2(CN(C(=O)CCOc3cccc(F)c3)C)CC2)CCCC(F)C1 CCCCC(C(=O)NCCC1(NC(c2c[nH]nc2OC)=O)CC1)N(C)C N1(C(C2(SC)CCC2)=O)CCCN(CCNC(=O)Cc2cccc(C)c2)CC1 c1(C(N(C2CCN(C(C3(C)CC3(F)Cl)=O)CC2)CCO)=O)n[nH]c2c1CCC2 c1(CNCc2nc(C)sc2)ccc2occc2c1O.C12(CCC1)CC(=O)N2 C1(N(C)C)(C(=O)N)CCOCC1.C1(NC(C=CC)=O)CCC1N(C)C c1(CN(C)CC2CCN(C(C3C(C)CCC3)=O)C2)nnc(S(C)(=O)=O)s1 c1(C(=O)NCC(CC=C)NC(=O)C(C)=C2CC2)cccc2cnccc12 C(=O)(C(C)(C)c1nncn1C)NCCC(C)NC(=O)CCCNS(C)(=O)=O Cc1nsc(C(N2CCC(C(=O)NC3CCC4CCC34)C2)=O)c1N N1(C(C2OCCN(CC)C2)=O)CC(NC(c2ccnnc2S)=O)CC(F)C1 C(C)(CCC(=O)N1CCCC1CNC(c1cnc(C2CC2)o1)=O)OC Clc1cccc2c1OCC2Nc1nccc(=NCCc2ccoc2)[nH]1 C1(CNC(CCn2c(C)ncc2)=O)CCCCC1NC(C1(CCF)CC1)=O c1(C(N(CCn2cc(C(N3CCOC3=O)C)nn2)CC)=O)cnc2[nH]cncc1-2 c1(C(N2CCN(C(CNS(CC)(=O)=O)=O)CC2C)=O)c[nH]c(C)c(Cl)c1=O C1(C2CCC2)(C(N(C(CNC(c2cc(O)cs2)=O)C2CC2)C)=O)CC1(F)F N1(C(C(C)OCCC=C)=O)CCN(C(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 CC1(NC(=O)Cc2ccsc2)CCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 N1(C(C2Sc3c(ccc(C)c3)C2)=O)CCC2CN(C(c3ccsn3)=O)CC2CC1 C1(NC(C(COC)C)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 N1(C(CC(C(C)C)C)=O)CC2(CCC(CNC(C34CC(CO)(C3)C4)=O)O2)C1 c1(C(=O)NC(C2CCCCN2C(C2CN(C3CC3)C2)=O)C)cccc(Cl)c1 C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(=O)C(O)CC2CCCC2)CC(O)C1 c1(C(=O)NCC2(NC(C3(CO)COC3)=O)CC3CCC2C3)ccn2nccc2n1 N1(C(CCCCOCC)=O)CCCCC12CN(C(=O)Cc1cc(C)on1)C2 Cn1cc(Cl)cc1C(=O)NCC(C)(C)OCC(=O)NCC1CC(C)(O)C1 N1(Cc2nc(C(F)F)sc2)CCCC(c2ccc(Cl)cc2)C1 N1(C(C(N(C(c2cc(C)c(C)s2)=O)C)C2CC2)=O)CC(C)(C)C2COCC12 C1(N=[N+]=[N-])(C(=O)Nc2c(C)cc(O)nc2)CCN(C(c2cccs2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)cc[nH]c2=N)=O)F)ccnc2ccc(F)cc12 S(=O)(=O)(c1cn(C2CC2)nc1C1CC1)Nc1c(C(=O)OC)ncs1 N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)Cn2cc(Br)cn2)C2(CC2)C1 c1(OC)ncc(Br)c(C)c1C(N1CCCCC1)=O.N12CCCC(C1)NC(=O)C2=O c1(CCC(=O)NCC(C)CNC(=O)CC2COC(=O)N2)ccncc1 c1(OC)cc(-c2nc(-c3cccnc3)nn2C2CC3CCC2C3)ccc1C(=O)O N1(C(CCNC(CCOCCOCC)=O)=O)CCC(CO)CC1C C1(C)(CNC(c2cnc(OCC)nc2)=O)CCC(NC(=O)CC2CCCC2)CC1 c1(OC(C)C(N2CC=CC(NC(=O)C(C(C)O)N(C)C)C2)=O)cc(F)cc(F)c1 Cc1cc(=N)[nH]cc1C(N1CC(CCNC(=O)C=CC(C)C)OC(C)C1)=O CC(C)CS(=O)(=O)CCC(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O N1(C(C(=O)NCC)=O)CCC2(NC(=O)C(F)CC(C)(C)C)CCCCCC12 N1(C(c2nc(CCCC)sc2)=O)CCCCC1C(C)NC(=O)C(C)=C(C)C N1(C(C2(CSC)CC2)=O)CC(C(N2CC(O)(CN(C)C)C2)=O)C(F)(F)C1 C(=O)(C(F)CCCCC)NC(C(=O)N(CCCCCC=C)C)COC C1(NC(c2ccc(OC)s2)=O)CC(O)CN(C(c2nocc2C)=O)C1 c1(C(N2CCCC(NC(CC(C)CF)=O)C2)=O)cccc(O)c1[N+](=O)[O-] C=CCC(C)(C)C(=O)NCc1ncc(C(=O)O)s1 Cc1cc(C)c(C(=O)NCC2CC(NC(c3ccc(C#N)cc3F)=O)C2)c(=O)o1 C1(CCNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(C2CC2)n1)=O N1(CC(=O)NC(CC)CN(C)C)c2ccccc2CS1(=O)=O CC1=CCC=CC1C(=O)NC1CCC(C(=O)Nc2scc(C)c2C)C1 Cc1nc(N(CC(O)CN(C)C(c2cc(C(N)=O)ccn2)=O)C)c2c[nH]nc2n1 C1(CNC(CC(=O)NCC)=O)CN(C(c2c(Br)noc2C)=O)CCO1 Cc1nc(C(N2CCCCC2CN(C(=O)CC2COC(=O)N2)C)=O)c(C)s1 C1(CC(=O)N(C2CCN(C(c3ccon3)=O)CC2)CC)CC2(CCC2)CCO1 c1(CCC(=O)NCC(C2CCCN(C(C3CCOC3)=O)C2)(C)O)cncnc1O c1(C(=O)NCCCN(C(CC2CC(CC)OCC2)=O)C)c(C)nn(C2CC2)c1Cl c1(OC)nn(C)cc1C(N1CCCC(CCNC(=O)C=CC2CCCN2C)C1)=O CC1CC2CCC(C1)N2C(C1COCC1NC(c1occ2c1CCC2)=O)=O N1(C(c2ncn(CCNC(Cc3ncn(C)c3)=O)c2)=O)CCCC(CCO)CC1 c1(CC)nccnc1C(=O)NCCC(O)CNC(=O)C=C1CCCCC1 Cc1cc(CNC(=O)C=CC(C)NC(c2ccc(C)c(O)n2)=O)nc(C)c1 c1(C(=O)NC2CN(C(=O)CCNC(N)=O)CC2F)ccc2cncc(Br)c2c1 C1(C(=O)NC2C=CCN(C(CC3(OCC)CCOCC3)=O)C2)CCCC2(CC2)C1 CC(C)CC(C(=O)N1CC(C)(O)C1)N(C(=O)CC1CCCC1O)C N1(C(c2c(OC)cccc2)=O)CC(NC(=O)C(C)C(C)(F)F)C2(CC2)C1 C1(C(N2C(C(C)NC(C(C)NC(COC)=O)=O)CCC2)=O)C(C)(C)C1(C)C C#Cc1cnc(C(N2CCC(C3CC3)C2C(=O)NOCC2CC2)=O)c(C)c1 CC(CC(C)(C)C)C(=O)NCCCO.C1(N2CCC2=O)CCN(CC2CC2)C1 N1(C(CC2C(C)(C)C2)=O)CCN(C(=O)CN2CCN(C3CCO3)CC2)C2(CCC2)C1 N1(C(CNC(=O)COCCNC(=O)COc2cn[nH]c2)=O)CCC(C2CCC2)C1 C1(C(=O)NC(CCO)C2CCC2)(CNC(CCSC)=O)CC=CC1 C(C(C)(C)CC)(c1nnnn1C1CC1)NCC1(CC)CCCC1 N1(c2nc(N3CCS(=O)CC3)c3c(n2)scc3)CCCCC2(CCCC2)C1 c1(OC)ccc(C=CC(=O)Nc2ncc(Cl)nc2Br)cc1S(N)(=O)=O c1(CN(CCC)C(C2CCCN2C(=O)C=CC2CCCC2)=O)ccccc1 C1(NC(CC#N)=O)CCN(Cc2cc(Br)co2)C1 Cc1ccc(C(N2CCCC(NC(C3(C4CC4)CCC3)=O)C2)=O)cc1C CC1CCN(C(C2(C(C)(C)C)CCC2)=O)CC1CNC(c1nccc(N)c1Cl)=O c1(CN2CCC(N(C(CC(CC)O)=O)C)C2)cc(OC)ncc1Br N1(C(C(=O)N(C)C)=O)CCN(C2CCC(NC(=O)COC3CCCCC3)C2)CC1 CC(C)(C)CC(F)C(=O)NC1(C(N2CC(NC(=O)C3CC3)C2)=O)CCCCC1 N1(C(c2cc(OC)ns2)=O)C2CCC1CN(C(=O)C(C)(O)C1CC1)C2 O=C1CCC(C(=O)NC23CC2CN(C(=O)C(F)=C2CCCC2)C3)n2cccc21 Cc1cc(C(=O)NC(C)(CNC(=O)COC(F)F)C(C)C)c(C)o1 C1(C(=O)NCC(C)C#N)CCCC(NC(=O)C=CC2CCCN2C)CC1 N1(C(C2C(COC)C2)=O)CCN(C(=O)C=Cc2cncc(O)c2)C(CC(F)F)C1 Cc1sc(=O)n(CC(N2CCC(NC(C3CCN(C)C3=O)=O)C(O)C2)=O)c1C C1(C)(C(=O)NCc2n(CC)cnc2)CN(C(=O)C(C)CC#N)C(C)(C)C1 c1(NC(C2(CCNC(CC3CCCC(=O)N3)=O)CC2)=O)cncc2ccccc12 N1(C(C2CC3N(C(C4C(C)C4C)=O)C(CC3)C2)=O)CCCC12CCNC2=O C(CCOCCO)(C(=O)NC1CCCC1CCSC)NC(CSCC=C)=O C#CC1(O)CC(C(N2CCC(CO)(CNC(=O)C(C(C)C)SC(C)C)C2)=O)C1 CC1=C(C(=O)N(CCCCCNC(C2(C3CC3)CC2)=O)C)Cn2ncnc2N1C C(=O)(CCCCN=[N+]=[N-])NC1(C)CCN(C(=O)C#CC2CC2)C1 C12(C(N(CCN(C(=O)C(COC)OC)CC)CC)=O)CCCN(CC1)S2(=O)=O n1(C(CC)CC)nc(-c2ccc(N)cn2)nc1CCc1ncc(C)o1 c1(NC(C)=O)ccc(C(C)C(=O)OCc2nc(-c3ccccc3)no2)cc1F Cc1ccc(NC(C2CC3CCN(C2)C3)=O)c(-n2cc(C3(C)COC3)nn2)c1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NC2CN(C(=O)C=CSC)CC3CC23)c1 C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(C2CC3(CC(=C)C3)C2)=O)(CO)C1 C1(NC(c2cc(Cl)sc2Cl)=O)(CNC(C2(CO)CC2)=O)CC2CCC1CC2 C1(NC(=O)COC2CCC2)CN(C(=O)CCCc2cncs2)CC2(CCC2)C1 C(=O)(C1=CC2CCCCCC12)N1CC(CNC(C2CC3(CCC3)CO2)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)CC2CCCN2C(C)C)nccc(OC)n1 N1(C(CN2CCCC(CC)C2)=O)CC2(NC(=O)C(COC)OC)CC1C2 N1(CC)CC(C(=O)NC2CC(NC(=O)C=CC(=O)N(C)C)C2)NC1=O c1(N(C)Cc2ccc(C)s2)nc2cc[nH]c2c(=NC2CC2c2c(Cl)cccc2Cl)[nH]1 CC(C)C(C(=O)N(C)CCNC(C1CC(F)(CO)C1)=O)NS(C)(=O)=O C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C)C(c2ccc(C(N)=O)nc2)=O)C1 C1(NC(C2C(C#C)C2)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CC1C=C CCC(C(=O)OC)C(=O)NCc1csc(C(=O)NC2CC2c2cnn(C)c2)c1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CC2CCC1C(NC(C1CCCOC1)=O)C2 Cc1cnncc1C(=O)NC(CNC(=O)CCCNC(=O)C1CC1)CC(C)C CCCCCCCN(C(=O)CCN(CCCO)C(c1conc1C)=O)C N1(C(CC(C=C)CCC)=O)CCN(C(c2cnc(O)cc2OC)=O)C2(CCC2)C1 CCC(C(C)(C)C(=O)OC)NC(=O)CCCCCn1cc(C(O)C(C)C)nn1 O=C(CCCCC(F)(F)F)NCCC1CCN(C(=O)C(F)OC(F)(F)F)C1 CSC=CC(=O)N1CCC(OCCNC(C2(F)CCOC2)=O)C1 CCC(O)C(C)C(=O)N(C(C)CCNC(=O)C(c1ccc(Cl)cc1)C)C CC1(NC(=O)CCC2CCCCN(C(=O)CCCC3CC3)C2)CCCC1(F)F n1(CC(=O)N(CCN(C(C=C(CC)C)=O)C(C)C)C)ccc2c(C)cccc12 Cc1cc2ncnc(N3CCC(NC(C4CC(O)C4)=O)C(C)C3)c2[nH]1 C1(C(N2C(C)CN(C(=O)CCC(C)(F)F)CC2)=O)CCC2(CCC2)CO1 c1(C(N2CC(C)(C)CC2C)C(=O)NCCOC)ncc(Cl)cc1F N1(CC(N2CCC(C)C(CNC(C3(C)CCC3)=O)C2)=O)CCc2sccc2C1 c1(C(=O)NCC2CC(NC(CS(=O)(=O)NC)=O)C2)cc(=O)c2ccc(Cl)cc2o1 CCC1=NOC(CC(=O)NC2(CCC(N3CCC(CCOC)C3)=O)CCC2)C1 C(C(C)(C(=O)NC(C)COCCOC)NC(C1CC1C(C)(C)C)=O)SC Cc1ccc2ncc(C(=O)NC3CC4CCC3(NC(=O)C(F)C3CCC3)C4)n2c1 Cc1cc(=NCC2CCCC23CCC3)[nH]c(N2CCN(C3CCCC3O)CC2)n1 C(CN=c1[nH]c(N2CCC(CN3CCOC3=O)C2)nc2c1CCC2)N(C)C c1(SC)cc(N2CCCC(CNC(=O)CCc3cnc[nH]3)CC2)nc(SC)n1 C1(C(=O)NC(C)CCCNC(=O)Cc2n[nH]c(=N)s2)CN2CCC1(C)CC2 C(CC(=O)N1CCN(C(c2cc(N)cc(O)c2)=O)CC1CO)(C(N)=O)NC(C)=O c1(C(=O)OC)ccc2c(c1)CC(C)N2C(c1ccc2cnc(C)n2n1)=O Cc1cnc2c(Br)c(C(=O)NNC(=O)Cc3cccc(O)c3)nn2c1 Cc1c(C(=O)NC2CC3(NC(=O)COCC4CC4)COC2C3)cc(C(C)C)n1C c1(OC)cnc(C)cc1C(=O)NCC1CCN1C(=O)Cc1sccc1Cl CCC(O)(CC(=O)Nc1cccc(NC(c2nsnc2O)=O)c1)c1ccccc1 c1(CC)c(C(=O)NCC2(C(F)F)CCN(C(c3cnccn3)=O)C2)cccc1F C=CC(C)(O)CC(=O)NCC1CC(NC(c2sccc2Cl)=O)CCO1 C=CCC(CC(=O)N1CC(c2ccccc2)C1)NC(=O)C(C)CC(=O)OCC Cn1ccnc1CCC(=O)NCC(C)(C)CC1CC1.C12CC(O)C1CC(=O)N2 c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)c2c(nn1C)CCSC2 N(C1c2ccccc2OCC1OCC)CC1(COCC=C)CCCNCC1 Cc1nc2cc(C(=O)Nc3ccc4c(c3)CCCC4O)c(F)cc2[nH]1 c1(OC)cc2cnccc2cc1C(=O)OC(C1CCN(C2CC2)CC1)C C1(NC(Cc2ccc(OC)cc2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC1C c1(OCC(=O)N(CCNC(=O)CC2(CO)CC2)CC)nc(Cl)c(Cl)cc1Cl c1(C(=O)NC(CNC(c2cc(C)cc(O)n2)=O)CC(C)C)ccnc2[nH]nnc12 Cc1ccnc(C2CCN(C(=O)C(N3CCCC(CN(S(C)(=O)=O)C)C3)=O)C2)c1 c1(C(N2CC(C)(C(=O)NC(C)CCO)C2)=O)ccc(F)cc1Br N1(C(C2OCCN(C)C2)=O)CCCC2(C1)CN(C(c1nn(C)cc1N)=O)CCO2 C(=O)(CCS(C)(=O)=O)NC(CCOCC)C(=O)NCC(O)C(F)(F)F N1(C(C(CC)(C)OC)=O)CCN(C(c2cccc3cncn23)=O)CC2(CC2)C1 c1(C(=O)OC)cncc(C(N2CC(CC(=O)Nc3c(Br)cnn3C)C2)=O)c1 c1(OC)nccc(C(=O)NC2CCCC2NC(c2cnc(-c3ccco3)s2)=O)n1 C#CC(C)(C)C(=O)NCC(CCC)NC(=O)C(C1CCCCC1)O c1(OCC)c(C(C)NC2CCN(c3ccc(Cl)cc3)C2)c(C)nn1C c1(C(C(=O)NC2CCC(NC(C3CC=CC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(-c2cccc(CNC(=O)NCc3cc(C)no3)n2)ccc(NC(N)=O)cc1 Cn1cnc2cccc(CNC3(c4nnnn4C4CCCC4)CC4CCOC34)c12 C=C(Cl)C(C)(C)C(=O)N1CC(CC(C)NC(=O)CSCc2ccccc2F)C1 CCC(C)(C)C(C(=O)NCC(C)NC(=O)COc1ccccc1C#N)OC c1(C(C)NC(CCCC#C)c2nnnn2C2CC2)c(F)cccc1Br C1(C(=O)NC2CCC(F)CC2)CC2(CC2)CN1C(c1nc[nH]n1)=O c1(C(N(CC(=O)NCC(=O)NCC2CC2)CCC)=O)sc(C)cc1C Cc1cc(F)sc1C(=O)NC(c1ccccc1)CNC(=O)C(C)NC(C)(C)C c1(C(=O)NCCCN(C)C(c2ccnc(CO)c2)=O)ccc([N+](=O)[O-])nc1 n1(CC(=O)NC(C(C)NC(c2ccn(C(C)(C)C)n2)=O)(C)C)cccnc1=O CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(CO)N(C(c2ccccc2)=O)C1 N1(C(c2cnc(C)s2)=O)CC2OCC(NC(c3ccccc3CO)=O)C2C1 CN1CCCC(C(C)(C)C(=O)NC2(c3ccccc3)CC(F)(F)C2)C1 N1(C(CC(CC)C2CC2)=O)C2CCC1CC(N(C)C(c1cc(=O)c(C)c[nH]1)=O)C2 c1(C(N(CCNC(c2c(C)n(CCN(C)C)nc2)=O)C)=O)cccc(F)c1C C12(C(=O)Nc3c(OC)cc(C(N4CCOCC4)=O)cc3)CCC(F)(CC1)CC2 C1(CCC)CN(C(=O)CNC(=O)NC)CCN1C(c1cnn(C)c1N)=O Cc1ccc(C(N2CCC(NC(=O)CC34COC(CF)(C3)C4)CC2C)=O)c(N)c1 C1(C(N(CC(C)NC(CCc2cc(C)[nH]n2)=O)C)=O)CCC(=O)N1C N1(C(CC(C)NC(c2ccccc2)=O)=O)CC(F)CC1C(C1(C)CCC(=O)C1)=O Fc1cccc(-c2ncc(CNc3ccccc3N3CCCC3)s2)c1 Cc1nc(CNC(=O)CC2CCC2)oc1C(=O)NOCCOCCF C(CCCCC(=O)N(C(C)C(N1CCC(C(C)O)CC1)=O)C1CC1)OCC C(CC(C)CCNC(=O)C(O)c1ccsc1)NC(Cc1nc(C)[nH]n1)=O N1(CC(=O)OC)CCC2(CC1)CC2C(N1CC2CCC1(C)C2)=O C=CC(CC)CC(=O)N1CC(CNC(c2cc(Cl)n[nH]2)=O)C(F)(F)C1 C1(CCC)CCCN(C(c2cc(CNC(C3(OC)CC3)=O)ccn2)=O)CC1 c1(C(=O)NCCC2(C)CCN(C(CC(=C=C)C)=O)C2)c(C)cccc1N C(=O)(C(=O)N=c1ccn(CCC#N)[nH]1)N(CC(C)C)CCN(C)C S(=O)(=O)(c1ccc(Cl)c(OCC(F)F)c1)Nc1cn(C)c(=O)c(Br)c1 C#CC1(C(=O)Nc2cncc(Cl)c2)CCN(C(=O)C(CN(C)C)CC)C1 C1(C(=O)NCCCc2ccco2)C2CN(C(C3(O)CC(CF)C3)=O)CC12 CCC(CCC(=O)NCCN1C(=O)CNC1=O)NC(c1ccc(Cl)cc1)=O c1(C(N(CCCNC(=O)C(O)C(C)C)CC)=O)cc(C2CC2)ncc1Br C1(C(N(CCCN)CCS)=O)CCCN1C1CCCC1.N1(CC(=O)CC)CC=CC1 c1(NC(c2ccc(-c3c(C)cccc3)cn2)=O)ncc(F)c(Cl)n1 C#CCCCCC(=O)NCc1ccc(CCNC(=O)CC2CCC(C#N)C2)cc1 N1(C(COC(C)(C)C)=O)CCCC(CC(=O)NC2CC(N(C)CCO)C2)CC1 C#CCC(C)(C(=O)NC(c1nccs1)C)NC(=O)CC1CC(CC)=NO1 c1(OC)ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)Cc2cccc(Cl)c2)c1 c1(C(=O)NC(C)C)cc(C2=CCC(C(C)(C)C)CC2)[nH]n1 C=CC(F)(F)C(=O)NC(C1CCCN(C(c2cc(F)n(C)n2)=O)C1)C N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(=CC3CCCC3)C)CCC2C1 c1(C(CN2CCCC(CN(C(C)C(N3CCOCC3)=O)C)C2)O)ccc(F)cn1 N1(C(CC=CC)=O)CCC2(CC1)CC2(CO)CNC(=O)C(C(C)C)n1cncn1 c1(C(N2CCC(CC)C2C(=O)NCC2(CF)CCC2)=O)cc(O)cc(F)c1 C(=O)(C1CCCn2ncnc21)NC1CC(C)N(C(c2scnc2Cl)=O)CC1 CC1=NOC(=O)C1CC(=O)NCC=C1CCN(C(c2cc(Cl)ccn2)=O)CC1 C1(C2CN(C(C3(c4cc[nH]n4)CC3)=O)C2)(NC(C(c2cccnc2)C)=O)CC1 N1(C(CC(=O)OC)=O)CCN(C(c2cncc(SC)c2)=O)CC1C c1(C(=O)NC2C(NC(C3C(SCC)CCC3)=O)CCC2)ccnc2c1ncn2C c1(CNC(C2CNC(=O)N2)=O)ccc(C(N2CCC(N3CC(O)C3)C2)=O)cn1 C1(C(=O)NCCN(C(=O)CC2CC2c2ccccc2)CC)COC(=O)N1 N1(C(C)C)CC(C(N2CCN(C3CCN(C(=O)C=CBr)C3)CC2)=O)CC1=O C12(C(=O)NCCOCCC(C)C)C(NC(=O)CCS(N)(=O)=O)C3CC1C2C3 N1(C(CC(C)C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)CCC1CCCO1)C2 n1(CCC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(CF)C2)nn1 C12(C(=O)NC(CCCC)CNC(c3sccc3CC)=O)CC(C)(C1)OC2(C)C c1(C(=O)NCCOCCN(C(=O)CC2CCC(=O)O2)C)cnn2c1OCCC2 CCCCC(C)CCC(=O)N1C2CCC1CN(C(C1(P(C)(C)=O)CC1)=O)C2 N1(C(c2nc(C)c(C)s2)=O)CCC(C(=O)OCc2c(Br)cnn2C)CCC1=O N1(c2nccc(OC)n2)CCN(C(c2cccc(F)c2I)=O)CC1OC(C)=O C(=O)(C1CCCc2ccccc21)NCCC1CC(NC(c2cc(C#N)oc2)=O)C1 CCC(CC(=O)NCC1(NC(=O)Cc2ccn(C(F)F)n2)CC1)CC(F)(F)F N#CC1CCCC(C(=O)NCc2ccsc2C(N2CCC(O)(CO)C2)=O)C1 n1(CCC(=O)N(CC(OC)OC)CC(F)F)cnc2sccc2c1=O CC1CN(C(=O)Cc2cncnc2)CCC1NC(C1C2(CC2)C12CC2)=O C1(C(N(CC(C)N(C(=O)C=CC(=O)NC2CC2)C)C)=O)CCCCS1(=O)=O C(=O)(CCCNC(c1occc1C)=O)NCC(COC)O C1(O)(CNC(c2n(C=C)nnc2)=O)CCCN(C(C2(N(C)C)CCCCC2)=O)C1 Cc1ccccc1CN(CC(O)CN(C)C(c1ocnc1C)=O)C C1(CNC(=O)C2=CCC2)C2CCC(C2)N1C(=O)Cc1cccnc1O N1(C(CCNC(C#CC(C)(C)C)=O)=O)CCC2CCC(C1)N2C CC1CCN(C(=O)C(=Cc2cccn2C)F)CCN1C(C1CCCNS1(=O)=O)=O N1(c2c(C#N)cncc2)CC(NC(=O)C2COc3ccccc32)C2(COC2)C1 N1(C(=O)CC(F)F)CCOC2(CCN(C(C3CCN(C4COC4)C3)=O)CC2)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(CC)OC)c(C)cc[nH]c1=N Cc1cc(C(N2CCC(C)(NC(=O)COC3CC3(F)F)C2)=O)cnn1 N1(C(C=CC)=O)CCC2C(NC(c3cc(C(C)(C)C)oc3C)=O)C2CC1 N1(C(c2cc(CC)[nH]n2)=O)CCC2(CCCC2C(=O)Nc2ncccn2)C1 C1(NC(CCc2onc(CC)n2)=O)CCCCC1CNC(c1c(Cl)n[nH]c1C)=O c1(CC)ccc(C(=O)NCCC(O)CNC(C2(C(C)(C)C)CCCC2)=O)c(C)n1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NCCCc1ccccc1)C2 N1(C(C(c2ccc(OC)cc2)O)=O)CC2CN(C(=O)C=CC(C)C)CC12 c1(C(=O)NC(CC)C(N2CCCCC2COC)=O)ccc(C)n1C N1(C(c2c(C)cc(OC)c(OC)c2)C(=O)NC2CC2)CCC2(C=CCO2)C1 C1(C(N2C(CC)CN(C(=O)CN(CC)CC)CC2)=O)CCCC2(CCOCC2)O1 C1(CC#C)(C(=O)NC(CNC(=O)CCn2cnnn2)C2CCC2)CCCCO1 C(CCN(C)C)(C(=O)N1CC(CC(N)=O)C1)NC(C(C)CC1CCCC1)=O C1(CCC)CN(C(C2CC(=C(F)F)C2)=O)CCN1C(C1CCN(C)C(C)C1)=O N1(CC)CC(C(N2CC(OC)C(NC(c3ccoc3Br)=O)C2)=O)CC1=O C1(CNC(CN(CC)CC)=O)CCN(C(c2scnc2C2CC2)=O)CC1 c1(C(=O)NCC2(CNC(c3ccc(CCC)s3)=O)CC2)ncccc1OC(C)C c1(C(=O)NC(C2CCN(C(=O)CC3(C#N)CC3)CC2)C)cc(O)cc(O)n1 C#CCC(CC(F)F)C(=O)NC(CCC(C)C)C(=O)NCCCNC(=O)C(C)(C)C C1(C(=O)NCc2nc(COC)sn2)CC2(CCC2)CN1C(=O)OC(C)(C)C C#Cc1ccc(OC)c(C(=O)NCC2CCN(C(=O)C(=O)NC3CC3)CC2C)c1 n1(CC)nncc1C(=O)NC1CCC(CC(=O)NCC2CC2c2ccncc2)C1 C(=O)(C1=COCCO1)NC(C1CCCN1C(=O)C(O)CCN(C)C)C C12(CNC(c3n(CC#C)ccc3)=O)CC1CN(C(C1C=CC=CC=C1)=O)C2 c1(CNC(C2(F)C(C(=O)O)C2)=O)cnn(C2CCOCC2)c1.C12CCN1C2=O Cc1ncc(Br)c(C(=O)NCC(C(C)(C)C)NC(=O)CC2CC=CC2)n1 c1(C(N2CC(CC(=O)NC3CSC(C)C3)(OC)C2)=O)cc(C)c(C)o1 Cc1ccc(C)c(OCC(N2CCC(O)(NC(=O)COC(C)(C)C)C2)=O)c1 N1(C(C(C2CCCCC2)C)=O)CCCC1CCCNC(=O)CC1CCC(O)C1 C1(C(=O)NCC(COC)(F)F)C(C)CCN1C(c1ccc(C#N)[nH]1)=O N(C1COc2ccc(Cl)cc21)C(c1ccc(C)s1)c1nnnn1C1(C)CC1 c1(C(=O)NC2(C3CCCN3C(c3cc(C4CCC4)on3)=O)CC2)cccnc1O S(=O)(=O)(C(C)CN=c1[nH]c(=NCC2CCCCC(F)(F)C2)[nH]c2cc[nH]c12)NC C1(CC#C)CCCCN1C(=O)C(c1ccnn1C)NC(=O)C(C1CCCCC1)C C1(O)(C(C)NC(C2CC(C(F)F)C2)=O)CCN(C(c2csc(Cl)c2)=O)C1 c1(C(=O)NC(CCC)CCCNC(C2CC=CCC2C)=O)n[nH]c2c1CCSC2 c1(OC)ccc(CC(C)C(=O)N(CCCNC(=O)C=Cc2ccoc2)C)cc1F c1(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2(C)CC2)ccn(C)c(=O)c1O CCCCCS(=O)(=O)CC(=O)NC1CN(C(c2cnc(CC3CC3)s2)=O)CC1O c1(C(N(C2CC(C(N)=O)C2)C)=O)coc2c1CN(C(=O)C(C)(C)F)C2 C1(C(=O)NC2(C(N3CCC(CCOC)CC3)=O)CC2(C)C)CCCC12CCC2 N1(C(=O)Cn2cnnc2O)CC2(CNC(C3CC34CC(F)(F)C4)=O)CC1CO2 C1(NC(C2(COC)CCC2)=O)(NC(=O)C(=O)NC2CC2)CC(O)C1 C1(CNC(c2ccc(Cl)nc2)=O)CCCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 c1(CC)cccc(C(=O)NCC2CN(C(=O)CC34COCC(C3)C4)CC2C)n1 C1(CNC(c2ccnc(-c3cccnc3)n2)=O)C2CN(CC3CS(=O)(=O)C3)CC12 Cc1nccnc1C(=O)N(CCN(C)C(C1COCCC1C)=O)C(C)C N1(C(C(C2CCC2)NC(CCCC(CC)C)=O)=O)CCc2nnnn2CC1 CCCCS(=O)(=O)NC1C2CN(Cc3scnc3C)CC12 N1(C(c2c(OC)ccc(O)c2)=O)CCN(C(=O)C(C)=C2CCC2)CC(C)(F)C1 c1(C(N2CCC(NC(Cc3c(OC)cccc3)=O)C2C)=O)cc(O)c(F)cc1N C1(O)(NC(C(C)N(CCCCCNC(c2c[nH]nc2C(F)F)=O)C)=O)CCOCC1 N1(C(CNC(CNC(C)=O)=O)=O)CC2CN(C(c3cnsc3C)=O)CC2(C)C1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1cc(CO)[nH]n1)=O C(=O)(CCC(C)CN(C)C)NCCC1(O)CN(C(C(C(=O)OC)C)=O)C1 C(CC(=O)N1CC2=C(C1)CN(C(c1c(C)nsc1N)=O)C2)(C(F)(F)F)OC N1(CC(=O)NCCN(C(=O)C=C(C)CCC)CCC)CC=CC1 CN1CCc2ccc(C(=O)NCCC3CN(C(C4CC4(C)C)=O)CCO3)cc21 N1(C(C(CC)CC)=O)C2CCC1CC(NC(=O)C(O)Cn1cncn1)C2 CC(N=c1nc(N(CC(F)(F)Br)C)c2c([nH]1)CCS2)c1cnc2n1CCCC2 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(C(CC)(F)F)=O)CC1C C1(C(=O)NC2C(CNC(Cc3n(C)ccc3)=O)CC2)CC2(C1)CC(F)(F)C2 c1(CC)nc(CNC(=O)C(=O)NC2(c3ncon3)CCC2)c(Br)s1 N1(C(CC2C(C)CCC2)=O)CC2(CCCC2NC(C2CN(C)C(=O)N2)=O)C1 C1(C(N(CCCN(C(COc2ccc(OC)cc2)=O)C)C)=O)CCC2C1C2(F)F C12(C(N(CCCCC(=O)NC(CCOC)C)C)=O)CCC(C1)OC2C C1(CNC(C(C2CCC2)OCC)=O)(NC(=O)CC2OCCO2)CCCCC1 O=C(C1=CC2CCCCC12)NC1CC(CNC(=O)C(O)CC2CC2)C1 Cc1ccnc(O)c1C(N1CC2CC(NC(=O)CC3CCS(=O)(=O)CC3)C2C1)=O C1(NC(c2cccc(OCCC)c2)=O)CCCCN(Cc2ccc(SC)s2)C1 c1(C(N2CCC(C)(CNC(C(C)(C)CCF)=O)C2)=O)nc2ncccn2n1 Cc1cc(C(F)F)oc1C(=O)NCC(C)CNC(c1ncc(C(F)(F)F)n1C)=O C1(C(N(CC(C)(C)C(=O)NC2CC3CCCC3C2)C)=O)Cc2ccccc2C1 c1(N(CCN(C)CC2CCSC2)C)nnc(-c2ccccc2F)n1CCC#N c1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)c[nH]c2cc(F)c(F)cc2c1=O Cc1nc(C)n(O)c1C(N1CCN(C(=O)CC(C)C)C(c2nccn2C)C1)=O CON(C)S(=O)(=O)c1ccc(C(N2CCN(C(c3cc(F)c[nH]3)=O)CC2)=O)cc1 c1(C(N2C(C)CC(NC(=O)C(C)C(F)(F)F)CC2)=O)ccc2cnccc2c1 N1(C(C(C)n2cccn2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 c1(N2CCN(C(=O)OC(C)(C)C)C2)nccc(=NCc2cc(F)cnc2Cl)[nH]1 N1(C(C(C)(N(C(Cc2ccc(C)nc2)=O)C)C2CC2)=O)CCCC(C)C1CO CC(O)C(C(=O)NC1CCN(C(=O)Cc2ccccn2)C1)NC(=O)OC(C)(C)C C1(C(=O)NCCN(C(C2CCC2c2nc[nH]n2)=O)CC)CCNC(=O)C1 C(CCC(C(=O)NC1CCOC1)N1CCC(O)CC1c1ccccc1)OC C1(C(=O)NCC(C(=O)OC)C)CCN(C(=O)C=CC(C)C)CC1C(N)=O N1(C(CC(=C)Br)=O)CC2(CC(NC(c3cn(CC)nc3C)=O)CO2)C1 C1(NC(C(c2cnn(C)c2)OC(C2C(C(=O)OCC)C2)=O)=O)CCN2CCCC2C1 C1(CNC(c2csc(C(F)F)n2)=O)CCCN1c1nc(C2CC2)ns1 C1(C(C)C)CC(CNC2CCN(c3ccccc3)C2)CCO1 N1(C(CC2N(CC)CCOC2)=O)CC2CCC(C1)N2C(=O)C(O)CN(C)C C#Cc1cccc(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)c1Cl C(=O)(C1=CCN(C(c2ccc(C)c(C)c2)=O)CC1)NC(C1CCOC1)C#C Cc1cc(C(=O)NC2CC(C(=O)NC(CO)CCO)C2(C)C)n(C)n1 C(CS(=O)c1ccccc1)SCc1nc(C(C)C)on1.c12ccccc1OC2=O Cc1nc(C(C)(C)C)ncc1C(=O)NC1CC1NC(C1CC(=O)N(C)C1)=O C1(CC(=O)NCC2(C)CCN(C(CC3CC(OC)C3)=O)C2)Cc2ccccc2O1 c1(CC)ccccc1S(=O)(=O)N1CCCC(CCN)C1 N1(CC(=O)N(CC=CC(=O)NC2CCC(OC)C2)C)CCC(C)CC1 C(=O)(C(C(C)C)N(C)C)N1C(C(C)NC(CC2(CSC)CC2)=O)CCC1 C12(C(N3CC(N(C(C4(CC)CCCCC4)=O)C)C3)=O)CCC(F)(CC1)CC2 c1(CC(C)OC)nc(C2=NOC3(CCOC3)C2)n(-c2c(F)cccc2F)n1 CC1(C)CC2(CC(NC(=O)CN3CCN(CCC(=O)NC4CC4)CC3)C2)C1 C12(C(=O)NC(C)CNC(=O)C=CC(CC(F)(F)F)=O)CCOC1CCOC2 CC(C(=O)NCc1csc(C(=O)NC(C(N)=O)C(C)O)c1)S(N)(=O)=O c1(CCC(=O)NC2C(C)N(C(c3sccc3F)=O)CC2)ccc(Cl)c(F)c1 C1(NC(c2nc(C)sc2)=O)CC12CCN(C(=O)C(F)CCNC(C)=O)CC2 C(CCC(C)(C)C(=O)NC(CC)C(C)O)NC(CCC=C=C)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC1CN(C(=O)C(C)N(C)C)CC1O Cc1c(O)ccc(C(N2CCC(CNC(=O)CCC3CC3(C)C)C2(C)C)=O)c1C N1(C2(CS(=O)(=O)N(CC(=O)OC)C)COC2)c2ccccc2Sc2ccccc21 c1(OC)cc2c(c(S(=O)(=O)NC3c4ccccc4C4CC3C4)c1)OCC2 c1(-c2cn(CC(=O)Nc3coc(-c4ccc(Cl)cc4)n3)nn2)cnccc1OC c1(C(=O)NCC2N(C(Cc3c(C)n[nH]c3)=O)CCCC2)ccc(Br)cc1C#N CC(C)(C)CC(C(=O)N(CCC#N)CCN1CCOCC1)N1CCC1c1cccs1 c1(CC)c(C(=O)NCC2CCCC(NC(c3cc(C)on3)=O)C2)nnn1CC N1(CC)N=C(C(=O)N2CC(OC)C(NC(=O)C(C)CO)C2)CCC1=O CN1CCN(CCN(C(=O)CC2CCN(C(=O)C(C)(C)NC(N)=O)CC2)C)CC1 C1(NC(C2C=CCN(C(c3c(C)cccn3)=O)C2)=O)CCC(O)C(O)C1 c1(C(N2CCN(C(C3C(=C)C3)=O)C(C3CCCC3)C2)=O)cc(Cl)c(F)cc1N Cc1cc(C(F)F)nn1CC(=O)NC1CC1NC(C1(F)CCC1)=O CC1(C)CC(C(=O)NCC2(C)CCCN2C(C2CC3(CCC3)C2)=O)CCO1 Cn1cc(C(=O)NC2CN(C(c3cnc(OCF)cn3)=O)CC2F)c2ccccc12 c1(OCC#C)ccc(C(=O)NCc2cc(C3CC3)on2)cn1.C1(=O)C(=O)NC1 C1(CNC(CC(=O)N(C)C)=O)Cc2ccccc2CN1C(c1c[nH]c(C#N)c1)=O CCC(CCCC(=O)N1CCSC(C)CC1)NC(c1cnnn1C)=O Cc1cccc(OCC(=O)NCC2(NC(=O)CC(C)C3CC3)CCOCC2)c1 N1(C(C(CCOC)C)=O)CC(NC(c2ccnc(C)c2N)=O)CC(C)C1 N1(C(C2N(C(C(C)N(C(C)=O)C)=O)CCCCCC2)=O)CCC2(C=CCO2)CC1 c1(C(N2C(C)CC(NC(C3(COCC)CC3)=O)C2)=O)cncc(Br)c1C N1(C(C(CCCC)C)=O)CCCC2(CCN(C(=O)C(c3c(C)noc3C)C)C2)C1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 c12ccc(Cl)c(c1N)N(C(=O)CCOC)C2=O.C(C(=O)OC1CCC1)SCC#C C1(C(=O)NCCn2c(C)nnc2)CC2CC1CC2NC(=O)COC(C)C N#Cc1cc(F)ccc1C(=O)NCC1(F)CC(CNC(C2(C3CC3)CCC2)=O)C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)CNC=O)C4CCCCC34)cc12 C1(N(C(=O)CCn2cnnn2)CC)CCN(C(=O)CN2CCOCC2)C1 C(C(=O)Nc1cn(C)nc1C)(C(C)C)NC(CCc1onc(C)n1)=O C(=O)(CCC(C(=O)N(C1CN(C(c2cc(C)ccc2Cl)=O)C1)C)N(C)C)OC c1(CC(=O)NCCC2(C(=O)NC(c3cn(C)nn3)C)CC2)nc(=N)cc[nH]1 C1(C(C)C)CN(C(=O)Cc2nccn2C)CCC1NC(=O)CN(C)S(N)(=O)=O C1(C2CCCN(C(=O)C(c3cccnc3)O)C2)(NC(=O)C(F)(F)C2CC2)CC1 C1(C(NOCCC(=C)C)=O)C2CN(C(C3CCC(C)(C)C3)=O)CC12 N1(C(C2OCCC(C)C2)=O)CC2CCCC(C1)N2C(=O)C=CSc1ccccc1 CCC(F)(F)C(=O)NC1CCCCC1CNC(c1nncs1)=O C(=O)(C(C)(C)C(=O)NCCCN(C)C(C1CCS1(=O)=O)=O)OCC c1(C2(C(=O)NCC(CNC(C(F)=CCC)=O)F)CCCC2)c(F)cccc1F C1(C)(CCC)CCN(S(=O)(=O)Cc2ncoc2CCC)C1 O=C1OC(C(=O)OCCOC2CCCC2)Cc2ccc(F)cc21 c1(CC)cc(C(N2CCC(CN(c3ncc(C)cn3)CC)CC2)=O)c(C)nn1 C(CCC(C(=O)NCCc1cccc(O)c1)NC(=O)Cn1nc(C)oc1=O)OC C(CC(C)C(=O)NCCCN(C)C(c1ccc(CO)cc1)=O)=CCC c1(C(=O)NCC2OCCN(C(C=C(CCC)C)=O)C2)ccc(Cl)c(C(=O)OC)c1 N1(C(CNC(=O)NC)=O)CCC(C2CCCN(C(C3CC4(C3)CC4F)=O)C2)C1 N#Cc1cccnc1NC(C1CCN(Cc2cc(-c3cc[nH]n3)ccc2F)C1)=O CC1(C)C(C(=O)NCC2CC(NC(=O)Cn3cccn3)C(O)C2)CCS1(=O)=O C(=O)(C1=NOC2COCC12)NC1C2CC(NC(c3cc4n(n3)CCO4)=O)CC21 c1(C(=O)NC2C(C)CN(C(c3cn(CC(F)(F)F)cn3)=O)C2)cc2[nH]ccc2s1 N1(CC(=O)NC(C)C(CO)NC(=O)CC2CC2(C)C)C(=O)CNC1=O c1(C(N(C)CC2(O)CN(C(c3cc(CC(C)C)on3)=O)C2)=O)ccc(O)c(F)c1 c1(C(C)(C)F)cc(C(=O)NCC2C=CCN2C(c2cncc(F)c2)=O)ccc1F O=S(=O)(c1ccc(NCCO)c2cnccc12)NC1CC(Cl)(Cl)C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCOCC(NC(C2(C)C(C)CCC2)=O)C1 CC(F)(F)C(C)(C)C(=O)NCC1(C2(O)CN(C(=O)C(c3ccccc3)O)C2)CC1 C(CCN=C(NCC1CCCC1O)N1CCC(C2CC2)C1)OC c1(C(=O)OCC)cc(C(C)NC(C2(c3ccn(C)n3)CC2)=O)c[nH]1 C(=O)(C1=NOC2(CCC2)C1)NC(C(C)(C)C)CNC(=O)COCc1cccnc1 C(CC1=CCN(C(=O)CN(C2CCCC2)C)CC1)NC(C(C)OCC=C)=O c1(CC)sc(C(=O)NC(C)(C)C(C)NC(c2ccc(OC)o2)=O)cc1Br c1(C(=O)NCC2N(C(C(CN(CC)CC)F)=O)CCC2)cc([N+](=O)[O-])ccc1O CC12CCCCC1CN2C(C1CN(C(C2CC2Cl)=O)CC12CC2)=O CCC(C)CC(=O)C(=O)NCCCN(C(=O)Cc1cnsc1)CC C(CCCN=[N+]=[N-])NC(C(C)N(C(=O)CSc1cn[nH]c1)C)=O c1(-c2n(C)ccc2)ccc(C(N2CC3CC2C3CNC(c2ccc[nH]2)=O)=O)cc1 CCC(C(=O)N(C1CC1)CC)N(C(=O)CN1CCOCC1)C c1(C(N(CCC(N2CC(C)(O)C2)=O)C)=O)cc(O)nc(O)n1 N1(C(C(Cn2cncn2)NC(c2cnsn2)=O)=O)CC2CC2(CO)C1 C1(C)(CNC(C2CC(C)OCC2)=O)CCN(C(=O)CCSCC(N)=O)CC1 N1(C(c2cnc(C)s2)=O)CCCCC(C(=O)NCC(O)(CO)CO)C1 N12CCC3(CC(C3)C1=O)C2.C1(NC(c2c(C)non2)=O)CC(C)N(C2CC2)C1 C1(=O)CC(C)CO1.C1(CCC)CCN(c2nnc(C)s2)C1 c1(C(N(CCCNC(=O)C(C)CO)CCC)=O)ccnnc1C C(=O)(C(C)(C)C1=CCSCC1)N1CC(O)(C(C)NC(C2CC3CC2CC3O)=O)C1 c1(CC(=O)NC2CCN(C(c3coc(Br)n3)=O)C2)ccsc1Br C(=O)(C(CNC(=O)C(F)=C(C)C)CC1CC1)N(CCN(CC)CC)C Cc1cccc2sc(NC(=O)C(N3C4CC5CC(C4)CC3C5)C)nc12 C1(F)(CNC(CCSCCCC)=O)COCCN(C(=O)CC(O)CC)C1 C(=O)(CC1=CCN(C)CC1)NC12CN(C(c3cccc(C)n3)=O)C(C1)C2 N1(C(C(C)c2ccco2)=O)CCC2(CCN(C(c3nnc4ccccn34)=O)C2)C1 N12CCCC(C1)CC2=O.Cn1ncnc1CNNC=O N1(C(c2onc(CC)n2)=O)CC2CC(NC(C3CCCS3)=O)C2C1 Cc1c[nH]c(C(=O)NCCC(C)NC(c2cn[nH]c2)=O)c1C CCC(C)C(O)CC(=O)NC(Cc1ccco1)C(N1CCCC2COCC12)=O N(C1c2cc(OC)c(OC)cc2CCCC1(C)C)C(C(CC#C)C1CC1)=O c1(C(C)C)ccc(C(=O)NCCCN(C(=O)CC2CCCOC2)C2CC2)cn1 Cc1nn(C)c(C)c1OCC(=O)NC(C1CCN(C(=O)CCn2ccnn2)C1)C C(N=c1[nH]c(N2CC3CC2CN3C(C)(C)C)nc2c1SCC2)c1n(C)ncc1 C(=O)(C(C)(C)C(=O)NCC(CNC(=O)C(CC1CC1)CC1CC1)CO)NC CS(=O)(=O)C1(C(N2CCCC(F)(CNC(C3CC3Cl)=O)C2)=O)CCC1 c1(C(c2cccs2)NC(COCC)C(C)C)cc(C)c(OC)cc1C C(=O)(CC(C)(C)CNC(c1cncn(C)c1=O)=O)NCC(=C)Cl C(=O)(CCCCCCCBr)NCC1N(C(c2[nH]cc(C)c2C)=O)CCCC1 CCCCC(O)C(C)C(=O)NCC1N(C(c2cncc(OC)c2)=O)CCC1(C)C C1(C(N2CCC(NC(C3CC(OC)(OC)C3)=O)(CF)C2)=O)CCn2ncnc2C1 c1(C(=O)NCC(C)=CC(=O)NCC(C)(CO)CO)cnc(O)cc1C C1(C(=O)OC)CC2(CC(NC(=O)N(CC(C)OC)C)CCO2)C1 N1(C(c2cccc(C(N)=O)n2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 c1(C(N2C(C(=O)NCc3cnc[nH]3)CC(O)C2)=O)ccc2nc(Br)sc2c1 c1(C(N2CCC(F)(C(=O)NC3(CCC)CC3)C2)=O)c(O)cccc1F N1(C(c2cnc(CC)[nH]2)=O)CC(CO)C2(CCN(c3nnc(O)s3)CC2)C1 c1(N2C(C(=O)Nc3ccc(N(CC)CC)cc3)C(C)CC2)ncnc2[nH]c(C)nc12 C1(C(N2CCC(C(C)NC(=O)CSCC#N)CC2)=O)CCC2C(CC1)C2(F)F c1(NC(c2ccc(Br)cc2I)=O)cc(Oc2ccccc2)nc(Cl)c1 Nc1cc(F)cc(C(N2CCCC(CO)(NC(c3coc(Cl)c3)=O)C2)=O)c1N CCC(C(=O)NCCn1cc(CNC(C2CN(C3COC3)C2)=O)nn1)C(C)O c1(NC(N2C(C(CC)O)CCC2)=O)cc2cnccc2nc1C C(=O)(CC(C)(C)CNC(C1(F)CCCCCC1)=O)NC1CCCC(C(C)C)C1 C(C(C)(C)CCNC(c1cscc1C(=O)Nc1cnc(C2CC2)o1)=O)OC C1(NC(c2nc(C)sc2C)=O)CN(C(c2ccnc(C)c2C)=O)CCC1CO CN1C(C(=O)NC(C2CCCC2)CNC(=O)CC2(C3CC3)CC2)CCS1(=O)=O C(C1CN(C(C2CN(C)CCO2)=O)CC1C(=O)NCCOCC(F)F)=CC C(CCCC(=O)NCC1CCC1NC(c1cncn1C1CC1)=O)SC C#CCC(CC#C)C(=O)N1CC(CCCCNC(C2CC2(Cl)Cl)=O)C1 c1(CNC(C2(COC)CCN(C(=O)C=CCCC(C)C)C2)=O)nc(C)ccc1C N1(C(C2CCN(OC)CC2)=O)CCN(C(c2csc3nnsc23)=O)CCC1C N1(C(CNC(CC)=O)=O)CC(CNC(=O)Cc2sc(O)nc2O)CC12CCC2 C(c1ccc(O)cc1)=CC(N1CCC(C(C)(C)C)(CNC(C(N)=O)=O)C1)=O c1(CC)cccc(C(=O)NCCCC(CO)NC(C2CCC(N(C)C)C2)=O)n1 c1(OCCC(=O)NC)cccc(Cl)c1.C1(C(N2CC(O)C2)=O)C(F)(F)C12CC2 Cc1c(C(=O)NC2CN(C(=O)C(F)C3CCC3)C3(CCC3)C2)c[nH]c2nccc1-2 C1(C(=O)OC)CCCC(C(=O)N(CC(C)CNC(=O)C(C)Cc2ccco2)C)C1 N1(C(C(C=CCCC)O)=O)CCC2(CCCN2C(C2CCSC(C)C2)=O)C1 C(CC(C)(C)C(=O)N1CC(NC(C2CC=CCC2)=O)C(C(F)F)C1)SC c1(C(=O)NC(C(C)NC(C2C(C=C)C2)=O)(C)C)cc(Cl)c(Cl)cc1C C=CC1(C(=O)N(CC(C)(C)C#N)C)CCN(C(c2cc[nH]c2C)=O)C1 Cc1[nH]c2ccccc2c1C(=O)NC(C)Cn1ccccc1=O Cc1cc(NC(C2CCCCN2C(=O)CCc2ccccc2)=O)c(N(C)C)nn1 CN(C)NC(=O)CCC(=O)NCC#CC(=O)NCc1cc(O)ccc1F Cc1cc(F)c(C(N2CCC(N3C(=O)CNC3=O)C2)=O)cc1C(F)(F)F C(C1=NOC2CN(C(=O)CSCCOC)CC12)NC(c1onc(CC)c1C)=O N1(C(CSCC)=O)CC(NC(=O)CCCc2sccc2C)CC(O)C1 C=CCC(C(=O)N1CCC(CNC(=O)C(N2CCSCC2)C)(COC)C1)N(C)C N1(C(c2ccc(C#C)cn2)=O)CC2CCC(CNC(=O)Cc3cnc(C)[nH]3)C2C1 C1(C(N2CC(N3CCN(C(CCCCC)=O)CC3)C2)=O)CCc2nnc(O)n2C1 C1(C(N2CCCC(CNC(C(C=CC)O)=O)C2)=O)CNc2ccnn2C1 C1(CC(=O)NCC(C)N(C(=O)C(C)(C)C#N)C)CCC(F)(F)CC1 Cc1cc[nH]c1C(=O)N(CC(O)CN(C(=O)C(F)CC1CCOC1)C)C Cn1cnn(CC(=O)NCC(C(C)(C)C)NC(C2C=CCC2)=O)c1=O c1(C(=O)NC(CC(C)NC(=O)Cc2c(F)cncc2Cl)C)csc([N+](=O)[O-])c1 CCC1(CC)CNC(=O)N(C(=O)C=C(C)CN(C)C)CC(=O)N1.C(C)(C)(C)O.CC CCCCC(C)CCC(=O)NCCC(C)(C)C(=O)NCCCCN(C)C1CC1 c1(C(N2CC(N(C(=O)CCNC(N)=O)C)C(C)(C)C2)=O)c[nH]c2cc(F)ccc12 C1(NC(C2CC(=C)C2)=O)(CF)CCN(C(c2cnn(CCOCC)c2)=O)C1 c1(CC(=O)NC2(C)CCCN(C(C3CC(SC)C3)=O)C2)ccc2c(c1)CCC2 C(CN=c1cc(NC2CC2c2nc(C(F)(F)F)cs2)nc(C)[nH]1)NS(CC)(=O)=O N12CCC1(C)CC2=O.C(CC(=O)N(C(C)(C)CO)CC)=CC=C N1(c2c(C)ccc(C)n2)CCC(CSc2ccccc2)CC(C)(C)C1 CC(CC(F)(F)F)C(=O)NC1CCCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C1(C(N2CCCC(C)(CNC(c3sccc3Cl)=O)C2)=O)CC2(C1)CC21CCC1 C1(CN(C(c2nc(C)sc2)=O)C)C2CN(OC(F)F)CC12.c12cccc(c1)N2 c1(OC)ccccc1N1CCC(NC(=O)CNCC2(F)CC2(F)F)C1 N1(C(NOCC(C)(C)C)=O)CCCCC1c1ccc(C2(O)CCCCC2)o1 N1(C(C(CCC)=CCC)=O)CC(NC(C2(n3cccn3)CC2)=O)CC(O)C1 c1(C(N(CC(=O)NCC)C)=O)cnn(CCNC(C2(C)CCOC2)=O)c1 N1(C(CC(COC)C)=O)CCN(C(=O)Cc2ccsc2C)CCC1C N1(C(Cc2cc(C)sc2)=O)CCC(C(=O)NC(c2c(C)noc2C)C)CC1C c1(C(=O)NCCN(C(C2C3C4CCC(C4)C23)=O)CC)cc2cnccc2[nH]1 CC1CC(C(=O)NCC(C)(C)CO)CN(C(C2(CO)CC3(CC3)C2)=O)C1 C12(C(c3ccccc3)=O)CCCC(C)(C1)OC2.C1(OC)C=CC(NC(=O)CCC[NH+]([O-])CC(=O)O)C1 C1(C(N2CC(C)(C(N(CCNC(C(C)C)=O)C)=O)C2)=O)C2CCCCCC12 C1(NC(CN(CCC#C)C)=O)CC2CCC(C1F)N2C(=O)C(C)Cn1ccnc1 C1(CNC(C(C)OCOC)=O)CCCCN(C(C2C3CCCCCC23)=O)C1 c1(NCc2cn(CC)nc2)cccc2cc(O)ccc12.C(=O)CCCCCBr CC1(C(=O)NCCC2CCC(F)(F)CC2)CCCN(Cc2ccc(F)nc2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCOCC(NC(C(c2ccccc2F)OC)=O)C1 CC1CCCc2c(C(N3CCC(Cc4ccccc4F)CC3)=O)cnn21 c1(C(N2CC[Si](C)(C)CC2)C(=O)NCC2(C(=O)OC)CC2)sc2ccccc2c1Br C(=O)(C(CCS(C)=O)N(C)C)N1CCC(CN(C(C=Cc2ncc(C)[nH]2)=O)C)C1 c1(OCC(=O)NC(C)CCCNC(=O)CC(=O)NC(C)(C)C)nn(C)cc1[N+](=O)[O-] C1(CNC(C(C)OCCOC)=O)CN(C(c2oc(SC)cc2C)=O)CC(C)(C)C1 c1(C(N2C(C(=O)NC3CCCCC3)CSCC2)=O)c(F)cc(Cl)cc1Cl c1(C(N2CCOCC2)=O)ccc(C)s1.n12cc(nn1)CCC(=O)NCC(OC)C2 CS(=O)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(=O)Cc2cncnc2)s1 c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1nnc(O)nc1O)=O C1(C(N2C(CNC(C(COC)C)=O)CC2)=O)CCC(NC(C)=O)CC1 CCCCC(O)C(C)C(=O)N1CCC1C(=O)Nc1ccc(C2CC2)nc1 N1(C(C2CCN(C(c3cnn[nH]3)=O)C2)=O)CCCCCC1CCO N1(c2cc(SC)ncn2)CCCC(CNC(c2ccc(C)cc2)=O)CC1 C1(=O)CCC(=O)NCC(NC(C2CCCN2C=O)=O)CN1.c1(COC)nccs1 C=CC(C)C(=O)N1CC=CC1C(=O)NC(C)Cc1nncn1C c1(C(N2CCCC(CCNC(C(CC#C)O)=O)C2)=O)ccnc2cc(C)ccc12 N1(c2ncc(C)cn2)CCN(C(c2ccc(OC(C)C)cn2)=O)CCC1C Cc1cc(OCCC(=O)NCCN(C(=O)C2=CCCC2C)C)c(C)c(C)c1 CC(C)(C(=O)NC(c1ccccc1)CC1(Cl)CCC1)c1cc[nH]n1 C(=O)(CCCCC#N)NCC(C)CNC(C1CCCCCC1)=O N1(C(CN(CCN(C)C)CC)=O)CCCC(CC(=O)NCC2(C)CCCCC2)C1 c1(C(=O)NCC(C)CNC(C23CCC(CC2)CC3)=O)ccc2sc(O)nc2c1 N1(C(c2cncc(C)n2)=O)CCCC(C)C1CCNC(=O)C(F)(F)CC1CC1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(O)CCNC(c1coc(OC)n1)=O CC(C)C(O)C(=O)N1CCCCC1CCN(C(=O)CC(C)O)C N1(C(c2cccc(SCCCC)c2)=O)CC2CCN(C(=O)C(C)C(C)O)C2C1 C1(C)(CC)CC(NC(=O)C2CC2)CN1C(C1(c2cccnc2Cl)CC1)=O C#CCC(C)(C(=O)N(C)CC1CC1C)NC(=O)CCNC(=O)CC c1(C(=O)Nc2ccnc(OC(C)C)c2F)ccc2c(c1)C(=O)N(C)C2=O c1(CC(=O)NCC2CCN2C(c2cc(Br)cc(F)c2F)=O)ccc([N+](=O)[O-])cc1 c1(CC(=O)NCC(C)NC(C(CCC)C)=O)c(C)nn(C)c1C C12(CNC(c3n(C)ncc3Cl)=O)CC(CO1)N(C(=O)CC(C)(C)C1CC1)C2 C1(CC(=O)N(CCCN(C)C)CCNC(C(C)n2ccnc2)=O)CCCC1(F)F c1(C(N2C(C)CC(CNC(C3(C(N)=O)CC3)=O)C2)=O)cc2ccc(F)cc2s1 C1(C(=O)NC(C=C)(C)C)CCC(C2CC2)N1C(c1cnn(CCO)c1)=O C1(C)(C(N(CCCNC(c2ccc(C)s2)=O)C)=O)CCc2ccccc2C1 CC(CC(=O)NC(C)(CNC(C1(c2ccncc2)CC1)=O)C1CCC1)NC(N)=O O=C1OC2CN(C(C34CSCC3C4(F)F)=O)CC2O1 c1(C(C(=O)NCCCSCC)N(CCCN(S(C)(=O)=O)C)C)ccc(F)c(I)c1 N1(C(C(C(C)C)SCC)=O)CC(NC(C2CCC(C)(C)CC2)=O)C2CC2C1 Cc1cc(NC(=O)N(C)C(c2ccco2)c2ccco2)c(Br)nc1C C(=O)(C1=CCS(=O)(=O)C1)NCCC1OCCN(C(c2cc(C#N)sc2)=O)C1 CC(C(=O)NCCCN(C(=O)C(C)(C)Nc1ccccc1)C)C1=CCCC1 c1(OC)ccc(C(N2CCN(CCN3C(C)CCC3C)CC2)=O)cc1C(F)F N1(C(CCSC)=O)CC2(C(=O)NCCc3ccon3)CC1CO2 C1(C(C)NC(c2cc(CCCO)on2)=O)CCCN(C(=O)COC2(C)CCC2)C1 N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(c3ccn4cncc4c3)=O)C2)C1 N1(C(CCC2CCCN(C(=O)Cn3ccc(O)n3)C2)=O)CC2CCCC(C2)C1 C1(NC(=O)CC2(CO)CC2)CCN(C(=O)CNCc2ccccc2)C(C2CC2)C1 CC1CN(C(c2ccsn2)=O)CCN1C(C1CC2C=CC1C2)=O c1(N2CCC(C(=O)NC)C2)ncnc(NCC2CCC(C)(C)O2)c1C C1(NC(C2(CS(N)(=O)=O)COC2)=O)CCCCN(C(C2CC23CCOC3)=O)C1 C(=O)(CCCCCC#N)N1CC(CC(C)NC(c2c(CC)nc(C)o2)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1csnc1Br)=O N(C(=S)N1CCC(N2CCOC2=O)CC1)CC(=O)N(C(C)C)C1CC1 c1(C(=O)NC(CNC(CC2(C(=O)OCC)CCC2)=O)C2CC2)n[nH]cc1Cl c1(CC)cccc(C(N2CCC(C)(CC(=O)NCCC3CC(=O)N(C)C3)C2)=O)n1 C(=O)(C1=CCCC1C)N1C(CN(C(CN(c2ccc(Cl)cn2)CC)=O)C)CCC1 C(=O)(CC(C)(C)CC(F)F)N1CCC(C)(NC(C(CCCCC)O)=O)C1 N1(C(c2n(C)nnc2)=O)CC(CNC(c2cnc(C3CC3)nc2)=O)N2CCC1C2 N1(C(c2ncc(OC)nc2)=O)CC(O)CCC1C(=O)NCCc1ccco1 Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)N2)=O)ccn1C(C)C C1(CC(=O)Nc2cccc(C(C)C)c2)CC2(C1)CN(Cc1ccncc1O)C2 C(=O)(C(C)(C)CC1CCOC1)N1CCC(C(C)(C)NC(CCN(CC)CC)=O)C1 CCC(CC)CC(F)C(=O)NC12CCC(C(=O)NCCCc3ncco3)(CC1)C2 CCC(CC(=O)NOCCC(F)F)NC(=O)CNc1cnn(C)c1 c1(C(=O)NC(CNC(c2c(CCC)occ2)=O)C2CCC2)ccc(CSC)cn1 CC1C(C)N(C(CC2CCC(C)(C)O2)C(=O)NCc2cccs2)CCS1=O CCC(C)CCCC(=O)NCCCNC(=O)CC1CC2CCC(C1)N2C C1(NC(C(C)C2CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)CC1F c1(C(=O)NCCC(=C)CNC(=O)Cn2ncnn2)cc(S(=O)(=O)CC)cnc1O c1(C(N(CC(CC)NC(C2CCCCN2CC(F)F)=O)C)=O)c(C)n[nH]c1C N1(C(CS(CC)=O)=O)CCC(C2CC(NC(=O)CSC3CCCC3)C2)CC1 c1(-c2cncc(NCc3cc(OCC)cc(C)c3)c2)cc(F)c(F)c(F)c1 c1(C(N2CC(OC)C(NC(c3cnc(O)o3)=O)C2)=O)ccc2nc[nH]c2n1 c1(C(N2CC(OCCNC(=O)CCc3ncc[nH]3)C2)=O)cccc2c1CCOC2 c1(C(c2ccc(Cl)cc2)N(C(C(=O)NC(CCSC)C)=O)C)ccccc1C CC1(F)CN(C(C2(CF)CCC2)=O)CCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(CCN(CCC)C)=O)CCn2nc(CNC(c3sc(C)cc3Cl)=O)cc2C1 N1(C(C2=CCC(C)CC2)=O)CC2CC(NC(=O)CCC3CCOCC3)CC(C2)C1 C(=O)(CCCC(CC)CC)NCCN(C(C(CC#C)C)=O)CC1CC1 C1(C(N(CCCN(C(=O)CCCc2ccsc2)C)C)=O)CCc2nnnn2C1 N1(C(c2ccc(C)cn2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC12 C(=O)(C1OCCn2ccnc21)NCC1N(C(c2cc(C)nc(C)n2)=O)CC1 c1(C(=O)NC(C(=O)N(C)Cc2cncnc2)C2CCCO2)ccc2nccn2c1 C1(C(=O)Nc2cnc(F)nc2)(CC)CCN(C(c2cnn(C)c2Cl)=O)C1 c1(C(=O)NCC2N(C(CC=C)=O)CCC2)cnc(NCC)nc1 C(=O)(CCCn1cc(CCC(C)O)nn1)NC(CNC(=O)OC)(C)C c1(C(C)=O)ccc(C(=O)NCC2(O)CN(C(c3coc(C(N)=O)c3)=O)C2)cc1F CC1(C)CC(CNC(C2(C)CC=CCC2)=O)CN1C(=O)CC1CC(=O)NC(=O)C1 C#CC1(O)CC(C(N2CCCC2C2(NC(c3cnoc3CC(C)C)=O)CC2)=O)C1 Cc1c(C(N2CC(c3cccc(C(=O)O)c3)C2)=O)nnn1C1CCCCC1 Cc1sc(C(=O)NCCCN(CCCNC(C2CCN(C)CC2)=O)C)c(C)c1C c1(C(=O)NC2(CNC(CN(S(C)(=O)=O)C)=O)CCOC2)ccc(=N)[nH]n1 n1(CC)cc(Br)c(C(=O)NCCN(C(=O)CN2CCC(C)CC2)C2CC2)n1 C(=O)(C1c2ccccc2CN1c1c(C)cncn1)Nc1cc2ccccc2n1C c1(OC)cc(C)c(C(=O)NCC#CCNC(c2nc(C)sc2Br)=O)cn1 C1(C(=O)NCC2C(CNC(C3(C#N)CCC3)=O)C2)CN2CCN1CC2 N1(C(CCc2nnc(C)o2)=O)CCN(C(=O)C(C)C(O)CC)CC(C)(F)C1 C1(C(=O)NCCCNC(C(c2cccc(Cl)c2)OC)=O)Cc2cc(F)ccc2O1 c1(C(=O)NC2CC(CC)(CC)N(C(=O)NC)C2)[nH]c2ccc(C(=O)O)cc2c1C N1(C(C(=O)N(C)CCC2CCCCC2)=O)CCc2c(cnn2C)C1 N1(C(c2cc(COC)sc2)=O)CC(NC(=O)C(CC)(CC)OC)C2(CC2)C1 N1(C(c2cn(C)c(=O)cn2)=O)CCCC2CCN(C(=O)C(C)(C)CC(F)F)CC12 Cc1ccc(SCC(=O)NCCC2CC(N(C)C)C2)cc1.C12(C)CCN(C1)C2=O N1(C(C2CC=CCC2)C(=O)NC(C2CCCCCC2)C)CCc2sc(Cl)cc2C1 Cc1cc(Cl)c(C(=O)NC2CC3C2CCN3C(=O)C(C)c2ccco2)c(Cl)c1 N1(C(C(C)(C)c2cscn2)=O)CC2CC(NC(C3(C)CCC(F)(F)C3)=O)C1C2 c1(C(=O)NC(CN(C(C2CCCOCC2)=O)CC)C)cc(C)cc(OC)c1C CCCCCC(=O)NC(c1ccccc1F)CNC(c1nc(C(C)C)oc1C)=O N1(C(CC(CC)SC)=O)CCCN(C(c2cc(O)n(CC)n2)=O)C(C(C)C)C1 Cc1cc(C(N2CCN(C(c3sccc3CO)=O)CC(C)C2)=O)c(F)cc1F N1(C(CC2CCCC(OC)C2)=O)CC2CC(C1)CN(C(c1ccsc1Cl)=O)C2 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(C2CC2F)=O)CCC1C(F)(F)F N1(C(C(=O)NC2CCOCC2)=O)CCCCC1C(N1CCSCC1)=O CCC(C(=O)OC)C(=O)N1CCCC(N(C(=O)COCCNC(C)=O)C)C1 c1(CC)cc(Br)cc(CC)c1Cc1ccccc1.C(=O)(CC(C)(C)CC)N N1(C(C=CCOC)=O)CC2(CC(NC(=O)C=Cc3cc[nH]c3)C2)C1 C#CCCCCCC(=O)N1CCCC1C=CC(N1CC(n2ccnn2)C1)=O C(C(=O)NCc1ocnc1C(=O)NC1(CF)CCCC1)(C(C)C)SC CC(=O)C(C)CC(C)C(=O)N1CC2(C(N3CC(C)(C)CCC3CO)=O)CC1CO2 C(=O)(C1=CCCC1(C)C)N1CCN(C(CCCC(=C)C)=O)C(CCOC)C1 Cc1cc([N+](=O)[O-])cc(C(=O)N(CCCNC(=O)CC2CCCCCC2)C)c1Cl C1(C(N2CC(CC(C)NC(=O)CCCc3nc(C(C)C)no3)C2)=O)CCC2CC2C1 n1(C(CC)CC)nccc1C(=O)NCC(C1CC1)N(C(=O)CNS(N)(=O)=O)C CCC(CC(=O)NC1(CF)CCN(C(c2ccc(C(C)C)cc2)=O)C1)C(C)(C)C C(=O)(CC(C)C(F)F)NCC1CCC(C(=O)NC(c2cn(C)nn2)C)CC1 C=C(C)CCC(=O)NC1C2CCN(C(C3CC3c3ccccc3)=O)C12 C1(NC(C2C(CCC)CN(C(C3(O)CCSCC3)=O)C2)=O)CCCC1C1CC1 N1(C(c2ccc(CCCCCC)s2)=O)CC(NC(C2CCC(=O)N2C)=O)C(SC)C1 C1(CN(C(C(C)OCCC=C)=O)CC)CCN(C(c2cccc(C)c2)=O)CC1 C1(C(N2CCC(O)(CN(C(C3(CCC=C)CC3)=O)C)C2)=O)CCS(=O)(=O)C1(C)C c1(C(F)F)cc(N(C2CCC2)C2COC2)n2ncnc2n1 CN1C(=O)NCC1C(=O)NC1CCC(NC(=O)CN2CCNC(=O)C2)C1 c1(-n2cc(C3CN(C(c4c(CC)n(CC)nc4)=O)C3)nn2)ccc(F)c(F)c1F c1(C(=O)OC(C)C(=O)Nc2nccs2)n[nH]c2c1COC2 N1(C(C(C)NC(C)=O)=O)CC2(CCN2C(c2cnc(O)c(F)c2)=O)C1 Cc1c(CC(N2CCC(c3cc(Br)no3)CC2)=O)ccc(Cl)c1Cl N1(C(C23CCC(OC)(CC2)C3)=O)CCC2(CCN(C(=O)C(F)C3CCC3)CC2)C1 C(C)(c1ccccc1OC)=CC(=O)N(C)CC1N(C(CC(=O)NC)=O)CCCC1 c1(C(N2C(C(=O)Nc3cccc(Br)c3Cl)CC(C)C2)=O)cc2ccccn2n1 C1(NC(C(COCC)C)=O)CC=C(C(=O)N2CC(C(C)CC)C2)C1 Cc1cncc(CCC(=O)NC(C)CCN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)c1 N1(C(C2CC(C#C)(O)C2)=O)CCCC2CN(c3nc(CC)nc(Cl)c3F)CCC12 N1(C(c2ccc(OC)c(F)c2)=O)CCN(Cc2ccc(C(C)C)cc2)CC1C#N N1(C(C(CC=C)C)=O)CC2CCC1C(NC(=O)CNC(c1cscn1)=O)C2 c1(OC)cc(C(=O)NC2CN(C(=O)CCCCCO)CC2F)cc(Br)c1Cl C(=O)(C1CCCn2ccnc21)N(CCC(c1cccs1)NC(=O)C=CCO)C N1(C(CC2N(C(C)=O)CCC2)=O)CCN(C(c2cc(C(C)(C)C)no2)=O)CC1C c1(OC(C(=O)N(CCC(C)NC(=O)C=C(Cl)Cl)C)C)ccc(C(F)(F)F)cc1 C1(NC(C(C)NC(N)=O)=O)(CO)CCCN(C(c2ccc(CO)o2)=O)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CN(C(c3cc(F)c(Cl)cc3F)=O)CC2C1 CCC(C)C(O)CC(=O)N1CCC(CCC(N2CC3CC(OC)C(C3)C2)=O)C1 N1(CCC(C)C(F)F)C(=O)CCN(Cc2ccc(OCC#N)cc2)C1=O C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NC1(CNC(=O)CCCCC2CC2)CCC1 C1(NC(C(C(C)C)(C)C)=O)CN(C(=O)C(C)(C)c2ccccn2)C2(CCOC2)C1 C(CNC(=O)C(C)CC)(CC(F)(F)F)NC(c1c(CC)c[nH]c1)=O N1(C(CCCCNC(Cc2ccn(C)c2)=O)=O)CCC(O)C(F)C1 CC(C)C(C)C(CNC(=O)Cc1csnn1)NC(c1cn(C2CCC2)nn1)=O Cc1c(Br)ccc(CN=c2ccc(C(=O)Nc3ncc(C(C)=O)s3)c[nH]2)c1F N1(C(C(C)=CC)=O)CCCCC(CNC(C23CC(CC(F)F)(C2)C3)=O)C1 c1(C(N(CC(C)N(C(C(CC#C)C2CC2)=O)C)C)=O)cc2n(n1)CCCC2=O N1(C(c2ccc(C(OC)OC)o2)=O)CCCCCC(NC(=O)CCS(C)=O)C1 C1(CC(=O)N)CCC2CC12.O=C(C(O)c1ccsc1)NC1(CC2CC2)CC1 CC1C(C)N(C(c2nncn2C)C(=O)NC(C)(C)C)CCS1(=O)=O C1(CNC(C(CC)n2ccnc2)=O)C2CN(C(=O)Cc3n[nH]cc3Br)CC12 C12(CNC(c3cnc(O)c(F)c3)=O)CCC1CN(C(c1csc(Cl)c1)=O)C2 N1(S(CCCC)(=O)=O)CCN(Cc2c(C)cccc2Br)CC1C#N c1(CC)onc(C(=O)NC(c2ccccc2)C(=O)NCC#CC#CCO)c1C CC1(C)CCCC(CN=C(NCC(F)F)NCC2CC(C(F)F)C2)O1 Cc1cccc(N2CCCC(NC(N3C(C)CC3(C)C)=O)C2)c1 C(CCCC(=O)NC(CCC1CC1)C(=O)NC(C)CCC(C)C)OC N(C(=NCc1cccc(N(C)C)c1)NC(c1cccs1)C)C(CC)C c1(OC)ccc(C(=O)NC(CNC(c2cscc2F)=O)C2CCC2)cc1 C1(O)(CNC(c2cncc(N)c2)=O)CCN(C(c2cnc(Cl)cc2Cl)=O)CC1 c1(-n2ccc(C)n2)cccc(C(=O)NCC2CC2CO)c1 C=CCC(C)(C)C(=O)NC1CCC(CNC(c2c(C)nn(C)c2C)=O)CC1 Cc1cc(C(N2CC3CC(NC(c4cccnc4C)=O)CC3C2)=O)c(F)cc1F c1(OCc2cn(CCn3cc(C(=O)OC)nc3C)nn2)ccc(C#N)nc1C c1(CC(=O)N(C2CCN(C(=O)Cn3cncn3)CC2)C)ccc2ncsc2c1 C1(NC(COCCC(C)C)=O)CC(CNC(c2cc(F)ccc2Cl)=O)C12CCC2 c1(C(N2CCC(CCOC)(NC(CCOCC)=O)C2)=O)nncc2c1CCCC2 N1(C(C(C)CC(N)=O)=O)CCCCC2(C1)CN(C(c1ccncc1N)=O)C2 C1(C)(NC(C(C)NC(=O)Cn2cnnn2)=O)CCCN(C(c2occc2Cl)=O)C1 N1(C(C(CCC)N(C)C)=O)CCC2C(CCN2C(c2cc[nH]n2)=O)C1 n1(C(C)C)cc(C2CC2C(=O)N(CC(C)CNC(=O)COCCCOC)C)cn1 C1(CNC(c2c(C)nco2)=O)CC2(CCN(C(=O)CC3(O)CC3)CC2)CO1 N1(C(C2(C)C(C)C2)=O)CCC(F)(F)C(CNC(=O)C(C2CC2)C2CC2)C1 C(=O)(C(O)CSC)NCC(COCC)N.C(=O)(COCCOCCO)OC C(=O)(C(F)CC(C)(C)NC(=O)CN1CCCCC1)NCC(C)(C)CO c1(C(N2CCC3(C(NC(C(COC(C)C)(C)C)=O)C3)C2)=O)cccn2cncc12 N1(C(c2cc(CC)nn2C)=O)CC(C)CCC1CNC(c1csc(COC)c1)=O C1(C(=O)O)(CN(C)Cc2cncn2C)CCCN1C(=O)C=CC(C)(C)C CCCC(C(=O)NCCC1CCCN1C(=O)C=Cc1ccc(CC)o1)NC(C)=O CC1CCC(=CC(=O)NC(C)(C)CC=CC(=O)NC2COCC2F)CC1 c1(NC(C2CCN(C(c3cc(F)ccc3CO)=O)C2)=O)ncc(Cl)cc1Cl C1(NC(c2c(C)n(C(C)C)cc2)=O)CCC(C)N(C(c2c[nH]cc(Cl)c2=O)=O)C1 C(=O)(CC(C)(C)C(=O)NCC1CN(C(=O)COC2CCOC2)CC1O)OC CCCC(C)(O)C(=O)N(C)CC1CCN(C(=O)CCCCN2CCOCC2)CC1 C1(CNC(C2CN(C(C=C(CC)CC)=O)C2)=O)CN(C(C2CCCCO2)=O)CCN1C C12(CNC(C3C(C)OC(C)C3)=O)CC(CO1)N(C(C13CC(CO1)C3)=O)C2 N1(C(C2N(C(CSCC#C)=O)CC=C2)=O)CCOC(C(=C)C)C1 C1(C(N2CCC(CN(C(C34CCCC3C4)=O)CC)CC2)=O)CC(=O)NC(=O)N1 c1(NC(C2N(Cc3cccc(C)c3)CCNC2)=O)cc(Cl)cc(Cl)c1Br C1(C(N2CC(C(=O)NC(C)C(=O)NC(C)(C)C)C2)=O)CC(F)(F)CN1C(N)=O C=C(C)CC(C(=O)N1CCC(C)(CNC(C2CCCC23CC3)=O)C1)OC C1(C(N2CCC(CN(C)CC)C2)=O)COC2(C1)CN(C(=O)C(C)(C)CN(C)C)C2 C1(NC(=O)C=Cc2ccncc2)CC(C2CCN(C(=O)Cc3cnns3)C2)C1 c1(C(N2CCC(O)(CN(C(c3c(C)n(C)nc3)=O)C)C2)=O)ccc(F)cc1Cl c1(C(=O)Nc2ccccc2OCC(F)F)cc(Br)cnc1Br c1(C(=O)NC(C(=O)NCC(C)(C)SC)CC2CC2)c[nH]c(=O)cn1 N1(C(Cc2cnc(C)o2)=O)CC2CCCC(NC(c3ncc(Cl)n3C)=O)C2C1 C1(C(=O)NC2C(C(=O)NCc3c(C)noc3)COC2)CCCC(=O)N1C c1(CNC(C2C(C)(C)C2)=O)nnc2n1CCN(C(=O)Cc1cc[nH]c(=N)c1)C2 N1(C(c2c(CC)scc2)=O)CCCC(C)(NC(=O)CC2(COC)CC2)C1 N1(C(C(Cn2cccn2)NC(C(C=C)OC)=O)=O)CCOC(CF)C1 C1(Cc2cn(C3(C(=O)NCc4cnc(C)nc4)CC3)nn2)CN2CCN1CC2 c1(C(=O)OC)nc(=NCCN(C(c2cc3sccc3cn2)=O)C(C)C)c(C)c(C)[nH]1 N1(C(C2(C(F)F)CCC2)=O)CC2CCC(C1)N(C(=O)Cc1ccsn1)C2 c1(C2C(C(=O)NCCN(C(C)C)C(C3CCC4CC34)=O)C2)cccc([N+](=O)[O-])c1 c1(CC(N2CCCC(NC(c3n[nH]cc3F)=O)C2)=O)c(Cl)cccc1Cl c1(C(=O)NCC2CC(NC(C(COC)C)=O)C2)ccc2c(c1)S(=O)(=O)NC2 N1(C(=O)CCc2ccccc2)CCN(C(C2CCCN2C2CC2)=O)CC1CF N(C1CCOc2c(C)cccc21)C(c1n(CC=C)nnn1)CCC Cc1cc(C(=O)NCC(C)(C)CNC(c2cc(O)n(C)n2)=O)cnn1 c1(OCC=C)ccccc1CN1CC2C(C(=O)NC3CCC(C(=O)O)CC3)C2C1 c1(Nc2scc(C(=O)Nc3ccc([N+](=O)[O-])o3)n2)c(C(F)(F)F)ccc(Cl)c1F C=CCCCC(C(=O)OC)NC1CC(C(=O)OC(C)(C)C)C(O)C1 C1(NC(C(CC=CC)CC)=O)CCN(C(=O)Cc2c[nH]nc2O)CC12CCC2 O=C1NCc2c(C(N3CC4CC(NC(C56CC5C6)=O)CC3C4)=O)cccc21 c1(NCC2CCN(CC)C2)[nH]c(=NCc2ccc(C)o2)nc2sccc12 c1(OC(C)C(=O)NCC2CCCCN(C(=O)CNC=O)C2)cc(Cl)cc(Cl)c1 CC1CCC(NC(=O)Cc2cnoc2)CN1C(=O)CCOC1CC1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(C1(c2cc[nH]n2)CC1)=O C=CC1(CNC(=O)CC=CCNC(C2(Cl)CC2C(C)=O)=O)CCOCC1 C1(=CC(N2C(CNC(C=CCOC)=O)CC2)=O)CCN(C)C1 CC(C)CC(C(=O)NC1C=CC(CNC(C2CCCC2C)=O)C1)C(N)=O c1(CC)ncnc(NC(C2C(C(N3CCCC3c3ccc(Cl)cc3)=O)C2)=O)c1F c1(C(=O)NCC(C)(CC)NC(C(C)OCC)=O)cc(-c2ccccc2)ccc1O CC(CN=c1[nH]c(=N)[nH]c(=NCc2cccc(Cl)c2F)[nH]1)C(C)(F)F C(=O)(C(CC)CC(C)C)NC1(CC=C)CN(C(C2(OCC)CCSC2)=O)C1 n1(CCC(=O)NCCC(C)NC(c2n(CC)ncc2)=O)ccc2cc(Cl)ccc12 O=S(=O)(C=Cc1ccc(F)cc1)Nc1cn2ncccc2n1 c1(OC)cc(Cl)ccc1C(=O)NCCNC(C1(CN)CCCNS1(=O)=O)=O c1(OCCC(=O)N(CCCNC(C2C3CCCC23)=O)C2CC2)ccccc1Cl O=C(C1=Cc2ccccc2C1)N1CC2CC1CCC2NC(C1CC(O)C1)=O c1(C(N2CC(C(=O)OC)C(C)(C)C2)C(=O)NCC(F)F)cc(Cl)c(F)c(Cl)c1 C1(CC)CN(C(=O)CC2CN(C(c3ccnc(OC)c3)=O)CCO2)CCN1C c1(C(=O)NC2CC(CCNC(C3OCCN(CC)C3)=O)C2)csc2c1CCCC2 c1(C(N2CCC(CNC(=O)Cn3ccnn3)C2)=O)ccc(C(O)CF)cc1 c1(N2CCCC(CNC(CCOCCN(C)C)=O)CC2)ccc([N+](=O)[O-])cn1 CC1(C2CCCN(C(C34CCCC3CCN4C(C3CCNC3=O)=O)=O)C2)CC1 S(=O)(=O)(c1ccc(N2CCC(CC(F)F)C2)cc1Br)N1CC(C(C)(C)C)OCC1 C1(NC(C2(OC)CCOC2)=O)CCN(C(c2cnc(C(C)=O)s2)=O)CC(C)(C)C1 N1(C(C2CC(OCC)C2)C(=O)NC(C)CC)CCOCC1 Cc1sc(Cl)nc1C(=O)NC(CNC(=O)CCCC1CCC1)CO CC(C(=O)NCC1CCC(NC(c2coc(CO)c2)=O)CC1)C(=O)N1CCOCC1 c1(OC)cc(CC(=O)N(CCCCN(C(=O)C#CC(C)C)C)C)cc(OC)c1O CCC(C)(C)C(=O)NC1CN(C(c2coc(-c3ccccn3)n2)=O)C2CC12 c1(C(N2CCCCC(NC(C(CC)=CC)=O)C2)=O)cnc(O)c2cncn12 C1(C(=O)NC(CNC(C2(COC)CCC2)=O)C)COc2cc(Cl)ccc2O1 c1(C(N(CC(C)N(C(C(CCSC)OC)=O)C)C)=O)cc2c(F)c(F)ccc2[nH]1 C1(NC(CC(C)C)=O)(CF)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 CC(CCO)C(=O)NC(CNC(=O)Cc1nncn1C)CO C1(N(C(CN(C(C)=O)C)=O)C)CN(C(=O)C(F)C2CCOC2)C1 N1(C(C(C)Cc2ccco2)=O)CCC2(CC1)CC2NC(c1ccc(CO)cc1)=O C(=O)(C1=CCCCC1C)N1CCCC(C(N(CC=C)C)=O)C1 C12(NC(CC)=O)CCN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC1C2 c1(C(N2CCC(COC)C2)C(=O)NCc2cccs2)cc(Br)cc2cccnc12 c1(C(=O)OCC)ncccc1NC(=O)C(N1CCCC1C1CCCCC1)=O C(CCC(=O)NCC(CC)NC(C1(C(=O)OC(C)(C)C)CC1)=O)=CCC=C c1(NC(C2CCC(NC(C3(CCCF)CC3)=O)CC2)=O)cc(Cl)ccc1O N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CC(C)C)CCC1 c1(C(=O)NCC#CCNC(c2c(CC)nns2)=O)cnc2c(ccn2C)c1 C(=O)(C(C#N)CC1CC1)N(C(C)CCn1cccn1)C1(CCN2CC(OC)C2)CC1.CO c1(C(C)OCC)nc(-c2cc(COC(C)C)n(C)n2)n(CC2(C)CCCC2)n1 C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C(CN(C)C)C1)=O)(C)C c1(CNC(c2ccc(N3CCOCC3=O)cc2)=O)ccc(S(=O)(=O)CCO)cc1 C1(CCC(N2CC(CC=C)(NC(c3csc(C4CC4)n3)=O)C2)=O)CCCCN1C CC1(C)COCCC1C(N1CCOC(c2cn(CCCCO)nn2)C1)=O N1(C(C2CC(=C)C2)=O)CCN(C(c2nc(C)oc2-c2ccccc2)=O)CCC1C CC1(C)CN(C(C2C3COCC23)=O)CCC1C(N1CCC(CC(F)F)C1)=O c1(C(N2C(C(N(C)CCF)=O)C(C)(C)CCC2)=O)ccc2cc[nH]c2n1 C(=O)(C#CC1CCCOC1)N1CCN(C(C2(CC)CC2)=O)C(c2cccnc2)C1 Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCCS2)=O)[nH]c1C c1(C(N2CC3C(C(=O)NCCC=C)(CC3)C2)=O)cc2cc(F)ccc2s1 C(=O)(C(C)(C)CNC(c1cc(C(C)C)no1)=O)NC1(CCCC)CC1 C1(NC(c2cn(CC=C)nc2)=O)CC(O)CN(C(=O)Cc2cncn2C)C1 C(=O)(CC(C)C(F)F)N1CC(c2cn(C(c3cccc(CO)n3)C)nn2)OCC1 C(=O)(C1=CC2CCCCC12)N1CC(CCNC(=O)C=Cc2ccco2)C1 C12(CNC(C3CC(OCC)C3)=O)CCC(CN(C(=O)Cc3ncn(C)c3C)C1)C2 CC1C(NC(=O)C(CO)c2ccccc2)CCN1C(=O)CCC1CCCCO1 C(C(C)(O)CC(=O)N1CCOCC(CNC(=O)CC2CC3(CCC3)CO2)C1)OC C1(CC(N2CC(CC=C)(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)CCCC(=O)N1 C1(C(C(N2CCCC2C2(O)CN(C(C3(n4cccn4)CC3)=O)C2)=O)O)CCOCC1 Cc1ccc2cc(C(N3CCC(N(C(=O)C(C)(C)C(C)C)C)CC3)=O)oc2c1 C1(C(=O)NCCCN(C(=O)C(C)CCOC)CC)CCC(N(C)C)CC1 c1(SCCC)cccc(C(=O)NC2CCCC2CNC(c2cccnn2)=O)c1 Cc1cc(C#N)sc1C(=O)NC(c1ccccn1)C(C)C C(=O)(C#CC1CCOCC1)N1C(C)CCC(NC(c2c(O)nnc(C)c2C)=O)C1 c1(C(N(C)CC2N(C(CS(CC)=O)=O)CCC2)=O)ccc2cnnc(O)c2c1 N#Cc1cc(C(=O)NCC2(CO)CCCCCC2)ccc1Br N1(C(Cn2c(C)csc2=O)=O)CCN(C(=O)Cn2cccc2)C2CS(=O)(=O)CC12 c1(OCCCNC(c2sc(Br)nc2C)c2n(CCC)nnn2)ccccc1Cl Cc1cc(NC(c2cc(Br)cn2C)c2nnnn2-c2ccccc2)cnc1Cl C1(C(=O)NCCNC(C2CC=CCO2)=O)Cc2cc(F)cc(F)c2O1 CN1CC(C(=O)NCC(C2(O)CN(C(c3cnc(S)nc3)=O)C2)(C)C)NC1=O C#CCCCCC(c1nnnn1CC(F)F)NCc1occc1C CCC(CCC(=O)NC1(CCNC(c2ccc(OC)c(Cl)c2)=O)CCCC1)OC c1(CN2C(c3cccs3)CCC(C)C2)n[nH]c2ccccc12 c1(CC)ccc(C(=O)NC(C)C(C)NC(=O)CN(C2CCC2)C)cc1F C1(C(=O)NC(CC)CNC(=O)CCCn2cncn2)CCC(CO)CC1 Cc1nc(C(=O)NC2CC(NC(=O)COC3CCCC(C)C3)C2)c(=O)[nH]c1C N1(C(c2cnc(-c3ccccc3F)s2)=O)CCC12CCSCC2 c1(CC)nc(C(N2C3CCC2CN(C(=O)CSCC(N)=O)C3)=O)c2ccccn12 c1(OC)cc(CN=C(NCC(C)(C)C)NC2CCS(=O)(=O)C2)cc(OC)c1C C1(NC(=O)COCC(F)F)(CF)CCN(C(=O)CCc2cccnc2)C1 c1(OCCCC)ccc(C=CCC2CC(NC(C)C)C2(C)C)c(C)c1 CCC(C)C(=O)C(=O)N1CCC(C(N2CC(CC)(CO)C2)=O)O1 N1(C(C(C(C)C)SC)=O)CCC2CCC(NC(c3cc(C)nc(Cl)c3)=O)C1C2 C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2cn(C)nn2)C12CCC2 c1(C(N(C2CCC(NC(CC3C(C)CCO3)=O)CC2)C)=O)cc(F)cc(Cl)c1 CCCCCCC(CC)(CC)C(=O)N(CC(CC)NC(C1CCC12CCC2)=O)C N(C1CN(C(=O)CCCC2CCCC2)Cc2ccccc21)C(C(C)C(F)F)=O C1(NC(C(CC)CC)=O)COC2C(NC(c3nc(C)n(C)c3C)=O)COC12 C1(OCC)CN(C(=O)C(C(C)C)N2CCCC2=O)CC1(C)C C1(CNC(C(CC#C)O)=O)(NC(=O)CC2CCC3(CC3)CO2)CCCCCC1 Cc1nnsc1C(=O)N(C(C)(C(=O)NC(CO)C1CC1)C1CC1)C C1(NC(C2(C)CCC(C)C2)=O)COC2(C1)CN(C(c1cnn(C)c1C(F)F)=O)C2 c1(C(=O)NC2(C)CCCN(C(C(CC)(C)CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C(=O)(CC(C)(C)C1CC1)N1CC(CC(C)NC(CC(C)F)=O)C1 C1(C(=O)NC2C(CC=C)CC2)CCC(CNC(c2ccc(C)o2)=O)C1 C12(CNC(C3ON=C(C)C3)=O)CC(CNC(=O)C(C)(C)n3cnnn3)(CO1)C2 N1(C(C2C(NC(C(C)(C)n3ccnn3)=O)CCO2)=O)CCOC2C(O)CC12 CC(C)CC(C)(CO)NC(C1CCCCN1C(C1OCC2CCCC12)=O)=O C1(CC(N2CC(NC(c3nc(CCC)oc3)=O)C2)=O)CCCCN1C c1(CC)nccnc1C(=O)NCC1CC1C(=O)NC(COC)CCO c1(C(N(C2CCN(C(=O)COc3ccsn3)C2)C)=O)cc(Cl)cc2ccncc12 C(CCCCCNC(C1CCS(=O)(=O)C1)=O)NC(=O)CCc1ncccn1 N1(C(C2C(C)N(C(C3CCOCC3)=O)CC2)=O)CC2CCCCC2C1C c1(C(=O)NC2CCN(C(=O)C=CCN3CCCCC3)C2)ccc(Cl)c(F)c1 c1(N(C)C)cnc(C(=O)NCC(=C2CN(C(=O)CC3CCS(=O)(=O)C3)C2)F)cn1 CC#CCC(C)NC(=O)C(C1CC1)N(C(=O)C(c1ccn(C)c1)C)C C1(NC(CCC(=C)Cl)=O)CCCN(C(c2cccc(C(F)(F)F)c2O)=O)C1C c1(OC)nccc(C(N2C(C(=O)NCc3cnccc3C)CC2C)=O)n1 CC(C)(C)C(O)C(=O)NCC12CC1CN(C(=O)Cc1nc[nH]n1)C2 C(CCCC(C)C)(C(=O)Nc1ccc(F)cc1C)N(C(C#C)C)CCCC Cc1nc(CCC(N2CC(CNC(=O)Cc3cc(Cl)cs3)C(O)C2)=O)oc1C c1(C(N2CCC(OCC(=O)NC3COCCOC3)C2)=O)cc2ccccn2n1 c1(C(=O)NC2(CNC(c3nc(Br)c[nH]3)=O)CC2)c(Cl)ccc2ncccc12 c1(C(=O)NC2C(C(=O)NC3C(=O)NCC3)CCCC2)ccc2nccnc2c1 Cc1cc(C(N2CCOC(C3(O)CC3)C2)=O)nc(N(C)CS(N)(=O)=O)n1 N1(C(c2c(C)nccn2)=O)CCCC(C)(C)C1CNC(=O)CC(C)(F)F c1(C(=O)NCC2C(C)CCN(C(=O)C(N)=O)C2)ccc2sccc2c1 C1(F)(CNC(C(C2CCCC2)OC)=O)CN(C(=O)C(C)Nc2nc(C)cs2)C1 c1(N2C(C)CCC2C(=O)Nc2ncc(F)cc2Br)ncnc2c1CCCC2 N1(C(CC(C(CC)(C)C)C)=O)CC(NC(=O)C2CC2)C2(CCS(=O)(=O)CC2)C1 c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)c[nH]c2nccc(Cl)c12 C1(NC(c2n(CCCOC)nnn2)c2sccc2OC)CCCCCC1 C1(C(N(CCC(O)C(=O)NC2CC(C)(C)C2)C)=O)CCCC2(CC2)C1 N1(C(C(CC)NC(N)=O)=O)CCC(C)C(NC(=O)CC(C(F)F)n2ccnc2)C1 N1(C(CC2C(NC(C3(OC)CCSC3)=O)CCCC2)=O)CC(C)CCCC1C C(c1ccccn1)=C(C)C(=O)NC(C)CNC(c1ccnc(N(C)C)c1)=O n1(CC)ncc(Cl)c1C(N1CCCC(C(C)(O)CNC(=O)Cn2nccn2)C1)=O c1ccccc1C(N1CCCC1)=O.C(=O)(CN(CC(=O)NC(N)=O)CC)OCCC C1(NC(c2ccc(OC)cc2OC)=O)CN(C(=O)C(O)C(C)(C)C)C2(CCC2)C1 c1(CNC)cccc(N(C)C)c1.C12CCCN1C(=O)NCC(C)C2 N1(C(CC2(N(C)C)CC2)=O)CCC2(C=C(C(=O)NCCC3CCN(C)C3)C2)C1 c1(C(=O)NC(c2ccccn2)CC)nc(CNC(C2C(C)(C)C2(F)F)=O)oc1C N1(C(CCCN(C(C)C)C)=O)CC(O)CC1(C)C(=O)NC1(c2cccnc2)CC1 C1(C(N2CC(CCCCNC(C(CC)OC)=O)C2)=O)CN(CP(C)(C)=O)C1 c1(C(N2C(C)CN(C(=O)Cn3cc(C(F)F)cn3)CC2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(CCCN(C(C)=O)C)=O)CCC2)cc(Cl)cc(Cl)c1 c1(OC)cc(C(=O)NC(C2CCCN2C(C2OCC2(C)C)=O)C)ccc1C(N)=O N1(C(c2cc(Br)nn2C)C(=O)NCCCOC)CCC(S(C)(=O)=O)C1 CC1(C)CN(C(C2CC(F)(CO)C2)=O)C1C1CCN(C(C2C=CCC2)=O)CC1 N1(C(CCC(=O)NC)=O)CCN2C(=O)C(NC(c3cc(C)cnc3N)=O)CC2C1 n1(CC)nc(C)c(C(=O)NCC2CCCN(C(=O)C(F)=CC3CC3)C2)c1Cl c1(CC(N2C(C(C)C)CN(C(C34CC(C3)C4)=O)CC2)=O)cc(F)c(F)cc1F C1(C(N2CC3CC2C3)C(=O)NCCSC)CCC(CCC(C)C)CC1 C1(NC(c2sccc2C2CC2)=O)(CNC(=O)CC2CCC2)CCCC1 CC1OCCC1(C)C(=O)NC1CC(NC(c2cccc(C(N)=O)n2)=O)C1 CC(C)C(C(=O)N1CC2CCN(C(C3CC4CC3CC4(F)F)=O)C2C1)C(C)C CCC(CC)C(C(=O)NC(C)CC1CN(C(c2c[nH]nc2C(C)(C)C)=O)C1)OC c1(CNC(CCN(C)C)=O)csc(C(=O)NC2CCN(CCCO)C2)c1 C1(CC(=O)N(C2CC(NC(c3c(CCC)nco3)=O)C2)C)SC2=NCCN2C1=O N1(C(c2c(OC)cccc2)=O)CC(CNC(=O)C(C)N(C)C(C)=O)C2(CC2)C1 c1(NC(NCC(CC)(C)OC)=NC)nncc2c1cnn2C.OC Cn1cc(C(=O)NC2CC2NC(C23CCCCC2NC(=O)C3)=O)c(=O)n(C)c1=O C1(C)(C(=O)NCC(CC)NC(=O)C(O)Cc2cnc[nH]2)CCCCNC1=O C1(CC(=O)NCc2c(C)nn(C)c2)CN(C(C2CCC3CC23)=O)C(C)(C)C1 c1(C(=O)NC2CCCCN(C(CCCC=C)=O)C2)c[nH]c2ccc(O)cc12 C1(C)(C(N2C(C(C)NC(c3n[nH]c(O)n3)=O)CCC2)=O)CCCCCC1 C(C)(C)(CCC(=O)NC(C(=O)NCCCCS(C)=O)C(C)O)OC n1(CCC)cncc1CNC(=O)NC12CC(NC(=O)NCC(C)(C)C)C1C2 c1(C(=O)NCC2N(C(C3C(F)(C(=O)OC)C3)=O)CC2)cc(-c2ccncc2)[nH]n1 N1(C(=O)CCc2ccccc2)CCC2CN(C(C3CCCC(F)(F)C3)=O)CC2C1 Cc1cc(NC(=O)Cc2ccccc2O)ccc1NC(C1CCS1(=O)=O)=O c1(C(=O)NCC2CC(NC(C3CCCCC3)=O)C2)cnc2ccc(Cl)cn2c1=O C1(CCCC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CCCc1ccc(C)s1 Cc1cc(C(=O)N(C(C(=O)NC2CC3(CCC3)C2O)C2CC2)C)c(O)nn1 C=CCC(C)(CC)C(=O)N1CCC(C(=O)NCC2CCC(O)C2)O1 Cc1cccc(C(N2CC(NC(=O)CSc3nncn3C(C)(C)C)C(C)C2)=O)c1 c1(CC)c(C(N2CCOC(CC(=O)NCc3nnn(C)n3)C2)=O)nnn1C C1(C(N2C(CNC(COc3c(C)occc3=O)=O)CC2)=O)CC(C)CC(C)(C)C1 C1(C(=O)NC(C(=O)NCCCS(C)=O)Cc2cc[nH]n2)CC2(CC2)CO1 Nc1cnc(C(=O)NCCCCC(=O)NCCC2(O)CCC2)cn1 CC1(NC(c2ccc(O)nc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1 C1(CCNC(CCN(CCC)C)=O)CCN(C(c2snnc2CC)=O)C(C)C1 C(=O)(C(C)C(C)(C)C)N1C(C(=O)NCc2c(C)ccs2)C=CCC1 N1(C(CCC(C)NC(=O)CNC(=O)CP(C)(C)=O)=O)CCc2ccccc21 N1(C(COC2CC(NC(c3c(CC)cncc3)=O)C2)=O)CCOC(C)(C)C1 Cc1cc(NC(=O)C(c2ccc(Cl)cc2Cl)O)ccc1NC(=O)C1=CCC1 C(=O)(N=c1[nH]n(C(C)(C)C)cc1C)C1(C)N(C(c2cccc(C)c2O)=O)CCC1 c1(C(N2CCC(C(C)C)C2)=O)ncncc1F.c1(C(=O)N)nn(C)cc1Cl N1(C(C=CCCC)=O)CC2CCC2(CNC(c2c[nH]nc2C2CCCO2)=O)C1 N1(C(CCCC#C)=O)CCC2CCC12CNC(=O)COCCC c1(C(N2C(CCOC)CN(C(=O)C=CSC)CC2)=O)cc2cccnn2n1 C#CCCCC(=O)NCCOCCN(C(=O)C(CC)CC)C.C1(=O)CN1 C1(C(N2CCC(F)(F)C2)=O)CN(C(=O)CCc2nncs2)C2(CCC2)C1 Cc1cc(C(=O)NCC(C)NC(=O)C=Cc2cccc(F)c2)c(N)c(C)c1 Cc1nc2c([nH]1)CC(C(=O)NCCOC1CCN(C(=O)C=CC(C)(C)C)C1)CC2 c1(CC(=O)NCC(C)CN(C)C(c2c(F)ccnc2F)=O)cn2c(n1)CCCC2 CN(S(N)(=O)=O)CC(=O)NC1COCC1NC(=O)CC(O)c1ccccc1 c1(OC)nc(Br)ccc1C(=O)NCC1CCCN1S(=O)(=O)CCc1ccccc1 N1(C(C2C(C)C2)=O)CCN(C)CC1CNC(=O)C(c1ccccc1)C Cc1cc(=NCC2C=CCC2)[nH]c(NC(C)COCC2CC2)n1 Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Cl)o3)=O)C2)=O)ccc1C(C)C c1(CC(=O)NCC(C2CC2)NC(C2(OC)CC2)=O)c(Cl)cccc1Br C(CC(C(=O)N1CC2CCC1C2)NC(c1cnccn1)=O)N(C)C N1(CCOCC)CC2(CN(C(c3n[nH]c4c3CCC4CCCC)=O)CCO2)C1 C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CNC(=O)C(F)C(F)(F)F)(CO)CC1 c1(CC)ncc(C(=O)NCC(C)(CO)NC(=O)CC2(NC(C)=O)CC2)[nH]1 c1(NC(C2C3(CCN(Cc4ccc(C)s4)CC3)C2)=O)n[nH]c2ccc(C#N)cc12 C(C(=O)NCCC#N)(C1=NOC2CCCCC12)N1CC(C)(C)C2C1CCC2 C1(C(C)NC(C(C)(C)C)=O)CN(C(=O)CCCCc2cccs2)C12CCC2 N1(C(CC(CNC(C(C)C(F)(F)F)=O)C)=O)CCC(F)(F)C(O)C1 c1(C(N2CCCC(NC(C3CC4C(C)(C)C4C3)=O)CC2)=O)ccc(Cl)c(Cl)c1O CC1CN(C(C2CC2(C)C)=O)CCC1C(=O)NCC(C)(C)CC1CC1 C1(C(=O)NC2C(NC(CC(CC)(C)C)=O)CCC2)CCn2c(cnc2C)C1 C1(NC(COCCC=C)=O)C2CCN(C(c3cnc(C(C)C)nc3)=O)CCC12 c1(SC)ncc(C(=O)NCC(C2(O)CN(C(=O)C(C)(O)C3CC3)C2)(C)C)s1 C1(C(N(C2CC(NC(c3nc(OCC)oc3)=O)C2)C)=O)CCC(C)CC1 CC1(C2CCCN(c3cc(NC4CC(C)C4)ncn3)C2)NC(=O)NC1=O Cc1cc(C(=O)NC(C2CC=CCC2)C(=O)Nc2csnc2C)cnn1 C1(OC(=O)CC2CCC23CCC3)CCOC2(CCC2)C1 C12(CC)CC(CC(=O)NCC(C)CNC(C3CCN(CC4CC4)CC3)=O)(CO1)C2 C1(CNC(CCC2CCC(NC(=O)CCCC3CCCO3)C2)=O)CC2C=CC1C2 C(CCC(=O)NCc1occc1C(N1CCC1CO)=O)=CCC=C N1(C(C(CC(=O)OC)(C)C)=O)CC2COCCC2(NC(c2ccc(Cl)s2)=O)C1 CCC(CN(C)C)CC(=O)NCCC1(CNC(c2ncoc2C)=O)CC1 N1(C(C(C2CCN(C(C3(C)CCC3)=O)CC2)C)=O)CC2CCCCCCC12 N1(C(C2(SC)CC2)=O)CC2CCC2(CCNC(c2c(C3CC3)noc2C)=O)C1 CC1CCN(C(c2cnc(C(C)(C)C)nc2)=O)CCN1C(=O)Cn1nccn1 c1(C(=O)NC2(C(N)=O)CN(C(c3c(=N)[nH][nH]c3)=O)C2)cccc2cc[nH]c12 C12(C(=O)NCC3(OC)CN(C(=O)CC(F)F)C3)CCCCC1C2(F)F C1(C(=O)OC)CN(C(c2nccc3c[nH]nc23)=O)C2CCCCC12 c1(N(CCc2ccc(C)cc2)C)nc(=NCP(C)(C)=O)[nH]c2c1CCCCCC2 C(C(=O)NC(C)C)(C(C)C)SC.C1CN(C(=O)C(=O)NCC2CC2)CC1C N12CCC(F)(CC1)c1cn(nn1)C1(CC1)C2=O.C1(CC)CN(C)C(C)(CO)C1 N1(CC(N)=O)CCN(C(c2scc(Cl)c2Cl)C(=O)NCCC2CC2)CC1 C12(CNC(C=C(CCC)C)=O)CCCCC1CN(C(=O)CNS(N)(=O)=O)C2 c1(C(N2CC3C(C(=O)NC4CCC(COC)CC4)C3C2)=O)c(F)ccc(F)c1F N1(C(c2c(OC)cncc2)=O)CC=C(CNC(C23COCC(C2)C3)=O)CC1 N1(C(C(COC)COC)=O)CC2CC1CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(C(N2CCC(N(C)C(c3ccccc3O)=O)C2)=O)[nH]nc2ncc(Br)cc12 c1(N(C(CCC#CC)=O)C)ccc(OC)cc1O N1(C(C(C)(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(F)(F)C(C)(C)O c1(NCC2C(=C)C2)nc(C)cc(=NCCn2cc(C3CCOC3)cn2)[nH]1 N1(C(C)=O)CCN(C(c2ccnc(NC3CCC3)c2)=O)C(CO)C1 c1(CNC(COCCC)=O)cc[nH]c1C(N1CCC(C(=O)OC)C1)=O c1(C(N(CCNC(C2(C)CC(=C)C2)=O)C)=O)c(C)ccc(F)c1Br C=CC(CC)CC(=O)N1CCC1CNC(C1(n2cnnn2)CCCCC1)=O C1(CNC(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CC(F)F)C12CCC2 c1(C(=O)NCCNC(C2CN(c3ccc(C)cc3)C(=O)C2)=O)cc(C)nc(C)c1 c1(C(=O)NC(C#C)C2CC2)cnn(CCNC(=O)CCOCCOC)c1 N1(C(C2(C)COC2)=O)CCCC(F)(C(=O)NCC(CC2CC2)CO)C1 C1(O)(CCNC(c2cn(CC)nc2)=O)CCCN(C(=O)COCCCC(C)C)C1 C12(C(N3CCN(C(CC4OCC(C)(C)OC4)=O)CC3)=O)CCN(CC1)S(=O)(=O)C2 C1(C(N2CCC(O)(COC)C2)=O)(NC(C(C)SCCCC)=O)CCN(C)C1 C12CCCCN1C(=O)COC(C)(C)CNC2=O.c1(CC)cnc(CC)[nH]1 C1(CNC(C(CC)C)=O)CCN(C(C2(SC)CCC2)=O)CCC1(F)F Cc1nc2c(C(=O)NC3CCCCC3CNC(c3n[nH]cc3Br)=O)cccc2o1 c1(NC(C2CCC(NCc3ccc(C(=O)O)[nH]3)CC2)=O)onc2ccccc12 CC(C)CC(C(=O)NCCC(C)N(C(=O)CN1CCC(O)CC1)C)C(N)=O C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(C(=O)NC(C)C(=O)NC(C)C)cc1 N1(C2C(CCC=C)C2)CCCN(C(c2ccccc2)CC)CC1 CC#CCCC(=O)NCCCC1CN(C(C2(CN(C)C)CCCC2)=O)CCO1 c1(OC)c(C(=O)NC23CC(Nc4ncc(Br)cn4)(C2)C3)ccc(Cl)c1Cl c1(C(CC)C(=O)NC(C)C(C)NC(c2cc[nH]c2C(C)C)=O)ccc(F)cc1 CC1(C)CCCC1C(=O)NC1C2CC(NC(c3ccns3)=O)CC12 C(CO)(CCC)NC(COCC(=O)NC(C#C)(C)C1CCCC1)=O N1(C(CC2(C)CC2)=O)C(CNC(C23CC(C)(C2)OC3(C)C)=O)CC2CCCCC12 Cc1cc(C(N2CCNC(C(N3CCC(C(F)F)CC3)=O)C2)=O)nc(C)c1 C(=O)(CCC(=O)NN(C)C)NCc1c(C(=O)NCC(CC(=O)OC)C)scc1 c1(C(=O)NC2CCC(NC(=O)OC(C)(C)C)C2)ccc2cc(F)c(F)cc2n1 CCCCC(O)C(=O)NCCCCCNC(=O)C(CN(C)C)C(C)C Cc1cc(CCC(=O)NC(C)(CNC(C2(C3(C)CC3)CC2)=O)C2CC2)cc(C)n1 CC1=C(c2ccc(NCc3cc(OC(F)(F)F)ccc3Br)s2)CCCC1 Cc1cccc(C(C)NC(=O)C(CCC2CC2)NC(c2conc2C)=O)n1 c1(NC(=O)NC2(c3ccccc3)CCC2)ccc(=NCc2ccc(Br)cc2)[nH]c1 C1(c2onc(-c3cnc(C)[nH]3)n2)C2CCCOC12 Cc1ccc(NC(=O)NC2C=CCC2)nc1 CC(CCCC(=O)NCCNC(C1(C#N)CC1(C)C)=O)c1ccccc1 [N-]=[N+]=NCCCCCCCNC(=O)NCCOC(COC(F)(F)F)CC(=O)O c1(C(=O)NC(c2ccc(F)cc2)c2ccc(C)s2)c[nH]ccc1=N C(=O)(CCC(CC1CCCC1)NC(=O)NC1(O)CCN(C(=O)NC(C)C)CC1)OC N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(C1C3CN(C)CC13)=O)C2 C12(NC(CCc3ccc(C)c(C)c3)=O)CCOCC1CN(C(c1cccs1)=O)C2 N1(C(c2ccccc2F)=O)CCN(C(c2cscc2Cl)=O)C(C2CCC2)C1 c1(C(N2CC(F)(CNC(c3ncn(C(C)C)c3)=O)C2)=O)c(F)cc(Cl)cc1F C1(NC(C(CSC)O)=O)CCN(C(=O)CNC(c2ccc(C)c(C)c2)=O)CC1O C1(C)(C(=O)NC(CNC(C(CCSC)(C)C)=O)CO)CC(C(C)(C)C)=NO1 C1(CC)CCC(C)CN1C(c1ccc(C2CC2)cc1)C(=O)NC1CC1C1CC1 Cn1c(Cl)cnc1C(F)(F)C(=O)NCC1(NC(c2ncc(Cl)s2)=O)CCCC1 C1(C)(C(=O)NC(C)CCN(C)C(c2cccc(=O)o2)=O)CC(C(C)(C)C)=NO1 C1(OC)CC(CNC(c2c(C)ccn2C)=O)N(C(c2cc(C(C)=O)cn2C)=O)C1 N1(C(CCN(C(C2(C)C(C)C2)=O)CC2CC2)=O)CC(CO)CC(C)(C)C1 c1(CC(=O)NC(C(CC)C)CC(=O)O)c(C)nc2cc(O)nn2c1C.C1C(=O)N1 c1(SCC)c(C2CC(F)(CNC=O)C2)nnn1CC.C(=O)(CN(CC)CC)CC c1(-c2nn(C)c(-c3cccc(-n4cnn(C(F)F)c4=O)c3)n2)cc(F)cc(F)c1 C(=O)(C(=O)C(C)(C)C)NC(C)CCC(=O)N1CCC12CCC2 C(=O)(C1c2ccccc2NC1C)NC1(C=C)CCOCC1 CCC(C)(C)C(O)C(=O)NCC1CCCN1C(c1cc(F)cc(OC)c1N)=O C#CCC(C)(C(=O)NCC1(C)CSC(C)=N1)NC(C1CC1(C)C(F)F)=O N1(C(C(CC=C)NC(C)=O)=O)CCN(C(=O)C=C2CCC(C)C2)CC1CCO C1(NC(C(C(C)(C)C)O)=O)COC2C(NC(=O)CCc3n[nH]c(=N)s3)COC12 N1(C(c2ccc(N(C)C)cc2)=O)C(CNC(C23CC2C3)=O)CC2COCC12 C(=O)(C1OC(=O)c2ccccc21)NCC(C)(C)NC(Cc1ccc(OC)cn1)=O c1(CCC)ccc(C(=O)NCCCCCN(C)C(c2cc(OC)no2)=O)cc1Cl N1(C(C(CCCC)NC(N)=O)=O)CCC(NC(C2CCCSC2)=O)C(CO)CC1 Cc1cc2c(c(NC(=O)CCCO[Si](C)(C)C(C)C)c1C)CCCC2 C12(NC(CCCOC)=O)CCCCCC1N(C(c1cc(C)cnc1N)=O)CC2 C1(C(=O)NCCN(C(=O)C(c2cccnc2)C)C(C)C)CCC2(CC2)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CCNC(c2ccco2)=O)CC12CCC2 C(CC(=O)N1CCC1CNC(=O)C(OC)OC)SCCCC C(=O)(C1=COCCO1)N(C1CCCC(N(C(CCCOC(C)C)=O)C)C1)C c1(C(N2CCC(c3nc[nH]n3)C2)=O)cc2scc(Br)c2[nH]1 C1(C(N(CCNC(=O)CC2SC(=N)NC2=O)CC)=O)CN(C)C(=O)CCO1 c1(C(=O)NCC2CCCC(NC(C3(C)C=CCC3)=O)C2)nccn2nccc12 N1(C(CC2ON=C(C)C2)=O)CCC(CC(C)NC(c2occc2F)=O)CC1 C(=O)(CCC(=O)NC1CCN(C(c2cc(O)nn2C)=O)C1)N(CC)CC Cc1cc(C(N2CC3(CCN3C(=O)C(C(C)C)N(C)C)C2)=O)c(S(N)(=O)=O)s1 C1(C(=O)NCCCCCNC(C(c2cncc(F)c2)C)=O)CCC(CO)CC1 C1(NC(C2C(C)(C(C)C)C2)=O)CCC2(CCc3ccccc32)CC1 N1(C(C(C)(O)CSC(=N)N)=O)CC2(CCCN(C(=O)C(O)Cc3cnc[nH]3)C2)C1 Cc1c(C(=O)NCCOCCN(C)C(C2CCCC2O)=O)cccc1Br c1(CNC(C(C2CCC2)NC(C(C=CC)O)=O)=O)cccnc1F C1(C(N(C)CCc2ccncc2)=O)CC12CCN(c1nnc3ccccn13)CC2 C1(NC(C(C)OCCOC)=O)CC2C(NC(c3cc(SC)c(C)o3)=O)C2C1 N1(C(=O)C(O)c2ccsc2)CC2C3CCC(C2C1)N(C(c1cc(O)cs1)=O)C3 CN1CCc2[nH]nc(C(=O)NCC34CCC(CC3)N4C(=O)C=CBr)c2C1 N1(C(CC2CC(=C)C2)=O)CCC(C(=O)NCCOCCCF)(C(C)C)C1 CC(C)CC(C(=O)NC1CCCC(NC(c2ccoc2)=O)C1)C(N)=O S(=O)(=O)(c1ccc(Br)cc1NCC(C)(C)CS(N)(=O)=O)NC(CN(C(C)C)C)C CCCCCCCC(=O)NC(CC(N)=O)C(=O)NC(CC)C(C)C c1(C(N2CCCC(NC(c3ccc(CC)o3)=O)CC2)=O)ccc2c(c1)OCCC2 Cc1n[nH]c(C)c1SCC(=O)N(CCN(C(=O)CC(C)F)C)C(C)C N1(C(C2N(Cc3c(Br)cn(C)n3)CC3(CC3)C2)=O)CCC2(CC1)CC(C)(O)C2 CC1(C(=O)NCC(CO)NC(c2ccccc2OC(F)F)=O)CCC(=O)N1 S(=O)(=O)(c1cnn2ccc(=NCc3cc(Cl)n(C)n3)[nH]c12)N1CCC(C(C)O)C1 C1(SCCCC)CCCCN1C(=O)Nc1cccc(NC(=O)CC2CCCC2)c1 C1(NC(c2csc(CO)n2)=O)CCCCCC1C(N1CCC2CCC12)=O c1(C(=O)NC2CC(N(C)C(c3cncc(N)c3)=O)C2)ccc(Br)c(F)c1F c1(C(N2CCC(C)C2c2cn(CC3(O)CCC3)nn2)=O)c(F)ccc(F)c1Cl c1(C(C)=O)ccc(C(N2CC(n3cc(C(O)C(C)(C)C)nn3)C(C)C2)=O)cc1F N1(C(C2CC(N(C)C)C2)=O)CCC2CCN(C(c3cccc(CO)c3)=O)CC12 N1(C(CC(C)(F)F)=O)CCCC(C2CCCN(C(=O)CCC3CCC3)C2)C1 c1(C(=O)NC23CN(C(c4cccc(OC)c4)=O)C(C2)C3)c[nH]c2nccc-2c1 C1(C(N2CC(C(C(=O)NCc3c(C)con3)O)C2)=O)CN(C)CCO1 Cc1cc2[nH]c(C(N3CCCC3(C)CNC(=O)CCc3ccncc3)=O)cc2s1 c1(CC)ccc(C(C)C(=O)NC2CCC(Nc3nccc(OCC)n3)C2)cc1 C(CCCCCCSc1cnn(C)c1)NC(N(C)Cc1cnc(C)s1)=O N1(CC2(NC(C(C=CCCC)O)=O)CC2)CCN(C(C2CC3CCC3C2)=O)CC1 C1(NC(C2CCN(CC)C2)=O)CC2CC(NC(C3(CC(C)=O)CC3)=O)C2C1 N1(C(c2c(C)cc(F)c(Cl)c2)=O)CCC2(CC1)CCN(C(C13CC(C)C1C3)=O)C2 N#CC1(C(N2CCN(C3CCCC4(CC3)CC4)CC2)=O)CCCC(=O)C1 C1(OC)CCn2cc(C(=O)NCCn3c(C(C)C)nc4ccccc34)nc2C1 N1(C(C(C(C)(C)C)=O)=O)CC2CC(C(=O)Nc3cc(Cl)cnc3O)C(C2)C1 C=CC1(O)CN(C(=O)CCOCCNC(=O)C=CC2(C)COC2)C1 c1(C(C(=O)NCC2CC(O)(CNC(c3coc(Br)n3)=O)C2)O)ccc(F)cc1 CC1OCCCC1C(=O)N(CCNC(c1cnc(C2CCCO2)s1)=O)CC1CC1 c1(CN(C(=O)NCC2CCN(C(C)C)CC2)C)nn(C)c(Cl)c1Br c1(C(N2C(CN(C(C(C)=CC3CC3)=O)C)CC(F)C2)=O)ccc2n[nH]c(C)c2c1 CCC(C(=O)NCC1CCCC1NC(=O)CCNC(N)=O)OCc1ccccc1 C(=O)(C1=CC2(CCN(C(c3sccc3OC)=O)C2)C1)N(CCF)CC c1(OCCCn2cc(CCCC)nn2)ccc(C(=O)N(C2CC2C)C)cc1 c1(C(=O)OC)cncc(C#CCNC(C2CCC(c3ccccc3)O2)=O)c1 CCC(C(=O)NCCC1(O)CN(C(=O)C(=O)Cc2ccccc2)C1)C(C)O CCC(CC)CCC(=O)N(C(C)CCNC(c1cc(C(C)(F)F)ccn1)=O)C c1(CC(=O)NCCCCN(C)C(C2(C)CC(F)C2)=O)cc(F)ccc1F C1(CNC(=NCCC)NC(C)COC)CCc2nncn2C1 CCC(C)CCCCC(=O)NCC1(C)CC(F)(F)CN1C(c1cc(OC)cs1)=O C(=O)(C(CC)C(C)(F)F)NC(CC=C)CNC(c1cc(C)n(C2CC2)n1)=O c1(CC(=O)NCC2CC2NC(C2CCO2)=O)ccsc1Cl CCC(C)C(O)CC(=O)N1CC(F)CC1C(=O)NCC1(C#N)CC1 N1(C(C(c2ccc(C)cc2)OC)=O)CCc2ncsc2C1.C1(=O)NOCC12CC2 N1(C(C2(COC)CC=CCC2)=O)CCC2(CC(NC(=O)Cn3nccn3)C2)C1 c1(CCC(=O)NCC2CC3CCC2N3C(C2CC(O)C2)=O)ccc2nc[nH]c2c1 c1(N(C)Cc2c3cc(C)[nH]c3ccc2)nc(=NCC2(C)CC2(F)F)[nH]c2c1CCC2 C(=O)(C(O)CC(N)=O)NC(COC)CNC(c1cc(C(C)C)oc1C)=O C1(c2n(CCOCC)nnn2)(NCc2cc(OC)ns2)CCSC1C c1(CC(=O)NC2CCC(CNC(c3sccc3Cl)=O)C2)ccc(F)cn1 C1(C(=O)NC(C)C(=O)NCC2(O)CC(O)C2)CCN(C)C1=O N(C(=NCCCCl)NCc1c(F)cc(F)cc1F)C(C)CCc1ccccc1 N1(C(C)C(N2CCCCC2SC(C)C)=O)CCCC(CNC(=O)C2CC2)C1 c1(C(=O)NC2CN(C(C(CC)CC3CCCC3)=O)CC2O)cn2cccnc2n1 N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(C1(CN(C)C)CC1)=O)CC(C)O2 N1(C(c2c(OC)n[nH]c2)=O)CCN(C(c2cc(Br)co2)=O)C(C2CCC2)C1 C1(C(C(=O)NC2CCCC2)N(C2CCOCC2)CCN(C)C)CCCOCC1 C1(C)(CNC(C2(COC)CCOCC2)=O)CN(C(C2CCCO2)=O)C(C)(C)C1 C1(C(=O)NC(C2CN(C(C3(C)CCCC3)=O)C2)C)(COC)CCCO1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CC2CN(C(=O)C#CC(C)C)CC12 N1(C(C(CC)N(C)C)=O)CCC(C(F)CNC(=O)Cc2ccsc2Cl)CC1 O=C(CCCNC(=O)NC1(CCO)CC1)NCc1cc[nH]c1 C#CCC(C(=O)Nc1ccc(C(C)C)nc1)NC(c1csc(C)n1)=O C=C1CN2C(=O)CCC2(C(N2CCC(C)(NC(c3cn(CCO)nn3)=O)C2)=O)C1 N1(C(C(N2CCCCC2=O)C)=O)CC(NC(=O)CC2CS(=O)(=O)C2)C2CC2C1 N1(C(C(CC)C#N)=O)CC2(CCN2C(c2ccc(C(C)(C)C(F)(F)F)cc2)=O)C1 C1(C(=O)NCC(CC2CC2)OC)(NC(c2cc(C(C)C)on2)=O)CCC(C)(C)C1 c1(CN(C(=O)NCC(COC)C(C)C)C)c(C)cccc1F N1(C(c2ccc(C)c(N)c2)c2n(-c3c(C)cccc3)ncc2)CCCCCCC1=O C1(C(=O)NC(c2ccc(Cl)cc2)c2n(C)ccn2)C2CCC1(C)C2(C)C CCCC(C(=O)OC)C(=O)NC(C)(CNC(c1cccc(C)c1C)=O)CC C(=O)(C1CCCc2nn(C)cc21)N1CC2N(C(C3C(C)C3)=O)CC(C2)C1 C12(C(N(C)CCNC(=O)CC3(O)CCCCC3)=O)CCC(C)(CC1)CO2 CCC(C)CC(C)C(=O)NCc1cccc(CNC(=O)C(c2ccccc2)O)c1 N1(C(C23CC(C)(C2)C3)=O)CC2=C(C1)CN(C(c1c[nH]cc1Br)=O)C2 N1(C(C2(COC)CC=CC2)=O)CC(C)C(NC(=O)Cc2c(C)noc2Cl)C(C)C1 N1(CC(=O)NCCC2(O)CN(C(CCc3ccc(C)o3)=O)C2)CCCCC1C N1(C(c2cc(C)c(Cl)s2)C(=O)NC)CCCC(N2CCOCC2)CC1 c1(C(=O)NCC(C(C)O)C)ccc(CNC(c2ccc(Cl)cc2)=O)cn1 Cc1ncc(C(=O)N(CCCCN(C(=O)CC2(N(C)C)CC2)C)C)cc1N N1(C(c2cccc(NC(CC3CCCC(C)O3)=O)c2)=O)CC2CCCC(C2)C1 c1(OC)cc(NC(C2CC(F)(F)CN2C(c2ccc(N(C)C)s2)=O)=O)nc(Br)c1 N1(C(CS(CC)(=O)=O)=O)CCC2C(CCCN2C(=O)CCP(C)(C)=O)C1 C(C)(CCC(=O)NCC1CC(F)(CNC(C2COC(=O)N2C)=O)C1)SC n1(CC)nc(C(C)C)cc1C(=O)N(C)CCNC(C1C2CCC(=O)C12)=O C(=O)(C(C)(C)CS(C)(=O)=O)N(CCN(C)C(c1ccc(Cl)c(C#N)c1)=O)C N1(C(C(C)NC(CC)=O)=O)CCCN(C(C2(OC(C)=O)CCOC2)=O)CC1 C1(NC(C2(C)CCCO2)=O)CN(C(c2ccc[n+]([O-])c2)=O)C2(CCOCC2)C1 c1(C(N(C)CC2N(C(C3OCCC(C)C3)=O)CCC2)=O)cccc(N=[N+]=[N-])c1 C(=O)(CC1=NNC(=O)C1)N1C(CNc2n(C(CC)CC)ncc2)C(C)CCC1 C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCCNC(COC)=O C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)CC(F)CN(Cc2occc2Br)C1 C12(COC1)CC2.C(C(C)(C1CC1)NC(c1cscn1)=O)NC(=O)OC(C)(C)C c1(C(=O)NCCC(CNC(C(COC)C)=O)O)cc(C)c(C)cn1 Cc1ccc(C(=O)O)cc1C1CC1.c12cc(ccc1F)NC(=O)CCn1cc-2nn1 C12(CN)CCC(C(N3CC(c4ccccc4)C(N)C3)=O)(CC1)C2 Cc1ccc(CC(N2CCOC(CC(N3CCC(O)C3)=O)C2)=O)cc1[N+](=O)[O-] c1(N2CCCC(CSC)C2)ncc(S(=O)(=O)NC2CCSCC2)cc1Cl CCCC(C)C(=O)NC(CNC(=O)Cc1nnc(O)s1)CC Cc1c(NCc2ccc(C(N)=O)cc2)ncnc1NC1CCOCC1CC(C)C C1(C(=O)NC23CC(NC(=O)CNC(c4cccnc4)=O)(C2)C3)OC2CCC1C2 N1(C(c2c(C)oc(CNC(=O)C(C)CC3CC3)n2)=O)CC[Si](C)(C)CC1 N1(C(CN2CC(CC)C2)=O)CCC2(CCN(C(=O)C=C(C)C3CC3)CC2)C(C)C1 c1(C(=O)NCCC(C)NC(C2=CC(C)CC2)=O)ccc2oc(O)nc2c1 C(=O)(C(C)CC(C)(C)C)N(CCCNC(CCc1c(C)noc1)=O)C1CC1 O=C1NC2CCCC1CN(CC(c1ccc(OC(F)F)nc1)N1CCCC1)C2 CC1(C)CCCN(C(c2cc3ccccn3c2)=O)C1C(N1CC(F)(CO)C1)=O N#Cc1cc(C(=O)NC2(CNC(c3ccc(CO)nc3)=O)CCOCC2)on1 C=CCCCCCC(c1nnnn1C1CCC(F)(F)CC1)NC1(CC)CCOC1 N1(C(c2nc(Br)c[nH]2)=O)CCN(C2CCN(C(C3CCOC3)=O)C2)CC1 C(=O)(CCC(C)C)NC1(CC=C)CN(C(c2cncc(C)c2)=O)C1 c1(C2CN(C(C3CC(n4cc(CCOCC(N)=O)nn4)C3)=O)C2)cccc(F)c1 N1(C(COCCOC)=O)CCC(C(N2CC(C3CCCO3)C2)=O)(C(C)C)C1 C1(NC(C2CC3CCC(C2)C3F)=O)CC2CCC(C1)N2C(c1ccns1)=O Cc1cc(NC(c2cncnc2C2CC2)=O)ccc1NC(=O)CN(S(C)(=O)=O)C C(=O)(CCCC(C)(F)F)NCCC1CCCN(C(CCC(=C)Br)=O)C1 C1(CNC(C(CC=C)C)=O)CCC2(CN(C(=O)Cc3cccc(C(C)C)c3)C2)O1 Cc1cc(O)ccc1C(N1CCCCC1C(=O)NCc1ccnc(Cl)c1)=O N1(C(CCC)=O)CCC2CN(C(C3(Cl)CC3C(=O)OC)=O)CCC12 c1(N2C(Cc3ccccc3)CNC2=O)csc(C)c1.CCCCOCC(=O)OC c1(C(N2CCC(N(C(=O)C(C)C3CC3)CCC)CC2)=O)c(F)cc(F)c(O)c1F C(CCN(C)C(c1cc(CSC)on1)=O)(C(C)C)NC(CC1N(CC)CCC1)=O C(C)(c1ccc(F)cc1F)=CC(=O)NCC1(F)CC(CNC(C(C#C)(C)C)=O)C1 c1(Nc2c(C)c(N3CCN(C)C(C4CC4)C3)ncn2)cnn2c1OCCC2 C(C(O)CC(=O)N(c1cccc(C)c1)C(C)C)NC(C1CC(OC)(OC)C1)=O c1(OC)cccc(C)c1C(N1CC(CNC(c2cc(C)sn2)=O)C(C)C1)=O CC(C)CC(C)(CNC(c1c[nH]nc1C1CC1)=O)NC(=O)C(=O)NCCC(N)=O N1(C(c2nnc(C)s2)=O)CCOC2(CCN(C(=O)CCOCC3CC3)C2)C1 CC1(C#CC(=O)NCC(C)(C2CCC2)NC(=O)CCOCC2CC2)CC1 C1(OC)CCN(C(=O)C(CNC(c2ccc(C(C)=O)[nH]2)=O)C(C)(C)C)CC1(C)C C12(COC)CCC(C(N3CCCN(C(=O)CNS(=O)(=O)CC)CC3)=O)(CC1)CO2 c1(C(N2CC3C(NC(CC(C)N(C)C)=O)C3C2)=O)cc(Cl)cc(Cl)c1O C=CC1(CC(=O)NCCCC(C)NC(C2CCCC2c2ccccc2)=O)CCC1 NS(=O)(=O)c1cc(C(N2CCCC(Cn3cc(C4(O)CC4)nn3)C2)=O)cc(Br)c1 Cc1ccccc1-n1nccc1NC(=O)NCCNS(N)(=O)=O Cc1ccn(CC(=O)NC2C3CC2N(C(=O)C(C)c2ccco2)C3C)c(=O)c1 N1(C(C(CSC)O)=O)CCCC(n2cc(CSc3nccs3)nn2)C1 CCC(C)CCCCC(=O)NCC1CC1NC(=O)CSc1cccc(OC)c1 C1(C(=O)OC)CC(C)N1C(=O)C(C1CC1)NC(c1cn(C(C)C)cn1)=O c1(C(N2CC3C(Cn4cc(-c5ccn(C)n5)nn4)(CC3)C2)=O)n[nH]c2c1CCOC2 c1(N2C(C)C(NC(C3CC34CCSCC4)=O)CCC2)ccc([N+](=O)[O-])cc1 Cn1oc(C(N2CCC(C(F)F)(CNC(C3(c4ccno4)CC3)=O)C2)=O)cc1=O c1(C(C(=O)NC)N(C)Cc2nc(C)ccc2C)cnc(OC)c(F)c1 C1(C(=O)NCC(C(C)C)NC(c2ccncc2O)=O)C2CCN(CC2)S1(=O)=O C=CC(C)(C)C(=O)NCCC(=C)CNC(=O)Cc1ccc(CO)cc1 CCC(C)(COC)C(=O)NCCC1(O)CCCN(C(=O)CCc2ccon2)C1 c1(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCOC)ccc2nc(C)[nH]c2c1 N1(C(c2ccn(CCCC)n2)=O)CC2CCC(CNC(=O)CCSCC)C2C1 CC(C)C(C(=O)N1CC(CN(C)C(C2CCS2(=O)=O)=O)C1)n1cccc1 N1(C(C(C=C)C)=O)CCOC(CCNC(=O)Cc2c(C)cnn2C)C1 C12(CNC(C(N3CCN(C)CC3)C)=O)CCC(CN(C(=O)COC3CC3)C1)C2 C1(NC(C(c2nccc(C)c2)(C)C)=O)CC12CCN(C(C1(N(C)C)CCC1)=O)CC2 c1(C(=O)NC2(C)CC(NC(c3ccc(C(C)=O)[nH]3)=O)C2)ccc2cnccc2n1 C1(CCNC(CC(=C)C)=O)CN(C(c2ccc(C)c(Br)c2)=O)CC(C)O1 CC(C)CC(F)(F)C(=O)NC1CC1CNC(=O)CC12CCC(CC1)C2(C)C C(=O)(C(C)(C)C(N)=O)NC(CCN(C(c1nc(C(C)C)sc1)=O)C)C C(CCN=c1[nH]c2ncc(Cl)cc2s1)N(C)C(C1(C2CCCO2)CC1)=O N1(C(CCC=C)=O)CCCC(CC)(NC(c2cnccc2N2CCOCC2)=O)C1 C1(NC(Cc2c(C)nc[nH]2)=O)CC2CC(C1)N(C(=O)CN1CCC(C)C1)C2 C1(C(=O)NC(CC(C)NC(C2(C)C(C)(C)C2(C)C)=O)C)CCc2nncn2CC1 c1(C(N2C(C)CCC(NC(=O)C=C(Cl)Cl)C2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C1(NC(C2CC(C)OC2=O)=O)(CNC(c2coc(Cl)c2)=O)CCC(F)(F)CC1 N1(C(C2N(C)C(=O)CC2)=O)CCCC2CN(c3c[n+]([O-])ccc3[N+](=O)[O-])CCC12 CC1=NOC2(C1)CC(C(N1CCCCC(CNC(=O)C(=O)C(C)C)C1)=O)C2 c1(C(=O)NC(C(=O)NC(CCC)C(C)(C)C)C(C)O)c[nH]c2ncccc12 C1(CNC(=O)C=CC=C(Cl)Cl)CC2CCC1N(C(=O)CCC1CC1)C2 c1(C(=O)NC(C(=O)NC(C)CC2CCCCC2)CCC2CC2)cncn(C)c1=O c1(CC(=O)NC(CCNC(c2c(C)c(N)n(C)n2)=O)C)cn2c(C)cncc2n1 N1(C(Cc2c(CC)noc2CC)=O)CCCN(C(=O)C(F)C(F)(F)F)C(C)C1 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C(F)(F)F)o2)=O)CC1OC C1(C(=O)NCC2CC(C(=O)NC3(CCCF)CC3)CO2)CC2(C1)CC2(F)F C(=O)(C(C(C)(C)C)NC(C1CC2CC2C1)=O)N1CC(N(C)C(=O)OC(C)(C)C)C1 C=CC1(C(=O)N=c2ccn(CC(C)C)[nH]2)CCN(C(=O)Cc2ccc(C)s2)CC1 c1(C(N2CCC(CC=C)(NC(=O)CCc3cn[nH]c3)C2)=O)cc(=O)n(C)cn1 CC1CC2(CCN(C(=O)NC3CNC(=O)C(C)(C)C3)C2)CO1 c1(C(=O)NC(CCOC)CNC(=O)CN(C2CCC2)C)cc(SC)oc1C CC1C(NC(c2cnn(C)c2C#N)=O)CCCN1C(=O)CCOC1CC1 c1(C(=O)NCCc2ccc(Cl)c(Cl)c2)nc(Br)n2c1CCCC2 C1(NC(C(C)O)=O)CCCN(C(c2ncsc2Cc2ccccc2)=O)C1 c1(C(=O)NCCCN(CCO)C(c2nnc(O)nc2O)=O)cc(F)c(F)cc1Cl N1(C(c2c(CC)onc2C)=O)CC2CCCCC2(CNC(=O)CS(=O)(=O)NC)C1 C(C(COC)C(=O)NCCCCCCN(C(=O)CC1SC(=N)NC1=O)C)OC c1(CC(N2CCC(C3CCCN3C(=O)Cc3ccsc3)C2)=O)ccc(O)c(F)c1 CC1CCCN(C(=O)C(=O)NCc2nc(CNC(c3cn[nH]c3)=O)cs2)C1 CC1CCN(C(=O)CCCC(=O)C2CC2)CC1NC(C1CN2CCC1CC2)=O CON1CCC(C(=O)NC(C)CCN(C)C(c2ccc(C#N)cn2)=O)CC1 c1(OC)cccc(CC(=O)NCC(C)CN(C(=O)C(n2nccc2C)C)C)c1F C1(C#N)(C(=O)NC(CC)CNC(=O)Cc2nncn2C(C)C)CCCOC1 C1(C(C)NC(C2(CO)CCCC2)=O)CCCN1C(C1CC(N(C)C)C1)=O C1(OCC)CCC(C(=O)NCCCNC(=O)C(c2ccnn2C)C)CC1 CC(CNC(=O)C(F)n1ccnc1)CC(=O)N1CCCC1CC1CC1 C(=O)(C1=C(C)OCCS1)N1CCN(C(CCSCCCC)=O)CC1CCC C#CCC(C(=O)NCC1CCCNC1=O)NC(c1ccn(C2CC2)n1)=O N1(C(c2c(C(C)C)onc2)=O)CCC(N(C(=O)CSc2cnn(C)c2)C)C(C)C1 N1(C(c2ccc(C)cc2C)=O)CC2CC(NC(=O)C(C)NC(N)=O)CC2C1 C1(CNC(CC2C(CNC(CCCOC(C)=O)=O)C2)=O)CCOC1(C)C CC1COc2ccc(C(=O)NCC(C)(C)NC(=O)C(C)C(C)O)cc21 C1(NC(C2N(C(c3ncn(CC)c3)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N12CCC3CC1CN(C3)CC2=O.c1(CCOC)ccc(C(=O)OC)cc1 C=CC(C)(O)CC(=O)NCC1CCCC1NC(C1CC(C(F)(F)F)C1)=O CN1CC(F)CC1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O c1(C(=O)NCCC(C)N(C(CCc2scc(C)n2)=O)C)cnc2sccn12 Cc1nc(NC(C2CSCCN2C(c2ccc(O)c(I)c2)=O)=O)c(C#N)n1C O=C(CC1=CCCCC1)NCCC1CN(C(C2CCc3nnnn3C2)=O)C1 CCCCC(CC)CC(=O)N1CC(NC(=O)CC(C)(C)O)C(C)(C)C1 C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCNC(=O)NC)=O)C1 c1(C(N(CCC(C(C)C)NC(CC2(C=C)CCC2)=O)C)=O)ccc(C)nc1C Cc1ccc(C#N)cc1C(=O)NCC1(NC(C2C3CC4C(C3)C24)=O)CC1 c1(C(N(CCC=C)CC)=O)cc(CC)no1.C(=O)(CC1(CO)CC1)NCCN C=CCC(C)(C)CC(=O)N1CCC(NC(c2cc(C(N)=O)cn2C)=O)C12CCC2 CC1(C#CC(=O)NCC2CC3CCC2N3c2ccnc(C3CCC3)n2)CCCO1 C1(Cl)(C(N2CC(C(N)=O)(CNC(C3CCCC3O)=O)C2)=O)CC12CCC2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)OC)C2(C)C)cnc(Cl)n1C c1(C(=O)NC2CC3CN(C(Cn4c(C)cnn4)=O)CC32)ccnc2c1CC(=O)N2 c1(CNC(C2CCC(C#C)CC2)=O)nc2c(s1)CN(C(=O)CC1CCOC1)CC2 CC1CC(C(=O)NCC2(C(=O)NC(=O)CCCNc3cccs3)CCC2)CO1 C1(OCC)(CNC(N2CCC(O)C2)=O)CCCCC1.C(CC(C)C)CCN(C)C CC(=O)CC(C)(C)CC(=O)NC(CNC(c1ccc(Cl)cc1C)=O)C1CC1 C1(C(=O)NCCc2ccncc2)CCN(C(c2cccc(F)c2O)=O)CC1O c1(OC(C)=O)ccc(C=CC(N2CC(C(=O)Nc3c(F)cccc3I)C2)=O)cc1 C1(CCNC(c2[nH]cc(C(N)=O)c2)=O)CCCCN1C(=O)Cc1cccc(Cl)n1 N1(C(CN(CCC)C)=O)CCC2(CC1)CC(C)N(C(C1CC3CCC3C1)=O)C2 N1(C(CC=CC=C)=O)CCC(NC(C2CCCN2C2CC2)=O)CC1C c1(OC)c(Br)cc(CNC(C2CCN(c3nccc(C)n3)CC2)=O)cc1[N+](=O)[O-] CC1CCC(C(=O)NCC2(C3CC3)CC2)CN1C(C1(CF)CC1)=O N1(C(c2c(C)oc(Cl)n2)=O)CCC(C(=O)NCC2OCC3CCC2C3)C12CCC2 C1(C(N(C(CN(C(c2cncc(OC)n2)=O)C)C)C)=O)CC2C(C1)C2(F)F CC#CC1CCN(C(=O)C(C)(CNC(=O)COCC2CCOC2)CC)C1 Cc1nc2c(o1)CCN(C(C1CCC(C)C(C)C1)=O)C2 C1(N(C(C2CC2c2ccco2)=O)CC)CCN(C(=O)CC2CCC(=O)N2C)CC1 C1(CNC(c2c(C)nc(CCC)o2)=O)CN(C(=O)CC2CCC(O)C2)CCN1C N1(C(C=C(C)C2CC2)=O)C2CCC(C2)C1COC(C)(C)C.C12(CC1)C(=O)N2 c1(C(N2C(C(=O)NCCOCC(C)C)C(C)CC2)=O)cc2cccnn2c1 c1(C(=O)NCCCN(C(=O)C(CO)C(C)(C)C)CC)cccc2ccoc12 C(=O)(C1=NOC2(CCN(Cc3cc(Br)ncc3Cl)C2)C1)N1CCC(OC(C)=O)C1 N1(C(=O)Nc2ccc(C(=O)OC)o2)CCC2CN(Cc3cc[nH]n3)CCC12 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCN(C(=O)C(c2ccc(F)c(C)c2)=O)CC1 C1(N(c2cc(C)nc(C(C)(C)C)n2)C)Cc2ccccc2C1C c1(NC(C)=O)ccc(C(=O)NCCN(C(=O)CC2CC2(Cl)Cl)C2CC2)nc1 C1(NC(CC(=O)NCC)=O)C2CC3C1C3C2C(=O)NC(c1nc(C)c(C)[nH]1)C c1(OCCC(=O)N(CC(CC)NC(c2ncccn2)=O)C)ccccc1O N1(C(C(C)OC)=O)CC(O)CC1CNC(C1C2CCC1CC2)=O C(=O)(C(C)(C)C1=CCSCC1)NCC(C)N(C)C(C1CCN(C)S1(=O)=O)=O c1(C(=O)NCc2ccc3occc3c2)n[nH]c2ccc(-c3ccnc(F)c3)cc12 CC1(C)CCC(CC(=O)NCCC2(O)CN(C(c3cc(Cl)nc(=N)[nH]3)=O)C2)OC1 CN1CCCCC(C(=O)NCC2CC3CCC2N3C(C2CCCCN2C)=O)C1=O N1(C(N(CCC)CCc2cc(C(F)(F)F)cs2)=O)CCCC1CC c1(C(N(CCC(C)NC(Cc2cnc(C)o2)=O)C)=O)n[nH]c2c1CCC2 CC(C)(C#Cc1cn(CCCOC(=N)O)nn1)NC(=O)C(C1(O)CCCCC1)O N1(C(C(C)(C)SC)=O)CCC(C2CN(C(=O)C(CO)C(F)(F)F)C2)CC1 CCCCCCC(=O)NC(CCCOC)C(=O)N(C1CCC1)C1CCC1 C1(=O)C(C)(C)C(=O)Oc2c(sc(C)n2)C(=O)NCC2CC(C2)N1.C(C)(C)(C)OC N1(C(C2CC(C(=O)NC3C(O)CC3O)C2)=O)CC(O)(CO)C1 C1(C(N(CCOC)CCNC(=O)CC(C)(C)C2CCCCC2)=O)C(C)OC(C)C1C N1(C(C2(NC(=O)C3CC3)CC2)=O)CC2CC(C1)CN(C(c1coc(O)n1)=O)C2 n1(CC(=O)NC23CCN(C(C4(O)CCCC4)=O)CC2C3)cnc2ccccc12 N1(C(COCCC(C)C)=O)CC(NC(=O)C(C2CCOCC2)C)C(F)C1 c1(C(=O)Nc2c(C)cccc2)ccn2c1CS(=O)(=O)CC2 N1(C(c2ncc(CC)s2)=O)CCC(NC(=O)C(C(C)C)NC(=O)COC)C1C N1(c2cc(F)nc(-c3ccccn3)n2)CC2C3CCC(CC3)C2C1 c1(OCC)cc(NCc2cccc(NC(=O)C(c3ccnn3C)O)c2)nc(C)n1 N1(C(C(CC2CCCC2)OC)=O)CCOCC1CCNC(=O)Cn1cnnc1O c1(-c2nc(C(c3ccccc3)COC)on2)ccc(C2(n3cc(Br)cn3)CC2)cc1 C1(Cl)(C(COC(CSCC)=O)=O)CC1C(=O)NC1CC1 C1(C(C)(C)NC(=O)Cc2ccsc2)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 c1(C(=O)NC2C(CNC(CCCCC#C)=O)COC2)cc(C)c(OC)c(C)c1 CC(=O)CCCC(=O)NC1CCCC(NC(C2CCCC23CC3)=O)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(c2ccc(C#N)c(C)n2)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)F)NC1CC(CNC(CC=CCC)=O)C1 Cc1ccc(N2CC(C(=O)NCC(O)CCNC(=O)C=CCO)CC2=O)cc1 CC1(CCNC(c2cccc(Cl)c2)=O)CCN(C(C2CCCC3CC23)=O)C1 Cc1scnc1C(=O)NCCC(C)(C)NC(=O)CCc1nccn1C N1(C(N(c2ccccc2)CC)=O)CCC(C)CC1CNC1CCC1 C=CCCCCCC(=O)N1CCC(N(C(=O)CCCSc2ccccc2)C)CC1 C#Cc1cc(C(=O)N(C2C3CN(C(c4cnc(O)n4CC)=O)CC23)C)cc(F)c1 N1(C(=O)CCc2ccncn2)CCC2CC12C(N1CCC(F)(F)C1)=O CN1C(=CC(N2CCc3sc(C(=O)O)cc3C2)=O)C(C)(C)c2ccccc21 CC1CN(C(c2cc(Cl)cc3cc[nH]c23)=O)c2cccc(Cl)c2O1 C(=O)(C(C)S(C)(=O)=O)NC(CC(C)C)CNC(=O)C=CCOc1ccccc1 c1(C(N(C(CNC(C(C(C)C)NC(N)=O)=O)C2CC2)C)=O)cccc2c1COC2 N1(CC)CCOC(C)(C(=O)N(c2ccc(OC)cc2)Cc2occc2C)C1 C1(CC(=O)Nc2cc(-c3cccs3)on2)CCCN(C(=O)C(C)(C)OC)C1.CC C1(NC(c2cocn2)=O)CCN(C(C2CCC(C(N)=O)C2)=O)C12CC2 CC1(C)CCC(O)(C(=O)NC2CC(F)(CNC(=O)CCNC(N)=O)C2)CC1 N1(C(CC(C)(C)OC)=O)C(CNC(=O)C(C)(C)C(C)(F)F)CC2COCC12 CC1CN(C(c2cnc[nH]2)=O)CCC1NC(c1cnnc(O)c1)=O CN1C(=O)CCC1C(=O)NC1C2CC1N(C(=O)C=Cc1ccccc1)C2 C1(NC(c2ccc(C3CC3)nc2O)=O)CCCCN(C(C2(O)CCCC2)=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(N(C(=O)CC2C=CCC2)C)CC1 c1(CCNC(=O)NC2CN(C(=O)OC(C)(C)C)CC2O)c[nH]c2cnc(Cl)cc12 N1(C(C2(CCOCC)CCCC2)=O)CCC2(COC(CNC(=O)CNC=O)C2)C1 C#Cc1ccc(C(=O)N(C2CN(C(c3csc(CC)n3)=O)CCC2C)C)cc1C C1(C)(CC(=O)NCCCOC=C)CCN1C(=O)CCOCCOC CN1CCC(C(N2CC(N(C)C(c3cscn3)=O)C(C)(C)C2)=O)S1(=O)=O C(=O)(C(CCc1cnn(C)c1)N1CCCC1COC(C)(C)C)NC(CC)C C1(CCOC)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CO)n2)=O)CC1 c1(C(=O)NCCN(C(C)C)C(C2CC23CCC3)=O)cc(C(F)F)cc(F)c1 C1(C(N2CCC(N(C(CCOC)=O)C)C2)=O)CCC(C(C)(C)O)CC1 N1(C(C2CCC(OC)CC2)=O)CC(C2CCCN(C(=O)C(F)n3cccn3)C2)C1 CC1CC(CNC(C2(F)CCCCCC2)=O)CN(C(C2(CN(C)C)CC2)=O)C1 c1(CC(=O)NCC2(NC(c3n[nH]cc3C(F)(F)F)=O)CC2)csc(C2CC2)n1 c1(C(N2CC(C=C)C(NC(=O)C(O)CC(C)C)C2)=O)c(C)cc(C)oc1=O CC(CNC(c1ccn(C(F)(F)F)n1)=O)(CO)NC(=O)C=C1CCSCC1 CCCCC(O)CC(=O)N1CCCCC(NC(c2cc(OC)ccc2F)=O)CC1 CCCCC(O)C(=O)NCc1cc(O)nc(CNC(c2cc(O)n(C)n2)=O)n1 N1(C(CCN2CCN(C)CC2)=O)CCCC(O)(CNC(=O)CCn2cccc2)C1 N#CC1(C(N2CC3CC3(CNC(=O)CCC3CCC3)C2)=O)CCCOC1 c1(C(=O)NCC23OCC(CNC(C4C(C)OCCC4)=O)(C2)C3)cc2ccsc2s1 N1(C(CSSC)=O)CCC2(CCCN2C(=O)Cc2cnccn2)C1 c1(C(=O)NC2CC(CNC(C(C(C)O)C)=O)C2)sccc1S(N)(=O)=O C1(CC(=O)N(CCC(c2cccs2)NC(C(C)C2CCC2)=O)C)CCC=CCC1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(=O)NC2CCC(OCC)CC2)C1(C)C c1(OC)cccc(C(O)C(=O)NCC(C)NC(=O)Cc2cnc(C)[nH]2)c1 N1(C(Cc2nc(CC)sc2)=O)CC2CCC(CNC(=O)C(C)(C)C#N)(C2)C1 CCCCCC(O)CC(=O)N1CC(CNC(C2OCC3CCCC23)=O)OC(C)C1 N1(C(CC)CCC(=O)O)CC2(C=C(C(=O)NC3(C)CCC4(CC3)CC4)CO2)C1 N1(C(c2cccc(C(=O)NC)c2)=O)CC2CN(C(=O)C(C)n3cnnn3)CCC12 c1(C(N(C2CCCC2)CCOC)=O)cc2c(s1)CCC(C(C)C)C2 C(C(=O)NCC12CC(NC(=O)CC3CC(=O)NC3=O)(C1)C2)(C(C)C)SC N1(C(C(C)O)=O)CCC2CCCC12C(=O)NC1CCC(N=[N+]=[N-])CC1 CCC(C(=O)NC1(CO)CN(C(C2(O)CCC2)=O)C1)C1CCOCC1 CC(CC(=O)c1ccccc1F)C(=O)NCC(C(F)F)n1cccn1 CP(C)(=O)C(CC(=O)N1CCC(O)(CCNC(c2ccc[nH]2)=O)CC1)C(F)(F)F C1(CNC(c2cc(C)n(C)n2)=O)CCN(C(c2sc(N(C)C)nc2Cl)=O)C(C)C1 CS(=O)(=O)C1CN(C(C)(C)C)CC1C(=O)NS(=O)(=O)CC1CCC(F)(F)CC1 c1(CC)c(C(=O)NCC(O)CN(C(=O)C(F)=C2CCC2)C)ccn1C C=CCCCCCCCC(=O)NCCC1CCC(NC(c2[nH]cnc2C#N)=O)C1 C1(N2C(=O)OCC2)CN(N2CCC(CNC3CCCN3)CC2)C1 Cc1ccc(S(=O)(=O)NCc2ccc(F)cc2C(F)(F)F)cc1C C1(C(=O)OC)C2CC(O)C1N(C(c1cc(O)ccc1C)=O)C2 c1(C(N2CC(C(N)=O)CC(F)(F)C2)=O)cccc2c(I)n[nH]c12 C1(C(=O)NC2CCN(C(C3CC(C)(CC)C3)=O)C2C2CC2)CCc2c[nH]nc2C1 N1(C(c2c(C)nn(-c3ccc(Cl)cc3)c2)=O)CC2(N)CCCC2(F)C1 C1(C2CC2)(C(=O)NC(C(C)(C)C)CNC(=O)COCC2CCCO2)CC=CC1 N1(C(C2(CC=C)CCCCC2)=O)CC2CC(C1)CN(C(c1n[nH]cc1Cl)=O)C2 C(=O)(C(F)(F)CC)N(CC(C)N(C(C1C(CC)C1)=O)C)C CC(C)CC(O)C(=O)NC1CN(C(c2cc(-c3ccncc3)no2)=O)CCC1F C1(OC(C)C)CCC(C(=O)NC(=O)Nc2ccccc2SC(C)C)CC1 c1(C(=O)NC2CCN(C(c3c(C)snc3)=O)C(C)C2)c(F)ccc(N)c1F Cc1cccc(C(N2CCCCC2CCN(C(=O)CC(C)(F)F)C)=O)n1 c1(C(N2CC(N(C(CCC=C)=O)C)C3(C2)CC3)=O)ccc(O)c(C)c1C N1(C(c2n[nH]c(CC)c2C)=O)CC(NC(=O)CN2CCC(C)CC2)CC1(C)CC N1(C(CC2CC(=C)C2)=O)CCC2CCN(C(c3ccc(O)c(N)n3)=O)CC2C1.OC C1(CCOC)CCN(C(=O)CCN(C(C2(CO)CCOC2)=O)C(C)C)CC1 c1(OCC)cccc2c1OCC(C(=O)NC(C)C(C)NC(=O)CN(C)C(N)=O)C2 C12(C(=O)NC(CN(C(C=NOC)=O)C)C)CC=CCN1CCC2 C1(C(C)NC2(c3n(CCCC)nnn3)CCOC2)CC2(CCC2)C1 Cc1ncnc(C(N2CCN(C(=O)CC(F)(F)F)C(C3CCC3)C2)=O)c1C N=c1[nH][nH]cc1C(=O)NC1CC(CNC(c2[nH]nnc2C2CC2)=O)C1 CC(C)CCCCCC(=O)NC(C)CCCNC(=O)Cc1ccccc1CC#N c1(C(=O)NC2(CCOC)CCN(C(=O)C=C(C)Cl)CC2)n[nH]c2c1CC(C)CC2 C1(CNC(CNC(CC2(CC(=O)OC)CC2)=O)(C)C)CC2CC1CO2 c1(C(=O)NCCNC(C2CCCN(C(=O)OCC)C2)=O)ccnc(Br)c1N c1(OCC)cc(OC)cc(C(N2C3CN(Cc4cc(Cl)cc(I)c4)CC23)=O)c1 CCC(C)C(C(=O)NC1CCC(C(C)O)CC1)N(C)C(c1cc(C)cs1)=O C12(C(=O)NCCOCCN(C(C(C)CSC(F)(F)F)=O)C)CCC(CO)(CC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(=O)CN1CCN(C)C(=O)C1 C1(OCC)CCOCC1NC(=O)C(=O)NCC1CCC1COC C(=O)(CC1=CCOCC1)N1CCCC(CNC(=O)Cc2ccsc2Cl)C1 C(=O)(C(CC)C(=O)OC)N1CC(C(=O)NCc2ncc[nH]2)(CC)C1 c1(C(C)C(N2CCCC2Cc2cn(CCNC(N)=O)nn2)=O)ccccc1F CCCCCCCC(=O)NC(CC)CC(=O)Nc1cnc(C)c(CC)c1 C1(CC2C(N(C(CC=CCC)=O)C)CC2)CCN(C(=O)C=CC(C)C)CC1 N1(C(c2ccc(CNC(C(C3CCOC3)OC)=O)o2)=O)CC(CO)C1(C)C C1(NC(=O)Cn2ncnn2)CC2(C1)CC(C(=O)NCC(O)(CO)CO)C2 C=CC(F)(F)C(=O)N1CC(O)(CN(C(=O)COCCOC)C)C1.c12ocnc1C2 O=C1CC(CC(N2CCC(O)(C(=O)Nc3sncc3C(=O)O)C2)=O)C(=O)N1 c1(C(=O)NC2C(NC(c3cnc(C)nc3)=O)CCC2)cc(C)c(F)cc1Cl Cc1sc(N(C(c2ccn(C(F)F)n2)C(=O)NCC(F)F)C)c(C)c1C N1(C(CC2C(C)C2)=O)CC2CN(C(C34CC=CC(C3)OC4)=O)CC2C1 c1(C(n2nnnc2C(C2CCOCC2)NCC)C2CC2)ccc2c(c1)CCOC2 Cc1ccc(CN(C(C2CC2)C(=O)O)CCCOC(C)(C)C)cc1Br CCCCC(C(=O)NCC(C)(C)CNC(=O)C(CCC)N(C)C)NC(N)=O C1(CNC(=O)Cc2ccsc2)CC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)CO1 CC1Cc2cc(NC(=O)NCCCCCN(C)C)ccc2O1 Nc1ncccc1-c1cn(CC2CCCN(C(=O)CNC=O)C2)nn1 C(=O)(CCCC(=O)N1CCOC(CN(C)C(C2CCCC2)=O)C1)NCCC Cc1cc(NC(c2csc(NC(c3ccccc3Cl)=O)n2)=O)n(CO)n1 C(C(=O)NC(C)C)(C(C)(C)C)NC(C1(C)CN(C(C(C)OCOC)=O)C1)=O S(=O)(=O)(c1ccc(N(C)Cc2cnccc2Cl)nc1)NCC(CCCCC)(C)C c1(C(=O)NCC(CC=C)NC(C23CCCC2C3Br)=O)cc(C#N)cn1C N1(C(CC(C)(C)O)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1c1cn[nH]c1 c1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)cc(Br)c2nccnc2c1 C1(CC)CN(C(c2ccsc2C)C(=O)NC)CCO1 c1(OCC)cccc(C(=O)NCC(C2CC2)NC(c2cnnn2C2CCC2)=O)c1 N1(C(CC=C=C)=O)CCCC(NC(=O)CCc2cnn[nH]2)C1 c1(C(N(C2CCN(C(=O)Cn3cc(C#N)cn3)C2)CC)=O)c(C)nn(C)c1C C(C(O)C(F)(F)F)NCC1N(C(c2ccccc2)=O)CC1 CCN=c1cc(NC2CCCC2CNC(=O)OC(C)(C)C)cc[nH]1 N1(C(CC(COC)C)=O)CC2CCN(C(c3ccc(F)cc3OC)=O)C2C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(OC)CN(C(=O)C(O)CC(C)C)C1 N1(C(C(CNCC)c2ccccc2)=O)CCC2(CCN(C(=O)C3=CCCCO3)C2)C1 c1(C(N2CCC(N(C(=O)CCc3nncn3C)C)C2)=O)ccc2oc(=O)oc2c1 c1(C(=O)NCC2N(C(C(C)C)=O)C3C(C2)C3)nc2c(Br)cccn2n1 N1(C(C(CC#C)NC(C2CCCCCCC2)=O)=O)CCOC(C2(C)N=N2)C1 CCC(C)(C)CCCC(=O)N1CCCC(C)(C(N2CC(=O)NC(=O)C2C)=O)C1 CC(C(C)(C)C(=O)NCC1CCC(=O)O1)NC(C1CCOCC1(C)C)=O C1(NC(CC=C(C)C)=O)CC(CNC(c2cncc(C(F)(F)F)n2)=O)C12CCC2 c1(C(N(CC(C(=O)NC)(F)F)C)=O)ccc(S(=O)(=O)NCCC(=O)NC)cc1 CC(C)C(C(=O)NC(C1(O)CN(C(=O)C(c2ccc(Cl)cc2)CO)C1)C)C(C)C c1(C(=O)NC2CCN(C(C(CC)n3ccnc3)=O)C2)cc(C)c(N)cc1Cl C1(CNC(c2csnn2)=O)CC2(CCN(C(c3cn4ccnc4s3)=O)C2)CO1 c1(C(=O)NCCN(C(C(CC=C)(C)C)=O)CCOCCO)cccc2nc[nH]c12 N1(C(C(CC)N(C)C)=O)CCC2CCN(C(c3cc(O)n(CC)n3)=O)C2C1 c1(CNC(C(CCOCCO)NC(C(C)CO)=O)=O)ccc(=O)n(C)c1 c1(C(=O)NC)ccc(C(=O)NC2(CO)CN(C(=O)Cc3cncs3)C2)cn1 Cc1cc(=NCC2CC2C2CCCC2)[nH]c(=NCC2CCN(C)CC2)[nH]1 C1(N(C(=O)C(C2(O)CCC2)NC(=O)CC#N)C)CCCCC1O N1(C(C2CCSCC2)=O)CCC2C(CCN2C(c2cnc3[nH]ccc3n2)=O)C1 C(=O)(C(CC(F)F)N(C(=O)COC(F)F)C)N1CCC(N(C)C)(CC)C1 N1(C(CC(C)SC)=O)CCCC2(CCN(C(=O)Cc3nc(C)sc3C)C2)C1 C(=O)(CCCCCNC(c1cccc(OC)n1)=O)NC(CCC)C(=O)N(C)C CCS(=O)(=O)CC(=O)NC(CNC(=O)COc1ccc(C#N)cc1)CO c1(C(N(C(C)C(=O)NCc2ccns2)CCC)=O)cn(C)nc1OCC C(=O)(C(=O)C(F)(F)F)NC(C1CN(C(C2(C)COC2)=O)C1)C C(CC(C(=O)NCC(C)CNC(c1ccc[nH]1)=O)N(C)C)SC Cn1ncc2cc(C(N3CC4CCC(C3)C4NS(=O)(=O)CC(F)(F)F)=O)ccc12 O=C(C1=CC2CCC=CCCC12)N1CC2(CCN(C(C34CC(F)(C3)C4)=O)CC2)C1 C(=O)(C(C)CCC(C)(C)C)NC(c1cn(C(CCC)c2cnn[nH]2)nn1)C C1(CNC(C=CCOCCOC)=O)CC(NC(C2CCCCC2)=O)C1(C)C c1(CCCO)nc(-c2cc(Br)c[nH]2)n(CCOc2ccccc2F)n1 C12(NC(c3cnc(C(C)C)s3)=O)CCCC1N(C(=O)CCCn1ccnn1)CC2 C=CC(C)(CC)C(=O)OCCOCC1(C#N)COC1 c1(OC)ccc(F)cc1C(=O)NC1(CNC(c2c(C)ccnc2O)=O)CCOC1 CN1CC2C(C(N3CCOCC3CC(=O)NC3CC(Cl)(Cl)C3)=O)C2C1 C1(C(N(C2CCN(C(C(CC)OCC)=O)CC2)C)=O)CCCC(C)CC1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(=O)CSc1ccc(F)cc1 C#CC1CCN(C(=O)COC2CCN(C(c3ccc(C)cc3)=O)C2)C1 C1(CC(=O)NC(CN(C(C2CS(=O)(=O)C2)=O)CC)C)CCC(C(C)C)CC1 C(CC(O)C(=O)NC1CC2(C1)CC2NC(=O)CC1(c2ccccc2)CC1)N(C)C N1(C(CC2CCC(C)C2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 c1(C(N2CC(C3CN(C(CC(C)O)=O)C3)C2)=O)cc2n(n1)CCCC2O C(CNC(=O)C(C1(O)CCC1)NC(=O)C(F)F)(C(F)(F)F)OC C(=O)(C1=CCCOCC1)N1CCC(NC(c2c(C)ncnc2)=O)C1(C)C S(=O)(=O)(c1ccc(Cl)cc1)N1CC(C(=O)NCCCN2CCOCC2)SCC1 C1(CCC)(NC(=O)CCS(N)(=O)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 CCC(C(=O)OC)C(=O)NCC12CC1CN(C(c1cc(C(F)F)no1)=O)C2 C1(N(C(C(C)N(C(C)=O)C)=O)C)CCCN(C(=O)C=CCF)CC1 c1(C(N2CCN(C(CC(C)(F)F)=O)C(C3CC3)C2)=O)cncc2c(O)nccc12 c1(C(N(C)CC2CCCN2C(C2CCCCC2)=O)=O)ccc(F)c(O)c1 c1(SC)ccc(CC(=O)N(C2C3CN(C(C4CCC(=O)N4C)=O)CC23)C)cc1 C1(N(C)C(c2scnc2C(C)(C)C)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1 C(C(Cc1ccc(Cl)cc1)C(=O)NC1CCN(C(=O)CSCC(=O)OC)C1)OC C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)CSCc2ncc[nH]2)C1 C1(NC(=O)C2=CCCC2)CN(C(c2ccc(Cl)c(F)c2)=O)CC2(CCOCC2)C1 CCCCCCCCOCC(N1CC2CC(NC(=O)C(C)(C)CCOC)C1C2)=O c1(C(=O)NCC2CC3(CCC3)CN2C(c2ccsn2)=O)cc(Cl)c2n[nH]cc2c1 CN=c1nc(N2CCC(CSC3CCOC3)C2)[nH]c(=NCC(C)(C)SC)[nH]1 C1(NC(CCn2c(C)ncc2)=O)CCCC12CN(C(=O)C(C(C)C)N(C)C)C2 N1(c2c(C)c(NC3C=CCCCCC3)ncn2)CCC(C)C(F)(F)CC1 C1(C(=O)NC(CSCC)C(N2CCC(O)(C(F)F)C2)=O)Cc2nccn2C1 N1(C(c2cccc(CC)c2)C(=O)NCc2ccccc2Cl)CCNC(=O)CC1C C(=O)(C1=NNC(=O)CC1)N1CC(C)(C)C(NC(c2cc(-c3cccs3)on2)=O)C1 C(=O)(C1OCCc2c(O)cccc21)NC(C)(CO)C(F)F c1(NCC)cncc(C(=O)NCC2CCCCC2NC(c2cncc(C)n2)=O)c1 c1(C(C)C)ccc(O)c(C(=O)NC(C)C(C)NC(=O)C2=CCCSC2)c1 c1(CC(N2CC3N(C(c4nn(CC)c(C)c4)=O)C3C2)=O)ccc2c(c1)OCO2 c1(N(CC(=C)Br)C)nc(N2CC(C(N)=O)C3(CC3)C2)c2c(n1)CCCCC2 C1(=O)CCC(=O)NCCC2CC(C2)N1.C(=O)(C(F)Cc1ccccc1)NC(C)=O C1(CNC(C2(NC(C3CCCO3)=O)CC(CO)C2)=O)CC2(CC2)CO1 N1(C(c2ccn(CCC)n2)C(=O)NCC(=C)C)CCC2CC(O)CCC2C1 C(CCCCCNC(=O)CN1CCCS1(=O)=O)N(C(=O)C1=CCCS1)C C1(C(N2CC(C)C(NC(=O)C(C)C3CCCC3)C2)=O)CC2(COC(=O)N2)C1 CON(CCC(=O)NC(C)CC(C)(C)O)C(=O)Cc1ccccc1F c1(OC)csc(C(N2CC(O)(CCNC(C3CC(CF)C3)=O)C2)=O)c1OC Cc1ncc2c(n1)CCC(C(N1CCCC1(C)CNC(=O)Cc1cncs1)=O)C2 C(=O)(C(O)CC(C)(C)C)NC(C1(O)CN(C(c2cccc(SC)c2)=O)C1)C C(=O)(C(C)(C)CNC(=O)CN1CCCCC1=O)N(CC(COC)O)C c1(NC(C2C(CNC(CCCCN(C)C)=O)CCC2)=O)ccc2c(c1)OCO2 c1(C(=O)Nc2nc(C)c(C(=O)NCC3(F)CCC3)s2)cc(Br)ccc1Cl C(=O)(CCS(C)(=O)=O)NC1CN(C(c2c(OCC=C)cccn2)=O)CC1C c1(C(N2CC(O)CC(NC(CP(C)(C)=O)=O)C2)=O)ccnc2cc(Cl)ccc12 C(=O)(C(CCOCCO)NC(c1nonc1N)=O)NC1CC(C)(CC)C1 N1(C(c2ccc(CC)cc2)=O)CC2(CC2)CC1CC(=O)NCc1cc(C)ns1 c1(N(c2ccccc2)C(=O)NCC(=O)NCc2nc[nH]n2)ccc2c(c1)COC2=O N1(C(c2c(CC)cncc2)=O)CCC(O)(CCNC(=O)CCCCSC)CC1 C(N=c1[nH]c2c(c(=NCC3CC(n4ccnc4)C3)[nH]1)CCC2)c1snc(C)n1 CC1(C(N2CCC(n3cc(C(C)(C)O)nn3)C2)=O)CCCCCC1 C(=O)(C(COC)COC)N1CCC(N(CCC)C(C2CC2c2ccccc2)=O)C1 CC1CCN(C(c2ncccc2N)=O)C1CNC(=O)C(C)(C)c1cnsc1 CCC(C(C)O)NC(=O)C(C)(C1CC1)N(C)C(C1CC(=C2CC2)C1)=O C#CCCCCCC(=O)N1CCC2(NC(=O)CC(C)(O)C3CC3)CCCC12 Cn1ccc2sc(C(=O)NC3(C)CCCN(C(c4ccnn4C4CC4)=O)C3)cc12 c1(N(CC(N)=O)C)nc(=NC(CCO)C2CCC(F)(F)CC2)[nH]c2ccsc12 CCCC(C(C)CC)(c1nnnn1CC1CC1)NCc1cccc(OC)c1 c1(C(=O)NC23CC(NC(=O)C4=CCCS4)(C2)C3)ccc2c(c1)Cc1ccccc1-2 C1(O)(CC(=O)NCCCOCCC(=O)NC(C#CC)(C)C)CCOCC1 CCCC(CNC(c1cnc(C)cn1)=O)C(=O)N1CCC1CC(N1CCCC1)=O CC1CC(NC(C2(C)CC2)=O)CN1CCSc1cccc(N2CCCS2(=O)=O)c1 N1(C(CCOCCCOC)=O)CCC(CNC(C2CCOC2C2CC2)=O)C(O)C1 CC1=NCC(C)CCCC2CN(SC=NN1)CC(=O)OC(=O)N2 c1(C(C)NC(=O)C=CC(=O)N(C)C)ccc(NC2(CO)CCC(C)C2)cc1 Cc1ccn2cc(C(=O)NC3CC4CCC3N4C(C3C(C)(C)C3(C)C)=O)nc2c1 c1(OC)cc(=NC(=O)C(C2(O)CCC2)NC(=O)CC2(O)CCCCC2)[nH]n1C C1(C(N2CCC=C2C(=O)N2CCOCC2)=O)CCc2cnccc2N1 C1(NC(C(COC)(C)C)=O)CCC2(CC1)CC(NC(=O)CSC)C2 C1(C(=O)NCc2ccc(C)cc2)CN2CCN1CC2C.c1(OC)cccc(Cl)c1N CCC(C)(C)C(C(=O)N1CCC(NC(=O)C(C)(C)c2ccno2)CC1)OC c1(C(=O)NC2C(NC(=O)C=Cc3cn[nH]c3)CC2)cc2cc(F)ccc2o1 C1(CNC(C(CC)(F)F)=O)C2CCC1CN(C(c1cccc(OC)c1F)=O)C2 N1(CC(C)C)CCOC(CNc2cc(NCCC34CCCC3C4)ncn2)C1 N1(C(C(C)(C)OCC)=O)CC2C(C(=O)NCc3ccncc3)C2C1 c1(OC)cccc2[nH]c(C(=O)NC3CN(Cc4cnc(Cl)c(Cl)c4)CC3F)cc12 C(=O)(C1=CCCN(C(C2CCCCCC2)=O)C1)N1CCCC(CC(C)C)C1 c1(C(=O)O)cccc2c1CN(Cc1cn(COc3ccco3)nn1)C2 c1(C(N2CC(O)CC(NC(CCC(CC)CC)=O)C2)=O)cnc2n1CCCCC2 C(C)(CCC#N)(c1n(C(C)C)nnn1)NC(C)Cc1ccco1 C1(CC(=O)OCCNC(=O)NC2CCCCC2)CC2CCC1CC2 C(=O)(CCC(C)(C)F)NCC(CO)NC(c1nn(C)c(C(C)(C)C)c1)=O Cc1[nH]nc(CO)c1C(N1CCC(C(=O)NC(C)Cc2cn[nH]c2)C1)=O C(=O)(C1CSc2ccccc21)N1CC(C(N)=O)(CNC(CCC=CC)=O)C1 c1(OCC)ccc(C(C)NC(C2CNCCN2Cc2ncc(Cl)s2)=O)cc1 c1(C(C(=O)O)NC(C(c2cnn(C)c2)NC)=O)ccc(C)s1 C1(N(C(c2c(CCC)nco2)=O)C)CCCN(C(=O)COCC(F)(F)F)CC1 c1(CC)cc(N(C)Cc2ccnn2C2CC2)n(C)n1 O=C(CC(O)C(Cl)(Cl)Cl)NC1CCOCC1NC(c1cc(C2CC2)[nH]n1)=O C(C(=O)N1CCC(C(=O)N(C)C(C2CCOCC2)C)O1)(OC)SC C1(CC)CN(C(C2CC(O)C2)=O)CC1NC(C1CC=CCC1)=O C1(CNC(CSCCC)=O)CN(C(=O)CCn2ccc(C)n2)C2(CCC2)C1 c1(CC)onc(C)c1C(=O)NC1CCCC(NC(=O)CCCN2CCCCC2)C1 CCCCCC(C)(CC)C(=O)N=S1(=O)CCC2(CC1)CN(C(=O)C(C)C)CCO2 CC(C)C(C)CC(=O)N1CCC(OCC(=O)NC2CC3(CCC3)C2O)C1 C(=O)(CCC(C)(C)C)NC1C(n2cc(C(C(=O)OC)(C)C)nn2)CCC1 CC(C)CC(F)C(=O)N1CCN(C)C(CNC(=O)CNC(C2CCOCC2)=O)C1 c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(O)C2)cccn2nncc12 c1(C(C)C)c[nH]nc1C(=O)NC1CCC1NC(=O)CCC1CCCCC1 C1(C(=O)NCC(C)(C)NC(C2C(COC)(C(C)C)C2)=O)C(=O)ON=C1C c1(C(=O)OC)cc2c(nc1O)CCN(C(c1cnn(CCC(C)C)c1CO)=O)C2 N1(C(c2c(CCC)[nH]cc2)=O)CC2CCOCC2(NC(=O)C(=O)NCC)C1 c1(CN(C(=O)CN2CCC2C)CCOCC)cc(OC)c(OC)cc1Br C1(C(=O)NCC(C)(C)NC(=O)CC2CCCC(CC3CC3)O2)CCCCC1O C1(CC)(NC(C2C=CCCC2)=O)CCN(C(=O)C(O)COC)CC1 c1(C(=O)NCC2C(NC(c3cc(OC)cc(F)c3)=O)C2)cc2n(c(=O)c1)CCS2 O=C(C1=Cc2ccccc2C1O)NC1CC(CNC(C2(CO)CC2)=O)C1 C1(C(=O)NCC2N(C(CCNC(N)=O)=O)C3CCC2C3)CCCC2(CCC2)C1 N1(C(c2n[nH]c(C)c2O)=O)CCCN(C(=O)Cn2cccn2)CC1C(C)C c1(NS(CC)(=O)=O)ccc(SCCN(C)CCC2CC2)nc1 C=C(C)CN=C(NCC(F)(F)C1CCC1)N1CCN2C(=O)NCC2C1 N1(C(c2cc(C#N)cc(C)n2)=O)CC(C)CN(C(=O)CN2CCCCC2)C(C)C1 N1(C(C)CNC(=O)Cn2cc(Cl)c(C(F)(F)F)n2)CC(C)OC(C)C1 CC1CC=C(C(=O)NC(CCC2CC2)C(=O)N(CCCn2ccnc2)C)CC1 C=C=CC(C)C(=O)N1CCCC(CNC(=O)C(C)OCOC)C1 N1(C(c2c[nH]nc2Br)=O)CC2OCCN(C(c3cnn4c3OCC4)=O)C2C1 N1(C(C)=O)CCc2cc(C(=O)N(C)C)ccc21.C12CCCCN(C1)CCCN2 C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(NC(CC(c2ccc(F)c(F)c2)C)=O)CC1 c1(C(N2CC(NC(C)=O)C(C)C2)c2cccnc2)cc2ccccc2cc1N N1(C(CC(C)C)=O)CC2CC1(c1cn(CCC3(OCCON)CCC3)nn1)CO2 Cc1cc(C(=O)NCC(N2CCC(C)C(CN)C2)=O)ccc1Cl C(CN=C(NCC1CCC(C(N)=O)O1)N1CCN(C2CCCCCC2)CC1)SC CC1(C)CCN(C(c2c[nH]nc2-c2ccccc2)=O)CC1NC(=O)C=CCO C1(CNC(C(C)N(CC)CC)=O)CCN(C(=O)CCNC(C)=O)CC1(F)F N1(C(C2CC(N(C(=O)C=Cc3cc[nH]c3)C)C2)=O)CC(C)N(C)C(C)C1 C(=O)(C(O)CCNC(C1CC(O)C(F)C1)=O)NC1C(OC)C(O)C1 CC1OCCOC1C(=O)NC1CCC(F)(CNC(C2(C3CC3)CC2)=O)C1 CCC(C)C(=O)C(=O)NCc1csc(C(N2CCSCC2C)=O)c1 C1(NC(C2N(CC)CC2)=O)CCN(C(=O)C(COC)OC(C)=O)CC1O CCCCC(O)C(=O)NCC(C)(C)CN(C(=O)Cc1ncccc1C)CC c1(C(=O)NC(CNC(C2SCCS2)=O)CO)ncnc2ccsc12 N1(C(CCCCOC)=O)C2COCC1CC(NC(=O)CC1CCCCN1C)C2 c1(OC(C)C(=O)NC2CC(NC(=O)C(C)(F)F)C2)ccccc1N1CCOCC1 C1(C)(C(N(CCOCCC(=O)NC(C=C)C2CCC2)C)=O)CC2C=CC1C2 CCC(CC(=O)N1CCCC1CN(C)C(C1CCCC(C)C1)=O)C1CCC1 C(CC(C)C)(C(=O)OC)C(C(=O)NCCOC)N(CCC(=O)OCC)C C1(NC(C(=O)NC(COC)C)=O)CCCN(c2ccccc2Cl)C1 C=CCCC(C(=O)N1CC(N(C)C)C(O)C1)NC(C1CC2(CC2)C1)=O C(c1ccc(F)c2ccccc12)=CC(=O)Nc1c[nH]nc1Cl CC(C(=O)N(C1CC1)CC1CCCN1C(=O)CC12COC(CF)(C1)C2)C(C)(F)F CC1CCC(NC(=O)CS(=O)(=O)NC(C)(C)C)CN1C(=O)C1=CCCS1 c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)conc1-c1ccccc1 C(=O)(CC(F)(F)C(F)(F)Br)NCC(C)N(C(=O)Cc1cocn1)C N1(C(c2cnn(CC)c2)C(=O)NCCC(=O)OCC)CC(CO)OC(C)(C)C1 c1(C(=O)NC2CC(F)(CNC(c3scc(OC)c3)=O)C2)c(CO)noc1C c1(C(=O)NCCN2CCC(C(=O)NCc3c(C)scc3)CC2)c(F)cccc1F c1(Cc2c(C(=O)NCc3cn(C(C)C)nn3)cccc2)ccc(Cl)c(Br)c1 c1(C(C(=O)NCCC)N(C)Cc2ccoc2)nc2ccc(Br)cc2s1 N1(C(C(CC)COC)=O)CCC(NC(=O)CCc2cccs2)C(F)(F)CC1 C(c1ccncn1)=CC(=O)NCC1CC(NC(C2(c3cccs3)CCCC2)=O)C1 c1(OC)ccc(F)cc1CC(=O)NCC(C1CCCC1)NC(=O)CSC1CC1 N1(C(C=CCC)=O)CCCC2CN(C(C3Cc4ccc(C)cc4C3)=O)CC12 c1(-c2onc(C(C34CCCC3C4(F)F)C)n2)cc(F)ccc1OC(F)F C(=O)(C(C)CC(C)(C)C)N1CCC(NC(c2c(C)nc(C3CCC3)o2)=O)C1C c1(CC(=O)NCC2C(NC(C=CC=CCC)=O)C2)cccc(C(C)C)c1 c1(CC)c[nH]nc1C(N1CC=CC1C(=O)NCCOCC1CCC1)=O C1(CNC(c2cn(C3CCOC3)cn2)=O)CCCCCN1C(=O)Cc1cnns1 CC(C)(C(=O)O)C(C1CC1)NS(=O)(=O)CCCOC C1(CNC(CCOCC)=O)CC2CCC1N(C(c1ccc(=O)n(C)n1)=O)C2 N1(Cc2c(CC)noc2C)CC2CCN(C(c3cccc(F)c3)=O)C2C1 c1(CC)ccc(C(=O)NCCC2CCCN(C(C3(C)COC3)=O)C2)cc1N c1(CNC(=O)NC(c2cnn(C)c2)C(=O)OCC)nsc2ccccc12 C1(NC(C(C)C(C)(F)F)=O)CC1C1CCN(C(=O)CC(C)(C)O)CC1 c1(C(=O)NCCN(C(=O)CCOc2cccnc2)CCOC)cc(Cl)nnc1O N1(C(CN(CCC#C)C)=O)CCCC2(CCCN2C(=O)C#CC2CCCCO2)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CCN(C(c3ccno3)=O)CC2C1 C1(CN(C)C)CCCN(C(=O)Nc2c(C)cnn2-c2ccc(C)cc2)C1 N1(C(C(N2CCSCC2)C)=O)CCC2C(NC(C3(Cl)CC3(F)F)=O)C2C1 c1(COC)ncc(C(N2CC3C(CN(C(=O)C(C)(C)SC)C)C3C2)=O)c(O)n1 c1(NCCC(=O)NC(C)C)[nH]c(=NCC2CC3(C2)CC32CCC2)nc2scnc12 c1(C(=O)NCC2N(C(CC(CCC)C)=O)CC2)cc(Cl)c(C)c(Br)c1 N1(C(CC(OCC)OCC)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C1(NC(=O)NCc2cccc(OC(C)(C)C)c2)C2CC3COC1C3C2 C1(C(=O)NC2C3CC2N(C(=O)COCC2CCOC2)C3)CC1C1CCOCC1 CC1COC(C)(C)CN1C(=O)C(Cc1ccco1)NC(=O)Cn1[nH]cnc1=N C(C(Cc1ccccc1)C(F)(F)F)NC(N1CCCC(NCCO)C1)=O N1(C(c2cnc(SC)c(C)c2)=O)CCC2(CCC(CNC34CC(CC)(C3)C4)C2)C1 Cc1ccc2c(c1)CC(C(=O)NCCCNC(c1cccc(P(C)(C)=O)n1)=O)O2 C1(CN(C(=O)CC(C)(C2CCC2)N(C)C)CC)CCCN(C(C2OCCO2)=O)C1 C1(CC(=O)NC)CN(C(=O)Cn2cccn2)CCN1C(c1cocn1)=O N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)CC2NC(C1(CO)CCCCC1)=O C(=O)(C(O)CC(F)(F)F)NCCCNC(=O)COc1ccc(F)c(Cl)c1 N1(C(C2NC(=O)C(F)C2)=O)CC2CCCC(C1)N2C(=O)COc1cccc(Cl)c1 Cc1c(C(N2CCC(CCNC(C34CCCC3C4)=O)C2)=O)cnn1C(C)(C)C Cc1cc(O)nnc1C(=O)NC1CN(C(c2cc(Cl)ncc2O)=O)CCC1CO c1(C(=O)NC2SCCN(S(CCC)(=O)=O)C2)ccc(OC)cc1C C1(CNC(C2CC3CCN(c4noc(C5CC5)n4)CC23)=O)CCn2cncc2C1 N1(C(C(C)Cc2ccccc2)=O)CCC(NC(c2scnc2C2CC2)=O)CC1C C#CC1CCN(C(C2COCCN(C(=O)Cc3cnoc3)C2)=O)CC1 N1(C(C2(F)CC2)=O)CC2(CCNC(C3(c4ccno4)CC3)=O)CCC1CC2 C1(NC(COCCOCCOC)=O)CN(C(c2c(O)cccc2Cl)=O)CC(C)(C)C1 N1(C(CNc2scc(C)n2)=O)CC(CNC(=O)CC2CC=CC2)OC2COCC12 c1(OC)c(C(N2CCC(NC(c3ccoc3C3CC3)=O)C2C)=O)ccc(Cl)c1C C1(NC(C(C)(O)C2CC2)=O)CCC(F)(CNC(=O)CCCc2ccccc2Cl)C1 CON1CCC(CC(=O)NCC2CC2CNC(=O)C=Cc2ccccc2C)CC1 N1(C(c2c(N(C)C)cccn2)=O)CC2CC(NC(c3sccc3F)=O)C1C2 CCCCCC(O)C(C)C(=O)NC1CCC1NC(C1Cc2ccccc2O1)=O C1(C(=O)NC2(CO)CN(C(C3(CCCC)CC3)=O)C2)COC2(CO)CC1C2 CCC(C)(CNC(C1CCCC1)=O)NC(C1C=CCCC1)=O c1(NCC2C(NC(C(C)C)=O)CC2)ccc(C(=O)NC(C)(C)C)s1 C1(CNC(C2(CC#C)CC2)=O)CC(NC(=O)Cc2c(C)cnn2C)C1(C)C CC12CCC(C(=O)NC3CN(C(=O)CCS(C)(=O)=O)CC3F)(CC1)OC2 c1(CC(=O)NC(CC=C)CNC(C2CC23CCC3)=O)ccnc(C(F)(F)F)c1 CC(O)(C(=O)N1CCN(C(C2CN3CCC2CC3)=O)C(C2CC2)C1)C(F)(F)F c1(NCCCN(C)C2CC2)ccccc1NC(c1ccccc1)=O C=C=CCC(=O)NCCCOCCNC(=O)CCCc1ccccn1 O=C1CCCC(CC(N2CC=CC(NC(=O)CCCc3cc[nH]n3)C2)=O)C1 C1(C(=O)NCC2(SC)CC2)CCC(O)CN1C(C1CC=CC1)=O C(=O)(CCCCC(F)F)N1CC(CNC(C2CC(C)(C)C2)=O)C(C)(C)C1 C#CCC(C)(C(=O)NCCCC1C=NNC1=O)NC(=O)C(COC)COC CC(C)CCCCCC(=O)NCCCCNC(=O)CC1C=CCCC1 C(=O)(C#CC1CCCO1)N(C(C)CN(C)C(c1cnc(C2CC2)s1)=O)C CCCCC(C)C(=O)NC(C)CCN(C)C(c1cnn(CCO)c1C(C)C)=O C1(C)(C(=O)NCCCN(C)C2CC2)CCN(C(C2CC2C2CCCC2)=O)CC1 C(=O)(C(F)C(F)(F)F)NC(CCCCNC(C1(C(=O)OC)CC1C)=O)C CC1CCC(CO)CN1C(=O)COC1CC(NC(=O)C=Cc2ccco2)C1 C1(C(=O)NCc2nc(C)c(C)o2)(C(=O)OC(C)(C)C)CCC2CCCC12 N1(C(C)=O)CCCC(O)(CNC(=O)C(Cc2cnc[nH]2)CNC(C)=O)C1 CCC(CNC(=O)C(C)C#N)(CC)NC(c1cc(C2(C)CC2)n[nH]1)=O N1(C(C(C)=C2CCCC2)=O)CCC(O)(C(C)NC(=O)CCC2CCC(O)CC2)C1 c1(C(N2CC3C(NC(c4ccc(CC)o4)=O)(C3)C2)=O)ccc2ccncc2c1 C1(C(=O)NCC2CCC(CNC(CNS(C)(=O)=O)=O)CC2)CCCCNC1=O c1(NCC2C(C(N3CCC(SC)C3)=O)C2)ccc(O)c(C)c1 C1(NC(c2cc(CCC)oc2C)=O)CCN(C(c2sc(OC)nc2C)=O)CC1F C=CCCCC(=O)NCC1CN(C(c2ccc(CC)cn2)=O)C2CC12 C1(CC(N2CC(F)(C3CC3)C2)=O)CC2(C1)CN(C(c1cncc(O)c1)=O)C2 C#CCCCCC(=O)N1CC(NC(=O)CSc2nnnn2C)C2CC12 C(=O)(C1=NNC(C(F)(F)F)C1)N1C(CCSCC(=O)NCC2CC2)CCC1 c1(C(=O)OC)ccccc1OCC(C)CNCC(=O)O.C12CCCN1C2 C1(CNC(C23OCC(CC)(C2)C3)=O)C2CCCC1N(C(=O)CCc1ccc[nH]1)C2 C12(NCC=C(C)C)CCC(CC1n1cc(COc3c(C)ccnc3Br)nn1)C2 N1(C(CC(CC)(F)F)=O)CCN(C(c2cnn(-c3ccccn3)c2)=O)CCC1C n1(CC)nnc(C(N2CCC(C3(C)N=N3)C2)=O)c1C Cc1oc(CNC(c2cc(C3CC3)on2)=O)nc1C(=O)N(C1CN(C)C1)C C#CC1CN(C(C2CCN(C(=O)Cn3cnnn3)CC2O)=O)CCN1C c1(C(N(C(CCNC(CCOCCCCC)=O)C)C)=O)ncoc1CC N1(C(c2ccc(CNC(C(CC=CC)C)=O)s2)=O)CC2C=CCC(C2)C1 Cc1cc(C(=O)NC2CN(C(=O)Cn3cccn3)CCC2C)nc(O)n1 c1(CCCCCC)cccc(N=c2[nH]c3cccc(OC)c3n2C)c1 c1(C(=O)NC(C(C)C)(C)CNC(C2(CCO)CC2)=O)ncc(F)cc1F C(=O)(CC(C)CC(C)(C)C)N1C(C)C(C(=O)NC2CCC3(CCCC3)C2)CCC1 c1(C(N(CCC)CCNC(=O)CCn2cccn2)=O)csc(C(C)(C)C)c1 C1(N(C(c2c(C)n(CCO)nc2)=O)C)CN(C(c2cc(Cl)ccn2)=O)CC1(C)C C1(OC)CC2CCC(C1)N2C(C1(N(C(=O)CC2CCCOC2)C)CC1)=O c1(C(=O)NC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ncc2ccccc2c1O C1(C(=O)NC2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)CN(S(N)(=O)=O)C1 Cc1ccc(C)c(-c2nc(C3CC34CC4)nn2CCN(c2ccccc2)C)c1 Cn1nc2c(c1C(N1CCN3CCCC3C1)=O)CN(Cc1cscn1)CC2 C(=O)(C(CO)C(C)(C)C)NC1(CNC(c2c(C)nc(CCC)o2)=O)CCC1 C1(C(N(CC(C)OC)C)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1O C1(NC(C(C)(C)Cc2ccccc2)=O)C2CCN(C(=O)CC3CC3)CCC12 c1(C(N(CC(C)NC(=O)C(C)(Cl)Cl)CC)=O)oc2c(OC)cccc2c1C N1(C(C(C)OC(C)(C)C)=O)CC(C(C)(C)O)(CNC(C2CCCCS2)=O)C1 c1(NC(CC2OCCN(S(CCCC)(=O)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1C C=CCC(C(=O)NCCCCC(C)NC(=O)C(c1ccccc1OC)O)C(C)C c1(C(N2C(CC(=O)NCC3CCC(CO)C3)COCC2)=O)cccc2c1CCN2 CC(F)(F)C(C)(C)C(=O)N1CC(CN2CCN(C(=O)CCC(F)(F)F)CC2)C1 c1(C(=O)NCCCC2N(C(C(CC)N(C)C)=O)CCC2)noc2c1CCCC2 c1(N2CC(NC(c3cccc(CO)c3)=O)C(O)C2)ncnc2cc(Br)sc12 N1(C(COCC(=O)OC)=O)CC(CNC(C2(C)CCNC(=O)C2)=O)C2(CC2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC2CNC(=O)C=C(C)c1ccccc1C N1(C(CC2C(C)=NNC2=O)=O)CCC2(CC2C(=O)NCCCc2ccco2)C1 C(C(=O)N=c1ccc(C)c(Cl)[nH]1)Cc1c(C(=O)OC)nn2ccccc21 N1(C(CCCn2ncc(C)c2)=O)CC(F)CC1CN(C(=O)C(O)CC1CCCC1)C C(=O)C(O)CC(C)C.N1CC(C2C(c3cn(C4C(SC)CCC4)nn3)C2)C(F)C1 c1(-c2cn(CC3CN(C(C4(C=C)CCOCC4)=O)C3)nn2)cc(Cl)cc(Cl)c1Cl c1(C(=O)NCCC2CCCN2C(c2sc(F)cc2Cl)=O)ccc2cccnc2n1 c1(C(N)=O)ccc2c(c1)CCC2NC(=O)N(CCO)CC1CC2CC1C2 C12(NC(c3nnc(C)o3)=O)CCC(CC1)N(C(=O)CCOC1COC1)C2 c1(OC)cccc(C(c2ccccc2)NC(=O)NC2CC(C#N)C2)c1 c1(C(N2CCC(NC(CC3(N(C)C)COC3)=O)C2)=O)ccc(O)nc1Cl N1(C(c2cc(C)c(CO)cn2)=O)CC2(CCCCN(C(C3CCCC3)=O)C2)C1 Cc1cccc(Cl)c1CC(=O)NC1C=CCN(C(=O)C=CCN(C)C)C1 c1(CNC(C2CCC(C)C(C)C2)=O)nc2c(s1)CN(C(=O)CC1(CO)CC1)CC2 N(C)(S(=O)(=O)N1CCNC(C2CCC2)C1)CCN(C)C C1(Cc2onc(CCCS(C)(=O)=O)n2)CC2C=CC1CC2 C1(OC)CC(CNC(C2CCC(F)CC2)=O)N(C(c2n[nH]c(C)c2Cl)=O)C1 c1(CN2CC(CC)N(CC(F)F)CC2)cc(OC)c(OC)c(Cl)c1 N1(C(=O)Nc2c(C(=O)OC)ncs2)Cc2c[nH]nc2C(C)C1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCCN2C(=O)C(=O)N=S(C)(C)=O)CC1 c1(C(=O)NCC2C(CNC(CCOCCCOC)=O)C2(F)F)c(C)n[nH]c1C c1(CCC(=O)NCCNc2ccc(C(N)=O)s2)ccc(O)nn1 Cc1c(C(=O)N(C)CC2CCN(C(C3CC3C3CCC3)=O)CC2)cncc1Br C#Cc1ccc(C(=O)NC2C3CC4C2C4C3C(=O)NC(c2nccs2)C)cc1 c1(CC(C)C(=O)NCC2CC3CC3N2C(=O)CS(C)(=O)=O)ccc(O)c(O)c1 N1(C(c2cn(C3CC3)cn2)=O)CC2(C(N3CCC3CO)=O)CC1CCO2 C1(OC)CC(NC(=O)CCC(C)SC)CN(C(c2ccc(CO)cn2)=O)C1 N=c1ccn(CC(=O)Nc2nc(N3CCNC3=O)no2)[nH]1 N1(C(C2(COC)CC2)=O)CCC2CN(C(c3ccc(Cl)nc3)=O)CCC12 C(=O)(C(F)C(C)CC(C)(C)C)NC(CNC(C(C)SC)=O)C1CCC1 c1(CSC)ccccc1NC(C)(CCn1cccn1)c1nnnn1C(C)C CC1(C)CC2(CC(NC(=O)C(CC3CCOCC3)NC(c3ccsc3Cl)=O)C2)C1 N1(C(CC(=O)N(C)C)=O)CC2COCC2(C(=O)NC2CN(C(C)=O)CC2(C)C)C1 Nc1c(C(N2CCC(C(F)C(=O)NC3CC=CC3)C2)=O)cccc1F C1(C(N(C(C)C)CCN(c2nc(Cl)c(C#N)s2)C)=O)CS(=O)(=O)CC(=O)N1 c1(C(=O)NCCC2(C(=O)NC3CCC(C(C)O)CC3)CC2)cc(O)ccc1F Cc1nc(O)c(C(=O)NC2CCCCCN(C(=O)CC3C=CCC3)C2)nc1C c1(CC)c(C(=O)NC2CCN(C(=O)C(O)CCSC)CC2)csc1C N1(C(CCC#C)=O)C(C(=O)Nc2cccc(CCC)c2)CCC12CC2 Cc1nc(C(=O)NCC(C)(C)NC(=O)CC(C)C(F)F)ccc1C#N C12(CCOCC1)C(=O)NCCO2.c1(C(=O)CNCC2(CC=C)CC2)cn(C)nn1 C1(C(C)NC(C2(C(F)(F)F)CC2)=O)CCN(C(=O)CNC(=O)C2CC2)CC1 c1(OCCN(CC)CC)cccc(SCCc2ccccc2F)c1.C(C#N)O Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CN(C(c2cc[nH]n2)=O)CCC1C C1(C)CCC(=O)N1.C1CCC(CNC(=O)CN(C)C(C)=O)CC1.CCCCC1CC1 c1(C(=O)NCCOCc2cn(-c3nccc(C)n3)nn2)cc2n(c1)CCC2 CCC(C)CCC(O)CC(=O)NCC(C)(C)OCCNC(=O)CNC=O CC(C)C(C(=O)N(CCc1cccnc1)CC1CCCC1)Sc1ccccc1 C1(OC)CN(Cc2cscc2Br)C2(CCC2)C1 c1(C(=O)NCC2C(CNC(CCCCCC=C)=O)C2)oc(P(C)(C)=O)cc1C c1(C(=O)NC(C(=O)NCCC(CCC)O)CCOC)cc(C#N)ccc1N c1(SCC)nccnc1C(=O)NC1CC1CNC(c1ncn(C(C)(C)C)n1)=O Cc1ccc(C=CC(=O)NC(C)CCNC(=O)CC(C)(C)O)cc1Cl c1(C(=O)NC2CCC(N(C(=O)CC3(C#N)CCC3)C)C2)ccc(F)c(F)c1 C(=O)(C(O)CCOC)N1C(C(=O)NCC2(OCC)CN(C)C2)CC2CC21 Cc1cc(C(N2CC(N(C)C(C3CC(=O)C34CCC4)=O)C(C)(C)C2)=O)cnc1C c1(CCN=C(NC(C=C)C)NCc2ccsn2)c[nH]c2cc(F)c(F)cc12 N(C(=NCC1CCOC1)N1CCC(O)C1)CC1C(C)(C)CCCC1(C)C C(=O)(CC(C)C(=O)NCC1CN(C(C2(OC)CCSC2)=O)CC12CC2)OCC C1(C(N(C2CN(C(c3c[nH]c(=N)s3)=O)CC2(C)C)C)=O)CCCCCS1(=O)=O C=CC(C)(C)CC(=O)NCc1csc(CNC(=O)CCCOCCC)n1 N1(C(c2cc(COC)[nH]n2)=O)CC2(CCCC(CNC(=O)C(C)(C)CSC)O2)C1 N1(C(c2sccc2OC(F)F)=O)CCC2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(C(c2cc(OC)c(O)cc2F)O)=O)CC2CCCCCCC2C1 N(C1CCC(NC(=O)C2CC2)c2ccccc21)C(c1onc(CC)c1C)=O c1(CC(C)OC(CNC(=O)OC)=O)ccc2c(c1)CCC2 C1(C)(CC)C=C(C(=O)NCC2(O)CCN(C(=O)Cc3csc(C(C)C)n3)CC2)C1 C12(C(=O)NCC(C(N3CCC4CC34C)=O)OC)CC(C#N)(C1)C2 N1(C(CCCCOCC)=O)CCc2c(ccnc2C(=O)O)C1 c1(OC)ncc(NC(c2cc(F)cc(F)c2)C)cc1Br N1(C(c2ccccc2)C(=O)OC)CN(Cc2ccccc2)CC1CO C1(CC(C)(C)C)CN(C(c2cnns2)=O)CCN1C(c1ccc(C#N)s1)=O c1(CC(N2CCN(C(c3c(SC)nccn3)=O)CC2)=O)ccc(C)c(Cl)c1 C1(C(=O)NC2CCCN(CC)C2)CN(C(=O)C(O)C(F)(F)F)CC1(F)F N1(C(C(n2cnc(C#N)n2)C)=O)CCC2(CC1)CC(NC(=O)C(C)CO)CCO2 c1(NCCn2c(C(C)C)nnc2)ccc(S(=O)(=O)NCCCN2CCCC2)cn1 C(=O)(C(C)(C)C(C)(C)C)NC(CC1CN(C(C2(C)ON=C(C)C2)=O)C1)C C#Cc1ccc(CC(N2CCCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)cc1 c1(N2CCC(C=C)(COC)C2)cc(Cl)c(Br)cc1C c1(CC)ccc(C(N2CC(OCCNC(=O)C(CC)OC)C2)=O)c(Cl)c1 C(=O)(CCC1=NNC(=O)CC1)N1C(C)CCN(C(=O)C(F)CC2CCC2)CC1 C(CC(=O)NC(C)(C)CC(C)(C)C)(C(F)(F)F)NC(C1C(=C)C1)=O CC(CC(C)(C)C)C(=O)N1CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 c1(N2CC=C(C)CC2)nc(=NCc2cc(C)cc(Cl)n2)[nH]c2c(F)cc(F)cc12 CCC(C)CCC(=O)N1CC(C(=O)NCc2cnn(CCF)c2)CCC1C CN1CC=C(C(=O)NCC(C)(O)CNC(=O)C(C(C)(C)C)C(=O)NC2CC2)C1 C1(NC(c2cc(CC(C)C)on2)=O)COC2CN(C(=O)CS(N)(=O)=O)CC12 N1(C(c2cn(C3CCCC3)nn2)C(=O)NCCCF)CCCCC12CC2 c1(SC)nc2ncnc(NC3CCCN(C(=O)CNC(C)=O)C3)c2s1 C(=O)(C1CCCc2nc[nH]c21)N1CC2C(N(C(C=CCN(CC)CC)=O)C)C2C1 c1(C(N(CC(C)(C)NC(C=CC(=O)OCCCC)=O)C)=O)cnncc1O N1(C(C(C)=C(CC)C)=O)CC2CCCN(C(c3ncnc4c3CCC4)=O)C2C1 N1(C(Cc2c(C)non2)=O)CCCC(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C(=O)(CS(=O)(=O)CCOC)NC1C(CC)CN(C(=O)C(C)OCCOCCO)C1 C1(CC(=O)NC(C2CN(C)CCO2)C)CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 c1(-c2c(C)c[nH]n2)nc(=NC(=O)NCCSCCc2ccsc2)s[nH]1 N1(C(C2(CCCC)CC2)=O)CCC(C)(C)C(NC(=O)CCCCC(=O)NC)C1 Cc1cc2[nH]c(C(=O)NC3CC3CNC(=O)CC=Cc3cccc(F)c3)cc2o1 Cn1ccc(C(=O)NC2CCCC2(C)NC(C2CC2c2ccco2)=O)cc1=O C1(NC(C(C(C)C)N(C)C)=O)CN(C(=O)CC(C)P(C)(C)=O)C2(CCCCC2)C1 c1(CN(CC(C)NC(C(C)OCCC=C)=O)C)ccc2c(c1)CC(C)O2 c1(C(=O)NCC2CCC(C(NOCC#C)=O)O2)csc(C)c1C c1(OC)ccc(Cl)c(C(c2nnnn2C2CC2)NC(C)CC2CCOCC2)c1Cl c1(-c2n(-c3cn(C)nc3)nc(CCC3CCCN3C)n2)cc(C2CC2)nnc1O C1(CNc2c(C)c(N3CCC=C(Br)C3)ncn2)CCCC2(CNC2)O1 N1(C(CN(C(=O)CCc2ccn(C)c2)CC#C)=O)CCCC(O)(CO)C1 C1(C(=O)NCC(CC=C)NC(=O)C=CC)CC2CC(=O)C1O2 C12(C(N(CC(COC)O)C)=O)CCCC1N(C(=O)CC1CC(C)C1)CC2 C1(CC=C)(NC(=O)CCC2CC2CC2CC2)CCN(C(C2COC(=O)N2C)=O)CC1 N1(C(CCC(=O)NCC)=O)CCC2CCCC12CNC(c1nccnc1CC)=O C1(CC(=O)N(C2CCCC2)CCCC)CC(O)CN1C(=O)CC1CCCC(=O)C1 C(C(CC(=O)N(C1(C(N)=O)CC1)C)OC)NC(C1(CCC)CCC1)=O c1(N2C(CCCN(C(Cc3c(C)cccc3)=O)C(C)C)CCC2)cc(C#N)ccn1 c1(OC)cc(C(=O)NC2(CF)CCN(C(=O)C(C)(C)C3(O)CCOC3)C2)n(C)n1 C1(NC(CC(c2cccc(OC)c2)C)=O)CCCCN(C(=O)C(O)C(C)(C)C)C1 C1(C(=O)NC(CC)CNC(c2cc(C)c(SC)o2)=O)COCC2(CCC2)O1 c1(C(=O)NC(CC=CC)C(=O)N(C)Cc2cnccn2)nccc(C)c1N N1(C(c2c(C(C)C)ccc(O)c2)=O)CC2OCC(NC(=O)C=CC3CCC3)C2C1 c1(C(n2cc(C3(NC(=O)C(C)CC#N)CCC3)nn2)(CC)C)ccc(Br)cc1 n1(CC)cc(C(=O)NC2(CCNC(=O)CCC3CCCN3C)CC2)c(C)n1 c1(N)nc(C(F)(F)F)ccc1C.C1(CC=C(C)C)CCC(SC)O1 C(=O)(CCCC(=O)NC(C)CC(=O)N1CCC(CF)C1)OCC C(CC(C(=O)NC(c1ncc(C)cn1)C)NC(c1sc(O)nc1C)=O)OC c1(CN2CCC(CC(=O)NC(C(C)O)CO)C2)c(F)cc(Cl)cc1Br C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(=O)C=CC(F)(F)F)CCOC1 c1(N2CC(NC(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)nc(C2CC2)nc2c1CCC2 C1(F)(CNC(CCSCC)=O)CCCN(C(c2cc(O)ccc2Cl)=O)C1 c1(C(=O)NC(C)(CNC(=O)Cc2cccc(O)c2)CO)coc2c1COC2 N1(C(c2cc(C(C)=O)on2)=O)CC(N(C(=O)C(c2cccnc2)C)C)C2(CC2)C1 c1(CC)ccc(F)c(C(N2CCCCC(NC(=O)C(N)=O)CC2)=O)c1F c1(NC(C2C(C(=O)NCc3ncn(C)c3)C2)=O)cc(F)c(Cl)cc1Cl C1(CNC(C2CCOCC2)=O)CC2(CCN(C(c3c(F)cccc3F)=O)C2)CO1 c1(C(=O)NC2(C3CN(C(c4cc(C)sc4)=O)C3)CC2)cc(F)cc2nn(C)cc12 O=S(=O)(c1cnc(NC2COCCC2O)c(Cl)c1)NCc1cc(F)ccc1F C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCOCC1NC(C1CCOCC1)=O C(=O)(C1=CCCOCC1)N1CCCN(C(c2c(C#N)ccs2)=O)CC1 C1(CCNC(C(C)n2cncn2)=O)CCCCN1C(c1n[nH]cc1C(F)(F)F)=O c1(C(=O)OCC)nnc(SC)nc1N1CC2CC2(C(=O)NCCSC)C1 O=C1CC(C(=O)NCC23CCC2CN(C(=O)CN2CCCC2)C3)=NN1 N1(CC(=O)NCC(C2CCCC2)C)CCN(C(=O)CCc2nncs2)CC1 c1(C(N2C(C(=O)Nc3ccc(Br)nc3I)C(O)CC2)=O)ccc2occc2c1 C(CC#CC(C)(C)C)NC(CCC(C)NC(=O)CC1CC(=O)NC1=O)=O C1(C(N2CC(C)(CC)C2)=O)N(C(=O)C(C)N2CCCC2)CC12CCCC2 C1(NC(C(=Cc2ccco2)C)=O)C2CC(O)C1N(C(c1cnnc(O)c1)=O)C2 CC1CCC(O)(CNC(C23CC(CN(C(=O)CC4CC5CCC4O5)C2)C3)=O)CC1 C1(C(N2CC(C)(N(C)C)C2)=O)CC2CC1CN(C(C1CCC(C)(O)CC1)=O)C2 CC(C)(C)CCC(=O)N1CCC(CC(=O)NC2(c3ccncc3)CC2)C1 N1(CC)CCC(NC(=O)C=CC(C)(C)SC)CC1.c12sccc1CNC2=O c1(C(=O)NCCC2(CNC(C3CC4CC3CO4)=O)CC2)ccc([N+](=O)[O-])cn1 C1(C)(C(=O)NCCCC2N(C(c3cc(OC)n(C)n3)=O)CCC2)CCCC1(F)F n1(C(C)C)cc(C(=O)NC2CN(C(=O)C(CO)N(C)C)CC23CC3)c(O)nc1=O C#CCC(C)(C(=O)Nc1cncc(F)c1)NC(=O)CC(C)C(F)F CC1(C)C2CCC1(C(=O)NCC1CC1CNC(=O)CCSc1ccccn1)CC2 C1(CNC(c2nc(OCC)oc2)=O)CC(C)N(C(c2cnn(CC)n2)=O)C1 c1(C(=O)NCC2CC2CNC(C23C=CC(CC2)C3)=O)cccc2nncn12 N#Cc1nccc(N2CCC(O)C2c2ccccc2OC(F)(F)F)n1.C1(=O)CO1 c1(C(N2C3(CN(C(c4cncc(C(=O)OC)c4)=O)C3)CC2)=O)cc2sc(C)nc2[nH]1 Cn1cc(C(N2CCC(CO)(NC(=O)CC3(C#N)CCC3)C2)=O)c2ccccc12 N1(C(C2(SC)CC2)=O)CC2CCN(C(c3cn(C)nc3C)=O)CC2C1 [N-]=[N+]=NCC(F)CCNC(C1(NC(=O)CC2CCCC2O)CC1)=O C(=O)(CCCCC(F)(F)F)N(C1CCCN(C(C2N(C(=O)OC)CCC2)=O)C1)C C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(C2)CC(O)C3)=O)C2(CCC2)C1 CC(C)CC(C(=O)NCC(O)C(C)O)ONC(C1CCC2(CCC2)O1)=O c1(SCC2C(C(=O)OC)C2)nn(CC(C)SC2CCOCC2)c(=O)o1 C1(C(N2CCC(NC(C=CCC)=O)(CF)C2)=O)Cn2c(C)nnc2CN1C c1(SC)cc(F)ccc1C(=O)NC(CO)C(C)NC(=O)Cn1ccc(C(F)F)n1 C1(C(N(C2CC(=C)C2)C)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 C1(C(=O)NCCCN(C(C2(CC3CC3)CCOC2)=O)CC)CC(OC)C(OC)C1 N1(C(C(C)OC)=O)Cc2[nH]nc(C(=O)NCCN3CC(C)(O)C3)c2C1 N1(C(CC=CC)=O)CCC(C)(CNC(C2C=CCS2)=O)C1 N1(C(CC2C(C)CCCC2)=O)CC(C)C(N=c2ccc(C#N)c[nH]2)C(C)C1 N1(C(c2c(C)nsc2)=O)CCCC(CNC(C2CC3CCC2C3)=O)C1 c1(C(N2CC(CC)C(NC(=O)C(=O)NCC(F)F)CC2)=O)c([N+](=O)[O-])cnn1C CP(C)(=O)c1cnc(C(=O)NCC2CCC2NC(C2COCCC2(F)F)=O)nc1 N1(C(CC(=O)NCC)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 Nc1ccc(O)cc1C(=O)NC1(CNC(c2ccc(C(F)F)o2)=O)CCOCC1 N1(C(=O)OC(C)(C)C)CC2CC(F)C1C2C(=O)NCc1ccco1 C1(C(N(C)CC2N(C(C=CC(CC)=CC)=O)CC(F)C2)=O)CC2CCC(C1)C2O C(C(O)CC(=O)NCC1=NOC(C)C1)NC(c1cn(CC=C)nn1)=O c12cc(c(Br)cn1)C(=O)N2.N1(CC)CCCCC1C#N.c12cncc(c1)C(=O)N2 N1(C(C(CCSC)OC)=O)CCC2(CCCN(C(c3ccc(CO)o3)=O)C2)CC1 Cc1cc(CCNC(=O)C(=O)NCC(c2ccsc2)N2CCCC2)c(C)s1 n1(CC)nc(C(=O)NCc2cnn(C)c2C(=O)NOCC(N)=O)c(C)n1 N1(c2ncc(C)s2)CCC2(CC1)CCN(C(=O)COc1ccc(Cl)cc1)CC2 S(=O)(=O)(c1ccc2c(c1)COC2)NCC(=O)NC1C(NC(COC(C)C)=O)CC1 S(=O)(=O)(c1ccc(F)cc1Br)NC(C(c1cc[nH]c(=N)c1)(C)C)=O c1(NC(C2CCN(C(CC3CC(=C)C3)=O)C2)=O)cccc(N=[N+]=[N-])c1 C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(c1nnc(C)s1)=O N#Cc1cccc(NC(C2(NC3(c4ccccc4)CCC3)CCCC2)=O)c1 C(C(F)(C(=O)N(c1ccsc1)C)C(C)C)NC(C(C1CC1)OC)=O C12CCCN(C1)C(=O)CO2.C1(COC)CCN(C(=O)COC2CC2)C1 C1(NC(C(C2CC2)OCC)=O)CC2CCC(C1C)N2C(=O)C(CC)CCOC N1(C(c2n(CC#C)ccc2)=O)CC2CC2(C(=O)NC(C)CCC2CC2)C1 CCCC(O)(CN(CC(=O)Nc1cccc(CNC(C)C)c1)C)C(F)(F)F C1(NC(=O)CC2COCCO2)CN(Cc2ccc(F)nc2F)CCC1(F)F c1(C(N2C(CNC(C(c3ccc(Cl)cc3)CC)=O)CCC2)=O)cccc(F)c1N C(N=c1[nH]c(Cl)ncc1Cl)C1C(C)CCCN1C(C1CC2(CSC2)C1)=O c1(C(N2C(CCNC(c3c(C)nsc3C)=O)CCCC2)=O)ccc(N)c(F)c1 N(C1CCC(NC(c2cscn2)=O)c2ccccc21)C(=O)C1=CCOC1 CC1CC(NC(=O)Cn2cccn2)CCN1C(=O)CCc1cc(F)ccc1F c1(CC(=O)NCC(C)(CNC(C2(C)CCCC2O)=O)OC)ccc(C(N)=O)nc1 n1(CC(=O)NCC(CNC(C(C)(F)c2ccccc2)=O)F)nc(O)ccc1=O Cc1cc(C(=O)N(CC(C)(C)CNC(=O)CCN2CCCC2)C)cc(C)c1O c1(C(=O)NCC2(CCNC(c3ncc(CC)s3)=O)CC2)cn2c(n1)CC(C)CC2 N1(C(C2OCCN(C)C2)=O)CCC(NC(c2cn[nH]c2)=O)C12CC2 C1(C(C)NC(c2cncn2C)=O)CN(C(c2cc(Cl)cs2)=O)CCO1 N1(CC(=O)NC(CN(C(=O)CC(=O)N(C)C)CC)C)C(=O)NC2(CCCC2)C1=O C(CS(=O)(=O)C(C)(C)C)NC(C1CCN(c2nc(C(=O)OC)[nH]c(=N)c2)CC1)=O C1(NC(c2cc(NC(C)=O)ncc2)=O)C2CCCC1CC(NC(C1(C)CC1)=O)C2 C1(CNC(C(C)OCC)=O)CN(C(c2cn(C)nc2C(C)(C)C)=O)CC1C C=C=CCCC(=O)N1CC(C2CN(C(c3cnc[nH]3)=O)CCO2)C1 C1(F)(C(=O)NCCOC)CCN(Cc2ccc(C(=O)O)o2)C1 N1(c2ccnc(SC)n2)CC2CC(NC(c3cnc(C(F)(F)F)s3)=O)CC2C1 c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ns2)=O)ccc(CCF)cc1 c1(CC(=O)N(CC(O)CNC(=O)C(C)(C)S(C)(=O)=O)C)ccc2c(c1)CCCO2 C1(C(N2CC(C)(NC(c3cc(-c4cccnc4)[nH]n3)=O)C2)=O)CCCS1(=O)=O C(=O)(C(F)(F)C(C)(C)O)NC1CCN(C(Cc2ccc(C)cc2Cl)=O)CC1F CCC(CC(=O)NC1(C)CC(NC(=O)CCN2CCCCC2)C1)OC CC1(C)CCCC(C(=O)NC(CNC(=O)CCCCN2CCCC2)(C)C2CC2)C1 c1(SCC(=O)N(CCN(C(=O)Cc2nccs2)C(C)C)C)cccc[n+]1[O-] CC(C)CS(=O)(=O)CC(=O)N1CCOC(CNC(c2cc(C(C)C)n(C)n2)=O)C1 C(C)(C(C(=O)NCC(C)(C)CNC(=O)C(=Cc1ccccc1)OC)N(C)C)OC c1(NC(c2nnc(O)o2)C)nc(N(C)Cc2nn(C)cc2Cl)nc2sccc12 c1(N(C)C)nc(C(=O)NC2CC(CNC(=O)CCc3ccccc3)C2)[nH]c(=N)n1 CC1CN(C(=O)CCC2CCOC2)CCCN1C(c1ccc2nn[nH]c2c1)=O c1(C(=O)OCC)cc(CNC2CCC3(CC3)C2)c(C)o1 N1(C(CSCC)=O)CCC2(NC(c3nc(C)nn3C)=O)CCCC12 Cc1cc(C(=O)NC(CN(C)C)C(=O)NCC(O)C(N)=O)nc(C)c1 c1(C(N(CC(=O)NC(C(O)CO)C2CC2)CCC)=O)c[nH]c(C#N)c1 c1(NC)c(C(=O)NCC2CCN(C(c3scnc3COC)=O)C2)cccc1F c1(OC)ncnc(C(N2CC3CC(NC(c4cnoc4C4CC4)=O)C2C3)=O)c1F C1(CNC(C2(CCCC)CCCC2)=O)COCCN(C(c2cc(C#N)no2)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cnc(C)cc1C c1(C(=O)NCCC(C)NC(C2C(C)C2C)=O)nn(C)c2c(=O)[nH]cnc12 c1(CN2CC(C(=O)NCCc3ccccc3)(CO)C2)c(F)ccc([N+](=O)[O-])c1F C(Cc1ccco1)(C(=O)NCCC1CC(F)C1)NC(C(C1CCOCC1)C)=O C(=O)(C(C)(CNC(=O)C=CCF)CC)NCCC(CC)C C(=O)(CC1OCCc2sccc21)NC1C(C)N(C(=O)C=CC(C)(C)C)CCC1 C=C1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)NC(C)CC2CCCCC2)C1 c1(CCNC(CN(C(=O)C(c2cnn(C)c2)C)CCOC)=O)ocnc1CO C1(CNC(CC2C=NN(C)C2=O)=O)CN(C(=O)CCCn2cccn2)CC1(C)C C1(CNC(=O)CNc2nccs2)CN(C(=O)Cn2cc(F)ccc2=O)CC12CC2 CC1CC(C(=O)NCC2(C(=O)NC3CC3C3CC3C)CC3(CC3)C2)CN1C C(=O)(C(C)CN(C(=O)CCN(C(=O)CNc1ncccn1)CCO)C)NC c1(CCC)cc(C(=O)NCCN(C(=O)CC(C)COC)CC2CCCC2)ccn1 CC1CN(C(=O)COC2CCC2)CCC1NC(c1cccc(-n2cccn2)c1)=O C(C(CNC(C1CCCC(C)(C)O1)=O)S(C)(=O)=O)NC(C1(CC)CC1)=O C1(NC(CC2(C)CCOCC2)=O)CC2CCC1CN2C(c1ccnc(S)c1)=O c1(CC(C)C)ccc(CCNC2CCCC(NS(C)(=O)=O)C2)cn1 C(=O)(CC(C)C(F)F)NCC(CO)NC(CN(C(=O)OCC)C)=O N1(C(C2(C#C)CCC2)=O)CC2CC(NC(=O)C=C3CCSCC3)CC2C1 c12ccc(cc1)[nH]c2=O.C1(NCCNC(C=CC(C)C)=O)CC(CN(C)C)C1 c1(C(N2CC(OC)C(NC(=O)C(c3cnccc3C)C)C2)=O)ccc(F)c(Cl)c1 C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]nc1Br)NC(C(C)=C(C)C)=O N1(C(C=C(COC)C)=O)CCC2CCN(C(C3SCCS3)=O)CC2C1 N1(C(C(C)n2cnnn2)=O)CCC(C(F)C(=O)N(CC(O)CO)C)C1 c1(CC(=O)NCCc2c(CNC(C3CC(C)OC3)=O)nco2)ncccc1F c1(C(=O)NCC(CC=C)NC(c2ccsc2C(F)(F)F)=O)cc2n(c1)CCC2 Cc1c(C(=O)OC2CCOC(C)(C)C2)[nH]c2cc(Cl)ccc12 N1(C(Cc2ccc(C)o2)=O)CC(C)CN(C(=O)CCc2nc(C)no2)CC1C N1(C(=O)C#CC2CCOC2)CC2CCN(C(c3ccc(Cl)[nH]3)=O)CCC2C1 C1(NC(Cc2ccc(OC)cc2)=O)CCN(C(C2CCCCN2N=O)=O)C12CC2 c1(C(=O)OCC)nc(=NC2CCCCC2NC(C23CC2COC3(C)C)=O)cc[nH]1 c1(C(=O)NC2CC3CC(C2)N(c2nncs2)C3)ccc2ncc(=O)[nH]c2c1 c1(C(N(CCC(C)NC(C2(O)CCC2)=O)C)=O)ccc2nc(O)cn2c1 C(=O)(C(C(C)C)N(CCO)C(C)=O)NCCN(C(C=C(C)Cl)=O)C1CC1.C(C)(C)(C)O C1(CC(=O)NCCOC(CC)(C)C)CCCCC1NC(=O)C(N)=O C(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccncn2)=O)C2C1C2)=O C1(C(=O)NCC(CCC)NC(=O)CC(C)CC)(CO)CCOCC1 c1(C(N2CC3C(CNC(Cc4cc(C)on4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C1(NC(C(C)CSC(F)(F)F)=O)CCCCN(C(c2cn(C3CCC3)nn2)=O)C1 N1(C(c2nc(CC)[nH]n2)=O)CC(CNC(c2ccccc2F)=O)CC1C C(C(=O)N(CCC(=O)N(C(CO)C1CC1)C)CCO)(C(C)C)OCC c1(C(=O)NCc2cncc(C(=O)NCC(C(C)C)CO)c2)cnn(C)c1C#N C1(OCCNC(=O)COC2CC=CC2)CCN(C(=O)C(O)Cc2ccccc2)C1 N1(C(CCOCC#C)=O)CCC2(CC1)CC(NC(=O)CC1SC(=N)NC1=O)C2 C1(CNC(C(C)O)=O)CN(C(c2ncc(OCC3CC3)cc2F)=O)CC(C)(C)O1 N1(CC)C(C)CN(C(C2CCN(C(C3CC(=O)CCO3)=O)CC2)=O)CC1C N1(C(Cc2ccc(C)cc2C)=O)CCC2(CC1)CN(C(=O)C(C)CF)CC2CO Cc1cccc(NC(=O)CC2CN(Cc3cccc(CC(=O)O)c3)CCO2)c1I C(CC(C(=O)NC(C)C(=O)NCCOC)NC(c1ccoc1C)=O)OC c1(C(N(CCN(C(Cc2cc(C)c(CO)cc2)=O)C)C)=O)cc(C#N)ccc1F C(C(=O)NCC(C)(C(C)C)NC(=O)CCn1ccnc1C(C)C)(C(C)C)OCC N1(CC(=O)NCC2CC(NC(C(C)SCCCC)=O)C2)CC2CC2C1 c1(C(=O)NCC2CCCN(C(C3(C)CCCCO3)=O)C2)cc2ccccc2s1 C(=O)(C1SCCc2ccccc21)N(CCCNC(=O)CC1CC2(CC2)CO1)CC C(=O)(N1CC(n2cc(-c3cncs3)nn2)CO1)c1cc(C#N)[nH]c1 Cc1cncc(C(=O)NCC2(O)CCN(C(=O)C(N)=O)C2)c1C C(=O)(CCCC(C)(C)CC)N(C1CCCN(C(C(c2ccccc2)OC)=O)C1)C C12(C(=O)NCC(C3CCN(C(c4cnco4)=O)CC3)F)CCCC1OCC2 CC(C)C#CC(=O)NCC(C1CC1)NC(=O)CCCOc1ccccc1Br C#Cc1ccc(OCC(=O)NC(C(F)(F)F)c2cnn(C)c2)cc1 N1(C(CC(c2ccc(OC)cc2)C)=O)CCC(C)(C)C(NC(c2ccco2)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(CC2CC(=C)C2)=O)cc(C(=O)OC)n(C)c1 N1(C(C(COC)C(F)(F)F)=O)CCC2C(=O)OCC12C c1(OC)cccc(NC(C2CCN(Cc3cc(C4CC4)[nH]n3)CC2)=O)c1F C1(C(N2CC(SC)C(NC(c3ccc(C)cc3)=O)C2)=O)CC2(CCO1)CC2 N(C1CCCc2occc21)C(C1(NC(c2ncc(C)c(C)c2)=O)CCN(C)C1)=O CN1CC(O)CC1C(=O)NCCCCCCN(C)C(C1CC2CCC2C1)=O C1(C)(C(NOC(C=C)C)=O)CCN(C(C2CCC(CC)C2)=O)CC1 C1(C(N(CCCCCCNC(C(C(=O)OC)C)=O)C)=O)CC(=O)N(OC)C1 CC1=C(C(=O)N2CC3CC2CCC3NC(=O)Cc2coc(C)n2)CCCO1 C1(NC(C=C(CC)C)=O)CC2CC1CN(C(c1n[nH]c(CC)c1Br)=O)C2 c1(CNC(=O)NCC2(C)CCOCC2)ccc2c(c1)CC(=O)N2 C(C)(CN=c1ccc(S(=O)(=O)NC2CC(CC#N)C2)c[nH]1)c1c(C)noc1C Cc1ccccc1C=CC(N1CCN(C(c2cccn2C)=O)C(C)C1)=O C#CCC(CC(=O)NCCCO)NC(=O)CCCCC=C c1(OC)cc(NC(C2CCOCCN2C(C2CCC2C#N)=O)=O)cc(F)c1 C1(C)(CC)CCN(C(C2(CNC(c3cnc(C)cn3)=O)CC=CC2)=O)CC1 c1(-c2ccc(C(=O)NC(C(=O)OC)Cc3ccccc3)o2)cc(F)ncc1F c1(C(=O)NCC2CN(C(C3(C(N)=O)CCC3)=O)C2)cc2nn[nH]c2cc1F C1(OC(=O)NCC(n2cncn2)C)CCN(C(c2cnc(C(C)OC)s2)=O)CC1 c1(NCCCCCC)ccc(-c2csc(C(C)=O)c2)cc1.N12CCC(CC1)C2 C#CC1(C(=O)N2CC=CCO2)CCN(C(=O)CSC(F)F)CC1 CC(C)(CS(C)(=O)=O)NC(=O)CCC(c1ccc(F)c(F)c1)=O n1(CC(N)=O)cc(C(N2CC(CO)(NC(c3coc(Br)c3)=O)C2)=O)nn1 C1(C(N(CC(CC)O)C)=O)(CC)CCN(C(=O)CCC(C)C)CC1 C(C1Cc2ccccc21)OC(c1ncc(C#C)cn1)=O c1(NC(C(CC2CC2)NC(C2CN(OC)C(=O)C2)=O)=O)cccc2c1CCC2 c1(C(N2C3CN(Cc4ccc(CO)o4)CC23)=O)cc(F)c(Br)c(F)c1 C1(CC)CN(C(c2cn(C)cn2)=O)CCN1C(c1[nH]cnc1-c1cccnc1)=O n1(CCC(=O)N(CCCCCC)CCNC(C2C(C)C2C)=O)ccccc1=O C1(C)(C(=O)NCCN(C2CCCC2)C(c2ccc(SC)o2)=O)CC2CC2C1 Cc1ccc(F)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)CC1O c1(C(=O)NCC2CCCN(C(CCCCC)=O)C2)cnn2c(Cl)cccc12 C1(C)(C(=O)NC(c2nc(C(=O)NC3CN4CCC3CC4)co2)C)CCCN(C)C1 c1(CC)ccc(C(=O)NCCCOCCNC(c2ocnc2C)=O)c(OC)c1 N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(C1CC3CCC1O3)=O)C2 C1(OC)CC2CC(C(N3CCN(CCCNC(C4(C)CCCC4)=O)CC3)=O)CC12 c1(C(=O)NCC2(C)CCN(C(=O)C(F)=C3CCC3)C2)cnn2c1S(=O)(=O)NCC2 O=S(=O)(c1c[nH]ccc1=NCC1CCC12CCOCC2)NCCc1nncs1 N1(CC(=O)NC2C(CNC(CCS(C)=O)=O)COC2)C(=O)CC(C)(C)C1=O N1(C(C(C)O)=O)CC2CC1CN(C(c1ccn3c1CSCC3)=O)C2 C1(NC(c2cc(CF)on2)=O)CC2(CCCCN2C(=O)CCC[N+](=O)[O-])C1 Cc1ccc(F)c(NC(C2(C)CCN(C(C3CC3C3CC3)=O)C2)=O)c1 O=C(CCCC(F)(F)F)NCCC1CCN(C(=O)CCC2CCOC2)C1 c1(C(N(C)CCOCCNC(C2CC2(C)C(F)(F)F)=O)=O)c(F)ccc(N)c1F C(C)(C)(CC(F)C(=O)NCc1cnc(C)n1CC)NC(C(C(CC)O)C)=O c1(NC(CC2CCN(C(C(CCC)CCC)=O)C2)=O)ccc2ccccc2c1Cl C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)CCN(C)CCc1ccccc1 c1(OC)cccc(C2(NC(C3CN(C(=O)Nc4ccc(=N)[nH]n4)C3)C)CC2)c1F C(C1C(C(=O)N(CCO)CC23CC(NS(=O)(=O)CCCCl)(C2)C3)C1(C)C)=C(C)C Cc1ccn(CC(=O)NC2COCCN(c3nnc(C)s3)C2)c(=O)c1 c1(C(C(=O)NC(C)CCNC(=O)COCC(C)(C)C)(F)F)nc2ccccc2s1 CC1(C)C(CNC(c2ccncc2)=O)CCN1C(C1COCCO1)=O Cc1ccc(C(=O)NCC2(NC(=O)CSC(C)C)CCCC2)c(=O)n1C CC1CCn2cc(C(N3CCCC(c4nnc5ccccn45)C3)=O)nc2C1 c1(NC(C)=O)cccc(C(=O)NCC(CC(C)C)NC(=O)Cc2nccn2C)n1 CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(C3CCCCCCC3)=O)C2C1 N1(C(C)=O)CC2CCCC2(C(=O)NC2CC(=C3CCC3)C2)C1 c1(CN2CCC(CC(=O)Nc3c(CC)n(C)nc3)C2)ccc([N+](=O)[O-])cc1Br CC1CN(C(=O)C(c2ccc(F)cc2)=O)CC1NC(=O)CC1CCC(=O)N1 C1(CNC(C(CC)(C)CC)=O)CN(C(=O)CCCc2csc(C)n2)C2CCN1C2 CCC(C(=O)NC1CC(NC(=O)C(=O)Nc2ncc[nH]2)C1)C1CCOCC1 CC1(C)CCN(C(C2CCCC2NC(c2ccc(OC(F)(F)F)cn2)=O)=O)CC1 C1(F)(CNC(C2CC=CCC2)=O)CCC(CNC(C2CC(O)C2)=O)C1 C1(NC(CCCC#CC)=O)COC2CN(C(C3C=CCCC3)=O)CC12 CCC(O)C(F)(F)C(=O)NCC1CN(C(c2ncccc2Cl)=O)CC1(F)F C1(CC=C)(C(=O)NC(c2csnn2)C)CN(C(=O)CCC2CC2(C)C)C1 C1(CC(C)C)COCCN1C(c1sccc1CNC(c1cc(Cl)n[nH]1)=O)=O N1(C(C(C)CC2CCC2)=O)CCC(C(C)(O)CNC(C2(O)CCC2)=O)CC1 CC(C)CC(C)C(=O)NCC(C)(C)CNC(C1CSCN1C(=O)C(C)(C)C)=O C1(C)(CC=C2CCOCC2)CCN(C(C(C)NC(C(n2ccc(-c3ccccc3)n2)C)=O)=O)CC1 C1(NC(C(C)Oc2ccccc2)=O)C2CCC(C2)C1c1nn[nH]n1 CN=c1cc(C(=O)NCCCC(=O)N(C)Cc2nncn2C)cc[nH]1 c1(-c2c(C)nc(=N)[nH]c2)cc(C)c2c(C(N3CCC(F)C3)=O)n[nH]c2c1 c1(CC(N2CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)ccc2ccccc2c1 C1(CNC(C=Cc2nc(C)sc2)=O)CN(C(=O)C(C)C2(O)CCC2)C2(CCC2)C1 CC1CCC=C1C(=O)NCC1(CNC(=O)COC2CC(F)(F)C2)CCC1 CC(C)(CNC(=O)CC1C(NC(=O)Cc2cc[nH]n2)CC1O)CC(F)F C1(C(=O)NCCCCNC(c2occ(C)c2)=O)CSC(c2ccccc2)=N1 C1(CNC(=O)NC2(C(N)=O)CCOC2)CCCOC1C1CC1 c1(C(C(=O)NCCCSCC)N(C(C(=O)OCC)C)C)cc(CC)n(C)n1 C1(CNC(C2(CC)CCC2)=O)CN(C(=O)Cc2cc(C)no2)CC12CC2 c1(C(C(=O)NCCCOC)N(CC(=C)Br)CC)cc2ccccc2o1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2ccoc2)=O)C1 c1(C(c2nnnn2C2(C)CC2)NC(C)Cc2cccc(F)c2)ncc(F)cc1F N1(C(COC(CNC(COCCOC)=O)(C)C)=O)CCSC(C)CC1 C1(NC(CN(C)C(C2CCC(C)(C)C2)=O)=O)CCN(CCO)CC1 C1(C(=O)NCC2N(C(c3c(NC)cccc3)=O)CCC2C)CC(=O)NC1(C)C CCCCC(C(=O)NCc1ccccc1)N1CCC(C)(CC)CC1 Cc1conc1C(=O)NC(CNC(c1csc(-c2nc[nH]n2)n1)=O)C(C)C N1(C(C(C)OC)=O)CCC2(CC2C(=O)NCCCC(O)CO)C1 CC1CN(C(c2ccc(N)c(O)c2)=O)CCC1CNC(=O)CCNC(N)=O C1(O)(C(C)NC(C(C)n2cnnn2)=O)CCN(C(=O)CC(C)NC(N)=O)CC1 C1(NC(=O)CN2CCCC2=O)CCC2CC1CN2C(C12CCC(C1)OC2)=O c1(OC)cccc(CCC(C(=O)NCC(F)Cl)N(C(C)CS(C)(=O)=O)C)c1 N1(C(CCCCCC)=O)CCCCC1C1CCCN1c1cc(O)ncn1 N1(C(c2ccc(F)s2)=O)CCOC2CN(C(C3(F)CC3)=O)CC12 C12(C(=O)NC3CC(CCNC(C(C4CCCC4)SC)=O)C3)CCC(O)(CC1)CC2 C1(CCOC)CN(C(c2coc(Br)n2)=O)CCN1C(=O)CCS(N)(=O)=O c1(OC)ccc(-c2ccccc2C(=O)N(C)C)cc1C(F)F C(=O)(CCC(=O)NCC1CC(NC(c2cc(Cl)ns2)=O)C(O)C1)NCCC c1(N(C)CC2(CC(N3CC(C(=O)NC)(OCC)C3)=O)CC2)cn(C)cc1C(N)=O N1(C(C(C)C2(O)CCC2)=O)CCCC(C(N2CCCC2)=O)CC1 Cc1ccc(Cl)c(C(C(=O)NC2COC2)N(C)CC2CC2)c1 N1(C(C(CC)Br)=O)CCC(N2CC3CC3C2)C(C)CC1 CC1OCCC12CN(C(C(=O)NC1CC1)C1CC1c1ccnn1C)CCO2 C1(NC(c2cc(C(=O)OCC)n[nH]2)=O)CCCC(NC(C2CNC(=O)N2C)=O)C1 c1(C(=O)NCC2(CC(=O)N(C3CCCCC3)CC#C)CC2)nnc(O)nc1O C12(C(N3CC(CNC(C4CC=CCC4)=O)OCC3)=O)CCC(F)(CC1)C2 c1(C(=O)NC2CC(C)N(C(=O)C(C)CC(C)(C)C)C2)ccc2cncn2c1 N1(C(CC(C)F)=O)CCC(C2(O)CN(C(=O)CC(C(F)F)C(C)(C)C)C2)CC1 CC1(OCC(=O)NC2(CNC(=O)C=CCF)CC2)CCOCC1 CC(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(=O)CCCN(C)C)CCO1 C1(C(=O)NCCCCC(C)NC(CCC(=C)C)=O)CN2CCCC2CO1 C1(CNC(CC(CN(C)C)O)=O)CC(C(=O)NCCC(N)=O)=NO1 C1(CNC(COCCOC)=O)CC(F)(F)CN1C(c1cc(C(C)C)ccc1C)=O CCC(CC)(CCNC(C1CC(C(C)C)=NO1)=O)NC(C1C2CC(=O)CC12)=O C1(NC(=O)NC2CCOCC2C(=O)O)Cc2ccccc2C1 N1(C(C2CC(OC)C2)=O)CCCC(C2CCN(C(=O)Cc3cccnc3Cl)C2)C1 Cc1c(C(=O)N(C(C)CNC(C2OCCC2(C)C)=O)C)csc1Br CCN=c1[nH]c(C(=O)NC2CN(C(=O)CC=C(Cl)Cl)C(C)(C)C2)cs1 c1(C(C)OCC)noc(CCC(=O)N(CCCCNC(C2(Cl)CC2(C)C)=O)C)n1 c1(CC)nc(C)c(CC(=O)NC2CC(=O)N(C3CN(C(=O)C(C)C)C3)C2)c(C)n1 c1(OCC(N2CC(C)(NC(=O)NC3CN(C)C3)C2)=O)ccc(F)cc1F c1(CC)nocc1C(N1CC(C(C)NC(c2cc(CO)[nH]n2)=O)C1)=O C1(C(N2CCC(n3cc(-c4ccc(=N)[nH]c4)nn3)CC2)=O)(OC)CCCOC1 N1(C(C(C(C)C)SCC)=O)CC(CNC(=O)Cc2nonc2C)C2(CC2)C1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C)SC(C)C)C2)cnc1O CC1CCc2c(C(=O)NC3(C)CCC(NC(=O)CC4CC=CC4)CC3)csc2C1 c1(C(=O)NC2C(C(N3CC(C(=O)OC)C(F)C3)=O)CCCC2)ccc(Br)c(Cl)c1F c1(C(N(c2nccc(C)n2)C2CCNCC2)=O)ccc2c(c1)c(C)c(C)n2C N1(C(C(F)=CCC)=O)CCC2(CCN(c3nc(CC)nc4sccc34)C2)C1 C1(NC(c2c(CC(C)(C)C)cccc2)=O)CC2CC1N(C(c1cncs1)=O)C2 C=C(Cl)CC(C(=O)NCC(=O)N(CC)OC)NC(=O)COCCCC(C)C c1(C(=O)NC2CC(NC(C(CC)(C)F)=O)C2)nc(OC)ccc1C c1(C(=O)NCCN(C(C(CC)NC(N)=O)=O)CC(C)O)cnn2c1NCCC2 C1(C(N2C(C)CCCC2C(N2CCOCC2)=O)=O)Cc2cccnc2C1 c1(C(C(=O)NCC2CCCO2)N(C(C2CCC2)C)C)ccc(CCCC#N)cc1 N1(C(c2nc(CC)[nH]n2)=O)CCCC12CCN(C(=O)C(F)C(C)C(F)(F)F)CC2 N1(S(CC)(=O)=O)CC2(CCC(NC(c3cc(Br)c(C)cc3O)=O)CC2)C1 N1(C(c2cc(C)c(O)nn2)=O)CCCCNC(=O)C(F)(F)C1 C1(C)(CNC(c2cc(COC)sc2)=O)CCCN1C(c1c[nH]nc1C)=O c1(CN(C(c2csnc2C)C(=O)NCC)C)cccnc1OC Cc1nn(CC(=O)NC2COCC2NC(C2CCC(C)(C)O2)=O)c(=O)n1C C1(NC(C2CCCC2(F)F)=O)CC(CO)N(C(c2cncc(F)c2)=O)C1 c1(OC)ccc(F)c(C(N2CCN(C(=O)Cn3cnnc3O)C(CO)C2)=O)c1N c1(C(=O)NC2C=CCN(C(C3CCN(C)C3=O)=O)C2)c[nH]c2nccc-2c1 C#CCCC(C(=O)NCC1(O)CCCC1(C)C)NC(=O)CCCCC CCCCC(CC)C(=O)NC1(CO)CCN(C(=O)Cc2nc[nH]n2)C1 c1(C(N(CC)Cc2ccco2)=O)cc(Cn2cccn2)on1 N1(C(C(CC)OC)=O)CCN(C(=O)COc2cccc(C#N)c2)CC1C1CCC1 c1(C(N2CC3C(NC(c4cnc(Cl)[nH]4)=O)(C3)C2)=O)cc2c(Cl)nccc2o1 N1(C(C=Cc2n(C)cnc2)=O)CC2(CCCCN(C(c3cccnn3)=O)C2)C1 c1(CNC2CCC(NC(c3ccc(OC)c(I)c3)=O)C2)ccc(Br)cc1[N+](=O)[O-] Cc1c(C(=O)NCCCCNC(C2(C)CCC(C)(C)CC2)=O)nn2ccccc12 Cc1ccc(F)c(-c2cn(C(C)CNC(=O)C(C)(C)CC3CCOC3)nn2)n1 C(=O)(C1=CS(=O)CCC1)NCCCNC(C(N1CCC(C)CC1)C(C)C)=O c1(C(=O)NC2C(CC=C)C(O)C2)ccnc(OC)c1Br C(=O)(C(C)(C)C1=CCN(C(=O)CCCCSCC)C1)NCCc1n(CC)cnn1 N1(C(C2(CC)CCC(O)CC2)=O)C2CCC1CC(CNC(=O)CC1CN(C)C1)C2 CC1CC2CN(C(=O)CC(C)(F)F)CC2N1C(=O)Cc1cccc2ccncc12 C1(CNC(C2(SC)CC2)=O)CN(C(C2CC3(CCC3)C2)=O)C2CCCCC12 Cc1cc[nH]c1C(N1CCC(N(C)C(c2csc(CS(C)(=O)=O)n2)=O)C1)=O C=CC1COCCN1C(C1CC(O)CN1C(c1ncccc1N)=O)=O N1(C(C(C)OC)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(OC)C1 C1(C(N2CCC(CC=C)(NC(C3CC3=C)=O)C2)=O)C2CCCCCCC12 CCCCCCCCN(C(=O)C(C)(C)NC(=O)COC(CC)CC)C Cc1c(CNC(c2nc(CC3CCCC3)nn2C)=O)noc1-c1ccc(Cl)cc1 c1(C(N(CCC=C)CCOC)=O)cc2ccc(-c3cc(C)nn3C)cc2o1 C1(C(=O)NCCCn2c(C)ncc2)CC12CCN(Cc1c(F)cncc1F)C2 C(=O)(C(CNC(C1CC1Cl)=O)N(C)C)NCCCOC C(=O)(N=c1ccn(C)[nH]1)C1(O)CCN(C(c2c(C)nc[nH]2)=O)CC1 C1(CC(=O)NCC(C)(C2CC2)NC(c2cnc(C3CC3)o2)=O)CCCOC1 c1(CC)ncncc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(C(N)=O)co1 N#Cc1cccc(C2(C(=O)NC3CCCC(NC(=O)Cn4nccn4)C3)CC2)c1 N1(C(CCC(C)NC(c2cc(=O)n(C)cn2)=O)=O)CC2CC1C(F)(F)C2 C1(C(=O)NCCn2c(C)ncc2)CC(O)CN1C(C1COC(=O)N1)=O C(=O)(C(F)(F)C(C)O)N(c1ccc(CC(=O)NC)cc1)CC.C1(C)(CO)CCCC1 c1(C(N(C(CCNC(CCC(C)CN(C)C)=O)C)C)=O)cc2n(n1)CCCO2 c1(C(=O)NCC(O)CNC(C2OCCCO2)=O)n[nH]c2c1COc1ccccc1-2 C1(C(=O)NCc2ccncc2N2CCOCC2)CCc2ccccc2N1 C(C(=O)N1CCC(NC(=O)CC2CCC2(C)C)CC1)(C(C)C)NC(=O)OC c1(C(=O)NC2(C)CC(NC(C=CC)=O)C2)ccc(C(C)(F)F)nc1 c1(C(N2CCC(C(C)NC(c3ccc(O)nc3)=O)C2)=O)ccc(O)nc1Cl C#CCC(C)(C)C(=O)N1CCCC1CNC(=O)C(c1cccc(C(F)(F)F)c1)(C)O C(C(C)(C)CC(=O)NC1C(C(=O)NCCCN(C)C(C)C)C1(C)C)OC(C)=O c1(C(=O)NCCC2OCCN(C(C(C)OCC3CC3)=O)C2)cc(N)nc(Cl)c1 c1(CN2C(C(N3CCC(C#N)C3)=O)CC3CC32)nc(Br)ccc1F C1(O)(C(=O)NC2C(NC(=O)C=Cc3ccco3)CC2)Cc2ccccc2C1 CC(C)C(C(=O)N1CC(NC(c2ccc(CSC(F)F)o2)=O)C1)c1cnn(C)c1 C1(C(=O)NC2CCCN(C(C3(C#N)CC(C)C3)=O)C2)CCC2(CCC2)CC1 c1(C(CC)NC(C(CC(=O)O)=O)=O)ccc2nccnc2n1.OCC C(CCCCC(=O)NC1(CN(C)C(C2(C)CCCC2C)=O)CC1)=CC c1(NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)cc(=O)n2ccccc2n1 c1(SC)ccc(CC(=O)NC2CC(C)(NC(c3ccc(C(N)=O)o3)=O)C2)cc1 C(=O)(CCC(C(C)C)NC(C1C2CCC(F)C12)=O)N1CC(C#C)C(O)C1 C(=O)(C(F)C(C)C)NCC(C)(C1CC1)NC(c1c(C(C)C)nns1)=O C(=O)(C1=CCCSC1)N1CCC(CCNC(C(C(C)C)SC)=O)C1 c1(C(N2CCC(O)(CCNC(C(CCC)(C)C)=O)C2)=O)cccc2occc12 c1(C(=O)OCC)cc(Br)ccc1N(C)Cc1sc(C)cc1C c1(N2CCC(C)C2CNC(=O)C(C)(C)CO)cc(Cl)nc(-c2ccc(F)cc2)n1 C1(CC=C)(NC(=O)C(C2CCOC2)NC(=O)Cc2cc(C)[nH]n2)CC2CCC1C2 C(C(C)C(C)(C)C)N(C(C(CSCC)NC(c1cnsn1)=O)=O)C C1(C(=O)NC(CNC(CC(=O)NCC)=O)(C)C2CCC2)CCC2CC1C2(C)C N(C(=NCCCF)NCC1(C2CC2)CC1)Cc1c(OC)nccc1 c1(NC(C(C)N(C2CCCC2C)C)=O)cccc(-c2nc(Br)ns2)c1 CC(CC(=O)NC1C2CC1N(C(c1ccc3c(c1)CC3)=O)C2)CC(C)(C)C c1(C(C(=O)NCCCN(C(c2c(CC)csc2)=O)C2CC2)OC)cccc(Cl)c1 CC(C)(CC(F)(F)F)C(=O)NC1COCCC1NC(=O)CN1CCCOC1=O C(C)(CN=c1[nH]nco1)(CC(C)C)NC(c1cc(OC)c(Cl)cc1)=O N1(C(c2nc(CC)oc2)=O)CCCC(CNC(=O)C(C(C)(C)C)C2CCC2)CC1 c1(C(N2CC(C=C)OCC2)C(=O)NC2CCCC2)cccn2ccnc12 N1(C(C(CC=C)OC)=O)CCC(=C)CC1C(=O)NCC1CC(CF)C1 O=C(C#CC1CCCCC1)NC(C(=O)N)C1CCCO1.C1CCC(=O)O1 C1(C(=O)NCCC2CC(NC(c3ncn(CC)c3)=O)C2)(CC)CC=CCC1 c1(OC(=O)NCC2(COC)CCC2)ccc(C(=O)OC(C)C)cc1O C1(OC)CC(C(N2CC(NC(c3cc(CCO)on3)=O)C(CO)C2)=O)CC1OC N1(C(c2ccc(OCC)cc2)=O)CC2CC(C1)N2C(c1ccc(C)cc1O)=O N1(C(C(CC)(C)O)=O)CC2CCN(C(C3(N4CCCC4)CCC3)=O)CC2C1 C1(NC(C(C=C)O)=O)CN(C(=O)CCCOc2ccc(C(C)(C)C)cc2)CC1C C1(C(=O)NC2CC(CO)N(C(C3CCCN3c3nccs3)=O)C2)C2CCCCC12 c1(NC(CCN(CC#C)C(C2CN3CCC2C3)=O)=O)cc(C)cc(O)c1 c1(CC(n2cc(C3COCCN3C(C3(C)CC3)=O)nn2)C)ccccc1F c1(C(N2C(C)CC(CNC(=O)C#CC3CC3)C2)=O)ncc2ccccc2c1O N1(C(C(C)C(=O)N2CCOCC2)=O)C2CCC1CN(C(C1(CF)CC1)=O)C2 N1(C(C(CNC(=O)C(C)(C)OC(C)=O)OC)=O)CCC2(CCOC2)C1 C(c1ccc(F)cc1)=CCC(=O)NCC1CCCC(NC(=O)C2=CCCOC2)C1 c1(C(=O)NC2CCCC2CNC(C2(F)CCC2)=O)cccc2cccnc12 c1(Cc2n(C)c(C3CC3)nn2)ccc2c(c1)CN(S(=O)(=O)C1CCOC1)CC2 Cc1nc(NC(C2C3(CC3)C23CC3)=O)c2cnn(-c3ccc(F)cc3)c2n1 N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)C=C2CCCCC2)CC1CC1CC1 c1(OC)cc(C(=O)NC(CNC(=O)C(=O)NC(C)C)C2CCC2)cnc1O c1(CCNC(CCN(C(=O)CC(=O)NC2CC2)CC#C)=O)ccccc1 Cc1cc(CNC(C2CCN(C(=O)CSc3nnc(C)s3)CC2)=O)cc(C)c1 c1(N(CCOCCNC(C(C(C)(C)C)SC)=O)C)cc(C)ccc1[N+](=O)[O-] C1(C(=O)OC)CCC(CN2CCC(c3ocnc3C(=O)NC(=O)NCC)C2)CC1 c1(SCC(N2CC(CC(C)NC(=O)Cc3nc[nH]n3)C2)=O)ccccc1O N1(CC(=O)N(CCn2cc(Cn3ccnc3)nn2)CC)CCOCC1=O C1(NC(c2n(C)cc(F)c2)=O)CCCN(Cc2ccc(Cl)cc2Br)CC1 CCCCC(C(=O)NCCn1cnc(C(N2CCCC(OCC)C2)=O)c1)C(C)C C1(CC(=O)N(CCC)C)CCCCN1C(c1cccc(F)c1)=O C(=O)(CCCCC#N)N1CCC(C(=O)NOCC(=C)C)(CC=C)C1 c1(C(N(C)CC2N(c3snc(C)n3)CCC2)=O)cc2cccc(Cl)c2o1 C(C)(CC(=O)NCCCCN(C)C(c1cn(C(F)(F)F)cn1)=O)SC C1(CNC(c2ccc(C)s2)=O)CN(C(=O)C(C2CCOCC2)F)C(C)(C)C1 CC(C)C(F)C(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(C(=O)NCC(=O)N(CCN(C(C(C)O)=O)C)C)cc(F)ccc1F c1(NCC2CCC(NC(C(c3ccc(C)cc3)=O)=O)C2)ccc(C)cc1[N+](=O)[O-] C1(OC(C)(C)C)CC2(C1)CC2NC(=O)OC(C)(C)C.c12nnc(s1)c(=O)o2 C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2coc(CO)c2)=O)CC12CCOCC2 c1(C(=O)NC2CCCC(NC(c3onc(C)c3C)=O)C2)c2c(c[nH]c1=N)CCC2 C(=O)(C(C(C)(C)C)c1cnno1)NCC1(F)CN(C(C2(C)CCCS2)=O)C1 N1(C(C(CC)C#N)=O)CCCC(N(C(=O)C=Cc2cccs2)C)CC1 CN1CCCCC1C(N1CCC(O)(CNC(C2(C(F)(F)F)CC(F)(F)C2)=O)C1)=O C(=O)(CC1COc2ccccc21)OCC1(CNc2c(SC)ccc(OC)c2)CC1 c1(NC(C2C(O)CCN(C(CCOC)=O)C2)=O)ccc2occc2c1O CC1COCC(CC(=O)N(CC(CO)(CO)NC(=O)COCc2nc[nH]n2)C)O1 N1(C(C(C)c2cccs2)=O)CSCC1C(=O)NC1CCNC1=O C#CCC(C(=O)N(C)CC1(F)CCC1)NC(=O)Cn1ccccc1=O C12(C(N(CCSC)C)=O)CC1CN(C(C1COCC1(C)C)=O)C2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)N1CC(CCNC(c2c(C)cco2)=O)OCC1 N1(C(C2C(CC)C2)=O)CC2CC1CCC2NC(=O)CC1COCC(C)(C)O1 n1(CC(=O)NCC2(C(N)=O)CN(C(CNC(CCC)=O)=O)C2)ccccc1=O N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)C(N1CCCCCC1)C)C2 N1(C(C(OC)OC)=O)CCN(C(=O)C(c2cncn2C)O)CC1c1ccncc1 CCCC(C(=O)NC1CCN(C(=O)C(C(C)O)N(C)C)CC1)NC(N)=O C(=O)(C1=CCCCC1)N1CCCC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1 Cc1ccc(N)c(C(=O)N(CCCNC(=O)C(C)C)Cc2cccnc2)c1F C(=O)(CCC(=O)NC1CCCCC1CNC(C1CN(C(C)C)CCO1)=O)NC C1(NCc2c(CC)cccc2)CN(C(C2CC=C(C)CC2)=O)CCC1F C(=O)(C(=O)NNc1ncc(Br)cn1)Nc1c(C(=O)OCC)ccs1 c1(CN2C3C(C(=O)NCCc4nn[nH]n4)C(C3)C2)ccc(F)c(O)c1 C(=O)(C1=CCS(=O)(=O)C1)NCC(CNC(Cc1c(CC)cccc1)=O)O C1(C(=O)NCC2C(NC(c3ccc(CC)cn3)=O)CCC2)CCC(C#N)CC1 C1(CNC(C(C)(C)OC)=O)CC2(CCOCC2)CN1C(c1cnc(C)n1C)=O C1(C(=O)OC)N(C(C(=O)Nc2ccc(F)cc2C)C2CC=CC2)CCSC1(C)C CC1CC(CC(=O)NC(C)CC(C)(C)C)CN1C(=O)CNc1cccnc1 c1(C(N2CCC3(C2)CN(C(c2cc(O)no2)=O)C3)=O)cn2ncccc2n1 C(CC(=O)N1CC(CNC(=O)C(C2CC2)SC)C1)NC(=O)OC N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC1CN2C(C1CC1(C)Br)=O c1(-c2onc(C)n2)ccc(NC(=O)NCC(C(F)F)N2CCCC2)cc1 c1(C(=O)NCCN(C)C(C23CC(C(C)(C)C)(C2)C3)=O)ncn(C(F)F)n1 CCC(C(O)C(C)C)NC(C1C2CC3C(C2NC(=O)CCc2ccnn2C)C13)=O c1(C(C)(CO)NC(=O)CC2CC3CCC2O3)ccccc1Cl C1(N(C(CCCC)=O)C)CN(C(c2cccc(N(C)C)n2)=O)CCC1O C(=O)(C1=CCN(C(=O)CCOC2CCC2)CC1)NC1CCCN(C)C1 c1(NCC2C(C)CCNC2=O)ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1Br C1(CNC(CNC(c2c(C)occ2)=O)=O)CCCCCN1C(C1CC(C#N)C1)=O N1(C(c2c(Cl)cccc2Cl)=O)CC2CCCC(C1)N2C(=O)C(F)Br N1(C(Cc2cc(C)c(Cl)cc2)=O)CC(CNC(=O)C2=NNC(=O)C2)C2(CCC2)C1 c1(C(=O)NC(CCCNC(c2c(OC)cccn2)=O)C)noc2c1CCCC2 C1(C(N2CCC(SC(F)(F)F)CC2)=O)(OC)CCN(Cc2ccccc2C)CC1 N1(C(C2CC=C(C)CC2)=O)CC2(CCC2NC(=O)C#CC2CC2)C1 C1(CNC(c2ccc(CCC)cc2)=O)CC(NC(c2cnc(C)[nH]2)=O)C12CCC2 C(c1cc(F)c(O)c(F)c1)=CC(=O)NCC1CCN(C(CNS(NC)(=O)=O)=O)C1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC2CCC1CN2C(=O)CCn1ccnc1 N1(C(C(=O)NCC2CCN(C(c3c(C(C)C)n[nH]c3)=O)C2)C)CCP(C)(=O)CC1 N1(C(c2cc(C(C)C)nn2C)=O)CC(NC(C2CC2(C)Br)=O)C2(CCOCC2)C1 N1(C(CC=C(C)C)=O)CCCOC(CCNC(=O)CN2C(=O)CNC2=O)C1 CC(C1CC1)=C(F)C(=O)N(CCOc1ccsc1)CC1CCCO1 N1(C(C(=O)C2CC2)=O)CC2(CCCN2C(=O)CCN2C(=O)C=CC2=O)C1 c1(C(N2CCC(CCNC(C)=O)C2)=O)ccncc1F.c12nnnn1C1CN2C1 c1(C(N2C(CCNC(C3(SC)CCC3)=O)CSCC2)=O)ccc2cnccc2c1 c1(C(N2CC(C)OCC2)=O)ccc(-c2ccccc2C#N)c2c1OCO2 C(C(C)NC(=O)C=CCN(C)C)N(C(C1CC1CC(C)C)=O)CC n1(CCC)nc(C)cc1C(N1CCOCC1CCNC(C1CCCO1)=O)=O CC12OCC(NC(c3ccc(C(=O)N(C)C)cc3)=O)(CO1)CO2 c1(C(=O)NCC(C(C)(C)C)NC(CC2(COC)CC2)=O)ccc(Br)c(N)n1 N1(C(CN(C(c2ccccc2)C)CC)=O)C2CCC1CN(C(C1CCC1)=O)C2 C1(NC(=O)CC2CC(F)(F)C2)CCC2(CCN(C(=O)C(O)C3CC3)C2)C1 c1(C(N2CC3C(CNC(=O)CCc4nnc(CO)o4)C3C2)=O)cccc2[nH]ccc12 C1(F)(CNC(CSCCOC)=O)CCC(NC(=O)C(c2cccc(C)c2)C)C1 Cc1cccc(CC(=O)NC(C)(CNC(c2c[nH]nc2C)=O)CO)c1Cl C(c1ccc(C)cc1)=CC(=O)NCCN(C(C=COCC)=O)CC C1(CCCNC(C(N)=O)=O)CN(C(c2ncoc2C2C3CCCC23)=O)CCO1 N1(C(CC(CC)C)=O)CCC(CC(N)=O)(NC(C2CCCS(=O)(=O)N2)=O)CC1 N1(C(c2cc(COC)[nH]n2)=O)CC2CC3CC2C1C3NC(C1CCC1(C)C)=O c1(C(N)=O)ccc(C=CC(=O)NCCC2CC(NC(C3C4CCC3CC4)=O)C2)o1 Cc1ccc2cc(S(=O)(=O)N3CC(S)CC3(C)C)ccc2c1 c1(C(N2C(CC#N)CN(C(c3sccc3Br)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NC(C(=O)NCCC2CCC(C)(C)C2)CC2CC2)CCCCC(=O)N1 N1(C(c2cn(CCC)nn2)=O)CCCC(C2(NC(C3C=CCC3)=O)CC2)C1 CC(C)(CC(=O)NCC(C(F)(F)F)N1CCN(C(C2CSC2)=O)CC1)C1CC1 C1(C(C)(C)NC(C2C(C)C2)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(NC(C2CCC3(CN(C(C(CC)C)=O)C3)O2)=O)cnc2ccc(Br)cc2n1 c1(C(N2CC3C(CNC(C(C)OC)=O)(C3)C2)=O)ccc2c(n1)CCOC2 c1(C(C(=O)N(CCOC)Cc2c(C)noc2C)(C)C)ccccc1C(F)(F)F Cc1ccc(C=CC(N2CC(NC(=O)C3=CCOCC3)C3CCCC23)=O)c(C)c1 C1(CCNC(c2nc(CSC(C)C(N)=O)sc2)=O)COCC1(C)C N1(C(C)=O)CCC(C)(C)CC1C(=O)NCC1C2CCCCC12 C1(NC(Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)CSCC(N)=O)CC2 c1(CC)ccc(C(=O)NCCOCCCNC(C2CC3CCC2O3)=O)cc1 C1(C(=O)NC2(CC=C)CN(C(c3cc(C)nn3CCC)=O)C2)CC12CCOCC2 C1(C(N2CC(NC(C(C)CC3CCC3)=O)C2)=O)CCN(c2cccc(Cl)c2)C1=O Cc1ccn2ncc(C(=O)NC(C)CCNC(C3(NC(C)=O)CCCC3)=O)c2c1 C1(CC(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)(NC=O)CCCCC1 C1(NC(C2(NC(c3c(C)csn3)=O)CCSC2)=O)CCCCCC1CO c1(NC(=O)NCCc2c(C)ccs2)cc(F)cc2ccoc12 c1(C(=O)NC2CC(F)(CNC(CN(CCOC)C)=O)C2)ccc(C(C)(F)F)nc1 n1(CC)c(C(N2CCC(CNC(C3(CCOC)CC3)=O)C2)=O)cnc1O Cc1ncnc(C)c1CC(N1CCN(C(=O)CC2CCC3(CC2)CC3)CC1C)=O N1(CC2C(C(C)C)C2)C(=O)CN(Cc2cc(Br)cnc2-n2cccn2)C1=O C1(CNC(C2(CCNC(C(COC)C)=O)CCC2)=O)C2CCCCCC12 c1(C(N2C(C(=O)Nc3cccc(C#C)c3)C3CC3C2)=O)cc2cccnc2[nH]1 Cc1c(C(N2CC3CC2CN(C(C2(F)CCOC2)=O)C3)=O)oc2ccc(Cl)cc12 Cn1cc(NC(c2coc(C(F)F)n2)=O)c(C#N)n1.C12CC1CNC2=O C1(C(=O)NCC2CC(NC(C3(CC#C)CC=CCC3)=O)C2)COC(C)(C)CO1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)=C3CCCC3)C2)C)c(F)c1 C1(CNC(C)=O)CC2CCCC2N1C(c1cccc(OC)c1O)=O C=C(C)CCC(=O)N1CC(O)(C2CCCN2C(=O)CC(C)(C)SC)C1 N1(C(C2CCN(C(=O)C3CC3)CC2)=O)CCN(C(c2cnns2)=O)C(CF)C1 C1(C(=O)NC(CNC(c2cc3ccccc3o2)=O)CO)CCc2ncccc2C1 C1(NC(C=C(CC)CC)=O)CCCC(CNC(=O)CCCc2ccc(Cl)cc2)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(=O)Nc2ccc(S(C)(=O)=O)c(C)c2)CC1)OC n1(CC(=O)N(CCCNC(C(N)=O)=O)C2CC2)cc(Br)c(O)nc1=O C(CNC(C1CC2C=CC1O2)=O)(CC(F)(F)F)NC(CC(C)(F)F)=O C=CCCCCCC(=O)N1CCN(C(=O)CC(O)CN(C)C)CC1CCO C1(C(=O)NCC2(CC(F)F)CC2)CCCN(C(=O)Cc2ccco2)C1 c1(C(N2CC(CC(C)NC(CN3CCC(C)C3)=O)C2)=O)cc(F)n(C)n1 C1(Cn2cc(C3N(C(Cn4cc(C(C)=O)nn4)=O)CCC3)nn2)CCCCCC1 c1(C(=O)NC2C3CN(C(CCS(C)=O)=O)C2C3)cncc2ccccc12 CCC(C)C(O)C(=O)N(CCNC(=O)C(F)=C(C)C)CCOCCO.C(C)(C)(C)O CC1CCCCN(C(=O)C=CC(C)(C)NC(=O)CC2(O)CCC2)C1 N1(C(c2c(C)cccc2)=O)CC(C)N(C(=O)Cc2ccc(O)nc2)CC1C CCCC(CC(=O)NCc1nocc1CC)NC(=O)C(C)(C)C(=O)N(C)C Cc1cc(F)ccc1C(=O)NCCCCNC(C1COCC1c1ccccc1)=O CCCC(CC)CC(=O)N1CCC(CO)(NC(=O)CCCC#N)C1 c1(-c2nnc(NC(C3C(C)C(=O)C3)=O)s2)cccc(F)c1 N1(C(C(C(C)C)F)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C1CCCC1 Cc1ccn(C)c1C(=O)NCC(C1CC1)NC(=O)C(C)CF c1(OC)nsc(OC)c1C(c1nnnn1C1CCC1)NC(c1cc(C)no1)C C12(C(N3CC(NC(c4cnn(CCF)c4)=O)C3)=O)CCN(CC1)C2 N1(C(c2nc(C3CC3)cs2)=O)CCc2c(F)ccc(Br)c2C1 C(=O)(C(CCS(C)(=O)=O)OC)NC1C(NC(CC2CCC(CCCC)CC2)=O)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC2(NC(=O)C=Cc3cccn3C)CC2C1 C12(NC(C(=O)NC(C)C(c3ccccc3)N(C)C)=O)CC(C1)C(C(F)(F)F)O2 N1(C(C=C(CC)C)=O)CCCC2(NC(c3cn(C)cn3)=O)CC2C1 C1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)COCCN1C=O CC1CCCCC1(CNC(=O)C=Cc1ccncc1)NC(=O)CCc1cc[nH]n1 CCC(F)(F)C(C)(C)C(=O)NCC1CC(NC(c2ocnc2C(F)F)=O)C1 N1(C(C(c2ccnn2C)C)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 C1(C(N2CCC(F)(CNC(C(F)=C(C)C)=O)CC2)=O)Cc2ccccc2C(=O)O1 CN1C(=O)C(=O)N(CC(=O)NC2CC(CCNC(C3(C)CC3(F)F)=O)C2)C1=O c1(C(=O)NCC2(CNC(C=C(C)C3CC3)=O)CC23CCC3)cc2n(n1)CCO2 c1(C(C(=O)NCCC(C)NC(=O)C(C)(C)CF)O)ccc(F)c(Cl)c1 c1(C(=O)NCC2(O)CN(C(C3C4CCCC34)=O)C2)cncc(O)c1 c1(C(=O)NC2CN(C(CCOCC#C)=O)C2)cncc(SC)c1 C(C1=NOC2OCCCC12)NC(=O)NCc1nnc(CC)o1 c1(C2CN(C(=O)NCc3nc(CC)c(C)s3)C2)ccnc2ccccc12 Cc1cc(CCC(=O)NCCOCC(=O)Oc2ccccc2)cc(C)n1 C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(=O)CS(N)(=O)=O)C1 Cc1nsc(C(N2CC=CC(NC(c3ccc(C(F)F)nc3)=O)C2)=O)c1N N1(C(C2C3N(C(C(c4ccn(C)n4)C)=O)C(CC3)C2)=O)CCCCC(C)(F)C1 c1(C2C(C(=O)OC(C)(C)C)C2)ccc(Cl)c(Cl)c1.c12n[nH]cc1C(=O)N2 c1(C(=O)NC2CC3CN(C(C(CC)(CC)CO)=O)C2C3)cc(=O)n2ccsc2n1 c1(C(N(CCCNC(CC=C=C)=O)Cc2cccnc2)=O)cccc(CC)c1 c1(C(C)C)ccc(O)c(C(N2CC3C(NC(C4CCCCO4)=O)C3C2)=O)c1 c1(C(N2CC(CCNC(C(CC(=O)OC)C)=O)OCC2)=O)ccc2ccoc2c1 Fc1cc(CNCC2CC23CCOCC3)cc(Br)c1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)C3)C)CCC2)=O)ccc2cnnn2c1 C(CCC(C)(C)C)(c1nnnn1C(C)C)NCc1cnn(CC)c1C c1(NC(c2ccccc2C(F)F)=O)ccc2c(C(=O)NC3CC3)ncn2c1 Cc1cc(=NC(C)C2CN(C(c3nccc4[nH]ccc34)=O)CCO2)[nH]c(C)n1 c1(NC(C(N2CCC(C)(C)C(c3ccccc3)C2)=O)=O)c[nH]c2ccc(F)cc12 C(=O)(CCNC(c1ccsc1)=O)N(CCNC(=O)C=C1CCC1)CC C1(CC#C)(C(=O)N(C)CCN(C)CCO)CCN(C(=O)CN2CCC(C)C2)C1 C(=O)(C#CC1(CC)COC1)NC(CC#CC)C(=O)NC1CCC(=O)NC1 n1(CC(=O)N(CC(C)N(C)C(c2cc(=O)n(C)o2)=O)C)cnc2sccc2c1=O N1(C(C2N(C)CCC2)=O)CCN(C(CNC(c2cn(C)cn2)=O)C(F)(F)F)CC1 C(CN=c1nc2sccc2c(NCCOCCOC)[nH]1)OCCCC CCC(C)C(C(=O)NCC1CC1CNC(=O)C(C1CCCCC1)F)N(C)C C(=O)(C(O)CC(N)=O)N(CC(C)NC(c1n(CC)nc(C(C)C)c1)=O)C CCCC(CNC(c1cc(C2CC2)[nH]n1)=O)C(=O)NCC(C1CCC1)OCC N1(C(Cn2nnc(C)n2)=O)CC(O)CC1CNC(c1cc(Br)n(C)c1)=O CN1CCCC1C=CC(=O)NCCC(O)CNC(=O)CC1CCN(CCF)CC1 c1(C(=O)NCC(CN(C(c2ccc(C#C)cn2)=O)C)O)ccc2nccnc2c1 C1(C(N(CCOC)CCOC(C)=O)=O)COCC1C(N)=O.C1CC(=O)N1 c1(NC(=O)NCCC(=O)N(CC)CC)nc(Cl)c2ccnc-2[nH]1 C1(C(=O)NC(COC)C)CC12CN(C(C1CCN(C3CCSC3)CC1)=O)C2 N1(C(C2C(CC)N(C(=O)CC(C)(C)C(F)F)CCC2)=O)CCCC(C2CC2)CC1 Cc1cc2[nH]c(CN3CCn4c(C5CC5)nnc4C3)cc(=O)n2n1 C1(CC)CC(CC(=O)NC2CN(C(C3(C)CCCC3)=O)CC2C)CCO1 N1(C(C(CC#C)C2CC2)=O)CC(C(=O)NC2CC(O)C(F)C2)C(F)(F)C1 N1(C(C(CC)NC(N)=O)=O)CC(C2(NC(c3nccc(OC)c3F)=O)CC2)C1 c1(C(N2CCN(C(CCNC(C)=O)=O)CC2CCO)=O)[nH]nc2ncccc12 Cc1c(C(=O)N(CC(O)CNC(C2CC2c2cccc(O)c2)=O)C)c(Cl)nn1C Cc1cc2c(NC3CCN(C(=O)CN4C(=O)CSC4=S)CC3F)ncnc2[nH]1 C1(CN(c2nc(C(C)(C)C)ns2)C)CCCN(C(=O)COc2cccc(Cl)c2)C1 C1(NC(C=C(C)C)=O)COC2(CCCN(C(c3cc4cc(Cl)ccc4[nH]3)=O)C2)C1 O=C(N=c1nc(Cl)[nH]s1)N=c1ccn(-c2ccc(F)cn2)[nH]1 Cc1ccc(N)c(C(=O)NCC2(CNC(C3(C)CC3F)=O)CC2)c1F C1(C(=O)NCC2N(C(Cc3nn(C)c(Cl)c3)=O)CC2)CCc2ccnn2C1 Cc1cn2cc(C(=O)NC(CNC(C3COC4(CCC4)C3)=O)C3CCC3)nc2s1 C12(CNC(C(C)(C)n3cnnn3)=O)CC1CN(C(=O)CCc1ccncc1)C2 C(CC1CCc2ccc3c(c21)CCO3)NC(C1CCC2(CN(C(CC)=O)C2)O1)=O c1(CC)ccccc1C1CC1C(N1CC(OC)C(NC(=O)C(CC)OCC)C1)=O c1(OC)ncc(Br)c(=NC(=O)C2CC3CC3N2Cc2occc2C)[nH]1 N1(C(CCc2n(C)cnn2)=O)CC(CNC(c2ccc(F)s2)=O)CC1(C)C N1(C(CC2(COC)CCOCC2)=O)CCC(COC)(NC(C2(C)CC2F)=O)CC1 C1(CNC(Cc2n(C)ccc2)=O)C2CN(C(=O)CCNC(C3CCCO3)=O)CC12 C(CCCCC(=O)NCC12CCC(F)(CC1)C2)N(C(=O)C(O)C1CC1)C Cc1cn2c(C(=O)NCC3CCCCN(C(C4C5CCCC45)=O)CC3)cnc2s1 c1(NC(C(C)S)=O)cncc(C2=CCC(C(F)(F)F)CC2)c1 C=C=CCCC(=O)N1CCC(N(C(=O)CSC(F)(F)F)C)C1 N1(C(c2c(CC)nccc2)=O)CC(NC(c2cnoc2C2CC2)=O)CCC(O)C1 Cc1nc(O)c(C(=O)NCC2CCCCN(C(C3(CF)CC3(F)F)=O)C2)nc1C N1(C(c2c(CC)c[nH]c2)=O)CC2CC(C(=O)NC(C)CC3=CCCCC3)C(C2)C1 N1(C(C=CC(C)(C)C)=O)C(CNC(C2(C)CNC(=O)C2)=O)CC2CCCC12 N1(C(=O)CCC2CCN(C(=O)COCCCOC3CCC3)C2)CCC2CCCC12 O=C(N=c1ccnc2[nH][nH]cc1-2)C1C2CCC(C2)N1C(c1c(Cl)cccc1Cl)=O c1(C(=O)NCC2CN(C(CC(C)C)=O)C(C)C2)cnc2c(c1)N(C)CCO2 c1(C(N(C2CC(C#N)C2)CC(=O)NCC(CC)(C)COC)=O)cc(C)ccc1F C1(C(=O)NCC2CCCCCN2C(c2ccc(Cl)cc2)=O)(OC)CCC12CCC2 Cc1ccccc1C(=O)NCCOCCC(=O)NCC1CC1 CC1(C(=O)NCC2(F)CCN(C(=O)C(F)=CCCF)C2)CCCNC1=O C(C(CC(C)C)C(=O)NCC1CC2CCC1N(C(=O)Cc1cncnc1)C2)OC Cn1ncc2c(NC3CCCC3CNC(=O)CCn3ccccc3=O)ncnc12 C1(N(C)C(C2(CNC(c3ncncc3N)=O)CC=CC2)=O)CC2CCC1O2 CCCCC(O)C(=O)N(C1CCCC1NC(=O)C(c1ccc(Cl)cc1)=O)CC C1(CNC(c2cnc(C)[nH]c2=N)=O)CC2CCC(C1)N2C(=O)C(F)CCC(C)C C(C(C)(C)CC(=O)NC1(CN(C)C)CCC1)NC(C1CCN(C)CC1)=O C(=O)(CS(=O)(=O)C1CC1)NC(C)CC1CN(C(=O)CCS(C)(=O)=O)C1 N1(C(Cn2c(C)ncc2)=O)C(C(N2CCC2C(N)=O)=O)CCC1C CC1CCC(CC(=O)NC2C3CC2N(C(=O)CN(CC(C)(C)C)C)C3)CC1C C1(=CC(N2CC3(N(C(c4ncc(C)cn4)=O)CC3)C2)=O)CCOc2ccccc21 N1(C(c2c(COC)noc2)C(=O)Nc2ccc(Cl)cc2F)CCCC(F)(F)CC1 CCCCC(CC)CC(=O)NCc1ccccc1CNC(C1(O)CCCC1)=O C1(CNC(C(C2CC2)OCC)=O)CC2(CC2)CN1c1ccnc(C)n1 c1(CNC(COC)(CC2CCOCC2)c2nnnn2C)cc([N+](=O)[O-])ccc1C C1(C(=O)NCc2ncc(C(F)(F)F)[nH]2)CC2(C1)C(C(=O)O)C21CCC1 C(=O)(C1=NOCC1)NC(C1(CNC(=O)CCCn2cccc2)CC1)C C1(N(C(Cn2c(CCC)ncc2)=O)CC)CCCN(C(C2CSCCS2)=O)C1C c1(C(=O)NCCN(C(C23CC(CO2)C3)=O)CC)c2ccccc2cc2ccccc12 C(=O)(C(CCc1cn[nH]c1)OC(C)=O)OC.N12CCCC(C1)NC2=O c1(C(C(=O)N(CC(C)N(C)C(c2ccc(CO)o2)=O)C)(F)F)cc(Cl)ccc1Cl c1(-c2c(C(=O)NCCCN(C(=O)C(C)=C3CCC3)CC)nco2)ccc(C)cc1 c1(C(=O)OC)c(C)noc1NC(C1CC(O)CN1C(c1cc[nH]n1)=O)=O C(=O)(CCCCN1CCOCC1)NCCC1CN(C(CN(CCC)C)=O)C1 C1(C(N2C3C(CNC(CC(C)n4ccnc4)=O)C(C3)C2)=O)CCOCC12CCC2 c1(CCNC(=O)NCCC2CCCSC2)cccc2[nH]ccc12 c1(CC(=O)NC2CCCN(C(CC3CCC(=O)NC3)=O)C2)cc(F)ccc1Cl N1(C(c2c(C)nc(N(C)C)s2)=O)CC(C2(NC(=O)COC(C)(C)C)CC2)C1 c1(NC(C2CC(NC(c3cc(C(C)C)no3)=O)C2)=O)cnccc1[N+](=O)[O-] c1(CCOC)nc(C(C)NC(c2ccccc2C)=O)n(-c2cnc(C)s2)n1 C(=O)(C(C)(C)C(F)(F)CC)N1CCC(C(C)NC(CCC(CC)OC)=O)CC1 C1(C)(CC)CC(C(N2CCC(C)C(CN=c3[nH]nc(O)s3)C2)=O)CCO1 C1(c2nnnn2-c2ccccc2)(NC(CCCC=C)C2CC2)COC2(COC2)C1 C=CCC(F)(F)C(=O)NCC1CC(C)N(C(c2ccoc2Br)=O)C1 Cn1c(=O)c2cc(C(=O)NC3CC3c3ccc(Br)c(F)c3)n(C)c2n(C)c1=O CCCC(C(=O)N1CCCC(Cn2cc(CN(C)CCO)nn2)C1)C(=O)O N1(CC(=O)Nc2nc(-c3ccc(Cl)cn3)cs2)CCCSCC1C1CC1 C12(OC(C3CCOC3)=O)C3C4C1C1C2C3C41C.CCC1CCC(=O)OCC(=O)O1 C(C)(CCCNC(C1(COC)CCOC1)=O)NC(C1C(=C)C1)=O c1(C(=O)NCCCCCN(C)C(c2c[nH]cc(Cl)c2=O)=O)ccn2nnnc2c1 C1(CNC(Cn2c(C)ccn2)=O)CC(C(C)C)CCN1C(=O)C(C)NC(N)=O c1(C(C(=O)NC2CCN(C(C3(C4CCC4)CC3)=O)CC2)O)ccc(F)c(Cl)c1 N1(C(C2C(C(N)=O)COC2)=O)CCOCCC1C(=O)NC12CCC(CC1)C2 C1(N(C(=O)CNC(c2ccccn2)=O)C)CCCN(C(C2CCCNC2=O)=O)C1 C1(CN(C2(CC(=O)O)CCCCC2)C)CCCN(C(=O)CC2CC2C2CC2)CC1 C1(NC(C=CCC)=O)CC2C1CCN2C(=O)CCCc1cccc(C(F)(F)F)c1 C1(OC)(CNC(c2ccnnc2O)=O)CCN(C(=O)C2CC2)C1 Cc1cc(C(=O)NC2CCC(C(=O)NCC3CC4C=CC3O4)C2)ncn1 N1(C(c2c(C)n(C)cc2)=O)CC(NC(C2(C3CCCO3)CC2)=O)C2CCCCC12 C1(C(N2CCC(C)C(NC(C3(CC4CC4)CC3)=O)C2)=O)CC2(COC(=O)N2)C1 c1(C(NC(=NCC)NCC2(OC)CCCOC2)C)ccc(C)cc1SC c1(CCN(c2nnc(-c3ccco3)n2CC2CCCCO2)C)ccc(F)c(F)c1 c1(CC(N2CCC(CCCC3CCCNC3)CC2)=O)ccc(F)cn1 C(C(C(=O)N1CC(O)C(O)CO1)OC)NC(CC(CC)(F)F)=O C1(C(=O)NCCC(C)N(C(c2c(C)n(C)nc2)=O)C)CC2(CCCO2)C1 Cc1ccc(C)c(C(N2CCCC(NC(=O)C=Cc3ccccc3F)CC2)=O)n1 c1(C(N2CC3(C2)CN(C(c2cc(Cl)c(F)cc2F)=O)C3)=O)ccc2nn[nH]c2c1 N12Cc3cc(OC)c(cc3C1)O2.N1(c2cc(CC)on2)C(=O)OC2CNCC12 N1(CC(=O)NC(C2CCOC2)CNC(c2nn[nH]c2Cl)=O)C(=O)CCC1=O C1(C(N)=O)CC(O)CN1C(C1CSCCN1Cc1ccncc1Br)=O N1(C(c2ccc(N)c(OC(F)F)c2)=O)CC2OCCN(Cc3ccccc3)C2C1 C=C(C)C(C)(C)C(=O)N1CCCC(CCC)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC2(O)CCCN(C(=O)C(O)CF)C2)c1C C(c1cc(F)cc(F)c1)=CC(=O)N(CCCN(C(C1CC(C)OCC1)=O)C)C c1(C(=O)NCCC(C)NC(C(CC)F)=O)cc(C(F)(F)F)ccc1F c1(C(N(CC(C(=O)N2CC(CC(=O)OCC)C2)(C)C)C)=O)ccc(F)cc1F C#CCCN=C(NCc1oc(CC)nc1C)NCc1ccsc1Cl c1(C(=O)NC2C(CC)CN(C(c3nnc(C)s3)=O)CC2)cnc2c(Cl)cccn12 C1(C(N2CC(NC(c3ccc(CCF)cc3)=O)C2)=O)CCC2(CCC2)OC1 C1(C(=O)OC)(NC(c2ccc(F)c(N)c2)=O)Cc2ccccc2C1 c1(C(N2CCC(CNC(C(c3cn(C)nc3)O)=O)C2)=O)cnc2ccc(F)cn12 c1(OC)ccn2c(C(=O)NCC3(c4ccc(Br)cc4)CC3)cnc2c1 C=CC(C)(C)C(=O)NCC1CCCCC1NC(=O)CNC(=O)NCc1ccco1 C1(NC(CCOCCOCC)=O)CC(OC)C12CCC2.C12CCCC1CC(=O)N2 C1(C(=O)NC(C)CNC(c2cnoc2-c2cccs2)=O)CCC(=O)N(C2CC2)C1 CC12CC3(CCN3C(=O)NC1)C2.C1(OC)CCCC(c2ccccc2)CC1 C1(C(=O)NC(C)C(CO)NC(=O)C(O)C(C)C)(OCCCCCC)CCOCC1 CC1CN(C(C2(NC(=O)COC3CCC3)CC2C)=O)CCN1CCO c1(NC(=O)NC(CC)(COC)c2ccccc2)cc(OC)cc2ncccc12 N1(C(c2c(C)ccnc2)=O)CCC(O)C(NC(=O)Nc2cccc(Br)c2)C1 C1(CNC(c2ccc(C(=O)OC)cn2)=O)CCN(C(C2COCCO2)=O)C1(C)C Cc1cc(F)c(C(=O)NC(c2ccc(Cl)cc2Cl)c2ccccc2)c(F)c1 C(C)(C(=O)NCCC(C)CO)(N(C(C(C)OCC)=O)C)C1CC1 CCC(C)(C)C(=O)N1CC2CC1C2NC(c1c(C2CCCC2)noc1C)=O CC1OC(C)C(C)C1C(=O)NC(C1CCN(C(c2ncc(F)cn2)=O)CC1)(C)C c1(OCC)ncccc1C(N1CC(NC(c2ncoc2C)=O)C(C(F)F)C1)=O C(CN=c1[nH]c(N2CCCC3(CC3)C2)nc2cc(C)ccc12)(CC(C)C)OC C(=O)(CCCN(C)N=O)NC(CCC)CCCNC(c1ccc(C(C)O)cc1)=O C(C(F)(F)F)(C(F)(F)F)NC(c1cc(CC(C)C)on1)=O CC1(C)CC2CN(C1)C2.c1(CN2C(C(=O)NC(N)=O)CCC2)ccc(F)cc1F N1(C(c2cc(C)ns2)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 N1(C(CC2(NC(C(C)NC=O)=O)CCC2)=O)CC2COC(=O)C2C1 N(C1CCc2cc(CNC(C3CC3C)=O)ccc21)C(C(C)Cc1ccccc1)=O N1(C(C(CCOC)NC(C2(C#C)CCCC2)=O)=O)CC(C)(C)CCC1C CCC(CCc1ccccc1)C(=O)NC(C)CC(C)NC(=O)CN(C)C Cc1cnc(C(N2CC(C(F)(F)F)CCC2C)C(=O)NC(C)C)cc1Br C1(CNC(c2n(C)nnc2)=O)CCCCN1C(C1(c2cccnc2Cl)CC1)=O c1(CNC(C2(CO)CC2)C)cc(C2(C)CC2)on1 CN=c1[nH]cc(C(=O)NCCc2n[nH]cc2C(=O)NCC2(C)C=CCCC2)s1 n1(CC(N2CCN(C(Cc3cc(C)c(Cl)cc3)=O)CC2)=O)cc([N+](=O)[O-])nc1C C1(CNC(C2CN(C(C)C)C2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 CC(C)(C)CC(C)(C)C(=O)N1CC2CCC2(CNC(C2CC2C2CCC2)=O)C1 c1(C(CC2CC2)NC(c2ccc(Cl)s2)CC)nnnn1C1(C)CC1 C(=O)(C1=C(C)S(=O)(=O)CC1)N(C)CC1CN(C(c2cc(OCC)c(C)cc2)=O)C1 c1(C(N2CCC2CC2(CC(=O)NCn3cccn3)CC2)=O)csc(-c2ccco2)n1 N1(C(CC2CC(C)C2)=O)CCC2C(NC(=O)CN(C3CCCC3)C)C2C1 N1(C(CCSC)=O)CCCN(C(c2cc(Cl)cnc2Cl)=O)CC1 CCC(C)CC(C(=O)NCc1cccc(F)c1F)NC(=O)CCSC C(=O)(C1=CCCN(C(c2ccc(O)nc2C)=O)C1)N(CCCC)CCOC Cc1c(C(N2CCC(N(C)C(C3CCCSC3)=O)C2)=O)oc2c(F)cccc12 C(C1=NOC2CCCC12)NC(C1C(C)N(C(c2ns[nH]c2=O)=O)CC1)=O Cc1nccc(C(=O)N(CC(C)(C)C(=O)NC2COCC2N(C)C)C)n1 C1(C)(CNC(C(N2CC(C)(NC(=O)OC(C)(C)C)C2)=O)=O)COCCO1 N1(C(C2C(OC)C2)=O)CC(NC(c2csc(-c3ncccn3)n2)=O)CC12CCC2 C1(COC(c2nc(C(N3CCCC3)C)sc2)=O)CCOCC12CCC2 c1(C(=O)NC2CN(C(C(CC)NC(C)=O)=O)CC2C)cnn2c1CCC2 c1(CC)c(C(=O)NCC(CNC(c2cc(C3CC3)sn2)=O)OC)cnn1C c1(-n2cc(C(CC(N)=O)NC(C3(C)COC3)=O)nn2)ccc(Br)cc1 C1(C)(NC(CCCOCCC)=O)CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)C1 CC1CCC(CNC(=O)Cn2ncnn2)N(C(=O)C=Cc2cnn(C)c2)C1 CC12CC(C(N3CC4C(CNC(C5CC(F)C(=O)N5)=O)C4C3)=O)(C1)C(C)(C)O2 N1(C(CSC)=O)CCCC(N(C(=O)CN(C2CCCCCC2)C)CCF)C1 c1(-c2c(C)ccs2)nc(C2CSC2)nn1CCC(F)(F)F N1(C(Cn2c(C)nnn2)=O)CCC(C)(CC(=O)NC(C)CC2(O)CCC2)C1 N1(C(C2(C=C)CCC2)=O)CC2CC(C(=O)N=c3ccn(C4CC4)[nH]3)C(C2)C1 c1(C(N2CC(C)(C)C(NC(=O)COC3CCCC3)C2)=O)cnc2[nH]ccnc1-2 N1(C(=O)C(F)=C2CCC2)CCCCC1C1CCCN(C(=O)C(O)C2CC2)C1 N1(C(=O)C=Cc2ccco2)CCN(C2CCC(NC(=O)Cc3ccco3)C2)CC1 N(C(=NCCC(=O)N(C)C)N1CCC(C(C)OC)C1)CCS(=O)(=O)NC C12(F)CCN(CC1)C(=O)C(C)(C)CCOC2=O.C1(N(C)C(C)=O)(CC)CCC1 c1(C(=O)NC2C(C)(C)C(CNC(c3cn[nH]c3)=O)C2)sc(C#N)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(c1nn[nH]c1C(N)=O)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CCC(C)NC(=O)CC1Cc2ccccc2O1)C C1(C(N(CCN(C(C2CCN(C)C2=O)=O)CC)CC)=O)CCOC2(CCCC2)C1 C#Cc1ccc(C(=O)NCC(c2ccccc2)CNC(C2CC2CC)=O)c(C)c1 N1(C(C(CC)C)=O)CCC(O)(CCNC(=O)CCc2cn(C)nc2C)C1 C1(C(N2CCC(=CCC)C2)=O)CCCCCN1C(C1CN(C(=O)NC)C1)=O CC(C(=O)N(C)Cc1ccc(Br)cc1)C(F)(F)F N1(C(c2c(C)c(Cl)ccc2)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)C1)=O)C3 N1(C(CCCCOC)=O)CCOC(C)C1C(=O)NCC1(C)CC(C)=NO1 c1(C(=O)NC2CN(C(C3C(SC)CCC3)=O)C2)c[nH]c(=NC2CCOCC2)cn1 N1(C(c2n(C)ncc2Cl)=O)CCC(C(=O)NC2(C)CCOCC2)CC1(C)C C1(O)(c2cn(CC(CNC(C(C)CC3CC(F)(F)C3)=O)(F)F)nn2)CCOCC1 C(=O)(C#CC1CCOC1)NC1C(Cn2cc(-c3cccc(N)n3)nn2)C1(F)F Cc1[nH]c(=NCc2cc(C3CC3)no2)sc1C(=O)Nc1ccc(Cl)cc1C(N)=O c1(C(=O)NCC(C2CC2)NC(C(CC=CC)CC)=O)cc2c(C)n[nH]c2cn1 C12(NC(C#CC(C)(C)C)=O)CCOCC1CN(C(C1(c3ncco3)CCC1)=O)C2 Cc1ccc2c(C(N3CC4(CCC(CNC(=O)COCCOO)O4)C3)=O)n[nH]c2c1 N1(C(CCC2(NC(C3C(C)OCC3)=O)CCC2)=O)CC2CSCC2C1 c1(C(N2CCC(NC(=O)CSC(F)F)(CF)C2)=O)c(Cl)ccc2ccncc12 c1(C(CC(=O)NCCC(C)NC(c2cnn(C)c2C2CC2)=O)C)ccc(F)cc1 c1(CC(=O)NCC(C)(CO)NC(C=C(C)C(C)C)=O)cc(C)sc1C N#Cc1cc(C(N2CC3CC(C2)C3(F)F)=O)c(O)nc1S c1(N(CCOCC=C)C)cc(C)c(S(=O)(=O)NCC2CC(C)(C)CO2)cn1 C1(NC(=O)NC2CC(c3cn(C)nc3)OCC2)CCc2c[nH]nc2C1 N1(C(C2N(C)CCOC2)=O)CCC2(CCCN(C(c3cc[n+]([O-])cc3)=O)C2)CC1 CC1Cc2cc(CC(=O)NCC3CC(NC(=O)C(F)(F)CO)C3)ccc2O1 N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCCC2(C)CCOCC2)C2(CC2)C1 Cc1ccc2c(C(=O)NC3CN(C(C4COC(=O)O4)=O)CC(C)(C)C3)c[nH]c2c1 c1(-n2ncc(C(N(C3CN(C(c4cn(CC)nn4)=O)C3)C)=O)n2)ccc(C)cc1 N1(C(CCC#C)=O)CC(CNC(=O)CSCCc2ccccc2)OC2CCCC12 N1(C(c2cc(OCC)no2)=O)CCC(O)(C(C)NC(=O)C(CC)SC)CC1 c1(CCNC2CCC(O)C2)ccc(Br)cc1 c1(C(=O)NC2CCC(NC(c3c(C)nc(CC)o3)=O)C2)cncc2ncccc12 C(=O)(C(CC=CCl)c1ccccc1)NCC(CNC(=O)Cc1nonc1C)OC C(=O)(CCCC(C)NC(C1CCC2CC12)=O)NCC(C(C)C)(C)C N1(C(c2n(C=C)nnc2)=O)CCCCC2(CCN(C(c3nccnc3C)=O)C2)C1 Cc1cn2c(n1)C(C(=O)OC(C)C(=O)NC(c1cccnc1)C)CCC2 C(=O)(C(C)(C)C(N)=O)N1CC(OC)C(C(N2CCC(C)(N(C)C)C2)=O)C1 c1(C(N(CC(C)(C)CNC(c2cnn(C)c2F)=O)C)=O)c(F)ccc(F)c1Cl c1(C(=O)NC2CCCC(N(C)C(c3cc(F)n(C)n3)=O)C2)cncc2n[nH]cc12 N1(C(c2cccc(C#N)n2)=O)CCN(C(=O)CSCC(F)(F)F)C2(CCC2)C1 C12C(NC(=O)C(O)C(C)C)CCN1C2=O.c1(CC)ccnc(OC2CCC2)c1 C1(CNC(CC2CC(=C)C2)=O)CC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(CNC(=NCCC=C)NC2CC(OC)C23CCC3)ccc(S(N)(=O)=O)cc1 C1(CC(=O)NCC(CC=C)NC(C2(C)CCCCO2)=O)CCC2(CCCC2)CC1 C(=O)(C(C)(C)CCNC(C1C2CCCCC12)=O)NCc1cc(C)ncn1 C(C)(CCCCNC(=O)Cn1nnc(C2CC2)n1)NC(c1n(C(C)C)ccn1)=O c1(C(=O)NC(C2CCCN(C(=O)Cc3ccccc3)C2)C)c(F)cc(O)cc1F C1(NC(=O)Cn2cccn2)CCC2(CC1)CN(Cc1ccc(F)c(Cl)c1)C2 C1(NC(CC(C)OC)=O)CC2(C1)CN(C(=O)CCNC(C1CCCO1)=O)C2 CC1CCN(Cc2ccccc2SCc2ccccc2)CC1c1ccc(O)cc1 Cc1nnccc1C(=O)NC1CC(F)(C(=O)NC2(c3ccc(Cl)nc3)CC2)C1 Cc1ncnc(C)c1CC(=O)NCC#CCNC(c1ccc(N)c(Br)n1)=O c1(C(=O)NCCC2CCN(C(Cc3cn(CC)nn3)=O)C2)c(SC)cnn1C C1(N(C)C)CN(C(=O)Cc2cccc(Cl)c2)CC1CNC(C1CCC(O)CC1)=O C1(NC(C=C(CNC(CSCC)=O)C)=O)CC2CC1OC(=O)N2 N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CC2(C)CCC2)CC(C)(F)C1 N1(C(CC=C)=O)CC(NC(=O)CCNC(c2cc(C)nn2C)=O)CC1C N1(C(Cc2cnc(C)s2)=O)CCC(CO)C(NC(c2sc(C(C)C)nc2C)=O)C1 C(C1(O)CCc2ccccc21)NC(CC(C)C)c1nnnn1Cc1cccs1 c1(C(N2C(C(C)NC(C3(C(F)F)CC3)=O)CCC2)=O)n[nH]c2ccccc12 c1(C(=O)NCC(CC)NC(c2coc(Cl)c2)=O)sc(N(C)C)nc1C c1(C(N2CC(OCCNC(c3cc(OC)no3)=O)C2)=O)cc(Cl)cc(Cl)c1F C1(CN(C(C2N(CC)CC2)=O)C)COCCN1C(c1nc(C)sc1C)=O C1(NC(C(=O)N(C)C)=O)C(CNC(c2ncc3[nH]ncc3n2)=O)CCC12CCC2 N1(CC)CCN(C(=O)Cc2cccc(OC(c3ccncc3)=O)c2)CC(O)C1 c1(COC)nc(C)cc(=NC2CN(C(=O)CC3CCCNC(=O)C3)CC23CCC3)[nH]1 N(C(=NCCCF)N1CCC(C2CCC2)C1)Cc1scc(C)n1 c1(NC)ccc(C(C)(CN(CC(F)(F)F)CCSC)NCc2ccccn2)cc1 CC1CCN(C(=O)CC(C)(C)O)CC1CC(=O)NCc1nnc(O)o1 c1(C(=O)NC2C(CNC(C3CCC(C)C3)=O)CCC2)cc2c(cn1)CCCC2 C1(C)(C(=O)NC(CC(C)C)CNC(=O)CCc2cnn(C)c2)CCS(=O)(=O)CC1 Cc1cc2ccc(C(=O)NC3CN(C(c4cc(Cl)c5n[nH]cc5c4)=O)C3)cc2o1 N12CCC(CC1C)n1cc(nn1)C2.c1(-c2cc(C)nnc2)cc2sccc2[nH]1 C=CCCC(C)(C)C(=O)NCCC1CCCCN1C(=O)C(C)OC C(c1c(Cl)nc2ccc(Br)cn12)=Cc1c(C)ccc(C)c1 Cc1cccn2cc(CC(=O)OCC3(C)CC3Br)nc12 O=C(O)CC=CCNC(=O)NC1CC1(F)Cl C(=O)(C(CO)C(C)(C)C)NCCN(C(CSc1ccc(C)c(C)c1)=O)C N1(CCCNC(CN2CC(C)(C)C2)=O)CCN(C(c2sccc2F)=O)CC1 CC1CCCC1(C(=O)NCCOC(=N)O)NC(c1cc[nH]c1C1CC1)=O n1(CCC)ncc(C(=O)NCCC2(O)CN(C(c3cccc[n+]3[O-])=O)C2)c1Cl Cc1nccnc1-n1cc(CC2CCCN(C(=O)C(C)Cc3cnn(C)c3)C2)nn1 c1(C(N2CCC(C3N(C(C(CC)F)=O)CCC3)C2)=O)ccnc(C2CC2)n1 CCC(C)C(O)CC(=O)NC(C)(CNC(=O)CSC(C)(C)C)Cn1cccn1 N1(C(C2(C#N)C(C)C2)=O)CC(C2(NC(=O)C=CCF)CC2)C1 C=C1CC2(C1)CC(C(=O)NC1CN(C(c3ccc(Cl)nc3OC)=O)CCC1C)C2 c1(-c2cn(CC(=O)NCc3c(C)nc(C)o3)nn2)c[nH]c2nccc-2c1 C1(O)(CNC(c2cnc(O)o2)=O)CCCN(C(=O)C2=CCCS2)CC1 c1(CC)nc2c(C(N3CCCC3(C)CNC(=O)CS(C)(=O)=O)=O)ccnc2[nH]1 C(C(=O)NC(c1nc(C(N2CCCC2CNC(N)=O)=O)co1)C)(C(C)C)SC CCC(O)C(C)(C)C(=O)NCCCN(CCO)C(c1cc(C(=O)OC)ccn1)=O c1(CCC(=O)NC2C(CNC(Cc3c(C)ncs3)=O)C2)c(C)n[nH]c1C N1(C(C(CCC#C)O)=O)CCCC(C2CN(C(c3ccnn3CC#N)=O)C2)C1 N#Cc1cccc(CNC(=O)Nc2nc(C(F)(F)F)cs2)n1 C1(N(C(CCN(C(c2cscn2)=O)CC)=O)C)CCCCCCC1 CC1(C(=O)NCc2cccc(O)c2)CC(O)CN1C(=O)CN1CCCCC1 CC1(C)OCC(c2cn(CCCC(=O)NCCN3CCC(CC#N)C3)nn2)O1 c1(C(=O)NCC2CCN(C(CCCCSC)=O)CC2)cccc(SC)c1O C1(C(N2CCC(CC)OCC2)=O)COC2(C1)CN(C(c1coc(C)n1)=O)C2 C1(C(=O)OC)CCOC1C(=O)NC1(CNC(C2(N(C)C)CC2)=O)CCOC1 C1(CNC(C2(CC(C)C)CC2)=O)C2CC1N(C(c1cncn1C(F)(F)F)=O)C2 c1(OC)ccc(CN2CC3C(C2)N3C(C2CCC(=O)NC2)=O)cc1C(C)C C(=O)(CC(C)(C)CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)SC)OC.C(=O)NCC N1(C(c2c(C)[nH]cc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(Br)o2)C1 c1(C(=O)NC2C(NC(=O)Cc3ccnc(Br)c3)CC2)n[nH]c2c1CCCC2 c1(OCC(=O)N)ccccc1.C(=O)(C(C)C1CCCO1)NCCNC(C)=O.C1CO1 C#Cc1cc(NC(C2CCOCCN2C(c2cc(O)cc(F)c2)=O)=O)cc(F)c1 CC(C(=O)NCC(O)CNC(C1OCCCC1(C)C)=O)S(=O)(=O)C1CCOCC1 c1(C(N2C(COC)CN(C(=O)C(C)(F)C(=O)OC)CC2)=O)ncn2c1CCCC2 C(=O)(C1=CS(=O)(=O)CCC1)NCCCCC(C)NC(=O)C(S(C)(=O)=O)C1CC1 C(=O)(CC(C)(C)COC)NCC1CC(NC(C(C=C)c2ccccc2)=O)C1 c1(CC)ccc(C(N2CC(C)C2C(=O)NC(C)Cc2cn[nH]c2)=O)cn1 Cn1nnc2ccc(C(=O)NC3CC(C)(NC(=O)C=Cc4cccs4)C3)nc12 CC(C)CCC(O)C(=O)N(C)CCOCCCNC(c1ccc[n+]([O-])c1)=O c1(C(=O)NCC2N(C(C(C)OCOC)=O)CC(F)C2)cc2cccnc2cc1F C1(C(=O)NC(CC(=O)NC)C)(CF)CCN(C(C2CCCN2C)=O)C1 Cc1ccc(F)c(CCC(=O)NC(C2CCCC(C)C2)C(=O)O)c1 C(=O)(C(C)CN(C(=O)CCCN(C)C(C1CCCN1C)=O)C)OC CCCCC(COC)NC(=O)CCN(C(=O)CCc1ccn(C)c1)CCO c1(C(=O)NC2CN(C(C34OC(C)C(CC3)C4)=O)C2)cc(Br)c(F)cc1N c1(OC)cc(F)cc(C(=O)NCC2CCN(C(c3ccns3)=O)CC2C)c1N C1(CNC(C2C(CNC(=O)Cn3ccnc3)C2)=O)CC1C1CCC1 Cc1ccn(CC(=O)NC2CN(C(c3cccnc3)=O)C2)c(=O)c1 N1(C(CCN(C(=O)C(C(C)C)SC)CC)=O)CCOC2COCC12 C1(NC(C(C)c2ccco2)=O)CCCCN(C(=O)CN2CCC(F)CC2)C1 CCCCCC=CCC(=O)N(CC(=O)NC(C1CCOCC1)C)CC c1(C(=O)OC)cc(F)cc(S(=O)(=O)NC2CCc3cc(F)ccc32)c1 CCCC(C(O)C(=O)N(CCCO)C1CC1)NC(c1cc(C)nnc1C)=O Cc1nocc1C(=O)NCC(F)CNC(C1C=CCCC1)=O N1(C(c2ccc(Cl)nc2)=O)CC2CCN(Cc3cccc(O)c3)C2C1 CC1(C)CN(C(c2cc(NC(C3CC4CC4C3)=O)ccc2N)=O)CC1NC(N)=O c1(C(=O)NC(C2CCCC2)CNC(=O)C2=CSCS2)nccc2cccnc12 C1(NC(c2c(C(C)C)ocn2)=O)COC2(C1)CN(C(=O)COCC1CCOC1)C2 N1(C(C2(CCC)CC2)=O)CC2(C)CN(C(=O)CCCC(C)O)CC2(C)C1 c1(C(N2CCCC(C(C)(O)CNC(=O)Cn3ccnn3)C2)=O)ccc(O)c(Cl)n1 c1(C(=O)Nc2cnc3[nH]ncc3c2)nc2n(c1Cl)CCN(C(=O)CC(F)(F)F)C2 n1(C(CC)C)ccc(=NC(=O)C2C(C3CC3)CCN2C(c2cccnc2O)=O)[nH]1 c1(C(=O)NCCC2(O)CN(C(c3cnccn3)=O)C2)cc(Cl)c(F)cc1Cl C1(C(=O)NC2C(C)CN(C(c3ccc(F)c(Cl)n3)=O)C2)CCC2C(C1)C2(F)F CCC(CC(=O)NC(CNC(c1cn(C2CC2)nc1C)=O)C1CC1)C(F)F C(=O)(C(CC(F)F)N(C)C)N1CC2C(C(=O)NCc3ccc(OC)cn3)C2C1 C1(CC)CN(C(c2cnc(F)c(C)c2)=O)CCN1C(=O)CCc1ccccc1F c1(OCCC(=O)NC2CCC2NC(c2cc(C(F)F)no2)=O)ccc(F)cc1 N1(C(CC(C)NC(N)=O)=O)CCC(C2CCOCC2)(CNC(=O)C(C)(C)CF)C1 C(CSC)(C(=O)NC1CC(NC(=O)Cc2ccnn2Cc2ccccc2)C1)OC C(=O)(C(CO)C(F)(F)F)NC(C)CNC(c1ccn(C(C)(C)C)c1)=O c1(C(N2CCN(C(c3c(C)nsc3)=O)C3C2C3)=O)c(F)ccc2cnn(C)c12 c1(C(N2CC(O)(CCNC(c3cc(Cl)n[nH]3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C(c1ccccn1)=C(C)C(=O)NC1CC12CC(NC(=O)CC13COCC(C1)C3)C2 c1(OCC)ccc2c(c1)CC(C(=O)Nc1ccc(C=CC(F)(F)F)cc1)CO2 N1(C(=O)C2CC2)CCCC(N=c2[nH]nc(C3CC3)s2)CC1 C(=O)(C1CCCc2nc[nH]c21)NCC(CN(C(C1C=CCCC1)=O)CC)(C)C N1(C(CCOCC)=O)CCCC(CNC(C2(C)CC(C)=NO2)=O)CC1 C=C1CCN(C(=O)CC(CC)CC)C(C(=O)NCc2ccn(CC)n2)C1 C(=O)(CC(C)C(F)(F)F)NCC(CC=C)NC(=O)C(c1ccc(Cl)cn1)(F)F C1(CC#C)(C(=O)OC)CCN(C(c2csc(Cl)c2)C(=O)NCCCF)CC1 C1(n2c(C(C3COCCO3)N(CCOCCF)C3CC3)nnn2)CCCCCC1 C12(CC(N3CC(c4cc(COCC(=O)OCC)[nH]n4)C3)=O)CCC(CC1)OC2 S(=O)(=O)(c1ccc(C#N)cc1)N1CCC(O)(C(=O)Nc2cc(OC)nc(C)n2)C1 N1(C(C2C3CCC2CC3)=O)CCCC(C2CCCN(C(c3cnc(O)o3)=O)C2)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(c2ccc(C)cc2)F)CC1SC)OCC c1(C(C(=O)NCCCSC)N(C(C#C)C2CCC2)C)ccc(C#N)cc1 Cc1cc(-n2cc(C3(C)CN(C(C45CSCC4C5)=O)C3)nn2)cnc1Br c1(OC)cc(Br)nc(NC(=O)C(=O)Nc2ccc(OCC3CCCCC3)cc2)n1 c1(C(=O)NC2(CNC(C(C)NC(N)=O)=O)CC2)cc2n(n1)CCO2 c1(OC)ccccc1C1CC(O)CN1Cc1cn(C)nc1C1CC1 C1(C(N2CCC(CC#C)CC2)=O)CC2CN(C(=O)C(C)(C)C(N)=O)CC2C1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 c1(C(N(C)CC2(NC(=O)Cn3cnnc3O)CC2)=O)ccc(-n2ccnc2)cc1 C(=O)(C(C)(C)C(C)(C)CO)NCc1c(C(=O)NCCOCC(=O)OC)nco1 n1(Cc2nn(CCOC)c(C=Cc3c(C)noc3C)n2)c(=O)oc2ccccc12 c1(C(N2CC3CCC3(OCC(F)(F)F)C2)=O)cccc2oncc12 C1(CC)COCCC1C(N1CCC(CC)(CO)C1)C(=O)NC C1(C(N(C)CCNC(=O)C(c2ccccc2Cl)(C)C)=O)CC2(C1)CC(F)(F)C2 CCC(O)(CNC(=O)C=CC1CCCN1C(=O)C(C)C(F)F)CC N1(C(CCCCC#C)=O)CCCC2(C1)C(NC(=O)CC1CC=CCC1)CCN2C C=CC1(C(N2CC(CC(F)C(=O)NCCOC(=N)O)C2)=O)CCCCC1 C12(C(NOCCOC)=O)CC(CO)(CN1C(c1ccncc1Cl)=O)C2 C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(=O)CCc2nc[nH]n2)CCN1C N1(C(COC(=O)CO)=O)CC(O)CC1CNC(C1(F)CCCCC1)=O c1(CC(=O)NC2C(CNC(COCC#C)=O)C2)ccc(OCCOC)cn1 N1(C(C2C(C)CCO2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)C2(CC2)C1 C1(CC)CN(C)C(=O)CN1C(c1cc(CNC(=O)C(C(=O)OC)OC)no1)=O Cc1nc(N2CCC(NC(c3cnn(CC(F)(F)F)c3)=O)C2(C)C)c(F)c(C)n1 c1(C(=O)NCC2(O)CN(C(C3C(F)(F)C34CCC4)=O)C2)ccc2c(c1)NCCC2 CC1OC(C)(C)N(C(=O)OC(C)(C)C)C1CNC(C1CS(=O)(=O)C1)=O c1(CC)ccc(O)c(C(=O)NCC2CCC2NC(c2ccc(C(F)F)s2)=O)c1 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)N(C(C)C)Cc2ccco2)CC1 c1(OC)ccccc1C1CCCN1C(=O)CC1CC(=O)NC1=O N1(C(CNc2c(C)cccc2C)=O)CC2(CCCC2NC(=O)Cn2ccnn2)C1 N1(C(C2CCN(C)C2=O)=O)CCOCC(F)(CNC(=O)CSC(F)(F)F)C1 C1(C#N)(C(=O)NCCC2CCN(C(COCC(C)(C)C)=O)CC2)CC12CCC2 N1(C(C(=O)NCCCC(C)NC(=O)C=Cc2cccnc2)C)C(C)CCC1C c1(NC(C)(CNC(=O)COCC2CCC2)c2nn[nH]n2)cncc(C2CC2)c1 c1(NC(C(COC)NC(C2CCN(C)CC2)=O)=O)cnn(C(C)C)c1C c1(C(=O)NCC2(CC)CCCOC2)ccccc1S(=O)(=O)C(F)(F)F C(C1=C(C)CCC1)NC(c1nn(C)nc1Br)c1n(CC(=C)C)nnn1 C1(F)(C(N(CC(CN(C(C2(CC(C)C)COC2)=O)C)O)C)=O)CCOC1 c1(N2CC(NC(C(C)(F)F)=O)C(O)C2)ncnc2c1CCCC2 C(C(C)(C)C(=O)N(CCC(=O)NC(=O)CC(C)(C)C(F)F)OC)OC CCCCN(c1ccsc1)C(=O)CC1CCN1C(=O)C=C(C)C C1(CNC(c2cn(CC)nc2)=O)(COC)CCN(C(=O)C2=CCCS2)C1 N1(C(C(C=C)(F)F)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CCC2)CC1 CC1(OCC(=O)NCC2CC(NC(=O)CCc3nc[nH]n3)C2)CCCC1 Cc1cc(Cl)cc(C(N2CC(C)(NC(=O)CCNC(C3CCCO3)=O)C2)=O)c1O CC(CCC(=O)NCC1(O)CN(C(c2ccccc2C(F)F)=O)C1)S(C)(=O)=O c1(CC)ncncc1C(=O)NC1(C)CCN(C(=O)C(F)n2cccn2)C1 c1(CS(C)(=O)=O)nc(Cc2ccc(C(F)(F)F)cc2)n(-c2ccnc(Cl)c2)n1 c1(C(=O)NCC(CCOC)NC(C2CCN(C)C(C)C2)=O)ccc2c(c1)CC2 c1(-c2cn(C(C(=O)NC(c3ncc(C)s3)C)C)nn2)cnn(C)c1C c1(SCC)cc(C(=O)NC2CC(C)(OC)C2)c2c(c1)CCO2 N1(C(C)=O)CC(CN(C)C(c2ccccc2OC2CCCC2)=O)C2(CC2)C1 Cc1ccc(O)nc1CNC(C1CNC(=O)CN1C(=O)CN1CCC(C)CC1)=O C1(C(N2CC(O)(C(C)C)C2)=O)CCC2(CC2)N1C(C12CC1CNC2=O)=O c1(COCC(=O)NC2CC(F)(NC(C(C)SCC)=O)C2)ccc(OC)nc1 c1(CC)ccc(C(=O)NC(C(=O)NCC2(CO)CCC2)C2(C)CC2)o1 c1(C(C)N(CC(F)(F)C2CC2)C2CC2)cccc(C(F)(F)F)c1 c1(C(N(C(C)CNC(C2CCc3cncn3C2)=O)CC)=O)c(Cl)ccc(C)c1N c1(CC(=O)N(C2CCCC2)CCNC(CSCC)=O)ncn2c1COCC2 C1(CNC(C2(C=C)CCC2)=O)CN(C(=O)C(C)Cc2ccco2)CC1C Cc1cc(Cl)ccc1OCC(=O)NC(C)CCN(C)C(c1ccc(N)c(Cl)c1)=O c1(C(=O)NCCN(C(c2coc(Cl)c2)=O)C2CC2)ccc(OC(F)(F)Cl)cc1 N(C(=NCC1CCCCO1)NCC(C)(C)C(=O)NC)C1CCN(CC)C1 c1(NC(C)=O)cccc(NC(C2CC(C)N2C(=O)C#CC2CC2)=O)c1C C(C1CN(C(c2c[nH]c(=N)o2)=O)CC1C(N1CCC(C)(C(C)C)CC1)=O)=CC N1(C(CC2CN(C(C)=O)C2)=O)CCN(C(=O)CC2(O)CCOCC2)CC1C1CC1 CCCCC(CNC(C1CCC1CNC(c1ccc(O)nc1C)=O)=O)CC C(=O)(CC(C)P(C)(C)=O)NCCN(CCOC)C(C1CC(C)OC(C)C1)=O C1(C(C)NS(C)(=O)=O)(NC(C(C2CC2(C)Br)N(CC)CC)=O)CCCCC1 c1(C(=O)NC(CC=C)CNC(=O)CCCOC(C)C)cc(C(F)F)cc(F)c1 c1(C(=O)NCC(CNC(C(N)=O)=O)F)cnc2cc[nH]c2c1 C1(NCC(=O)NCC(S(C)(=O)=O)c2ccccc2)CCc2nnnn2C1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(C)C1CNC(=O)C=Cc1ccc(C)nc1 C(=O)(CCCCNC(=O)C(F)n1ccnc1)N(CC(C)O)CCO C1(NC(c2cccc(C(C)C)c2)=O)CC2CCC(C1)N2c1ncnc2[nH]ccc12 CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CCNC(=O)CCn1cncn1 c1(CC(=O)NCCn2cc(CN(C(C)C)C(C)C)nn2)c(F)cccc1Cl c1(C(=O)NC(CCC)CCCNC(c2ccoc2C)=O)ccc([N+](=O)[O-])cc1F CC(C#N)CCC(=O)NCC(O)CN(C)C(c1ccnc(-n2cccn2)c1)=O C1(CC(=O)NC(C#C)C2CCC2)COCCN1C(=O)C(C(C)C)OCC C12(C(=O)NCc3cc(CC)on3)CCCC1CCN2C(c1cnn(CCO)c1)=O C1(NC(=O)CC2(N3CCCC3)CC2)CN(C(=O)CC2C=CCCC2)CC12CCC2 C1(C(=O)NCc2c(C)nn(C)c2)CS(=O)(=O)CC12CC2 C(=O)(CC(C(C)CC)NC(C1(OC)CCSC1)=O)NCC(C=C)O C#CC(CC(C)(C)C)NC(C1(F)CCN(C(c2cc(C)n(C)n2)=O)C1)=O c1(CN(c2ncc(C(N(C)CC3CC3)=O)cc2Cl)CC(=O)O)cccc([N+](=O)[O-])c1 C1(CNC(COCCC=C)=O)C2CC2CN1C(C1CC1C(=O)OC(C)(C)C)=O c1(CC)oc(C)cc1C(=O)N(C(C)(C)CC(=O)NC(c1nccc(O)n1)C)C N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(C3CC(SC)C3)=O)CC12 C1(C(N2CCC(OCC)C2)=O)C2CCN(C(C3OCCC3(C)C)=O)CC12 C12(C(=O)NC(CN3CCN(C(C=NOC)=O)CC3)C)CCCN(CCC1)C2 c1(C(C)C)cccc(F)c1C(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1 CC1CCCC(C(=O)NC2CCC(N(C)C(c3nccnc3N)=O)CC2)CC1 Cc1oc(Br)cc1C(N1CC=CC1CN(C(=O)COC1CCOCC1)C1CC1)=O N1(C(c2cccc(OC)c2)C(=O)NCC=C)CCC2C(C1)C2(F)F C(CCCCCC(=O)N1CC(O)C(O)C1)NC(C(C)(C)c1ccno1)=O c1(OC)ncc(C(N2CCC(C)(N3CCOCC3)C2)C(=O)NC2CCOC2)cn1 N1(C(=O)NC)CCCC1C(=O)NCC(CNC(c1cc(C(C)C)[nH]n1)=O)CO c1(C(c2n(CC=C)nnn2)NCC2CC=CC2)cnn2cc(Br)cnc12 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(c2sc(SC)cc2C)=O)CCC1C c1(C(=O)NC2CC(NC(C3C(C)CC3)=O)C2)ccc(CN2CCCC2)cn1 c1(C(N2CCN(CC(=O)Nc3ncc(OCC)cn3)CC2)=O)cn2c(n1)COCC2 N1(C(COCC#C)=O)CCCC(C2CN(C(c3ccc(O)cc3F)=O)C2)C1 c1(C(N2CC(C)C(NC(C3CC34CCC4)=O)C2)=O)n[nH]c2cc(Br)ccc12 CN1N=C(CC(=O)NC2(C(=O)NCCC3CCC(C)(C)O3)CCN(C)C2)CC1=O C1(CNC(C2CCCC(C)(C)C2)=O)N(C(c2csnc2Cl)=O)CCCC1(C)C C(=O)(C(O)C1=CCCCC1)N1C(N(C(N2CCCC2CF)=O)CC)CC1C CC1CN(C(=O)COc2ccccn2)CC(C)N(C(c2cccc(=S)n2O)=O)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC23CCC3)ccc(=O)n2c1COCC2 CCCCC(CC)C(=O)N1CCOC(C)(CNC(C23CCC(C)(CC2)OC3)=O)C1 Cc1ccccc1-c1cccc(NC(=O)NC2CCC2CN)c1 C(=O)(C(C)C(C)COC)NCCN(CCC)C(c1cncc(N)n1)=O C1(C(=O)NCc2cncc(C(=O)NC(C)CCC3CC3)c2)CCCCC1(C)C C1(CNC(C(COC)C)=O)CCC2(CCC2)CN1C(=O)C=C1CN2CCC1CC2 C=CCC(C(=O)N1CCC(CCNC(c2c(N)cc(Cl)nc2Cl)=O)C1)C(C)C C1(CC(=O)NC(CNC(c2c(C(=O)OC)coc2)=O)CO)CCC(=O)NC1 C1(C(=O)OC)CCC(C(=O)OC)CN1Cc1cccc(OCCOC)c1 CC(C)CC(C(=O)N1CCC=CC1C(=O)NC1CCN(CCCO)C1)N(C)C N1(C(Cn2c(C)nc(C)n2)=O)CC2CC(NC(C3(S(C)(=O)=O)CC3)=O)CC2C1 N1(C(CSCC)=O)CC(CCNC(c2cnc(SC)nc2)=O)C(C)C1 C1(C(=O)NC2(C)CC(F)(F)C2)CCOCCN1C(C1CCC(F)(F)C1)=O C(C)(C(=O)NCC1CCCC1N(C)C)(C1CCC1)NC(C(C)=CC(C)(C)C)=O C1(C(N(C)CC2(O)CCCN(C(=O)CNC=O)C2)=O)CCC2(CCCC2)C1 N1(C(C2CC(C)(C)C2)=O)Cc2nccn2CC(NC(=O)CN2CCC(C)(O)C2)C1 N1(C(C2CC(C#C)(O)C2)=O)CC2CCC1CN2C(=O)Cc1cc(C)cs1 Cc1oc(S(=O)(=O)Nc2cc(Cl)nc(Cl)c2Cl)cc1S(C)(=O)=O N1(C(c2ccc(NC)cn2)=O)CCN(C(c2cc(C)cc(C)c2)=O)C(CCO)C1 c1(C(=O)NC2C(CNC(CCP(C)(C)=O)=O)CC2)cc(F)c(F)cc1Br c1(C(N(CCOC)CCNC(=O)Cc2cccc(F)c2)=O)cc2sc(C)nc2[nH]1 c1(C(N2CC(C)C(NCc3nncn3C)CC2)=O)cnn2ccncc12 c1(CC)ccc(C(F)(F)F)c(F)c1.c12ccc(s1)CN(C)C2C(=O)NC1CCOC1 N1(C(C(c2cncn2C)N(C)C)=O)CCC(C)(C)C(NC(=O)Cn2ccnn2)C1 c1(C(=O)NCC(=O)NCC2CCCN(C(c3cscn3)=O)C2)[nH]cc2c1CCC2 N1(C(c2cc(CNC(=O)CCc3csnn3)sc2)=O)CCOC2(CC2)C1 C1(NC(C=C(C)Cl)=O)CC1C1CCN(C(c2cccc3sccc23)=O)CC1 N1(CC=C)CCCN(C(=O)C(CNC(c2ccncc2)=O)CC2CCCC2)CC1 C#Cc1cc(C(=O)NCC2CCN(C(C3CC3F)=O)CC2(F)F)cc(Br)c1 CC(C)(C)C(C(=O)NC1CCN(C(C23CC4CC2C3C4)=O)C1)N1CCCC1 c1(C(N2CCCC(N(C(=O)CCc3cnn(C)n3)C)C2)=O)cc2cccnc2o1 C1(C(N(C(CC)C)C)=O)CCCCC1(C)NC(c1c[n+]([O-])c(C)cn1)=O C1(C(C)NC(c2c(CC)c[nH]n2)=O)CN(C(=O)C(c2cccnc2)C)CCO1 c1(N(C(C(C)NC2C3COCC23)=O)S(C)(=O)=O)cc(-c2ccccc2)nn1C c1(OC)cc(NC(=O)C(C2CCN(C(=O)CCC(C)SC)CC2)C)cc(OC)n1 N1(C(C2C(C)C(=O)C2)=O)CCOCC1CNC(c1ccn(C(F)F)n1)=O CC1(C)CCN(C(=O)CN(C2CCC2)C(C2CCCC23CCC3)=O)CC1CO CC(C(N)C(=O)NCCC1(C#N)CCCC1)C1CC1 C1(C(C)C)CN(C(=O)CSCC(F)F)CCC1NC(=O)C=Cc1cccnc1 N1(CC(=O)N(C2(CC(=O)NCc3occ(C)n3)CC2)C)CCCCC1=O N1(CCNC(c2cccnc2)=O)CCC(=O)N(Cc2cc(C(F)(F)F)ccn2)C1=O N#CC1(CC(=O)NCC(C2CCC2)NC(c2cccc(C(F)F)c2)=O)CCCC1 Cc1nsc(C(N2CCCC(CC(=O)NCc3ccnn3C)C2)=O)c1N c1(C(N2CC(CC)SCC2)=O)ccc(F)c(-c2cn(-c3ccccn3)nn2)c1 Cc1c(C(N2CC3CC(O)C2C3NC(=O)C2=CCOC2)=O)oc2ccc(F)cc12 C1(CNC(COC)=O)CC2(CCN(C(c3c[nH]nc3OC)=O)CC2)CO1 N1(C(CC2(CC=C)CCCC2)=O)CCCC(CCNC(C2CNC(=O)N2)=O)CC1 c1(NC(CC2(C(=C)F)CN(C(=O)OC(C)(C)C)C2)=O)ccc2c(c1)COC2 n1(Cc2cc(OCC)on2)c(N2CCC(OC)C2)nnc1-c1cnc(CCO)s1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(CCC2NC(C2CC(C)N(C)C2)=O)CC1 C(C(=O)N(C1CCCN(C(=O)N(C)C)C1)C)(C(C)C)SCC.C12CC(C1)NC2=O CCCC(C=O)C(=O)NCC1CCCC(CNC(C2CC2COCC)=O)C1 C1(OC2CN(C(C3(CC=C)CCC3)=O)C2)CCN(C(C2(C)CCCCO2)=O)CC1 C(=O)(CCCCCCCBr)NC(C1CCN(Cc2cc(F)c(F)cc2Cl)CC1)C C(c1cnc(O)nc1O)=CC(=O)NCCCCCCNC(C(C)CS(C)=O)=O CC(C)C(O)C(C)C(=O)N1CCC(CF)(NC(=O)CNC(=O)CN(C)C)C1 CCCN=C(NCC(C)CN(C)C)N1CCC(CSC)C1 N1(C(CCCc2onc(C)n2)=O)CC(C)(C)CC1CNC(c1ncccc1O)=O N1(CC(C)NC(c2nc(C(C)C)oc2)=O)CCN(C(=O)COC(C)(C)C)CC1 CCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CCN(C(C)CC(=O)OC)CC1 c1(C(=O)NC(CNC(c2cc(CCCO)on2)=O)CO)ccc(Cl)nc1O C1(N(C(=O)C=CC(=O)N(C)C)C)CCCN(C(=O)C(C)OC2CCCC2)CC1 N1(C(COC2(C)CNC2)=O)CCCN(CC(N)=O)CC1.C(C(C)(C)C)N(C)CC c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(C2(c3cc[nH]n3)CCC2)=O)CC1 N1(C(C#CC2(CC)CC2)=O)CCN(C(c2nc(C)c(C)s2)=O)C(C)CC1C N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(CNC(c3ccc(COC)o3)=O)(C2)C1 C12(CN)CCN(CC1)C2=O.c1(OCCOC)ccc(C2CCC2)cc1 c1(C(=O)NC(C(=O)NC(C)CC(F)(F)F)C2(O)CCC2)cc2cccnc2[nH]1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(C(N2CCC(C(CNC(CC(=C)C)=O)O)CC2)=O)ccc(NC(C)=O)c(F)c1 N1(CCC(=O)NCCc2cn(CCO)nn2)CCCS1(=O)=O.c12cnc(s1)NC2 c1(N2CC(C)C(NC(c3cccnc3F)=O)C2)nc2ncc(Cl)cc2o1 c1(C(N2CC(OC)CC2(C)CNC(c2sccc2C)=O)=O)cc2n(n1)CCOC2 N1(C(CCC(=C)Br)=O)CCCC(N(C(=O)CC2CCOC2)CC)CC1 c1(C(N2CCC(C)(CC(=O)NC3CCC(C)(O)CC3)C2)=O)ccc2[nH]ccc2c1 C1(NC(CC=C=C)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]c3ccccc13)C2 CCCC(CCC)CC(=O)N1CCCCC1CCCNC(C12CC(OC)C1C2)=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(N=c2nc(C(F)(F)F)[nH]s2)(CO)C1 CC1CCCN(Cc2ccccc2NC(=O)COCc2ccccc2)C1 C(C(=O)N(CCC(=O)NCC(=O)NCCCO)CC(C)O)(OC)OC.C1CC1 C1(C(N(C(C)C(C)(C)C)C)=O)(CF)CCN(C(=O)Cc2ccc[nH]2)C1 c1(CCNC(C(C)n2cnnn2)=O)ocnc1CNC(=O)Cc1ccco1 c1(NC(C2CCN(C(c3c(C)cc(Br)cn3)=O)C2)=O)ncc(S(=O)(=O)O)cc1Br C1(CNC2(c3nnnn3CC3CC3)C(C)CSC2)CCCCC1(F)F.C1CC1 Cc1sc(Br)nc1C(=O)N(C1CC(NC(C2(C3CCCO3)CC2)=O)C1)C C1(CNC(Cc2n(C)nnc2)=O)CN(C(C2(C)CCOC2)=O)CC12CCC2 N1(C(CCc2cn(C)nc2)=O)CCCc2c1cnn2C1(CC(=O)OC(F)F)CC1 N1(C(c2ccc(C)s2)=O)CC2(NC(c3cc(C)n(C)c3)=O)CC1C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NC1CCC1CNC(=O)C(=O)NC1CC1 C1(C(CC)CC)CCC(NC(=O)N(C)CC2CCOC2)CC1 C(CCC(=O)N(CCCc1ccco1)C(C)=O)N(CCCC)CCC c1(C(=O)NC(C(C)(C)NC(CCN(CC)CC)=O)C)nc(C2CC2)oc1C C(=O)(C(C(C)(C)C)N(C)C)NC(c1ccc(C)o1)C1CCCCC1 CCC(C(C)C)C(C(=O)Nc1ccc2c(c1)OCO2)N1CCCC1c1ccsc1 C#Cc1ccc(C(=O)NC(C)CCCNC(C23CCC(CO)(CC2)C3)=O)cc1C Cc1cnc(NCC2CC(CNC(C3COCCC3(F)F)=O)CO2)c([N+](=O)[O-])c1 C(C(CC1CCCC1)C(=O)NC(c1ccns1)C)NC(CCCC)=O c1(NC(CNC(C23CCC(C2)OC3)=O)C2CCC2)cc(O)ncn1 N1(C(CN(C2CCC2)C)=O)CCCC(NC(c2cocc2C(N)=O)=O)C1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OCC)csc3)C2)cc(Br)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1CN(C(=O)C=CC(F)F)CCC1C N1(C(C2(C)N(C)CCC2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 CC(C)CCC(=O)N1CCCC(NC(c2cc(C(F)F)cs2)=O)C1 C1(C(N2C(C(=O)NC3(CC#C)CCC3)CC2)=O)(COC)CCCO1 c1(OC)ccc(C(N2CC3(CCC3)C2C2CCOCC2)=O)nc1N c1(COC)nc(=N)[nH]cc1C(=O)NC(C)CN(C)C(C1CCCCC(=O)N1)=O C1(NC(c2cn(CCN(C)C)nc2)=O)CC(O)CN(C(C2(C(N)=O)CCC2)=O)C1 N1(C(c2ccc(F)cn2)C(=O)NCC)Cc2ccccc2C(c2ccccc2)C1 CC1(C)CCCC1(C)NC(C1CN(C(c2ccnc(O)c2)=O)CCO1)=O c1(NC(=O)Nc2c(C(C)C)nccc2)cc(F)c(Cl)c([N+](=O)[O-])c1 c1(Cn2cc(C3(O)CN(C(=O)CCCCC4CC4)C3)nn2)cc(Cl)ccc1Cl N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(O)(CNC(=O)C(F)C2CCC2)C1 c1(CSCC(=O)NC2(C(=O)CCOCC3CCC3)CC2)ccncc1.C1CO1.NC C1(NC(=O)CC2CCOC2)CCCC2CN(C(c3ccc(O)c(Cl)c3)=O)CC12 c1(NC(CSC)C)ccc(S(=O)(=O)NCC2CCOC3(CCC3)C2)c(Cl)c1 c1(OC(C2C(c3ccc(C)cc3)C2)=O)cc(F)ccc1C C(c1cc2ccccc2o1)=CC(=O)NC1CN(C(c2cn(C)[nH]c2=N)=O)CC1O C1(C)(N(C)C(C2CN(C(=O)C3CC3)C2)=O)CCN(C(=O)COCCCN=[N+]=[N-])C1 N1(C(c2c(OC)csc2)=O)CC(NC(C2CC23CCOCC3)=O)CC(F)(F)C1 c1(N2CCCC(CN(C(c3c(CC)occ3C)=O)C)C2)nc(OC)c(F)c(C)n1 N1(C(C(CO)OC)=O)CCC(C)(CC(=O)NCCc2ccco2)C1 c1(C(c2cn(C3C=C3C)nn2)C)ccccc1.C12CC(C1)CCN2 C=CCC(C(=O)N1CCC(F)(F)C(CNC(=O)Cc2cnoc2)C1)C(C)(C)C C(=O)(CC(CCCC)NC(=O)CCc1cncnc1)N1CCCC(C#C)C1 CCCCCC(O)CC(=O)N1CCN(C(C2CC2C(N)=O)=O)CC1C1CCC1 C#Cc1ccc(C(c2nnnn2C2CC2)NC(C2CC2)C2CC2)nc1 c1(C(N(C)Cc2onc(CCC)n2)=O)cc(OC)nn1C c1(OCC#C)ccc(C(=O)NCC(C)(CO)NC(=O)CCC=CC(C)C)cc1 C=CCC(C(=O)OC)NC(=O)CCOCCN(C)C(C1C2CCCC12)=O N1(C(c2ccc(COC)o2)=O)CCC(NC(C2CCN(C)C(=O)C2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC2CNC(=O)C(C(C)C)N2CCCCC2)c(O)nc1C CC1CN(CC(c2ccccc2Br)O)CCN1c1ccncc1 C1(NC(c2nn(C)c(O)c2)=O)CCN(C(=O)C(c2cccnc2)O)CC1(C)C C(=O)(CC(C)C(C)(C)NC(c1ccn2ccccc12)=O)NC(c1nc(=O)o[nH]1)C c12ccc(nc1)SCC(O)CNC2=O.c1(C(N)=O)ccncc1.C1CC(=O)N1 N1(C(C=CC=CC)=O)CCN(C(=O)C(c2cccc(Cl)c2)O)CCC1C c1(C(=O)NC(C)C(C)NC(C2(C#N)CC2)=O)ccc2nn(C(F)F)cc2c1 c1(C(=O)NC(C)C(CO)NC(c2ncncc2C#N)=O)ccccc1[N+](=O)[O-] N1(C(c2ccc(OC)c(I)c2)=O)CCCc2cc(OC)ccc21 C#CCC(CC(=O)OC)NC(=O)C(CC(C)C)NC(C1CC1C(F)(F)F)=O C1(CNC(=O)CN2CC3CC3C2)CN(C(=O)CN2C(=O)CNC2=O)CC1O N1(C(C2CCN(C)CC2)=O)CCC2(CCN(C(C3(C)CC=CCO3)=O)C2)C1 Cc1cc(NC(C2CCCN2Cc2ccc3cc[nH]c3c2)=O)c(F)cc1F c1(OC)cccc(NC(C2(C)CCCN2C(c2cc(C#N)cs2)=O)=O)c1O N1(C(C=CC(=O)OCC)=O)CCC(C(=O)NCCSCCC(F)(F)F)C1 c1(OC)ccc(CC(N2CC(NC(=O)CCn3ccccc3=O)C(C)C2)=O)cc1 c1(CN(C2(c3cccc(OC)n3)CC2)C=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(CCC(=C)C)=O)CC(C)(C)C2)cc2c(o1)CCCC2 N1(C(CCCCOCC)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NCCC2CC(NC(C3(OC)CCC3)=O)C2)cnc(C)nc1 C1(O)(CNC(C2(CNC(c3cc(C4CC4)on3)=O)CC2)=O)CCSC1 c1(CNC2(c3ccccc3)CN(C(c3c(C)onc3O)=O)C2)cnc(O)c(F)c1 c1(C(c2noc(-c3cc(C4CCCN4)[nH]n3)n2)C)ccc(CC(N)=O)cc1 N1(C(C2(C)CCCCCC2)=O)CCCC(C2CN(C(C34CC5CC3C4C5)=O)C2)C1 OCC(Cc1ccoc1)CN=c1nc(N2C3CCCC2COC3)c2c([nH]1)CCC2 Cc1cn2nc(C(N3CC(CN=c4cc(C)nc[nH]4)C(C)(C)C3)=O)cc2c(=O)[nH]1 c1(C(C(=O)NCCOCC(=O)NCC(CO)C2CCC2)O)cccnc1 C1(C2(O)CCOCC2)(C(N2CC3CCN(C(=O)C4=C(Cl)CCCC4)C3C2)=O)CC1 C1(CNC(CCCN(C)C)=O)CN(C(c2c[nH]nc2C2CCCCC2)=O)CCO1 c1(C(=O)NC2C(CNC(C=CC(C)C)=O)CC2)cc(C(C)(C)C)n(C)n1 c1(CNC(=O)Cc2cnsc2)ncccc1C(=O)NCCCCCC1CC1 n1(CCCC(=O)NCCC(=C)CNC(=O)C(C)C2CC2)ccc2ccccc12 C1(CNC(=O)CC2CCOC2)CC(NC(c2cnc(-c3cccs3)o2)=O)C(O)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(NC(c2ncc(Br)cn2)=O)C1 C(=O)(C(CC#N)c1ccccc1)NCC(CN(C(=O)COCCOC)C)O N1(C(C(CC)N(C(=O)C=Cc2cnn(C)c2)C)=O)CCC2CCN(C)CC12 O(NC(=O)C1CC(=O)N1)CCCOC.c1(COC(C)=O)ccccc1 CC1(C)CC2(CC(CNC(C3CCN(C(=O)C(C)(C)O)CC3)=O)C2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1(F)CN(C(C2CC2c2cccc(Cl)c2Cl)=O)C1 CC(F)(F)C(F)C(=O)NCCOC1(CC=CC(=O)NCC2CCC2)CCC1 C1(c2n(CCC)nnn2)(NCc2cn(C3CC3)nn2)CCC(CC)C1 N1(C(C(n2cc(-c3cccc(C)c3Cl)nn2)C)=O)CCC(O)C(C)(C)C1 N1(C(CC2CN(C(c3ccc(CC)nc3)=O)C(C)C2)=O)CCC(F)(C#N)C1 c1(C(N2CCC(CN(C)Cc3onc(CCC)n3)C2)=O)c(C)ccnc1O C#Cc1ccc(OCC(=O)NC2CC3CC(NC(C4(CO)CCC4)=O)CC23)cc1 N12CC3CC1C3C(=O)NC(C)(C)C=CC2=O.C1(SC)CCCC1N(C)C N1(C(C(=O)NCCCCC2CCCC(C)C2)=O)CC(N)CC2(CC2)C1 C1(C(=O)NCc2c(C(=O)NCC(CC)C)n[nH]c2)CN(C)CC(C)O1 C1(c2n(C(CC)(C)C)nnn2)(NC(C)(C)COC)CN(C)CC1C c1(C(=O)NCC2(O)CCCN(C(CC3(COC)CC3)=O)C2)ccc2occc2c1 CC1CC2CN(C(C3CCCC3NC(C3CC(=O)OC3(C)C)=O)=O)CCN2C1 N1(C(C2CC(OC)C2)=O)CCN(C(c2oc(CO)cc2C)=O)CC1CS(C)(=O)=O Cc1nn(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)c2cnccn2)c(=O)o1 c1(C(N2C3(CN(C(=O)CCBr)C3)CCC2)=O)ccc(I)c([N+](=O)[O-])c1 N(C1CCC(NC(=O)CC(C)(C)O)c2ccccc21)C(CC=C=C)=O c1(CN(C2CCCC2)CC(C)C)c(F)ccc(C#N)c1F C1(NC(CC2(OC)CC2)=O)COC2C(NC(c3cc(C(C)=O)oc3C)=O)COC12 N1(C(C(F)=CCC)=O)C(CC(=O)N(C)CC2CCOC2)C2CCCC12 N1(C(CCOCC)=O)CCCCC(NC(C2CC(F)(CO)C2)=O)C1 CS(=O)CCC(=O)NCCC1(Cn2cc(CNCc3ccc(C#N)o3)nn2)CC1 C1(C(=O)NCCS(=O)(=O)NC)CN(Cc2cnc(C(C)C)s2)CCC1(F)F Cc1ccc(C(N2CCN(C)C(C(=O)N(C3CCN(C4CC4)C3)C)C2)=O)cc1O C1(C(=O)NCC2OCCC(NC(=O)Cc3cscn3)C2)CCCC2(CCC2)C1 CCCC(C)C(=O)N(C(C)(C(N1CCC(C)(CCC)C1)=O)C1CC1)C N1(C(c2scc(C(C)=O)c2)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(CCC(=O)NCCC)=O)CCOCC(NC(c2cc(Br)ccc2C)=O)C1 Cc1ccnnc1C(=O)N(CCCCCNC(=O)CCC1COC(C)(C)O1)C N1(C(CCCc2onc(C)n2)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 CC1(NC(=O)CC2CC(F)C2)CC(NC(=O)CC2(C3CC3)CC2)C1 C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2ccc(C3CC3)nc2O)=O)CC1F C1(C)C(C)(C)C(=O)NCC(C2CCC2)OC(C)CCC(=O)N1.CCOCC Cc1ccccc1OCCCC(=O)NC1CCN(C(C2CCSC2)=O)C1 C1(OC(C)C)CC(NCCCc2ccccc2)C1(C)C c1(CC(N2C(C)CC(CNC(CCOC)=O)C2)=O)c(Cl)cccc1Br C1(C(=O)N(C)CC2(C(=O)NC(C)C)CC2)CCCN(C)C1.C12CCCN1C2=O c1(C(=O)NC(CNC(c2c(C)c(N)cnc2)=O)C)cc2cc(F)cc(F)c2[nH]1 C1(CNC(c2c(C)cc(C)s2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(N(CCCNC(C2CC2C)=O)CC)ccnc(C2CCC2)n1 N1(C(C2CC(C)SCC2)=O)CCN(C(=O)CC(=O)OCCC(C)C)CC1CCO Cc1cc(C(N2CC3CC3(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)c2c(C)nn(C)c2n1 C1(CC=C)(NC(C23CC(F)C2C3)=O)CN(C(c2ccn(C3CCCC3)n2)=O)C1 C1(C(=O)NCCCC)CCCN(CCCOC(=O)N(C)C)C1 c1(OC)nccc(C(N2CCC(C)C(NC(=O)CCc3cn[nH]c3)C2)=O)c1Br c1(C(=O)NCC2CCN2C(C2(N3CCOC3=O)CC2)=O)cnncc1O Cc1nc(N2C(C(N3CCC(O)C(F)(F)C3)=O)CC3CC23)nc2ccc(Br)cc12 C1(CC(=O)NCCC2CCCC2COC)(CC)CCOCC1.C12(CC1)C(=O)N2 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)N=c2cc(C)n(C)[nH]2)CC1 c1(C(=O)NCC(CC)NC(=O)CCCS(N)(=O)=O)cccc2oc(=N)[nH]c12 C1(c2nccs2)(OC(c2cnc(C(=O)NC3CCCO3)s2)=O)CCOCC1 C1(NC(C(C)N(C(=O)C(F)OC(F)(F)F)CCC)=O)CCCCC12CCC2 C12(CC)CN(C(C3CC=C(C)CC3)=O)C(CNC(=O)Cc3cnccc3Cl)(C1)C2 O(NC(=O)C1CCc2c[nH]nc21)C(CC(C)C)C(=O)NCCCCCCF C(=O)(C1SCCc2sccc21)NC(C(C)C)(C)CNC(c1cnnn1C)=O C1(OCC)CC2(C1)CC2NC(C1(C(=O)Nc2cccc(OCC)c2)CC1)=O C12(CNC(C(CCO)C3CC3)=O)CC(CO1)N(C(=O)CCc1nc(O)n[nH]1)C2 c1(CC(=O)NC23C(CN(C(CS(CC)=O)=O)C2)C3)ccc2nc[nH]c2c1 O=C(C1=COc2ccccc2O1)NC12CCC(CF)(C1)OC2 C(C1(C)COC1)=CC(=O)NC1(CN(C(=O)Cn2ccc(Br)n2)C)CC1 c1(C(=O)NC(CN(C)C(C2CC3(CC3)CO2)=O)(C)C)ccccc1SCCO c1(C(=O)NCC2(C)N(C(c3nc(C)c(C)s3)=O)CCC2)cccc(F)c1Cl CCCC(C#N)C(=O)NCC1CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)C(C)C1 c1(C(=O)NC(C(C(C)C)NC(CCNC(=O)OC)=O)C)cc2c(s1)CCCCC2 c1(C(=O)NCCC(C)CCNC(C2CCC(C#N)CC2)=O)ccc2cncn2c1 C1(C(N2C(C(=O)OC)(COC)CCC2)=O)CCCc2ccccc2C1 C1(CC=C)(NC(c2cnc(CCC)s2)=O)CN(C(C2CC2F)=O)C1 Cc1nc(C(N2CCC(O)(CCNC(C3CC(F)C3)=O)C2)=O)c2n1CCCC2 CCC(CC)CCC(=O)N1CC2(C1)CN(C(c1cncnc1)=O)C2 C1(CNC(c2c(C)nco2)=O)CC2CCC1N2C(c1scc(Br)c1C)=O N1(C(C(CC(C)C)OC)=O)CCCN(C(c2cncc(N)c2)=O)C(C(=O)O)C1 N1(C(C(CC#C)O)=O)CCCC(NC(c2ccc(-c3nnc(C)o3)cc2)=O)C1C C(CC(C)C)(C(=O)N1CCC=C(F)C1)C(=O)NOCC1(COC)CCC1 C1(CN(C(c2ccc(CCC)[nH]2)=O)CCC)CN(CC(C)C)CCO1 c1(C(C=O)N2CCCC2c2c[nH]nc2-c2cnccn2)nc(Cl)c(Cl)s1.CC1CC1 C(C)(CO)(CC(C)C)NC(c1cc(CNC(c2ccc(OC)s2)=O)ncc1)=O Cc1ccc(C(N2CCN(C(c3ncncc3Cl)=O)C3CC23)=O)cc1OC(F)F CC(C)S(=O)(=O)C(C)C(=O)NC1CN(C(c2ccccn2)=O)CC1F c1(C(C)=O)cc(C(=O)N(C2CCCCC2)CCCNC(=O)C(C)N(C)C)co1 C1(N(C)C(c2cc(=O)cc[nH]2)=O)CCCCN(C(=O)C(CN)c2ccccc2)C1 O=C1CC(NC(c2coc(CNC(=O)CC3CCCCO3)n2)=O)CC(=O)N1 CCC(CO)CCNC(C1CCN(C(c2ccnn2C)=O)C1CC)=O c1(NC2C(NC(c3n[nH]c(C)c3C)=O)CCCC2)ncnc2scnc12 c1(C(CC(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)C)ccc(F)cc1F C#CCC(C)(CC)C(=O)NCC(CCNC(=O)C(n1cc(C)cn1)C)OC C1(C(N2C(CN(C(c3c(CC(=O)OC)ccs3)=O)C)CCC2)=O)C2CCCCC12 c1(C(=O)NC2C(NC(CC3C(C)(C)CCC3)=O)CC2)cc(Cl)c2n[nH]cc2c1 N1(C(c2ccc(C(C)C)s2)=O)CCC2(NC(c3nc(Cl)sc3Cl)=O)CC2C1 C1(CN(C)C(c2ccn(C)c2)=O)CCCN(C(=O)COCC2CCCC2)C1 C1(C)(NC(c2cc(SC)oc2C)=O)CCN(C(=O)CNc2nccs2)CC1 O=C(CCCCCn1cc(C2(O)CC2)nn1)NC(CN1CCC1)CC1CCCCC1 C1(C)(CC)CCCN(C(=O)C(CCC2CC2)NC(c2ccc(CO)cc2)=O)CC1 N1(C(C2CC(OCC)C2)=O)CC(C(N2CCC(C(C)(C)C)C2)=O)C2(CC2)C1 C(CC1=CCCCC1)CNC(CCCC=C)c1nnnn1C CC1=CCC(C(=O)NCC2(NC(c3ccc(Br)cn3)=O)CCC2)CC1 C(c1ccc(F)cc1F)=CC(=O)NCC1CCCCN1C1CC1 S(=O)(=O)(c1cccnc1NCc1ccc(Br)cn1)NCC(n1c(C)cc(C)n1)C c1(C(N2CCCN(C(C(CCC)(C)CC)=O)CC2)=O)cnc2c(c1)CCCC2 c1(C(N2CCCC(CC(=O)N(C)C)C2)C(=O)NC(C)C)cc2n(n1)CCCCO2 C12(CNC(=O)CCC3CCCC3)CC(C1)C(NC(=O)Cc1cnns1)CO2 C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(C(CC)C)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CCCN(C(=O)C=C2CCC2)CC1 CC1CC(C(=O)O)CN1C(=O)NCCC1CCCOC1 S(=O)(=O)(c1cccc(F)c1)NCC(CCNC(=O)NCCC1CCCC12CC2)O c1(CCC(N2C(CN(C(c3cnsc3)=O)C3CC3)CCC2)=O)ccc(O)cc1 c1(OC)c(NCC2CCCC(NC(=O)C(C)C(C)C)C2)ncnc1Cl C#CCC(C(=O)N(C)Cc1cccs1)NC(c1cnn(CC)c1C)=O c1(C(N2CCCCC(COC)C2)C(=O)NC(CC)(C)C)cc(Cl)c(F)cc1F Cc1ccc(Cl)c(C(=O)NCC2(C(F)F)CCN(C(=O)COC(F)F)C2)c1 C=CC1(C(N2CCCC2CCCO)=O)CCN(C(=O)CS(C)(=O)=O)C1 C1(CNC(CC(C)n2ccnc2)=O)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)CSCc1cccs1)C2 C1(NC(c2c(Br)n[nH]c2C)c2n(CC(=C)C)nnn2)CCn2ncnc2C1 C=CC(C)(CC)C(=O)NC1C2CCN(C(c3ccnn3CC)=O)CC12 c1(C(CC(=O)NCC(CNC(C(C)(C)OC(C)C)=O)F)O)nc2ccccc2[nH]1 c1(CCCCNC(=O)C(N2CC(CCO)C(O)C2)=O)ccc(O)cc1 n1(CC)nc(C(N2CC(C(C)NC(C3CCC(=O)N3C(C)C)=O)C2)=O)ccc1=O c1(C(c2n(CCOCC)nnn2)NCc2ncccn2)cc2c(s1)CCC2 c1(C(=O)NCC2(CC(=O)NCC(C)(C)OC)CC2)cn(C2CC2)nc1C CCC(CC)CCCC(=O)NOC(CC(C)C)C(=O)N1CC(C)(OC)C1 C#CCCCCCCCC(=O)NCC1CCC2CN(C(C3CNC(=O)N3)=O)CC12 C(=O)(C(F)C(=O)Nc1cn(C)nc1C(C)C)OCC.C123CC(C1)(C2)CNC3=O c1(OC)cc(C(N2CC(CNC(c3cncs3)=O)CC2C)=O)ccc1OC(C)C c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)N(C)Cc1cc(Cl)cc(Br)c1 C(C(CC1CC1)C(=O)NCC(C)(O)C(C)C)NC(COCC(=O)NC)=O N(C1CCc2cc(CNC(c3cnnn3C3CC3)=O)ccc21)C(CCOCC)=O C1(C2CC2)CC(=O)NCCCO1.C(CC(=O)NC1CC1)NC(COC)=O CC1C(NC(C2(CO)CC2)=O)CCCN1C(c1cc(C(F)(F)F)cnc1O)=O c1(C(=O)NC2(CCNC(c3cncc(CC)c3)=O)CC2)cc(N)ccc1Cl N1(C(c2ccc(C(C)=O)o2)=O)CCC(CN(C(=O)C(O)CCN(C)C)C)CC1 C=CCCN=C(NCC=CCl)N1CCc2c(cc(F)c(F)c2F)C1 N1(C(CC2(C=C)CN(C(=O)C(O)C3CCC3)C2)=O)CCS(=N)(=O)CC1 c1(NC(C2CCC(N(C(=O)CCCNC(N)=O)C)CC2)=O)cc(F)c(F)cc1O C(=O)(C1=CS(=O)(=O)CCC1)NC1C(CC)CN(C(=O)C=Cc2cnc(C)s2)CC1 CC1(C)CC(CNC(c2ccccn2)=O)N(C(=O)COc2cc(F)cc(Cl)c2)C1 C#CCC(CC(F)(F)F)C(=O)N1CCC(Oc2cccc(C)c2)CC1 C12(C(=O)NC(CC=C)(C)C)CC(CN1C(=O)Cc1csc(C)n1)C2 C1(C(C)NC(CSCCOC)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 C(CCC)(C(=O)NCC(c1ccc(F)cc1)NC(C1CS(=O)(=O)C1)=O)=CCC C1(NC(C(C)OCC)=O)CC2CC(C1)N(C(=O)C(c1noc3ccccc13)C)C2 Cn1cc2c(n1)CCCC2C(=O)N1CC(O)(CNC(=O)C(C2(O)CCCC2)F)C1 c1(-c2nnc(N3CC(OC)C3)n2C)cc(C)c2ncccc2c1C c1(C(N2CCC(NC(C3C(C=C)C3)=O)CC2)=O)ccc(C)c(S(=O)(=O)NCC)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC(NC(=O)CC2(C(=O)OCC)CC2)C1 c1(C(=O)NC2(CO)CN(C(C3C(=C)C3)=O)C2)cccc(N2CCCC2)n1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(CCNC(c2cn(C)nc2Cl)=O)C1 c1(CN(C)Cc2ccccc2OCc2ccco2)cc(C=O)ccn1 C(=O)(C(C)CCC(C)(C)C)NC1(C(=O)NCC(COCC)O)CCSC1 Cc1ccc(CC(=O)NC23CCN(C(c4ccsc4)=O)CC2C3)c(C)c1 N1(C(C2C(CCC)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(C)N(C(C2CC(F)(F)C2)=O)CC)CCC(=C2CCC2)CC1 c1(C(=O)NCC(CC)NC(c2c(Cl)n[nH]c2C)=O)cc(F)c(N)cc1F c1(OC(C)C(=O)NC2CC(CNC(C3CC(=O)N3)=O)C2)ccc(Cl)cc1 N1(C(C(c2c(C)cccc2Br)NC(C2CC2C2CC2)=O)=O)CC(C)(C)C12CCC2 O=C(CCCCOCc1ccccc1)OCC(C1CC2CCCC12)=O c1(CNC(=O)NCC23CCCN(CCC2)C3)cccc2nn[nH]c12 C1(CNC(c2ccc3cc[nH]c3n2)=O)C(C2CC2)CCN1C(=O)C=C1CCC1 N1(C(c2n(C)nc(Cl)c2)=O)CCC(c2ccccc2)(NC(=O)CC(F)(F)Cl)CC1 c1(C(N2CC(C)OC(CO)C2)=O)noc2c1CN(C(=O)CCC(N)=O)CC2 CCCCS(=O)(=O)N1CCC(C(=O)NC2CC2CNC(c2ccc(C)s2)=O)CC1 C(CCCCC(=O)N1CC(c2cc(C)cc(C)c2)C1)n1cc(CNC)nn1 C12(NC(c3c(Cl)cn(CCC)n3)=O)COC(C1)C(NC(=O)CNC(N)=O)C2 C1(C)(NC(C(C)Cn2ccnc2)=O)CCCN(C(c2ccc(O)cc2)=O)C1 N1(C(C(CC)OCC)=O)CC2CCCC2(NC(=O)CSc2ccccn2)C1 C1(NC(=O)CCCn2ccnn2)(CF)CCN(C(c2ccc(C3CCC3)o2)=O)C1 CC#CCCC(=O)N1CCC(C2CCCN2C(C2CSCN2C(=O)CC)=O)CC1 N1(C(c2cnn(CC)c2C)C(=O)NCCOCCOC)C2CCC1CN(C)CC2 c1(C(C)=O)cccnc1C(=O)N(CCCN(C(=O)CNC(=O)CC(F)(F)F)C)C c1(C(=O)NCC2(F)CC(NC(c3c(C)coc3C)=O)C2)ncn2c1CCCCC2 c1(C(=O)NC2C(CNC(c3c(C)ccs3)=O)C2)cccc(-c2ncn(C)n2)c1 C(=O)(C#CC1(C)CCCO1)N1CCC(C=C)(C(=O)N(C)Cc2nnc(C)o2)C1 c1(SC2(C(=O)NCC(C(C)C)NC(c3noc(CN)n3)=O)CC2)ccccc1F N1(C(C(C)N(C)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)CC1CO c1(CC)n[nH]cc1C(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 N(C=CC(=O)C(F)(F)F)C(C1CC2(C1)CN(C(c1cc3ccoc3s1)=O)C2)=O C(CN=c1ccc(Br)c(S(=O)(=O)NC(C)CC(C)O)[nH]1)c1scc(C)n1 CCCCC(CCC)N=c1[nH]c(N2CC3C4C=CC(CC4)C3C2)nc2ccsc12 C(C)(CO)(C(=O)NCC(C(C)(C)C)NC(=O)CCNSCC1CCCC1)OC C1(N(C(=O)Cc2ccsc2)C)CN(C(=O)C=C2CCSCC2)CCC1O C1(N(C(c2ccc(C)cc2)=O)C)CN(C(c2onc(C)c2C)=O)CC12CC2 c1(C(=O)NCC(C)NC(=O)CCCn2ccnn2)c(C(F)(F)F)sc2c1CCC2 C1(C(=O)NC2(C)CN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CCc2n[nH]c(C)c2C1 N1(C(=O)CC=C(Cl)Cl)CC2(C1)CN(C(C1CCOC3(CCC3)C1)=O)CC2CO N1(C(=O)OC(C)(C)C)CC2C3C=CC(O3)C2C1.O=C1CC(O)CN1.C(CO)N CCC(C)C(C(=O)NCC(C)C)N(C)C(c1cc(C)on1)=O c1(CC)cc(OC)ccc1C(=O)NC(C)C(C)NC(=O)CCCCN(C)C(C)C N1(C(c2cnc(OC)c(Cl)c2)=O)CCOCC(F)(CNC(c2cnco2)=O)C1 c1(N(CCC)CCNC(C2(OC)CCSC2)=O)nc2cccc(OC(F)F)c2s1 C#CCC(C)C(=O)NC(C1CCCC1)CNC(c1ccc(C(F)(F)F)s1)=O c1(NC)ncccc1C(N1CCCC(CCC(=O)NCC(C)F)C1)=O C(C(COC)C(=O)NC1(c2ccccc2)CCN(C(c2cc[nH]n2)=O)C1)OC c1(C2C(C(=O)NCC(C)NC(CCCc3onc(C)n3)=O)C2)cccc(F)c1F C1(NC(C(=Cc2cccnc2)C)=O)CC12CCN(C(c1cc(C)sc1)=O)CC2 c1(C(N(CCCNC(CC(C=C)C)=O)CC)=O)ccc(C(C)C)cc1O C1(CNC(c2cc(C)sc2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1O CN1C(=O)CSC1=CC(=O)NC1CCCN(C(c2cccc(Cl)n2)=O)C1C C1(C(=O)NCC2C(CNC(c3c[nH]cc3C3CC3)=O)C2)CC1C1CCCC1 N1(C(c2sccc2F)=O)CCN(C(c2cc(C(=O)OC)ccc2O)=O)C2(CC2)C1 N1(CCCC)CCCC2(CCN(C(=O)CCc3c(C)noc3C)C2)C1 N=C1NC(=O)C(CC(N2CC3CC2C3NC(c2ccc(SC(F)(F)F)o2)=O)=O)S1 C1(C(N2CC(C)(NC(=O)C=Cc3ncc[nH]3)C2)=O)(COC)C=CCC1 c1(NC(C)=O)cccc(C(=O)NCC(C)NC(=O)C(C)(C)N2CCCC2)n1 Cc1nn(CCO)cc1C(=O)N(CC(O)CNC(=O)CCc1cnoc1)C Cc1ccc(OCC(=O)NC(C)CC2CCN(C(=O)C3=CCCS3)CC2)cc1 C12(NC(c3scc(C(N)=O)c3)=O)CCN(C(c3cnc(Cl)s3)=O)CC1C2 C1(C(=O)NC(CC#C)CC)CCC(C)(C)N(C(=O)C(CC)C(=O)OCC)C1 CCCC(C(=O)NC1CCCCC1CC(=O)N(C)Cc1nncn1C)OC CCCC(C)(C)CC(=O)N1CCN(C(C2CCCC(CF)C2)=O)C(CC)C1 C(=O)(CCCCN=[N+]=[N-])NCCC(C(=O)NCC1CCC(C)CC1)OC c1(NC(C2CSCCN2C(c2cnccc2Cl)=O)=O)ccc(Br)nc1F N1(C(C(C=C)O)=O)CC2(CCN(C(c3cnc(C)nc3C3CC3)=O)CC2)C1 N1(C(c2c(C)oc(C(C)C)n2)=O)CC(NC(C2CCCSC2)=O)C2CCCCC12 N1(C(CCN(C(c2c(C)cnnc2)=O)C2CC2)=O)CCOC(C)(C(C)C)C1 C1(NCc2ccc(C)c(C)c2C)CCOC2(CCS(=O)(=O)C2)C1 C1(CC#C)(C(=O)Nc2csnc2C2CC2)CCN(C(C2CCC3(CC3)C2)=O)C1 C(CC(F)(F)Cl)NC(C(C1CCCC1)NC(C)=O)=O c1(CN2CC(N3CCN(C(C(CC)CC)=O)CC3)C2)cc(=O)n(C)c(=O)n1C C1(CNC(C(N2CC(C)C2)C)=O)CN(C)CCN1C(c1ccc(C2CC2)cc1)=O c1(C(=O)Nc2ccsc2)cc2n(n1)CCCN(C(C1(F)CCCC=C1F)=O)C2 C=C(C)CC(C)C(=O)Nc1nnc(-c2ccccc2Cl)o1 Cc1cc(C(=O)NCC2(CNC(=O)C(C)(C)NS(C)(=O)=O)CC2)ncc1Cl N1(C(CCc2c(C)n(C)nc2)=O)CCC2C1CCCN2C(=O)CN1CCOCC1 N1(C(CCC=C)=O)CCCOC(CNC(c2occc2C(=O)OC)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2CNC(C2CC3CCC3C2)=O)C1 C1(CC=C)(NC(=O)C(CCC)OCC)CCN(C(=O)Cc2cccc(Cl)c2)C1 CC1CN(C(=O)CC2CCOC2=O)CC(C(=O)NCC(CO)N(C)C2CC2)O1 c1(C(=O)NCC2(C(N3CC(CC)OCC3)=O)CCCCC2)ccn2cncc2c1 Cc1ccc(C(=O)NC2CC(NCc3cnc4ncccn34)C2)cc1[N+](=O)[O-] N1(C(C2N(C(CCC=C)=O)CC(C)C2)=O)CCCC(O)(c2ccccc2)CC1 N(C1CCCc2c[nH]nc21)C(C(C)CN(C(=O)CCc1nccs1)C)=O C12(CNC(C(CC)N(CC)CC)=O)CCC(CC1)N2C(c1cc(F)ccc1C)=O C1(CNC(C(C)N(C(=O)CNC(=O)OC)CC)=O)CCC(=O)N1 Cc1cccc(N)c1C(=O)NC1CC(F)CN(C(C2CC2CF)=O)C1 C(CN=c1[nH]c(Cl)nc2c1CS(=O)(=O)C2)c1ccc(OC)c(F)c1 c1(-n2cc(-c3cnc(CC(=O)N)s3)nn2)ccc2[nH]ncc2c1.c1(S)ccccc1 C(C)(C)(CCC(=O)NCCCCCCNC(=O)C(c1cnn(C)c1)O)OC C(=O)(C(F)CC(C)(C)C)N1CCC(CC=C)(C(=O)NCC2(CO)CC(C)C2)C1 C1(CN=c2[nH]nc(CO)s2)(NC(c2cc(CCC)oc2C)=O)CCCCC1C C(=O)(n1c(SCCC)cc(=O)n(C(=O)c2cc(F)cc(I)c2Cl)c1=S)OCCC C1(C(N(CC=C)Cc2ccccc2)=O)CN(C(=O)C(F)C(CC)CC)CC(C)(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC(CNC(C1(CC)CCOCC1)=O)CO CC1CCC(NC(=O)CC2(n3cnnn3)CCSCC2)CN1C(=O)OC(C)(C)C c1(C(=O)NC(C)CC(C)NC(C2CN(C3CCOC3)C2)=O)csc(=NC2CC2)[nH]1 CCC(CC)C(F)C(=O)NCC(C)(C)CC(=O)NC(COC)C(C)C c1(CC(=O)NCC(C)(C)NC(CSCC)=O)ccc2c(cnn2C)c1 c1(C(=O)NC2(CNC(CC=C=C)=O)CC(OC)C2)csc(=NC)[nH]1 C1(N(C(c2c(C)n(C3CC3)cc2)=O)C)CCN(C(C2(F)CCOC2)=O)CC12CC2 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1 c1(COC)cccc(NC(=O)C(=O)NCC2CN(C(=O)OC(C)(C)C)C2)c1 c1(C(N)=O)ncccc1C(N1C(C(N)=O)CC2CC12)=O N1(C(C(C)C2CCCC2)=O)CCN(C(N2CC3(CC3)C2)=O)CC1 c1(C(=O)NC2C(C)(C)N(C(c3cc(Cl)ccc3F)=O)CC2)occ2c1CCOC2 C1(CCCC(=O)NCC(CC)(C)NC(=O)CS(=O)(=O)N(C)C)CCC(C)C1(C)C c1(CC)cc(C)ccc1C(=O)NCCC1CC(NC(c2cc(O)ccc2Cl)=O)C1 C1(CC)CCN(C(=O)Cc2cc[nH]n2)C1C(N1CCC(OCC(N)=O)C1)=O C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(C)NC(C1(C(F)F)CCCCC1)=O C1(NC(c2ncc(C)c(Cl)c2)=O)CC2CCC(C1F)N2C(c1cccc[n+]1[O-])=O c1(C(N2CCN(Cc3cnc(CCC)s3)CC2C)=O)cc(F)cc(F)c1Br O=C(C#CC1CCCC1)NCc1cccc(NC(c2ccsn2)=O)c1 CCC(O)C(C)(C)C(=O)N1CCN(C2CCN(C(=O)CCCN=[N+]=[N-])C2)CC1 c1(SC)nc(Cl)c(NC(C23CC2CN(Cc2cn4cccnc4n2)C3)=O)c(Cl)n1 C1(NC(CS(CC)=O)=O)CC2CN(C(=O)C(O)C(C)(C)CC)CC2C1 N1(C(c2c(C)oc(C)c2C)=O)CCN(C(c2cncs2)=O)C2(CC2)C1 C1(CN(C(=O)Cc2cccs2)C)C2CN(C(=O)C(C3CC3)C3CC3)CC12 CC1CN(C(=O)CC(C2CC2)C2CC2)CCC1NC(c1cc(Cl)ccc1F)=O C1(NC(C2C(C(=O)OC)CN(C(=O)OC(C)(C)C)C2)=O)CCCC2(CCC2)C1 C(=O)(C(C)CC(=O)N(C1(CC(=O)NCC2(F)CCCCC2)CC1)C)OC N1(C(CONC(C2C(C)CCO2)=O)=O)CCSCC1CO C(=O)(CCC(O)C(C)(C)C)NCC12N(C(C3(C)CCN(C)C3=O)=O)CC(C1)C2 c1(C(N2C(C)C(C(=O)NC3(C(F)(F)F)CC3)CC2)=O)ccc2cc[nH]c2n1 C1(C(=O)NCc2ccc(CC)o2)CC12CC(NC(=O)Cc1ccsc1C)C2 C12(CNC(CC(CC)SC)=O)CN(C(c3ccc(F)cc3Cl)=O)CC(F)(C1)C2 C1(CNC(=O)C=CCF)CN(CC(=O)N(CC)Cc2ccccc2)CCO1 c1(C(=O)NC(CCN(C(c2c(SC)cccc2)=O)C)C)cc[nH]c2nccc1-2 Cn1cc(C#N)cc1C(=O)NC(C(=O)NCCn1ncccc1=O)C(C)(C)C Cc1ccc(Br)c(NC(C2CC23CN(C(=O)Cn2cc(C)nc2C)C3)=O)n1 c1(CCC(=O)NC(CNC(C(CCC)OC)=O)CO)cc(C)cc(C)c1 c1(CNC(=O)NC2(n3cnnn3)CCOCC2)ccnc(-c2ccccn2)n1 O(NC(=O)C(C)(C)CC(F)F)C(CC(C)C)C(N1CCC2(CN(C)C2)C1)=O C(=O)(C1=CC2CC(C1)CC2O)NC12CC(CNC(c3c(CC)ccs3)=O)(OC1)C2 N1(C(C=CC)=O)CC(C2CCCN(C(c3c(Br)cc(Br)c(O)c3Br)=O)C2)C1 c1(C(=O)NC(C)CC2CN(C(=O)C(C(C)O)N(C)C)C2)ccc2ccsc2c1 c1(C2(N(C(C3C(=C)C3)=O)C3CC3)CCC2)cn(Cc2ccno2)nn1 C1(CNC(c2cc(C3CC3)[nH]n2)=O)C2CN(C(c3sccc3F)=O)CC12 Cc1nc2c(F)cccc2cc1C(=O)NCCN(C(c1ccon1)=O)CC1CC1 c1(NC(C(c2ccnn2C)C)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(C(=O)NCC(C2CCOC2)NC(CCC=C)=O)c(C)coc1C CCCN=C(NCc1ccsc1S(C)(=O)=O)N1CCC(C(F)(F)F)(C(=O)NC)C1 c1(C(=O)NCC(CNC(CCCOC)=O)CO)cnc(C)nc1 C1(C(=O)NCC(C2CCCC2)NC(COCCCC)=O)CCC(N(C)C)CC1 c1(C2C(C(=O)NC(CNC(C=C3CCN(C)C3)=O)(C)C3CC3)C2)ccccc1Cl C1(C(=O)Nc2ccc(-c3ccc(C)cc3)cn2)(CN)CCC(F)(F)CC1 c1(OCC(=O)NC2C(C(=O)OCC)C2)ccc(C(F)(F)F)cc1.N12CCCC1C2 CC(C)CC(CNC(=O)OC(C)(C)C)C(=O)NCCCOC1CCN(C)CC1 C1(C(=O)NC(COC)(C)CO)CC2(CC2)CO1.C12(CCCC1)CCC(=O)N2 N1(C(C(C)N2CCC2)=O)CCC(NC(c2occc2CN2CCOCC2)=O)C1C C(=O)(CCC(=O)c1cc(C)sc1C)N1CC(O)(CCNC(CCNC(C)=O)=O)C1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCCS2(=O)=O)=O)C(C(C)C)C1 c1(C(N2C(CCNC(c3c(CC)n(C)nc3)=O)CCCC2)=O)ccc(O)c(Cl)n1 c1(CCN=C(NC(C=C)C)NC2CC23CCCC3)cccc2cc[nH]c12 CC(C)CCCCC(=O)NC1CCCC(N(C(=O)CS(=O)(=O)C2CC2)C)C1 c1(CNCc2n(C(C)C)cnc2)cc(-c2ccccc2)c2c(c1)OCO2 Cc1cn(C(C)C)cc1C(=O)NC1C2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 C(=O)(C#CC(C)(C)CNC(C1CC12CCC2)=O)NCc1c(OC)cccn1 c1(CNC2CN(C(CC(C)O)=O)CC23CC3)n[nH]c2ccc(Br)cc12 Cc1nc(N(C2CCCNC2)C(C2CCC(O)CC2)=O)c2cc(Br)ccc2n1 C(=O)(C(=O)CC(C)C)N1CCC(C(=O)NCc2cscc2C)(OC)C1 C=CC(CC)CC(=O)N(C1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC1O)C N1(C(C(C)NC(=O)NC)=O)CCC2C(C1)CN2C(=O)Cc1c(C)nn(C)c1Cl Cc1c(C(N2CCCC(C)C2CNC(=O)C(C)C)=O)sc2ccccc12 N1(C(C2CCC(=O)N2)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 c1(OCCC(=O)NCC(C)CNC(C2CCC3(CC3)C2)=O)ccc(Cl)cc1Cl N1(CC)CC(NC(=O)C(C2CCN(C(=O)CCC3OCCO3)C2)C)C(C)C1 C1(NC2C3CC4(CO)C(C3)C42)CC2CCC1CC21OCCO1 n1(CC=C)nnnc1C(c1cc[nH]n1)NC(C1CCOCC1)C N1(C(CC(=O)NCC(F)(F)F)=O)CCOC2CCN(C(C3(F)CCCC3)=O)CC12 N1(C(C=C(C)C(F)F)=O)CCC2CN(C(C3CC=CC3)=O)CCC2C1 C(=O)(C1=CC2(CCN(C(=O)C(C)(C)n3cnnn3)C2)C1)N(CC=C)C1CC1 C1(NC(CN(CCNC(CC(C)n2cccn2)=O)C2CC2)=O)CCS(=O)(=O)C1 CC1=C(C(=O)NC(CNC(C2CCS2(=O)=O)=O)C2CC2)CC1 C=CCC(C)(C)CC(=O)NC1CS(=O)(=O)CC1NC(=O)COCCN=[N+]=[N-] C1(C(=O)N(C(CNC(c2ncc[nH]2)=O)C2CC2)C)(OC)CCOCC1 N1(C(C(C=C)(C)C)=O)CC2CC(C1)CN(C(C1CNC(=O)CC1C)=O)C2 CCCCC(O)C(C)C(=O)N1CC(O)CC1(C)C(N1CCC(N(C)C)(CC)C1)=O C1(NC(CC=CC)=O)CC(O)CN(C(c2ncncc2Cl)=O)C1 c1(CCC(=O)NC(CC)CNC(C2(CCOC)CC2)=O)ccc2ncsc2c1 c1(CN(C2CCN(c3ncnc4[nH]ccc34)C2)C)c(F)ccc(F)c1O C=CCCC(C(=O)NCC(C)C#N)NC(c1ccc(OC)nc1)=O n1(CC)nc(C(N2CC(F)CC2CNC(c2cnsc2C)=O)=O)c(Br)n1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CC(NC(C2(F)CCOC2)=O)C1 C(c1cncc(O)c1)=CC(N1CC(NC(c2n(CC)nnc2)=O)C(C(F)F)C1)=O N(C(=NCCC(C)=O)NCc1c[nH]nc1-c1cccs1)C1CC(OC)C12CCC2 C1(C(=O)NC(C(C)C)CCNC(C2CCC(=O)N2C)=O)CCc2ncncc2C1 c1(C(=O)NC(CC)CNC(C2CCN(C3COC3)C2)=O)ccc(C)c(C)n1 CC(CCCCNC1CC(C)(F)C1)N(C(=O)CC#N)C(C12CSCC1C2)=O Cc1ccc(CN(C(=O)C(CC(C)C)ONC(=O)CCc2cn[nH]c2)C)c(C)c1 C1(C(=O)OC(C)(C)C)CCN(C(=O)OC(COC)CO)C2(CC2)C1 C12(OC)CCC(C(=O)NC3CN(C(C4CC(F)(F)C4)=O)CCC3O)(CC1)C2 CC1COCCC1C(=O)NCCCCC1CN(C(c2cnn(CCN(C)C)c2)=O)C1 C1(NC(CN(CC#C)C(C2(SC)CC2)=O)=O)CCC(CC(N)=O)CC1 Cc1cc(C#N)cnc1C(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Cl)o1)=O Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(=O)C=Cc2cccc(Cl)c2)C1)=O C(=O)(C(C)(C)CNC(C)=O)NCC(C)(C1(NC(=O)OC(C)(C)C)CC1)OC c1(OC)ccnc(O)c1C(=O)NCCCCC(C)NC(C1(Br)CC1)=O C=CC1CN(C(=O)CCOCCNC(c2cccn2CC)=O)CC1O CCC(C)C(C)C(=O)N(C1CCN(C(=O)C=CSC)CC1)CC1CC1 CC(CC(N)=O)C(=O)N(C)CC1CCCC1NC(c1ccc(=O)n(C)n1)=O CC1CCN(C(c2cscc2C#N)=O)CC1CNC(c1cncnc1)=O Cn1nc2c(c1C(=O)NC1CC(C)(NC(c3cnn(C(C)(C)C)c3)=O)C1)CCC2 CC1(C)CCC(C(=O)NC2(C(=O)NCCOC3CCC3)CSC2)C1 C=CCC(F)(F)C(=O)NCC1CC2CN(C(=O)CCCOC)CC12 N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)(OC)CC1 c1(-c2cccc(C)c2F)cn(CC(F)(F)F)c(=O)nc1O c1(OC)ccc(C)c(C2CCCN2C(=O)C(=O)OCCN2CCC(F)CC2)c1 N1(C(CSCCC(C)C)=O)CC(NC(=O)C#CC2CC2)C2(CCC2)C1 C1(=O)C(C(C)(C)C)OC2CCN1C2.C=CCC(C)(C)NC(=O)COC CN1N=C(CC(=O)NCC23CC2CN(C(C2(C(F)F)CCC2)=O)C3)CC1=O c1(C(N2C3CC(CNC(C4(OC(C)=O)CC4)=O)C2CC3)=O)cc2occc2n1C C1(C)(CNC(c2ccc(COC)cc2)=O)CN(C(=O)CC(C2CC2)C2CC2)CCO1 C12(OC)CCCC1N(C(=O)CCc1ncc(-c3ccccc3)o1)CCC2 Cc1cnc(N2CC3C(C(=O)Nc4c(C(F)(F)F)cccc4Cl)C3C2)nc1C C(=O)(CCC(=O)N1CC(OC)CC1CNC(C1CCCO1)=O)NCC N1(N(C(c2c(OC)n[nH]c2)=O)C)CCN(C(=O)CCN(CC(F)(F)F)C)CC1 C(=O)(C1=CC2C=CC(C1)C2)N(CCN(C(c1ccc(C)c(O)c1)=O)C)C CC(C(=O)NCCCC1CN(C(=O)Cc2ccc(O)cc2)CCO1)C(F)F C12(C(=O)NCC(C)N(C(C(C)=CC)=O)C)CCC(O1)c1ccccc12 n1(CC)ccc(CC(N2CC(C)C2C(=O)N(CC(C)OC)C(C)C)=O)n1 C(=O)(CC1OCc2ccccc21)N(C(CCNC(c1cn(C(C)C)nc1)=O)C)C C1(C(C(=O)NC2CCC(CNC(c3c(C)snc3)=O)C2)O)CCCCCCC1 N1(C(Cc2ccc(C)o2)=O)CCCC(N(C)C(C2CCCOC2)=O)C1 C12(CNC(C(C)NC(C)=O)=O)CN(C(C3CC(N(C)C)C3)=O)CC1CCO2 C1(NC(c2cc(C)nn2C)=O)CCC2CCN(C(=O)CCCc3cc(C)no3)C12 C1(OCCn2cc(C(N(c3ccccc3)C)=O)nn2)CC(C)(F)C1.C1CO1.C1CO1.C1CO1 O=S(=O)(c1c[nH]ccc1=NCCCc1cccs1)NCCC1(OC)CCOC1 C=CC(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccccc1C C1(CC(=O)NCc2c(C)nsc2)CN(C(=O)CCn2ccnc2C)CCO1 N1(C(C2C(CN)CC2)=O)CC(O)C(C#N)C1 c1(C(=O)NC23COC(C2)C(NC(=O)C(O)C(F)(F)F)C3)coc(=O)c2ccccc12 C#CCCC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(c1cccc2[nH]ncc12)=O C#Cc1cnc(C(N2CCC(C(=O)OC(C)(C)C)CC2C)=O)c(C)c1 C1(NC(c2c(CCC)nco2)=O)CN(C(=O)CC2CN3CCN2CC3)CC1(C)C C1(n2cc(-c3ccc(=N)[nH]c3)nn2)(C(N2C(C)(CC)CCC2)=O)CCCCCC1 c1(NCCC2CCN(C(c3ncn(C(C)(C)C)n3)=O)C2)ncnc2c1SCCC2 c1(C(=O)NC(CCOC)C(=O)NC2CC(=C3CCC3)C2)cnc(C)c(C#N)c1 c1(C(N2CCN(C(CCC3(C)CC3)=O)C(C(C)(C)C)C2)=O)cnc2ccnn2c1 C#CC1CN(C(=O)CC2CN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C2)CCN1C c1(CC)nccc(C(=O)NC2CCC(NC(=O)CCc3cccc(F)c3)CC2)n1 CCC(CC(=O)N1CCCC(c2n[nH]c(CNC(=O)CCF)n2)C1)C(C)C S(=O)(=O)(c1cccnc1)N1CC(CC(N2CCCC(N3CCCC3=O)C2)=O)C1 c1(C(N2CC(F)(CF)C2)=O)cc2n(n1)CCN(C(C1CCCO1)=O)C2 C1(OC)CN(C(c2nsnc2O)=O)CC1NC(c1cccc(-n2cncn2)c1)=O c1(C(=O)NC2(CNC(C(C)N(CC)CC)=O)CCC2)cccc2ccnn12 CC1=NN(C)C(=O)C1CC(=O)NC1(CO)CCN(C(=O)C#CC(=O)N(C)C)CC1 C#CCC(C(=O)NCC1=NOC(C)C1)NC(C1CCOC1(C)C)=O C1(C(=O)NCC(CC(C)C)O)CC(O)CCN1C(=O)COCCN(C)C N1(C(C(C)C2CN(C(=O)OC(C)(C)C)C2)=O)CC2CCC(C1)C(=O)O2 c1(C(N2CCCC(CCCO)C2)=O)cc(O)nc(O)n1.c1(N)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C(NC(COCCCC)=O)CCCC2)c(OCC)ccnc1O C1(CNC(C=CCNC(CNC(C2C(C)C2)=O)=O)=O)CC(=O)N(C)C1 N1(C(C2CCN(C(C)=O)C2)=O)CCN2CCN(C(C3COC(=O)N3)=O)CC2C1 C1(C)(C(N(CC(=O)NC2CC(CC(C)(C)C)C2)CCOC)=O)CSC1 c1(N2CCC(N(CCCC)C)C2)nc2c(c(=NCC3(CCCO)CC3)[nH]1)CSC2 CC(CC(=O)NC1(C(=O)NCc2cccnn2)CCN(C)C1)C(F)F C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CC(O)C(F)C1 c1(N(CCNC(c2cc(OCC)no2)=O)CC)ccnc(COC)n1 c1(C(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)(CO)CO)nccc2cc[nH]c12 c1(C(N2CC(CNC(CNC(C)=O)=O)C2)=O)ccn(C)n1 C12(C(=O)NC(CC)(C)CO)CC1CN(C(=O)CC=CC(C)(C)C)C2 Cc1cc(=O)n(C)cc1C(=O)NC1COCCC1NC(C1CCC(C)(F)CC1)=O N1(C(c2c(-c3ccc(C(=O)NC(C)(C)C)nc3)ncs2)=O)CC2COCC2C1 c1(NC(C2CC2F)=O)c(SC2CCN(C(=O)Cn3ccnn3)C2)cccc1F S(=O)(=O)(c1ccc(S(=O)(=O)NC(C)(CCO)C(=O)O)cc1)CN(C)C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(=O)C(F)C(C)(C)O)C1 N1(C(C(C)=C2CCC2)=O)CCC(C)C(NC(=O)C=Cc2ccc(C3CC3C)o2)C1 CCC(C)CCC(=O)N1CCC1CNC(C1(COC)CCCC1)=O C=CCCC(C)C(C(=O)NCCCC)N(C)Cc1ccsc1 N1(C(COCCC=C)=O)CCC(F)(F)C(C(=O)N(S(C)(=O)=O)CCO)C1.C1CN1 N1(C(c2nc(C(C)C)sc2)=O)CCCC(NC(=O)CCc2cccn2C)C1 c1(C(N2C(C(N(C(C=C)C3CC3)C)=O)C=CC2)=O)cc2ncccc2[nH]1 CC1OCCC1CC(=O)NC(CC1CCC1)C(=O)NCCc1ccon1 c1(C(N(CC(CC)NC(=O)C(=O)C(C)(C)C)CC)=O)cccc(C#N)c1F C#CC1(C(=O)NC2CCC(=O)N(CC)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(N2CCC(C)(CCNC(CC(CC)OC)=O)C2)=O)cnc2cccc(C)n12 Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC1CC2NC(c1ccco1)=O)=O Cn1cnc2[nH]c(=NCCC3CC(C(C)(C)C)C3)nc(N3CC4CC4(CO)C3)c12 C(C(C)N=c1cc(C)[nH]c(=NCC2(OC)CCCC(C)(C)C2)[nH]1)N(CC)CC C1(CNC(c2cc(C)n(C(C)C)n2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1(C)C C(=O)(C1CC(=O)Nc2ncccc21)NC1(CNC(C(COC)(C)C)=O)CCOC1 C(=O)(C(C)C(C)C)NC(C1N(C(c2c(C)nc[nH]2)=O)CCC1)(C)C c1(C(=O)OC)cc(=NC(=O)C2CCN(Cc3cc(Br)c(F)cc3O)CC2O)[nH][nH]1 c1(C(N2CCCC(N(C(=O)COC3CC3)CC)C2)=O)cc(F)c(N)cc1OC C(=O)(C1=CC2CCCCC12)NCC1(F)CCCN(C(CSCC=C)=O)C1 Cc1nc(C2CC2)nc(C)c1C(=O)NC1CN(C(C2CN3CCN2CC3)=O)C1 C1(C)(C(=O)NCCc2nc(C)c(C)s2)CCCN(C(=O)C(C)O)C1 N1(C(c2ccc(CNC(c3ccc(C(C)C)o3)=O)s2)=O)CCCC(F)(F)CC1 C#CCCN=C(NCC(C)(C)OC)N1CCN2C(=O)NCC2C1 CC1CCN(CCc2cccs2)CC1NC(c1nc(Cl)sc1Cl)=O C1(C(=O)NCCC2CC(C(=O)NCCC(C=C)C)C2)COCCN1C C(c1cccc(F)c1F)=CC(=O)NC1CCC(NC(c2c(C)scn2)=O)CC1 c1(NC(CC)=O)ccc(C(N2CC3C(CNC(=O)COC(C)=O)C3C2)=O)cc1 CC1=C(C(=O)NCC2=CCN(C(c3ncc(C(F)(F)F)cc3N)=O)CC2)CCO1 C(=O)(C1=CCCOC1)NCC(C1CCCN(C(CCN(CC)CC)=O)C1)(C)O CC1CC(NC(=O)CCCCC2CC2)CCN1C(C1C2COCC12)=O C(=O)(CCCCc1cnn[nH]1)N(C)CC1C(NC(C(C)OCC)=O)CCC1 N1(C(C(CC)(C)CNC(=O)CC(COC)COC)=O)CCCOC(C)(C)C1 C1(NC(CCC=C)=O)CCCOC1C1CCN(C(=O)CCc2cncn2C)CC1 CC(C)CCCCC(=O)N1CCCC(O)(CCNC(C2CC3(C2)CC(C)C3)=O)C1 c1(OC)cc(CC(N2CCOC(CNC(=O)C(C)(C)CO)C2)=O)ccc1O C(=O)(C(C)(C)CN(C(=O)CC(=O)N(C)C)C)NCc1n(C(C)C)ccn1 N1(C(NS(=NCC=C)(C)=O)=O)CC(OC(C)(C)C)C2CCCC12 Cc1nc(C(=O)NC(C2CCCN2C(c2ncccc2O)=O)C)n(C)n1 C(=O)(C(C)(CO)NC(c1scnc1Cl)=O)N(C)CC1(C#N)CC1 N1(C(c2c(OCC=C)cccn2)=O)CCCC2CN(C(=O)C(C)(C)CC)CCC12 c1(C(=O)OC)ccc(F)c(C(N2CCCC(C)(NC(c3cnsc3)=O)C2)=O)c1 C(=O)(C(C)(C)C(=O)OC)NC(CC(=O)N1CC(C(=O)OCC)C1)(C)C C=CCCC(C)(C)C(=O)NCCCC1CCCCN1C(c1[nH]c(C)nc1C)=O N1(C(CC2C(CC)C2(F)F)=O)CC2CC1C2NC(c1n[nH]c(C)c1Br)=O CCC(CCC(F)(F)F)C(=O)NC1CC(CCN)C1 CC(CCCNC(=O)C(C)OCc1ccccc1)NC(c1csc(C2CC2)n1)=O C1(C(=O)NC(C=C)(C)C)CN(C(C2CC(OC3CC3)C2)=O)CC1F c1(CN(S(N(CCC)CC)(=O)=O)C)c[nH]c2c(Cl)cc(F)cc12 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)NC1CC(C=C)C1 c1(NC(=O)Cc2ncccn2)ccc2c(c1)CN(C(=O)C1=CCCCO1)CC2 N1(C(C2N(CC)CC2)=O)CCC(C)(CC(=O)NCC(C2CC2)OC)C1 c1(C(c2c(NC(C3CCN3C3CC3)=O)ccc(F)c2)=O)c[nH]c2ncc(F)cc12 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)C3CC23)=O)c2c1CCCN2 c1(CN2CCCN(C(c3c(C)noc3)=O)C(C)C2)cc([N+](=O)[O-])ccc1O N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(C3(CO)COC3)=O)CC2C1 C1(N2CCN(C(=O)OC)CC2)CCN(C(c2ccc(CO)o2)=O)CCC1C C#Cc1ccccc1CC(N1CCN(C(c2n[nH]c(=N)s2)=O)C(C2CC2)C1)=O CC(C)(CNC(c1ccc(C(F)F)o1)=O)CCNC(=O)C=CC1CC1 c1(C(N2CC3C(NC(C4CNC(=O)O4)=O)C3C2)=O)cc2cccc(Br)c2[nH]1 C(C(F)F)(C(C)CC)Nc1nnc(SC(C(=O)NC)C)n1-c1ccccc1 C1(CNC(c2cc3ccccn3c2)=O)CCCC2CN(C(c3cncs3)=O)CC12 C1(F)(CNC(=O)CN2CCC(O)CC2)CCN(C(=O)C(=O)NCC(F)F)CC1 N1(C(C(C)(C)SC)=O)CCN(CC2CN(C(c3nsnc3O)=O)C2)CC1 N1(C(C=C(CC)CC)=O)CCC2(CC1)CCN(C(C1CNc3ccnn3C1)=O)CC2 N1(C(=O)NCCCCCCCC)CCOC2(C1)CN(C(c1ccsc1C#N)=O)C2 C(C(C(=O)NCCN1C(=O)CNC1=O)C(C)(C)C)NC(c1n(C=C)ncc1)=O c1(C(=O)OCC)cc(C)nnc1N1CCC(CNC(c2occc2C)=O)C(C)C1 c1(OC)c(C)cc(C(=O)NCCC2CC(NC(C3CC(C)CO3)=O)C2)cc1C O=C(CCC[N+](=O)[O-])NC1C=CCN(C(C2(c3cc(F)ccc3F)CCC2)=O)C1 CC(Cc1ccccc1Cl)N=c1nc(N2CCC(C)(F)C2)c2c([nH]1)CCC(C)C2 CC(O)CC(C)(C)CNC(C1CCCCN1C(=O)Cc1cncnc1)=O Cc1ccc(CC(N2CCC(N(C)C(c3n[nH]cc3Cl)=O)C2)=O)cc1C CS(=O)(=NC(=O)c1ccc(CN2CCOCC2)o1)C1CC(c2nn[nH]n2)C1 Cc1cc(C(N2CC3CCC2CN3C(C2(C)CCC(C)C2)=O)=O)c(C)nc1C N1(C(C(=O)NCc2c(N(C)C)cccc2)=O)C2CCC(C2)C1CCO Cc1cc(C(N2CC(N(C)C(c3[nH]cc4c3CCC4)=O)C(F)C2)=O)ccc1Cl Cc1ccc(NC(=O)NCCC2CC3C=CC2C3)c(-n2cc(Cl)cn2)n1 C=CCC(CC(=O)NC(C)CCF)NC(C1(C=C)CCCCC1)=O c1(C(CC(=O)NC(c2nccc(=N)[nH]2)C)N)cccc(F)c1 c12nnc(C3COCCN3C)n1CC1CCN2C1.N(CC)CC.C1(COC)CC1 CC(C)CC(C)C(=O)NC(C)(CNC(c1c[nH]cc(Br)c1=O)=O)C1CC1 C1(NC(CNC(CC(C)(C)C)=O)=O)CCCC12CCN(C(c1sccc1F)=O)C2 C=CC(CC)C(=O)N1CCC(C(=O)N(CC(O)C2CC2)C)(CO)C1 c1(NC(C(C)NC(CCC2CC(OC)C2)=O)=O)ccc2ccoc2c1 c1(C(CF)NC(N(c2cccc(OCF)c2)C(C)C)=O)ccc2c(c1)OCO2 N1(C(C2(C#C)CN(C(c3csc(CC)n3)=O)C2)=O)CCOC(C)C1CO N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)Cc3c(O)ncnc3O)CCC2C1 C(=O)(C1=COCCO1)N1CCC(CN(C)C(C2(c3ccc(F)cn3)CC2)=O)C1 c1(C(N2C3(CNC(c4n(C)ncc4)=O)CCC2CC3)=O)c[nH]c2cccnc12 CC(C)C(CCNC(C1(C)CCOCC1)=O)NC(=O)C(C)NC(C)(C)C c1(C(C)NC(C(C)NC=O)=O)nocc1C(=O)NC1CC2CC2C1 c1(C(N2CC(CNC(COc3c(OC)cccc3)=O)C2)=O)cc(S(C)(=O)=O)co1 n1(N(CCN(C2CCC2)C(c2ccccc2)C)C)ncccc1=O c1(N(CCCCNC2C=CCCC2)C)ncccc1S(=O)(=O)Nc1cnn(C)c1 N1(C(CN(CCC)C)=O)CC2CCC1C(CNC(=O)Cc1ccccc1F)C2 C1(N(C(c2cnc(CC)s2)=O)C)CCCC(NC(=O)C(C)(C)NC(C)=O)C1 N1(C(C2C(CNC(c3cncc(CO)c3)=O)C2)=O)CC2CCC(CO)(C2)C1 C1(CNC(C=CC=CCC)=O)COC(CNC(=O)CCC2CC(OC)C2)C1 c1(CC(=O)NCC(c2ccc(F)cc2)NC(c2c(C)nc[nH]2)=O)ccc(F)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC(C)CNC(c1cccc2c1CCO2)=O C1(NC(c2c(C)coc2C)=O)CN(C(=O)C(C)c2ccsn2)C2(CCCC2)C1 C1(CCC)CN(C(=O)C(N2CCNC2=O)C)CC1NC(c1cc(OC)n(C)n1)=O N1(C(CC2C(C)(C)C2)=O)CC(C(=O)NCc2ccc(Cl)cn2)CCC1(C)C C1(NC(C2C(=C)CC2)=O)C2CN(C(C3C4(CC4)C34CC4)=O)CC12 C=CC(O)C(=O)NC1CCCC1CNC(=O)CC1(O)CCCC1 c1cccc2cc(C)oc12.c1(OC)cccc(C#N)c1.N1(C2CN2)CCC(O)C1=O CCCC(C)CC(=O)NCCCCN(CCCNC(=O)Cc1cccn1C)C O=C(N=c1ccn(C2CN(C=O)C2)[nH]1)c1cc2c(s1)CCC2.C1(C(F)(F)F)CC1 C1(C(N2C(CCCNC(C(C)S(C)(=O)=O)=O)CCCC2)=O)CC2(C1)CC(F)(F)C2 Cc1nn(CC(=O)N(C2CCCC(NC(c3ccc(=O)oc3)=O)C2)C)c(C)c1Cl C1(CNC(C(C)N(C)C)=O)CN(C(c2n[nH]cc2Cl)=O)C2COCC2O1 N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(=O)N(C)CCF)c2C1 N1(C(Cc2cc(OCC)ncc2)=O)CCC2CCN(C(c3ccsc3C)=O)C2C1 C(=O)(CC(O)CNC(=O)C(C)CNC(=O)CC(C)F)OC C(CCN=c1cc(C)nc(NC(C)CS(N)(=O)=O)[nH]1)n1ncc(C)c1 c1(CNC(C2CSCCN2C(c2cc(Cl)sc2Cl)=O)=O)ncccc1Cl N1(C(C=CCN(CC)CC)=O)Cc2[nH]nc(C(N3CCC(C)C3C)=O)c2C1 N1(C(CCC(C)OC)=O)CCN(C(c2cccnc2)=O)CC1CN(C)C C1(NC(C(C)(C)c2ccns2)=O)CN(C(C2CCC(C)CC2)=O)CCC1CO C1(N(CC(F)F)C(=O)OCC(C)O)C=CCN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC(CC=C)(C)C)CCCN(C(C2(N(C)C)CCCC2)=O)C1 C1(C(N(C)CCN(C)C)=O)(NC(=O)CC(=O)NCC#N)CC1(C)C C12(COC)CC(CNC(=O)CC(C)F)(CN1C(c1ccc(C)s1)=O)C2 c1(COC(c2ccc(C)cc2Br)=O)ccc([N+](=O)[O-])cc1Br C1(CC(N2CC(CC(=O)NC(c3ccccc3)C)C2)=O)NC(=O)NC1=O CC1(C)CCN(C(c2c[nH]nc2Cl)=O)C1CC(=O)NCC1CCC=CO1 C(CC(C)C(=O)N1CCC(C(=O)N(CCC(N)=O)C)C1C)OC c1(C(N(C)CC2N(C(C(=O)NC(C)C)=O)CCCC2)=O)nc[nH]c2ncnc1-2 Cc1ccc(C(=O)NC2CC(C(=O)NC3CCCC(F)C3)C2)nc1 C(=O)(C(CCC(N)=O)N(C)C)NCC1N(C(Cn2c(C)csc2=O)=O)CCN(C)C1 c1(C(=O)Nc2scc(-c3ccc(C#N)o3)n2)c(Br)ccnc1Cl N1(C(c2ccc(C=C)cc2)=O)CCC(NC(=O)C(N2CCCCC2)C)C(C)(C)C1 C1(OC)(OC)CC(C)(C(N2CCCC(CNC(C3(C4CC4)CCCO3)=O)C2)=O)C1 C(=O)(C(c1cccs1)=Cc1cccc(Cl)c1)NC1CCN(C(C(C)N(C)C)=O)C1 C1(NC(c2c(CC)ocn2)=O)CCN(C(=O)C(C2CCOC2)OC)CC1C N1(C(c2cn(CC)nn2)C(=O)NCCCC)CCOCC(CO)C1 C1(CC)(CC)CC(C(=O)NC2CC(CCNC(=O)CSCc3cscn3)C2)C1 N1(C(C2C(CCC)C2)=O)CC=CC1C(=O)NCC1(O)CN(C)C1 C1(CNC(CCCOC)=O)CN(C(=O)Cc2cn(C(C)C)nn2)CC(C)(C)C1 C(=O)(CC1OCCc2ccsc21)NC1C2(CC(NC(CCC(=C)C)=O)C2)C1 c1(OCC)c(CC(N2CCCC(CNC(C3CC(SC)C3)=O)C2)=O)cccc1Cl C(=O)(CCCC(=O)N1CC(NC(=O)CCn2ccnc2C)CC1C)OCC c1(SC)cscc1CNC(c1nnnn1CC(F)F)(C1CCOCC1)CF C1(CNC(c2cc(Cl)sc2Cl)=O)C2CCCC1N(C(=O)CC1CC=CC1)C2 c1(C(=O)NC(C)CNC(=O)CC2CCC(=O)C2)ccnc(C(F)F)c1 c1(C(N2C3C(NC(c4c(C)scc4)=O)CC(C3)C2)=O)ccc2c(c1)C(=O)NC2 Cc1sc(Cl)c(C(=O)NC2(CNC(=O)CC3CC(C)C3)CCOC2)c1C Cc1cc(O)c(F)cc1NC(C1CN(C(c2[nH]cc(C)c2C)=O)C2(CCC2)C1)=O c1(C(=O)NCC2CC(F)CN2C(c2cc(F)n[nH]2)=O)cnc2c(c1)CNC2=O C1(NC(c2c(C)onc2C(F)(F)F)=O)CCC(C)N(C(C2C3CCCCC23)=O)C1 CCC(C)(C)C(C)CC(=O)NCC1C=CCN1C(=O)CSc1ccc(OC)cc1 c1(C(=O)NCC(C)N(C(C(c2c(C)cccc2)C)=O)C)ccc(F)c2ccsc12 CC1CC(C(=O)N(C)CC2CCCC2(C)C)CN(C(=O)CCc2ncccn2)C1 N1(C(CCC2N(C)CCC2)=O)CC=C(C(=O)NC23CCCC2OCC3)C1 Cc1ccc(C=CC(=O)NCCCCCNC(=O)C(C)C(F)(F)F)cc1C N1(C(C(C(C)C)c2cn(C)nn2)=O)CCS(=O)(=O)N2CCOCC12 CC1=C(C(=O)NCC2(C)CCN(C(=O)C(c3ccccc3)F)C2)C(=O)OC1(C)C CCC(O)C(C)C(=O)NCC1CN(C(C2(c3cccc(Cl)c3)CCCCC2)=O)C1 c1(NCC(=O)N(CCNC(c2c(CCC)nns2)=O)C2CC2)ccc(C)cc1 c1(C(N2CCC(C(=O)NC3(C(F)(F)F)CC3)C(F)C2)=O)nc2ccc(F)cn2n1 C#Cc1ccc(C(N2CC(CNC(=O)CC3CCC(=O)NC3=O)C(C)C2)=O)cc1 c1(C(N(CCNC(C(CC)OCC)=O)C2CC2)C)ccc(C(F)(F)F)cc1 CC#CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C1CCC1 Cc1c(N)ccc(C(N2CCOC(CNC(=O)CC(O)CC3CC3)C2)=O)c1Cl c1(C(N(C(C)CN(C)C(C2(O)CC2(C)C)=O)C)=O)cnn2cccnc12 C(N=C(NC1CCCCC1)N1CC(C)CC(C)C1)C1Cc2c(ccc(CO)c2)O1 CC1(C)CC(n2ccnc2-c2cccc(C(F)(F)F)n2)C(=O)N1 C1(NC(CCCc2onc(CC)n2)=O)CCN(CC2CCC(C)O2)C(C)C1 c1(CC(=O)NC(C2CC2NC(=O)CNC(=O)CC(C)(C)C)C)ccc(O)nc1 c1(SC)ccc(O)c(C(=O)N(C2CN(C(=O)COc3cccc(C)c3C)C2)C)c1 Cc1cc(N)ccc1C(=O)NCCN1CCN(C(=O)CC2COCCOC2)CC1 c1(CC(C)OC)nc(-c2ccc(C(F)(F)F)nc2)n(C(c2ccccn2)C)n1 c1(OC)nccc(=NC(=O)C2(C)CCN(Cc3ccc(Br)nc3Br)C2)[nH]1 C1(NC(C(CC)CCOC)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)=O c1(OC)cc(Cl)ccc1C(=O)NCCCCNC(=O)C(F)(F)CN(C)C CC1CCN(C(=O)Cc2cc(O)no2)C1c1cn(CCO)nn1 c1(OC)cc(C(=O)NCc2nc(CNC(=O)CCC(C)C)cc(O)n2)ccc1C O=C1NC(C(=O)NCC2(O)CCN(C(=O)CCC(=O)c3ccc[nH]3)C2)C2CCC12 C1(C)(CNC(C(CCC)NC(=O)C(C)OCCC(C)C)=O)CCCC(C)(C)C1 CCS(=O)(=O)C=CC(=O)N1CCC(OCCNC(=O)CC2=CCCCC2)C1 CCC(CC)CN=c1[nH]c(=NCC2(C)CC3(C2)CC(F)(F)C3)c2cccc(F)c2[nH]1 CCC(CCC(=O)NCC1CC(C)=NO1)NC(=O)CCCOC(C)(C)C C1(CC(=O)N(C2CCSC2)CC)(NC)CCCN(c2ncc(OC)c(C)n2)C1 c1(C(C(N2CC3(CC(NC(C(C=C=C)C)=O)C3)C2)=O)C)cccc2ccccc12 C1(NC(c2c(NC)cnnc2)=O)(CO)CCCN(C(=O)CC2=CCCC2)C1 C1(CC)CN(C(C23CCC(C2)C3(C)C)=O)CCC1NC(=O)CCCC1CC1 C(=O)(CC(C)CF)N(CCC)CCNC(=O)C(F)(F)c1csc(C)c1 C1(C(=O)NC2C(OC)CN(C(=O)C(C(C)C)SC)C2)CC2CCC1C21CC1 Cc1ccc2c(c1)CC(C(=O)NCCCCCCN(C(=O)C(C)(C)C)C)S2 c1(NC(C(CC2CCC2)NC(CCC=C=C)=O)=O)ccc(F)c(OC)c1 Cc1ncc(C(=O)NCC2CC3CCC2N3C(=O)Cc2ccccc2C)c(C)n1 c1(C(=O)NCCC(C(C)C)NC(=O)CC(O)C2CC2)nccc2occc12 c1(C(N(C2CCCN(C(=O)CCC(C)SC)CC2)CC)=O)cn2cc(C)sc2n1 C(=O)(C1=CCCCC1C)NC1CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC21 C1(C(=O)NCCS(CC)=O)CCCCN1C(=O)Cc1cncnc1 c1(C(=O)NC2CC(NC(C3CCOCC3)=O)C23CCC3)ccc2[nH]ccc2c1 C1(CC(=O)NC(c2nccs2)C)CCCC(NC(=O)Cc2cccnc2)C1 c1(CC)ccc(C(=O)N(CCCCCCNC(C2(C#N)CCCO2)=O)C)cc1Cl C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(C2COC(=O)O2)=O)CC1)CC c1(C(C(=O)NC(C)CCNC(c2ccc(C(F)F)cc2)=O)O)ccc(F)c(Cl)c1 CCCCC(C)(CO)NC(c1ccc(C)c(C(=O)O)c1)=O C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cccc(F)c2C)=O)C(F)(F)C1 c1(C(N(C2CCN(C(=O)C(C)(C)CO)C2)CC)=O)oc2c(Cl)cccc2c1C C(C)(C)(CCC(=O)NCCN(CC)CC)NN(CCC)CCN(C)C C1(NC(c2c(C)nc(O)cc2)=O)CC2CC(NC(C3CCC(C)CC3)=O)CC2C1 Cc1ccc(C)c(C(=O)NCC2CC2NC(c2cnc(O)c(F)c2)=O)c1O C(CO)(C(C)(C)C)NC(c1nnnn1CCC1(C)CC1)(COC(C)C)C C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(C2CC2C)=O)C2(CCCC2)C1 Cc1cc(C(=O)NC2CN(C(=O)CSCC(C)C)CC2C)nnc1O N1(C(C(=O)NCCN(CCOC)C)=O)CCCCNCC(F)(F)C1 C1(CC(N2CCCCC2C2(NC(=O)COC(F)(F)F)CC2)=O)(CC)CCOCC1 N1(C(C(CCSC)OC)=O)CC2CCN(C(c3sc(F)cc3Cl)=O)CC2C1 O=S(=O)(c1ccc(NC2CC2c2cccc(F)c2)nc1)NCCC1CC(O)C1 S(=O)(=O)(c1cccs1)NC(CCSC)C(=O)Nc1cc(CS(C)(=O)=O)nn1C C(CC(C(=O)N1CCN(c2ncccc2Cl)CC1)OC)OC N1(C(C(C)OC)=O)CC2(C1)C(NC(=O)Cn1cccc(C)c1=O)CCS2(=O)=O N1(CCC)CCN(C(=O)Cn2cc(C(=O)OC)nn2)C(C)C1=O C1(NC(c2cnc(Cl)s2)=O)COCCN(C(=O)C(C2CCS(=O)(=O)CC2)F)C1 CC1OC2(CO)CC1(C(=O)NCCN(C)C(C1CCCN(CC(F)(F)F)C1)=O)C2 N1(C(C(C)O)=O)CCOCC1CCNC(=O)CSc1ccccn1 c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2OC)=O)nnn(C(C)(C)C)c1CC c1(C(=O)NC(CC)(CC)C(N)=O)n[nH]c2c1CN(C(=O)C(C(C)C)SC)C2 Cc1c(Cl)cnn1CC(=O)NC(C)C(C)NC(=O)Cc1sc(O)nc1O C1(C2CCN(C(c3cnn(CC)c3C)=O)CC2)(NC(CC(C=C)(C)C)=O)CCC1 C1(C(N2C(C)CN(C(C34CCCC3C4(F)F)=O)CC2)=O)CCc2ccccc2C1 C(=O)(CS(=O)C(F)(F)F)N1CC(OCCNC(CC(C)N(C)C)=O)C1 C(=O)(CCCN=[N+]=[N-])NCCCC(=O)NC(C)CC1(O)CCC1 N1(C(C(C(C)(C)C)CO)=O)CCC2(CC1)CCN(C(c1csc3nnsc13)=O)C2 c1(CC)cnsc1C(=O)NC1COCC1n1cc(C(CC)OC)nn1 c1(C(=O)NCC23OCC(CNC(C(C)=CC)=O)(C2)C3)cnc2cccnn12 CN1CCN(C)CC(C(N2CCCC2CCNC(C2(C)CC2(F)Cl)=O)=O)C1 C1(C(C)NC(=O)CCOCc2ccccc2)CN(C(c2cc(O)cs2)=O)CCO1 CCC(C(=O)NCC1CCN1C(c1cc(C(N)=O)no1)=O)Oc1ccccc1 c1(C(=O)NCC2(CN(C(C)C(=O)O)CC)CC2)c[nH]nc1-c1ccoc1 Cc1ccn2c(=O)c(C(=O)NCC3(NC(=O)C(N)=O)CCCCC3C)cnc2c1 CCS(=O)CC(=O)N(C(c1ccccc1)CNC(c1cc(Cl)on1)=O)C N1(C(C(c2cc(C)sc2)(F)F)=O)C2CCC1CN(C(c1cc(O)cc(O)n1)=O)C2 N1(C(CCC(=O)OC)=O)CCC(NC(=O)Cc2ccc(Br)cc2I)C(F)C1 CCCCC(c1nnnn1CCCSc1cccs1)NCCCn1cc(C)cn1 C1(C(N2CC3CC(NC(C4CC(O)(C#C)C4)=O)C3C2)=O)(CC)CCC(F)(F)CC1 C1(N(C(CCCC#C)=O)C)CC2CCC(C1)N2C(C1CCC(C)C1)=O CC1CCCCN1CCNC(=O)C(C)(C)NC(=O)CC(C)N(C)C C1(CC=C)(NC(C(C=C=C)C)=O)CCCN(C(=O)CCCCCOC)C1 N1(C(CCCCC=C)=O)CC(CNC(c2cnc(C)[nH]2)=O)CC12CCOCC2 N1(CCC(=O)N(CC(C)(C)NC(C(C2CCOC2)OC)=O)C)CCOCC1=O C1(C(=O)NC(CC#CC)C(=O)NC)CN(C(=O)C(CCC)N(C)C)CCC1(C)C c1(C(=O)NC2C(NC(COCC=C)=O)CCC2)cc(F)cc2nc[nH]c12 C(=O)(C1CCc2cccnc21)N1CCC(CNC(C=Cc2c(C)cccn2)=O)C1 CC(C)(F)CN=c1[nH]c2c(c(=NCc3ccc(Br)cc3N)[nH]1)CC(C)CC2 CCC(C)(CCNC(=O)C(=Cc1cccnc1)F)NC(=O)C(O)CSC c1(OC)ccc2c(=NCC=CBr)[nH]c(=NCc3ccc(=N)[nH]c3)[nH]c2c1 CC1(C)CC(CC(N2CCCC(C)(NC(c3coc(O)n3)=O)C2)=O)C(=O)O1 C(=O)(C1=NN(CC)C(=O)CC1)NC(C1(C)N(C(CCC=CC)=O)CCC1)C n1(CC(=O)NC2CC(NC(=O)CCC3CCCC(O)C3)C2)ncc2ccccc12 C(=O)(CCC(=O)N1CC(O)(CN(C(=O)C(c2ccc(C)cc2)(C)C)C)C1)NC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C(C)NC(c1ocnc1C1CC1)=O)C C1(CCNC(COCCCCC)=O)COCCN1C(=O)C(N1CCC(C)C1)=O c1(C(C)C)cc(C(=O)NCC(C)NC(c2ccncc2Cl)=O)cc(F)c1 C1(NC(C(C)(C)CF)=O)CC(F)CN(C(c2c[nH]nc2C2CCOC2)=O)C1 CS(=O)(=O)c1ccc(NC(=O)C(=O)Nc2ccc(C(N)=O)c(Cl)n2)cc1 C(=O)(C(O)C(C)CC)N(CC(CNC(CCCCC)=O)(C)C)CC C1(N(C)C)CN(C(C2CCC(NC(=O)Cc3ccsc3)CC2)=O)CCC1O C=CCCCC(C(=O)NCC(CC)N(C)C)NC(=O)C#CC(C)(C)C Cc1cc2ncc1S(=O)(=O)N2.C1(NCCN(C)CCO)CC=CCC1C(F)(F)F c1(C(N2CCCC2C(=O)NC(C)(C)C)C(=O)NC)cc(Cl)cc(Br)c1F c1(C(=O)O)cc(COC)cc(S(=O)(=O)NC2CC(c3ccc4c(c3)OCO4)C2)c1 N1(CC(=O)NCC(CNC(c2cc(C)cc(O)c2)=O)C)C(C)=CC(C)=NS1(=O)=O C1(NC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)CCC(CNC(=O)C(C)CF)CC1 CS(=O)C=CC(=O)NC1CCCN(C(=O)CCc2ccc(-c3ccccc3)o2)C1 N1(C(N2C(c3onc(C)n3)CCC2)=O)CC(=O)Nc2cc(C(F)(F)F)ccc21 N1(C(C(CC)n2ccnc2)=O)CCC(NC(c2ccc(N)c(N)c2)=O)C(C)C1 c1(C(N2CC(NC(C3CC(C)(F)C3)=O)C3(C2)CCC3)=O)cc(O)ccc1[N+](=O)[O-] c1(CC)ccoc1C(=O)N(C)CCOCCC(=O)NC(c1cnsc1)C C1(NC(Cc2cc(C)on2)=O)COCCC1NC(=O)C(C)c1ccco1 C1(C(=O)NCCc2scc(C)n2)CC2CCC(C1)N2C(C1C2CC3C(C2=O)C13)=O CCCS(=O)(=O)C(C)C(=O)N1CCN(CCN(C)C(c2cc(C)nn2C)=O)CC1 N1(C(C(CCC)F)=O)CCC(NC(c2cccnc2OC)=O)C(C)C1 c1(OC)ccc2oc(C(N3CCC(NC(C4(O)CCSC4)=O)C3)=O)c(C)c2c1 C(C(=O)NCC1(O)CN(C(C2(C)CCN(C(C)=O)C2)=O)C1)(C(C)C)SCC c1(NCC2(O)CCN(C(CC(=C)C)=O)CC2)ncnc2sc(C)c(C)c12 c1(COC)c(C(=O)NC2CCCCC2NC(C2(C)CCC23CCC3)=O)cnn1C Cc1cc(C(F)(F)F)ccc1CC(N1CCC(NC(c2n[nH]c(C)c2C)=O)C1)=O c1(OCC)ccc(NC(=O)CCC2CCN(C(=O)C=CCO)C2)cn1 c1(C(=O)NC(C)CNC(=O)CCCCO)cncc(N=[N+]=[N-])c1 C1(CS(C)(=O)=O)CN(C(=O)CCCc2ccccn2)CCN1C(C1CC1(F)F)=O c1(-c2ccc(C(=O)NC)cc2)ccn2nc(C(=O)NC(CO)CO)cc2c1 n1(CC(=O)NC(C)(C)CC2CCCC2)cc(CNS(=O)(=O)C2CC2)nn1 CCCCC(F)C(=O)N1CCCC1CCC(=O)NCc1cccc(F)c1O N1(C(C(C)=O)=O)CC(NC(c2n[nH]c(C)c2F)=O)C(F)C1 C#CCCCCCCC(=O)N1CC(NC(c2ccn(CCC)n2)=O)C(O)C1 C1(C(=O)NC)CCN(C(C2CN(C(=O)CN3CSCC3=O)CCO2)=O)C1C N1(C(C(C)c2cccs2)=O)CCN(C(C2(F)CCCC2)=O)CC2(C)CCCC12 C(C)(C(C(=O)NCc1ccc(C#N)cc1)C(C)C)NC(C(C1CCCC1)OC)=O C1(NC(CCC(C)=O)=O)CC(NC(=O)C=Cc2ccnn2C)C12CCC2 c1ccc(F)cc1.C1(COCC)CCN(Cn2cc(C(N)=O)cn2)C1 C1(C(C(=O)N(C2CCN(C(c3cnc[nH]c3=N)=O)C2)C)O)CCS(=O)(=O)CC1 N1(C(CN2CCCC(c3nnc(C)o3)C2)=O)CC(C)OC(C)C1 c1(C(C)OCC)nc(C)c(C(N2CCC(C)(NC(c3snnc3CC)=O)C2)=O)s1 c1(N2CC(c3ccc(C)o3)OCC2)nc(=NCCC2CC2)[nH]c2cccc(F)c12 N1(C(c2cncc(C)c2C)=O)CCC(NC(C2(F)CC=CC2)=O)C(CO)CC1 O=C(C#CC1CCCC1)NC1CCCCN(C(=O)CCc2nccs2)C1 c1(CC)cc(C(N2CC(CNC(c3ccn(CC(C)C)n3)=O)CC2C)=O)ncn1 Cc1cccc(C(N2CCCC2C2(C(=O)NC3CC4C=CC3CC4)CC2)=O)c1O N1(C(CC2(OC)CCC2)=O)CCC(F)(F)C(NC(=O)CCCc2ccccc2)C1 C1(C(=O)NC2CC(NC(CC)=O)C(O)C2)CCc2nc(C)nc(C(F)(F)F)c2C1 CCC(CC(=O)N(C)CCOCC(C)(C)C)NC(=O)C(C)C1CCCC1 Cc1nc(N2CC(NC(=O)CCCCCNC(N)=O)CC2C)c2scc(C)c2n1 c1(CC(C)NC(C(=O)NCC2C(OCC)C2)=O)c(F)cccc1Cl O=C1CC(NC(C2CC(O)CCN2C(C2C3CCC(F)C23)=O)=O)CC(=O)N1 C1(C(=O)NC(C(=O)NCC(CC)(C)Cl)CO)C2CC3C(C2)C13 c1(-c2nc(C(=O)NC3CC(OCCOCC)C3(C)C)on2)cc2ccccn2n1 C(CC(=O)N1CC(C)CC1CC)(C(F)(F)F)NC(C(CC)C)=O Cc1nc(N)c(CC(=O)NCC#CCNC(=O)CC2CC2(C)C)c(O)n1 c1(CC)cnc(CNC(=O)CC=CCNC(=O)CSCCC#N)o1 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)C(CCS(C)=O)N(C)C)C(C)(C)C1 C1(CNC(C=NOC)=O)CN(C(c2cc3n(n2)CCC3)=O)C2CCCCC12 N1(C(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)COC(F)F)C2CCC12 C1(NC2(c3n(CCCC)nnn3)COC2)CCCC(n2nccn2)C1 c1(CC(C(=O)N2CCC(OCCF)C2)NC(=O)CN2CCCC2)ccccc1Br C1(C2(O)CN(C(=O)C(CC(C)C)NC(=O)NCC(C)C)C2)(C(=O)OC(C)(C)C)CC1 C(C(C)C(F)C(=O)N1CC(C)(C(N)=O)C1)NC(CCc1cnc(C)o1)=O C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(c2nocc2Cl)=O)C1 Cc1ccc2scc(CC(=O)NCCN(C(=O)CC3CC=CCC3)C)c2c1 c1(CC(=O)N(CCC(C(C)C)NC(c2cnn(C)c2)=O)C)c(F)cccc1F C1(C(=O)NC(CCNC(C2(CC)CCC2)=O)(C)C)CC(Cc2ccccc2)=NO1 C1(CC(=O)NCCCCCN(C(=O)Cc2ccc(Cl)nc2)C)CCC(C)CC1 Cc1c(F)ccc(C(=O)N(CCCS(C)(=O)=O)C)c1N C(=O)(C(C)(C)CCCc1ccccc1)NCC(CNC(CC1(CC)CCC1)=O)F C1(=O)CCCCCC(=O)O1.C1(C)(COCC)CCN(C(=O)CC)CC1 C(=O)(CCCCC(C)(C)C)N1CCC(CNC(CCC(C)C)=O)C(F)(F)C1 C1(NC(C2C(C(=O)OC)C=C2)=O)CN(C(c2cc(C)cc(O)n2)=O)C2CCCC12 c1(N2CCCC(CC=C)(NC(=O)C(C)OC3CCCC3)C2)ncnc2[nH]ccc12 c1(C(N2C(CNC(CCCC)C(=O)OCC)CC(OC)C2)=O)nccc2occc12 N1(C(C2CC(C)C2)=O)CC2CCCC1C2CNC(c1c(Cl)n[nH]c1C1CC1)=O C1(NC(C2C(C(C)C)C2)=O)CCC(NC(c2csc(Cc3ccccc3)c2)=O)C1 N1(CCCCCCSC)C(=O)CN(CC23CCCC2C3(F)F)C1=O c1(CC(N2CCOCC(NC(CCC(N)=O)=O)C2)=O)c(F)cc(F)cc1F N(C1CN(C(c2ccc3c(c2)CC3)=O)Cc2ccccc21)C(CCOCC#C)=O C1(NC(c2c(CC)c(C)ccc2)=O)CCCCN(C(=O)CNC=O)CC1 Cc1cccc(C(N2CCOC(CN(C(=O)C(C)OCC3CC3)C)C2)=O)c1C C1(C(=O)NCCCOCCNC(=O)CCc2cn[nH]c2)C2CC3C(C2=O)C13 Cn1cc(C(=O)NC2CC(NC(=O)CCC3CCCC(=O)N3)CC2O)ncc1=O N1(C(c2ccc(Cl)c(Cl)c2)=O)CCN(C(C2CCc3nnnn3C2)=O)CC(O)C1 N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ncncc2C)=O)C(CCOC)C1 N1(c2scc(C)n2)CCN(C(=O)CC(C)C2CCC(C)O2)CC1 N1(Cc2cnc(C)s2)CC(NC(=O)C(C)Sc2ccccn2)C(C#N)C1 c1(C(=O)NCC(C)(CO)NC(=O)CC2C=CCCC2)ccc(F)cc1Br Cc1nc(C)c(C(N2CC(NC(=O)C(C)Cc3ccco3)CC(F)C2)=O)c(C)n1 C(=O)(C(C(C)(C)C)NC(N)=O)NC(C1CCN(C(Cn2ccc(C)n2)=O)C1)C N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C)CN(C(c3cnn[nH]3)=O)CC2(C)C1 c1(OCC)ccc(OCC(=O)NC2CCC(NC(=O)CC(CC)OC)CC2)cc1 c1(C(=O)NCCC2(OC)CN(C(=O)Cc3cnnn3C)C2)nccc2ccsc12 CC(C)CC(CNC(=O)C(C)(O)C1CCC1)NC(=O)CSc1ccc(F)cc1 c1(-n2c(C(c3ccc(C)cc3)NCC(C)CO)nnn2)c(C)cccc1C c1(NCc2c(C)scc2)ccc(C(N2CCC(Br)C2)=O)cn1 CC1CCCC=C1C(=O)N(C)CC1CCCN(C(=O)C(F)(F)c2cscn2)C1 C1(C(=O)NCC2CN(C(c3cccc(COC)c3)=O)C2)(OC)CCCC(C)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)c(F)c2)cc(O)nc(OC)n1 N1(C(c2c(C)snn2)=O)CCOC2(C1)CN(C(=O)CCC1CCCC1)C2 C1(C(N(CC(=O)NCC(O)CO)C)=O)CCCC(F)C1 C1(NC(C(C)OCC2CC2)=O)CN(C(=O)C(C2CCC2)C2CCC2)CC1C N1(C(=O)OC(C)(C)C)C(C(=O)NCC2(CO)CC2)C2CC1(CC1CC1)C2 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C(=O)N(C)C)C(F)(F)CC1 c1(CC(=O)NC2CC(NC(c3cscc3F)=O)C2)cn2c(n1)CCCC2 C1(C(=O)NCC2CC2NC(C2C=CCS2)=O)CCC(F)(F)CC1 N1(CCOC(C)C2CC2)CCC(Cc2ncoc2C(F)(F)F)C1 CC1(C)C(NC(c2n[nH]cc2F)=O)CC1CNC(=O)CCOC1CCOCC1 c1(-c2ccc(CNC)cc2)cc(C(N2CC3COCC3C2)=O)nc(=N)[nH]1 c1(Cc2nc(C(C)(C)NC(C)=O)sc2)cccc(S(=O)(=O)C(N)=O)c1 C#CCC(C(=O)NCC(=O)NC(C)(C)C)NC(=O)C(CC)N(C)C C(=O)(C1=NOC2(CCC2)C1)NC1CC(C)CN(C(c2cccn3nncc23)=O)C1 N1(C(CC2CC(OC)C2)=O)CC(C(=O)OC)CC2CCCCC12 C(=O)(CC(O)CC(C)(C)C)N1C(CCNC(C2(NC(C)=O)CCC2)=O)CCCC1 CC(CS(C)(=O)=O)C(=O)NCCC1CCCN(C(=O)C2=CC3CCCC23)C1 CC1CC2(CCN(C(c3cncc(C(C)(F)F)c3)=O)CC2)CN1C(=O)C1=CCC1 C(CN=c1cc(Cl)c(O)n[nH]1)(N(C(C(CCSC)O)=O)C)C1CC1 N1(Cc2cnc(SC)nc2)CCC2(CC1)CC(C(=O)N=c1cccn[nH]1)CO2 N(C1CCCn2cnnc21)C(CC1(C)N(C(C2(CCN(C)C)CC2)=O)CC1)=O c1(C(=O)NCCC2CCN(C(=O)CCC(F)F)C2)ncc(Cl)cc1Cl c1(C(=O)NCC(CC)NC(c2sc(COC)nc2C)=O)noc2cc(F)ccc12 C12(NC(C3(C)CCCCC3)=O)CCCN(c3nncs3)CC1C2.c1(C)cn[nH]c1.N C(=O)(C(O)CCNC(=O)C(C#N)CC)NCCCCCC Cc1ccc2nonc2c1C(=O)NC(C)CCNC(=O)CCCc1n[nH]c(=N)s1 CC(c1ccco1)=CC(N1CCN(CC2CN(C(=O)OC(C)(C)C)C2)CC1)=O c1(C(N(CCOC)CCNC(C2C3COCC23)=O)=O)cc(Cl)cnc1OC c1(C(N2CCN(C(C3CCc4nccn4C3)=O)CC2)=O)c[nH]c2nc(Cl)ccc12 CC1CN(C(=O)CS(=O)(=O)NC(C)(C)C)CC(C)C1NC(=O)Cn1nccn1 C1(C)(CC)NC(=O)N(CC(N2CC(NC(c3cccn4nncc34)=O)C2)=O)C1=O CC(C)(CCC#N)C(=O)N1CCCC2(NC(C3CCOC3)=O)CC2C1 C(=O)(C1CCCn2nccc21)NCC(C)N(C(C(C)Sc1ccccc1)=O)C C1(SC)CCC(N=c2[nH]c(=NCc3nncn3C(C)C)c3ccccc3[nH]2)C1 c1(N2CC(S(C)=O)C2)ncnc2c1ncn2CC1(C)CC1(F)F C#Cc1ccc(C(=O)N(CC(C)O)CCNC(C2(C)CCCS2(=O)=O)=O)cc1Cl C1(N(C)C(=O)NC2CCN(S(C)(=O)=O)C2)CCCC(N)C1 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CC2)cnc2ccccc2c1OC c1(C(=O)NCC2(COC)CN(C(=O)CN3CC(C)C3)C2)ccc(O)cc1.C1(C)CC1 C1(F)(CNC(C2C(CC)C2)=O)CCCN(C(c2cnc3n2CCS3)=O)CC1 C1(C(=O)NCC(CC)NC(C2(C)COCCO2)=O)CC2(CCC2O)C1 CC1CC(N(C(=O)CCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)C1 N1(C(c2nc(N(C)C)oc2)=O)CC(F)(F)CC1CNC(C12CCC(F)(CC1)C2)=O CC(C)(CNC(c1conc1CNC(C1CCCC(=O)CC1)=O)=O)CCCO Cc1cccc(O)c1C(=O)NC(CCCNC(=O)C(C)(C)F)c1ccccc1 Cc1c(F)ccc(C(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)C2)c1N N1(C(c2c(C)nncc2)=O)CCC(C2CCN(C(C3(F)CC3C)=O)C2)CC1 c1(C(N(C2CCN(C(C3COC(=O)C3)=O)C2)C)=O)cnn(-c2ccccc2)c1F c1(C(N(C2CCN(C(c3nncn3CC)=O)C2)CCC)=O)ncc(Br)cn1 C1(C)(C(=O)NC2C3CC(NC(c4n(C)cnc4)=O)CC32)COC(C)(C)CO1 C(=O)(CCC(CC)CCCC)NCC(CNC(CCC(=C)Cl)=O)(C)C N1(C(c2occc2C)C(=O)NC)CC2C3CCC(C3)C12 c1(CNC(C2CC2C(=O)NCc2ccnn2-c2ccccc2)=O)cccc(O)c1 N1(C(C(C)CF)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 C(CC(CO)C(C)C)NC(C(C(C)C)NC(=O)C=CC1CCCN1C)=O N1(C(C)=O)CCOCC1C(N1CC(CNC(=O)CC2CCC2)C1)=O N(CP(C)(C)=O)(CC(N1CCCC(c2n[nH]c(=N)o2)C1)=O)C(=O)OC(C)(C)C C1(C(=O)NCC(C(C)(C)C)NC(c2cscc2C#N)=O)CC2CCC1CC2 C(=O)(NN1CCCC1C(=O)NCC1(C)CCC(=O)N1C)c1c(C)n(C)nn1 c1(C(=O)NC(CC)(CNC(=O)C(F)n2cccn2)CC)c[nH]c2cc(F)ccc12 C1(N(C(C=C(C)C)=O)C)CC2CCC(C1)N2C(=O)CCc1ccc(O)c(O)c1 C1(NC(C2NC(=O)OC2)=O)(CNC(C2(O)CCOCC2)=O)CCCCC1 N1(C(c2cc(C(=O)OC)n(C)n2)C(=O)NC2CCCCC2)CCC2CCN(C)CC12 C(=O)(C1=CCCCO1)NC1CN(C(CCOc2ccc(C(N)=O)cc2)=O)C2C1C2 c1(C(=O)NCC(CC=C)NC(C2(C(C)C)CNC(=O)C2)=O)ccc([N+](=O)[O-])cn1 c1(CC)noc(CC)c1CC(=O)NCCC(C)(C)NC(c1occc1CSC)=O C(=O)(C#CC(C)(C)C)N(C1CCCN(C(c2ccc(NS(C)(=O)=O)nc2)=O)C1)C C1(N(C(=O)CCC2(CC3CCCC3)CCOC2)CCC)CCc2c[nH]nc2C1 c1(C(N2CC(C(N3CCC(C#C)CC3)=O)C(C)C2)=O)cccc2c1CCC2 N1(C(n2ncc(C)c2N(C)C(=O)C2CC2)=O)CC2CCC(CSC)C2C1 C1(CC(=O)N(CC)Cc2cncn2C)CN(C(c2c[nH]nc2C)=O)C(C)(C)C1 N1(c2cc(OCC)ncn2)CCCOC(CNC(=O)CN2CC(=O)N(C)C2=O)C1 C(=O)(C1CCCn2c(Br)cnc21)N1CCCN(C(C(C(C)C)(C)O)=O)CC1 c1(C(=O)NCCOCCNC(c2nc(CC)oc2)=O)n[nH]c2c1CC(C)CC2 c1(C(=O)NC2(CC=C)CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)ccn(O)c(=O)c1 C(=O)(C1=CC(O)C(NC(=O)C#CC2(C)COC2)C1)Nc1c(OC)nsc1 N1(C(C(C)C)=O)CCN(C(C2CC2C(=O)NC(c2ccc(F)cc2)CO)=O)CC1 CCC(CC(=O)NC1CN(C(c2cnncc2OC)=O)C2CCCC12)CC(C)C CCCC(CNC(=O)COCC(F)F)C(=O)NCc1cn(CCC)nn1 CC1(C)C2CNC(c3ccc(SC(F)(F)F)cc3)C12 C1(NC(C=CC)=O)CCN(C(c2cc(CCO)on2)=O)C1C1CC1 C1(O)(CCNC(C(C)CC2CCCO2)=O)CCN(C(c2ccoc2Cl)=O)CC1 Cn1ncc(C(=O)NC(C(=O)NC2CCN(C(N)=O)C2)C2CCCO2)n1 C#CC1CN(C(=O)CSCCC)CCN1C(C1CCS(=O)(=O)N1C)=O c1(C(N2CCC(CN(C(CCOCC)=O)C)CC2)=O)nc(O)nc(O)c1N c1(NC(=O)CC2CN(Cc3ccc(O)c(F)c3)CCO2)nccc(Cl)c1I c1(C(C2CCCN2C(c2ccc(Oc3ccccc3)s2)=O)=O)ccnc(Cl)c1F c1(CC(N2C(CN(C(C3(COCC)CC3)=O)C)CCC2)=O)cnn(C)c1C C1(C(N2CC(CC(C#C)C)C2)=O)CCC(NC(=O)CC2CCC(C)CC2)CC1 c1(NC(c2n(CCOC)nnn2)C2CCCSC2)ccc(N(S(C)(=O)=O)C)cc1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(Cc2c(C)nn(C)c2Cl)=O)CC1 CC(C)(C(=O)N1CCC(C2CCCN2C(C2CCCC2)=O)C1)C(F)(F)F N1(c2n(Cc3c(Cl)cc(Cl)cc3)nnn2)CCc2nc[nH]c2C1c1ccc(Br)cc1 N1(C(C(C(C)C)(C)C)=O)C(CNC(=O)CN2CCNC(=O)C2)CC2COCC12 c1(C(=O)NC(C)(C)CNC(=O)CCn2ccnc2)cccn2nncc12 N1(C(c2c(C)n(C(C)C)nn2)=O)C2CCC1CN(C(c1c[nH]ccc1=N)=O)C2 C1(O)(CCNC(C(Cc2ccccc2)NC(N)=O)=O)CCCN(C(=O)C(F)F)C1 C1(C(=O)NCC(C)CCCO)CCCN1NC(=O)C1(C#N)CCCC1 C1(C(=O)NCC(C)Cc2cn[nH]c2)COCCN(C(=O)C2=CCCC2C)C1 N1(CC(=O)N(C(=O)C(C)Sc2ccc(Cl)cc2)CC)CCN(CCCOC)CC1 c1(C(C)C)nn(C)cc1NC(=O)CCCCN(C)C(c1cc(C2CC2)[nH]n1)=O C1(NC(c2onc(CC)n2)=O)CN(C(=O)CCc2cncc(C)c2)CCC1C Cc1cc(C(=O)NC(C)(CO)C(=O)N2CC(F)(C#N)C2)oc1C N1(C(C(c2n(C)ccn2)(F)F)=O)CCOC(CCNC(=O)CCN2CCCC2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(N2CC(CSC)C2)=O)(CF)C1 c1(OC)cncc(C(=O)NC2CCC(CNC(C3CC4CCC3O4)=O)C2)c1 C1(C(=O)NCC2CCC(F)(CNC(C3C(=C)CC3)=O)CC2)CC2(CC(C)=NO2)C1 C1(CC(C)(C)C)CCN(C(C23CC(n4cc(CNC(N)=O)nn4)C2C3)=O)C1 c1(CC(=O)NC2CN(C(=O)CCC(F)(F)F)CCC2F)c[nH]c2ccccc12 N1(C(C(CC)CCOC)=O)CCCC2(C1)CN(C(=O)CCc1cccc(O)c1)C2 N1(C(CC(CNC(c2n(CC)nnc2)=O)C)=O)CCOc2ccccc21 c1(C(N2CCCC(NC(CCC=C)=O)(CC)C2)=O)cc(Cl)ccc1[N+](=O)[O-] C=CC1CN(C(c2cc(C)ccc2OCC)=O)CC1NC(=O)C(C)(C)CO C1(CNS(CCC)(=O)=O)(NC(=O)C(Cc2ccccc2)N(C)C)CCOCC1 N1(C(CCc2ccc(C)o2)=O)CCC(C)C(NC(=O)CCSc2n[nH]c(C)n2)C1 C1(CC(N2CCC(C)(NC(c3cnccn3)=O)CC2)=O)CCn2cncc2C1 N1(C(Cn2cc(C(=O)NC)nn2)=O)CCN(C(=O)C2=NOC(C)C2)C(CF)C1 C(CN=C(NCC1CC(F)(F)C1)NC(C1CCCO1)C)c1c(C)nccn1 C(=O)(C1=CC2(CCN(C(=O)C(=O)C(C)C)C2)C1)NC(CCCC)CC CC(C)CCC(O)C(=O)N1CCCCC(CNC(=O)CCc2ccc(Cl)nc2)C1 C1(O)(C(C(=O)N(C2CCCO2)CC)F)CN(C(=O)COC(C)(C)CC)C1 N1(c2nnc(Cc3cccc(OCC)n3)n2CCOC(C)=O)CCCC(C)CC1 Cc1cc(C)c(C(=O)NCC2CC3CCC2N(C(=O)C(C)O)C3)cc1Br c1(C(=O)NCC2CC(NC(C(C3CC3)SC)=O)C2)c(C)nc2sc(C)cn12 C(=O)(C1OC(=O)c2ccccc21)N(CCN(C(CC1(C=C)CC1)=O)C)C N1(C(CCC2C(C)(C)C2)=O)CCOC(CNC(c2ccoc2Br)=O)C1 C(=O)(C1CCCn2nccc21)N(CCNC(c1cc(OC)c(O)c(Br)c1)=O)C N12CCN(CC1)c1ccnc(n1)COC2=O.c1(CCNC(C)(C)C)cnc[nH]1 N1(C(c2oc(C)c(CO)c2)=O)CC(CNC(=O)C(F)C2CCOC2)CCC1C N1(C(CNC(CC)=O)=O)CCOCC(CNC(C2(C)CCOC(C)C2)=O)C1 N1(C(C(CC)SC)=O)CCCC(C2CCN(C(c3nc(C)ncc3Cl)=O)CC2)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(c1ccc(=O)oc1)=O c1(C(N2CC(NC(COC)=O)C(O)C2)=O)c(Cl)ccc(F)c1C c1(OCC=C)ccc(CNc2cccc(N3CCOCC3=O)c2)cc1Cl C1(NC(C2=CCN(C)C2)=O)COC2C(NC(C3CC34CC4)=O)COC12 C1(C(=O)NC(C2(C(=O)NCc3ccc(F)cc3)CC2)C)CC(C(C)C)=NO1 c1(C(=O)NCCCNC(c2cscc2C(F)F)=O)ccc2c(c1)OCO2 C12(CNC(c3c(C)csn3)=O)CCCC1CN(C(c1cccn1C)=O)C2 Cc1ccc2sc(CN(C3CCN(C(=O)COc4ccsn4)C3)C)nc2c1 CCC(F)C(=O)NCC(O)CN(C)C(c1cnn(C(F)(F)F)c1)=O C1(N(C(C2N(C(C(CC)OC)=O)CCCC2)=O)C)CCCC(C)(C)C1 c1(COC)sccc1C(N1CC(C(C)NC(C2CN(CC(F)(F)F)C2)=O)C1)=O C1(C(N2CC(O)(CNC(CNS(CC)(=O)=O)=O)C2)=O)CC2CCC1C2 O=S(=O)(c1ccc(OC(F)F)c(Cl)c1)NCc1ccc(F)cc1F C=C1CC2(C1)CC(C(N1CCOCC(NC(=O)C(c3ccc(C)s3)C)C1)=O)C2 CC1(C)CCCN(C(c2cnc(Cl)c(N)c2)=O)C1CNC(=O)Cc1cccnc1 C1(C(=O)NCc2oc(C(=O)NCc3c(C)ccs3)c(C)n2)CC(C2CC2)=NO1 C1(CNC(C(C)=C(CC)C)=O)CN(C(=O)C=CCN(C)C)C2(CCOCC2)C1 c1(C(N2CC3(CN(C(C(C(COC)C)C)=O)C3)C2)=O)ccc2ccncc2n1 c1(C(N(C(CN(C(C(CC)=CC)=O)C)C)C)=O)ccnc(N2CCN(C)CC2)n1 c1(C(=O)NC(CC)(C)C(N)=O)nc(C)c(C)cc1N C1(CNC(COCCCC)=O)CC12CCN(C(c1ccsc1CC)=O)CC2 Nc1c(-c2cn(CC3CCN(c4ccc(F)cc4F)C3)nn2)cccc1O c1(C(N2C(CNC(c3c(C(C)C)onc3)=O)CCC2)=O)cccn(C)c1=O N1(C(CN(CCCCCC)C)=O)CCC2CCN(C(=O)Cc3nc(C)cs3)CC12 CC(CC(C)C(F)F)NC(C1CC(C)CCN1C(=O)CC1CCCC(C)O1)=O C(c1ncccc1C)=CC(=O)NC1C(CNC(c2c(COC)cco2)=O)CCC1 c1(NC(C2CN(C(CNC(CCC(C)C)=O)=O)CC2O)=O)ccc(F)cc1Cl c1(C(N(CC(CNC(Cc2cc(C)on2)=O)(C)C)C)=O)cccc([N+](=O)[O-])c1Cl N1(C(C(c2ccc(F)cc2)CC)=O)CCC(NC(=O)Nc2cnncc2C)CC1 N1(C(CCC(C)OC)=O)CCCCC(C(=O)NC(CO)CCC2CC2)C1 N1(C(CCC)=O)CCC2(CCCCC2NC(=O)CN(C)CCO)C1 O=C(CCC(F)(F)F)NC1(CCCCNC(=O)COC2CCCO2)CC1 c1(C(=O)NC(C(=O)NC(CC)C2CC2)Cn2cncn2)cc(C)sc1N c1(C2(NC(C3C(NC(C4C(CCC)C4)=O)C3)=O)CC2)cccc(OC(F)(F)F)c1 c1(C(=O)NCCC2CN(C(C(C)(C)C3CCCO3)=O)C2)ccc(N)cc1Cl c1(-c2ccn(CCCC3(F)CCN(C(=O)OC(C)(C)C)C3)n2)cc(F)ccc1F CCC(C#N)C(=O)N1CC(O)(CCNC(=O)C2CC2)C1 c1(OCCC)cccc(C(=O)NCC2(O)CCN(C(=O)Cn3ccc(C)n3)C2)c1 c1(C(N(CCCCNC(C=C(C)C)=O)C)=O)sc2cccnc2c1Cl C(=O)(CCC(N)C(=O)O)N1CCCC(C(=O)NC(C)CC(N)=O)CC1 C1(C)(C(=O)NCCN(C(CNC(C(CC)CC)=O)=O)CC)OC(C)(C)OC1C C#CCCCCCCC(=O)N1CCC(C(N2CCC(OC)CC2)=O)C1CC c1(OC)cc(C(N2CC(O)(CNC(c3c(C)ccnc3O)=O)C2)=O)nc(C)c1 c1(C(=O)NC(CC)CN(C)C(C23CCCC2(C(N)=O)C3)=O)ccc(O)c(C)c1C c1(CC(=O)NC2C(NC(C(CCOC)C)=O)CCCC2)ccc2c(c1)CCCO2 c1(CC)cc(NC(c2nnnn2C2CC2)CC2CCOC2)ccc1C c1(OC)cc(C(N2CC(NC(c3nc(=N)cc[nH]3)=O)CCC2C)=O)cc(C)n1 C1(CNc2ccnn2CC(F)F)CNCC1(F)CO.O=C(C(=O)C1CC1)NCC1CC1 c1(NC(c2ccc(C3CCCCO3)cc2)=O)cc2cc(Br)ccc2s1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCN(C(c2cc(Br)no2)=O)CC1O C(=O)(CC(C)(C)CCOC)NC1CC2(CC(CNC(C3C(OCC)C3)=O)C2)C1 C1(C(N2C(C#C)CC2)=O)CCN(C(c2cccc(OC)c2)=O)C(C)(C)C1 N1(C(C(CNC(C2(CCOC)CC2)=O)O)=O)CC(C)(C)C1C(N)=O Cc1ccc(NC(C2(NC(=O)C(c3ccnn3C)C)CCN(C)C2)=O)cn1 N1(C(CCCSC)=O)CC(C(=O)N(C)CCn2cnnc2)C(C2CC2)C1 c1(C(N2CC(C)CC(NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)ccn2c1CCCC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CC1)CCN(C(C1CCCC1C)=O)C2 n1(CC(C)C(N2CCC(O)C(NC(=O)C=C3CCC3)C2)=O)ncc2c1CCCC2 c1(C(N2CCC3CCNC(=O)C23)C(=O)NCC=C)sc2ccccc2c1Br c1(C(C)OCC)nc(CC(=O)NCC(O)CNC(=O)Cn2cn[nH]c2=N)cs1 N1(C(=O)C=CC2CCCO2)CC2CCCC(NC(C3CC(F)(CO)C3)=O)C2C1 C12(C(=O)NC(C3CCCCC3)C#C)CC(CO1)N(C(c1ccc(CO)s1)=O)C2 Cc1ccc(CC(=O)N(C)CCN(C(=O)C=Cc2nc(C)co2)C)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)C=CC(C)C)C(C2CC2)C1 C1(CC(N2CCN(C3CCN(C(CCC#N)=O)C3)CC2)=O)CC2CCC1CC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCC(C1)N2C(=O)C(=CC1CCCC1)C C1(NC(C(CC)F)=O)CN(C(=O)CON=C2CCCCCC2)Cc2ccnn2C1 N#CC1(C(=O)NC(CNC(C2CC3CCC2O3)=O)CC(F)(F)F)CCCCC1 Cc1cc(C)n(CC(N2CCCN(C(=O)CCCC(C)(F)F)C(C)C2)=O)c(=O)n1 C=CC(C)(O)C(=O)N1CC2CC2(NC(=O)C=CC(CC)=CC)C1 Cc1ccc(NC(C2CCCN(C(=O)Cn3cccnc3=O)C2C)=O)cc1C CS(=O)CCC(=O)NC(C1CCCC1)CNC(=O)C=Cc1cc(C(N)=O)co1 CCCCCCCNC(=O)COC1CC(NC(=O)C(O)CC2CCCC2)C1 c1(C(=O)NC)ccc(Cl)c(NCc2cn(C)nc2C(F)(F)F)c1 CCC(C)C(CNC(=O)COCCNC(=O)CNC(C)=O)OC C1(N(C(CN(CCC)C)=O)C)CN(C(=O)CNC(=O)NCC2CC2)C1 c1(C(=O)NCCC(C)N(C)C(c2cc(Cl)on2)=O)ccncc1F c1(C(N2CC(O)(CNC(CCc3c(C)n[nH]c3C)=O)C2)=O)ncnc2c1CCC2 C1(NC(c2ccc(C)c(C)n2)=O)CN(C(=O)C(C)Cc2ccco2)CC(F)(F)C1 N1(C(COCC=C)=O)CCOC2(CCC(NC(c3cc(O)ccc3C)=O)CC2)C1 N1(C(CNC(Cn2c(C)ncc2)=O)C)CCN(C(=O)C(C)SC(F)(F)F)CC1 C1(F)(C(=O)NC(C)C(=O)NC(C)(C)C)CCN(C(C2CCC(=O)N2C)=O)C1 N1(C(CC(=O)NCC)=O)CCN(C(C23CC(CC(C)O2)C3)=O)CC1CCO C(=O)(CC(C(F)(F)F)NC(=O)C(F)(F)C(C)(C)O)NC(C)CC(C)(C)O CC(C(=O)NCC(C(=O)N1CCC(CC(C)(C)C)C1)N(C)C)C(C)(C)C c1(CNC(C(CC)N(C)C)=O)cccc(C2CCC2)c1 N1(c2cc(NCC3(Br)CC3(F)F)nc(C)n2)CCCNC(=O)C(F)(F)C1 c1(NC(C(C(C)(C)C)NC(C2=C(C)CC2)=O)=O)ccc2c(c1)OCC2 c1(C(=O)NCC(CC=C)NC(=O)Cn2nnc(C)n2)cc(C)nn1C c1(CCC)cc(C(=O)NCC(C)(C)CNC(=O)CC(C)n2cccn2)[nH]n1 c1(C(=O)NCCNC(c2nc(C)oc2)=O)cc2c(C)nn(-c3ccccc3)c2s1 N1(C(C(C)OCC#C)=O)CC2CC(C(=O)NCC3CC3CC)(C2)C1 c1(C(=O)NC(CC(C)C)CNC(C2(F)CCCN(C)C2)=O)cncc2c[nH]nc12 N1(C(c2c(C)nc(CC)o2)=O)CC(N(C)C(C2CC2c2ccsc2)=O)C(C)(C)C1 C1(C2CCOCC2)(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)CC1(F)F n1(CC(N2CC(N3CCN(C(C=C=C(C)C)=O)CC3)C2)=O)cc(F)ccc1=O C(C(C)(C)C#CC(=O)NC1CCCN(CC)C1)NC(c1c(CC)non1)=O c1(CNC(CC(N2CC3CC2CS3=O)=O)Cc2cccs2)cccc2c1OCCO2 C1(NC(C2(C)CCC2)=O)COC2(CCCN(C(C3CC(F)(F)C3)=O)C2)C1 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(=O)Cc1cnc[nH]1 C=CCC(C(=O)N(CC(=O)NC1CC1)C)NC(C1CC2CC2C1)=O C1(CC(NOCC2CC(=C)C2)=O)CCCCN1C(=O)C(n1ccnc1C)C N1(C(C2C(CC)OCC2)=O)CCC(CCNC(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(N(C2CCCN(C(=O)CC3(CO)CCC3)CC2)C)=O)CC12CCOCC2 CC(Cc1cnco1)C(=O)NCCCC(C)NC(=O)CSc1ccccc1 C1(CNC(C2CC=CC2)=O)CCN(C(c2cc(O)ccc2Br)=O)C12CCC2 C1(CNC(=O)Cc2cccnc2)COCCN(C(c2cn3c(n2)SCC3)=O)C1 c1(CC)cnc(N(C2CCNCC2F)C(=O)Cc2ccccc2Br)nc1 O=C1CCC2(C(=O)NCCNC(c3ccc4occc4n3)=O)CCCCC2N1 C(c1ccc(Cl)cc1)=CC(N1CCC(F)(c2ccccc2)CC1)=O C1(OC)Cc2ccccc2N(Cc2cnc(C(C)C)s2)C1C C(=O)(C(C(C)(C)C)N(C)C)N1CC2C(CNC(c3c(C)ccs3)=O)(C2)C1 Nc1c(C(=O)NCC(O)CNC(c2cnn3cnnc3c2)=O)ccc(Br)c1F CC(C(C)(C)C(=O)NC1(C2CC2)CC1)NC(c1cnc2n1CCC2)=O C(=O)(CC(C)(C)CNC(c1ccc[n+]([O-])c1)=O)NCC(C)N(C)C1CC1 N1(C(C(C)NC(C)=O)=O)CC2(CO)CC1(C(=O)NCc1cncn1C(C)C)C2 C1(C(=O)Nc2cc(C(N)=O)ncc2)CN(C(c2c(Cl)cccc2Cl)=O)CCC1O c1(-c2cn(C(C(=O)NCC(C)OCC=C)C)nn2)cc(OC)ccc1Br Cn1nc(C(=O)NCC2CCN2C(c2conc2C2CCC2)=O)c2c1CCSC2 C(c1cncs1)=CC(=O)NC(CC1CCOCC1)C(=O)NCCC1CC=CCC1 C1(C(N(CCCOC)CCO)=O)C2CCC(C2)N1C(=O)C1=NOCC1 Cn1c(=O)n(CC(=O)NCCC(C)(C)NC(=O)CCP(C)(C)=O)c2c1CCOC2 N1(CC(=O)NCCOCCN(C(c2c(SC)n(C)nc2)=O)C)CCN(C)C(=O)C1 N1(C(Cc2c(C)n(C)cn2)=O)CC2COCC2(C(=O)NOCCCC(F)(F)F)C1 N1(C(=O)OCC(C2CCC(C)C(C)C2)=O)CC(C(=O)NC(C)(C)C)C2(COC2)C1 N1(C(C2(C)CC=CC2)=O)CCC(F)(C(=O)Nc2cnc(Cl)nc2)CC1 N1(CCN(C(CC(C)C2CC2)=O)C)CCN(C(c2cnc(C3CC3)nc2)=O)CC1 CCCC(CC)C(=O)N1CCC(CNC(C2(C(F)F)CCCC2)=O)C(O)C1 CC1(CCC(N2CC3(CC3)C2)=O)CCCN1C(=O)CCn1cncn1 C1(CC(=O)NC(c2ccc(C(NOC(C(C)C)CO)=O)o2)C2CC2)CCC(=O)NC1 N1(C(CCOCC#C)=O)CC(CNC(=O)CN2CCNC(=O)C2)C(F)(F)C1 C12(CC(=O)NCCC(C)N(C(=O)CC3C=CCC3)C)CCC(CC1)C2 c1(C(=O)NCCNC(C2CC=CCO2)=O)nc(-c2ccccc2)oc1C1CC1 C1(C(=O)NCC2CCC(NC(CC(=C)C)=O)CC2)CCn2c(C)nnc2C1 N1(C(=O)CCc2ccsc2)CC2CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2C1 C1(CNC(=O)C(F)=CCCF)CCCC12CCN(C(C1(O)CCCCC1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2CC2(Cl)Cl)=O)CC)noc2c1COCC2 N1(C(c2ccc(=N)[nH]n2)=O)CC(C(=O)NCC2CCCC(CO)C2)C(F)(F)C1 CC1(NC(=O)C(CCC2CC2)NC(=O)CCc2nncs2)CC2CCC1C2 C(N=c1nc2scnc2c(N(CCC)C(C2(CO)CCCOC2)=O)[nH]1)CCC=C N1(C(CCSCCC)=O)CC2CCOC2(CNC(c2cn(C)nc2O)=O)C1 C1(CC(=O)NCCCCN(C)C(c2cn(CC3CCOC3)nn2)=O)COC2(CCC2)C1 C1(NC(c2cc(Cl)sc2Cl)=O)CN(C(=O)CCN2CCC(F)C2)CCC1F C(=O)(C(F)C(C)CNC(C1(CC)CCOCC1)=O)N(CC#CC)C c1(-n2cc(C3C(OC)CN(C(C4(CCC)CC4)=O)C3)nn2)nnc2ccccn12 C1(NC(C(C)C2(O)CCC2)=O)CC(C(=O)NCc2ncc(CO)[nH]2)CC1O c1(C(N(CCC(C)NC(=O)CC2COCCO2)C)=O)cnn(C(C)C)c1F c1(C(N2C(CNC(=O)CCn3cc(Cl)cn3)CC2)=O)cc(Br)sc1Cl c1(NC(C2CC3(CC(OC)C3)C2)=O)ncnc2c1CCC2 c1(C(=O)NCC(CO)NC(=O)C(c2ccccc2)=O)ccccc1C(F)F CCCCCC(C)(C)C(=O)NC1CS(=O)(=O)CC1NC(=O)Cc1ccc(C)cc1 C#CCCN=C(NCC1(C2CC2)CC1)NCC(C)(O)CC C(=O)(CCC1=NNC(=O)CC1)NC1CCCN(C(C(CC#C)O)=O)CC1 C1(CC)CN(C)CCCN1C(C1CN(C(=O)Cc2ccc(C)nc2)CCO1)=O c1(-c2c(OC)cncc2)ccn2cc(C(=O)Nc3cnc[nH]3)nc2c1 CC(=NO)C1CC(C(=O)NCC2(C)CCN(C(=O)CC34CC(C3)C4)CC2)C1(C)C Cc1cc(=NCC(C)C#N)[nH]c(N2CCC(O)(c3cccc(F)c3)CC2)n1 C1(NC(=O)CCn2cccn2)CCOCC1NC(c1nccc(C(F)(F)F)n1)=O CC1=CCSC1C(N1CCC(OCC(=O)NC2CC(F)(F)C2)C1)=O c1(CC)cccc(NC(=O)CONC(=O)Cc2ccon2)n1 CC(C)CC(C)CC(C)C(=O)NCC1CC(C)N(C(=O)C(C2CC(F)(F)C2)O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)CNc3cnn(C)c3)C2(C)C)c(F)c1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C(n2ccnc2C)C)C1 CCC(C)C(CC(=O)NCCCCC1CC1C)NC(c1cocn1)=O C1(C(=O)NC(CC)(C)CC)Cc2cccc(OC)c2O1 C1(C)(NC(CCc2cc(C)[nH]n2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 c1(C(N2CC(C(C)(C)O)(SC(C)C)C2)C)cc(SCCC2(F)CC2)ncn1 N1(C(CCN(C)CC)=O)CCOC2(CCN(C(C3CCC(=O)N3CC)=O)C2)C1 C1(O)(C(=O)NC2C(C(C)NC(c3coc(C(F)F)n3)=O)CCC2)CCSCC1 N1(Cc2ccc(COCC)o2)CCC(C(=O)NC(c2ccncc2)CO)C12CC2 c1(C(N2CCN(C(C3N(C=O)CCC3)=O)C(C3CC3)C2)=O)n[nH]c2c1COCC2 N1(C(CC=CC(=O)NCCC)=O)CC2CC2(C(=O)O)C1 C1(CC(=O)OCC)Cc2ccccc2CN1c1cc(F)cc(F)c1[N+](=O)[O-] c1(C(c2nnnn2C)NC2(COC)CCCC2)ccccc1C(=O)N(C)C CC(C)C(CCC(=O)NCC1CC2(C1)CC(O)C2)NC(C1COCCN1C)=O c1(SC)ccc(CN2CCCCC2C(=O)Nc2ccc(C(=O)OC)cc2)cc1 C1(NC(C(C(CC)C)N(C)C(c2sccc2C)=O)=O)CCCCC12CCC2 c1(C(C2CC2)OC)cn(C2CC3(C(=O)N(C)Cc4cnoc4)CC23)nn1 N1(C(Cc2c(C)n[nH]c2C)=O)CCCCCC1CNC(C1COCCN1C=O)=O N1(C(C2CCN(C(C(C=C)CC)=O)CC2C)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC(CC(=O)NC(C2CCCC2)C)OC)ncc(F)cc1F c1(C(C)NC(C(CC)CNC(C(C)(C)OC=O)=O)=O)ccc2c(c1)CCO2 C1(NC(=O)C=Cc2cnc[nH]2)CCC(NC(c2ccncc2C2CC2)=O)CC1 c1(OCC)ccc(NC(=O)C(N2CC(O)C(O)C2)=O)cc1S(N)(=O)=O c1(C(N2CCC3CN(C(C4(C)CC4)=O)CC3CC2)=O)cccc2nc(O)ccc12 C(=O)(CC1=NNC(=O)C1)N(C1(C(=O)NC2(C)CCN(C(C)=O)C2)CC1)C1CC1 C1(NC(CN(C(C=C(CCC)CCC)=O)C2CC2)=O)CCOC12CCCC2 c1(SCC(N2CC(COC)(CNC(C3CC34CCCC4)=O)C2)=O)nc(C)cc(C)n1 c1(CCN=C(NC2C(C)C2)NC2(CO)CCCCCCCCC2)ccc([N+](=O)[O-])cc1Cl c1(C(N(C(CN(C(c2cncc(NC)c2)=O)C)C)C)=O)scc2c1OCCO2 Cc1cc(N(C)C)ccc1C(N1CCOCC1c1cn(CCO)nn1)=O c12nc(cc(Cl)n1)NC(=O)NC2C.c1(CNC2CC(OCCN(C)C)C2)ccccc1 c1(C(=O)NC(C2N(C(C3C(C=C)CC3)=O)CCC2)C)cc(C)c(Br)cn1 N1(C(C2(C)N(C(C3CCN(CC)CC3)=O)CCC2)=O)C2CCC1CC(=O)NC2 Cc1cc(C(=O)NCCC2(O)CCCN(C(=O)COC(F)F)C2)c2occc2c1 C12(C(N3CCCC(NC(C4C(C)(C)CO4)=O)CC3)=O)CCC(O1)c1ccccc12 C(CCCC(=O)N(C1CCN(C(=O)Cc2cccc(C(N)=O)c2)C1)CC)OCC c1(C(=O)O)ccc(Br)c(CNC2C=CS(=O)(=O)C2)c1F C(=O)(C(C(C)(C)C)NC(c1cnn[nH]1)=O)N(C(C1CCCC1)C)C C(=O)(CC(CC)C(C)C)CC.N1(C(CC2CO2)=O)CCOC(C)(C)C1 N1(C(CCC#C)=O)CCC(C)(C)C1C(=O)NCCN1CCCCC1 C1(C(N2CCCC2(C(=O)O)CO)C(=O)NC)C2CCCCC12 Cc1cc(C(N2CC3CC3(C(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(C#N)c1 N1(C(CC=C)=O)CCCC2C(NC(=O)CCOCCOC)C(C)(C)C12 C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(CNC(C(c2ccc(OC)cc2)(F)F)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC(O)C1C(=O)NC1(C)CCCC1C C=Cn1nncc1C(=O)N(C1CCN(C(c2ccc(C(C)=O)cn2)=O)CC1)C c1(NC(C2CC2C(=O)Nc2cc(O)ccn2)=O)cc(Br)ncc1[N+](=O)[O-] N1(C(c2cnc(CC)nc2O)=O)CC2CN(C(c3cc(Cl)no3)=O)CC2(C)C1 C(CC(O)CNC(C1CNC(=O)N1)=O)NC(=O)Cc1ccon1 c1(-c2onc(C3(OC)CCCOC3)n2)coc2c(F)cc(F)cc12 C=C(C)C1CN(C(C2CCCN(C(C3(F)CC=CC3)=O)CC2)=O)CCO1 C1(O)(CN(C(CC2(C=C)CC2)=O)C)CCCN(C(c2nc(Cl)sc2C(C)C)=O)C1 C(=O)(C1=CCCS1)NCC1C(NC(=O)NCC(=O)OCCCC)CCC1 N1(C(C(CC[S+](C)C)O)=O)CC2(CCCN(C(=O)CC3CC4(CC4)C3)C2)C1 Cc1cc(C(=O)NCC2CCN(C(c3ncoc3C)=O)C2)ncc1F c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)Cc3ccc(Br)cc3)CC2)c1 Cc1cc(Br)c(NC(C2CC3(C2)CN(C(=O)C(C)c2cccs2)C3)=O)cc1C C(=O)(C(C1=NOC2CC12)N(C1CC2(CCC2)C1)C)NCCC Cn1cc2c(n1)CCCC2C(=O)NCCOCCNC(=O)C1CCCc2c[nH]nc21 c1(NCc2c(C)nc(Cl)s2)cccc2cccc(Cl)c12 N1(C(c2cnn(C)c2C(F)F)=O)CC(NC(=O)C2=CCCC2)CC(C)(C)C1 C1(NC(C(CCOC)C)=O)CN(C(=O)CCCc2nc(C(C)C)no2)CCC1C c1(CC)cc(C(=O)N(C2CN(C(=O)CCC3CCCN3C(C)=O)C2)C)c(C)o1 N1(Cc2c(=O)cc[nH]c2)CC=CCC12CCOC2 c1(CCC)c(C(N2CCC(F)(c3cn(CC4CCCOC4)nn3)C2)=O)nnn1C n1(CC(=O)NCC#CCNC(c2cnc(C#N)s2)=O)nc(C(F)F)c2c1CCC2 C1(CNC(C2(CC=C)CCCN2C(=O)CC2CSCCO2)=O)CC2(CCO1)CC2 c1(NC(Cc2nc(C)oc2)=O)ccc2c(ccn2CC(=O)N(C)C)c1 c1(C(N2CCC(NC(c3c(C)cn(C)c3)=O)C(CO)C2)=O)cccn2nncc12 c1(C(N2CC(NC(C3N(C)CCC3)=O)C(F)C2)=O)cc(C(F)(F)F)nc(Cl)c1 C1(C(=O)NC(CCC)C2CCCC2)N(C(c2csc(C)c2C)=O)CCCC1(C)C c1(N(C)C(=O)OC(C)(C)C)cnc(C(N2CCOC(CCO)C2)=O)nc1 C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CCOC2(CCCC2)C1 C1(Cl)(C(N2CC(CC=C)(C(N3CCC3CC)=O)C2)=O)CCCCC1 c1(C(C)Nc2sc(Br)cc2N)cc(F)ccc1F c1(C(N(CC(CC)NC(c2ccnc(O)c2)=O)C)=O)cnc(C)c(C#N)c1 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(CCn2ncc(C)c2)=O)CC1 N1(C(c2cnc(C(C)OC)s2)=O)CC2CCCC(C1)N2C(=O)CSS(C)(=O)=O c1(NC(CNC=O)=O)[nH]nnc1SC(c1ccccc1)CNC(C1CS(=O)C1)=O C1(NC(C(CC=C)C)=O)CC2CC1N(C(c1c[nH]nc1-c1ccsc1)=O)C2 N1(C(c2c(Br)ccc(C)n2)C(=O)NC2CCOC2)CCC2(CC(C(F)F)=NO2)C1 c1(CC)ncsc1C(=O)NCC1CCCC1NC(=O)CC1C(CC)C1(F)F CC(CCCNC(=O)C(C)OC1CCCC1)NC(C1CC1c1ccccc1)=O c1(C(N2CCC(OCCNC(C(C=C)O)=O)C2)=O)nn(CC(F)F)cc1[N+](=O)[O-] C1(NCc2cncc(C)n2)CCCN(C(C2CCC(O)CC2)=O)CC1 Cc1cc(=O)c(C(=O)NC2(CNC(C3COC3)=O)CC2)nn1-c1ccccc1 C1(C(N2C(CNC(c3cnc(C)nc3C)=O)CCCC2)=O)CC2(C1)CS(=O)(=O)C2 C(CC(C(=O)Nc1ccc(OCC)nc1)NC(=O)CC1CNC(=O)O1)OCC Cc1cc(N)c(C(=O)NCC(F)CNC(C2CCC3CC2CO3)=O)c(F)c1 C1(C(=O)NCC2N(CC)CCC2)CC12CC(NC(=O)C(C)=C1CCC1)C2 c1(N2CC(NC(c3ccn(C(C)(C)C)n3)=O)C(F)(F)C2)ncnn2cc(Br)cc12 CN1CC(O)CCC1C(N1CC(CC(=O)NCc2ncc[nH]2)C2(CC2)C1)=O c1(CC(=O)NC(C)CCNC(=O)CSCC(F)(F)F)cc[nH]c(=N)c1 C1(C(=O)NCCOC2CCN(C(c3ccncc3F)=O)C2)CCC2(CC1)CC2 C(=O)(CCCCCCS(N)(=O)=O)N1CCC(C2(NC(C=COCC)=O)CC2)C1 C1(C(=O)NCC(COc2c(C)cccc2C)O)CCC2(COC2)OC1 C1(CC(C)NC(=O)C2CC2)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 c1(CC)c(C(=O)NC2CCC(NC(=O)C(C)P(C)(C)=O)C2)[nH]c2ccccc12 C1(NC(C2CC(OC)C(OC)C2)=O)CC(O)CN(C(c2c(Cl)n[nH]c2C)=O)C1 c1(OC)ccc(C(=O)NCC(O)CC2CCC2)c(N)c1F N1(C(c2c(CCCC)ocn2)=O)CCCC(CNC(=O)C(=O)NC2CC2)C1 C1(NC(=O)NCC(C#C)C(C)C)CS(=O)(=O)CN(C(C)(C)C)C1 C(=O)(C1COc2ccc(Cl)cc21)NC1C(CNC(C2CCC(C)C2)=O)CCC1 c1(OCC)cc(C(N2CCCC2CNC(=O)CC2CCC(F)(F)C2)=O)oc(=O)c1 C#Cc1ccc(OCC(=O)NCC2C3CN(C(=O)C(C)(O)COC)CC23)cc1 Nc1cccn(CC(=O)NC2CC(NC(c3cc(Cl)ccn3)=O)C23CCC3)c1=O c1(C(=O)NC2CN(C(Cc3cc(C(C)C)no3)=O)CC2F)ccc(S(C)(=O)=O)s1 C1(CC(N2CC(NC(=O)CN3CCCNC3=O)(CF)C2)=O)CCC2(CCC2)O1 c1(CC)nc(-c2nc[nH]n2)sc1C(=O)NCC(O)CNC(c1sc(F)cc1C)=O CC(CS(=O)(=O)c1cccc(Br)c1)NS(=O)(=O)c1ccc(Cl)s1 C(=O)(C1=CCC(C)CC1)N1CCC(CCOC)(NC(=O)C=CC2CCOC2)CC1 Cc1nc(C(N2CCC3(CCCN3C(C3CCC(=O)N3)=O)C2)=O)c2n1CCCC2 c1(NC(C23CC(C(=O)O)(C2)C3)=O)ccc2[nH]c(CN3CCC(F)(F)CC3)cc2n1 C1(C(N2CC(C)CC(NC(CN(C(C)C)C)=O)C2)=O)CCC(=O)C(C)C1(C)C CCCC(C)(C)C(=O)NC1CCCC(CNC(C2CC3CCC2O3)=O)C1 c1(NCC(CC)(CC)NC(=O)C(CC(C)C)OC)ccnc2nc(C)nn12 NC(=O)CCC(=O)NCC(CNC(c1cccc(OCC(F)(F)F)n1)=O)CO N1(C(C2CCC(CNC(C(C)(C)SC)=O)CC2)=O)CCOC2COCC2C1 C#CC1(O)CCN(C(=NCCc2c[nH]nc2C)NCC(=O)NC(C)COC)C1 N1(C(c2c(C)cno2)=O)CC2CCCC(CNC(=O)C3=C(Cl)CCOC3)(C2)C1 CC1=C(C(=O)NC(C2CCCCC2)CNC(=O)CCC(F)F)CCC1 c1(C(=O)NC2CC(N(C(C(C)SCC)=O)C)C2)c(F)ccc(Cl)c1[N+](=O)[O-] C1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)C(F)F)CCc2c(cnn2C)C1 CCC(C)(C)C(=O)NCCCCCN1CCN(C(=O)C=CC(C)C)CC1 c1(CC)c[nH]c(C(=O)NCC2(O)CC(NC(=O)C(C)OCC(F)(F)F)C2)c1 C1(CNC(c2ccc(OC)o2)=O)CC2CCC1N2C(c1cnnc(Cl)c1)=O C1(O)(CN(C(C=C(COC)C)=O)C)CN(C(c2csc(C(C)=O)n2)=O)C1 N1(CCOCC)C(=O)NC(c2cnc(N(C)C)s2)C(C(=O)OC)=C1C(C)CC C(=O)(C(C)CC(C)(C)C)NC(C(CO)NC(CC(C)NC(=O)OC(C)(C)C)=O)C C#CCCCC(C)C(=O)NC1CC2CC1N(C(=O)Cc1ccc(C)nc1)C2 O=C(CC1=CCOCC1)NCCC1CCC(NC(C2CNC(=O)N2)=O)C1 N1(C(Cc2c(OC)nccc2)=O)CCCN(C(c2ccnn2C2CC2)=O)CC1C CCCC(CCC)C(=O)NC1CN(C(c2ccc(N)c(Cl)c2O)=O)C1 O(NC(=O)C(C)(CSC)NC(=O)CC(C)C1CC1)C(COC)COC N1(C(c2cn(CCC)nc2C)C(=O)NC(c2nnn(C)n2)CC)CCC2C(O)CC12 C=C(C(=O)NC1CCCCC1NC(c1cccc(Cl)c1F)=O)C(F)(F)F C1(CC(=O)N(c2ncc[nH]c2=O)CC)CC(F)CN1C(C1CN(C(N)=O)C1)=O CC(C)C(CCC(=O)N1CC(CO)C1(C)C)NC(=O)C(C)CC1CCC1 N1(C(CCC=C)=O)CC(C=C)(CC(=O)NC(CC)C(=O)NC(C)C)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(C)Cc1cccs1 C1(C(=O)NCC(n2ccnn2)C)CC(C)(C)CCN1C(=O)C(N1CCOCC1)=O C(N=c1cc(C)nc(Cl)[nH]1)C1(C)CCC(NC(c2c(OC)cccc2F)=O)CC1 C(CCC(C(=O)N1CCC1C(=O)OC)NC(c1ccncc1Cl)=O)OC Cc1ccc2sc(C(=O)NC3CC4CC3N(C(C3(C)COC(=O)C3)=O)C4)cc2c1 c1(CCC)noc(CCCC(=O)NCCC2CCN(C(=O)CC3CC(F)C3)C2)n1 C1(C(=O)NCCCC2CC2)CCCCCCN1C(C1CC(O)C1)=O c1(CC(=O)NCC2C(C(=O)NCC(CCC)C)CC2)ccc(F)nc1 C(=O)(C1=CCCOC1)N1C(C)CC1C(=O)NCCCP(C)(C)=O C(C(=O)N1CC(C(C)NC(=O)CC(O)C2CCCC2)C1)(C(C)C)NC(COC)=O C(CCC(C)NCC(C)(C)C1CCOC1)N(CC#C)CC=C c1(C(=O)NCC2N(C(C(=O)NC3CC3)=O)CCOC2)ccc(CO)cc1F C(=O)(C1=CCC(C)CC1)NC1CCCCN(C(C(=O)NCCOC)=O)C1 c1(CC)c(C(=O)NCCC2CN(C(=O)CO)CCO2)cccc1C Cc1ccccc1-n1cc(-c2csc(C(=O)NCC3(C#N)CC3)n2)cn1 CCC(CCC(=O)NCC(O)CCO)NC(=O)Cc1ccc(O)cn1 N1(C(CC2CC(=C)C2)=O)CCC(C(F)(F)F)C(NC(=O)C=Cc2cscn2)C1 CC#CCCC(=O)N1CC(CC(C)(C)CNC(=O)C(C)OC(C)(C)C)C1 c1(CCC)ncoc1C(=O)N(CCC(=O)NC1CCSC1C)C(C)C N(C(=NCC1C(C(=O)OC)C1(F)F)NC(C)Cc1cccc(F)c1)C(CC)CC C(=O)(CC(CC)CCCC)N1CC2C(CNC(CCCCCCC)=O)(CCC2)C1 C1(C(N2CCC(C)(NC(=O)C#CC3CC3)CC2)=O)C2CCC(CC2)C1C(F)(F)F Cc1cc(C(=O)NNC(=O)C2CSC2)c(C)n1-c1ccccc1 c1(C(=O)NC2CCC(NC(c3cncc(O)c3)=O)C2)c(F)c(F)cc(F)c1F N1(C(CCOC)=O)CCCC1(C)C(=O)NC1CC(OC)CN1C(=O)OC(C)(C)C Cc1cc2c(C(N3CC4CC3CCC4NC(c3ccoc3C)=O)=O)cccc2o1 c1(NC(C2COCCN2Cc2ccc(CO)o2)=O)ncc(I)cc1C(F)(F)F Cc1cccn2ncc(C(N3CCN(C(=O)C(C)(C)C(C)C)CC3C3CC3)=O)c12 Cc1cnc2nc-2c(CCC(=O)N(c2nccc(Cl)c2Cl)C)c(C)[nH]1 C1(CNC(C(c2cnn(C)c2)OC)=O)CC2CCC(C1)N2C(C1C2CCCC12)=O CC1(C(=O)NCCCN(C(c2cscc2C2CC2)=O)C2CC2)CCCC1O CC1(C)CCCN(C(=O)CC2COCC2O)C1C(=O)NCC1=NOC2COCC12 C1(NC(C(CC#C)C2CC2)=O)CCC2(CCN(C(=O)CC(=O)OCC)C2)C1 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)C(F)(F)F)cc(F)c1Br C1(C(N2CC(C)(OCC(=O)NC(C3CCCCC3)C#C)C2)=O)CC(=O)NC(=O)N1 C1(C(N2CC(C)OC(C)C2)=O)N(c2nnc(COC)s2)CC12CCC(F)(F)CC2 N(C1CCc2cccnc21)C(c1[nH]c2c(Br)cccc2c1-c1ccccc1)=O c1(C(N2CCC(C(=O)Nc3c(C)cnc(F)c3)C2)=O)ccc(Br)c(O)c1Br C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(C2CC3(CC3)CO2)=O)CC(C)(C)C1 C1(OCC)CC2(C1)CC2C(N1CCCCC1CN(C(=O)CC(C)(F)F)C)=O C1(NC(C2C(=C)C2)=O)CN(C(C2CC(C)(C)CN2C)=O)CCC1C(F)(F)F N1(C(c2n(C(C)C)ccc2)=O)CCC2CN(C(=O)C=Cc3ccco3)C2C1 C1(N(C(CCSCCC)=O)C)CCC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC12 N1(C(C(C)SC)=O)CC(NC(=O)CCc2cnn(C)n2)Cc2ccccc21 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(c2cccnn2)=O)CCC1CO c1(-c2cc(NC3CNCC3F)ccc2)cccc2c1OCO2 C(=O)(NNc1ccc(Cl)c(C)n1)c1cnc(OC)[nH]c1=N c1(C(=O)NCCN(CC(C)O)C(=O)CN(C)C(=O)C2CC2)ccc(S(C)(=O)=O)o1 c1(C(=O)NCCC2(O)CN(C(c3c(CC)n(C)nn3)=O)C2)c(CC)nn(C)c1Cl C(=O)(CC1=NNC(=O)C1)NC(CN(C(C(c1c(C)n[nH]c1C)C)=O)C)C n1(CC(C)C(=O)NCCN(C(=O)C(C)(C)CN(C)C)C)ncc2ccccc12 N1(C(CC(COC)NC(=O)C(C)C#N)=O)CCC(C)(c2ccccc2)CC1 Cc1ccc(F)cc1C(N1CC(O)CC1C(=O)NC(c1nn(C)cc1O)C)=O CCCC(CNC(=O)Cc1cn(C(C)C)nn1)NC(=O)C=C(CC)CC c1(C(N(C)CCN(S(C)(=O)=O)C2CCC2)=O)ccc(C(C)C(F)(F)F)cc1 c1(C(=O)NCC(CNC(CC(CC)C)=O)C(F)(F)F)ncc2cc(Cl)ccn12 O=[N+]([O-])c1cc(Cl)c(Cl)cc1S(=O)(=O)NC1(c2ccc(OC3CC3)cc2)CC1 N1(C(CCC=C)=O)CCOCC1CN(C(=O)C(C)(C)COC)C C1(C(=O)NCCCOCC)CCCCN1C(=O)CC1CCC(C)CO1 C(=O)(C1CCc2ccccc21)NC1C(C(N(C(C)(C)C)CCN)=O)C1 c1(C(C)=O)cccnc1NC1CCN(C(c2cnn(CC3CC3)c2)=O)C1 N1(C(C(CN(CC)CC)F)=O)CCCC(C)(CNC(c2cnncc2C)=O)C1 C1(NC(C(C(CC)O)C)=O)CCCC12CN(C(c1c(C)ccnc1C)=O)C2 N(C(=NCCNS(C)(=O)=O)NCC1CC2CCC1O2)CC(C=C)(C)C C1(N(C)C(C2CC(F)(F)C2)=O)CCCN(C(c2cc[nH]n2)=O)C1 N1(C(C2(CF)CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)CC2CCCCC2C1C C1(NC(C(=O)NCCOCCCC)=O)CCN(C(c2ccccn2)=O)C(CC)C1 N#Cc1ccc(CN2CC(Nc3ncc(C4CC4)cn3)CC(CO)C2)c(Br)c1 c1(NC(C2C(c3n(C)cnc3)C2)=O)ccc(C(F)(F)F)cn1 c1(C(=O)NC2CN(C(c3ccc(C(=O)OCC)nn3)=O)C2)cc(OC)ccc1I c1(C(N2CCC(F)(CNC(C3CC(C)(CC)C3)=O)CC2)=O)c(F)ccc(F)c1F n1(C2(C(=O)NC3CC(NC(CCN(C)CC)=O)C3)CC2)cc(Cl)cn1 C1(NC(c2c(CC)nco2)=O)CC2CCC1CC2NC(=O)CCc1ncnn1C C1(CC=C)(NC(=O)C(c2ccccc2C)C)CCN(C(c2cscn2)=O)C1 O=C(C#CC1CCOCC1)NCC12CCC1CCN2C(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC23CC(COC)(N(C(=O)CC4C=CCC4)C2)C3)cccn2nccc12 c1(COC)ccc(C(=O)NC2CCC(NC(C3CCNC(=O)C3)=O)C2)cc1F c1(NC(=O)CC2(N)COC2)ccc(CNC(CC)=O)cn1.c1ccccc1 c1(C(=O)NCC2OCC(CNC(C(CC)(C)C)=O)C2)c(N)sc2c1CCSC2 C1(NC(C(CC)n2ccnc2)=O)CCC(C)N(C(c2ccc(Br)cc2)=O)C1 C1(C(N2C(C(C)NC(C3(C(C)C)CC3)=O)CCC2)=O)CCCCN1C N1(C(CC(CC2CC2)NC(Cc2cc(C)on2)=O)=O)C2CCCC1CN(C)C2 C1(c2ccon2)(CC(=O)N(C)CC2(CNC(C3CCS3(=O)=O)=O)CC2)CS(=O)(=O)C1 N1(C(C=CCOCCOC)=O)CCC2CCN(C(=O)CCCn3ccnc3)C2C1 C1(C(=O)NCC(C)NC(=O)OC)CC(C)N1C(C1CN(C(C)=O)C1)=O N1(C(C2(C)CCOC2)=O)CC2(NC(=O)COC3CC=CC3)CCC1CC2 C(=O)(CC1(O)CCOc2ccccc21)NCC(C)NC(CCCC#C)=O C1(C(N(C)CCNC(=O)CCn2ccnn2)=O)CCCCN1S(N)(=O)=O C=CCC(CC=C)C(=O)NC1CCN(CCCNC(=O)C(O)P(C)(C)=O)C1 C1(NC(c2csc(Cl)n2)=O)CC2(CCCN(C(=O)CC3CCCO3)C2)C1 C1(NC(C(CC)=CC)=O)CC(C)N(C(=O)C(CC)OC)C1 Nc1ccc(C(N2CCCC(c3cc[nH]n3)C2)=O)c(F)c1 C(=O)(C(O)CCCC)NCC1CN(C(CC=C)=O)CC1c1ccc(OC)cc1 c1(CNCc2ccc(CC)cn2)cn2c(C)cc(C)nc2n1 C=CCC(C)C(=O)NCc1ccc(CNC(c2cc(C(F)(F)F)ncn2)=O)cc1 C1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)CC(c2ccc(F)cc2)=NO1 C(C)(CCN=c1ncc(I)c[nH]1)NC(c1c(O)nc(CC)c(C)c1)=O S(=O)(=O)(c1c[nH]ccc1=NCC(F)c1ccc(Br)cc1)NC1C(C)(C)C(O)C1 C=C(C)C1CN(C(c2cn(CCNC(=O)C(C)C(O)CC)nn2)=O)CCO1 C1(CNC(CCCC#C)=O)CN2CCCCC2CN1C(c1cncc(SC)c1)=O c1(C(=O)NC(C(C)C)(C)CNC(C2(C)CCCNC2=O)=O)cnc2occc2c1 N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CC1OCCCC1(C)C c1(C(C2CCC2)NC(C2COCCN2Cc2ccccc2)=O)ccc(Cl)cc1O CCCCC(C)C(=O)N1CCCC(CCC(N2CCOCC2C(N)=O)=O)C1 C(=O)(C1SCCc2ccccc21)N1CC2(N(C(c3n(C)ccn3)=O)CC2)C1 C(=O)(C1=CC2(CN(C(C3C4CCCCCC34)=O)C2)OC1)NC1CCC(C)(C)CC1 c1(C(=O)NC(C)CCNC(c2ccc(N)cc2)=O)cc2c(=O)[nH]ccn2n1 C(=O)(C(F)(C(=O)OCC)C(C)NC(N1CC(C)C2CCCCC12)=O)OCC C1(N2CC(C(=O)NCC(CN(C)C(C3(C#N)CC3)=O)O)C2)CCOCC1 c1(NC(c2nc(C(=O)OC)oc2)=O)ccc([N+](=O)[O-])cc1Cl C=CCCC(C)(C)C(=O)NC(c1nocc1C(=O)NC1CC(C)(C)C1)C C1(C(=O)NCC(CC)(C)Cl)CC(O)CN1C(c1nccnc1C)=O O=S(=O)(c1nc[nH]n1)NCCCCCc1cccs1 N1(C(c2n(CC=C)ccc2)=O)CCC2(NC(=O)CCOC3CC(F)(F)C3)CC2C1 c1(-c2c(OC)ccnc2)n[nH]c2c1CN(C(=O)C(O)CC(C)C)CC2 N1(C(C(c2ccccc2)NC(C)=O)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1 C(=O)(CCCC(C)C)N1CC(CC(C)NC(C(CCSC)OC)=O)C1 C(CCC(N)=O)(C(=O)N1CC2CN(C(c3ccc(OCF)s3)=O)C2C1)NC(C)=O Cc1cccc(O)c1C(=O)NCCc1ccc(CNC(C2CC2CF)=O)cc1 c1(C(=O)NCCN(C)C(C2CCSC2)=O)ccc(N2CCOCC2)cc1F C1(C(=O)NC2CC(O)(CNC(c3ccc(Br)o3)=O)C2)CCc2nnc(O)cc2C1 C12(C(=O)NCC(C(=O)OCC)C)CC1CCN2C(=O)Cn1cncn1 c1(C(N(CC(CN(C(C(C)NC(=O)C2CC2)=O)C)O)C)=O)cc(O)cs1 c1(C(=O)NC(C2CCN(C(=O)CCOc3ccc(F)cc3)C2)C)c(Cl)cnn1C C(C(=O)NC1(C)CCC(C(N2CCC(CO)(CO)C2)=O)C1)(C(C)C)SC C1(C(=O)NCC(C)CNC(=O)C(O)Cc2cccc(Cl)c2)CC2(CCC2)C1 c1(C(=O)NC2C(NC(Cc3cnc(C)[nH]3)=O)COC2)csc2c1CCCCCC2 c1(C(N2C(C)CC(NC(=O)C(=O)N=S(C)(C)=O)CC2)=O)nccc2c1NCCC2 C1(C(=O)O)(CNC(C2CC2C2CCCO2)=O)CCS(=O)(=O)CC1 c1(CNC(C(CC)NC(=O)C(O)C2CCCC2)=O)cncc(C)c1 c1(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)CC2)n[nH]c2c1NCCC2 c1(C(=O)NCc2c(C)cco2)cc(C2CC2)ccn1 N1(C(CC(CNC(C(C=C)(C)C)=O)C2CCC2)=O)CC2(CNC(=O)OC2)C1 c1(C(=O)NCC(C)N(C(C(CCC)OCC)=O)C)c(OCC2CC2)cccc1Cl C1(C(C)C)C(=O)N2CCCC2CC1.c1(ONC(CC=CCC)=O)ccc(F)cc1.OC C1(CNC(Cc2cc(C)[nH]n2)=O)C(C2CC2)CCN1C(c1cnccc1C#N)=O CC1CN(CC(O)COCC(F)(F)F)CCN1C(c1coc(C2CCOCC2)n1)=O CS(=O)(=O)c1cccc(C(=O)NCC2C=CC(NC(c3ccsc3Cl)=O)C2)c1 c1(C(=O)NC(C2N(C(C=C(C)C(F)F)=O)CCCC2)C)cc(F)c(F)cc1O Cc1cccc2c(C(=O)NCC(F)CNC(c3ccnc(S)c3)=O)n[nH]c12 N1(C(C=CC(C)C)=O)CCN(C)CC1CNC(c1[nH]c(=N)ccc1C)=O N1(C(C(CC)(C)O)=O)CCC(C)(Oc2nn[nH]n2)CC1 Cc1cc(CC(=O)NCC2(C)CCN(C(C3CN(C(N)=O)C3)=O)C2)ccc1F Cc1cc(C)nc(N2CCCC(NC(=O)CCn3cccnc3=O)C2)n1 c1(C(N(CCN(C(C(C(=O)OC)(C)F)=O)C)C)=O)ccc(O)c(C)c1C Cc1csc(CNC(C2CC2c2ccc(-c3cncn3C)cc2)=O)c1C c1(OC)ccc(CC(C)CNC(=O)C(=O)N(C(C)C)Cc2ccoc2C)cc1F N1(C(C(CCC)CC2CCCC2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)C1 CC(C)C(C(=O)NCC1C2CC1N(C(=O)CC(C)c1cccs1)C2)n1cnnn1 C1(C(=O)O)CN(CC)CCO1.C(=O)(C(C)C)NC(=O)NCC Nc1cc(Cl)cc(Cl)c1C(=O)NC1CC(O)CN(C(=O)C=Cc2nccs2)C1 C1(C(C)(C)NC(C=C(COC)C)=O)CCN(C(c2ccncn2)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC(C)N(C(=O)CCC1CC1(Cl)Cl)C n1(CCC)nnnc1C(c1ccoc1C)NC(C)C(=O)OCC(C)C C1(NC(C2CCC2(F)F)=O)CC2C(NC(C3(C4CC4)CC3)=O)C2C1 Cc1cnc2c(S(=O)(=O)NC3COc4ccccc4C3=O)cccc2c1 N1(C(c2ncc(C#N)cc2Cl)=O)CCC2(CC(C(=O)N=c3onc(Br)[nH]3)=NO2)C1 N12CCN(CC1)CC2=O.Cn1ccnc1SCC(=O)NC1C2CCCC12 c1(C(N2CC3C(CNCc4n(C)cnc4)(C3)C2)=O)c(Br)ccc2c1OCO2 c1(CC)oc(C)cc1C(=O)NC(CN(C(C1(C(F)(F)CC)CC1)=O)CC)CC c1(CCN(C)C)ccc(C(=O)NNC(=O)c2ccc(N(C)C)cc2)cc1[N+](=O)[O-] Cc1nc(C(N2CCC(O)(C(C)NC(=O)CCCc3nncn3C)C2)=O)c(C)s1 C1(CC)CCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1)=O CC1CC(C)N(C(=O)CNC(N)=O)CCN1C(c1ccc2nc(O)[nH]c2n1)=O CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)COc2ccccc2C)C(C)(C)C1 C#CCCCCC(=O)N1CCC(C(C)NC(=O)CC2CC3(CCC3)CO2)C1 CC1(O)CCN(C(C23CC(C)(CN2C(=O)CCc2cncs2)C3)=O)CC1 N1(C(=O)C=C2CCCCC2)CCOC2(C1)CN(C(=O)CNC(C1CCOC1)=O)C2 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC(C(C)NC(c1c(CC)cno1)=O)(C)C Cc1cc(=NCC2C3CCCC23)[nH]c(N(C)Cc2ccc(OCC(N)=O)cc2)n1 c1(C(N2CCC(C3CCC3)C2)C(=O)NCCOCC2CC2)cnc2ncccn12 C1(C(=O)NC2CCC(NC(c3ccc(F)o3)=O)C2)CCc2nnc(O)n2C1 C12(C(N3CCN(C(C4C(C)OCCC4)=O)CC3C)=O)CC3CC1C2C3(F)F c1(C(=O)NCC(CC)NC(C2CC(F)(CO)C2)=O)cncc(F)n1 S(=O)(=O)(c1cccc(C(=O)N(C)Cc2ccc(S(N)(=O)=O)cc2)c1)N(CC)CC N1(C(c2c(C)cc[nH]2)=O)CC2OCC(NC(c3cccn4nccc34)=O)C2C1 C1(C)(CC)C=C(C(=O)NCC2CC(OC)CN2C(c2cc(SC)ccc2Cl)=O)C1 CC1=C(C)CC(C)(C(N2CC(CNC(=O)CP(C)(C)=O)C(C)(C)C2)=O)CC1 N1(C(C(Cc2cn[nH]c2)NC(CC2CC(OC)C2)=O)=O)CC2(CCN2C)C1 C=C(Cl)CC(C(=O)NCc1nc(C)cc(O)n1)NC(c1cc(C)nnc1C)=O CC(C)C(C(=O)N(CCC(C)NC(C1CC(C2CCC2)C1)=O)C)C(C)C c1(-c2cn(CCCC(=O)NC(COC)CF)nn2)cc(Cl)ccc1C(=O)O c1(C(N2C(CN(C(C=C(CC)C)=O)C3CC3)CCC2)=O)ccc(C)c(C)n1 C1(CNC(C(=Cc2ccco2)C)=O)COCCN(C(=O)C(F)CC2CCCC2)C1 Cc1ccc(CNC(=O)C(C)NC(c2cnccn2)=O)c(F)c1 C=C1Cn2c(C(=O)NC34COC(C3)C(NC(C3(C#N)CC=CC3)=O)C4)nnc2S1 c1(C(N2C(CCC)CN(C(=O)Cc3ccc(C)o3)CC2)=O)ccc2nnnn2c1 c1(C(=O)NCCC2(OC)CN(C(C3CCN(C)C3)=O)C2)sc(C)nc1C(F)(F)F N1(C(CCC=C)=O)CCCC2(NC(c3cnc(OCC)cn3)=O)CCCC12 Cc1cccc2cc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)[nH]c12 N1(C(CCc2n(C)cnn2)=O)C2CCC1CN(C(c1cc(C(N)=O)n(C)n1)=O)C2 C1(C(=O)NC2(CCCC)CC2)CCCCC1CNC(C1(C)CNC(=O)C1)=O C1(C(N2CCC(F)(CF)C2)=O)CCCN(C(C2CCCCS2)=O)C1 C#CC1CC2(CC2)CN1C(c1coc(CNC(=O)C(C)(C)CC(F)F)c1)=O CC1CC(C(=O)NCCC2CCCN2C(c2cnc(-c3cnccn3)s2)=O)=NO1 N1(C(c2ccn(CCCC)n2)=O)C2CC1CN(C(c1sc(C)nc1CC)=O)C2 N1(C(CCCC(=C)C)=O)CCCCCCC1C(=O)NC1CC(=O)N(C(C)C)C1 c1(C(N2C(C(NOCC)=O)CCC2)=O)ccnc2cc[nH]c12 C1(CC(=O)NCCCCC#CC)C2CCC(C2)N1C(c1cc(C)nn1C)=O C1(OC)C(N=c2[nH]c(=NC3CC(N(CC(F)(F)F)C)C3)[nH]c3c2COC3)CC1(C)C C1(C(=O)NCC2(O)CCN(C(c3cc(CF)on3)=O)C2)Cc2cc(Cl)ccc2O1 C1(N(C(C(=O)NCCNC(C)=O)=O)C)CN(C(C2CCNC2=O)=O)CC1(C)C C1(CCCC)CN(C(=O)C(C)CSC)CCN1C(c1nn(C)cc1C)=O CC1=C(C(=O)N2CCC(C3CC(NC(=O)CSC(F)F)C3)C2)C(C)(C)CCC1 C#Cc1cc(F)c(C(=O)NC2CC3(C2)CC3NC(c2cccc(C)n2)=O)c(F)c1 N1(C(C(CSC)O)=O)CCCC2CN(C(=O)CNC(=O)Cn3cncn3)CC12 c1(C(N2CCC(C(C)NC(c3cccc(CC)n3)=O)CC2)=O)ccc(N)c(F)c1 c1(C(=O)NC2(COC)CN(C(C(C)OC)=O)C2)ccc(C)cc1OC1CC1 C1(c2nocn2)C2CCCC2CN1N(CCO)CCCC.C1(C)(CC)CCC(C)O1 C1(NC(CCC=C(C)C)=O)CN(C(c2ccc(C)nc2O)=O)CCC1CO Cc1ccc(C(=O)NCC2(F)CCN(C(=O)C(C3CCCCC3)C)C2)nn1 c12cc(ccc1F)C(=O)N(C1CCCC1)CCS2.C12(C(=O)NC(C)C)CC(O)C1C2 Cc1cc(Br)cnc1C(=O)NCC(CC(F)(F)F)NC(C1CC1F)=O C1(NC(=O)C=CCF)CC1C1CCCN(C(=O)C=CCN(C)CCO)C1 C1(NC(c2cc(CC)nn2C)=O)CC2CN(C(=O)CC(=O)OC)CC12 C(=O)(N=c1ccn(C2CCC2)[nH]1)C1CC1.N1(C(C(C)C)=O)CCCC1C=O CN1CCN(C2CC(NC3(CNC(=O)OC(C)(C)C)CCC4CC34)C2)CC1 O=C1N(CC(c2nc(Cl)cs2)=O)CC2CCCCN12 C(C(CC(F)(F)F)NC(c1ccnn1C1CC1)=O)NC(c1c(C(C)C)[nH]cc1)=O C1(CC(C)C)(C(=O)NCC2CC(NC(c3nc(CCC)oc3)=O)C2)CCNC1=O c1(NCC(CCCCC)O)ncc(C)cc1S(=O)(=O)NC(c1cccc(Br)c1)C Cc1cc(C(=O)NC(CCNC(c2csc(Cl)c2)=O)C(C)C)nn1C1CC1 c1(C(N2C(CO)CC(NC(CNS(CC)(=O)=O)=O)C2)=O)cc2ccsc2n1C N1(C(c2c(OC)ccs2)=O)C2CCC(C2)C1C(=O)NCc1cccnc1SC CCC(CCCC(=O)NCCOCC(=O)OC)NC(=O)C=C1CCCCC1 c1(C(N2CCCC(NC(CCCC(N)=O)=O)(CO)C2)=O)cn2c(n1)CCCC2 C(C(C)CC(=O)NCC1(C(=O)NOCC=C(C)C)CC2(CC2)C1)OC c1(CC)ccccc1OCCOCC(=O)NCCN(C(=O)C(C)CO)C(C)C N1(CC)N=C(C(=O)N2CCC(=CCNC(=O)CCCCC(C)C)CC2)CCC1=O c1(C(N(C)CC2(O)CN(C(c3nc(COC)sc3)=O)C2)=O)cccc(Cl)c1C c1(C(N2CCCC(CC(N)=O)(NC(CCC)=O)C2)=O)cc2c(cn1)OCCO2 C12(C(N3CCC(OC(C)=O)C3)=O)CC(C)(C1)OC2C c1(C(=O)NC2CCN(C(C(CC(C)C)O)=O)C2)noc2cc(Br)ccc12 Cc1cccc(C2(C(=O)NCC(CO)NC(c3cccnn3)=O)CCC2)c1 c1(-c2cccc(NC(C3C4CCC(F)(F)C34)=O)c2)nnc2n1CCC2 CONC(=O)CNC(C1C=CCN1C(=O)COCC(F)F)=O c1(OC)ccc(N(C(=O)NNC(=O)c2cc(Br)c[nH]2)C)cc1 N1(C(C=CCC)=O)CCCC12CCN(C(c1cc(C)sc1C)=O)C2 c1(C(=O)OCC)ccc2c(c1)CC(NC(=O)C(=O)NCCCCCCCO)C2 CC1CN(C(C2CC3C=CC2C3)=O)CCC1CNC(=O)CC1COC(=O)N1 c1(CN2C(C(=O)Nc3ccc(C)nc3I)CCCC2)cc(F)cc(C#N)c1 Cn1c(=O)sc2cc(CNS(=O)(=O)c3ccc(Br)cc3Cl)ccc12 C1(CN(C(C(C)C)=O)C)CCCC(NC(=O)C=C2CCC(C(C)(C)C)CC2)C1 CC(CCc1ccccc1F)C(=O)N(CCCNC(=O)COCC1CCCC1)C c1(C(=O)NC2(CC)CCCN(C(=O)CCC(C)(F)F)C2)ccc2nc[nH]c2n1 CC1CCCC1(C)NC(N1CCN(C(=O)Nc2cnsn2)CC1)=O c1(C(=O)NC(C(=O)NC2CCN(C(C)=O)C2)Cn2cncn2)cc(C)c(F)cn1 N1(C(C(N2CCOCC2)C)=O)CC(CNC(c2nn(C)cc2N)=O)CC12CCC2 N1(C(C(CSC)O)=O)CC(NC(c2ccc[nH]2)=O)C(CC(C)(C)C)C1 C=CC1CCCCN1C(=O)CC1CCCN1C(C1CS(=O)C1)=O N1(C(C(CC)CC(C)C)=O)CCC(NC(=O)CC(F)(F)C(C)C)C2(CCC2)C1 C(=O)(C1=NOC(C)C1)N1CCN(C2CN(C(C(OC)OC)=O)C2)CC1 C1(NC(c2c(O)nc(CC)c(C)c2)=O)CCC2(CC1)CN(C(=O)C(C)(C)F)C2 c1(C(C(=O)NCCC#N)N(CCCC)CC)cc(S(N)(=O)=O)cs1 C(=O)(C(O)C(C)C)NC1C(OCC)C(O)C1.[nH]1nc(-c2ccccc2OC)cc1C c1(C(N2C(CNC(C(C=C)(C)C)=O)C(C)(C)CC2)=O)ccc2c(c1)CCN(C)C2 c1(SC(C)C(=O)NCCCOCCC(=O)N(C(C)CO)C)ccccn1 C=CCC(C)(C)CC(=O)NC1CCCC1CNC(=O)COC(C)(C)C N1(C(c2csnn2)C)CCC(O)CC1.C123CC(C1C2)n1cc(nn1)CNC3=O N1(C(CCC=C=C)=O)CC(CNC(=O)CC2CCC(=O)NC2)C2(CCOCC2)C1 N1(C(CNC(=O)OC)=O)CC2CCOC2(CNC(=O)C(CO)NC(N)=O)C1 N1(C(C2OCC(C)(C)C2)=O)CC(C(=O)NOCc2cncc(C#N)c2)C2(CCC2)C1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(C)C(NC(=O)Cc2nnc(C)o2)C1 CC1CC(NC(C2(C)CC(C)(C)C2)=O)CCN1CCCN1C(=O)CNC1=O S(=O)(=O)(c1cc(C(=O)NC(C2CCCN(C(=O)Cc3ccsn3)C2)C)co1)NC N1(C(CCc2cnc(C)o2)=O)CC(O)CC1CNC(=O)CCN1CCCCC1 N1(C(C(CNC(C2(O)CCOC2)=O)N(C)C)=O)CCn2ncnc2C1 C(=O)(N=c1cc(Br)n(C)[nH]1)C1CN(C(CS(CC2(C)CC2)(=O)=O)=O)C1 Cc1ccc(O)nc1CNC(=O)CN(CC(C)C)C(C1CC(=O)C1(C)C)=O C(=O)(CC1=NNC(=O)C1)NC1CC2C(NC(CC3(COC)CCOCC3)=O)C2C1 S(=O)(=O)(c1ccccc1)N1CCC(C(N(CCC)CCNC(=O)C2=CCC2)=O)C1 N1(C(C(CCCOC)C)=O)CCCN(C(=O)C(F)(F)CN2CCCC2)CC1C N1(C(C(CC=C)(C)C)=O)CCC(C2(NC(C3(C(C)(F)F)CCC3)=O)CC2)CC1 C(=O)(CCCCCC(C)C)N1CCCC(NC(c2n(CC)nc(C)c2)=O)CC1 Cc1nc2cccc(C(N3CCCC(NC(c4nscc4Br)=O)C3)=O)n2n1 CN1N=C(C(=O)N2CCC(OCC(=O)N3CC(C)(O)CO3)C(O)C2)CCC1=O c1(OC(CC)C)cccc(CN2CCC2)c1.C1(C(=O)N)C=CCN1.C(C)SC c1(C(=O)NC2CN(C(C3C(C)(CC)C3)=O)C2)ccc(CCc2ccccc2)[nH]1 n1(CCCC)nc(C)c(C(N2CC(O)(CNC(=O)CC3CCOC3=O)C2)=O)c1Cl C(=O)(CCCc1ccsc1)NCC(C1CCOC1)NC(C1(SC)CCC1)=O CCCCCCC(C)C(=O)N1CC2(C1)CN(C(c1cc(C)n(C)c1)=O)CCO2 C1(CCNC(=O)Cc2cnccn2)COCCN1C(=O)Cc1cncs1 C1(CNC(C(C)n2ccnc2)=O)CCCN(C(c2ccncc2C(F)F)=O)CC1 n1(CC)nc(C2CC2)cc1C(=O)NCCC1CC(OCCOCCO)C1 C1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)CC2O)CCCC2(CC2)C1 c1(CC(=O)N(C)CC2CCN(C(C3CC(O)C3)=O)C2)csc2nccn12 C1(C(F)(F)F)(C(=O)NC2CN(C(c3cc(C(F)(F)F)c[nH]3)=O)C2)CC=CCO1 CON(CCO)C(=O)COC1CN(C(=O)C=C(C2CC2)C2CC2)C1 C(CCCC(CO)NC(C12CCC1C2)=O)NC(C1CCN(C)CC1)=O c1(C(N2CC(O)(CNC(C3CCn4cncc4C3)=O)C2)=O)ccc(F)c(F)c1F N1(C(c2c(C)scc2)=O)CCN(C(=O)C(C(C)C)n2cncn2)C2CCC12 c1(C(C)=O)ccc(SC(C)C(=O)NCc2ccc(Cl)cn2)cc1 C#Cc1cn(C)nc1C(=O)NCC1CCN1C(c1cn(CC2CCOC2)nn1)=O C(=O)(C1(C)CCCc2ccccc21)NCCN(C(=O)C#CC(C)(C)O)CCC C1(NC(C2CC3CCC3C2)=O)CCN(C(=O)C(F)(F)C2(O)CCCC2)CC1 c1(CN(CC(CCC=C)O)C)cccn(Cc2ccccc2)c1=O CC(CC(=O)N(CC(O)C1CC1)C)C(C)(C)NC(c1cn2c(n1)CCC2)=O Cc1ccn(CC(=O)NCC2(O)CN(C(c3ccnn3CC(F)F)=O)C2)c(=O)c1 CCC(CC)C(C)C(=O)NCCCCNC(c1cnc2sccn12)=O c1(C(=O)NCc2c(CCNC(C(CC)OC)=O)ocn2)nnc(O)cc1O C1(NC(C(c2cncnc2)C)=O)CCCC(C(=O)NC2(CCF)CC2)C1 c1(CCC(=O)NCCC(=O)NC2CCCC2)nnc(C2CC2)n1-c1cccs1 N1(C(C=C(C)C2CC2)=O)CCC(C2CCCN(C(C3CCOC3)=O)CC2)CC1 c1(C(=O)NCC=C)ccc(-c2ccnc(N3CCN(C)CC3)c2)c(C(F)(F)F)c1 CC1(C)CCC(NCCCc2ccc(C(C)(C)C)cc2)c2ccccc21 N1(C(c2c(Cl)nc(N(C)C)s2)=O)CCC(CNC(=O)C(N)=O)C12CCC2 N1(C(c2c(NS(C)(=O)=O)ccs2)=O)CCC(O)C(C(N2CC(O)C2)=O)C1 c1(C(N2C(Cn3cc(-c4n[nH]c(C)c4C)nn3)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CCCC)ccc(C(c2nnnn2C(C)C)NCCc2cccnc2C)cc1 c1(NC(=O)Nc2nc(CCCC)sc2)ncc(Cl)nc1Br C1(COC)(NC(=O)CCSCC(=O)OC)CCCN(C(=O)C(C)(F)F)C1 CCCCCC(O)CC(=O)N(C)CCNC(c1cc(F)cc(Cl)c1)=O c1(C(N2CC(NC(c3cncs3)=O)CC3(C2)CC3)=O)cc(F)c(F)c(O)c1F C1(CNC(=O)C=Cc2ccco2)CC2CCC(C1)N2C(=O)CCC(F)F c1(COC)ccc(NC(=O)CC2CCCN(C(=O)C(=O)C(C)C)C2)cc1 C1(C)(NC(c2n(COC)ncc2)=O)CCCCC1C(=O)Nc1ccc(O)nc1 C1(C2CC2)(NC(C(F)=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(=O)Nc2ccnc(C(N3CCC(O)CC3)=O)c2)ncn2c1CCCC2 Cc1nocc1NC(=O)CC1CCN(C(C2(C)OCCO2)=O)C1 c1(CCC(=O)NCCC2(O)CCN(C(C3CCSC3)=O)C2)nc2cccnc2[nH]1 c1(C(CNC(C2CN(C3CN(C(CC)=O)C3)C(=O)C2)=O)=O)csc2cncn12 Cn1nc2c(c1C(=O)NCc1cncnc1)CN(C(=O)CCCCCCBr)CC2 C(=O)(C1=CCCOC1)N(C1CCCN(C(C=CC(CC)C)=O)C1)C C1(CCC)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)CCC1CCC(=O)N1 CC1CN(C(=O)C(Cc2cnn(C)c2O)NC(=O)CC(=O)NC2CC2)CCN1C N1(C(C2CN(C(C)C)C2)=O)CCC2(COC(CNC(C3CC3F)=O)C2)C1 C1(NC(C(c2ccccc2)NC(=O)OC)=O)CCOCC1NC(C1(Cl)CC1)=O c12cn(c(=O)nc1O)CC(=O)NCCCNC2=O.C1(CC)CCCCO1.C(C)C c1(C(=O)NC(CNC(C(CC)(C)C)=O)(C)CC)coc2c1CS(=O)(=O)C2 Cc1sc(C(N2CCCC2CCNC(=O)C(C)CC2CCCC2)=O)nc1O c1(CC(N2CCN(C(C(C(C)C)F)=O)C(C3CCC3)C2)=O)cccc2nonc12 N1(CCC(N2CCCC(N(C)Cc3cc(C)on3)C2)=O)C(=O)NC(C)(C)C1=O c1(C(=O)NC(C(=O)NC(c2n(CC)ncc2)C)CC2CC2)cccc2[nH]ccc12 C1(C(N2C(CN(c3c(C)cncn3)C)CCCC2)=O)CC(=O)NC1(C)C C1(C(=O)NCC2(CC(C)C)CC2)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 CCC(C)C(C(=O)NC1CC(CC(C)(C)C)C1)N(C(=O)Cn1ncccc1=O)C c1(C(=O)NC(C2CN(C(=O)C(F)C3CCC3)C2)C)ccc(OC(F)(F)F)nc1 N1(C(c2cc(C)on2)=O)CCCC12CCCN(C(c1cc(Cl)cn1C)=O)C2 C(c1c(Cl)cccc1Cl)=CC(=O)NC(C)C(C)NC(c1ccc2nc[nH]c2n1)=O CCC(C(=O)N(CCCNC(=O)Cc1cnn(C2CC2)c1)C1CC1)OC C1(CCC(=O)NCC(=O)OC(C)C)CCCN(C(c2cscn2)=O)C1 C1(CC=C)(C(=O)NCCCc2cnn(C)c2)CCN(C(c2cc(Cl)no2)=O)C1 C(CCCC(=O)N1CCC(NC(c2cc(C)c(C)s2)=O)CC1)OCCC=C CC1=C(C)CC(C(=O)NC(C2CCCN2C(c2nn(C)c(C)c2Cl)=O)(C)C)CC1 C1(NCc2cc(SC)c(Br)cn2)CCCC12CCOCC2 n1(Cc2c(C)cccc2)nc(C)c(NC(=O)C(C)C(C)O)c1C c1(NC(c2nc(C(N3CC(O)C3)=O)cs2)=O)cc(O)ccc1Cl c1(CC=C)ccccc1C(=O)NC1CCC1CNC(c1ccccc1OC)=O CCC(CC(=O)N(C)CC1(O)CCN(C(=O)CC2(C#N)CCCCC2)C1)C(C)C C1(S(C)(=O)=O)(C(N2C3CC(CNC(CC(C)F)=O)C2CC3)=O)CCOCC1 C1(C(N(CCNC(c2cc(CCOC)on2)=O)CCOCCO)=O)C2COCC12 N1(C(c2c(C)cnn2C)=O)CCCN(C(C2CC2C)=O)C(c2ccccc2)C1 c1(C(N(C2CCN(C(=O)C(C)CO)CC2)CC)=O)noc2ccc(Cl)cc12 N1(C(C#CC(C)C)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)N2CCCC2)C1 c1(C(=O)NCCC2CCN(C(CNC(=O)NC3CC3)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(NCc2cc(C)cc(C)n2)cc(Br)ccc1S(=O)(=O)NC(CCC)CSC CN=c1[nH]cc(C(=O)N(C(C)CNC(=O)CSCc2ccc(Cl)cc2)CC)s1 C12(C(=O)NC(C(C)O)CO)CCC(C(=O)Nc3nccc(Br)c3Cl)(CC1)CC2 c1(N2CC(C)C(NC(=O)CC3CCCC3(F)F)CC2)ncnc2sc3c(c12)CCC3 C(CC(C)(C)CNC(=O)C(C)Oc1ccccc1F)NC(C(CC)O)=O CCC(C)C(C(=O)N1CCC1Cn1cc(-c2ccc(OC)c(N)c2)nn1)N(C)C C1(CN(C2CCCCN(C(=O)OC(C)(C)C)C2)C)CCCCCCCCCCCC1 C1(C(=O)NCC2CCC(CC)O2)CCCCN1C(=O)C(CC)OC CCCCCC(C)(c1nnnn1C1CCOC1)NCc1cc(Cl)cs1 Cc1nn2c(c1C(=O)NCC1(C)CC(NC(=O)CC3CC=CCC3)C1)CCCC2 n1(CC(=O)NCC2CC(F)CN2C(c2cnsn2)=O)cccnc1=O N1(C(c2cc(CCC)[nH]n2)=O)CC(C(=O)NC2CCCSC2)C(F)(F)C1 c1(C(=O)NC2C(NC(C3CN(C(=O)OCC)C3)=O)C2)nnc(O)nc1O CC1CN(C(=O)CCN(C)CCO)CC(C)C1NC(c1ccc(S(C)(=O)=O)o1)=O C(CC(C(=O)N(C(C)(C)CC(=O)N(C1CN(C)CC1O)C)C)OC)OC c1(OC)ccccc1OC(C)C(=O)N(CC(C)NC(=O)CCc1cn[nH]c1)C CC1=C(C(=O)N2CC(C)(NC(c3ccc(-c4ccco4)nc3)=O)C2)CCO1 C12(C(=O)NCC(CC)NC(c3ccc(O)nc3Cl)=O)CC3CC(CC(C3)O1)C2 C12(NC(CS(CC)(=O)=O)=O)CCN(C(c3cnc(C(F)(F)F)nc3)=O)CCC1C2 C(C)(C)(CCC(=O)N(C1CC(CNC(C2CCOC2)=O)C1)C)OC C1(NC(c2nc(C)sc2)=O)CCCN(C(C23C=CC(CC2)C3)=O)CC1 C1(C(C2C=CCCC2)Nc2nnnn2CC2CC2)CCN(c2ncccn2)CC1 CN1CC(O)CC1(C)C(=O)NCCNC(C1CCCCN1C(c1ccccc1)=O)=O c1(OCC(=O)NCCC(C)CCNC(C2CC=CCC2)=O)nc(O)nc(O)n1 N1(C(CCC(=C)Cl)=O)CCCC(NC(c2cnc(C)c(Cl)c2)=O)C1C CC1(C)CC(CNC(=O)CC2(O)CCC2)CN(C(c2cnoc2C2CCC2)=O)C1 C1(NC(c2cc[nH]n2)=O)CN(C(C2(c3ccccc3)CC(O)C2)=O)CC1C1CC1 Cc1ccc2c(O)c(C(=O)NC(C)(CNC(=O)C(O)C3CC3)C(C)C)cnc2n1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)F)cnn2ccc(O)nc12 CCC(C)(C(=O)NCC1(O)CCN(C(=O)Cc2ccc(F)cn2)C1)C(N)=O C1(C(=O)NC(c2ccc(OC)cc2)CC)CC2COCC(C1)C2N c1(COC)ccc(C)cc1-c1cscc1C(=O)NCCC1CCCN1C c1(CC(CNC(=O)C=Cc2nccs2)N(C)C(C2CC2C(F)F)=O)ccccc1 C(=O)(C(F)(F)C(C)(C)O)N(C(CC)C(=O)NCC(O)COC)C c1(C(=O)NCC2CC(OC)CN2C(c2ocnc2C)=O)ccn2ccccc12 c1(N2C(C(=O)Nc3cc(C)c(Br)nc3)CC(F)C2)nc(S(C)(=O)=O)ncc1C N1(C(CC2N(C(C(C(C)C)O)=O)CC2)=O)CCOC2(CCC2)C1 c12ccc(cc1)C(O)NCCOCOC2=O.C(CCN(C)C)ON.CC C(=O)(CC=C(Cl)Cl)N1CC(CC(CN(C)C(=O)OC(C)(C)C)=O)C1 Cn1cc(C=CC(=O)NCCC(O)CNC(=O)Cc2cccc(Br)c2)nn1 Cc1sc(Cl)nc1C(=O)N(C)CCNC(c1cnn(C2CC2)n1)=O N1(C(c2nn(CC)c(=O)cc2)=O)CCc2nn(C)c(=O)cc2C1 C1(C(N2C(C(C)C)CC2)=O)(NC(C2CC(=O)C2(C)C)=O)CCN(C)C1 c1(OC)ccc2c(c1)OCC2NC(=O)NCc1cc(P(C)(C)=O)ccn1 C1(N(C(C2N(C(CCNC(C)=O)=O)CC(C)C2)=O)C)CC(C)CC(C)C1 C(C)(CO)(C(=O)N1CC(C(O)C(N2CCOC(C(C)(C)C)C2)=O)C1)OC c1(-c2ccc(C#N)c(F)c2)ccc2sc(C(=O)Nc3c(F)cccc3Br)cc2c1 c1(C(N2CC=CC(NC(c3cnn(C)c3F)=O)C2)=O)cc2nccnc2cc1F N1(C(C(C)(C)C)=O)CC2CCC(NC(=O)CCc3cccc(C(=O)OC)c3)(C2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(C)NC(C2(CO)CCCC2)=O)C1 C1(NC(=O)CSCc2cscn2)CN(C(C23COCC(C2)OC3)=O)CC1C1CC1 CC1=CCCN(C(C2CC(C)N2C(c2nccn2C)=O)=O)C1 CC(C)CC(CNC(=O)C(C)C(C)C)C(=O)N(C(C(N)=O)C1CC1)C c1(C(N2CCCC(C)(NC(=O)CN3CCC(F)(F)C3)C2)=O)ccc(F)c(N)c1F C(=O)(CC(CC)CCCC)NC(CC=CC)C(=O)NC(c1ccncn1)C c1(C(=O)NC2C(C)CCN(C(CC(=C)C)=O)C2C)cnc2ccc(C)cn12 N1(C(CC2OCCN(C(C(C)C)=O)C2)=O)CCCC12CCOC2 C1(C(N(C2CC2)CC)=O)CC(OC)CN1C(=O)CC1(OC)CCC1.C1(=O)CN1 C(=O)(C1=CC2C=CC1C2)N(C(C(=O)N(C(CC(CC)C)C)C)C)C N1(C(C)C)C2CCC1CC(N=c1ccn3ncc(S(=O)(=O)NC4CC4)c3[nH]1)C2 CCC(C(=O)NC(C)CCNC(C1(CC)CCC1)=O)OC1CCCC1 N1(C(CCCC(C)C)=O)CC2(CCC(C(=O)NCc3cncnc3)O2)C1 CCC(C)C(C(=O)N1CCC1CNC(=O)Cc1ccc(C)nc1O)NC(=O)OC CCN(C)NC(=O)Cn1cc(SCCOC(=O)COC2CCCCC2)nn1 C1(NC(CCOCC)=O)CC2CCC1C1CN(C(=O)C3=CCCC(C)(C)C3)CC21 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C(C)n2ccnn2)=O)c(F)c1 c1(CCC(=O)NC2CCCN(C(c3c(C)nccc3)=O)C2)ccc(Cl)cc1O N1(C(c2n(CC)ncc2C)=O)CCC2(C=C(C(=O)Nc3ccc(F)nc3C)C2)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(C)CC(C)(F)F)CC2)=O)c2sccc12 c1(CCC(=O)N(C(C(=O)OC)C2CCCO2)C2CC2)ccc(O)c(OC)c1 C1(NC(C2C(OC)CCC2)=O)CC(NC(c2cc(C3CC3)no2)=O)C(O)C1 C#Cc1ccc(NC(=O)Nc2ccccc2C(=O)NC2(C#C)CCCCC2)cn1 C(CC(C)C)(C(=O)NCCC(C)(C)C)N(C(C(CCCC)O)=O)C N1(C(C2(CC=C)CCCC2)=O)CC2CC2(C(=O)NCc2cccc(C3CC3)c2)C1 C1(NC(CC(C)(C)F)=O)CCCN(C(=O)CCc2ccc(Cl)cc2Cl)CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)(C)C1C(=O)NOCC1CCCCC1 C1(CNC(C=CC(C)C)=O)CN(C(=O)CCC2CC2(C)C)C2(CCOCC2)C1 CCC(C(C)(C)O)NC(C1CCC(NC(=O)CC2CCC(=O)C2C)CC1)=O CC1(C)Cc2cc(C(=O)NC3CCN(c4cc(F)ncn4)CCC3CO)sc2C1 C1(NC(CCOCC)=O)CCCC(C(=O)N(C)CC2(C#N)CCC2)CC1 CC(C)CC(C(=O)NCCn1ccnn1)ONC(=O)Cc1ccccc1Br c1(CC)nc(O)c(C(=O)NC2CCN(C(=O)CC3C=CCC3)CC2)cc1C c1(OC)ccc(C#N)c(NC(C2CCCC(NCC3(F)CCC3)C2)=O)c1 Cc1ccc(C(=O)NC(C)CCNC(C2(CC(C)C)CCC2)=O)cc1Cl N1(C(C(C)OCCOC)=O)CC2CCC(N(C(=O)Cc3cncs3)C)C2C1 C1(C(c2cn(C(C)(C)C(=O)O)nn2)C)C(=O)NCCN1CC1C=CCC1 O=NN1CCCC1C(N1CC(CCNC(C23CC(CN2C2CC2)C3)=O)C1)=O Cc1noc(C)c1C(C)CC(=O)N(C1CCN(C(=O)CCC2CC2)C1)C C1(C(=O)NCCC2(NC(COc3cc(C)on3)=O)CCCC2)CC(=O)N(O)C1 N1(Cc2c(C(=O)OCC)ccs2)CCSC(C(=O)Nc2ccnc(F)c2)C1 N1(C(c2ncn(CC)c2)=O)C2CCC1(CNC(=O)CC1CCCC(F)(F)C1)CC2 N1(C(CC=CCC)=O)CC(O)CC1C(=O)Nc1cnoc1 c1(N2CC(C(=O)Nc3c(OC)nccc3C)SCC2)ncnn2ccc(Br)c12 C=CCCCCC(=O)NC(C)CNC(C1CC1c1ccccc1)=O c1(C(=O)NC2CC(NC(Cc3c(C)cccc3)=O)C(O)C2)c(Cl)ccc(F)c1N C(=O)(C1=CCCSC1)N1CCC(N(C(=O)CCCNS(C)(=O)=O)C)C1 C(=O)(C1=CCCOCC1)N1CCC(CN(C(=O)CC2CCCS2(=O)=O)C)C1 CCC(CC)CC(=O)N1CC2CC(NC(=O)Cc3cc(F)ccc3C)C1C2 CC1=CCN(CCNC(=O)CCCCNC(C2CC2C2CC2)=O)CC1 N1(C(CN(C)C(=O)C2CC2)=O)CC2CCC1C2NC(=O)COC1(C)CCC1 Cc1ccc(Br)c(CC(=O)NC2CC2C(=O)NC2(c3cc(C)on3)CC2)c1 c1(C(N(C2CCN(C(C(CC#C)C)=O)C2)C)=O)ncc(C(=O)OC)cc1Cl C(=O)(CC(C)C(C)C)N1CC(CNC(c2nc(C)n(C)c2)=O)C(C(F)(F)F)C1 C1(OC)CCCCC1C(=O)NCC(C1CCCC1)NC(=O)C=CC1CCCC1 c1(C(=O)NCCOC2CCN(C(C3(C)CC(C)C3)=O)C2)cnc([N+](=O)[O-])n1C CC1CC(CNC(c2occc2CN(C)C)=O)CCN1C(C1CCSC1)=O N1(C(c2cncc(N)n2)=O)CCCCC(CNC(c2cc(Cl)cs2)=O)C1 C=CCC1CNC(=O)C2(CCOCC2)CN(CC)C1=O.c1(CO)ccc(Br)cc1 C1(CNC(C2(C(=O)NC)CCC2)=O)CN(C(=O)C=C(C)I)CCO1 Cc1cc(I)ccc1C(=O)NC1CC(NCc2c(Cl)ccnc2Cl)C1 c1(NC(CCC)C)ncccc1S(=O)(=O)NC1CC(NS(=O)(=O)NC)C1 C1(CC=C)CC(NC(C2C#CCCCCC2)=O)CC(CC(=O)OC)O1 Cc1ccc(CC(=O)NC2CC23CCN(C(C2CCC(C)C2)=O)C3)cc1F N1(C(=O)C(c2ccccc2)O)CCCN(C(C2(F)CC=CC2)=O)CCC1 C1(C)(C(=O)OCC)CCCN1CC1CCC(C(F)(F)F)CC1 C(C(=O)NCC1(C(N2CCC2CC(C)C)=O)CC2(CC2)C1)(C(C)C)OCC C1(COC)CC2(C1)CN(C(c1nc(OCC)ccc1C)=O)C2.C12(CCC1)C(=O)N2 N1(C(c2c(C)scn2)=O)CCCCCC1CNC(C12CCC(C(F)F)(CC1)C2)=O Cc1cnc(NCC(C)NC(c2nn(C)c(Cl)c2Cl)=O)nc1S(C)(=O)=O C1(c2sc3cc(C)sc3n2)CC2(CCN(Cc3ccc(N4CC=CC4)cc3)CC2)C1 Cc1ccc(COCCCCc2cn(CC(=O)NC3CCCC4CC34)nn2)cc1 CC(F)CC(=O)NC1CCCC1CNC(=O)C(F)(F)C1(O)CCCC1 C1(F)(CNC(C=CCOCCOC)=O)CN(C(=O)C(C)(C)c2ccsc2)C1 Cc1cccc2sc(C(=O)NC3CCC4CC3CN4C(=O)CCCC#N)c(Cl)c12 C1(CCNC(c2n(CC)ncn2)=O)COCCN1C(=O)CCOCCCOC Cn1ccc(=NC(=O)c2ccnc(CNCc3cccc(O)c3)c2)[nH]1 n1(CC(N2C(C)CCC(NC(=O)CCC(F)F)C2)=O)cc2ccccc2n1 N1(C(c2nncc(OC)c2)=O)CC2CCC1C(C(=O)NCC1CC(C(=O)OC)C1)C2 C=CCC(C(=O)N1CC2(CC(CC(=O)NCC3CCOC3=O)C2)C1)C(C)C N(C)(CP(C)(C)=O)C(C1(NC(c2cnc(C)o2)=O)CCSC1)=O Cc1ccccc1C(C)CC(=O)NC1CCC1CNC(c1c(C)cnn1C)=O Cc1[nH]nc2cc(C(=O)NCC3C4CN(C(C5CC5F)=O)CC34)ccc12 c1(C(=O)NC(CCCNC(C(CCSC)OC)=O)C)nc(C)c(C)nc1O CC1CN(C(c2cnc3[nH]cncc2-3)=O)CCCN1C(=O)CC1CC(C)(C)OC1=O N1(C(C2CC(OC)(OC)C2)=O)CC2CCC1C(NC(c1c(Cl)cnn1C)=O)C2 C1(COC)(CNC(=O)C(N)=O)CCN(C(=O)CC2CCCN2C(C)C)C1 C12(CNC(C(CC)(C)C)=O)CCCC1CCN2C(=O)CNC(=O)C(CC)CC c1(SC)cc(C(=O)NC2CCC(N(C(=O)CC3(CO)CC3)C)C2)ccc1F c1(C(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cnc(C(N)=O)cn1 C12(C(N(CC)CC3CCC3)=O)CCC(NC(=O)Cc3ccccc3F)(CC1)C2 O(N1CCC(N=c2cc(C)[nH]c(=NCC3CCC(C)O3)[nH]2)CC1)CC N1(Cc2ccn(CC=C)c2)CCC(O)C(C(=O)NC(C)Cc2ccccc2F)C1 c1(OC)cccc(C(=O)N(C)CCN(C(=O)C=C2CCC(C)C2)C(C)C)c1 C1(C(=O)NC(COC)CO)CC12CCN(Cc1nc(Cl)ccc1F)CC2 Cc1nc(C=CC(N2CCCC2CNC(C2CC(C)(O)C2)=O)=O)[nH]c1C C(CC(C)(C)CC(=O)N1CCCCC1CC(N1CC2CC(F)CC2C1)=O)OC C(C(CC1CCOCC1)CO)NC(=O)NC1CC(OC(C)C)C1 Cc1ccc2oc(N3CC(C)(C)CCC3CNC(=O)C(C(C)C)N(C)C)nc2c1 CC1=C(C(=O)NCC2CCCN(C(=O)Cc3cncc(C)c3)CC2)CCC1 N1(C(=O)OC(C)(C)C)CC2CC(C1)C2NCCN1CSCC1=NCl CCCC(C#N)C(=O)N1CCN(C(CNC(c2cc(C)c(C)o2)=O)C(F)F)CC1 c1(CCOC)nc(=NC(C)C2CCN(C(c3c(F)ccc(F)c3Cl)=O)C2)s[nH]1 c1(C(=O)NC(CN(C(=O)C(C)CC2CC2)CC)C)ccc(OC)cc1Br N1(C(c2c(C)nco2)=O)CC2CC2(NC(c2ccc(SC(F)(F)F)o2)=O)C1 c1(OC)cc(C(=O)NC23CC2CN(C(=O)COCc2ccccc2)C3)ccc1C N1(C(c2nc(COC)oc2)=O)CCCC(CCNC(C2CC3(CC3)C2)=O)CC1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(N(C(=O)Cc2cncc(F)c2)C)C1 S(=O)(=O)(c1cccnc1N1CCC(C#N)C1)NCC1OCCN(C(C)(C)C)C1 N1(C(c2c(OCC)n[nH]c2)=O)CCCCC1C1(NC(c2cccs2)=O)CC1 Cc1nc2cc(Br)cc(NC(c3ccc(CCc4cccs4)cc3)=O)c2o1 c1(C(N2C(C(=O)Nc3c(C#N)scc3)CCCC2)=O)c(Cl)cccc1Cl N1(C(c2cc(COC)[nH]n2)=O)CC2CCC2(CNC(=O)CCC(C)N(C)C)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(F)C3CCC3)C2)cc2cccc(F)c2s1 C(=O)(C(c1cccs1)=Cc1cccs1)N1CC(NC(C2CCN(CCC)C2)=O)C1 N1(C2CCN(C(C(F)=CC)=O)C2)CCN(C(C2OCCC2C(F)(F)F)=O)CC1 CC1OC2(CNCC(c3cccc(Cl)c3)O)CC1(CO)C2 c1(C(=O)NC(c2ccccc2F)CNC(c2ccc(C)s2)=O)cncc(N)c1 CC(C)(CC(=O)OC(C)(C)C)c1ccccc1.C12CN(CC1O)C1CN(C1)C2=O C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC2CCN(C(c3cn(C)nn3)=O)CC2C1 c1(OC(C)(C)C)cc(NCC2C3COCC23)cc(F)c1 C(=O)(CCCCC(C)C)NCC(CC=C)NC(c1cncc(C)n1)=O C1=CC(=O)OC(C2CCOC2)C(=O)NC1(C)C.C1(=O)C=CCN1.C(=O)(C=C)OC N1(C(C2CCN(C(CC3(OC)CCC3)=O)C2C)=O)CC2(CNC(=O)OC2)C1 CC(C)(C)C(C)(C)C(=O)N1CCC(=CCNC(C2Cc3nccn3C2)=O)CC1 Cc1cc(C)c(S(=O)(=O)NCc2ccc(F)c(S(N)(=O)=O)c2)cc1[N+](=O)[O-] c1(OC)ncccc1C(=O)C(=O)NCC1CC1CNC(C1(C)CC2CC2C1)=O c1(NC(CC(CNC(C2CC3C(C2)C3(F)F)=O)OC)=O)cccc2nccn12 C12(NCCN(C(C(Cc3ccc(C)cc3C)C#N)=O)C)C3C4C1C1C2C3C41C CC(C)CC(C)C(=O)NCC1(O)CC(C(=O)NCC(O)C2(Cl)CC2)C1 C1(CNC(=O)Cc2ccsn2)C2CN(C(C3CC3c3cccc(Cl)c3)=O)CC12 Cc1cnc(C(N2CCC(CCNC(C3(c4ccsc4)CC3)=O)CC2)=O)c(F)c1 c1(N(C(=O)CC2CCCN2C(c2n[nH]c(C3CC3)n2)=O)CCC)ccc(C#N)cc1 N1(C(c2cc(Cl)nc(Cl)c2)C(=O)OC)CCN(c2nccc(OC)n2)CC1C C1(CC(=O)NCCC(C)N2CCCC2)CN(C(C2CCCC(=O)N2)=O)C(C)(C)C1 c1(C(=O)NC2CCC(CNC(C3CC(C(C)C)C3)=O)C2)nccc2ncccc12 C(CNC(=O)CN1CC2CCC1C2)(CC(F)(F)F)NC(CC)=O N1(C(COC)=O)CC(NC(=O)CC(C)(C2CCC2)N(C)C)C2(CC2)C1 N1(C(C(C)=C2CCC2)=O)CC2CC(NC(=O)C(C)(C)c3cncnc3)C2C1 CCCS(=O)(=O)CC(=O)NCC12CN(C(=O)C(C)(C)n3cccn3)CC1CCO2 N1(C(C2C(C)=C2)=O)CCOC(C(C)NC(C2CC3C=CC2C3)=O)C1 C12(CNC(C3(C#C)CC3)=O)CCC1CCN2C(=O)Cc1ccc(C#N)cc1 c1(CC)cc(N2CCC(CCNC(c3oc(C(C)N)nc3C)=O)C2)ncn1 CC1CCSCCN1C(C1(NC(C2CCCC2O)=O)CCC(C)(C)C1)=O c1(CC)oc(C)cc1C(N1CCCC(CNC(c2ccc(C3CC3)cc2)=O)C1)=O C1(CC=C)(C(=O)NC(C)CN(C(C2CC(OCC)C2)=O)CC)CCC1 N1(C(C(C)NC(N(C)CC)=O)=O)CCCC(C(=O)NCCCc2ccccn2)CC1 c1(N2CCOCC(NC(c3c(C(C)C)cccc3)=O)C2)c(Br)cccc1[N+](=O)[O-] C#Cc1cccc(C(=O)NC2CCCC2NC(=O)CCCN=[N+]=[N-])c1 C1(CC)(CC)CC(NC(c2nnc(S)n2C)=O)CN1C(=O)CC1CC1(C)C n1(CCC(=O)NCCCN(C(=O)C(O)C(C)CC)CCC)c(C)c(C)sc1=O C(=O)(CC(=O)NCCCNC(=O)OC)C1(C(=O)NCC2C(OCC)C2)CC1 n1(CC(=O)OC)cc(C(N2CCC2CNC(C2CCCN(C)C2)=O)=O)ccc1=O CC1=C(C(=O)NCC2CN(C(c3cc(C)ccc3N)=O)CCC2C)SCCO1 C1(O)(C(C)NS(=O)(=O)CC2(C(C)(F)F)CC2)CCCC(C)C1 N1(C(c2ccc(CC)cn2)=O)CCOCC(CNC(=O)CC(C)c2ccco2)C1 O=C1CCC(C(N2CCCC(NC(=O)CSc3nc[nH]n3)C2)=O)CN1 c1(CC)ccc(C)c(NC(=O)C(F)C(C)CNC(=O)C(=O)NC2CC2)c1 N1(C(C2C(c3cn(C)nc3)C2)=O)CCCCC12CC(NC(=O)CC(F)(F)F)C2 CN1CCC(C(=O)NCCC2CCC3CC23)(NC(C2(C(=O)NC3CC3)CC2)=O)C1 N1(C(C(CC)(C)O)=O)CCCC2(CCN(C(=O)CC3CCCC34CC4)CC2)C1 c1(COCC(=O)NC(C2CCCC2)CNC(C2(CC)CC2)=O)cccc(Cl)c1 c1(NCC(C)CO)nc(N2CCCNC(=O)CC2)nc2ncn(C)c12 CC12CN(C(c3cccnc3O)=O)CC1(C)CN(c1ccnc(S(C)(=O)=O)n1)C2 N1(C(c2ccc(CC)o2)=O)CCCCC1CC(N1CCC(C)(F)C1)=O c1(OCC=C)ccc(C(=O)NCC(CO)NC(=O)C(C(C)C)NC(C)(C)C)cc1 C1(C(=O)NC2C(NC(CN3CC(C)C3)=O)COC2)CC(C2CCOCC2)=NO1 C(=O)(CC1=NNC(=O)C1)NC(CN(C)C)NC1CC(SC)C1 CCCC#CC(C)(C)NC(=O)C(C)NC(=O)C(C)n1cccn1 C(=O)(CS(=O)(=O)CCOC)N1C(C)(C(N(CC#C)CC=C)=O)CC(O)C1 c1(C(=O)NC2C(NC(C(CC)C)=O)C2)ccc(COc2ccccc2)cc1 C1(C(N2C(C)CN(C(c3cccn3C)=O)CC2)=O)CC(c2ccncc2)=NO1 c1(CC)ccccc1C(=O)N(C1CN(C(=O)CCN(C(CC)CC)C)CC1F)C C1(C(N(C2CC(C#N)C2)CC(=O)NC(c2cnsc2)C)=O)CC12CCOCC2 C1(C(=O)NCC2OCCC(NC(C(CN(C)C)(C)C)=O)C2)C(F)(F)C12CCC2 N1(C(Cc2ccc(OC)cn2)=O)CCC(C)(C)C(CNC(=O)C(O)C(F)F)C1 O(NC(=O)CN=c1ccnc(CCN2CCCCCC2)[nH]1)CCOCCOC n1(CC)ncc(Cl)c1C(=O)NC1CC(F)(CNC(=O)C(c2ccc(Cl)s2)=O)C1 c1(CN2CC(CCC)C(CO)C2)ccc([N+](=O)[O-])cc1F CC1CC=CCC1C(=O)N(CC(O)CN(C)C(c1ccc(OCCF)cn1)=O)C c1(C(N2CCN(C(COC(CC)C)=O)CC2C)=O)ccc2c(c1)nnn2CC c1(C(=O)NC2(CC(N3CCC(C)(O)C3)=O)CCC2)ccc2[nH]ccc2c1 c1(OC)cncnc1C(=O)NC1(CCC(=O)NC2CCC2O)CCC1 c1(C(=O)NC(CN(C(=O)C(C)NC(C)=O)CC)C)cccc([N+](=O)[O-])c1N c1(C(=O)NCC(C)CNC(=O)C(C)(C)c2ccno2)ccc2nccn2c1 C1(CNC(C2(c3cccc(Cl)c3)CC2)=O)CC2CCC1N2C(=O)CCCCO c1(C(CNC(C2CNC(=O)N2)=O)NC(c2ccco2)=O)ccccc1F c1(-c2cnc(OCC)nc2)cccc2[nH]nc(C(=O)NCCc3nn[nH]n3)c12 c1(CC(=O)NC2CN(C(c3cc(Br)no3)=O)C2)ncc(F)cc1F N1(C(CSCCCC)=O)CCC(C(=O)NC(C)C)C12CC2 Cn1cnc2c(NC(c3ncccc3NCC3CCCS3)=O)ncnc12 CCCCCC(F)C(=O)NCCNC(c1cc(O)ccc1F)=O C(=O)(CN=S(C)(C)=O)NCc1c(CN(C)C(C2CC2C(F)F)=O)cccc1 C12(C(N3C(C)CN(C)CC3)=O)CCC(CC1)N(C(c1cccc(F)c1)=O)C2 C1(CCC)CN(C(=O)C=C2CCSCC2)CC1C(=O)C.C1(=O)C(OCC)ON1 c1(C(=O)NCC2(NC(c3ccncc3Br)=O)CCC2)cc2cccnc2cn1 N1(C(C2CC2[N+](=O)[O-])=O)CC2CC(C1)N(C(c1ccc(-c3cccnc3)s1)=O)C2 c1(C(=O)NC(CNC(COCCOCC)=O)CC)c2n(c(=O)n1C)CCCC2 Cc1cnc(C(=O)NCCNC(c2onc(C)c2C)=O)cc1C CC(C)CC(c1nnnn1C1CCCC1)NCc1csc(Cl)c1 N1(C(Cc2cccc(C#C)c2)=O)CCC(F)(F)C(CNC(c2sccc2C)=O)C1 N1(C(c2c(CC)nccn2)=O)CCC2C(CCCN2C(=O)C(C)CSC)C1 C1(NC(CCCOC)=O)CC2CCC(C1)N2C(c1ncsc1C(F)(F)F)=O c1(C(=O)NC2C(CNC(C(C)CF)=O)CC2)ccc(C(F)(F)F)nc1 CC(C)CC(=O)C(=O)N1CC2C(NC(=O)COc3ccsn3)C2C1 CCC(C)C(O)C(C)C(=O)NC(COC)CC(=O)N(C)CCN1CCCC1=O C(=O)(C(F)(F)C(F)(F)F)N1CCCC(CNC(C(C)(c2ccccc2)OC)=O)C1 c1(C(N2CCN(C(C(CCCC)N(C)CC)=O)CC2C)=O)cc2cc(Cl)sc2[nH]1 C(=O)(CC(C)C(=O)N1CCCC(NC(=O)COCCO)C1C)OC CC(CC(=O)N1CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1)P(C)(C)=O Cc1cc(F)ccc1C(N1CC(=O)CC1C(N1CCC(F)CC1)=O)=O C#Cc1ccc(C(=O)NC2CCCCC2CNC(=O)C2=CCC2)nc1 C#Cc1ccc(F)c(C(C)NCC2CCN(c3ccc(F)cc3F)C2)c1 c1(C(=O)NCC2CCN(Cc3cccc(C)n3)C2)ccc(Br)nc1Br CC(C)(C)CCC(=O)NCC12CC(NC(C3CCCN3C3CC3)=O)(C1)C2 c1(CC(=O)NC2CC(C)N(C(=O)CP(C)(C)=O)CC2)cn(C)c2ccccc12 c1(COCC(=O)N(CCNC(=O)C(F)OC(F)(F)F)CC)ccc(F)cc1 N1(C(C(C)Cn2ccnc2)=O)CCC(CO)(CNC(=O)Cc2cn(C)cn2)C1 Cc1ccc(SCC(N2CC3CC3(NC(=O)C(O)C3CC3)C2)=O)c(C)c1 C12(CNC(C(C)N(C(=O)C(C)NC(=O)OC)CCC)=O)COC(C1)C(O)C2 Cc1cc(=NCCCC(C)O)[nH]c(N2CCC(c3c[nH]c(=N)[nH]3)CC2)n1 CCC(CC)C(=O)NCC(=O)NC(C)CNC(=O)C(C)(CC)OC CC(C)C(CNC(C1CC2COCC2C1)=O)C(=O)N1CCCC1CN(C)C c1(C(N2CC3C(NC(CN(CCC)C)=O)(C3)C2)=O)cc(Cl)cc2c1CCC2 n1(C(COC)C)nc(-c2ccc(N)cn2)nc1CCc1cc(C)no1 CC(N=c1nc(N2CC(=O)NC(C)(C)C2)c2ncccc2[nH]1)c1ccoc1 C1(C(=O)NCC2(O)CC(NC(C34COCC3C4)=O)C2)CCC2(CCCCC2)CC1 C1(NC2(CC(=O)OC)CCCOC2)CC2(CCCCCC2)C1 c1(OC)ccc(CNc2cccnc2C(=O)NCC2CCC(C)CC2)c(OC)n1 CCC(C(=O)NCCOCCNC(=O)Cc1c(C)nn(C)c1Cl)C(C)(C)CC C(=O)(C(C)(C)N=[N+]=[N-])NCc1c(C(=O)NCCc2nc(C)[nH]n2)occ1 C1(C(=O)NCC2CC(NC(c3cnn(CCO)c3)=O)C2)CCC(n2ccnn2)C1 C(=O)(CC1=CCCC1)NCCC1CCCN(C(CCCc2n(C)cnn2)=O)C1 N1(C(C2C3(CC(OCC)C3)C2)=O)CC(NC(C2CC3CC3C2)=O)CC2(CC2)C1 C1(C(=O)NCC2N(C(c3cc(N)cc(F)c3)=O)CC=C2)CCCC2(CCC2)C1 CCCCC(CC)CC(=O)NC1CCC(CNC(C2C3CCC(=O)C23)=O)C1 Cc1ccc(F)c(C(=O)NCC2CCCC(NC(=O)CN(C)C(=O)C3CC3)C2)n1 c12ccc(cc1)[nH]c2=O.c1(C(N2CCC(CC)C2)C(=O)OCC)cccc(F)c1 CC(=O)CCCC(=O)NC(C)(CNC(=O)CCCc1nncn1C)CO CCCC(F)C(=O)N1CCC2CC12C(=O)N(C)Cc1ccncc1 c1(CCC(=O)NCC(CO)NC(C2C(c3onc(CC)n3)C2)=O)cncnc1O CC(C)C(O)C(F)(F)C(=O)N(C)CC1CCCC1NC(=O)C(C)Cc1cnco1 C1(CNC(COC(CC)CC)=O)CCCN(C(=O)CCCC2(N(C)C)CCC2)C1 c1(C2(NC(C3CC(O)(c4cccnc4)C3)=O)COC2)cccc(Cl)c1 C(=O)(CCP(C)(C)=O)NCCC1(O)CCN(C(Cn2cc(CN(C)C)nn2)=O)C1 C(CCCCCCCO)=CC(N1CC(CNC(C(C(C)C)OC)=O)N(C)CC1)=O C(N=c1cc[nH]c(-c2nccs2)n1)C1CN(C(=O)NC2C(C)(C)CCC2)C1 c1(C(C)OC)nc(C)c(S(=O)(=O)N2CCCCC2C(=O)OC)s1 Cc1ccc(C(=O)NC2CCC(C(=O)N(CC(C)C(C)(C)C)C)CC2)nn1 C(N=c1ccn2nccc2[nH]1)C1CCCN(Cc2c(OC)cccc2F)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCN(c3ccc(S(N)(=O)=O)cc3)CC2)=O)c1 c1(C(N2CC(C)(C)C(C(=O)NCC3(C)CC4CC4C3)C2)=O)c[nH]c2cnccc12 N1(C(C(CC)OC)=O)CCCCC(C(=O)NC2CC2(C)C)C1 C1(NC(C(CCCC)O)=O)COC2(CCN(C(c3cncs3)=O)CC2)C1 Cc1ccc(C(C)NC(=O)C(CNC(=O)C(O)C2CCCC2)N(C)C)nc1 Cc1nc(=NCCCCC(C)NC(C2CCCN2C(N)=O)=O)[nH]cc1Br c1(C(C(=O)NC(C=C)(C)C)NC(=O)C(c2ccn(C)c2)C)cccc(OC)c1 C(=O)(C1CCc2c[nH]nc21)N1CCC2(C(NC(c3n(C)c(S)nc3)=O)C2)C1 C(=O)(C(C)CCO)NCC(C1CCCC1)NC(CN1C(C)CC1)=O C1(CNC(=O)Cc2csnn2)CCN(C(C2CCC(=O)N2C2CC2)=O)C12CCC2 c1(C(=O)NCC(CNC(CSCCC)=O)F)cnn(CCF)c1 C1(C2(NC(CC(=C)Br)=O)CC2)CCCCN1C(c1ccccc1SC)=O c1(C(N(CC(C)O)CCNC(C2N(C(C)=O)CSC2)=O)=O)ccc(C)n1C c1(OC)cc(C)c(C(N2CC3C(C2)N3C(=O)CCC(F)(F)F)=O)c(C)c1 N(C1CCCc2cc(N)ccc21)C(Cn1cc(OC)c(=O)cc1C)=O C1(CC)CCN(C(C2CCCS2)=O)C1CNC(c1cccc(OC)c1)=O c1(OCC)cc(C(N2CCS(=O)(=O)CC2)=O)c(-c2cc(O)cc(F)c2)cn1 Cc1cc(C(=O)N(C2CCSC2)C(=O)NC(C2CCCO2)C2CCC2F)cc(C)c1Cl N1(CC)CCOCC1CC(=O)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CC1 N1(c2ncc(C)cn2)CCOCC(CNC(=O)CC2CCCCCC2)C1 c1(C(CNC(C2C(C)C2C)=O)NC(=O)C=CCN2CCOCC2)ccccc1F N1(C(C(C)C(C)O)=O)CCCC(C)(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(NCc2c(C)ccc(OC)c2)ccc(=NCCN(C(=O)C(=O)NC)C)[nH]c1 C1(CN(C(c2cc(C(C)C)[nH]n2)=O)C)CCCC(NC(C2(Br)CC2)=O)C1 C1(NC(c2cc(OC)n(C)n2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1nccs1 c1(NC(c2n(C(C(=O)OC)C)nnn2)C2(CN(C)C)CC2)ccc(C)c(C#N)c1 CCC(CC(=O)NCC1CC(C(=O)NC(C)Cn2ccnn2)C1)OC C12(CC(=O)NCCNS(CC)(=O)=O)CCC1CN(C(=O)C(C(C)C)N(C)C)C2 S(=O)(=O)(CC(=O)N1CCC(O)(C(C)NC(=O)COCc2cccc(C)c2)C1)NC Cc1nc(N2CC(O)(CCNC(c3ccco3)=O)C2)cc(-c2ccco2)n1 Cc1cn2cc(C(N3CCC(=CCNC(c4cc5n(n4)CCC5)=O)CC3)=O)nc2s1 C1(C)(CC)CC(NC(=O)C2=CCCC2)CN1C(=O)CN1CCSCC1 c1(CC2CCN(C(c3ccn(C)c3)=O)C2)ccc(Oc2ccncc2)cc1 CCCCCCCCNC(=O)C(=O)NCC(c1ccc(OC)c(OC)c1)C C(=O)(C(F)C(C)C(F)(F)F)NCC(CNC(c1cc(C)c(C)s1)=O)O CCCCCC(O)C(C)C(=O)N1CC2CC(NC(C3COCCN3C=O)=O)C1C2 c1(C(N2CCC3CN(C(CCC(C)C#N)=O)CC32)=O)ccc2cccc(F)c2n1 C(=O)(C(O)C(F)(F)F)N1CCC(CNC(c2ccc(CC(C)C)s2)=O)C1 C1(C(=O)NCCN(CCC)C(C2(N(C)C)CC2)=O)CCCC(CF)C1 c1(SCC(N2C(c3cn(CCOC)nn3)CC2)=O)nc2ccccc2o1 c1(C(=O)NC(CNC(C(C)NC(=O)NC)=O)C(C)C)cc2ccccc2oc1=O C=CC1(C(=O)NC(C)CC2CCCCC2)CCN(C(=O)C=C2CCCCC2)CC1 CC1(C)CN(C(=O)CC=Cc2ccc(F)cc2)CC(CNC(=O)C(O)CF)O1 c1(OC)cc(CC(=O)NC(C)CCCNC(C2(CSC)CCC2)=O)cc(Cl)c1 C(=O)(C(CC(C)C)C(N)=O)NCc1ccc(C(N2CC(F)=C(C)CC2)=O)o1 C1(O)(CN(C(C2C(CCC)C2)=O)C)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 N#Cc1cnccc1COC(=O)C=Cc1cccc(-c2ccc(Cl)cc2)c1 O=C1NC(C(=O)NCC=CCNC(=O)C(c2ccccc2)C2CC2)CCO1 C(S(=O)(=O)CCNC(N1CCC(C(=O)O)C1)=O)c1cn(CCCC)nn1 c1(OC)ccccc1-c1nc(SC(C2CCCCC2)C)n[nH]1 C1(CNC(C(CO)N(C)C)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1 C#CC1(C(N2CCC(CCO)C2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C1 N1(CC(=O)N(CC)CC)CCC2(CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)C1 C1(C)(NC(c2cccc(OC)c2)=O)CCC(NC(=O)Cc2ccccc2Cl)CC1 c1(-c2c(C3(C(=O)OC)CC3)cccc2)cc(OC(C)C)c(F)c(F)c1 c1(CC)cc(C(N2CC(OCCNC(C3CC(C#N)C3)=O)C2)=O)c(C)o1 c1(C(N(CCCN(C(=O)C(C)(C)c2ccccn2)C)C)=O)cnn(C)c1N c1(C(=O)NC2CN(c3nnc(CO)s3)C3CCCCC23)cccc(C#CCO)c1 c1(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)sccc1Cl N1(C(c2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccc(F)nc3)=O)C2)C1 Cc1ccc(C#N)cc1C(N1CCC(C)C(CC(=O)NC(CF)C(F)(F)F)C1)=O c1(OC)cc(CCC(=O)NCCCCCNC(=O)C(c2ccc(C)s2)OC)on1 N1(C(C(=O)NC)C)CCCC(NC(=O)CC(C)OC)CC1 N1(C(CCC=CCC=C)=O)CCC(CNC(c2scc(C)c2C)=O)(OC)CC1 CC1(C)CCOC(C(=O)N2CCC(C(=O)NCc3cc(C(N)=O)no3)O2)C1 C1(C(=O)NCC=C)CC2C=CC1N(C(C1Cc3nccn3C1)=O)C2 N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)CN(C(c1ncc(C(F)F)s1)=O)C2 C1(C2(O)CCOC2)(C(=O)NC2C(C)(C)C(CC(=O)O)C2)CC1 c1(C(=O)NCC(CCNC(C(C)OCC)=O)O)ccnc2ccncc12 C(=O)(CCCC(=O)N(C1CCCN(C(c2coc3c2COC3)=O)C1)CC)NCC S(=O)(=O)(c1ccc(C(=O)N(CCC(C)NC(=O)C(O)CCSC)C)cc1)NC c1(C(=O)NCC2(OC)CCN(C(c3ccc(F)c(C)c3)=O)C2)sc(C)c(C)c1C c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)ccc(F)c(F)c1 N1(C(C2N(CCC)CCC2)=O)CCC(O)(C(C)NC(=O)CCc2ccsc2)CC1 c1(C(=O)NCC(C)N(C)C(c2cnn(CCO)c2)=O)cnn2c1OCC(C)(C)C2 N1(C(C2(C(C)C)CCCO2)=O)CC2CC1CN2C(=O)CN(S(C)(=O)=O)C C1(C(=O)N(CC(C)C(C)C)C)(CC)CCCN(C(c2ccc(C(C)C)o2)=O)C1 c1(C(N2CCC(NC(CCc3cn(C)nn3)=O)C2)=O)c(C(F)(F)F)cccc1O c1(CC)nn(C)cc1C(=O)NC1CN(C(c2sccc2C(C)(C)C)=O)CC1C N1(C2CCC(NC(COC)=O)C2)CCN(C(=O)CN2CCC(O)CC2)CC1 N1(c2c(C)c(NCc3ncsc3Cl)ncn2)CCC2(CCCN2C)C1 N1(Cc2c(C#C)cccc2)CCC(CNC(c2cc(F)cc(Cl)c2)=O)C(F)(F)C1 CC1(C(=O)NCC2C3CN(C(=O)Cc4cnco4)CC23)CNC(=O)C1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2O)c1C N1(C(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(C1CC1CF)=O C1(N(c2nccn2C)C(c2cc(C)n(C(F)F)n2)=O)CCC2(CCNC2)CC1 C12(NC(COCc3cccc(OC)c3)=O)CCCC1N(C(=O)COC(C)=O)CC2 C1(NC(CCCN(C)C)=O)CCN(C(C2CC3(CC3)CO2)=O)CC12CCC2 N1(C(C(CCC)OC)=O)CCC(C2CCCN(CCc3cscn3)C2)CC1 Cc1cccc2nc(C(=O)NC(C)(C)CCN(C(=O)C3=COCCC3)C)cn12 C1(C)(COC)CCCN(C(C2CCN(C(=O)CC3(C)CCOC3)C2)=O)C1 C(=O)(C(O)CCCNC(C1CC(C)N(C)C1)=O)N(CC(=C)C)C C1(C(=O)NCC2C(NC(=O)Cc3ccno3)CCC2)Cc2cccnc2C1 [N-]=[N+]=NCCC(=O)NCC1CN(C(c2cccc(C3CC3(F)F)c2)=O)CCO1 N1(C(CCNC(COC)=O)=O)CC(N(C)C(C2CC23CCCC3)=O)C(C)(C)C1 N1(C(CCCCNC(C(C)SCCCC)=O)=O)CC2CCC2(CO)C1 N=c1[nH]c2ccc(C(N3CCC(NC(=O)C#CC4CC4)CC3)=O)cc2[nH]1 N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CC(C#N)C1)=O)C3 N1(S(CC)(=O)=O)CCC2CCC(C1)N2C(c1cncc(CN(C)C)c1)=O CC1c2c[nH]nc2CCC1C(N1CCCCC(CNC(=O)Cc2ccns2)C1)=O N1(C(c2cnc(C(C)C)[nH]2)=O)CCC2(CCC(N(C)C(c3cnns3)=O)CC2)C1 C1(NC(c2cc(CNC(C3(CC)CCC3)=O)ncc2)=O)CN(C)CC1(F)F c1(C(N(CCC)CCNC(c2nsc(OCC)n2)=O)=O)c(CC2CC2)noc1C Cc1nc(N(C)C)sc1C(=O)NC1CC(CCNC(=O)C=CCF)C1 c1(C2C(NC(=O)NCCCc3cc(C)[nH]n3)CC2)cccc(Br)c1 N1(c2c(OCC#C)cc(Br)cc2)Cc2ccc(C(=O)O)cc2C1 c1(C(N2CC(O)(C(C)NC(CC=CCC)=O)C2)=O)cccc(C)c1Br C1(NCCCn2cc(CCNC(c3c(C(=O)O)csc3)=O)nn2)CCS(=O)(=O)C1 c1(OCC(C)C)ccc(SCC(N2CC(NC(=O)CNC=O)C3CC23)=O)cc1 N1(C(c2ccc(C)o2)=O)C2CCC1C(CNC(=O)CC1CCC1(F)F)C2 c1(C(C(C)OC(=O)C#CC(=O)N(C)C)=O)ccc(O)cc1 C12(C(=O)NCCC(C)NC(c3csc(-c4cnc[nH]4)n3)=O)CCC(CC1)CO2 C=C(C)CCC(=O)N1CCC(C(C)NC(=O)CS(C)(=O)=O)C1 C(=O)(C(C(C)NC(C1CCCC1O)=O)C(C)C)NCc1nccc(C)n1 c1(C(=O)NC(C)Cn2cc(CN3CC4CC4C3)nn2)c(Cl)nc2ccccn12 C1(OC(C)(C)C)CC2(CCC(COC(c3cccc(-n4nccn4)c3)=O)O2)C1 CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cnc(O)s1)=O c1(C(=O)NCCOCCCN(C(c2cc(OCC)n[nH]2)=O)C)ccccc1C c1(CC)nnc(O)c(C(N2CCC(CNC(=O)C(O)CCC(C)C)C2)=O)c1CC CCCCCC(C)(C)C(=O)NCC(C)(C)NC(C1CCCN(C(C)=O)C1)=O c1(NC(C(COCC)C)=O)cc(F)ccc1N1CC(C(=O)OC)OC1=O CC(C)C(F)(CNC(c1ccccc1C#N)=O)C(=O)NCCN1CCOCC1C N1(C(c2c(C)ccs2)=O)CCC2(CC1)CN(C(=O)C(C)(C)N1CCCC1)C2 C1(CNC(CSC(C)C)=O)CCCC1C(=O)NOCCCCCC1CC1 C12(Cc3occ(C(=O)NCCN(CCOC)C4CC4)n3)CCCN1CC(OC)C2 N1(C(c2c(C)nncc2)=O)CCC(C)C(CC(N2CC3CC(C)C3C2)=O)C1 Cc1cccc(C(=O)NC2(CCCCNC3CC4CC4C3)CC2)c1 N1(C(CC2CC(C)N(C(C34CCC(C3)C4(C)C)=O)C2)=O)CC=CCC(C)(C)C1 c1(COC(=O)NC(CC(C)C(C(=O)OC(C)(C)C)OC)C)cccn2c(C)cnc12 c1(C(N2CC(C)(OCC(=O)NCC(C#C)CCC3CC3)C2)=O)nnccc1C C1(OC(=O)CCNC(=O)OCCC(=O)NC(C)C)CCCCC1 c1(C(N2CCC(CNC(C(C)N(C(C)=O)C)=O)C2)=O)cc2c(nn1)CCCO2 c1(C(N2CC(NC(C(C=CCCC)O)=O)C(C(F)F)C2)=O)c(F)ccc(F)c1Cl N1(C(CC2C(C)CCN(C(c3cc(C)oc3)=O)C2)=O)CCC12CCOCC2 C(=O)(CCCCN(C(=O)C(=O)Nc1ccccc1)C)NC.C1(=O)C(C2CC2)N1 CC1(C)CC(O)CN1C(=O)CC1(C)CN(Cc2c(I)ccnc2F)C1 N1(Cc2nnc(C)o2)CC2(CN(C(c3ccc(F)c(O)c3)=O)CCO2)C1 c1(C(N2CCC(C)(NC(=O)C3=C(C#N)CCC3)C2)=O)cnn2c(Br)cccc12 CCS(=O)CC(=O)NCC1(F)CC(NC(c2cccn2-c2ccc(F)cc2)=O)C1 Cc1c(C2(CN(C(C34CC(CO3)N(C(=O)C(C)C)C4)=O)C3CC3)CC2)cccc1F C1(NC(c2csc(C)c2C)=O)CCCCCCC1NC(=O)CC1CCCN(C)C1 CCCC(C(=O)N1CC(CCNC(c2ccccc2SC(C)C)=O)C1)OC C(=O)(C(C(C)(C)C)c1cc[nH]n1)OCCOC(C)C#N C#Cc1ccc(Br)c(C(=O)NCCC2(O)CN(C(c3c[nH]nc3F)=O)C2)c1 N1(C(c2c(Cl)cnc(C)n2)=O)CC2OCC(NC(C3(CC(F)F)CC3)=O)C2C1 c1(C(=O)NC2CC(O)(CNC(C3CCC3(F)F)=O)C2)ccc(F)cc1Br c1(CN2CCC(CC(=O)Nc3ncc(OCCOC)nc3)C2)ccc(F)c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(C3OCCN(C)C3)=O)C2)ncnc(O)c1Cl O=C(CCC(=O)c1ccc(F)cc1)NC1CC1NC(C1CC2CC2C1)=O Cc1noc(C)c1CC(=O)NCC1C2CN(C(C3CC(=O)N3)=O)CC12 c1(CC(=O)NCC2(COC)CN(C(=O)C=Cc3cn(C)nn3)C2)cncc(SC)c1 C1(C(=O)NCC)CC(OC(C)(C)C)CN1C(CC(F)COC(C=CC=CC)=O)=O C(=O)(C#CC1CCCOC1)NCC(C(C)C)NC(C1(C(C)=O)CC1)=O N1(C(Cn2nnc(=N)[nH]2)=O)CCOC2(CCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 N1(C(CCC=C(C)C)=O)CC(NC(=O)CCOCC(F)F)CC12CCCCC2 CC(C)CC(CNC(=O)C(C1CCOCC1)F)C(=O)N(CCC(N)=O)C c1(N(C)Cc2cccc(F)c2)nc2ccsc2c(=NCCN(S(C)(=O)=O)C)[nH]1 C1(C(=O)NC(CNC(CC(=O)OC(C)(C)C)=O)(C)C2CC2)COCCN1C=O Nc1c(C(=O)NC2COCC2CNC(C2OCCC2C(F)F)=O)cc(Cl)cc1Cl C(c1cscn1)=CC(=O)NC1(CNC(C(C)=C2CCC2)=O)CCC1 N1(C(c2cc(CNC(c3n(CC)ncc3C)=O)on2)=O)CCC(O)CC1C C1(N2N(CCC(=O)O)C2=O)CC2CCC1CC2N(C)C.CCC(COC)CC C1(CNC(=O)Cn2ccnn2)CC2CCCCC2N1C(=O)CC1CCC(=O)N1 N1(C(C(C)S)=O)Cc2c([nH][nH]c2=NC(=O)c2c(Cl)ccnc2Cl)C1(C)C C(C(=O)N1CC(NC(c2cnco2)=O)C(C)C1)(C(F)(F)F)OC(C)=O c1(OC)cc2nc(C)sc2cc1OCC(=O)N(c1ccccc1)C c1(CN(c2c(C)scc2)C=O)c(OC(F)F)cccc1Cl c1(CNC(C(CC)N(C)C)=O)ccc(CNC(c2cncn(C)c2=O)=O)c(F)c1 C12(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCOCC1CN(C(=O)C=CCF)C2 CC1CCCC1(C)C(=O)NCC1CC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 C=CCC(C(=O)N(C(C)CNC(c1c(F)ccc(OC)c1F)=O)C)C(C)C c1(C(=O)NC)ccc(O)c(NC(C2CCCCC(=O)C2)=O)c1 C(=O)(C#CC(C)C)NCC1CC(NC(c2cc(C(=O)OCC)sc2)=O)C1 CC(=O)C(C)(C)CC(=O)N1CC2COCC2(C(N2CCOC(CC(N)=O)C2)=O)C1 C1(C(=O)Nc2sccc2CO)CC2(C(N3CCC(CCCO)CC3)=O)COC1C2 Cc1ccc(CC(=O)NCC(O)CNC(C2(C)COCCO2)=O)c(Cl)c1 Cc1cc(CNC(c2occc2CNC(C2(O)CCOC2)=O)=O)nnc1C C1(NC(=O)C#CC2CC2)C2CC3C(C2)C13C(=O)NCC1CC2(CC2)C(=O)O1 c1(C(N(C(CCNC(c2cc(CC)no2)=O)C)C)=O)cc(N(C)C)ccc1F C1(NC(CS(N)(=O)=O)=O)C2CCCC1CC(NC(c1cc(=O)cc(Cl)[nH]1)=O)C2 C1(C2N(C(=O)C(F)C3CCCC3)CCC2)CCN(C(C23CC(C2)C3)=O)CC1 CC1CCC(C(=O)NC(C2CCN(C(=O)C(CO)N(C)C)CC2)C)CC1 N1(C(c2cc(Br)c[nH]2)=O)CC2CN(C(c3cc(F)nc(F)c3)=O)C2C1 CON1CCC(C(=O)NC2(CC(=O)NCC3CCSC3)CC2)CC1 Cc1nc(C=CC(N2CC(NC(C3(C#N)CC3(C)C)=O)C(C)C2)=O)[nH]c1C N1(C(C(CC=C)OC)=O)CC2CC(C(=O)NC3CCCC3(C)N(C)C)(C2)C1 N1(C(C2CC(SC)C2)=O)CCC2CN(C(=O)CCCc3ccncc3)CCC12 C=C(Cl)CC(C(=O)NC(Cc1ccco1)CO)NC(c1cnc2n1CCC2)=O C1(CNC(c2c[nH]c(=NC)o2)=O)CCN(C(C2CC(OC)C2)=O)C1(C)C N1(C(C=C(CCN(C)C)Cl)=O)CCN(C(=O)C=CC2CCCN2C)CC1CF c1(CC)ccc(C(=O)NCC(CC)N(C(=O)Cc2ccnn2C)C)s1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2ccc(F)cc2C)C1 c1(CNC(C(=O)Nc2c(C)nn(C)c2)=O)ccc(Br)cc1I C(=O)(C1=NOC(CNC(=O)CC2CCCSC2)C1)NCCn1ncc(C)c1 c1(CC)nc(C)oc1C(=O)NCCOCCC(=O)N(C)Cc1occc1C CC(CC(C)(C)C)C(=O)NC1CN(C(c2csc(O)n2)=O)CC1C(F)F C(C1=NOC2CCCC12)NC(C1(C)CCCN(C(c2cc(Cl)cs2)=O)C1)=O C1(NC(C(=O)N(C)C)=O)CCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(C(=O)NC(C2CCCN2C(c2cc(N)ccc2Cl)=O)C)nccc(Cl)c1F c1(CC)cccnc1C(=O)NCC1CCCCN1C(=O)C=Cc1cn(C)nn1 c1(C(N2C3CC(NC(C4CC45CCC5)=O)CC2CC3)=O)c[nH]c2nc(F)ccc12 C#Cc1ccc(NC(C2CC(F)CN(C(=O)COC3CCCCCC3)C2)=O)cc1 C1(CC)C(=O)N(C)CCN1C(C1C(CNC(=O)CCOC2CC2)C1(C)C)=O Cn1ccc2c(C(F)(F)C(=O)NCC3CCCCS3(=O)=O)ncnc12 C1(CNC(CCCCC=CC)=O)CCC2CN(C(=O)Cc3ccn(C)c3)CC12 c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C2)ccc2nnc(O)n2c1 N1(C(C(C)CF)=O)CCC(CO)(CNC(=O)C(C)COc2ccccc2)CC1 c1(CCCC)ncc(C(N2CC(NC(C3(C(=O)NC4CC4)CC3)=O)C2)=O)s1 CN1C(=O)CCCC1C(=O)N(c1ccns1)C CC1CC2(CC(C(N3CC4CC(NC(=O)Cc5cocn5)C3C4)=O)C2)C1 N1(C(C(COC)C(F)(F)F)=O)CCc2sccc2C1CNC(=O)CCC(N)=O CCCCCCC(C(=O)NC1CC(NC(C2CNC(=O)C2)=O)C(O)C1)NC(C)=O C#CCCCCCC(=O)NC1(C)CCN(C(=O)CSc2cc(C)ccc2C)C1 c1(CC)cc(Cl)ccc1C(N1CCC(NC(C2CCN2CC)=O)C1(C)C)=O n1(C(C)C)ccc(C(=O)NC(C)(C)CNC(=O)CCCC2CCOCC2)n1 CN1C(=O)CCC1C(=O)NC1CN(C(c2cnc(N)cn2)=O)CC1O c1(-n2cc(-c3cn(C)nc3)nn2)cncc(C(N2CCC(CCO)C2)=O)c1 Cn1cnc2cccc(C(=O)NCC(O)CNC(c3cn(CCF)nn3)=O)c12 C1(C(N2C(CC)CC(C)C2)=O)(CC)CCCN(C(=O)Cn2ncn(C)c2=O)C1 CC(C)CC(CNC(=O)CCCC1CCCO1)C(=O)NCC1CCCC(C)O1 N1(C(C2C(C)CC2)=O)CCCC12CCN(C(c1cc3cccc(Br)c3o1)=O)C2 CCC(C)CCC(=O)N(C1CC2CC1N(C(=O)Cc1cc(Cl)n(C)n1)C2)C C#Cc1ccc(NC(=O)NCC2(NS(=O)(=O)C3CCOCC3)CC2)nc1C C1(NC(C(CCC)NC(N)=O)=O)CC2CC(NC(=O)CCCSC)C2C1 C1(C(=O)NCC2CC(NC(=O)Cc3nnc(C)o3)C2)(OC)CCCSC1 C12(CC(=O)NCCc3c(C)n[nH]c3)CCC1CN(C(=O)C(F)C(C)(C)O)C2 c1(C(=O)NC(CCCC)CNC(c2ccnn2COC)=O)cccc2c1COC2 c1(COC(C2(Cl)C(C(=O)OC(C)(C)C)C2)=O)cnoc1-c1ccccc1 C1(NC(CCSCCC)=O)CN(C(c2c[nH]cc2CC)=O)CCC12CCC2 C1(OCCNC(CCC=CCC=C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 C(=O)(CC(C)CC(=O)NC1CN(C(=O)C#CC(=O)N(C)C)CC12CC2)OC C1(C(=O)NC(CCCC)C)CC2(CNC2)CO1 Cc1nn(-c2ccccc2)c(NC(N2CCCC2C(O)C(F)F)=O)c1Br C(C(C)(C(C)C)NCC)NC(CC1CC(OC(=O)CP(C)(C)=O)C1)=O N1(C(C2C(C(N)=O)CC2)=O)CC=CC1C(=O)NCCF c1(C(N2CCC(C)N(C(C3CCCS3)=O)CC2)=O)c2c(nn1C)CCCC2 C1(C)(C(=O)NC(C)CNC(=O)CCCc2n[nH]c(=N)s2)CCCCC1(F)F C1(C(=O)NC(CCCNC(C(C=C=C)C)=O)(C)C)Cc2cc(Br)ccc2O1 N1(C(C)CNC(C2CNC(=O)C2)=O)CCN(C(c2ncncc2N)=O)CC1 N1(C(C2CN(S(C(C)C)(=O)=O)C2)=O)Cc2cccc(Cl)c2C1 c1(C(=O)NCCCOCCNC(CC=CC=C)=O)cnn(CC)c1C c1(C(C)C)nc(NCCSc2nccn2C)cc(N2CCC(C(C)O)C2)n1 c1(C(=O)NC2CC(CNC(C3(C)CC(=C)C3)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 C1(C(=O)NCc2nc(-c3ccco3)n[nH]2)CC2CCC(C1)C2(F)F N1(C(c2c(OC)cccc2)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CCC1 c1(NC(C(C)Cc2ccco2)=O)ccccc1SCCC(N)=O N1CCCNCC1.c1(-n2cc(C3(C)CC3(Cl)Cl)nn2)ccc(F)cc1 c1(C(C)CNC(=O)C(=O)NCC(C2CCCCC2)F)ccc(F)cc1 Cc1cc(C)n2nc(C)c(C(N3CCC3CNC(C3C(Cl)(Cl)C34CC4)=O)=O)c2n1 c1(NC(C2(CNC(c3ccc(Cl)nc3Cl)=O)CC2)=O)ccnc2ncnn12 c1(C2C(C(=O)NCC(CC)NC(c3n[nH]c(C)c3O)=O)C2)ccncc1Cl c1(C(=O)OC)cncc(S(=O)(=O)NCCc2ccc(Br)cc2F)c1 CCC(C)C(C)C(=O)NCCC1(C(=O)NC2CC(F)(F)C2)CCC1 C(=O)(CCN(OC)C(=O)C(CO)OC)N(C(CC)CC)C1CC1 C=C(C)C(C)(C)C(=O)NC1CCCCCC1C(=O)N(C)CCc1ncon1 N1(C(C(COC)NC(=O)CC2CCCC(=O)C2)=O)CCCC(C)(C)C1C c1(C(=O)NC2CC(C)N(C(=O)C(N)=O)C2)cc([N+](=O)[O-])c(F)cc1N C1(NC(C(C)OCC=C)=O)CN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CC1F C1(NC(C2OC3CCC2C3)=O)CCC(NC(C2C(Cl)(Cl)C23CC3)=O)CC1 c1(OC)ccc(C(C)C(=O)NCCNC(=O)C(c2cnn(C)c2C(F)F)C)cc1 N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(C(c2ccc(F)o2)=O)CC1C Cc1nnc2n1C(C(=O)NCC(C1CC1)NC(c1ccn3cncc3c1)=O)CC2 n1(CC)nc(C(=O)NCC2C3CC3CN2C(C2CC2F)=O)ccc1=O C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)CC(C)C)CC(C)(C)C1 N1(C(C(c2n(C)ncc2)O)=O)CCCN(C(C2(C(=O)N(C)C)CC2)=O)CCC1 C=CC1(CNC(=O)C(CC2CCC2)NC(=O)CC(C)n2cccn2)CCC1 Cc1cc(NC(=O)CC23CCC2CN(C(=O)C(O)c2ccsc2)C3)cnc1C C1(CC)(CC)CN(C(=O)CC(C2CC2)NC(=O)CC2CCC(O)C2)CCO1 c1(C(N2C(C(=O)NCCOc3cccnc3)CC(OC)C2)=O)ccc(O)cc1Cl C(=O)(C(C)(C)CC(C)(C)C)NCC(C)NC(CCOC(C)C)=O CN=c1nc(N(C)C(=O)N)cc(C)[nH]1.N1(CCC2ON=C(C)C2)CCC(C)(C)C1 C=Cc1cnn(C)c1C(=O)NCC=CCNC(=O)Cc1cnn(C)c1 N1(C(c2cc(OCC)no2)=O)CCC(C)(CNC(=O)CCNc2ccccn2)C1 C1(NC(CCc2onc(CSC)n2)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C c1(OC)ccnc(C(N2CCC(NC(C3CN(C(C)=O)C3)=O)CC2C)=O)c1OC C12(C(N3CCCN(C(CC4OCC(C)OC4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 Cc1ncc(Cl)cc1NC(C1OCCC1NC(=O)CC1CCC(C)(C)C1)=O Oc1c(CN2CCC(c3nn[nH]n3)C2)cccc1Cl C#CC1CCC(NC(c2ccc(CNC(C3CCC(N(C)C)C3)=O)nc2)=O)C1 C1(C(N2CCC(CCNC(C=C3CCN(C)C3)=O)C2)=O)CC(=O)OC1(C)C c1(OC)cc2nn[nH]c2cc1C(=O)NCC1CC(NC(=O)CC2(O)CCOC2)C1 Cc1nc2c(CCC(N3CC(NC(C4CCSC4)=O)CC3(C)C)=O)cccc2o1 Cc1c[nH]c(C(=O)NC(C)CCC(=O)NCCC(O)C(C)C)c1C c1(OC)c(C)cc(NC(=O)CC2(O)CCN(C(c3ccc(C)o3)=O)CC2)cc1C N1(C(c2n(CC)ccc2)=O)CC2(CCC2NC(c2ccc(OC(F)F)cc2)=O)C1 CC1(F)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(F)Cl)=O)C1 c1(C(=O)NC2CC(C)CN(C(C3C(C)(C)C3(F)F)=O)C2)ccc2ncnn2c1 N=c1ncc(C(N2CCOC(Cn3cc(CNC4CCOC4)nn3)C2)=O)c[nH]1 C1(O)(C(=O)NC23CN(C(C(C)(C4CC4)NC(C)=O)=O)C(C2)C3)Cc2ccccc2C1 Cc1cc(NC(C2CCOC(=O)CC2)=O)ccc1NC(C1(S(C)(=O)=O)CC1)=O n1(CC(N2CCN(Cc3c(O)cccc3O)C3CC23)=O)ccc2c(F)cccc12 c1(CC(=O)NCC(n2ccnn2)C)cc(=O)cc[nH]1 Cc1ccnc(C(=O)NCC2(O)CCN(C(=O)CN3CCCNC3=O)C2)c1O C1(NC(c2c(CC)scn2)=O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC(C)(C)C1 CC1C(NC(c2snnc2C2CC2)=O)CCCN1C(c1cc(C2CC2)on1)=O C(CN=C(NCc1ccc(C#N)cn1)NCC1(C)CCCOC1)SC Cc1sc(C(=O)N(C2CCCC2)CC(=O)NCCSc2cccc(Cl)c2)c(C)c1C CCCN=c1[nH]c(=NC2CCCCN(Cc3ccccc3)C2)c2sccc2[nH]1 C1(C(=O)NC2C(NC(c3n[nH]c(CC)c3C)=O)CC2)CC2OC1C1CC21 N1(C(C(=O)N(C)C)=O)CC2CCCC(N(C)C(c3cnc4sccn34)=O)C2C1 c1(C(=O)NC2(C)CC(NC(C3COCC(C)O3)=O)C2)ccc2nccnc2n1 Cc1nc(CNC(=O)C(CNC(=O)CC23CCCC2C3)N(C)C)sc1C CC(C)(CC#N)C(=O)N1CCC(NC(c2sccc2OC(F)F)=O)C(O)C1 c1(C(=O)NCC(C2CC2)NC(C(C)(C)OCC)=O)cc2c(F)ccc(F)c2s1 n1(CC(=O)NCC2N(C(Cc3nc(CC)on3)=O)CCC2)ccc2ccccc12 CC1CC(C(=O)NCC2CN(C(=O)CCCc3ccccc3N)CCN2C)=NO1 N1(C(c2c(C)nns2)=O)CCCC2(CCN2C(C2CCCSC2)=O)C1 C(=O)(C(F)C(F)(F)F)NCCCOCCNC(Cc1c(CC)cccc1)=O CCCCCC(O)C(=O)NCc1ncccc1C(=O)N(CCC(N)=O)C N1(CCC)CCCC1C(=O)NC(C)CCNC(c1cnoc1C1CC1)=O C(C(C)CC(=O)NCCCC(C)NC(=O)C(C)SCc1ccccc1)OC C1(C(N2CC(F)(F)CC2CNC(C2CC(CF)C2)=O)=O)CCOC2(CCCC2)C1 CC(C)CS(=O)(=O)CCC(=O)NCCCN(C(=O)CCc1cscn1)CCO N1(C(COC(C)=O)=O)CC2C(NC(c3ccc(CO)cc3)=O)C2C1 c1(OCC(=O)NCC(CC)NC(=O)C(C)(C)C2CC2)ccccc1C Cn1ncc2c(=O)n(C(=O)c3cnn(Cc4cccnc4Cl)c3)c(C#N)nc12 N1(CC(C)(C)CCCc2ccccc2)CC2CCC(O)CC2C1 c1(CNC2C(C(=O)ON)CCCC2)cc(C)ccc1OC1CCC1 c1(C(=O)NCc2ccsc2)n[nH]c2c1CN(C(=O)CN1CC=CC1)C2 O=S(=O)(c1ccc(NC(c2ccccc2)CO)c(Cl)c1)N1CCC=C(F)C1 CC(C(=O)NCc1cscn1)NC(=O)C(C)C1CCCC1 C1(C(=O)NCCC2OCCN(C(c3c[nH]c(=NC)o3)=O)C2)CC(C)(C)OC1(C)C C12(C(=O)NC(c3nc(C(F)(F)F)cs3)CC)CCCCC1C2Br C1(NC(C2(OC)CC2)=O)CCCC2CN(C(c3cnsc3C)=O)CC12 CCCCC(C)C(=O)N1CC(CNC(=O)CCC2(NC(=O)OC(C)(C)C)CC2)C1 N1(C(C(N(C)O)=O)=O)CCC(O)(CNC(=O)NC)CC1 C1(C(C)NC(C2CCCO2)=O)CCCN(CC(=O)Nc2ccccc2)C1 c1(CC)cc(C(=O)NCC2(O)CC(NC(=O)CC3CC=CC3)C2)c(C)nn1 c1(C(=O)NCCCCN(C(=O)CCn2cc(Cl)cn2)C)csc2nccn12 CC(C)(C#N)CC(=O)N1CC(NC(C2CCC(=O)N2)=O)C(O)C1 c1(CNC(C(=O)NCC(CNC(C=C(C)C(C)C)=O)C)=O)ccc(F)cc1 N1(C(c2n(CC(=O)OC)cnc2C)=O)CCCC(F)(CNC(c2cnn[nH]2)=O)C1 c1(CN(C(CCCOC)=O)C)cnn2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(CCCCC(=O)N(CCNC(=O)C2CC2)CCOC)nc2ccccc2s1 CC1(C(=O)NC2CCCN(C(C34CC3CCC4(F)F)=O)C2)COC(=O)OC1 Cc1cn2c(C=CC(=O)NCc3cnc(C#N)cn3)c(C)nc2s1 C=C(C)CC(C(=O)N1CCN(C)C(CNC(=O)C(O)CCSC)C1)OC CCC(CC(=O)NCC(c1ccc(F)cc1)NC(C12CC(F)(C1)C2)=O)C(C)(C)C C1(CC(N2CC(CSC)C2)=O)CC(F)CN1C(C1CC12CC2)=O c1(C(=O)NC2CC(O)(CNC(c3cc(CC)sn3)=O)C2)n[nH]c2c1CSCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)(C)C)NC(c1cnc(O)n(C)c1=O)=O c1(C(N2CCC(OCC(=O)OC)C2)=O)cc(C#N)[nH]c1C C#Cc1cc(NC(=O)C#CCNC(C2CCC(=O)N2)=O)ccc1C C(=O)(C(CN=[N+]=[N-])NC(C1CC2(C1)CC2(F)F)=O)N(C1CCN(C)CC1)C N1(Cc2ccn(C(C)C(=O)O)n2)CCC(c2nn[nH]n2)CC12CC2 c1(CN2CCCC(C(=O)Nc3c(OC)nnc(Cl)c3)C2)cc(C)c(Cl)c(C)c1 C(CN=c1[nH]ccc(=NC2CC2c2ccc(Br)cc2)[nH]1)N1CC=C(C)CC1 N1(C(C2(NC(C3C(C)C3)=O)CC(O)C2)=O)CCCCCC1 c1(C(N(C(C)C(N2CCC(C#N)C2)=O)CCC)=O)ccc(C)cc1 N1(C(C(C)OCC#C)=O)CCCC2(CNC(C3CC(C)=NO3)=O)CCCC12 Nc1cccc(C(=O)CCC(=O)NC2CC2NC(C23CCCC2C3)=O)c1 c1(C(N2C(CC)C(NC(c3cnncc3O)=O)CC2)=O)ccc(Cl)cc1O C=CCC(CNC(=O)COCC(C)C)NC(=O)C#CCN(C)C N1(C(CN(C(=O)OCC)C)=O)CCCC(CCC(=O)NCC(O)CC)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C2CC(CC)OCC2)=O)C2(C1)CC2 C1(C(=O)NC2C3(CN(C(c4cc(=NC)[nH]cc4)=O)C3)CC2)CC2(C1)CC(C)(C)C2 N1(C(C(CC)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)CC(C)(C)C1 C1(C(=O)OC)(NC(C2CC(N(C)C)C2)=O)CCN(C(=O)C(C)Cc2ccco2)C1 c1(OC)ccc(C(N2CCC(CNC(=O)CC(F)F)C2)=O)c(Br)c1F N1(C(C(c2ccccc2)C)=O)CC2CC(C1)CN(C(c1ocnc1C1CC1)=O)C2 c1(C(COC)(C)NCCN(CCOC)CC(C)C)nnnn1C1CC1 C1(C(=O)NC(C2CCCC2)C#C)CCCCC1(C)NC(=O)CC1(O)CCOCC1 CN1CCC(C)(C(=O)NCC23CC2CN(C(=O)CC2CSCCO2)C3)CC1 c1(OC)cc(C(C)OC)nc(-n2nc(-c3ccccn3)nc2C2CCCSC2)n1 C=CC(CC)C(=O)NC(CO)C(C)NC(c1cnn(CC)c1CC)=O N1(C(C2C(COC)C2)=O)C(C)CC2CN(C(=O)CCC3CCC3)CC12 c1(N(C)CC2CC2)ccn2ncc(S(=O)(=O)NC3(C)CCOC3C3CC3)c2n1 c1(C(N2CCCC(N(C(=O)CCC3(C)CC3)CC)C2)=O)c(F)ccc(C#N)c1F c1(C(N2CC(C)(NC(c3cc(COC)oc3C)=O)C2)=O)cccn2nnnc12 C1(F)(CNC(C(c2ccc(F)cc2)OC)=O)CCN(C(=O)CC2CCC(=O)N2)C1 C(CNC(c1cccc(COC)c1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O c1(CN2CC(N(C3C(C(=O)OC(C)(C)C)C3C)C(C)=O)C2)ccn(C(F)(F)F)n1 c1(OCC)ccc(C)nc1C(N1CCOCC(NC(C)=O)C1)=O Cc1cc(F)c(CC(N2CCC3(C2)CN(C(=O)CC2(O)CCCOC2)C3)=O)cc1F O=C(CCCCCCNC(c1ocnc1C1CC1)=O)NCCC(F)F C1(NC(c2ccnn2CCF)=O)CCCCC1CNC(C1CCCO1)=O CC1(C)C(NC(=O)Cc2ccc(F)cc2F)CCN1C(C1COC(=O)O1)=O C1(CNC(CC=C=C)=O)CCN(C(=O)CNC(C2CCCCC2)=O)CC1C Cc1nc(F)ccc1-c1cn(CC2CCN(C(C3C=CCC3)=O)C2)nn1 Cc1nn(C)c(N)c1C(=O)Nc1c(C)nn(CC(C)C)c1C N1(C(Cc2ccc(CC)cc2)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)C(C)C1 c1(OC)cc(C(=O)NCC2COCCN2C(c2ccsc2)=O)cc(C2CC2)c1 C1(NC(CC(CC)C)=O)CC2CC(NC(c3cc(CO)[nH]n3)=O)C1C2 CN1CCC2(CCN)CCCC12 C1(CCNC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(NC(CSCCCC)=O)C(C)CN(C(c2occc2CC)=O)CC1C C1(C2CCCN(C(=O)C=C(C)Cl)C2)(NC(CC2C(C)=NN(C)C2=O)=O)CC1 Cc1nn(C)c2cc(NC(=O)CC3CCC(C)C3)ccc12 C(c1nnn(C)n1)=CC(=O)NC1(C2CCN(C(C(N3CCOCC3)C)=O)C2)CC1 N1(C(C2CCOCC2)=O)CCN(C(C23CC(O)C2C3)=O)CC1CO N1(C(C2C(CC)C2)=O)CCOC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC12 C=CCC(C(=O)N1CCC(C(C)(C)C(=O)Nc2ccc(OC)nc2)C1)NC(C)=O N1(C(C(F)=C(C)C)=O)C(C(F)(F)F)CC2CCCCC12 c1(OC(C)(C)C)ccc(C(N2CC(NC(=O)C=C3CCCCC3)C3CC23)=O)cc1 C12(NC(CCOCC)=O)CC(C)(C1)OC21CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC12CC(NC(=O)CO)(C1)C2 c1(C(N2CCN(C(C(C=C=C)C)=O)C(CC)C2)=O)nnn2ccccc12 c1(NC(C2CCCC(NC(C3(Br)CCC3)=O)C2)=O)cccc(F)c1Br c1(CNC(c2nc(CNC(C=C(C)C(C)C)=O)oc2C)=O)cncc(C#N)c1 N#Cc1ccc(Cl)c(C(N2CCC3(CNC(c4cscn4)=O)CCCC23)=O)c1 CC(C)C(C)(CNC(=O)CCCN1C(=O)CNC1=O)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)F)NC(C)CC1CCCC(NC(c2cn(C)c(=O)cn2)=O)C1 N1(C(C(C2CN(C(C3(OC)CCOCC3)=O)C2)O)=O)CCCC(N=[N+]=[N-])CC1 C1(C(=O)OC2CC(c3ccccc3)C2)CCC2(C1)CC2(F)F c1(C(N2CC3CN(Cc4cnc(SC)nc4)C3C2)=O)ccc2c(c1)CCO2 C(=O)(C(F)(F)F)NCC(=O)N(C1CCN(C(=O)C(O)c2ccco2)C1)C Cc1ncnc(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)F)C2)c1C Cc1cccc2[nH]cc(CC(=O)NC3CCCN(C(c4coc(C#N)c4)=O)C3)c12 C=CCCCC(=O)NCC12CC(CN1C(=O)C=CSCc1ccco1)C2 Cc1cc(C(=O)NC(C)CCN(C(=O)CNC(=O)CCC(C)C)C)c(O)nc1C c1(NC(c2cccc(O)n2)=O)ccc(NC(c2ccc(O)cc2O)=O)c(F)c1 c1(OC)ccc(Cl)cc1CC(=O)NCCOC(C)(C)CNC(=O)CCCN(C)C C(=O)(C(CC)CCC)N1CCC(C)(NC(COCCCCOCC#C)=O)C1 C1(C(=O)NCc2ccc(C)o2)CC2C=CC1N(C(=O)CC1CCC(=O)C1C)C2 c1(C(C)C)cccc(C(=O)NCCOCCCNC(c2ccc(F)s2)=O)n1 N1(C(COC)=O)CC2(CCN2C(=O)CCc2ncccc2C)C1 C(=O)(CCCN=[N+]=[N-])NC(C(C)NC(C1N(C(C)=O)CCC1)=O)CO N1(C(C2C(C)(C)C2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccc(F)cc1 N1(C(Cc2nc(CC)sc2)=O)CCCC(C2CC2NC(c2cnsc2)=O)C1 C1(CC(=O)NC(CNC(=O)CC23CCC(CC2)OC3)C2CC2)CC2(CCC2)CO1 c1(CC)cc(C)nc(NC2CC(F)(CNC(=O)C=C(C)C(C)C)C2)n1 N1(C(C2(C)CC=CC2)=O)CCCC(CO)(NC(c2ccnc(O)c2)=O)C1 c1(C(=O)NC(CCNC(C=C(C)C(C)C)=O)(C)C)ccc2cnoc2c1 c1(C(N(C)CC2(NC(Cc3cncc(C)c3)=O)CC2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)CC1CNC(C1(CCO)CC1)=O c1(CC)cccc(Cn2cc(CCCNC(c3ccc(C)cc3F)=O)nn2)c1C C1(CC#C)(C(=O)NCCC(O)CO)CC=CCC1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(=O)C=Cc2cn(C)cn2)CC12CCCC2 C1(C(C(=O)NCC)C)CCN(C(c2ccc[n+]([O-])c2)=O)CC1 c1(OC)ccccc1OC1CN(C(=O)CC2(N)CCSC2)C1 N1(C(C(C)NC(C)=O)=O)CCC(CNC(=O)COc2ccc(C)cc2C)C12CC2 Cc1ccc(CNC(=NC(C)C)NC2CC(=O)N(C(C)(C)C)C2)c(=O)n1C C1(C(C)C)CCC(C)CC1CNC(=O)C1=NOCC1 C(=O)(C1=CC2CCCCCC12)N(C)CC1COCCN1C(C1CCCS1)=O C(=O)(CC(C)C(F)(F)F)NC1C(CNC(c2c(-c3ccc(C)o3)onc2)=O)CC1 c1(C(C)C)cnc(CNC(=O)NC23CSC(C2)C3)o1 CS(=O)(=O)c1ccc(C(=O)NC2(C3CCNC3)CC2)s1 C1(NC(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(C)c2ccon2)CC1 N1(CC(=O)NCCCOCCC(=O)NC2(CCCC)CC2)CCC(OCC)C1 CN1CC(C)(C(=O)NC2CCN(C(=O)CC3CNC(=O)O3)CC2)CC1=O c1(OC)cc(C)cnc1C(N1CC(CNC(C2CN(C(N)=O)C2)=O)C(C)(C)C1)=O C1(NC(C=C(CC)CC)=O)CN(C(C2CC2(COC)COC)=O)CC1C c1(C(N(CC(CNC(CCc2cc(C)on2)=O)O)C)=O)cccn2ccnc12 N1(C(c2cc(CC)no2)=O)CCC2(CCCCC2NC(=O)CCCN(C)N=O)C1 N1(C(CNC(CCCC)=O)=O)CCN(C(c2cnc(C3CC3)s2)=O)C(CCC)C1 c1(CCNCc2ccc(-n3c(C)cc(C)n3)nc2)cccc(F)c1F c1(C(N(CCCNC(c2cnccc2Cl)=O)CC)=O)cn2ncnc2nc1C C1(c2cn(CCNC(C(C)C)=O)nn2)COCCN1C(c1ncn(C)n1)=O C(=O)(C1=CC2CCC=CCCC12)N1CC(CCNC(c2ocnc2C)=O)(OC)C1 N1(C(CNC(=O)OCC)=O)CCC(F)C(NC(=O)C(C)(C)N2CCCC2)C1 C1(NC(C2CCCC(CF)C2)=O)CCCC2CN(C(=O)C=C3CCCC3)CC12 c1(C(N2CCCC(CNC(C3ON=C(C)C3)=O)CC2)=O)cc(C)cc(C)c1C CC1CN(C(=O)CC2CCCN(C)C2)CC1NC(c1cc(CCCO)on1)=O C12(C(=O)NCC(C)(C)F)CC(CO1)N(C(C1CCC=CCCC1)=O)C2 C=CCC(CC(F)F)C(=O)N(C)CC1(O)CCCN(C(=O)CCC(C)CC)C1 N1(C(C2(C#N)CC3CC3C2)=O)CC(NC(c2cnc(Cl)s2)=O)CC(F)(F)C1 Nc1ccc(S(=O)(=O)NCCC(=O)NCC2CCN2C2CC2)cc1 N1(C(C(CC)(C)F)=O)CC(NC(=O)CCn2cccn2)CC(F)C1 C1(C(N2CCCC(C(C)NC(CCC)=O)C2)=O)CCC(C2CCC2)CC1 c1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCCCC)ccc(COCC)cc1Br C(c1cn[nH]c1)=C(C)C(N1CCCC1C1(C(=O)NOCCCN(C)C)CC1)=O CC1Cc2cccc(O)c2N(CC2(C#N)CCCCC2)C1 CC1CC=C(C(=O)NC2CC3CC2N(C(=O)CCc2cnn(C)n2)C3)CC1 C1(CNC(CCS(C)=O)=O)CCN(C(=O)CSCc2ccc(F)cc2)C12CC2 C1(CC(=O)NC(C2CSC2)C)CCN(C(C2CC3C(C2)C3(F)F)=O)C1(C)C n1(CC)ncc(Cl)c1C(=O)NC(C)CC1CN(C(=O)C=C2CCOCC2)C1 C1(C(N2CC[Si](C)(C)C2)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 Cc1noc(Cl)c1CC(=O)NC1CCCC(CNC(=O)CCc2cncs2)C1 CCCC(CCNC(C1OCCC1CNC(c1occc1C(C)C)=O)=O)CCC N1(C(C(=O)NC(CCCCC)C(C)(C)C)=O)CCSC2(CCCCC2)C1 CC1CCOC(C(N2CCC(NC(c3ccc(C(F)(F)CF)cc3)=O)C2)=O)C1 C1(Nc2cc(N3CCC(C=C)C3)nc(C)n2)CCc2nn[nH]c2C1 c1(C(N2CCC(C)(CNC(c3cccc(F)c3F)=O)C2)=O)nsc2ccccc12 CC(C)(C(=O)N(CC(S(C)(=O)=O)C1CC1)C(C)(C)C)C(=O)N1CCCC1 Cc1c(Cl)ccc2[nH]c(C(N3CCCN(C(C4CCOC4)=O)C(C)C3)=O)cc12 O=[N+]([O-])c1ccc(F)c(Br)c1S(=O)(=O)N=S1(=O)CCC(C2CN(C(CCCl)=O)C2)CC1 N1(C(CC=CC=C)=O)C2CCC1CC(CNC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(C)NC(=O)NC(c2ccc(O)cc2)(C)C)cccc(O)n1 c1(N2C3CS(=O)C(C3)C2)nc2ccccc2c(=NCc2cccc3nc[nH]c23)[nH]1 C(=O)(C1CCC(=O)c2ccccc21)N(CCC(C)NC(Cc1scc(C)n1)=O)C CC(CC(=O)NCCCCC(=O)N1CC(C)C(O)C1)C(F)F c1(CC(=O)NC2CN(C(CSC)=O)CC2n2ccnn2)cncc(C#N)c1 CCC(F)(F)C(=O)NCC1(O)CC(NC(c2ccnc(NC(C)C)c2)=O)C1 Cc1cc(N(C(C)CNC(=O)C(C)C(C)S(C)(=O)=O)C)n2ncnc2n1 CCCCC(C(=O)N1CCC(F)(CNC(c2c(C)noc2CC)=O)CC1)C(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)OC2)Nc1c(C(=O)OC)c(F)ccc1 c1(CN2CC3C(C(=O)NCCN4CCCCCC4=O)C3C2)cnc2ccccn12 C1(CCNC(Cc2nc(C)sc2)=O)COCCN1C(=O)CC1C=CCC1 N1(C(C=CCCC)=O)C2CCC1C(NC(c1sc(Cl)c(Cl)c1C)=O)C2 C=CC(C)(CCOC)C(=O)NC1CCCN(C(c2cc3cscc3s2)=O)C1C CCCCC(C)C(=O)NCC1(CN(C(=O)CC2CCCC2O)C)CC1 c1(N2C(C(N3CCC(CCNC(COC)=O)C3)=O)CCC2)ccc(Cl)cc1 c1(-c2cccc(C(=O)OC)c2)ccc2c(c1)OCCN2C(=O)N(C(C)C(N)=O)C Cc1ccc(C(=O)NC2COCCN(C(c3cn(C)nc3C)=O)C2)c(I)c1 O=C(C1CCCCCc2ccccc21)NC12CC(NC(=O)C3=CCSC3)(C1)C2 Nc1cccnc1C(=O)NCC(c1ccccc1)CNC(=O)CNC=O c1(C(=O)NC2CCN(C(CC(=O)OC)=O)CC2OC)ccc2ncc(Br)cc2c1 CC1CCN(C(C2COC(C)C2)=O)CC1NC(=O)CNC(c1ccc(N)cc1)=O CCC(C(=O)NCCCCN(C)C(c1cn(C)[nH]c1=N)=O)C(C)(F)F N1(C(=O)C#CC2CC2)CC2(CNC(C3(CCN4CCCCC4)CC3)=O)CC1CO2 N1(c2ccnc(CC)n2)CCn2ncc(CN(C(=O)CCC(C)OC)C)c2C1 Cc1cnn(C(C)C(=O)NC(C)Cn2cc(COCP(C)(C)=O)nn2)c1 c1(C(N2CCOCC(NC(C(C)O)=O)C2)=O)c2c(nn1C)CCSC2 N1(C(C(C#C)(C)C)=O)CCC2(NC(=O)CC(COC)Cc3ccccc3)CC2C1 C(=O)(C(CC1CCC1)NC(=O)CC(C)F)NC(c1cnn[nH]1)C c1(C(N(CCNC(c2nc(CCC)sc2)=O)CC)=O)cnc2c(cnn2CC)c1 c1(NC(C2CC(C)(NC(=O)CCc3ccc(O)c(O)c3)C2)=O)ccc(C#N)nc1 C1(O)(CNC(C(Cc2cn(C3CCCC3)nn2)NC(=O)OC)=O)CCCN(C)C1 c1(C(=O)NCC2(C)CC(NC(c3c(OC)ccs3)=O)C2)cccc(C2CC2)n1 C1(C(=O)NC(CCOC)C)(NC(=O)CCC(N)=O)CCC(C)(C)C1 N1(Cc2n(C)c(C(=O)O)cn2)CCC(F)(c2ccccn2)CC1.c12ccc(cc1)[nH]2 N1(C(C2(C=C)CCC2)=O)CCN(C(=O)CC2=CCCC2)C(CF)C1 C1(C(=O)NCC(=O)NCC(C)C)C2CCC(C2)C1NC(c1cc(Cl)cn1C)=O C1(C(=O)NCC(COC)OC)CCCCCCN1C(=O)C1=CCCCO1 C1(NC(C=Cc2nc(C)sc2)=O)C2CC1CN(C(c1nc(O)sc1C)=O)C2 c1(C(N2CCC(C)(NC(CCN(S(C)(=O)=O)C)=O)C2)=O)nc(Cl)ccc1N Cc1[nH]c(C(=O)NC2CC2(F)F)c(C)c1C(N1CCC(O)(CF)CC1)=O N1(C(c2c(CC)n(C)nc2)=O)C2CCC1CC(NC(C1CCN(CC)C1)=O)C2 C1(CNC(c2cccc(C(C)C)c2)=O)(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC(C)N(C(C(CC)O)=O)CC)cccc(-n2ccnc2O)c1 Cc1[nH]nc2c1CCC(C(N1CC(C)(NC(c3ccccc3Br)=O)C1)=O)C2 c1(C(=O)NC2(C(=O)NC(C3CC3)C3CC3)C(C)(C)C2)ccc(O)cc1F C1(C(=O)NCCCC=C)CC12CCN(C(=O)CSC(C)(C)C)CC2 Cc1nsc(C(=O)NC2CCN(C(=O)C(n3nccc3C)C)C2)c1Br N1(C(c2c(C)cco2)=O)CCN(C(c2cnn(C(C)C)c2N)=O)CC(C)(F)C1 c1(-c2n(C(C)C(=O)NS(C)(=O)=O)c(S)nn2)cncc(C(F)(F)F)c1 Cc1nc(C(=O)NC(C)C(=O)N(C2CC(C)C2)C)ccc1C#N c1(OC)cccc(S(=O)(=O)N2CCC23CN(c2cc(C#N)ncn2)C3)c1 c1(CN(C)C(C2(CNC(=O)COC3CCCOC3)CCCO2)=O)ccncn1 N1(C(c2c(C)scc2)=O)CC(NC(=O)CC2CCSCC2)C(O)C1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)C1 c1(OC)cncc(C(=O)NCc2ccsc2C(=O)NC2C(C)(C)C2(C)C)c1 Cc1ccc2occ(C(=O)NC3CCCN(C(=O)C#CC4CCCO4)CC3)c2c1 C1(NC(c2c(C)[nH]cc2)=O)CC(O)CN(C(=O)CCCc2ccc(F)cc2)C1 c1(Nc2n(C)nnc2CNC(=O)COCCCN(C)C)cccc2c1CCO2 CCCC(CCCNC(=O)C(C)Cc1ccco1)NC(=O)CS(=O)(=O)NC c1(C(=O)OC)cnn2cnc(NC(=O)C(N3CCC(C(=O)OC)C(CO)C3)=O)nc12 N1(C(CC(=O)OCC)=O)CC(C(=O)NC(CC)C(C)O)C(C2CC2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(F)CC1CNC(=O)CC(C)(C)N(C)C C1(CCC)CN(C(=O)C(C2CCCC2)OCC)CCN1C(=O)C1=CCCSC1 Cc1cc(=NCc2ccn(-c3ccc(F)cc3)n2)nc(-c2ccncc2)[nH]1 C(=O)(CCC(=O)NN(C)C)NCC(CC=C)NC(c1cc(CO)ccn1)=O C(CC(C(C)(C)C)NC(=O)C(C(=O)OC)OC)N(C(C(C#C)(C)C)=O)C CC1CCC(CNC(c2ccc(CO)cc2)=O)CN1C(c1n[nH]cc1Cl)=O C1(NC(c2n[nH]c3c2CCCC3)=O)CCCCN(C(c2ccoc2)=O)CC1 C1(C(N2CCN(C)CC2)=O)C2CCC(C2)C1NC(C1CC=CC(O)C1)=O N1(C(C(C)(C2CC2)OC)=O)CCN(C(c2csnn2)=O)C2(CCC2)C1 C#CCCCC(=O)N(C)Cc1ccc(CNC(C2C3CNC(=O)C23)=O)cc1 Cc1cc(=NC(=O)C(F)C2CCN(C(=O)C3CC3)C2)[nH]n1C CC1=NN(C)C(=O)C1CC(=O)N(C)CCN(C)C(c1ccnnc1S)=O C#CC1(C(N2CCOCC(O)C2)=O)CCN(C(=O)OC(C)(C)C)C1 CC1C(NC(C2CC3(CC3)CO2)=O)CCN1C(=O)C(O)C1CC1 c1(N2CCC(N(C(=O)C3=COCCC3)CCC)C2)nccc(S(C)(=O)=O)n1 C(=O)(CC(C)(C)CNC(c1c(F)cncc1F)=O)N(C(CC(C)C)C)C1CC1 c1(SC)cccc(C(=O)NC(CNC(=O)CC2CC23CC3)C(C)C)c1Cl C(=O)(C1=CCCCCC1)NCC1(C(C)NC(c2coc(Br)n2)=O)CC1 C1(CNC(=O)OC(C)(C)C)CCC2(CC(C(=O)Nc3cncc(Br)c3)C2)O1 c1(OCC(=O)NC2CN(C(c3ncn(C(C)C)n3)=O)C(C)C2)cccc(C#N)c1 C1(NC(c2n(CC)ncc2)=O)CC(CNC(=O)COCCF)C1(C)C C1(NC(CC2(COC)CCCC2)=O)CC2CCC1N(c1ncc(C)c(O)n1)C2 c1(C(=O)NC2C(NC(C(C)CO)=O)CCC2)cncc(C(F)(F)F)c1 C1(C(=O)NCC2CCCCN(c3nnc(CO)s3)C2)CCCCC12CCC2 c1(C(=O)NCCCCCN(C)C(C2CC23CCOC3)=O)cncc(N)n1 c1(C(=O)NC2(C)CCC(NC(C(COC)OC)=O)CC2)cncc(C)c1C S(=O)(=O)(C1CCCCC1)NC(C1CC(c2ccc(Br)cc2)(C)C1)=O C=CCC(C(=O)N1CCC(=CCNC(=O)C(O)CC(=O)OCC)CC1)C(C)C c1(NC(C2C(C(N3CCN(CC(=O)NC)CC3)=O)C2)=O)c(C)cc(Br)cc1Cl C1(CNC(=O)CC2CC3(CC3)C2)CC2(CCN(C(=O)Cc3cn[nH]c3)C2)CO1 O=C1NC(=O)C(CCNC(C2CCCN(C(c3ccnc(C(F)F)c3)=O)C2)=O)N1 CCCC(C(=O)NCC12CCC(CN(C(c3cnnc(C)c3)=O)C1)C2)C(C)C C1(NC(=O)CCNC(c2ccsc2)=O)CN(C(C2COC(=O)N2)=O)CC12CC2 Cc1nc(C2CC2(F)F)sc1C(N1CCC1CNC(C1OCCCO1)=O)=O N1(C(C(c2ccccc2)SC)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)C2(CC2)C1 c1(C(=O)NC(C2CC2C(=O)N(CC(C)(C)CN(C)C)C)C)cc(F)n(C)n1 CCC(C(=O)NCC1CN(C(=O)CCOC(C)C)CCN1C)C(C)(F)F C1(NC(C(c2ccc(F)cc2)(C)C)=O)CCCN(C(=O)Cc2ccon2)CC1 c1(C(C)=O)ccc(C(=O)N(C(C)C(=O)NC(c2nc(C)cs2)C)C)o1 c1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(C)n2cccc2)cc1F C1(NC(C(C#C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CCOCC1(C)C C1(CN(C(c2cnc(C)s2)=O)C)CN(C(=O)CCc2cc(C)n(C)n2)CCO1 C1(NC(=O)CC2=CCOCC2)CCC2(CCCN(C(=O)CCCC3CC3)C2)C1 c1(C(=O)Nc2cc(C3CCCN3)[nH]n2)cc(Br)c(Cl)s1 C1(C(N(C(CNC(c2cc(CC)oc2C)=O)C2CC2)C)=O)CC2CC2CC1C C1(C(=O)NCc2occ(C(N(CC(C)(C)C)CCC#C)=O)n2)CN(C)CCO1 c1(C(=O)NCC2(OC)CCN(C(c3ccoc3)=O)CC2)ccn2c(C)cnc2c1 N1(C(c2cccc(Br)c2F)C(=O)NCC=C)CC2(CCCC2)OCC1C C(c1ccc[nH]1)=CC(=O)NC12CC(CNC(c3occc3C3CC3)=O)(C1)C2 C=C(C)CCC(C)NC(=O)CC1(N(C(=O)C(C)COCC)C)CC1 N1(C(=O)C(O)C2CCC2)CCN(C(C2CCCCN2C(c2ccsc2)=O)=O)CC1 N(C(=NCCF)NC1CCN(Cc2ccco2)CC1)CC1N(C)CC1 C1(NC(CCC=C)=O)(CO)CCN(C(c2cn(CC3CCCO3)nn2)=O)CC1 CC(C(=O)NCC1CC2(CC(NC(C3(CF)CC4(CCC4)C3)=O)C2)C1)C(F)(F)F N1(C(C(=O)NCC)c2ccns2)CCCCC1CNC(c1ccccc1)=O c1(C(=O)NC(CNC(C(CCCC)=O)=O)CCCC)cc(S(=O)(=O)N(C)C)c[nH]1 C1(NC(C(=Cc2ccccn2)C)=O)CCC2(CC1)CC2NC(=O)COCC1CC1 C(=O)(C1CCc2ccccc21)NC1CC(NC(c2n[nH]c3c2CN(C)CC3)=O)C1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCN(C(C2CCC3CC23)=O)CC1CCOC C12(NC(CC3CC(SC)C3)=O)CC1CN(C(=O)Cc1sc(O)nc1O)C2 c1(CC(=O)N(C2CCN(C(C(C)C)=O)C2)C)ccc(Br)cc1[N+](=O)[O-] c1(CC)nc(C(=O)NC2CC2CNC(c2cc(F)cnc2O)=O)c2ccccn12 C1(C(N2CCC(Br)C2)=O)CCc2nc(-c3ccc4n[nH]cc4c3)sc2C1 N1(C(=O)CCC2CCC(O)CC2)CC2CCC(C1)N2C(=O)CC1CC1 c1(C(=O)NCC2CCN(C(C3CC3F)=O)CC2(F)F)ccc2ccnc(O)c2n1 c1(C(N2C(C(C)NC(C3CCSC3)=O)CCC2)=O)cc2ncccc2cc1Cl C1(NC(C(CCCC)C)=O)CN(C(=O)COCC(C)C)CC2CCCC12 c1(N2CCC(NCc3c(Cl)cccc3)C2)ncnc2sc(Br)cc12 c1(OC)cc(C(=O)NCC2(O)CCCN(C(c3c(C)nsc3C)=O)C2)cc(Cl)c1 CC1=C(C(=O)N2C3CCCC2CC(CNC(=O)C(O)C(C)C)C3)CCC(C)(C)C1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc2cnccc2[nH]1 Cc1cnc(F)c(C(N2CCC(C(C)NC(=O)C(C)(C)C3(O)CCOC3)C2)=O)c1 c1(OCC)ccnc(N2CC(C(C)NC(C3(Cl)CC3)=O)C2)n1 C1(N(C)C(C2CC2C2CC2)=O)CN(C(=O)CC2CCCCC2)CC1O CC1=C(C(=O)N2CCOCC2CCNC(=O)CSc2nccn2C)CCC1 C(=O)(C1=CSCCO1)N(CC(C)NC(c1c(C)nc(C(C)C)o1)=O)C C1(NC(CN(C2CCC2)C)=O)COCCC1C(=O)N(C)OCC(F)(F)F c1(OC)cc(-c2ccc(CC(=O)NCCCn3ccnc3C)c(F)c2)ccc1C N1(C(C(C)(C)c2cnco2)=O)CC2C3CCC(C2C1)N(C(C1CC=CCC1)=O)C3 N1(C(CC2CCC(OC)CC2)=O)CC2CCCC(N(C)C(C3CCCS3)=O)C2C1 N1(C(c2ncc(C)nc2)=O)CCC(C)(C)C(CNC(c2coc(N(C)C)n2)=O)C1 CC1=CC(C)CN(C(c2cnn(C(F)F)c2)C(=O)NCCC#N)C1 c1(CC(=O)NCCN(C(=O)C(C)C2(O)CCC2)CC)cccc2nonc12 c1(C(=O)NCC(C)NC(=O)CC(=O)NC2CC2)ccnc2c1nnn2C C1(CN(C(C(C)NC(=O)NC)=O)C)CCCCN1C(=O)CC1(O)CCC1 N1(C(C(CCC)O)=O)CC(C)C(Nc2cc(C(N)=O)nc(Cl)n2)C(C)C1 c1(C(N2CCCC(NC(c3n(CC)nc(C)c3)=O)C2)=O)cc2ccccc2o1 C1(CNC(COC)=O)CCN(C(c2cccc(C)c2O)=O)CC1C C(=O)(CC(C)CC(C)C)N(CCNC(c1cncc(C(N)=O)c1)=O)CC C1(C(C)NC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)C(=Cc1c[nH]cn1)F N1(C(c2cnc(OC)s2)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 c1(NC(C2(C)CCN(Cc3ccc(C)cn3)C2)=O)cc(Br)c([N+](=O)[O-])cn1 N1(C(c2nc(C)oc2)=O)CC(CNC(=O)COCc2ccnn2C)C2(CC2)C1 C(CC1=CCN(C(c2cn(CCC)nn2)=O)CC1)NC(C(CCCC)O)=O N1(CC(C)(C)NC(Cc2c(C)ncs2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 N1(C(C2(C)CC3CCC2O3)=O)CC2(C1)C(NC(c1ccns1)=O)CCS2(=O)=O n1(CC(N2CC(C3(NC(C#CC4(C)CC4)=O)CC3)C2)=O)ccc(=O)c([N+](=O)[O-])c1 C1(CNC(=O)OC(C)(C)C)(OC)CCCO1.N12CCC(C1)n1cc(nn1)C2=O C(C(=O)OC(C)(C)C)(C(C)C)c1cnc(C)s1.C12CC(C1)OC(=O)C2 C1(C(N2CC(CNC(c3c(CC)n(C)nc3)=O)C2)=O)CCS(=O)(=O)C(C)C1 O=[N+]([O-])c1cc(OC)c(OCc2ccc(I)c(Cl)c2)cc1F C(C(=O)Nc1ccc(Cl)cc1F)(C1=CCCSC1)N(CCC)CC1CCOC1 N1(C(CSc2n(C)nnn2)=O)CC(C2CN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(CCS(=O)(=O)N1CCOCC1)N1C(NC(=O)CC=Cc2ccccc2)CC1 c1(C(=O)NC(CCNC(C(C)Cn2cccn2)=O)C)cc(Br)cnc1O O=C1Nc2c(C(N3CC4CN(C(C5CCCS5)=O)CC(C3)O4)=O)cccc2C1=O c1(OCC)ccnc(N2CCN(C(=O)CCN3CCOCC3)CC2)n1 C(=O)(C(O)CC(F)(F)F)NCC1C(C(=O)NCC(CC=C)(F)F)CCCC1 C#Cc1ccc(C(=O)NCC(CC=C)NC(c2ccc(F)c(CC)c2)=O)cc1Cl c1(NCC(CC)OC)ccc(S(=O)(=O)NC2CCOC3(CCCCC3)C2)cc1Br N1(C(c2ccc(N)cn2)=O)CCC(CNC(=O)CC(F)(F)C(F)F)C(F)(F)CC1 c1(C(=O)NCCCN(C2CN(C(N)=O)C2)C)csc(S(N)(=O)=O)c1 c1(OC)nc(NC(=O)CN2CCN(S(C)(=O)=O)CC2)ccc1-c1nn[nH]n1 Cc1cnc(NC(c2ccnc(-c3cccc(O)c3)c2)=O)c(Br)n1 C1(CNC(c2c(C)cnnc2O)=O)CCC2(CN(C(=O)Cc3cocn3)C2)O1 C1(C)(CC)C=C(C(=O)N2CC(F)(F)CC2C(=O)NC2CCC(C)CC2)C1 Cc1ccc(C(N2CC3CC2C3NC(=O)CC(C)C)=O)nn1 Cc1noc(C)c1CC(N1CCC(C(C)(C)NC(C2COCCO2)=O)C1)=O c1(NCC(N(C)C(C2CC2C2CCCCC2)=O)C2CC2)cc(S(C)(=O)=O)ncn1 Cc1ncn(C)c1C(=O)NC(C)CCNC(=O)CCCCC1CCCCC1 C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(C(CCC)(C)O)=O)CC1 C1(C(=O)OC)Cc2n[nH]cc2N(C(=O)C(c2ccc(Cl)cc2)O)C1 C1(CC(N2CC3C(NC(C4C5CC6C(C5)C46)=O)C3C2)=O)CCC2(CCC2)O1 c1(C(N(C)CC2(NC(=O)Cc3ncco3)CC2)=O)ccc(OCC(N)=O)cc1 CCCC(C)(CC)C(=O)N1CCC(O)(CNC(=O)COC)C1 C(CC(C)(C)C)(C(=O)N(C(C)C(=O)N(C1CCSC1)C)C1CC1)OC Cc1cc(N2CCC(CC(N3CCNCC3C3CC3)=O)C2)nc(C)c1 C(=O)(C1c2ccccc2C2CC1C2)N1C(CC)CN(C(=O)CC(C)SC)CC1 N1(CCC(=O)N(CC)Cc2ccccc2)CCc2nc(O)ccc2C1 CN(C)S(=O)(=O)N1CCCCC1CNCC(O)C1(Cl)CC1 C=CCCC(C(=O)OC)NC(=O)CC(C1CC1)NC(c1cnc(O)n1CC)=O C1(N(CC(O)COc2ccccc2F)C=O)CCCC(c2cccs2)C1 N1(C(CCCN(CC(C)N2CCC2)C)=O)CCC(NC(C)=O)CC1 C(C)(CC(=O)N1CCC1CC(=O)N(CC(C)CO)C)=C(C)C c1(C(=O)NCCCCCNC(c2cc(CC)sn2)=O)cc(C)nn1C(C)(C)C c1(COC)c[nH]c2cccc(-c3cnccc3C(N3CCN(CCO)CC3)=O)c12 C(CS(=O)(=O)N)(C1CCC1)N(C(CC(N)=O)c1ccsc1)C(C)C.CO O=C(C1CCCn2cnnc21)NC1CCN(C(C2CCCC3(CC3)C2)=O)CC1 C12(NC(C(CC)O)=O)CC(CNC(c3cnc(S)nc3)=O)(C1)OC21CCC1 N1(CC(=O)NC(CNC(CNC(=O)NC)=O)C2CCC2)CCCS1(=O)=O c1(C(=O)NCC(C2CC2)NC(C2(NCC)CC2)=O)ccc2cc(OC)ccc2c1 C1(C2CC2)(OC)CN(C(=O)CC(C)CNC(=O)OC(C)(C)C)C1 C1(C)(NC(C)=O)CCCN(C(c2cccc(-c3ccc(N)s3)c2)=O)C1 CC1CCN(S(=O)(=O)CC(=O)N(CCCNC(C2CC3(C2)CC3F)=O)C)CC1 c1(NC(CCc2c(C)ncs2)=O)cccc2c1N(CC(F)(F)F)CC2 c1(NC(C)=O)ccc(F)c(C(N2CC=CC2CNC(=O)C(O)C(C)(C)C)=O)c1 Cc1cccc2oc(C(=O)NCC3CCN(C(C4(C5CC5)CC4)=O)CC3O)cc12 c1(C(=O)NCCCN(C(C23CC(C)C2C3)=O)CC)cnc(C(C)(C)CF)o1 c1(OC(C)C(=O)N(c2cccc(CN3CCC(O)CC3)c2)C)cc(Cl)ccn1 N(C)(C1CN(C(=O)CCCCOC)CCc2ccccc21)C(C1C(OC)C1C)=O c1(Nc2ccccc2)cccc(P2(=O)CCCC2)c1.C12C(CC1O)NC(=O)N2 c1(CCCC)cc(C(N2CCCC2CN(C)C(C2(C#N)CCCO2)=O)=O)c(C)o1 c1(C(=O)NCC2CCN(C(=O)C(F)C3CC3)C2)cnc2[nH]nnc2c1 c1(NC(C(N2CC(CCOC)OCC2)=O)=O)cc(C)ccc1C(C)C C1(N(C(=O)CSCC2CCCO2)C)CCN(C(c2cscc2Cl)=O)CC1 C(C1CCCc2ccccc21)NCC(c1cccc(Br)c1)CO c1(C(N(CCC)CCNC(c2ccnn2C2CCC2)=O)=O)cccc2c1OCC2 C(C(CO)(CO)NC(=O)C(C)SC)N(C(c1c(CCCC)ocn1)=O)C c1(C(c2ccccc2)N(CC(C)C)CCCO)ccc(Br)c(C(F)(F)F)c1 N1(C(C2CCC(=O)O2)=O)CC2(C1)CN(C(C1CCCCS1)=O)CC2CO N1(C(C2CCN(S(c3c(C)n[nH]c3C)(=O)=O)CC2)=O)CCCC2(C1)OCC1CC21 C1(c2ccccc2)(NC(C(CC)n2ccnc2)=O)CCN(C(=O)CSC2CC2)C1 CC(CC(C)NC(c1ccnn1-c1ccccc1)=O)NC(=O)CCC1CCOC1 C1(C(=O)NC2CCCC(CNC(Cc3c(C)ncs3)=O)C2)CC2CC(=O)C1O2 C1(CCNC(c2cnc3cc(C)nn3c2)=O)CC(N=c2nc(C#N)[nH]cc2C)C1 N1(C(C=CC=CCC)=O)CC2CC(C1)C(CO)C2NC(=O)CCn1ccc(C)n1 c1(SC)c(C(=O)N(C2CC(NC(c3snc(Cl)c3Cl)=O)C2)C)cnn1C c1(C2(C(=O)NCC(CNC(C3(OC)CC3)=O)(C)O)CC2)ccc2c(c1)OCCO2 C1(C)(NC(CC2(OC)CCCC2)=O)CCN(C(c2nnc(C)s2)=O)CC1 Cc1cc(N(CCCNC(c2ccc(F)cc2C)=O)C)nc(CO)n1 C(=O)(C(CCF)NC(C1CCCN1C1CC1)=O)NCC1C(C)CC1 c1(CNC(c2c(CCC)n(CC)nn2)=O)nnc2n1CCN(C(C1CC1Cl)=O)C2 c1(C(=O)NC2(C)CCN(C(C3COC(C)(C)C3)=O)C2)ccc2c(c1)CCC2=O CC1CC(C(=O)NC2CC(C)(CNC(=O)CCNC(c3ccoc3)=O)C2)CN1C c1(CC(=O)NC2CCC(NC(C3(C)C(C)C3)=O)CC2)cccc2ncccc12 C#Cc1ccc(C(=O)NCC2(NC(=O)C=CC3CC3)CCCCC2)cc1 N1(C(c2c(CC)nccn2)=O)CC2CC(C1)CN(C(=O)CCCCCC(C)C)C2 N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(c1n[nH]cc1Br)=O)CC2CO n1(CC(=O)NC2CC(NC(CN3C(C)CCC3C)=O)C2)cc(P(C)(C)=O)cn1 CC(C)C(C(=O)N1CCOC(CC(=O)N(CC(O)CO)C)C1)C(C)C c1(NC(C2(CC=C)CC2)=O)cc(=O)c(NC(=O)NCCCNC(=O)NC)co1 Cc1cc(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)cc2ccoc12 C(=O)(CCCC(C(=O)NC1CCOCC1)N(C)CCSC)OCC C1(CC(=O)NC(C)C)CCCN(C(C2CC(=O)N(C3CCC3)C2)=O)C1 C#Cc1ccc(CNC(=O)CCC2CC(NC(C3CC(F)C(=O)N3)=O)C2)cc1 C(=O)(C(C)(C(C)C)NC(C)=O)NCC(CC=C)NC(=O)CCc1cn(C)nc1C C1(CC(=O)N(C2CCCN(C(C3(C(N)=O)CC3)=O)C2)CC)CCCC(=O)N1 Cc1cnc2c(C(N3CC(NC(=O)C(O)c4cnc[nH]4)CC(O)C3)=O)cnn2c1 c1(OC)ccnc(CN2CCN(CCCNC(c3cncc(O)c3)=O)CC2)c1 C(=O)(C(CCOCCO)NC(=O)C=CCN1CCCC1)NC1(C(=O)NC)CCCC1 C12(CNC(CN(C)C3CC3)=O)CC(C1)C(NC(=O)CCc1nnc(C(F)F)o1)CO2 N1(C(c2c(N)c(Cl)ccc2)=O)CC2(CCC(CNC(=O)CCc3cnn[nH]3)O2)C1 CCC(C)CC(C)C(=O)NCCNC(C12CCC(F)(CC1)C2)=O C=C(C)C1OCCC1C(=O)NC1CC(NC(=O)C(C)(C)C2CCCCC2)C1 N1(C(c2c(C)ccnn2)=O)C2CC1CN(C(=O)C(N1CCOCC1)C)C2 Cc1c[nH]cc(C(=O)NC(C2CCN(C(=O)CCCOC(C)(C)C)C2)C)c1=O N1(C(CCCc2cc(C)no2)=O)CCC2OCCN(C(c3csnc3C)=O)C2C1 Cc1cccc(C)c1CN(CCNC(C1CN(C)C1)=O)C1CC1 N1(c2nnc(C(=O)OC)s2)CC(C)(C)CC1CNC(=O)C(F)(F)CC1CCCO1 N1(C(c2nnn(C)n2)=O)CCC(C2CCN(C(c3snc(O)c3Cl)=O)CC2)C1 C1(C(=O)O)CC(c2ccccc2)CCN1C(C12COCC(C1)C2)=O c1(C(N2CC(NC(c3c(C)cccc3)=O)C(F)C2)=O)ncnc(O)c1Cl N1(C(C2CCC(C)(CC)O2)=O)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(C3C(C)(C)C3(C)C)=O)C2)cc(Cl)ccc1C(F)(F)F c1(C(N2CCC(N(C(=O)C(F)OC)CC)C2)=O)ccnc(C)c1C C(CC1=CCN(C(=O)CSC2CC2)CC1)NC(c1ccc(Cl)cc1C(F)F)=O N1(C(c2cc(C(C)C)on2)=O)CCOC2(C1)CN(C(C1(S(C)(=O)=O)CC1)=O)C2 C(CCCC(CO)NC(c1ccc(F)s1)=O)NC(COCCCCCC)=O CC(C(=O)N(C)CCOCCNC(=O)C(C)O)NC(c1cccs1)=O C(C(C)C(=O)Nn1ccccc1=O)N(C(CCC(C)(C)SC)=O)C C1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)CCOC2(CCOCC2)C1 N1(C(c2cnc(Cl)s2)=O)CCN(C(c2cc(O)ccc2F)=O)C(CC(F)(F)F)C1 Cc1cc2ncc(C(N3CCC(C(=O)Nc4ccc(CCO)cc4)C3)=O)cn2n1 C1(C(F)(F)F)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCOCC1 C(CC(C(=O)N1CC(C)(C(N)=O)C1)NC(=O)CN(C1CCCC1)C)=CC C(=O)(C1=CCCN(Cc2cnc(Br)s2)C1)NC(c1cccnc1)C(C)C N1(C(c2cc(CCC)on2)=O)CCN(C(C2CCN2CC)=O)CC1CS(C)(=O)=O Cc1nc(C(C)C)nc(O)c1C(N1CCC(CF)(NC(=O)C(C)O)C1)=O C1(CNC(C=CCC)=O)CC(NC(c2ccc(C(C)CC)cc2)=O)CCO1 C1(CNC(CN(C)CCc2ccccc2)=O)CN(C(=O)CC#N)C(C)(C)C1 C1(C(N(CC)CC2CCOC2)=O)CC(C)(C)CCN1C(C1CCCCC1(C)C)=O C(=O)(C(O)CC(F)F)N1C(CN(C)C(c2cccc(Cl)c2O)=O)CCC1 CC1=C(C)C(OC(C2(C(=O)Nc3ccccc3)CC2)=O)CCC1 C1(CC(=O)NCCC(CNC(=O)CCn2ccnc2)OC)CC2C=CC1C2 c1(CC)conc1C(=O)NCC1CCCC1NC(c1ccc(-c2ccco2)s1)=O N1(C(Cc2nc(C)sc2)=O)C2CCCC1CN(C(C1CCCC(F)(F)CC1)=O)C2 C1(C(N2CCCC(N(C(c3ncn(C)n3)=O)CC)C2)=O)CCCCC(=O)N1 CP(C)(=O)c1ccccc1C(=O)N(CCNC(=O)Cn1ncnn1)C1CC1 c1(C(C(N2CC(NC(C3CC3CF)=O)(CO)C2)=O)O)cccc(F)c1 S(=O)(=O)(CC(=O)N(CC(C)O)CCNCC)NC1CC1.C1CCN(CC(C)C)C1 c1(CNC(C2(COC)COC2)=O)cncc(C(=O)NCC(O)(CO)CO)c1 C(=O)(C1=COCCO1)NC1C(CNC(c2cnc(C(C)(C)C)nc2)=O)CCCC1 C1(OC)CN(C(=O)Cn2ncnn2)CC1C(=O)NC1(C)CCOC1=O C1(C)(CC(=O)NC2CCC(NC(C(CC)CC)=O)C2)CCS(=O)(=O)N1 N1(C(C2N(CC)CCC2)=O)CCC(O)(C(=O)NCC2CCCC(OCO)C2)CC1.C.N=C c1(C(N(CC(CNC(Cc2ccc(CC)cc2)=O)O)C)=O)ccc2nn[nH]c2c1 c1(OC)cccc(OC)c1C(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 O=C(CC1COc2ccccc21)N1CCOC(CCNC(C2(C3CC3)CC2)=O)C1 c1(C(N2CCC(CN(C(C(c3ccccc3Cl)C)=O)C)C2)=O)ccc(F)c(N)c1 C1(C(N2C(CNC(c3cc(C)n(C(C)C)n3)=O)CCC2)=O)CCn2cnnc2C1 C1(C(N(CC(C)CNC(C2CC3(C2)CC(CO)C3)=O)C)=O)CCC2C(C1)C2(F)F N1(C(CC(CC)CC)=O)CCC2(NC(c3ccc(SC)o3)=O)CCCC12 N1(C(C(CC)SC)=O)CC(CC(=O)NC2C(C)(C)C2(C)C)C2(CC2)C1 C1(C(=O)NC2COCCC2O)CC2(CC2)CN1Cc1ccncc1Br C1(NC(c2ccc(O)cc2)=O)CC(C(=O)NC2CC3CCC2O3)C12CCC2 N1(C(c2nc(C3OCCO3)c(C(C)(C)C)s2)C)CC2CCC1C2N C(=O)(CCC(C)(F)F)N1CC(C(C(=O)N(C)Cc2cncnc2)O)C1 C=CCC(C)(C)C(=O)N(CC)CC1CN(C(=O)CCOC(C)CC(C)C)CCO1 c1(C(N2CCN(c3ccc(C)c(C)c3)CC2)=O)cnc2c(Br)c(C)ccc2c1 C(N=c1[nH]c(=NCCOC2CC2C)c2ccccc2[nH]1)c1c(C)c(F)c(F)cc1 C1(F)(COC)CCN(C(c2ccc(-n3cnnn3)c(I)c2)=O)CC1 C1(S(N)(=O)=O)(C(N(C2CCCCC2)CCNC(CN(CC)CC)=O)=O)CCC1 c1(CC)nn(C)c(Cl)c1C(N1CCOCC(C(C)(C)C)C1)C(=O)NCCC#N N1(C(C(CCC)NC(=O)CCOCC(=O)OC)=O)CC(C)CCC12CC2 CCC(C)C(O)C(C)C(=O)NCC(C)(O)CNC(c1cccc(O)c1F)=O Cc1nc(Cl)nc(N2CCC(N3CCN(C(C4CCCN4C)=O)CC3)CC2)c1Cl CC(Cc1ccco1)C(=O)NCCOCCNC(=O)Cc1coc(C(F)F)n1 c1(N(C(C)C)C)ccccc1C(=O)NCC1CCN1C(C1CNC(=O)N1C)=O c1(C(=O)NCC2(CNC(C3CN(C)C(=O)CC3)=O)CC2)ccc2c(n1)CCC2=O c1(N(C(=O)NCCCC2CCOC2)CC)nc(C)nc(=N)[nH]1 c1(OC)csc(C(N2CCN(C(C3(C(N)=O)CCC3)=O)CC2)=O)c1OC C1(CNC(C(CC)F)=O)CN(C(C2(COC)CCOCC2)=O)CC(C)(C)O1 n1(CC)nc(C(=O)NC2(CNC(=O)CC3CCC(=O)NC3)CCCCC2)cc1O C1(NC(C(C)(C)OC(C)C)=O)CC2(C1)CC(C(=O)NC1C3CCCCCC13)C2 N1(C(c2c(CCC)occ2)=O)CC(NC(c2ccncc2Br)=O)CC(F)C1 c1(C(=O)NCCCC2N(C(C(COC)C)=O)CCC2)cccc2c1nc(O)n2C N1(C(c2c(C)ccs2)=O)CCN(C(c2cn(C)nn2)=O)CC1C1CCCC1 N1(C(Cc2c(C)cccc2)=O)CCN(C(=O)C(CO)c2ccccc2)C(C#N)C1 Cc1cncc(C)c1C(=O)NC1CCCC1NC(=O)CC(F)(F)F C1(CN(C(C(=O)NCC(=C)C)C)C)CCN(C(c2coc(C3CCC3)n2)=O)C1 C=CC1(C(=O)NC2CN(C(=O)C(C)CC3CCCC3)CC2C)CCOCC1 CCCC(C(O)C(=O)Nc1cc(C)ccc1C)NC(=O)C(C)(C)COC C=C1CC(C)(C(=O)NC(C)C(C)NC(=O)CCOCCOC)C1 c1(COC)csc(C(=O)N(CCCCNC(=O)CCc2nc(C)cs2)C)c1 C1(NC(C(C)(C)CC2CC2)=O)CCOC12CCN(C(C1(C)CC3CC3C1)=O)CC2 C(=O)(CCN=c1[nH]ccs1)N1CCC(CCNC(c2cnc(CC)[nH]2)=O)C1 c1(-c2cccc(CC(=O)NC(c3cscn3)C)c2)c(O)cccc1O N1(C(CCCC#C)=O)CC(CNC(c2nc(Br)c(C)s2)=O)C(F)(F)C1 C1(C)(C(=O)OC)CCCN(C(c2ccc(-c3ccc(C)c(OC)c3)nc2)=O)C1 CC1CN(C(c2cscc2C(F)(F)F)=O)CC1NC(=O)C(C)(C)c1cnn(C)c1 CC(CCC(F)(F)F)NC(=O)CCNC(C1CCCCC(=O)C1)=O Cc1c(C(=O)NCCN(C(=O)C(C(C)C)NC(N)=O)C)[nH]c2c(C)cccc12 N1(C(C(C)S(N)(=O)=O)=O)CC(C)CN(C(C2CCC(F)(F)CC2)=O)CC1C N1(C(C)C)CCCC(CC(=O)NC2CCCC(NC(=O)Cc3ncc(Cl)s3)C2)C1 O=C(CC(F)(F)C(F)(F)F)NC1CN(C(=O)COC2CCCCC2)C2CC12 C1(CCOCCO)C(=O)N1.C(CNC(C)=O)(C(=O)N1CCC(C)C1)OC.OC c1(C(=O)NCC2(NC(C3C(C)=C3)=O)CC2)ccc(F)c(C)c1Cl Cc1n[nH]c(C)c1CC(C)C(N1CC(CNC(=O)CSCCN(C)C)C(C)C1)=O c1(CN2CCC(NC(C(C3CC3)OCC)=O)C2)nc(Br)ccc1F c1(C(=O)NC(C2CCCN2C(=O)CC(C)(C)C#N)C)c(OC(F)F)cccc1Cl C(=O)(CC(C)C(F)F)N(CC1(CNC(CN(CC)CC)=O)CCCC1)C1CC1 CCCC(C)(CC)C(=O)NCc1cc(C)c(C(=O)NCCCN(C)C)o1 C(=O)(CC(C)C(=O)OC)NC1(C(=O)NCC(=O)OCC)CC1C C1(N(C(=O)C(O)C2CCCC2)C)CN(C(c2ccccc2Cl)=O)CC1O C1(C(=O)NCC(C(=O)OC)O)N(C(=O)CN2CCNC(=O)C2)CCC1(C)C c1(OC)ccccc1C(C)C(=O)NCCCCCCNC(C1(C)CC(F)C1)=O n1(CCN(CCNC(COc2ccc(OCC)cc2)=O)C)c(C)cc(C)nc1=O Cc1ccc(Cl)c(C(=O)N(C)CC2(NC(=O)C(c3ccc(Cl)cc3)CO)CC2)c1 N1(C(c2cc(OC)cc(OC)c2)=O)CCCCC12CC(NC(C1(O)CC1)=O)C2 C1(CC)C(NC(=O)CCc2ncccn2)CCCN1C(c1ccc(Cl)cn1)=O CCC(O)(CC)CCNc1ncnc(NC2COCC2OCC)c1C CC(C)(C(=O)NC1CC(O)(CNC(c2ccc[nH]2)=O)C1)Oc1ccccc1 c1(C(N2CCN(C(C(CCC)CCC)=O)CC2C)=O)ccc2c(C#N)c[nH]c2c1 C1(C)(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)CC2CCC(F)(F)C2)C1 CC1CCC(O)(C(=O)NCC2CCN2C(C2CCC(C)(C)C2)=O)CC1 C(N=c1cc(C)[nH]c(=NCC2CCCN(C)C2=O)[nH]1)c1c(CC)cc(F)cc1 c1(C(=O)NCC2(O)CN(C(C(C)NC(C)=O)=O)C2)[nH]nc2ncc(Br)cc12 N1(C(CCCSC)=O)CCC(C(F)(F)F)C(NC(c2cc(C(N)=O)no2)=O)C1 C1(C(N2CCN(CCCNC(c3ncc(C)nc3)=O)CC2)=O)CC(S(C)(=O)=O)C1 N1(C(c2c(C)cc(OC)c(Cl)c2)=O)CCN(C(=O)CNC=O)CC(C)(F)C1 c1(C(C)NC(C(C)OCCOC)=O)nc(C(=O)NCc2cncn2C2CC2)co1 c1(C2(CNC(=O)NCCC3C(C)OCC3)CC2)cccc(C(F)(F)F)c1 C(CCCC(=O)NC(CC(C)C)C(=O)N(C(C)C(C)SC)C)(OC)OC N1(CCCNC(CC(C)NC(N)=O)=O)Cc2ccccc2C1 C(=O)(C1=CCN(C(=O)C2=NOC(C)C2C)CC1)NC(C1CCOC1)C#C N1(C(CNC(CNC(C)=O)=O)=O)CCC(CO)(NC(c2n[nH]c(C)c2C)=O)C1 c1(NC(c2ccc(C(C)C#N)cc2)=O)cc(F)c(C(F)(F)F)cc1F c1(C(C2CCOCC2)N(C(c2cc(C)no2)=O)C2CC2)cnc(C(F)(F)F)nc1 N1(C(C)=O)CCCCC(CNC(=O)Cn2c(-c3ccccc3)c(C)sc2=O)C1 c1(OC)nccc(C(=O)NC2(C(=O)NCc3ccn(C4CC4)n3)CC2C)n1 c1(C(N(CCCNC(C2CC2(Cl)Cl)=O)C)=O)cnn(-c2ccccc2)c(=O)c1 C1(O)(CNC(CCSCC)=O)CCCN(C(c2cncn(C)c2=O)=O)C1 CC(C)(CO)CCN=c1[nH]c(=NCc2cccc(P(C)(C)=O)c2)[nH]c2c1CCCC2 C1(C(=O)NC(C(C)(C)NC(CCc2cnc(C)o2)=O)C)CC2OC1C1CC21 C1(C(=O)NC2(CN(C(C(C)OCCCC)=O)C)CC2)CC(c2ccccc2)=NO1 C(=O)(C(CCSC)OC)NC1CC(CCNC(CN(CCC#C)C)=O)C1 O(NC(=O)C1=CC2(CCN(C(=O)C(C)OCCC(C)C)C2)C1)CC(C(C)C)O C(CNC(c1cc(O)nn1C)=O)(CC(F)(F)F)NC(CC(CC)C1CC1)=O C1(CC=C)(NC(=O)CC2CC(C)(C)CO2)CCN(C(=O)CS(C)(=O)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)COCC(C)(C)C)C2C)nc(C)c1 N1(C(C(C)=C2CCCC2)=O)CC2CCC1CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(C(N2C(CNC(C(CC)COC)=O)CC2)=O)cc(Br)cc2cccnc12 c1(OC)cncc(OCC(C)OC(C2CCCC2c2ccccc2)=O)c1 N1(C(=O)NCCc2cccc(C(=O)NC)c2)CCC2(CC1)CC(O)C2 C1(C(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)CCn2ncnc2C1 CC(C)C(F)(CNC(=O)CN1CCN(C)CC1)C(=O)N1CCC1C1CCCC1 C1(O)(CNC(c2sc(C)c(O)n2)=O)CC2CCC(C1)N2C(C1(C)CCCOC1)=O CCCCCOCCC(=O)NCC(CO)NC(=O)C(=O)NCC1CC1 c1(C(=O)NC2CC(C)(NC(CC(CC)OC)=O)C2)cc(Cl)c2c(c1)OCCO2 c12ccc(F)cc1CN2C.C(O)(C(F)(F)F)C1CCC1.C12CC(C1)CNC(=O)N2 c1(NC(C(c2cccs2)NC(c2nc[nH]n2)=O)=O)cccc(OCF)c1 N1(C(c2c(C)nccc2)=O)CC(C)(C)OCC1CNC(C1(C2(O)CCC2)CC1)=O C1(C)(C(=O)NCCN(C(=O)COCC2CCCCO2)CC)CCN(C)C1 C12(NC(C(C)NC(=O)NC)=O)CCCC1N(C(=O)CCc1ncc(F)cn1)CC2 C1(CNC(=O)C(O)C2CC2)CC2CC2N1C(C1(F)CCCC1)=O c1(C(C)C)nc(NC(c2csc(C3CC3)n2)C)cc(N2CCC(Cl)=C(Cl)C2)n1 C(=O)(C(CC(C)C)C(C)C)NC1(CC)CCCN(C(c2cn(C)nn2)=O)C1 c1(OC)ccnc(C(=O)NCCC2CC(NC(C3(C)CC3(Cl)Cl)=O)C2)c1N N1(C(=O)CC2CC2)CC2CCN(C(c3cnn(C4CCOC4)n3)=O)C(C2)C1 N1(CCCNC(C(C)OCC#C)=O)CCN(C(C2(c3ccno3)CCC2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCC2(CCN(C(C3(n4cncn4)CC3)=O)C2)C1.C1CC1 CCCC(C(O)C(=O)NCC(=O)N(C)C)NC(C1CC(=O)CC12CCC2)=O N1(CC)CCN(C(=O)CC2CCC(NC(c3cc(C)ncc3Cl)=O)CC2)C(C)C1 c1(C(=O)NCC2CN(C(C3(C(F)F)CC(=C)C3)=O)CC2C)cc(C)c(C)nn1 c1(C(N(CCC)CC)=O)ccn(CCNC(=O)CCC2CCOC2)c1 C(C)(C(=O)NCC1(C(=O)NCC)CCC1)NC(COC)=O.C1(S)CC1 c1(C(=O)NCC(CC(C(C)C)O)C)cccc(S(=O)(=O)N(CCC(N)=O)C)c1 CC12CN(C(C3CC4CCC3O4)=O)CC1(C)CN(CCC1=CCCCC1)C2 Cc1nc2cc(C(=O)NC3CCC3NC(c3c[nH]nc3C(F)F)=O)c(F)cc2[nH]1 Cn1ccc2c(C(=O)NC3CN(C(=O)CC(C)(C)C)C4CC34)ncnc12 CC1(C)CC(C)(C(=O)NC2CCC(NC(=O)COC3CC=CC3)CC2)C1 N1(C(C(n2ccc(C)n2)(C)C)=O)CCCC(CNC(C2CCC(F)CC2)=O)CC1 C(C(C(=O)NC(C)C(C)C)NC(=O)C(C)=CC(C)(C)C)OCC c1(N2CCN(C(CC)=O)CC2CCO)ncc2sccc2n1 c1(C(N2CC(COC)N(C(C3CC3C3CCC3)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(c2cnn(C)c2F)=O)CCC(NC(=O)Cc2ccc(F)cc2F)CC(O)C1 N1(C(C(C)NC(COC)=O)=O)CC2(CC2)CC1CNC(=O)CC1CC2(CCC2)C1 N1(C(CCC=C)=O)CCC(c2ccccc2)(NC(=O)Nc2ccc(NC)cc2)C1 C(C(CCC)CC(C)C)NC(C(CCCOC)NC(CCCC#C)=O)=O C(CC(O)C(=O)N1C(C(=O)NCCC2CCN(C)CC2)CCC1C)N(C)C c1(CC(=O)NCC2CN(C(C34CCC3C4)=O)CCO2)ccc2c(c1)OCCCO2 N1(C(C=CC)=O)CC(CO)(NC(c2ccn(C(c3ccccc3)C)n2)=O)C1 c1(CN2C(C(=O)Nc3cc(OC)ncn3)CC2)ccc(F)c(F)c1Br N1(C(C(CCCCC)O)=O)CC2(C=C(C(=O)Nc3ccc(C)nc3C)CO2)C1 CN1C(=O)CCC(NC(C2COCCN(C(c3cc4n(n3)CCO4)=O)C2)=O)C1=O C1(NC(C(c2c(C)noc2C)C)=O)CN(C(=O)C2=CSCCO2)CCC1CO Cc1nc(C(=O)NCc2ccsc2C(=O)NCC2CCSC2)cc(O)n1 c1(NC2CC(OC)C2)cc(C)c(S(=O)(=O)N2CCCN3CCCCC3C2)cn1 N1(C(C2CCS(=O)(=O)N2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CCC2)=O)C1 C1(NC(c2ccccc2Cl)=O)COCCN(C(c2cc(Cl)ncc2F)=O)C1 N1(C(=O)CCc2ccc[nH]2)CCC2CCC(C1)N2C(=O)CCOC1CCOCC1 C(=O)(C(CC(F)F)NC(C1CC(F)(CF)C1)=O)NC(CC)C(C)(C)O N1(C(c2c(CC)ccs2)=O)CCCCC1CCC(=O)NCC(Cl)Cl C1(NC(C(C(C)C)NC(C)=O)=O)CCCN(C(c2cncc(C)n2)=O)CC1 Cc1ccc(C(=O)NC2CC(NC(C3CCCC3(F)F)=O)C2)c(C)c1 C=CCC(F)(F)C(=O)NCCC(CC)(CC)NC(C1CC(CF)C1)=O c1(C(N2CCCC(c3ccccn3)C2)C(=O)NC2CCOC2)cc2c(s1)CCC2 C12(NC(=O)CSCc3ccc(Cl)cc3)CCN(C(c3coc(O)n3)=O)CC1C2 n1(CC(=O)NC(CCN(C(CC(C)OC)=O)C)C)c(O)nc2ccccc12 C=C(C)C(C)(C)C(=O)NCC1(NC(c2cnns2)=O)CCOC1 N1(C(c2cnc(C)[nH]2)=O)CC2(CC2)CC1C(=O)N(C(C)C)Cc1cccnc1 C1(NC(C(C)C(F)F)=O)CC(C2CCN(C(c3c[nH]nc3C3CCC3)=O)CC2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(=O)C(C)Cn2ccc(C)n2)C(C)C1 c1(C(N2C(CC(=O)N(CCCCO)CCCC)CCC2)=O)cc(F)ncc1Br CC1CC(C)CN(CCN2CC(c3nn[nH]n3)CCC2=O)C1 c1(CSc2ccc(-c3cc(C(C)C)no3)s2)ccccc1.c1nc(C(C)C)no1 C1(NC(CSCC(C)C)=O)CCOCC1NC(=O)CC(c1ccc(F)cc1)O N1(C(C=COCC)=O)CC(CN=c2nnc(CC)c(CC)[nH]2)C2(CCOCC2)C1 CCC(CC(F)(F)F)C(=O)N(C)CC1(CNC(c2cccc3nc[nH]c23)=O)CC1 C(CCCC(=O)NC12CC(F)(C1)C2)N(C(CN(CC(C)(C)C)C)=O)C N1(C(c2c(C)ccnc2F)=O)CC2(CCC(C(=O)NCc3ccnc(Cl)c3)O2)C1 N1(C(C(CC)SC)=O)CCN(C(=O)CSC(C)C)C(c2ccc(OC)cc2)C1 CCC(CC(=O)NCC1CC1)NC(=O)C(C)OCC(C)C N1(C(C2(F)C(C)C2)=O)CCCC2(CCN(C(=O)CC(C)(C)CC(F)F)C2)C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cc(C)oc2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(C(F)=CC)=O)C2)ccc2sc(C)nc2c1 C1(CC=C)(C(=O)N(C2CCC3CC23)C)CCN(C(c2c[nH]nc2OC)=O)C1 n1(CC(=O)NCC2N(C(CCOCCN(C)C)=O)CCOC2)cc(F)ccc1=O S(=O)(=O)(c1ccc(N(C)CCn2cnc(Br)n2)c(Cl)c1)NC(C)CCO Cc1cn2cc(C(N3CCN(C(=O)CCCC4CCC4)C(C4CC4)C3)=O)sc2n1 C12(C(=O)NC(C(C)NC(C3CC=CCO3)=O)C)CC3CC(F)(C1)CC(F)(C3)C2 C(CCCCC(=O)N(C1CC1C)C)n1cc(-c2ccc(C)n2C)nn1 Cn1nc(C(=O)NC2(CCNC(C3CC4CC4C3)=O)CCC2)c(Cl)c1Cl C(CO)(C(F)(F)F)NC(=O)CC1CCC(NC(=O)CC2CC3(CC3)C2)CC1 C=CCCCC(=O)N(CCCNC(=O)CCCOOC(C)(C)C)C.N1C(=O)OCC1 N1(c2ccnc(C(C)C)n2)CCC2(CC(NC(=O)CC(C)c3ccncc3)C2)C1 N1(C(CSCC)=O)CCOCC1CN(C(=O)Cc1cc(C)no1)C C(=O)(CC1OCc2cc(Cl)ccc21)N1CCC(NC(c2c(C)ccnn2)=O)C1 N1(C(C(CC(=O)OC)(C)C)=O)CC2(C1)CN(C(C1C=CCCC1)=O)CCO2 C1(C(=O)NCCCCNC(C2COC3(CCC3)C2)=O)SC2=CCC1CCCC2 c1(COC2CN(C(CCCSC)=O)C2)cncc(CO)c1.c1(C(=O)N)occc1CO N1(C(c2cnn(CC)c2C)=O)CC(NC(C2CC3(CCC3OC)C2)=O)C2(CC2)C1 c1(C(=O)NC(C(=O)N(C2CCC2O)C)C2CCCO2)ccc(C#N)cc1 CCC(C(=O)N1CCC(CNC(c2nocc2C)=O)(OC)CC1)C(F)(F)F C(CCCCCNC(c1coc(-c2cccc(Cl)c2)n1)=O)NC(C(CSC)C)=O C1(CNC(CN(C)CC)=O)CN(C(C2(CF)CC(=O)C2)=O)CC1OCC c1(C(=O)NCC=CCNC(c2cnc(CCC)s2)=O)ccc(NC(C)C)c(F)c1 c1(C(c2onc(CCOC)n2)C(=O)OC)cccc(Br)c1 N1(C(c2[nH]c(=N)sc2)=O)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 C1(NC(CCc2onc(C(c3ccccc3)OCC)n2)=O)C(=O)OCC1(C)C Cn1nnc2cc(C(=O)NC3CCN(C(C4C5CCC45)=O)CC3)cnc12 CCC(CC)C(C)C(=O)NC1CCC(NC(=O)C(c2ccc(C#N)cc2)(C)C)C1 N1(C(C(CC)SC)=O)CC(NC(c2cc(Cl)c(Br)[nH]2)=O)C(C)C1 c1(C(N(C2CCN(C(C3CCCC3O)=O)C2)CC)=O)sc2cncn2c1C c1(CNC(CCCOCCC)=O)nc2c(s1)CCN(C(c1cncnc1)=O)C2 C1(C(N2CC(C(=O)N(CCCOC)C)(SC)C2)=O)CC1C1(C)COC1 c1(N(C2CC2)CC2N(C(=O)OC(C)(C)C)CCC2)cc2sccc2s1 c1(N2CCC(OC)CC2)nc2c(c(=NCC(C(C)C)N3CCCCC3)[nH]1)COC2 c1(C(=O)NC(CN(C(=O)CC2COCCO2)C)(C)C)n[nH]c(C2CC2)n1 N1(C(CCCN(C)C)=O)CCCC12CCN(C(=O)CCOC1CCOC1)C2 N1(C(C2OCC(=O)N(CC)C2c2cccnc2)=O)CCS(=O)(=O)C(C2CC2)C1 CC(CNC(=O)C=CCN(C(=O)C(C)n1cncn1)C)CO c1(C(=O)NC(C)(CNC(=O)C(F)C2CC2)CO)cc(F)ccc1F C1(C(N(CCC)CCC)=O)CCN(C(C2C=CCCC2)=O)C(C)(C)C1 CCCCCC(F)C(=O)NC1CC(CNC(=O)CCn2ccccc2=O)CC1O N1(C(C(CSC)C)=O)CCCC(CCNC(=O)C(F)CC2CCOC2)CC1 c1(N2CCCN(C(c3ccc(F)cc3)C)CC2)ccc2cnc(C#N)cc2c1 C=CCC(C)(C(=O)N1CCCC(CCNC(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C C12(NC(CCC(=O)NCC)=O)CC(CNC(C3CCC3C)=O)(C1)OC2(C)C c1(CNC(c2cc(C)ns2)=O)ccc(CN(C(=O)CC2C(C)(C)C2(C)C)C)cc1 c1(CC)ccc(C(C)C(=O)NC2C=CC(CNC(c3ccccc3)=O)C2)cc1 c1(OCC)ccnc2sc(C(=O)NCCC3CN(C(=O)C(C)OC)CCO3)cc12 c1(SC)nc2ncnc(N3CCCC(CNC(c4nccnc4Cl)=O)C3)c2s1 Cc1cc(NC(C2CCN(C(=O)c3ccon3)O2)=O)cnc1C c1(CNC(C2N(C(C=C=C(C)C)=O)C(C)C2)=O)ccc(C)cc1F CC1CCC2(CC1)CCN2C(c1cncc(CNC(=O)COCC(F)F)c1)=O N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C(F)C1 CCC1=NOC(C(=O)NC(C)CCCNC(=O)C(N2CCCCC2=O)C)C1 CC1CC(CNC(c2ccc(-c3cccs3)s2)=O)CN1C(c1cc(O)nn1C)=O CC1(C)CC(CC(=O)NC2(CO)CCN(C(=O)Cc3cnccn3)CC2)CCO1 Cc1ncc([N+](=O)[O-])cc1C(N1CC(C)(NC(=O)C=C2CCOCC2)C1)=O c1(C(=O)NC2CCCN(C(C3CC(C)N(C)C3)=O)C2)c[nH]c(=O)c2ccncc12 c1(NC(CC2N(C(CCOC)=O)CCC2)=O)c(Cl)cccc1Br c1(C(=O)NC(CC)CNC(c2csc(O)n2)=O)cc[n+]([O-])cc1 CC(C)CC(C)CC(=O)NC(C(=O)NCC(F)CO)c1cccs1 C1(NC(CCNC(N)=O)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 C#CCC(C)C(=O)N1CCCC1(C)CNC(C1(C(c2ccccc2)=O)CC1)=O c1(C(N2CCC(CCCNC(C(COC)(C)OC)=O)CC2)=O)cn2ccsc2n1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)(CNC(=O)Cc2nc[nH]n2)CC1(C)C c1(C(=O)NC(CCC(N2CCC(CC)(CO)CC2)=O)(C)C)cncc2[nH]ccc12 C1(Nc2ncc(C(=O)OC)cc2Br)CCC2(CN(C(=O)CC(=O)NC)C2)O1 N1(C(c2cn(CC)nc2C)=O)CCC2(C(N3CCCC(C)CC3)=O)CCCC12 C1(NC(c2c(OC)scc2)=O)CN(C(c2cn(CCCF)nn2)=O)C(C)(CO)C1 c1(C(C)=O)cccc(C(N2CCC(O)(CCNC(=O)CC(C)N(C)C)C2)=O)c1 c1(C(=O)NC2CC3CN(C(CCOCCN(C)C)=O)CC32)ccnc2[nH]nnc12 N1(C(c2c(OC)n(C)nc2C)=O)CCN(c2ncnc(=N)[nH]2)CC(O)C1 CN1CCCC(C(C)(C)C(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)N(C2CCC(CO)CC2)C)CC1)OC C1(C(N2C(C)(CNC(C3C(C)C3)=O)CCC2)=O)Cc2cc(Cl)ccc2O1 N1(Cc2cn(C)nn2)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1.C1(=O)CN1 C(=O)(C1=NOC2CNCC12)NC(C)Cn1cc(CC(C)(C)C)nn1 c1(C(N(CC(C)(C)CNC(=O)CC2=CCCC2)C)=O)cncc(P(C)(C)=O)c1 c1(OC)cc(C)c(Cl)cc1C(=O)NCC(C)(CC)NC(=O)C(N1CCC(C)C1)=O N1(C(CNC(C(CC)C)=O)=O)CC2CCCC(NC(=O)CSc3ccccc3)(C2)C1 N1(C(c2ccsc2Cl)=O)CC(CNC(=O)C(F)(F)C2(O)CCC2)C(O)C1 N1(C(Cc2n(C)ncc2)=O)CC2(CCN(C(=O)C=Cc3ccncc3)C2)C1 C#CC1(C(=O)NCC2CN(C(=O)C=C(Cl)Cl)CCC2C)CCOCC1 N1(C(C(CC)SC)=O)CCC(C2CCCN2C(c2ocnc2C)=O)CC1 c1(C(N2C(C)CC(CNC(C(C(CC)C)OC)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1OCCC1CN(C)C(C1CC(CCNC(=O)Cc2ccn(C)n2)C1)=O c1(C(=O)NCC(CC(C)C)NC(c2n(CC)nnc2C)=O)cnc(C)nc1C C(=O)(C(CC(C)C)C(C)C)NC1C(C(N2C3CC(=C)C(C3)C2)=O)COCC1 CC(CC(=O)NCC1CCOC1C(=O)N(C1CCCC(C)(C)C1)C1CC1)CC(C)(C)C c1(NC(C(CC2CCOCC2)NC(C(CCCC)F)=O)=O)cc(C)cn(C)c1=O N1(C(c2c(OC)cc(O)nc2)=O)CC2CC3CC2C1C3NC(=O)CS(C)(=O)=O Cc1cc(C(=O)NCC2CCC(NC(c3ocnc3C)=O)CC2)cc([N+](=O)[O-])c1 c1(C(N(C2C3CN(C(CC(C=C)C)=O)CC32)C)=O)cccc(=S)n1O C1(C(N2CCC(N(C(c3ccn(CC)n3)=O)CCO)C2)=O)CC2(C1)CC(F)C2 C1(C(N(CCCCCC)CCNC(=O)CNC=O)=O)CCc2n[nH]cc2C1C Cc1cc(C(N2CC3=C(C2)CN(C(C2(CO)CCCO2)=O)C3)=O)cc(N)c1O N1(CCC)CCCCC1C(=O)NCC(C)NC(=O)C(=Cc1c[nH]cn1)F N1(C(C(CC)O)=O)CCN(c2ccc(C(=O)N(C)Cc3cccs3)cn2)CC1 N1(C(C2(CC)CCNC2=O)=O)CC(C(=O)NCc2nn(C)cc2O)C2(CCC2)C1 C1(C(=O)NC(CC=C)CC=C)COCCN(C(=O)C(F)C2CCCC2)C1 NS(=O)(=O)c1cc(C(=O)NC2CN(C(C3CCCO3)=O)CCC2CO)cs1 c1(CC(N2CC(C)(NC(c3cc(I)c[nH]3)=O)C2)=O)cccc(C#N)c1 N1(C(CCCC#C)=O)CCC(F)(F)C(NC(c2cc(F)cc(F)c2Cl)=O)C1 c1(C(=O)NC2CC(NCc3ccc(C)nc3Cl)C2)cc(F)cc([N+](=O)[O-])c1Br Cc1ccccc1OCCCC(=O)NCC1(CNC(=O)CCC=CBr)CC1 C1(C)(C(=O)NC2(C(N(C)CCOCCO)=O)CC2)CCCC1 Cc1snc2sc(C(N3CC4C(C3)N4C(C3CCCCC3)=O)=O)cc12 C1(COC)CCN(C(=O)C(C)S(C)(=O)=O)C12CCC2.C1CCCCC(=O)N1 C(CC(C)(C)C(=O)N1CCC(O)(CNC(=O)CCSC(F)(F)F)CC1)OC N1(C(C2(CC)CC2)=O)C2CCC1CC(C(=O)NCC(C)Sc1ccc(F)cc1)C2 c1(CNC(C2(OC)CCC2)=O)nc2c(s1)CN(C(=O)CC1CCC(=O)N1C)CC2 CCC(=O)CCC(=O)NCC1CCCCC1C(=O)NCCOCC(C)(C)C c1(CC(=O)NCC(CCCC)NC(=O)C(O)CCSC)c(C)cccc1Cl c1(CC(=O)NCC2CCN(C(C(C3CC3)OCC)=O)C2)ccc(OC)c(F)c1 C(=O)(C(F)C(C)(F)F)NCC(N1CCN(C(=O)CCc2ncc[nH]2)CC1)C C(CC(N)=O)(C(=O)NC(C)CCC1CC1)NC(C1C(C(C)C)CCO1)=O C1(NC(CC2CCN(C)C2=O)=O)CCCCCC1NC(=O)CN1CCCC1=O C1(NC(C(F)OC)=O)CCN(C(=O)CNC(=O)CC2CCCC2)C12CCC2 N1(C(c2cn(CCC)nc2)=O)CCC(CNC(C2CCC2C(F)(F)F)=O)C12CC2 c1(C(C(CC)NC(C2(F)CN(C(=O)OC(C)(C)C)C2)=O)=O)cc(C)ccc1C C1(NC(c2cc3ccccc3o2)=O)CCN(C(C2CC(F)(F)C2)=O)CCC1CO C(=O)(N=c1ccn(CC2CC2)[nH]1)C1(CNC(C2C(C)(CC)C2)=O)CCC1 C=CCC(C)(C)C(=O)N(C(C)CNC(=O)COCC(C)(C)C)C CC1CN(C(c2cccnc2)=O)CC1(C)CNC(=O)CSCc1ccccc1Cl C1(N=c2[nH]nc(C3CC3)o2)(CCNC(CCCCC#C)=O)CCC1 C#CC1(C(=O)NC(C)CC2CCOC2)CCN(C(c2ccc(C)cc2)=O)CC1 C1(OC)C2CC3CN(C(C4CCC5(CCCC5)O4)=O)C1C3C2 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ncc(Br)cc1C N1(C(COCC=C)=O)CCC(C2CCN(C(c3cnc(C)nc3C)=O)C2)C1 c1(C(=O)OC)ncc(C(=O)NC2CC2NC(C2CC2C2CCCO2)=O)s1 N12CCC1C#CC(=O)OC2=O.C(=O)(N=c1ccn(C2CCCC2)[nH]1)C(C)(C)C C1(CC(N2CCC(F)(CNC(=O)CCOCC(F)F)C2)=O)CN2CCN1CC2 C1(CNC(CC(=O)N(C)C)=O)CCC(CN(C(=O)CC2CCC(=O)NC2)C)CC1 c1(NC(CC2CC(NC(=O)CCOC(C(C)(C)C)=O)C2)=O)ccc(F)cc1F N1(CC2CN(C(C(C)OCC(C)C)=O)C2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(C(N2CCOCC(NC(c3nn(CC)nc3C)=O)C2)=O)cccc2c1OCC2 c1(CC)n[nH]c(=NCc2ccc(C3(CNC(=O)CCC(C)OC)CC3)c(F)c2)o1 C1(NC(C2CCN(C)C2=O)=O)CN(C(=O)Cc2cnns2)C2(CCCCCC2)C1 Cc1cc(-c2ccc(C(F)(F)F)nc2)c[nH]c1=NCc1ccc(Br)c(Cl)c1Cl c1(C(=O)OC)nnc(-c2cnn(-c3ncccn3)c2)c2ccccc12 Cc1cc(CC(N2CC(CN(C(=O)C(c3cccc(F)c3)(C)C)C)C2)=O)n(C)n1 C1(C(N(CCCCN(C(C2ON=C(CC)C2)=O)C)C)=O)CC2(CCOCC2)CO1 C1(NC(c2cn(CCC)nc2)c2nnnn2CCCOC)CC(F)(F)C12CCC2 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)ccc(S(=O)(=O)N2CCCC2)o1 C(=O)(C(C#N)=CCl)N(CCC(=O)OC(C)CNC(c1cccs1)=O)C C(=O)(C(O)C(C)(O)CC)NCC(C(C)(C)C)n1cc(COCCCOC)nn1 c1(C(=O)NCC2(NC(=O)Cc3cc[nH]n3)CCC2)ccc2c(n1)CCCN2 C1(CNC(C(CC)C)=O)CC12CCN(C(c1sc(Cl)cc1Cl)=O)CC2 C(=O)(N=c1nc2n([nH]1)CC(C(F)(F)F)CC2)NC(CCCN(C(=O)OC)CC)C C1(C(=O)NCC2(F)CC(NC(=O)CCF)C2)CC12CCOc1ccc(Cl)cc12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)CN(C(=O)COC2CCCC2)C(C)C1 N1(C(CCC(C)OC)=O)CCN(C(=O)COc2cccnc2)CCC1C C1(N(C(=O)C=Cc2ccc(Cl)s2)CC)CCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(SC)cccc(CC(=O)NCCCCNC(=O)C(F)(F)c2ccccc2)c1 Cc1cc(CNC(C2CSCCN2C(c2cc3ncsc3[nH]2)=O)=O)ccc1Br C(CC(C(=O)NCC(C)(C)CSC)NC(c1cncnc1)=O)OCC C(=O)(C1=NOC2(CCC2)C1)NCCCCCCC(=O)Nc1ccc(CC)nc1 CCCCC(CC)CCC(=O)NCC1(NC(=O)CC(C)F)CCCCC1 C1(NC(=O)CCF)CCN(C(C2(N3CCCCC3)CCCCC2)=O)CC1F N1(C(COCCOCC#C)=O)CCCC(NC(C2CCN(C)C2=O)=O)C1C CC(C)C1=NOC(C)(C(=O)NCCCCNC(=O)CCc2ccn(C)c2)C1 c1(-c2cn(CC(=O)NCCOCC(=O)O)nn2)cc(F)ccc1F C1(NC(=O)Cn2cncn2)CN(C(C23CCCC(CO2)C3)=O)CC12CC2 c1(C(N2C(CNC(c3cnn(CC)n3)=O)CC2)=O)cc(OC)ccn1 C#CCC(C(=O)NCCC(C)NC(C1CC(N(C)C)C1)=O)C1CC1 C1(C(N(CCCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)NC(=O)OC1C S(=O)(=O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC1CCCCN1C)NC C(C(=O)N1CCC(C(=O)NCC2(C(N)=O)CCCO2)O1)C1(CCC)CC1 N1(C(CC2C(OC)COCC2)=O)CCC2(CNC(c3cnns3)=O)CCCCC12 C12(C(N3CC4C(C)(C)C4C3)=O)COCC1CN(C(c1ccn[nH]c1=O)=O)C2 n1(CC(N2CCC(C(CNC(C3C(C)C3)=O)F)CC2)=O)c(=O)oc2ccccc12 Cc1ccc(C(=O)NC2CCN(C(=O)Cc3cnoc3)C(C)C2)c(O)n1 c1(C(C)C)nnc2n1CCN(C(=O)C=Cc1nc3ccccc3o1)C2C CC(C(C)C(=O)N(C)CC1CCC(C)CC1)NC(=O)C=Cc1cncn1C c1(OC)ccccc1COCCNC(=O)N(C)CC1CCCSC1 C(c1cccc2ccccc12)=CC(=O)NC1C(NC(c2cn(CC=C)nc2)=O)C1 c1(C(N2CC3CCC(O)C3C2)C(=O)NCCCSC)cc(F)c(F)cc1F CC(CO)C(C)NC(=O)CCN(C(=O)CSC(C)(C)C)C c1(Cc2cc(N)no2)ncccc1C(=O)O.O=C(C(F)(F)F)N1CCN1 C1(NC(c2ccc(C)cc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C N1(C(c2c(C)[nH]c(=NCC)s2)=O)CCCC2CN(C(=O)C(F)C(C)(C)O)CCC12 c1(NC(c2nc(-c3c(OC4CC4)ccc(C)c3)sc2)=O)cccc(F)c1[N+](=O)[O-] C1(C(=O)NCC(C(=O)N(CCN2CC=CC2)CC)C)CCCC(=O)C1 Cc1ccn2nc(C(=O)NCCCCC(C)NC(=O)CCCCC3CC3)nc2n1 N1(C(c2cnc(C)nc2)=O)CCC(C)(C)C(CNC(=O)CN(C(=O)C(C)C)C)C1 NS(=O)(=O)CCCC(=O)N1CCCCC(CNC(=O)Cc2ccc(Cl)nc2)C1 c1(C(=O)NCCC2CC(NC(c3c(C)cn(C)c3)=O)C2)cc2c(s1)COCC2 C1(C(N2C(CNC(c3cccc(=S)n3O)=O)CC2)=O)CCC2CCCCC2C1 c1(C(N2CCCC(NC(C=C(CC)CC)=O)CC2)=O)ccc2snnc2c1 CCC(C(=O)N1CC(COC)(NC(c2cnn(C)n2)=O)C1)n1ccnc1 CCCCC(C(=O)NCCCN1CCCC1C)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCC(F)(F)F)N1CC2C(NC(C3CCC34CCOCC4)=O)(C2)C1 c1(CNC(=O)Nc2c(C)n(CCC(C)C)nc2)cccc2c1OCCO2 CC1(C2CC2C(=O)NCC2CCOC2C(N2CC3CC3C3CC23)=O)COC1 Cc1cc(Cl)cc(C)c1C(N1C2CCC1CC(NC(=O)C=CCO)C2)=O N1(C(CC(C)(C)C)C(=O)NCCCC2CC2)CCSC2(CCOCC2)C1 O=C(CCCN1CCOCC1)NC1CCC1CNC(C1(C(F)(F)F)CC(O)C1)=O C1(C(C)C)CCC(C(=O)N(C)CC2CCOCC2)N1C(C1CCN1C(C)(C)C)=O c1(CCC)c(C(=O)NC2CC2NC(=O)C(C)c2ccco2)cnn1CCO C1(NC(c2c(CC)occ2)=O)CS(=O)(=O)CC1NC(c1ccnn1CC#N)=O N1(C(C(CC)N2CCCC2=O)=O)CC2CCC2(CNC(=O)C(=O)C(C)(C)C)C1 c1(CC(N2C(CNC(CSS(C)(=O)=O)=O)CC2)=O)cncc(C#N)c1 C1(C)(CNC(C2(SC)CC2)=O)CCC(NC(=O)CCc2cccs2)C1 N1(CC(N2C(C(C)(C)CNC(=O)CC3CCC(O)C3)CCC2)=O)CC2CCC1C2 N1(C(C(=O)OC)C)CCN(CCCNC(c2csc(Cl)c2Br)=O)CC1 Cc1nc(Cl)ccc1CC(=O)NCCC1CC(NC(c2cccc(F)c2)=O)C1 c1(N2CCC(CCOC)C2)nc2c(c(=NCC(C)(C)N3CCCC3)[nH]1)COCC2 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCCCN(C(c2cc(N)ccc2F)=O)C1 S(=O)(=O)(c1ccc2[nH]c(=NCC3CC(O)C3)sc2c1)N1CC(C(C)C)SCC1 c1(CNC(C2CC(OC)C2)=O)c[nH]nc1C1CCN(C(c2c[nH]c(=N)s2)=O)C1 c1(NC(C2CC(NCC(F)(F)F)C3CC23)=O)cc(Br)ccc1OC(F)F C(=O)(C1CCCc2nncn21)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C1 C1(N(C(CC(CCC)C)=O)C)CCC2CN(C(=O)CN(C)C(N)=O)CC12 N1(C(C(c2ccc(F)cc2)C)=O)CCC(CF)(NC(c2cc(Cl)ns2)=O)C1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1sc3ncccc3c1Cl)=O)CCO2 C(C(=O)N(OC)C1CCS(=O)(=O)CC1)Cc1nn(CC)nc1Br N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC(CNC(=O)CC3CC3)C2C1 c1(CNC(C2(CNC(COCC)=O)CC2)=O)ccc(O)c(OC)c1 C(=O)(C(O)CCCNC(C12CCC(CC1F)C2)=O)NCC(C1CCCC1)OC C(=O)(CCC(C)(C)N(C)C)NC(CNC(CCCC#C)=O)(C)C1CCC1 N1(C(C2=NOC(C)C2)=O)CC2CCC1CN2C(=O)COCC1CCOCC1 C#CCC(CC(=O)N1CCC(O)(C(C)C)C1)NC(=O)Cc1sccc1C C(=O)(C(C)C(C)(C)C)N1CC(OC)C(NC(=O)CCn2cnccc2=O)C1 N1(C(C(=O)Nc2ccc(C)cc2Cl)C)CCS(=O)(=O)C(CNC(=O)CC2CC2)C1 c1(NC(C(C)OC(c2cccc(C3(C)CC3)c2)=O)=O)cc(C(F)(F)F)ccc1F C1(C)(C(N(CC)Cc2cccnc2)=O)CCCN(c2cc(OC)nc(C)n2)C1 c1(NC(C2N(C(c3cncc(OC)c3)=O)CC(C)C2)=O)ccc(Br)c(Cl)c1C c1(CC(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)CCOC)cnc(Cl)cc1C Cc1cc(C(N2CCC(NC(=O)CCc3ccn(C)n3)CC2C)=O)cc(C)c1Cl C1(C)(NC(C(CCC)O)=O)CCCN(CC(=O)Nc2cccc(C(F)(F)F)c2)C1 CCC(CC)CC(=O)NC(c1ccccc1F)CNC(=O)C(COC)CC CC(C)(C#N)C(=O)NCc1ccccc1CNC(c1ncccc1N(C)C)=O c1(NC(=O)OC(C)(C)C)cccc(CF)c1.c12ccc([nH]1)CCC(=O)N2 C1(CNC(C=C(C)C(F)F)=O)CC12CCN(C(=O)CN(C)CCO)CC2 c1(C(N(C(C)CNC(C2CCC(C)CC2)=O)CC)=O)nc(C(C)C)ncc1Cl N1(C(CC(C=C)CC)=O)CCCCC12CC(NC(=O)COC1CCC1)C2 C1(C(N(C)Cc2c(C)nsc2)=O)CC(NC(c2cncs2)=O)CCO1 C(CC(=O)NCC1CCCSC1)(C(C)(C)C)NC(c1c(C)nc(C)o1)=O Cc1ccc(C=CC(=O)NC2CCC(CCNC(c3ccc(C)nc3)=O)C2)nc1 N1(C(CN(C(C)C)CC)=O)CCCC(CNC(C2CCN(C(=O)NC)C2)=O)C1 C1(O)(CN)CN(C(C2CC(C(F)F)C2)=O)C1 c1(-c2cn(CCCC(=O)NC(C)CC3CC=CCC3)nn2)nccnc1C(=O)O C1(C(N(C2CCN(C(=O)CC3CCCOC3)C2)CCO)=O)COC2CC1C2 Brc1csc2c(Nc3n[nH]c4c3CN(Cc3ccc(C5CC5)cc3)C4)ncnc12 CCCC(C(=O)NCCN(CCC)C(C1CC2(C1)CC2F)=O)C(C)C C(=O)(CCC(C)NC(=O)C=Cc1ccnn1C)N(C(CCCC)C)C C1(NC(C=Cc2n(C)cnc2)=O)CCCC12CN(C(C1NC(=O)OC1C)=O)C2 c1(OC)cc(C(=O)NC2CCN(c3nccc(C(F)(F)F)n3)C(C)C2)cc(Cl)c1 C#Cc1ccc(CC(=O)NCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)c(F)c1 c1(OC)cc(NC(=O)C=CC(C)NC(=O)COCC2CCOC2)on1 C1(C(=O)NC(C2CN(C(C3(C4CCCCC4)CC3)=O)C2)C)CN2CCCN1CC2 C1(C(=O)NC(C)(C)CCNC(c2ccccc2CC#N)=O)CCc2ccnn2C1 C1(C(C)C)CN(C(c2ccc(O)nn2)=O)CCN1C(=O)Cc1nc[nH]n1 O=S(=O)(c1ccccc1OC(F)F)N1Cc2ccc(Br)cc2C1 CS(=O)(=O)CCc1cn(CC2CCCO2)nn1.c1(CN)nnnn1Cc1cccs1 c1(SC(C)(C)C)ccccc1C(=O)NC1CCC(Cn2cc(C(C)OC)nn2)C1 Cc1nn(C)cc1NC(=O)NCC(N1CCN(C)CC1)C Cc1cc(O)c(F)cc1NC(C1(CNC(=O)C(C)CO)CCOCC1)=O c1(C(=O)NC(C(C)NC(C(C)Cc2cnc[nH]2)=O)(C)C)cc(Cl)c(F)cc1O c1(NCC2(CO)CC(C)C2)cc(Br)ccc1S(=O)(=O)N1CCC2CC12 C(C(C)C(C)C(=O)NC1(CNC(=O)CSC)CCOCC1)OC C12(C(=O)NCCN(C(=O)COCc3nccn3C)CCC)CSCC1C2(F)F c1(CC(CNC(=O)C(C2CCCC2)SC)NC(C(F)OC)=O)ccccc1 c1(C(N2CCC(c3cn(Cc4cnn[nH]4)nn3)CC2)=O)ncccc1Br C1(CC)CCC(C)CN1C(=O)C(CC(F)F)N(C)C(c1cc(C#N)[nH]c1C)=O N1(C(C(=O)Nc2c(SCC)nccc2)=O)CC2(NC(=O)C(F)(F)F)CCC1CC2 c1(NC(C2N(C(C(C)C)=O)CCCC2)C)nccc(S(C)(=O)=O)n1 N1(C(C(=O)N(CC(C)OC(C)(C)C)C)=O)CC2CCCC12 Cc1nc(Cl)sc1C(=O)N(Cc1ccc(Cl)cc1)Cc1ccsc1 c1(CC(=O)NC2(CN(C)C(C3CCCCC3(C)C)=O)CC2)cc(O)nc(O)n1 N1(C(c2cc(C)c(O)nc2)=O)CCCC2(NC(c3cc(Br)co3)=O)CC2C1 N1(C(C(C(C)C)OC)=O)CC(C(=O)NC2CSC2)C(C)(C)C1 Cc1ccc(F)c(CNC(c2cncc(CNC3(C)CC3)c2)=O)c1 N1(C(C=CC(=O)OCC)=O)CCC(C2CC2)C1CNC(C1CC2C=CC1CC2)=O c1(C(C)C)ncc(C(N2CCC(NC(c3ccn(C4CCC4)n3)=O)CC2)=O)cn1 N1(C(C(CNC(C)=O)(C)C)=O)C2CCC1CC(N(C(=O)CN1CCCC1=O)C)C2 C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(CC(=O)NC)C)(COC)C=CC1 C12(C(N(CCCC=C)CC)=O)COCC1CN(C(c1ccc(C(N)=O)cc1)=O)C2 C1(OC)C(CN=c2[nH]nc(-c3ccccn3)o2)CCCN1C(C)=O CC1CCC(CO)CN1C(=O)NCc1csc(C(=O)O)n1 N1(C(CCC#C)=O)CCCC12CN(S(=O)(=O)CCC(=O)OCC)C2 C=CCC(C(=O)NCCCN1CCN(C(=O)CC2CCCCC2O)CC1)OC C1(CN(C(c2cnc(CC)s2)=O)C)C2CN(C(c3ccn(CCO)c3C)=O)CC12 CC(C)C(C)C(=O)N1CC(C)C1C(=O)NCCc1cocn1 N1(C(CCCCCC(C)C)=O)CCC2(CC1)CC(C)N(C(c1csc(Cl)n1)=O)C2 CCCC(CC)CCC(=O)NC1CC(NC(=O)CC(C)C2CC2)C1 C1(CC(=O)NCC2(Nc3nc(C)nc(O)c3)CC2)COc2ccccc2O1 Cc1cc(C(N2CC(C3CN(C(=O)C4=CCC4)C3)C2)=O)c(C)cc1Br C12(CNC(C3C(C)(C)C3)=O)CC(CCO1)N(C(C1CC3C=CC1O3)=O)C2 C1(O)(C(C)NC(CC(=C)C)=O)CCN(C(=O)CSCCN(C)C)CC1 C12(C(N3CC(C)(NC(c4n(C(CC)C)ncc4)=O)C3)=O)CCC(CC1=O)C2 C1(C(=O)NC(c2nnc(S)n2C)C)CC(C(=O)NC2CC(N(C)C)C2)=NO1 C12CCCCN(C1)C2=O.C1(CNC(c2c(CC)cco2)=O)CCCC1(C)C c1(C(=O)NC2C=CCC(C(=O)NC(CCCC=C)C)C2)c(C#N)ncn1C C(=O)(C(C(C)(C)C)N1CCCC1=O)N(C)CCc1cn(C2CCOCC2)nn1 c1(Cn2cc(CN3CC(OC)CC34CCC4)nn2)c(F)cc(Br)cc1F C1(CS(=O)(=O)NC(c2cccc(C)c2)CN(C)C)CC12CCCc1ccccc12 C1(O)(CNC(CSCC(N)=O)=O)CCCN(C(c2cncnc2C2CC2)=O)C1 C1(C(=O)NCC2(NC(c3[nH]cc(C)c3)=O)CCCC2)OC2CCC1CC2 c1(CN(C(C(=O)NC(C2CCOC2)C)=O)C)cnc(C(F)(F)F)s1 c1(OC)ncc(C(=O)NC2CCCN(C(C3CCCSC3)=O)C2)c(C)n1 c1(NC(C2(C(=O)OC)CCNC2)=O)ncnc2cc(C(C)(C)C)sc12 c1(NC(CCC2(NC(C3CC(OC)C3)=O)CCCC2)=O)ccccc1N=[N+]=[N-] Cn1nc(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(C)CC2(Cl)Cl)c2c1CCC2 C(=O)(C(C)(C)CNC(C1CCC(NC(C2CCCN2C)=O)C1)=O)NC C1(C(=O)NCC2(C)CSC2)CCCC(NC(c2nnsc2N)=O)C1 c1(COC)ccc(C(=O)NCC2(F)CN(C(c3ncoc3C3CC3)=O)C2)s1 C1(NC(C2(CC)CCNC2=O)=O)CCC2CC1CN2C(=O)Cn1cncn1 C1(CC(=O)NCCOCCNC(=O)CCC2OCCO2)CCCC(C(F)(F)F)O1 c1(C(=O)NCC2CCN(Cc3cc(Br)cs3)C2)cnn2cccc(F)c12 C12(NC(c3c(C)n[nH]c3)=O)CCCN(C(c3c(Cl)csc3Cl)=O)CC1C2 c1(SC)cc(C(N2CCCC2CCC(=O)NCC(C)(C)C2CCCO2)=O)co1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C C(=O)(C1=CS(=O)CCC1)NCCCCNC(CC(C(C)C)C)=O C1(N(C(=O)CC(C2CC2)C2CC2)C)CN(C(=O)CC2CC(F)(F)C2)CC1F N=c1[nH]c(CSCC(=O)NCC2CCC(NC(=O)C(O)C3CC3)C2)cs1 C(C(C)(C)C(=O)N1CC(C(=O)NC2C3CCCC23)C(C)C1)OC(C)C CC(CCCCNC(=O)CC1CC1(Cl)Cl)NC(C1CC(O)(C(F)(F)F)C1)=O c1(C(=O)NC2C(NC(CCc3nnc(CC)o3)=O)CCCC2)n[nH]cc1[N+](=O)[O-] c1(-c2c(CNC(N3CC(CC)OCCC3)=O)ccc(F)c2)ccc(C)cc1NC CCCC(C)(CCC)C(=O)NCC(O)CC(=O)NCC1Cc2ccccc21 CC1(C)CCC(C(=O)NC2CC(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)C1 CCCC(C(=O)NCCN(c1nccc(C(=O)OC)n1)CCOC)NC(N)=O c1(-c2ccc(CNCCCN3CCC(N(C)C)CC3)nc2)nc2ccccc2s1 C1(NC(C(C)CN(C)C)=O)CCN(CCNC(C2C3CCC2CC3)=O)CC1 c1(CCC(=O)NC2CCC(CCN(C(C(C)(C)C)=O)C3CC3)C2)ccnc(Cl)c1 C1(OC)CC(NC(=O)CCc2ccccc2)CN(C(C2CC23CCC3)=O)C1 Cc1cccn2nc(C(=O)NC3CCN(C(c4cncnc4)=O)C(C)C3)cc12 N1(C(c2cccc(C=CC(F)(F)F)c2)=O)CCC2CCC(F)(F)CC2C1 N1(C(=O)Nc2c(OCC#C)cccc2)CCc2[nH]c3ccc(F)cc3c2C1 c1(C(=O)Nc2cncc(C)n2)cnc2ccc(-c3ccc(F)c(C#N)c3F)cn12 c1(-n2c(C(O)C3CC3)nc(CC)n2)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(c2c(C)c[nH]n2)=O)CCC(NC(=O)C(C)NC(c2cccs2)=O)C1(C)C C1(OC)CN2CCCC2(C(=O)NCCC2(CNc3c(SC)ncnc3Cl)CC2)C1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2(CCCCN(C(=O)C3=CCCCO3)C2)C1 N1(C(CCSCCCC)=O)C(CNC(=O)CCc2csnn2)CC2CC12 CC(CCC(C)(C)C)C(=O)NC1CCCC(CC(=O)Nc2cc(O)ccc2F)C1 CC(C)C(O)CC(=O)N1CC(C)(C)CC1CC(=O)NCc1nn(C)c(=O)n1C c1(N2C(C)CN(C(=O)CC(=O)NCC(F)(F)F)CC2)nc2ccc(F)cc2o1 CCCC(C(O)C(=O)NC(C)(CC)CCO)NC(=O)C(O)CCN(C)C C1(NC(C#C)=O)C(C)CCCN1C(=O)C=CCOC c1(C(N(C(C)CCNC(=O)C(N2CCNC2=O)C)C)=O)ccc2nc(S)[nH]c2c1 c1(C(N2C(CNC(CSCC)=O)C(C)(C)CCC2)=O)cnc2n1CCCC2C C1(CNC(C(C2CC2)NC(C2C3(CC3)C23CC3)=O)=O)CCCC2(CC2)C1 c12cc(N(C)C)cc(c1)NC(=O)N2.Cc1n[nH]cc1CCOC(C)(C)C C1(C)(OC)CC(NC(=O)C(CCOC)NC(c2cc(C)nc(O)c2)=O)C1(C)C C1(=O)C2=CCN(C2)CC2CC(C2)N1C.C(=O)(CCC1CCC1)N.C1CC1 C1(CC(N2C(C=C)CC2)=O)CCN(C(C2CC(O)C(F)C2)=O)C1(C)C C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCNC(c1cncc(C=C)c1)=O)C C=C(CNC(C12CCCC1C2)=O)CCNC(=O)C(c1ccccc1)N(C)C c1(NC(C2(OC)CCSC2)=O)cc(NC(c2ccc[n+]([O-])c2)=O)ccc1C C1(CC(=O)NC(C)CN(C)C(C2CCN(C3CCCCC3)C2)=O)C(C)(C)C1(C)C CC1CC(C)CCN(C(C2C=CCN(C(c3ccnnc3O)=O)C2)=O)C1 c1(C(=O)Nc2c(C(=O)OC)c(C)cs2)ccc(-c2ccc(F)cc2)nc1C c1(CC)c[nH]cc1C(=O)NCC1OCCC1C(=O)NCc1ccsc1C C1(CNC(COCCCCC)=O)N(C(=O)CC(C)OC)CCCC1(C)C CC(C(=O)N1CC2CC(NC(=O)Cc3ccccc3Br)C1C2)C(C)(F)F CCCCC(C(=O)NC)NC(C12CC(CN1C(=O)CC1CC(C)(C)CO1)C2)=O C1(O)(CNC(c2c(CC)c[nH]n2)=O)CCCN(C(c2cc(OC)ccn2)=O)CC1 c1(OCC(=O)NCC(CNC(C(C)CC2CC2)=O)(C)C)ccccc1F n1(CC)ccc(=NC(=O)CCC2CCN(C(=O)Nc3ccc(F)c(F)c3)CC2)[nH]1 Cc1cccc(CCN(C2CCOC(c3ccncc3)C2)C)c1 N1(C(CCOCCNC(C(C)(C)OC)=O)=O)CC(=O)NC(C(C)C)C1 C=CCCC(F)(F)C(=O)N1CC2(CCCC2NC(=O)C(c2ccc(F)cc2)F)C1 N1(C(C2CC(C)SCC2)=O)CC2CC(C1)C2NC(c1c[nH]nc1C1CCOC1)=O S(=O)(=O)(c1ccccc1Cl)NC1C(NC(Cc2ccc(C)nc2)=O)C2CCC1C2 c1(C(=O)NCC2CCC(NC(c3c(SC)snn3)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C1CCCc2c[nH]nc21)N(C1CCN(C(=O)CSCCOC)CC1)CCC CC1=C(C(=O)N2CC3CC3C2C(=O)NCCCN(C)C)CCC1 C=CC1(O)CCN(C(C2CCCC(NC(=O)CCCCNC(N)=O)C2)=O)C1 CC1CCC(NC(C23CC(C2)C3)=O)CN1C(C1CCC(C(N)=O)C1)=O c1(C(=O)NCCC2(O)CN(C(CN(C)C)=O)C2)nc(C2CC2)n2ccccc12 c1(OC)ccccc1C.C1(C(=O)S)(NC(=O)C(C)n2cccn2)CCC1 O=C1CC(C(=O)NC(C2CC2)C2CC2)N(C(C2CC=CC2)=O)C1 C1(Cn2cc(-c3c(C)ccs3)nn2)CCCN(C(c2ccccc2Cl)=O)C1 N1(C(C(C)OCC=C)=O)C2CC1CN(Cc1ccc(CC)cc1)C2 C1(CNC(CN(C)C)=O)CC2CCC(C1)N2C(=O)CSCc1ccccn1 c1(C(N2CC(C)(CNC(CSCC)=O)OCC2)=O)cc2nccnc2cc1F C#CCCCCCC(=O)NC1CCC(C)(CNC(=O)CCc2cc(OC)no2)C1 C1(CNC(C(CC#C)C)=O)CC2CCC1N2C(c1cc(C)cc(F)c1)=O N1(c2ncc(C)cn2)CCC2(NC(=O)CCC3CCCCCC3)CCCC12 C=C=CCCC(=O)NC(C)CN(C(=O)CCC(C)c1ccc(Br)cc1)C c1(CC(N2CC(CNC(C3CCC(COC)C3)=O)C(O)C2)=O)noc(C)c1C#N CC(C)(C)[Si](C)(C)OC1CCCCC1CCCOC(=O)Cc1c(O)ncnc1O C(=O)(C1=C(C#N)CCC1)NCCn1cc(C(N2C3CN(C)C(C3)C2)=O)nc1 C1(NC(c2ccc(F)s2)=O)CN(C(c2cc3c(o2)CCCC3)=O)CC2CCCC12 Cc1cc(F)ccc1C(N1CC(C)(C)CC1CC(=O)NC(c1ccnn1C)C)=O C(C)(c1cccs1)=CC(=O)NC(C1CN(C(C(=O)N(CC)CC)C)C1)C Cc1cc(O)ncc1C(N1C2CCC(C2)C1C(=O)NCCC1(C)CCCO1)=O N1(C(CCCC#CC)=O)CCC2(C1)CN(C(C13CC(C1)C(C)O3)=O)CC(C)O2 Cc1n[nH]c(C)c1CC(N1CCCC(C(C)C(=O)N(C)CCO)C1)=O Cc1cc(=NC(CNC2(C(N)=O)CC2)CO)nc(-c2cccs2)[nH]1 Cc1cnnc(O)c1C(=O)NCCC1CC(F)(F)CN1C(c1ccnnc1O)=O CCC(CC(=O)N1CCC=C(C(=O)NCc2ncoc2C(C)C)C1)C(F)F N1(C(c2c(OC)cccc2)=O)CCN(C(=O)Cc2cccn2C)C(CF)C1 c1(C(=O)NCC2CCCN2C(C2CC23CCCC3)=O)n[nH]c2cc(Cl)ccc12 CC(C)CCCC(C)C(=O)N1CCC(O)(CN(C(=O)CC(=O)N(C)C)C)C1 Cc1nc(O)nc(C)c1CC(N1CCCN(C(C2OC3CCC2CC3)=O)CC1)=O c1(C(N(C(CNC(CC(CC)CC)=O)C)C)=O)ccc2cnnc(O)c2c1 Brc1ccc(-c2ccc(CN(CCCSC3CCCO3)C3CC3)s2)cc1 c1(C(N)=O)cncc(C(=O)N(C2CCCC2O)CCNC(=O)C=CC2CCCC2)c1 CC(C)C1=CCC(C(N2CC(C)N(C(c3cnn4c3OCC4)=O)CC2C)=O)CC1 Cc1cc(C(N2CC(C)CCC2C(=O)NCCC(F)=C(F)F)=O)ccc1C#N N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(C)(NC(c2nn(C)cc2Cl)=O)C1 C=CCC(C(=O)NCCC1CCCN1C(=O)C(=O)Nc1ncc[nH]1)N(C)C C=CCCCCCC(=O)NC1CN(C(=O)Cc2cncnc2O)CC1C c1(C(=O)NCC23CC(CNC(C(CC)O)=O)(OC2)C3)cccc(F)c1F N1(CCNC(c2c(NC)scn2)=O)CCN(C(C2(C)CCC(=O)C2)=O)CC1 C1(NC(C2C(C(=O)OCC)C2)=O)CN(C)CC1CC.c12n[nH]c(n1)CNC2=O c1(C(N2CC(C(C)NC(c3c(C)c[nH]n3)=O)C2)=O)cc2c(Br)cccc2[nH]1 CC(C)(CC(=O)NCC1CCCC(NC(c2cc(=O)cc[nH]2)=O)C1)CC(F)F c1(CCNC(C(N2C(C)COCC2)=O)=O)cc(C#N)ccc1I C1(C(=O)NC2(CSC)CC2)CC(O)CCN1C(c1cnnc(C)c1)=O CC1CCN(C(=O)CCS(C)(=O)=O)CCN1C(=O)C(C)CC1CCCCC1 C1(N(C(CN(CCOC)C)=O)C)CCCN(C(c2ccnn2C2CC2(F)F)=O)C1 C1(C(N(C(CNC(c2nc(C)[nH]n2)=O)C2CC2)C)=O)CC=CCC1C CC(C)C(N=c1[nH]c(Cl)ncc1Cl)C(C)NC(=O)OC(C)(C)C c1(C(C)=O)cc(C(=O)NC(COC)C(=O)NC2(c3n[nH]c(C)n3)CC2)no1 c1(CC)ccc(NC(c2cccc(OCC(F)(F)F)c2)=O)cc1S(N)(=O)=O C1(C)(C(N2C(CNC(C(CC)(F)F)=O)CCCC2)=O)CCCNC1=O C1(N(C(=O)C=C(Cl)Cl)CC2N(C(c3c(CC)nns3)=O)CCC2)CCC(O)CC1 Cc1cc(C(F)(F)F)ncc1C(=O)NCC=CCN(C(=O)C1=CCCC1C)CC c12ccc(cc1)SC2.C1(N(C)C2CC2)(CNC(=O)C(F)C2CCC2)CCC1 C123CCC(CC1)(OC2)CNC(=O)CCc1c(ccc(F)c1)C(=O)N3.C1(CO)CC1 N1(C(Cc2cc(C)ncc2)=O)CCOC2(CCN(C(C3CC4C=CC3C4)=O)C2)C1 c1(NC(CCC)CCCNC(C2(CO)CC2)=O)nc(O)n(C)c(=O)c1[N+](=O)[O-] N1(CCNC(C2CC3CCC2(C(F)(F)F)C3)=O)CCCC(C2CCCCC2)C1 c1(C(N(C(C)CN(C(=O)C(O)C2CCC2)C)C)=O)cccc(-c2ccco2)c1 c1(NC(C)=O)cnccc1C(N1CCCC1(C)CNC(=O)Cc1cc(C)cs1)=O c1(C(N2CCC(F)(C(=O)NCc3cccc(Br)c3)C2)=O)ccc(O)nc1 Cc1ncnc(C)c1C(=O)NCC1(NC(=O)CC2(O)CCOC2)CCCC1 CC(C)(CNC(=O)C(O)CC(N)=O)CC(=O)N1CC2C(C1)C2(F)F C1(NC(C(C)=CC)=O)CC2(C1)CC(CNC(=O)C(c1cccn1C)=O)C2 C1(C(=O)NCC2C(NC(Cc3c(C)cccc3C)=O)C2)CCn2nccc2C1 C(=O)(C(C)CC(C)C)NCC(C)(CNC(=O)C(c1c(C)n[nH]c1C)C)OC c1(NC(C(C)O)COC(C)(C)C)ccnc2c1CCO2 C1(NC(c2ccc(NCCOC)cc2)=O)CC2CC1N(C(=O)C(C)(C)CF)C2 C1(C(=O)NCCNC(C2(O)CCSC2)=O)(OC)CCCCCC1.C(C)(C)(C)NC(=O)O N1(C(CC2(COC)CC2)=O)CC2COCCC2(NC(c2csc([N+](=O)[O-])c2)=O)C1 C1(OC)CC(CNC(=O)CCCOc2ccccc2F)N(C(c2ccc[nH]2)=O)C1 NS(=O)(=O)c1cc(C(=O)NC2CC23CC(NC(C2CCC(F)(F)C2)=O)C3)co1 N1(C(C2CC(C)(O)C2)=O)CCC(N2CCN(C(C3CCC4CC4C3)=O)CC2)CC1 C1(C(=O)Nc2cccc(C(C)C)c2)CNC(=O)CN1C(=O)CCc1ccsc1 Cc1c(NCCF)nc[nH]c1=NCC(CC)(c1ccc(F)cc1)c1ccccc1 c1(OC)ccnc(N(C)CCN(C)C(C2CCN(Cc3ccccc3)CC2)=O)n1 N1(C(C2(C)COC2)=O)CCC12CN(C(=O)C(O)Cc1ccccn1)C2 N1(C(c2c(Nc3nc(C)c(C(=O)O)s3)ncnc2)=O)CCc2c(F)cccc2C1 N1(C(c2c(CC)nns2)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C(C)C1 Cc1[nH]nc(C(=O)NC2CCCC2CNC(c2sccc2Br)=O)c1C c1(C(N2CCC(CNC(C3CC4CC4C3)=O)C2)=O)c(Cl)cncc1Br c1(C(=O)NCC2(F)CC(NC(C=CC(C)(C)SC)=O)C2)cc(Cl)ncc1NC N1(C(C2OCCOC23CCC3)=O)CCC(C2CN(C(C3(F)CCC3)=O)C2)CC1 Cc1nc(C(C)C)nc(O)c1C(N1CCN(C(C2C3CCCC23)=O)CC1)=O c1(C(C)NC(=O)NCCc2cc(OC)c(C)cc2)cc(Cl)cc(Cl)c1O C1(NC(c2c(C)coc2)=O)CCCCC1CC(N1CCC(CC2CC2)C1)=O C=CCCC(C(=O)NC1CCOC(C)C1)NC(=O)CCC(C)(C)C c1(C(N(CCCN(C(C2C(CCOC)C2)=O)C)C)=O)ccn(-c2cccnc2)n1 C1(NC(C(CCNC(C2C(C)CC2)=O)(C)C)=O)CCC(C2CC2)CC1 c1(OC)cc(F)c(Sc2ccc(C(N3CC4CC(C3)C4O)=O)cc2)cc1F.O CC1OC(C)C(C)C1C(=O)NCC(C)CNC(C1CC(O)(C(F)(F)F)C1)=O c1(C(C)C(=O)NC2(C)CCN(C(=O)Cc3ccoc3)C2)ccc(C#N)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC1CC(NC(C(COC)C)=O)C1 C(CC(C(=O)NCC12CC1CN(C(=O)COCC1CCC1)C2)NC=O)SC C=CCC1C(=O)N1CC.C(C)(C(=O)NOCC1CC1)NC(C)=O C1(NC(c2cccc(CN(C)C)c2)=O)CCN(C(=O)COC2CCCC2)C12CC2 C(=O)(CC(C(F)F)CC(CC)NC(C)=O)NC(COC)C1CC1 Cc1ncncc1N(C(c1ncoc1C)C(=O)NCC1CCCO1)C C(=O)(CS(=O)(=O)CC)N1CC(C(=O)N(C)Cc2ccccn2)(SC)C1 CCCCC(CNC(=O)CCc1ccc(N(C)C)cc1)NC(c1ccnn1C)=O C1(F)(CNC(C2(C(=O)NC)CCC2)=O)CC(CNC(=O)C(C)COC)C1 Cc1ccnc2c(C(N3CC(C)CCC3CNC(=O)C(C)(C)C(C)C)=O)cnn12 Cc1cc(F)cc(C(=O)NC2CCC2NC(c2c[nH]nc2[N+](=O)[O-])=O)c1N Cc1cc(C(=O)NCCC(C)NC(C2CC2C(N)=O)=O)c(C)n1NC(N)=O CC(CN=C(NCC1CCCO1)NCC1CC2CCC1CC2)OC(F)F c1(C(N2CC(SC)C(NC(=O)C(C)(C)SC)C2)=O)ccc2ncn(C)c(=O)c2c1 c1(C(N(CCN(C)C(c2cc(Br)cnc2N)=O)C)=O)cc([N+](=O)[O-])nn1C c1(NC(C2C(CC)CN(C(=O)CC(C)SC)C2)=O)cc(CO)cc(F)c1 c1(OCC)cc(C(=O)NCCN(CCOC)C(C2CCC(C)C2)=O)ccc1O C1(C)(C(N2CCC(CCC(C)(C)C)C2)C(=O)NCCSC)CCC(=O)NC1 C(C(CCC)C(=O)NCC(C)(C)F)NC(COC1(C#C)COC1)=O C1(NC(C(C)OC(N)=O)=O)CCCC1Cn1cc(C(C)(C)N(C)C)nn1.C1CO1 c1(C(N2CC(NC(CC3(COC)CC3)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 C1(CC(=O)N(C2CN(C(CCCNC(=O)OC)=O)C2)C)CCCCC1F C(=O)(C1CCCc2nn(C)cc21)N(C)CCNC(=O)Cc1cnn(C)c1 N1(C(c2ccc(C(C)C)cc2)C(=O)NCCSC)CCC(C)C(CO)C1 CCCCC(=O)C(=O)N1CC(CC(F)C(=O)N(CCC(C)(C)C)C)C1 CC1(c2ccccc2)CCN(C(=O)C(N2CCOC(C3(N)CC3)C2)=O)C1 CCCC(C(=O)N1CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1)NC(N)=O C=C(C)CCC(C)N(CC(=O)NCC(c1ccc(Cl)cc1)=O)C C(CN=c1c(C(C)=O)c[nH]cc1C)OC.C1CO1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C#N)C2)=O)C2CCCC2(C)C1 c1(NCC(CC(C)C)N(C)C)[nH]c(=NC2C3CC(Cl)CC3C2)nc2sccc12 c1(C(C)=O)c(CCC(=O)N2CC(NC(C3CCC(C)C3)=O)C2)c[nH]c1C N1(C(C=CC)=O)CCN(C(c2ccccc2Br)=O)CC1c1cn[nH]c1 N1(C(C(CC)NC(N)=O)=O)CCC2(CC(C(N3CC(COC(C)=O)C3)=O)C2)C1 c1(SCC(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)ccc(C(F)(F)F)cn1 C(=O)(CCCC(F)(F)F)N1C(CNC(CC(C)NC(N)=O)=O)CCC1 c1(C(=O)NCCC2CC(NC(c3cc(OC)n[nH]3)=O)C2)nn(C)cc1Cl CC1=NN(C)C(=O)C1CC(N1CC=CC1CNC(C1(CC2CC2)CC1)=O)=O C=CC(C(=O)N1CSCC1C(=O)NCC=C=C)OC C(CCCCCNC(C1CCCC(=O)O1)=O)N(C(CC1N(C(C)C)CCC1)=O)C c1(OC)cc(C(N2CCC(CO)C(NC(=O)C(F)=CC3CC3)C2)=O)ccc1F CC1CN(C(=O)C=CC(F)(F)F)CCN1C(c1cccn(CC(F)(F)F)c1=O)=O C1(N(C(COCCC#C)=O)C)CC2CC1N(C(=O)C(C)(C)CCSC)C2 N1(CCC(CC)C)CC=C(CCNC(c2cc3oc(C(=O)OC)cc3[nH]2)=O)CC1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2ccsc2NCC)=O)C12CC2 c1(N(C2CC3CC2CN3)C(C(CC)NC)=O)ncc(OC(F)(F)F)cc1Br C1(NC(CN(C)CCO)=O)C2CC3CN(C(=O)CCCCN4CCCC4)C1C3C2 Cc1ccc(Cl)cc1C(=O)NCC1C(C)CCN1C(C1CN(S(C)(=O)=O)C1)=O Cc1cccc2nc(NC3(C(N)=O)CCCN(C(=O)CC(=O)N(C)C)C3)oc12 Cc1cnc(C)c(C(=O)NC(C)CC2CN(C(=O)C=Cc3cn(C)cn3)C2)c1 C1(NC(C(C=C)(C)C)=O)CC2CCC(C1C)N2C(=O)CCc1nnc(C(C)C)o1 C1(NC(c2c(OC)ccs2)=O)CCN(C(=O)CC2(O)CCC2)CCC1CO C#CC1(NC(=O)C(CC)N(C(=O)C(C)CC(C)(C)C)C)CC2CCCC12 C12(CNC(C3C(C(N)=O)C3)=O)CCC(CN(C(=O)CN3CC4CCC3C4)C1)C2 C12(C(N3CCCN(C(C(CCC)OCC)=O)CC3)=O)COCC1CN(C(C)C)C2 C1(C(N2CC(OCC(N3C(CNC(CC)=O)CCC3)=O)C2)=O)CCC(C)(O)CC1 CC1(C)CC(=O)c2[nH]c(=NC(C(N)=O)C(C)(C)C)oc2C1C(=O)O c1(OC(C(=O)NC(CN(CC(C(=O)OC)OC)C)C)C)ccc(Cl)cc1C C1(NC(C2C(OCC)C2)=O)CCC(F)(CNC(C2CN(C3COC3)C2)=O)C1 N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)CCS(N)(=O)=O)C(C2CCC2)C1 C1(NC(CCOCCC)=O)CCS(=O)(=O)C12CN(C(=O)CCCC(F)F)C2 c1(CC(C(=O)NC(CNC(c2c(CC)con2)=O)CC)F)ccc([N+](=O)[O-])cc1 C=CCCCCNC(=O)CC1(C)CN(C(=O)COC(C)(C)CC)C1 c1(C(N2CC=CC(NC(C(CO)NC(C(C)C)=O)=O)C2)=O)cc2occc2s1 c1(CCCOc2cn(C3CN(C(C(=O)OC)=O)C3)nc2)cccc(C)c1 c1(OC)nc(C)c(C(c2nnnn2C(C)C)NCCn2cnnn2)c(C)n1 Nc1sc2c(c1C(N1CC3(CCN(C(C4CCOCC4)=O)C3)C1)=O)CCC2 N1(C(CCC=C)=O)CCC2(CC1)CC2C(N1CCOCC(C(C)C)C1)=O C#CCC(CC(F)F)C(=O)NC1CC(C(F)F)(NC(=O)CN(C2CCCC2)C)C1 Cc1cc(F)cc(C)c1C(=O)NCC1CN(C)CCN1C(=O)C(C#N)C1CC1 Cc1ncc(C(N2CCCC2(C)C(=O)NCc2ccc(NC(C)C)cc2)=O)n1C C1(NC(c2ccc(CC)o2)=O)CN(C(C2CC(C)C2)=O)C2(CCCC2)C1 C(=O)(CC(C)(C)NC(=O)CCc1cncs1)NC(c1nccs1)C N1(C(COCC)=O)CC(NC(c2nc(C)n(-c3ccccc3)n2)=O)C(CC2CC2)C1 C(=O)(C(CC)C(F)(F)F)N1CC(OCCNC(c2n(C=C)nnc2)=O)C1 C1(CNC(CCCSc2ccc(C)cc2)=O)CCN(C(=O)CCC2CC2)C1(C)C C1(NC(C2(OC)CC2)=O)COC2CN(C(=O)CC3(O)CCCCC3)CC12 C(N=c1[nH]c(=NC2CCC3CCC23)[nH]c2c1CCC2)c1c(C)ccnc1 N(C1CS(=O)(=O)c2ccccc21)C(CC1C(C(=O)OCC)C1)=O n1(CC)nc(CNC(C2CC(NC(c3ccnn3C)=O)CCO2)=O)c(C)n1 N1(C(C2CC(C)(O)C2)=O)CC2CCC1CN2C(=O)C1=NOC(C2CCCC2)C1 C(C)(CCCC(=O)N1CCC(C(C)C)(CO)C1)NC(C(CC=C)C)=O C(C(=O)N1CCCC(CCNC(c2nc(C3CC3)oc2C)=O)C1)(C(C)C)OC c1(C(C(N)=O)NC(C2(F)CN(C(C3CC3F)=O)C2)=O)ccccc1Br C1(CC(=O)NC)CN(C(=O)CCCN(C)C(C)=O)CCN1C(=O)CC(C)C1CC1 Cc1ccc2c(c1)CN(C(C1(NC(=O)CC(=O)NC3CC3)CC1(C)C)=O)C2 C1(CC(=O)N(CCCCNC(c2c[nH]cc2Br)=O)C)CCOC(C)(C)C1 C=CC1(O)CCN(C(=O)COC2(C)CN(C(=O)C=C(C)C)C2)C1 C1(NC(C2(C)CCOC2)=O)CN(C(=O)Cc2ccc(O)cc2)CC2(CC2)C1 C(N=c1ccnc(N2CCN(CC(=O)N(C)C)CC2)[nH]1)c1c(C)nn(CC)c1C N1(C(C(C=C)(C)O)=O)CCOCC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(=O)Nc2cncc(OC)n2)cc(SC2(CC(=O)O)CCC2)ccc1[N+](=O)[O-] N1(CCC(=O)NC(C2CCN(C(=O)CSc3n[nH]c(=N)s3)C2)C)CCOCC1 c1(C(C(=O)NC(C2CCN(C(C3C=CCS3)=O)C2)C)=O)cccn1C c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cocn3)CC2(C)C)c2c(c1)CCO2 O=C(C1CCOc2ccccc21)NCC12CCCN(C(c3cscn3)=O)C1C2 C1(Cn2cc(C3C(c4cccc(C)c4)C3)nn2)CCC2(CC1)NC(=O)N(C)C2=O N1(C(CC2C(C)C(=O)CC2)=O)CCC2(CC1)CC2C(=O)NCC(=O)N(C)C c1(CNC(C2(COC)CN(C(=O)CC3CCCC3(C)C)C2)=O)ccccc1Cl Nc1c(C(=O)NCC(CNC(c2cncc(C3CC3)c2)=O)CO)cccc1F c1(OC)ccc(Cl)c(C(N2CCC(O)(C(N3CCCC(F)(F)C3)=O)C2)=O)c1Cl c1(OCC(=O)NCCCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CC1NC(=O)C(N(C)C)=C1NCC(O)C(C)(F)F C1(NC(c2n(CC)nnc2)=O)CCCN(C(c2cc(Cl)ccc2N)=O)C1C Cc1ccc(F)cc1CC(=O)NC1C2CN(C(C34C=CC(CC3)C4)=O)CC12 N1(C(c2c(C)csc2)=O)CCC(C)C(CC(=O)NCCCCc2ncc[nH]2)C1 CC1CCN(C(c2cccc(Cl)c2)=O)CC1NC(=O)CC1CC2CCC1C2 N#Cc1cc(C2CCN(c3ccccc3C#N)CC2)ncc1Br C1(C(=O)NCc2c(C)ocn2)CC(=O)CN1C(C1CC(=O)C1(C)C)=O CC1(C(F)(F)F)c2ccccc2CCN1C(CCC1CC1)C(=O)NCCCF c1(C(=O)NCC2CC(C)N(C(c3ccncc3)=O)C2)ccc(N=S(C)(C)=O)s1 c1(C(C)(C)C)nc(NC(=O)C=CCN2CCC(OC(C)(C)C)C2)cs1 C1(C(=O)NCC(C)(C)OC(C)C)CC12CCN(C(=O)CC1CCCCC1)C2 C(=O)(CCCCCCc1ccccc1)N(CCC)CCNC(=O)CCCCSC CC(C(=O)NCCCC1CN(C(c2cc(C(F)(F)F)c[nH]2)=O)CCO1)S(C)(=O)=O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)NC(c1ccc(N)cc1F)=O C12(C(=O)Nc3ncn(C)c3)CCC1CN(C(c1c(I)ccnc1Cl)=O)C2 N1(C(CC2N(C)CC=CC2)=O)CCC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(CC(C)CN(C)C)=O)CC2(C)CC1(C(=O)NC1C=CCCCC1)C2 N1(C(C#CC(C)C)=O)C2CCC1CC(NC(C1CCCCC1C)=O)C2 N1(C(C(CC=C)CNC(=O)CNC(=O)OCCOC)=O)CC(O)C(O)C1(C)C Cc1cn2c(n1)C(C(=O)NC1CCCC(NC(=O)CCc3cnoc3)C1)CCC2 C(C(C)C)(C(C)(C)O)NC(C(C1CCN(C(c2ccc(C)cc2)=O)C1)F)=O c1(CCC(=O)NCCCNC(C(C)OCCOCC)=O)cc(F)ccc1Br CCC(C)C(O)C(=O)N1CC2(NC(=O)C(N3CCC(C)CC3)=O)CC1C2 c1(CC(=O)NC(C(C(C)C)NC(=O)CCc2cnoc2)C)nc2c([nH]1)CCCC2 c1(OC)ccnc(C(=O)NC2(C)CC(NC(=O)CC3CC3(Cl)Cl)C2)c1OC c1(CC(=O)OCC(c2nnco2)=O)ccco1 N1(C(C2(Oc3ccc(F)cc3)CC2)=O)CCC2(C(=O)NC3CCC(O)C3)CC2C1 CC1(NC(=O)CCc2cc[nH]n2)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1ccc(O)c(C(C2CC(C)OC2C)COC(=O)C2CC2)c1 OC1(CNC(=NCC2CCOC2)NCc2nncs2)CCSCC1 C=CCCC(C(=O)N1CCCC(C)C1)NC(c1cc(C)cc(F)c1)=O C=CC1(C(N2CC(NC(c3ccoc3CC)=O)C2)=O)CCCCC1 C1(C(=O)NCCN(C(CN(CCC#C)C)=O)C)Cc2n[nH]cc2C(=O)N1 C1(C(N(c2ccc(Cl)cc2)C)=O)CCC(C)(C)N(C(=O)C2=CCCOC2)C1 N1(C(C=CC(CC)=CC)=O)CCc2sc(CNC(C3(F)CCCOC3)=O)nc2C1 c1(C(=O)NC2CCCCCC2NC(C2CCCSC2)=O)ccc2nonc2c1 N1(C(CCC#N)=O)CCC(NC(c2c(C(F)(F)F)cccc2F)=O)CC1C1CC1 N1(C(C)C(N2CCCC2CNC(C2(CC3CC3)CCCO2)=O)=O)CCCCCC1 c1(CC(=O)NC(CNC(CC(C)=C(C)C)=O)(C)C2CC2)ccc(F)c(C)c1 C1(NC(C2C(CC)CCO2)=O)CN(C(c2coc(Cl)n2)=O)CCC1C C(N=c1cc(C)nc(C)[nH]1)C1N(C(C(c2cccc(C)c2)(F)F)=O)CCCC1 Cc1ccc(C(=O)NC2CC2CNC(=O)C=CCN2CCC2)c(F)c1C C1(O)(C(=O)NCC2(NC(c3ccc(C)nn3)=O)CCC2)CCCC(C)CC1 C1(CNC(c2cc(=O)cc[nH]2)=O)CN(C(=O)CCc2nc(O)n[nH]2)C2CC12 C1(CCNC(C2(CNC(C(COC(C)=O)C)=O)CC2)=O)CC2CCC1O2 N1(C(C(F)OC)=O)CC2CN(C(c3cccc4c3OCC4)=O)CC2(C)C1 c1(C(=O)NCC(C(C)C)NC(C(C2CC2)OC)=O)sc(C)cc1C N1(C(C(C)n2cnnn2)=O)CCC2(CC1)CN(C(=O)CSC(F)F)C1COCC21 C1(F)(C(=O)NC(C)CCCCNC(C2CCC2C)=O)CCCCCC1 N1(C(CN(C)C2CC2)=O)CCC(CCCCCNC(C2(c3ncco3)CC2)=O)CC1 c1(CN(C(C2CCCN2Cc2ccco2)=O)CCO)cc(F)cc(Br)c1 c1(C(N2CC(C)C(NC(=O)CCCC(F)F)C(C)C2)=O)ccc2nc(O)oc2c1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 Cc1csc(C(=O)N(CCC(C)NC(=O)C(C)C2CC2)C)c1C N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CC(NC(c3cccc4nc[nH]c34)=O)CO2)C1 N1(C(CCCOC(C)=O)=O)C2CCC1CC(NC(=O)C(C)Sc1nncn1C)C2 Cc1c(C(=O)NC(CNC(C2(Cl)CCCCC2)=O)C(C)C)cccc1F c1(C(=O)NCC(=C)CCNC(=O)COC(F)(F)F)ccc(=O)n(C)n1 c1(N(C)CC)ccc(C(=O)N(C2CCN(C(=O)C(C)CC34CC(C3)C4)C2)C)cc1 C1(C(NNC(=O)CC2CCCCO2)=O)C(F)(F)C12CCOCC2 C1(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2)(NC(c2cnco2)=O)CC1 c1(C(N2CCN(C(=O)CC3C=CCC3)CC2C2CCC2)=O)nccn2ccnc12 N1(C(CC(CC=C)(C)C)=O)CCC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CCC12 c1(C(N)=O)cc(=NCC23CCCCC2CN(C(=O)CC2(O)CCC2)C3)[nH]c(Cl)n1 N1(C(c2oc(C)c(CO)c2)=O)CC(C(=O)NOCC(C)(C)C)CCC1(C)C C12(C(N(CC(C)NC(c3cc(CC)nn3C)=O)C)=O)CCOC1CCOC2 C(=O)(CC(C)NC(=O)CCC1CCC(NC(=O)CC(C)N(C)C)C1)OC C(=O)(C#CC1(C)CCCO1)NC(CCC=C)C(=O)Nc1ccc2ccccc2c1 O=S(=O)(NCc1cc(I)ccc1F)N1CCCC2(CCCNC2=O)C1 c1(C(=O)NCC2C(CNC(C(C)=CC3CC3)=O)C2)cnc(S(C)(=O)=O)s1 c1(C(C(=O)NC)N(C2CC3CC3C2)C)cc(C2CC2)[nH]n1 N1(C(C(CC)CC)=O)CC2CCC2(CNC(=O)C=CS(C)=O)C1 CCCCC(CCC)NC(=O)CN(C(=O)C(C)C1CCCC1)C1CCC1 C1(CC)CCC(C(=O)NC2(C)CN(C(C3(CF)CCOCC3)=O)C2)CC1 C(=O)(C(C)(C)CCCO)NCC1C(NC(c2c(=O)ccn(C)c2)=O)CCC1 N1(C(C2C(C)(C)OCC2)=O)CCC2(CCC2)C(NC(=O)C(=O)NCC(F)(F)F)C1 CC1CCC(NC(=O)CC2(O)CCCOC2)CN1C(c1cc(=O)n(C)cn1)=O Cc1oc(C2CC2)nc1C(=O)NC1CCCC(CNC(=O)COC(F)F)C1 CCCC(C)C(C)(c1nnnn1C)NCc1ccc(-c2cnco2)cc1 C1(NC(Cc2nc(CC)sc2)=O)CCCN(C(=O)C=CSc2nc[nH]n2)CC1F C1(C(C)C(=O)N2CC(C(F)(F)F)C2)CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(C(=O)NCCCC2CC2(Cl)Cl)=O)CCC2(CC1)CS(=O)(=O)C2 N1(C(c2c(CC)c[nH]n2)=O)CCCC(C)(NC(C2CN(C(=O)OC)CCO2)=O)C1 N12CC(O)(C1)CN(C)C(=O)C2=O.C1(C)(NC(=O)OC(C)(C)C)OCCO1 c1(NC)ccc(C(N2C(C(=O)NCC(C)(O)C3(C)CC3)CC2C)=O)cc1 CCC(C(=O)N(CCC(=O)N(CC(C)(C)N(C)C)C)CC)NC(N)=O Cc1ccccc1CC(=O)NC1CN(C(C2(CCCF)CC2)=O)CC1C(F)(F)F c1(OC)ccc(C(N2CCNC(C(=O)NCCC(C)C)C2)=O)cc1OC C1(Nc2nccc(OCC)n2)CN2CCN1CC2C.C12(F)CC(C1)CNC2=O c1(CC)c(C(=O)N(C)CC2COCCN2C(c2cnnn2CC)=O)nnn1CC c1(OC(=O)NCC(c2cncc(F)c2)(C)C)cccc(C#N)c1[N+](=O)[O-] c1(NCC2OCC(C)C2)[nH]c(=NCC2(C(F)(F)F)CC2)nc2c1ncn2C c1(N(c2sc(=NCc3ccccc3Br)[nH]c2C)CC)c(F)cc(Br)cc1[N+](=O)[O-] c1(C(=O)NC2(CCCNC(C3C(C)(COC)C3)=O)CC2)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2(C)CCN(C(C3(C)CC=CCC3)=O)C2)c(F)cccc1F N1(C(CC=C(C)C)=O)CC2=C(C1)CN(C(=O)Cn1nc(C)c(Br)c1C)C2 C1(CNC(Cc2c(C)nsc2)=O)(NC(=O)C(O)CC2CCCCC2)CCOCC1 c1(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)cnc2c(c1)COCC2 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCN(C(c2nnn(C)c2C(F)F)=O)CC1C C1(NC(CCCCC#C)=O)CC2(CCC(CNC(c3cnnc(C)c3)=O)CC2)C1 N1(C(C2C(C)(C)C2)=O)CCCC(C2CN(C(=O)C(c3ccc(Cl)cn3)(F)F)C2)C1 c1(CCC(=O)NCCCSC(C)(C)C)c(Br)cncc1Br N1(C(C(C)NC(=O)C2CC2)=O)CCCC2(C1)CC2(F)F Cc1ccc(C(=O)NC2CCN(C(c3cc(C(N)=O)cn3C)=O)CC2)cn1 c1(C(=O)OCC)cnc(NCc2nnc(CO)s2)s1 c1(C(N2CC3C(NC(CSCCC)=O)(C3)C2)=O)cc(SC)c(Cl)cc1Cl N1(C(C2CCC(C(N)=O)CC2)=O)CCCC(C2CN(C(=O)C3=NNC(=O)C3)C2)C1 CN1CCC2C(CCN2C(=O)CCC2CCCN(C(C3(C4CC4)CC3)=O)C2)C1 C12(NC(CC=CC)=O)CCOCC1CN(C(c1cccc(Br)c1)=O)C2 CCCCC(CNC(c1cnccc1N(C)C)=O)NC(=O)CC(=O)NCC1CC1 c12cccc(c1)CNC2=O.C(C)(C(C)=O)N(CC)CC Cc1sc(C(N2CC3CC2CN(C(=O)COC(F)F)C3)=O)cc1[N+](=O)[O-] C(=O)(CCCC(=O)N1CCCC(NC(=O)C(C)(C)n2ccnn2)CC1)OC C1(CCN(C)C(C2CCC2(F)F)=O)CCCCN1C(c1ccc(=O)oc1)=O C(CC1=CCCCC1)N(C)C(=O)NCc1cc(F)ccc1Br C1(CC=C)CCCCN1C(=O)CNC(=O)CC#N C1(NC(C2CCC(NC(=O)C3=CCCC3)C2)=O)CCC(C2CC2)C1 N1(C(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(=O)CCC1CCCO1)CO2 c1(NC(c2cc(OC)ns2)C)cc(C)c(S(=O)(=O)N2CCCC(O)CC2)cn1 c1(CCNC(CC(CNC)(C)C)=O)ccc2c(c1)COC2(C)C c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)cccc2cccc(O)c12 C1(NC(CC2(CSC)CC2)=O)(CF)CCN(C(=O)C(c2cccn2C)=O)C1 C1(OC)CC2(C1)CC(C(=O)NCC(c1ccccc1)NC(=O)CC(C)C)C2 C1(NC(C(CC)N(CC)CC)=O)CCC2CC1CN2C(=O)CCC(C)(C)OC CC1CN(C(=O)CSc2cn[nH]c2)CC1CNC(=O)Cn1nnc(=N)[nH]1 C1(C(N2CCC(SC)CC2)=O)CN(C(=O)C=CC(F)F)C2(CCC2)C1 Cc1cc(CNC(C2CCN(C(c3cc(C)nc(C)c3)=O)C2(C)C)=O)cc(F)c1 c1(C(=O)NCC2CCC(C)N(C(=O)COCCCF)C2)cccc2[nH]ncc12 N1(C(C(C)CCN(C)C)=O)CCOCC1(C)c1cn(-c2cccc(Cl)c2)nn1 C1(C(N(CC2=NOCC2)C)=O)C2CCCC2CN1C(=O)CC1CCC(=O)N1C O(N(CC)C(=O)C1CC=CC(NC(c2ccnc(OC)c2)=O)C1)CC C1(CCCNC(C(COC)OC)=O)CCCCN1C(=O)C=C(C)c1ccco1 C1(CCNC(CCC(=O)NCCC)=O)CCCN(c2nccc(CC#N)n2)CC1 N(C)(C(=NCCF)NC1COC2CC1C2)CC1(OCC)CCCCCC1 Cc1cccc2c1C(=O)NC(C)(C)N2C(c1noc2c1COCC2)=O CCCC(C)(O)C(=O)NC1CC(OCC(N2CCC(n3cnnn3)C2)=O)C1 O=C1CC2(CCC2)C(C(=O)ON2CCN(CCOCCO)CC2)CN1 c1(C(=O)NC2CC(NC(=O)CCNC3CC3)C2)cc2ncccn2n1 C(=O)(C1=CC2C=CC(C1)C2)NCC(CC=C)NC(=O)CCc1cnn(C)c1C Cc1ccnc(C)c1C(=O)NCC(CO)NC(=O)CC1CC(c2ccccc2)C1 C1(F)(CNC(C(n2ncc(C)c2)C)=O)CCN(C(=O)C(F)C(C)C)CC1 c1(C(=O)NC(CN(C(C2CC(O)C2)=O)CC)C)cc(O)c2ccsc2c1 c1(C(=O)NC2CS(=O)(=O)CC2NC(c2ncccc2O)=O)cnc2n1CCOC2 Cc1c(C(N2CCN(C(C3(C)CC3F)=O)CC2)=O)sc2[nH]cnc(=O)c12 C1(C(C)NC(=O)C(Cl)=CCl)CN(C(=O)CC2(O)CCC2)CCO1 N1(C(C2(c3cn(C)nc3)CC2)=O)CCN(C(=O)CC2CCCC23CC3)CC(O)C1 c1(CNC(=O)NCCC2CCOC2)ccc(CO)c(Cl)c1 N1(C(C2C(C(=O)OC)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CC2)C1 C(=O)(CCC(C)CN(C)C)NC(CCCC)CNC(=O)CCNc1ccccn1 C12CCCCN1C(=O)C1(CC1)NC2=O.C=CC(O)C(=O)NCc1ccccc1 n1(C2(C)CC2)nnnc1C(c1cc(Cl)cs1)(C1CCC1)NCCCCC1CC1Cl c1(SC)cc(C(N2CCC(NC(c3cccnn3)=O)C(F)C2)=O)cc(Cl)c1 N1(C(c2ccc(C)cc2C)=O)CC2CCCC1CN(C(=O)COC(C)C)C2 C1(CNC(C(c2ccc(F)cc2F)C)=O)CC2CN(C(C3CCC3)=O)CC12 C1(C(=O)NCC2(F)CN(C(C(CC=C)NC(C)=O)=O)C2)CCC2(CCOCC2)O1 c1(C(=O)NCC2CCC(NC(c3ccc(CC#N)cc3)=O)C2)cc2n(n1)CCC2 N1(C(c2n(C(CC)CC)ncc2)=O)CC2CC1C2NC(c1cnc(Cl)s1)=O c1(C2(C#N)CCC2)cccc(CNC(=O)CNc2ccccc2Cl)c1 C1(C(=O)Nc2c(C)c(-n3cccc3)ccc2)CNCC1C1CCOC1 N1(C(C(c2ccccc2F)(C)C)=O)CCC(CF)(NC(C2CCCO2)=O)C1 c1(C(=O)NC2(CC)CN(C(c3nncs3)=O)C2)coc2c1COC2 CC(C)(C)CC(O)C(=O)NCCCCCCC(=O)NCCCC1(O)CC1 C1(OC)CC2C1CCN2N1CC(c2nc(O)c3ccccc3n2)C1 C1(C(=O)Nc2cn(C3(CN)CC3)nc2)CCCC2(C1)CC2(F)F c1(C(N2CC(N(C(CCC#C)=O)C)C2)=O)c[nH]c2ccc(C#N)cc12 c1(C(=O)NC2C(NC(c3c(C)n(C)nc3)=O)COCC2)ccn2c1CCC2 c1(C(N2CCC(C(=O)Nc3c(C#N)scc3)C2)=O)ccc(O)c([N+](=O)[O-])c1 N#CC1(C(=O)NCCCCCNC(c2ccc(C3CCOC3)s2)=O)CC2CC2C1 n1(C(CC#C)C2CC2)c(N2CCC(CS(C)(=O)=O)CC2)nnc1-c1ccc(C)o1 O=C(C(F)(F)CCn1cc(-c2ncccn2)nn1)NCC1CCS1(=O)=O C1(NC(CC(=C)C)=O)CN(C(=O)CC2(OCC)CC2)CC1Cc1ccccc1 C1(CNC(CC2(CNC(=O)Cn3nccn3)CC2)=O)(OC)CC2CCCC12 CCC(CCCC(=O)NC(C)(CO)C1CCC1)NC(c1coc(C(C)C)n1)=O c1(C(N2C(CNC(c3cc(OC)ns3)=O)C(C)CC2)=O)cnc2[nH]c(C)nc2c1 c1(C(=O)OC)cc2c(s1)CCC2NC(=S)Nc1cccc(F)c1C c1(C(N(C2CCN(C(C(CC=CC)C)=O)C2)CCC)=O)ccc(C2CC2)c(Cl)c1 n1(CCOCC)nnnc1C(c1ncoc1C(F)F)NC1CC(C)C1 c1(OCC)cc(-c2nccn2Cn2cccc2)cc(C2CC2)c1O C(=O)(C(C)CCCC(C)C)N1CC(CC(=O)NC(CC)C(=O)NC)OCC1 CC(C)CC(CNC(c1ccc(C(O)CF)cc1)=O)NC(c1cc(Cl)n(C)n1)=O C1(C(=O)OC)CCC2(CCOCC2)CN1C(=O)Cc1csc(-c2ccc(Br)s2)n1 N1(C(C(C)=C2CCCC2)=O)CC2CC(C1)CN(C(=O)Cc1cnns1)C2 C(=O)(C1SCCc2sccc21)NCC(C1CCC1)NC(c1cc(C)n(C)c1)=O N1(C(CCC2CCCCN(C(c3cccc[n+]3[O-])=O)C2)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(F)=C2CCCC2)C1 C(CC(O)C(=O)NCC1CCN(C(C2CCCC2c2nncn2C)=O)CC1)SC N1(C(C2CCC(CNC(=O)COCC3CCCC3)CC2)=O)CC2CCOC2C1 Cc1nc(C=CC(N2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)=O)cs1 C12(NC(C=CC(C)C)=O)CCN(C(C3(c4ncc[nH]4)CC3)=O)CCC1C2 N1(C(CCC2OCC(C)(C)C2)=O)CC(C)(C)C(NC(=O)CSC(F)F)C(C)(C)C1 n1(CCC(=O)NCC(CC)NC(=O)Cc2cn(CC)nn2)ncn(C)c1=O C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)CC(N)=O)C1)C)OC N1(C(c2nc(OCC)sn2)=O)CCC2(CC(NC(C3(C)CCOC3)=O)C2)C1 C1(CC)CCC(Cn2cc(C(C(=O)NCCCF)N(C)N(C)C)nn2)CC1 Cn1nccc1C=CC(=O)NC(C1CCOC1)CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NC(CO)CC(C)(C)C)C(C)C1 C1(C2CCC2)(C(N2CCC(CNC(C3(CC)CC3(F)F)=O)C2)=O)CC1 N1(C(Cc2c(C)nsc2)=O)CCC2(NC(=O)Cn3ccc(O)nc3=O)CCCC12 CC(C)CC(O)C(C)C(=O)NC1CCCC(CC(N2CC(N(C)C)C2)=O)C1 C1(C(=O)NCCN(C(=O)CN2CCCC2=O)C)CC2CCC(C1)S2 C1(C(=O)NC2(CC(=O)NCCCn3cccn3)CC2)CCS(=O)CC1 c1(CC)ncc(C(=O)NC2CCCN(C(c3ccnc(Cl)c3N)=O)C2)c(C)n1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCN(C)C(=O)C1)=O N=c1[nH]c(CC(=O)NCC2(CNC(=O)C=CCF)CC2(F)F)cs1 C1(NC(C(C)C)=O)CCN(C(C2(CF)CC2)=O)CCC1(F)F c1(C(C)OCC)nc(NC(=O)NCc2nc(CN(C)C)ns2)cs1 c1(C(N(CCNC(CN2C(=O)CN(C)C2=O)=O)C2CC2)=O)nccc2cc[nH]c12 C1(CC)(NC(c2cc(F)cs2)=O)CCN(C(C2CCCNC2=O)=O)CC1 c1(C2(C(N3C(CC(c4ccc(Br)o4)=O)CCC3)=O)CC2)ccnc2ccccc12 C1(C(N2C(CN(C(CN(CC(=O)NC(C)C)C)=O)C)CCC2)=O)SC(=N)NC1=O Cc1c(C(N2CC(CNC(=O)Cc3ccsc3Cl)CC2C)=O)cnn1CCO C1(NC(CC(C)C2CC2)=O)(Cc2ccccc2)CCN(CC(N)=O)C1 C1(CNC(C(CC=CCC)C)=O)CN(C(c2cnc(CC)nc2O)=O)CC1(C)C CCCCC(CNC(=O)CC(C)CC)NC(C1CN(CC(F)(F)F)C1)=O c1(-c2ccc(OC)c([N+](=O)[O-])c2)cnc(N=c2[nH]c(C3CC3)cc(C)n2)nc1 c1(C(c2n(CC3CN(C(=O)OC)C3)nnn2)NCC)noc2c1CCC2 Cc1ccc(N(C(=O)CC2COC(C(F)(F)F)C2)C(N)=O)cc1 N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(c1cc(C2CC2)no1)=O N1(C(C(C)CF)=O)CCCC(C)C1CNC(c1cnn(C2CC2)c1)=O C1(NC(C2C(=C)CC2)=O)C2CC1N(C(C1(Cc3ccccc3Cl)CC1)=O)C2 Cc1cc(C(=O)NC2CCC3CC2CN3C(=O)CCNS(C)(=O)=O)cc(C)c1C N1(C(c2cnc(C)s2)=O)CC(NC(=O)Cn2cccnc2=O)C(C)C1 CC(C(=O)N(C1CN(C(c2cn3cc(Br)ccc3n2)=O)C1)C)C(F)(F)C(F)F N1(C(CCCC(=C)C)=O)CCC2CN(C(c3sccc3CC)=O)CC12 N1(C(c2c(C)n(C)cc2)=O)CCC(N(C(=O)CSC(C)(C)C)C)C(C)C1 C1(NC(c2n(CC)ncc2)=O)CCCN(C(C2C=CCC=C2C)=O)C1 Cc1nc(C(N2CCCC(N(C(=O)CCCc3ccc(Cl)cc3)C)C2)=O)nn1C c1(-c2onc(-c3cccc(SC)c3)n2)cnn2c(C)c(C)ccc12 c1(NCC)ccccc1C(=O)NC(CO)C(=O)NCC12CC(CCO1)C2 C123CCC(CC1)(CO2)CNC3.C(=O)(C(C)c1ccco1)OC(C)C.C12CC1NC2=O N1(C(C#C)C)CCN(C(=O)C(CO)NC(=O)CC(CC)SC)CC1 C1(C(=O)NC(C)CN(C(=O)CSCC2CCCO2)C)CNC(=O)CC12CCC2 N1(c2cc(COC)ncn2)CCC2(CC1)CC(NC(C1(OC)CCC(C)C1)=O)C2 C1(CN(C(C(COC)OC)=O)C)CN(C(c2cc(C)c(C)o2)=O)CCO1 c1(C(N2C(C(C)(C)NC(c3c(C)nc(C)o3)=O)CCC2)=O)coc(S(C)(=O)=O)c1 Cc1cccc(C=CC(N2CC(O)CC2C(N2CCC2C(C)O)=O)=O)c1 C1(CNC(C2(C(C)(F)F)CCC2)=O)CC2(CC2)CN1c1nc(CC2CC2)ns1 CC1(C)CCC(O)(CNC(C2(CNC(=O)CCC3(C)N=N3)CCCCC2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC12C(CN(C(c3c(N)c(O)ccc3Cl)=O)C1)C2 CC(C)(C)C(C#N)C(=O)N1CCC(C(N2CCCC3(CC3)C2)=O)(CF)C1 Cc1cnc(N2CCC(C)CC2)c(S(=O)(=O)NC2CCCCN(C)C2)c1 Cc1ccc(Cl)c(O)c1C(N1CCC(NC(C2CC(C)CO2)=O)CC1)=O c1(C(CNC(=O)CC2CNC(C(F)(F)F)CO2)=O)ccc2nccn2c1C.CO c1(C(N2C(CNC(CC(=C)C)=O)CCC(C)C2)=O)onc2c1CCCC2 N1(C(CC2C(C)=NOC2=O)=O)CCC(CNC(c2nc(C)oc2C)=O)C(C)C1 N#Cc1cc(C(N2CC3(C2)CN(C(c2cc4n(n2)CCC4)=O)C3)=O)ccc1F C1(C(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)CC2CCC(C1)N2C c1(OCC)c(C(=O)NCCNCCCN(C)Cc2cnccn2)cccc1Cl C(=O)(C#CC1CCCCC1)NC12CC(CNC(C3(C#N)CC3)=O)(C1)C2 c1(C(N2CCN(C(C(C)SC)=O)C(C3CC3)C2)=O)cccc2ccccc12 C=CC1(O)CCN(C(C2CC=CCN2C(C2CC(C3CC3)C2)=O)=O)C1 C1(CNC(Cc2cc(C)sc2)=O)CN(C(=O)CCCC(C)(F)F)CCC12CCC2 CC(C)C(C(=O)Nc1ccc2ncnn2c1)C(C)NC(=O)CCN1CCCCC1 N1(C(CCN(CCC)C)=O)C2CCC(C(=O)NCc3n[nH]c(C)n3)C1CC2 c1(N2CC(NC(c3c(OC)cncc3)=O)C(C)CC2)ncn(C)c(=O)c1Br c1(C(=O)NC2CN(C(CNC(C)=O)=O)C(CO)C2)cccc(N2CCCC2)c1 c1(OC)ccccc1OCCC(=O)NCC1(O)CCN(C(=O)C(C)NC(N)=O)C1 C1(NC(C(N(C(c2snc(C)c2N)=O)C)C2CC2)=O)CCc2c[nH]nc2C1 N1(C(=O)OC(C)(C)C)CCC(O)(COC(=O)NCCC2CCC(F)(F)CC2)CC1 c1(N2C3CN(c4c5ccn(C)c5ncn4)CC2CC3)ccnc2c1ccn2C N1(C(c2c(Cl)ncn2C)C(=O)NC(c2ccccc2)C)CCN(C)C2(CCC2)C1 C(=O)(C1=CCCN(C)C1)NCCC1(O)CN(C(c2c[nH]c(=NC)s2)=O)C1 C1(CC(=O)NCC2(COC)CCCO2)CC(C)N(C(c2cc(=N)[nH][nH]2)=O)C1 CC1(C)CC1(NC(c1cccnn1)=O)CC(c1ccccc1)C(=O)O C1(N(C(CSCC=C)=O)C)CC2CCC(C1)N2C(c1cnc(N(C)C)o1)=O Cn1c(C(N2CCCC(CCCCNC(=O)C(O)C3CCC3)C2)=O)ccc1C#N N1(C(c2c(CC)n[nH]c2)=O)CC(O)CC1(C)C(=O)NCC1CC(F)(F)C1 Cc1ccnc2c(S(=O)(=O)NCC(c3ccc(=N)[nH]c3)=O)cccc12 C1(C(=O)NC(CCC)C(=O)NCC2(C)CCC(=O)N2)CN(C)CC(C)O1 C=Cc1cc(C(=O)NCc2noc3c2CCCC3)cc(F)c1 c1(C(COC)NC(C2(c3ccc(Cl)cc3)CCC2)=O)ccccc1F C1(NC(CCNC(=O)OC)=O)CC2CCC1CC2NC(=O)C(N1CCOCC1)C c1(C(N2CC(CCNC(C(C)(CO)OC)=O)OCC2)=O)cc2ccsc2c(O)n1 Cc1coc(C(N2CC(O)CC2CNC(=O)CCC(=O)c2cccs2)=O)c1C CCC(C)C(C(=O)NCCCS(C)(=O)=O)N(C(=O)C(F)C(C)(F)F)C C1(CCC(C)(C)NC(=O)CNC=O)CCN(C(=O)C(F)C2CCC2)CC1 N1(C(C2N(C)C(=O)CCC2)=O)CC(F)(F)CC1(C)CNC(=O)CC1CCOCC1 CCC(C)C(C(=O)NCC(C)CNC(=O)Cc1ncc(C)s1)N(C(=O)OC)CC N1(C(C(CC(C)C)NC(CCCOC)=O)=O)CCC(C2CC2)CC1 CC1C(C(=O)NNC(=O)C2CCCN(CC3CC3)C2)CCN1C(=O)NC(C)(C)C S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(NC(c2scc(C)n2)=O)C(F)(F)CC1 c1(C(=O)NCC2CC(NC(C=CC(CC)=CC)=O)C2)ccc(N)c(C(F)(F)F)n1 c1(C(=O)NC2(CNC(C(c3cccc(Br)c3)C)=O)CC2)nc2ncccn2n1 C1(NC(c2c(CC)ccs2)=O)CCC12CN(C(c1csc(C(F)F)c1)=O)C2 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CCNC(c2cnc(SC)n2C)=O)CCC1 S(=O)(=O)(c1ccc(N2CCC3(CC(F)C3)C2)nc1)N1CC(C)(C)C(CO)C1 C1(C(N(C)CCOCCNC(c2cccc(C3CC3)c2)=O)=O)CC1C1CCCC1 [N-]=[N+]=NC1CCC(C(=O)NC(C2CCCOC2)C(=O)O)CC1 CC1CC2CN(C(=O)CCCC3(NC(=O)CN4CCNC4=O)CCC3)CC12 C1(O)(CC(N2CCCC2CO)=O)CCN(CC2(C3CCC3)CC2)CC1 c1(CN2C(COC)CCCC2)c(C)nn(C2CCS(=O)(=O)C2)c1Cl C1(NC(c2nc(C)[nH]n2)=O)CC(=O)N(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 N1(C(CCC=C(C)C)=O)CCC(C(=O)N(CC(N2CCCC2)C)C)CC1C C(=O)(C1=CCC2CCC1N2C(c1ccc(N)cn1)=O)NCCCC(C)C C=CC(C)N=c1[nH]c(=NCCN(CCCC)C(C)C)c2c(ncn2C)[nH]1 c1(C(=O)NCC(C2CCC2)NC(C(C)O)=O)ccc(S(C)(=O)=O)cc1Br Cc1cnn(CC(=O)NC2CCC2NC(=O)Cn2ccc(C)n2)c1 C(=O)(C1NCCc2nn(C)cc21)NCCc1c(C(=O)OC)cccn1 C1(C(=O)NCC(C)CNC(=O)CCc2csc(Br)c2)CCOC(C)(C)C1 C(C(CC1CC1)C(=O)N(C)Cc1cn(C)nn1)NC(C1(SC)CC1)=O c1(C(C(=O)NCC2(OC)CCN(C(CCC#C)=O)C2)C)cc(C)cc(F)c1 c1(CC)ccc(C(=O)NCCC2COCCN2C(=O)C(F)C(C)(C)O)c(F)c1 O=C(C(F)CC1CCOCC1)NCCCNC(C1(CC2CCC2)CC1)=O C1(NC(C2(C(N)=O)CC2)=O)CC2(CCC(NC(c3ccnn3C3CC3)=O)CC2)C1 C=CCC(CNC(c1scnc1C)=O)NC(C1CCCCO1)=O C(c1ccccc1)=C(OC)C(=O)NC1CN(C(c2cscn2)=O)C1 c1(C(NOCc2cn(CC(CC)O)nn2)=O)ccc2cc(N(C)C)ccc2c1 C(=O)(C(C(C)(C)O)NC(C1CCCSC1C)=O)NCCC(CCC)O C1(CCNC(CC=C=C)=O)CCCN(C(=O)CCc2ccc(CC)cc2)C1 c1(CC(C)C)nccc(C(N2CCC(C)(CCNC(=O)C(F)=CC3CC3)C2)=O)n1 N1(C(CCCC#N)=O)CCCCCC1C(=O)NCCn1cnnc1 C1(C(=O)NCC2CN(C(c3ccc(SC(F)(F)F)s3)=O)C2)CCCCCCC1 CC1N(C(C2CC23CC(NC(=O)COCCN(C)C)C3)=O)CCC1(C)C C1(CNC(c2c(OCC)scc2)=O)CCCCCN1C(=O)CC(C)C1CCCC1 c1(-c2onc(-c3ccc(Cn4cncn4)nc3)n2)ccc2n[nH]cc2c1 c1(C(N(CC(=O)OC)CC#N)=O)cc(C)c(C(=O)O)cc1C Cc1ccc(CNC(C2CCN(C(C3COCC3(C)C)=O)C2C)=O)cc1 Cc1cc(F)c(C(=O)NC2(C)CCN(C(=O)C(C)CF)C2)cc1N N#Cc1ccsc1C(N1CC(NC(=O)CSc2cccs2)C(C(F)F)C1)=O C1(c2n(CCCC)nnn2)(NCCOCCOC)CCC2CCCC2C1 C1(NC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)C(N2CCOCC2)C)CC1 c1(C(N2CCN(C(C3(C=C)CC3)=O)CC2CO)=O)cc2oc(Br)cc2s1 CN1CCOC2(CCN(C(C3(C)CCCN(c4ncncc4I)C3)=O)C2)C1 C(CCCC(c1nnnn1CCCSC)NCCC1CCSC1)OC c1(C(=O)NCC2N(C(c3noc(CC)c3C)=O)CCCC2)cc(S(N)(=O)=O)cs1 c1(C(N(C2CCN(C(=O)C(C)(C)CF)C2)CCC)=O)ccc(C(C)C)cc1F C1(C(N(CC(C)NC(=O)COCC(=O)NCc2cccnc2)C)=O)C2COCC12 C1(C(=O)NCC(C)CCl)COC2(CCN(C(c3cnn4c3CCCC4)=O)C2)C1 C=CCC(CC)C(=O)NCc1ccc(CNC(C2(Cl)CC23CCC3)=O)cc1 C1(SC)CCC(NC(c2cn(CCNC(C3(c4ccno4)CC3)=O)cn2)=O)C1 c1(OCC(N2CCN(C(C3(C)CC3)=O)CC2CCO)=O)ccc2c(c1)CCCC2 c1(C(CCC(N2CC(=O)NCC2)=O)=O)ccc2c(c1)NC(=O)CC2 c1(CNC(C2C(C)(C)CO2)=O)ccc(CNC(C2CCCC(O)C2)=O)c(F)c1 C1(C2CCOCC2)(C(=O)NC2CCN(C(c3c(C)cc[nH]c3=N)=O)C2)CC1(F)F c1(CCC(=O)N(C(C)CCNC(=O)CCC[N+](=O)[O-])C)c[nH]c2ccccc12 c1(C(=O)NCC(N(C(Cc2scc(CC)n2)=O)C)C2CC2)ccc(S(C)=O)cc1 CC1CCCC1C(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C c1(NC(C2C(C(=O)NCc3cn(C)nc3)C2)=O)cc(Br)cnc1I CCC(CC)C(=O)N1CCOCC1CC(N1CCC(CF)C1)=O c1(N2CC(C(N3C(C(=O)OC)CSCC3)=O)OCC2)nc(C)ncc1C#N c1(NC(c2ccccc2-n2cc(CCCO)nn2)=O)cccc(Cl)c1.N12CC(C1)C2 n1(Cc2ccc(C)cc2)cnc2cc(C(=O)NNC(=O)CCN(C)C)[nH]c2c1=O c1(-c2cn(C(CNC(COCCCC)=O)C)nn2)ccc(-c2cn[nH]c2)cc1 N1(C(c2cnc(C)[nH]c2=N)=O)CCC(C2CC2)C1CNC(c1nc(C)no1)=O N1(C(c2cnc(OC)nc2C)=O)CC2(COC(CNC(=O)C(C(C)C)SC)C2)C1 c1(NCc2c(OC)cnc(F)c2)ccc(C2=CCSCC2)cc1C c1(C(N(C(C)CNC(C2(n3ccnn3)CC2)=O)C)=O)cc2c(F)c(F)ccc2[nH]1 c1(C(=O)NC(CC)CNC(c2c[nH]nc2C(F)F)=O)cccc(C#N)c1C CC1CN(C(=O)CCc2ccc(C3CCC3)cc2)CC1CNC(=O)CCF N1(CC(N2C(C3(NC(=O)C=CCF)CC3)CCC2)=O)C(=O)CNC1=O c12cc(on1)COC2=O.C(=O)(C(CC1CCCO1)SC1CC(F)C1)OCC C1(NC(c2ncc(F)cn2)=O)CCC2(CC1)CN(c1cncc(Cl)n1)C2 c1(NC(C)=O)cccc(C(N2CCCC(C3CC(N)CCO3)C2)=O)n1 c1(C(=O)NCC(CC)NC(c2cnsc2C)=O)cnc(CC2CC2)s1 N12CC3(CCC1C3)CCNC(=O)c1nc(cs1)C2=O.C1(NC(C)=O)CC(O)CN1 N1(CCC(=O)N(C2CN(C(CC3ON=C(C)C3)=O)C2)CC2CC2)CCN(C)CC1 C1(CCNC(c2c(C)coc2)=O)CC(F)(F)CN1C(c1ncc(C(F)F)s1)=O c1(OC)cncnc1C(=O)NCC(C1CCOC1)NC(c1nncs1)=O C1(CC(=O)N(CCCCC)C)CN(C(C2(CC)CC2)=O)CCO1 c1(C(=O)NC2(C(C)(C)C)CCN(C(=O)C#CC3CCC3)C2)cccc2cncn12 C1(CC=C)(NC(=O)C(C)NC(=O)CC)CCN(C(c2c[nH]nc2C(C)C)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(=O)NC(C=C)C1CCC1)Cc1cc[nH]n1 c1(C(N2CC(NC(C(CC)CC3CCCC3)=O)C(C)C2)=O)cc(N)cc(F)c1 c1(C(N2CCN(C3CCN(C(C4C(C)C4)=O)CC3)CC2)=O)ccc(Br)nc1O c1(CC(=O)NC2C(NC(=O)C=Cc3cc[nH]n3)C2)ccc2ccccc2c1 c1(C(=O)NC(CCNC(c2cc(C)c(F)cc2N)=O)C)cc2c(s1)CC(C)(C)C2 CC1(C)OCC2CC12C(=O)NCC1CCN1C(c1nocc1Cl)=O c1(C(=O)NCC(C)NC(C2(C)CC2)=O)cc(-c2ccccc2)n(C)n1 CCCC(C=O)NC(=O)CSCC(N)=O.C(CF)N c1(C(=O)NC2CC(CC(C)C)OCC2)cc(S(C)(=O)=O)ccc1F CC1(C(=O)NC2CCCC2NC(C2CC(F)(CO)C2)=O)CCc2ccccc21 CC1(C(=O)NC2CCCC2NC(C2(C3CCCO3)CC2)=O)CC1(F)F c1(N(C2N(C(C(CCC)C)=O)CCCC2)C)cc(C(F)(F)F)nc2ncnn12 c1(C(N2CCN(C(C#CC3(CC)CC3)=O)C(C)CC2)=O)ccc2oc(=O)oc2c1 N1(C(c2c(C)nccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1C C(=O)(C(=O)N=c1ccn(Cc2cccc(Cl)c2Cl)c(O)n1)N(c1nccs1)C(C)C CC1C(NC(c2cc3c(F)cccc3s2)=O)CC2CCC1N2C(c1cnns1)=O c1(C(N2C3C(NC(c4c(COC)cc[nH]4)=O)C(C3)C2)=O)cccc2cnccc12 Cc1ocnc1CC(=O)N(C(C)CCNC(=O)CC1CC1C1CC1)C C=CCC(CC)C(=O)NC(CCC)CCCNC(C1(C2CCC2)CC1)=O C1(CN(C(C2CC(OC)OC2OC)=O)CC)COCCC1C1CC1 CCC(C(=O)NC1(CN(C)C(C2CCC(C(N)=O)CC2)=O)CC1)C(C)(C)CC N1(C(C2CCC(CC)CC2)=O)CCCC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 Cc1[nH]nc(C(N2CCC3(NC(C4C=CCC4)=O)CCCC23)=O)c1[N+](=O)[O-] C12(CNC(COCC)=O)CC(NC(=O)C(C)NS(C)(=O)=O)(CO1)C2 CC(=O)CCCCCCC(=O)N1CCC(NC(=O)C2=CS(=O)(=O)CCC2)C12CC2 C(=O)(CCC(=O)NCC1CCCCC1NC(=O)CSCC(=O)OC)NC C1(C)(C(=O)NCC(C2CCCC2)NC(C(N2CCOCC2)C)=O)CCCS1(=O)=O c1(C(N2CCC(OC)C2)C(=O)NC2CCCCC2)ccc(C)c(C)c1F CCC(COC)C(=O)N1CC(C(=O)Nc2csnc2C)(CC)C1 C(=O)(CCC(C)(C)F)NC(C1(O)CCN(C(C2CCC(C)O2)=O)C1)C N1(CC(c2cscn2)N(C)C)C(=O)NC(c2cccc(F)c2)C1=O c1(NC)ccc(C(=O)NC(CC2CC2)C(=O)N(C)Cc2nnnn2C)cc1 Cc1oc(SCC2(F)CC(NC(=O)OC(C)(C)C)C2)nc1NC(=O)CO c1(CNC(CC(C)C)=O)cnn(C)c1C(N1CCOCC1C(=O)OC1(C)CC1)=O c1(C(=O)NCCN(C(C=Cc2ncc(C)[nH]2)=O)C2CCC2)ccc(O)c(F)c1F C1(C)(CCC(=O)NCCCCC2C(C)C2)CCCN1C(C1CCCCCC1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC2(CCN(C(C3(F)CCOC3)=O)C2)C1 c1(C(N(CCNC(c2coc(OC(C)C)n2)=O)CC)=O)cc2cc(C)ccc2s1 N1(C(c2c(CC)n[nH]c2)=O)CCCCC1CNC(=O)Cc1nonc1C C1(C(=O)OC)Cc2c[nH]nc2CN1C(c1ccc(OCc2ccccc2)nn1)=O C1(C(=O)NCCCC2(CNC(C(C)OC3COC3)=O)CCCC2)CCCC12CC2 c1(C(=O)NCC(CO)NC(c2cc[nH]c2)=O)cc(Br)n[nH]1 c1(C(=O)NCC(C)(CO)NC(c2cccs2)=O)cccc(-n2ccnc2O)c1 O=C(C(O)CC(F)(F)F)NCC12CCC(CC1)N2C(=O)CC1CCCO1 C1(C(N(C(CNC(c2c[nH]c(=NC)o2)=O)C)C)=O)CC2C=CCC(C1)C2 COn1cnc(C)c1C(=O)NC1CCCCC1CC(N1CC(O)(CN(C)C)C1)=O Cc1cc(F)ccc1NC(=O)C(N1CCOCC1C1CC1)c1ccoc1 c1(NCCc2ccc(F)cc2)cc(=NCC2CCC(F)(F)C2)[nH]cn1 CC(Cc1ccncc1)C(=O)N(CCNC(c1[nH]ccc1C1CC1)=O)CC1CC1 Cn1nc(CNC(C2CCS2(=O)=O)=O)cc1C(=O)NCCn1ccc(=O)cc1 c1(OCC(=O)NC2(C)CN(C(c3scc(C)c3)=O)C2)ccccc1O C12CN(C3CCN1C3)C(=O)N2.CC1CCCCC1CC(=O)OC(C)(C)C c1(OC)ccc(Cl)c(C(=O)NC2CC(CNC(c3ccnn3C)=O)C2(C)C)c1 N1(C(c2c(C)c[nH]c2)=O)CC(NC(=O)CC(O)C2CCCC2)Cc2ccccc21 C1(NC(C2(C(=O)NC)CC2)=O)CCCC2CN(C(c3conc3CC)=O)CCC12 N1(C(c2c[nH]c(=NC)o2)=O)CCC(CNC(=O)C(C)CS(C)(=O)=O)C(F)(F)C1 CC(C(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC(C)(C)C1)C(C)S(C)(=O)=O Cc1cccc(C)c1C(N1CCC(C(C)C(=O)NC2CC(O)C2)C1)=O N1(C(=O)Nc2cccc(O)n2)CCCN(C(c2cnc(C(F)(F)F)cn2)=O)CC1 c1(NC(N2CCN(C(=O)OCC)CC2)=O)ccc(SC2CC2)c(N)c1 c1(NC(C)=O)cccc(F)c1-c1ccc(C(=O)N(C)CCN(C)C)nc1 C1(C(=O)NC(C(C)C)C)CC(NC(=O)OC(C)(C)C)CN1C c1(C(=O)NCC23CC(NC(CC(C)O)=O)(C2)C3)ccc(OC(F)(F)F)cn1 c1(C(C)=O)cccc(C(N)=O)c1.N1(C(CCCN)=O)CCN(CCCl)CC1 c1(CC(N2CCN(C(c3cccc(OC)n3)=O)CC2)=O)c(C)cccc1C CCC(CC)(CC)C(=O)NCC1CC(C)CCN1C(=O)CS(C)(=O)=O c1(OC)cccc(C)c1C(N1CCC(c2ccccc2)(NC(=O)COC(C)C)C1)=O N1(C(Cc2c(SC)cccc2)=O)CC(C)CCC1CNC(=O)CNS(N)(=O)=O c1(NC(C2(O)CCN(C(c3ccc(Cl)cc3Br)=O)C2)=O)ncc([N+](=O)[O-])cc1O Cc1cnn2cc(C(=O)N(CCC(C)(C)C=O)CC(C)C)cnc12.N(C)C C1(C(N2CC(OC)C(F)C2)=O)CC2(CC2)CN1Cc1ccc(OC(F)F)nc1 C(C)(C)(CCCF)NC(C(CN(C)C)NC(=O)CC1(CN(C)C)CCC1)=O c1(C(N(CCC)CCNC(c2sccc2Cl)=O)=O)ccccc1OCC(C)C c1(C(=O)NC(CN(C(=O)C2=CCCSC2)CC)C)cc(C(C)C)n(C)c1C c1(CC(=O)NCC2N(C(c3cc(CC)c(CC)o3)=O)CC2)ccc(C)cc1C C1(Cn2cc(-c3n(C)cnc3)nn2)CCN(C(C2CCNC(=O)C2)=O)CC1 CC1CC2CN(C(c3cnc(C4CC4)nc3)=O)CC2N1C(=O)C(CO)NC(N)=O N1(C(c2c(OC)ccs2)=O)CC2CCC(CNC(=O)CC3CCCC3O)C2C1 Cc1nc(-c2ccc(Br)cc2)sc1C(C)NC(c1cc(C2CC2)ccn1)C C1(NC(c2c(C)coc2)=O)CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 O=C(CS(=O)(=O)C1CC1)NCC1CCC(CNC(=O)COCC2CCOC2)C1 c1(C(N2CCC(OCCNC(CCC3C(C)C3)=O)C2)=O)ccc2c(c1)C(=O)OCC2 C=CCCCCCC(=O)N1CCC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)CC1 C=CCCCCC(=O)NC(C)(CNC(c1ccc(C(C)C)cn1)=O)CO C1(C(=O)NC2C(CNC(c3cccc(N)c3O)=O)C2)Cc2cc(F)cc(F)c2O1 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)NCC1CC(Cl)=NO1 C#CC1CCCCN1C(c1n[nH]cc1CNC(=O)C(CC)N(C)C)=O c1(Cc2n(CCCOC)c(N(c3ccccc3)C)nn2)cc(C)cc(C)c1 CC(=O)C(C)CC(C)C(=O)NC1CCCC(CC(=O)NCc2ccc(F)cc2)C1 C=CC1CC1C(=O)NCC1(CC(=O)OCC)CC1 c1(C(N2C(CCNC(C(C)=C(CC)C)=O)COCC2)=O)cnc2n1C(C)CCC2 N1(C(CCC=C)=O)CCN(C(=O)CSc2ccsc2[N+](=O)[O-])C2CCCCC12 C1(C(=O)OCc2ccccn2)CCC(=O)N1C(=O)CCN1CCCCCC1 C(C)(C1OCCc2ccccc21)N(C(C(C)Nc1ccc(OC)cc1)=O)C C1(C(=O)NC(C)CC(=O)O)C2CN(C(=O)CN3CC4CC4C3)CC12 c1(C(=O)NCC2(NC(CN(CCC)C)=O)CC2)ccnc2ccc(O)cc12 c1(C(=O)NCCNC(C2CCC(C)S2)=O)ccc(CN2CCOCC2)cc1 c1(CC)cccc(F)c1.C1(NC(C2CCC(F)(F)C2)=O)CC2CCC(C1)N2 C(=O)(CCCN=c1nccc[nH]1)NCCOCCNC(C(C(C)C)(C)O)=O n1(C(C)C)ncnc1C(=O)N(CC(C)NC(=O)CCC1CCC(=O)N1)C c1(-c2n(C)cnc2)ccc2nnc(C(=O)Nc3scc(O)c3C#N)n2c1 C(=O)(C1=CCC(C)(C)CC1)NC(C(=O)Nc1c(C)cc(Cl)cc1)Cn1ccnn1 N1(C(C=Cc2nc(C)sc2)=O)CCCCC(C2CN(C(=O)C3=NOCC3)C2)C1 C1(OC)CCCCC1C(=O)N(C)CCN(C(=O)C(F)(F)c1cccnc1)C C(C(=O)NCCOCCOCCNC(=O)CSC1CC1)=CC=CC c1(C(=O)NC(CNC(C2C(C=C(C)C)C2(C)C)=O)(C)C)ccc(S(C)(=O)=O)s1 C1(COC2CN(C(CC(=C)C)=O)C2)CCN(C(=O)CN2CCCC(CC)C2)CC1 O=S(=O)(c1ccc(NCCCSC(F)(F)F)cc1Br)NCC(C1CCCC1)O Cc1ccc2c(c1)CCN2C(C1CCC(F)CN1C)=O N1(C(C2C(CC)CCCC2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)(C)C2CC2)nc1C c1(C(=O)NCC2(NC(CC(CC)OC)=O)CCCC2)cccn2cncc12 C1(C(=O)NC2(CCC)CC2)C=CCN1C(=O)C=CCN1CCOCC1 C(=O)(C1=C(C)CCC1)C(c1cnn(CCNCC2CC(SC)C2)c1)=O C1(CC(c2nnnn2CCCF)NCc2cc(C)c(Cl)s2)CCCC(C)(C)C1 c1(-c2nnc(C3CCC(=O)N3)s2)ccc(-c2nc(-c3ccccc3Cl)no2)cc1 c1(C(=O)NC(CNC(C2OCCN(C)C2)=O)C2CC2)cc(F)cc(F)c1 c1(C(N(C2CCCN(C(=O)CN3CCCCCC3)C2)C)=O)ncccc1Cl N1(C(C2(CC=C)CCN(C(c3cnn(C)c3C)=O)C2)=O)CCC(=O)N(C)CC1 C(=O)(C(C)SC(F)(F)F)N(CCOCCN(C(=O)C=CCF)C)C C12(CNC(CC=CC)=O)CCC(CNC(=O)CCCC3OCCO3)(CC1)CO2 C1(CC)CC(C(=O)NCCCc2ccsc2)CCN1C(=O)CC1CC(C)(C)CO1 C#CC1CCCC(NC(C2CCCC2CNC(c2cnnc(C)c2C)=O)=O)C1 C(=O)(C(O)C(C)CC)NCC(CC)NC(C1(c2cccnc2)CCC1)=O Cc1ncc(C(=O)NCC2(NC(=O)C=CC(F)(F)F)CC2)n1C c1(C(N(CCCNC(C(C(CC)O)C)=O)C2CC2)=O)ncccc1N=[N+]=[N-] C(=O)(C1=C(Cl)CCOC1)N(C)CC1COCCN1C(c1cc(F)n[nH]1)=O C1(CNC(C2(NC(c3[nH]ccc3C(C)C)=O)CCC2)=O)CC12CCC2.CCOC C(CC(C)N=c1nc(-c2cccs2)[nH]c2ccccc12)NC(C(C)SC)=O Cc1cc(C)c(NC(=O)NCC(N2CCSCC2)=O)cc1O N1(C(CN2CCN(C)CC2)=O)CCC2CC2(NC(=O)Cc2ccnn2C)CC1 N1(Cc2ncn(C)c2)CCC2(CC1)CN(C(C1CC1F)=O)C2 N1(C(C(C=C)O)=O)CCN(C(C2CN3CCN2CC3)=O)C(c2nccn2C)C1 N1(C(CC=CC=C)=O)CCC2CCC12CNC(c1c(I)c(NC)n(C)n1)=O c1(CC(C(C)C)NC(=O)COC2(CO)CCCNC2)ccc(Cl)cc1 N1(C(c2ccccc2NCc2cc(I)cc(I)c2O)=O)Cc2ccccc2C1 CC(c1ccccc1Cl)=CC(=O)NC(C1CCCC1)CNC(=O)C#CC(C)C c1(C(=O)NCC2(C)CCCN2C(=O)COCC2(F)CC2)ccn2cncc2c1 CCCCC(CNC(=O)Cn1cnnc1O)NC(=O)CN(C)CC C=CCC(CC)C(=O)NC1(CO)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2CCC(NC(=O)CNC(N)=O)(C2)C1 C1(C(=O)NCC2ON=C(CC)C2)CN(C(C2CC2(C)C(F)F)=O)C2(CCC2)C1 c1(C(N(C)CC2CCCN2C(=O)C(c2cncn2C)O)=O)cccc(F)c1 N1(CC)CCc2cc(-c3ccnc(NC(=O)NC(C)CF)c3)ccc21 C(CC(CNC(=O)C=C(Cl)Cl)NC(=O)C(C)OC(C)(C)C)OC C1(CNC(CCCC(=C)C)=O)CCC(C)(C)CN1C(=O)C=Cc1ccccn1 c1(C(=O)NC(C(C)C)C(C)NC(c2c[nH]cc2Br)=O)cc2sccc2n1C CC1CC(C(=O)NCC2CCC(NC(=O)COc3cccc(F)c3)CC2)C1(C)C Cc1noc(C)c1C(C)C(=O)NC(CNC(=O)CC1(C)OCCO1)C1CC1 c1(NC(=O)NCC2C(SC)COC2)cnc2c(c1)c(C)nn2CCO c1(-n2cc(CN3CC(O)CC(C4(C=C)CC4)C3)nn2)ccnc(P(C)(C)=O)c1 Cc1nc(C)c(-c2nnc(N(C(c3ccccc3)C(=O)N3CCCC3)C)n2C)s1 N1(C(C2C(=O)NCCCC2)=O)CCCC12CCN(C(=O)COC1CC=CC1)C2 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC2O)c(C)nn2cc[nH]c(=O)c12 c1(OC)c(CC(N2CCC(O)C(NC(C3CC3C)=O)C2)=O)cccc1F N1(C(c2ccc(N)cc2O)=O)CCC(C2CC2)(NC(=O)CSCc2ncc[nH]2)C1 N1(C(C=Cc2c(OCCC)cccc2)=O)Cc2[nH]nc(C(=O)O)c2C1 C#CCCCC(C)C(=O)NCC1CN(C(=O)CN2CCCCCC2)C1 c1(CC)cc(C(=O)NC2CCCCC2CNC(=O)C(CC)CO)c(C)o1 C1(OCC)CCCN(C(=O)C(C(C)O)NC(C2(OC)CCSC2)=O)C1 N1(C(c2cccc(SCC)c2)=O)CC2CCCC2(NC(=O)CCF)C1 Nc1cnc(C(=O)OCc2cccc(C(F)(F)F)n2)cn1 C1(NC(C2CC(F)C2)=O)CCCCN(C(=O)Cc2cccnc2O)CC1 c1(OC)ccc(SCCC(=O)NCC2CCCN(C(=O)CN(C)C)C2)cc1 C1(C(=O)NC(C(=O)NC(CC(=O)NC)C2CC2)COC)C2CCCCC12 N1(C(C(C)(CO)OC)=O)CCOC(C)(CNC(=O)CSC)C1 C1(CC)SC(C)CC(N2CCC(O)C(C(N3CCC(N(C)C)C3)=O)C2)C1C C1(C(=O)NC2CCSC2)CCCCCN1C(c1n[nH]c2c1CCC2)=O C1(C(N2C(CNC(c3ccnc(C)c3N)=O)CC2)=O)Cc2ccc(F)cc2O1 Cc1c(Cl)nc[nH]c1=NCC(O)CNC(c1cc2cccnc2s1)=O CC1(C)OC(=O)CC1C(=O)NCCN(C(=O)CC1CCC1(F)F)C1CC1 N1(C(c2cc(C)no2)=O)CCC(CCNC(c2ccc(O)c(N)n2)=O)CC1C Cc1nn(C)c2c(NCc3ccn(C(C)C)n3)nc(N3CCC(C4CC4)C3)nc12 CC1(C(=O)COc2cccnc2Cl)CCCOC1.N12CC3CC3(C1)NC(=O)CC2=O c1(C(=O)NC(C)CC2CN(C(=O)C=Cc3cnc[nH]3)C2)cnc2c(c1)CCCC2 N1(C(c2c(C)n[nH]c2)=O)CCOC(CN(C(=O)C(F)CC2CCCCC2)C)C1 C12(C(N(CC(=O)NC(C)(C)C)C)=O)CC(CO)(CN1C(C1CC3(CC3)C1)=O)C2 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2=O c1(N(C2CCSCC2)C)cc(N2CCC(C(C)(C)C)(CO)C2)nc(C(F)(F)F)n1 CN(C1CCc2ccc(Cl)cc21)C(=O)C(=O)NCCc1ccc2c(c1O)OCO2 C1(NC(CC)=O)CCN(C(=O)C(C)ONC(=O)OC(C)(C)C)CC1F c1(OCCCC(=O)NCC(CCNC(C(C)(C)NC(N)=O)=O)O)ccc(Cl)cc1 N1(C(c2cn(CCNC(CSCC#C)=O)nc2)=O)Cc2ccc(O)cc2C1 c1(SC)ncc(CNC(c2nnnn2CC2CC2)CC2CCCC2)s1 c1(N(CCCCCC)C)cc(NCC(C)(C)COC)nc(C(C)C)n1 c1(C(N(CC(C)(C)NC(C2CC(C)OCC2)=O)C)=O)cnc(O)cc1C(F)(F)F C1(NC(c2cnc(CC(C)C)s2)=O)CC2CN(C(c3cnn4cc[nH]c34)=O)CC12 c1(C(=O)NCCCC(=O)NCc2nc(C)sc2C)ccc(C)c(C#N)c1 c1(CN(C(=O)CC2CCC(C)(C)C2)C(C)C)nc2ccccc2[nH]1 C1(CC(=O)NCC2CN(C(C)C)C2)CCCCN(C(=O)CC(C)O)C1 N1(C(C(CC)F)=O)CCC2(CCC2)C(CNC(c2cccc3cccnc23)=O)C1 c1(C(N(CC2N(C(CC(=C=C)C)=O)CCCC2)CC)=O)nnn2c1C(=O)NCC2 c1(C(=O)NCC(C)NC(C2CCCC23CCC3)=O)cccc(C(N)=O)c1F c1(OC)ccc(C=CC(=O)NC2(CF)CCN(C(C3(C#N)CC3)=O)C2)cc1F c1(OC)cccc2c(NC(C)CCNC(=O)Cn3cc([N+](=O)[O-])cn3)ncnc12 N1(C(C(CC)NC(C)=O)=O)CC2CC1CN2C(=O)C(c1cncn1C)O CC1(C)CC2(CO1)CC(NC(c1ccnc(F)c1F)c1nnnn1CC(F)F)C2 CC1CCC(C)(C(=O)NCC(C)(C)NC(=O)Cn2nnc(C(C)(C)C)n2)CC1 C(=O)(CC1=CCN(C(C2CC(F)(F)C2)=O)CC1)NC(C#C)C(C)C CC(CCS(C)=O)N(C(=O)C(=O)C1CC1)C CCC(C(=O)NCC(C(C)C)NC(=O)CCc1nc(C)no1)Sc1ccccc1 c1(C(N(CCC(C)NC(=O)Cn2nnc(=O)[nH]2)C)=O)coc(-c2ccccn2)n1 C1(C(=O)NCC2(CNC(C3CN(C4CCOCC4)C3)=O)CC2)COC(=O)C1 C1(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)Cn2ncc(Br)n2)C2CC12 c12ccccc1-n1nnnc1C(NC1(C)CCC1)CC2.C1(CC)(CO)CC(C)C1 S(=O)(=O)(c1cccc(Cl)c1)N(CCNC(C1CC1C(=O)NC1CC1)=O)CCO C1(CNC(CCC#N)=O)CCCCC1NC(c1nn[nH]c1Cl)=O C=C1CCN(C(=O)CS(=O)CC)C(C(N2CCNC(=O)CC2)=O)C1 c1(C(=O)NCCCCNC(C2C(C)(C(=O)OCC)C2)=O)cnc(C2CCC2)s1 O=C(C1=NOC2(CCOC2)C1)NC1CCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 c1(SC(C(CC)C#N)c2cccs2)cc(C)ccc1C(=O)OC Cc1nccc(C(=O)NCC(C)(C)CN(C)C(C2(C(N)=O)CCC2)=O)c1C C(CN=c1[nH]c2cccc(C)c2s1)C1C(NCc2c(OC)nccc2)CCCC1 C(=O)(CCCC(C)C)NCC1(CO)CCN(C(c2c(C)nc(C3CC3)o2)=O)C1 c1(CN2CC(C(=O)Nc3ncc(Br)s3)SCC2)c(O)cccc1Cl C1(CNCC(CC)(C)CC)(CO)COCCN1Cc1ccccc1 Cc1nc2cc(C(=O)NCCC3CCCNCC3)c(F)cc2[nH]1 c1(-c2scc(C(=O)NC(c3ccccc3[N+](=O)[O-])C)n2)cc(F)c(O)cc1F CCCCC(C)C(=O)NCC1(NC(=O)CCC2OCCO2)CC(OC)C1 N1(C(C(=O)NCC)=O)CCCC(NC(c2oc(C(C)C)nc2C)=O)C(F)C1 Cc1c(C(N2CCC(CN(C)C(C3CCC(N(C)C)CC3)=O)C2)=O)cncc1N c1(C(N2CC(CNC(C(c3ccc(OC)cc3)(C)C)=O)C2)=O)cc(Cl)ccc1F CC1CCC(CC(=O)NCCCCCCNC(=O)CCCN2CCCCC2)OC1 CC1CCN(C(=NCCC2(C)CC2(F)F)NCCF)C1 c1(CC)ccc(C(C)(C)C(=O)NCCCOCCN(C)C(C2CC2CC)=O)cc1 C1(NC(C(C=C=C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(C(C=C)CC)=O)CCN(C(C2CCCN2CCC)=O)C(CCC)C1 c1(CCC(C)C)cc(C(=O)OCC(CN2CCN(CC)CC2)O)nn1CCO c1(OC)cccnc1C(=O)NC1CN(C(c2cc(C3CCCC3)no2)=O)C1 C1(CNC(c2ccc(F)cc2O)=O)CC2CCCC2N1C(=O)CCC1CC1(F)F O(NC(=O)C(O)C(CCC)NC(C1(C#N)CCOC1)=O)CCCC=C c1(C=O)cccc(C)c1C.C1(F)(C(=O)NC2C(OC)CC2)CCN(C)C1 c1(C(=O)NCCN(C(=O)CC2CCCOC2)C2CC2)cnc2ccccc2n1 c1(C(=O)NC2CN(C(C3C(OCC)C3)=O)CC2C)cc2ccoc2cc1F O=S(=O)(c1cc(Cl)c(F)cc1Cl)NC1CCCCC1Oc1ccc(Cl)cc1 c1(OCC)ncc(C(=O)NC(C)CCCNC(=O)CC(C)SC)cn1 N(C(=NCCCF)NCC(C)OC)Cc1c(OC)nccc1 C1(CNC(C(CC=C)CC)=O)CCC12CCN(C(=O)C(C)(C)CC)CC2 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(Cn2cc(CCOC(C)=O)nn2)C1 N1(C(C2CC(NC(c3cccc(I)c3)=O)C2)=O)CCC12CCCCC2 c1(OC)csc(C(=O)NCC2CN(C(=O)CCOCC(F)F)CC2C)c1OC c1(OC)cc(Br)c(F)cc1C(c1nnnn1C)NCC(=O)Nc1ccc(F)cc1 c1(NC(CC2CC3(CN(C(C(C(C)(C)C)O)=O)C3)C2)=O)cccc2ncsc12 N1(CC)CC(CNC(c2ccc(CNC(C3CCO3)=O)s2)=O)CC1=O c1(NC(C2CC(F)CN2C(C2CCCS2)=O)=O)nc(Br)cnc1Cl c1(C(=O)NC(C(C)C)(C)C)cc2c(s1)CCOC21CCN(c2ncccn2)CC1 C(CNC(=O)C(COC)N(C)C)(CC(C)C)NC(C1(CC#C)CCOC1)=O C(=O)(CCCCc1cnn[nH]1)N(C1CN(C(=O)C=C(Cl)Cl)C1)C c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cccc2nc(O)n(C)c12 c1(CC)[nH]nc(C(=O)NC2CC(CNC(=O)COCC3(F)CC3)C2)c1Cl C(C(F)(F)C(=O)N1CCC(F)(CNC(=O)C=CCN2CCOCC2)C1)OC C(C(C)(C(C)C)NC(=O)CO)NC(C(CC)C)=O.c1(OCC)ccc(Br)cc1 C(c1cnn(C)c1)=CC(=O)N(C1CCN(C(CCc2onc(CC)n2)=O)C1)C C(=O)(C(CNC(c1ccc(O)nc1)=O)C(C)(C)C)NC(c1ccccc1O)C c1(C(N2CCC(NC(c3c(C)ccnc3)=O)CC2C)=O)cc2c(nn1)OCCS2 c1(CC)noc(C)c1CNC(C1(C)CN(C(C2C3CC4C(C3)C24)=O)C1)=O C1(NC(c2ccc(CC)nc2)=O)CC2CCC1C(NC(C1C3CNC(=O)C13)=O)C2 C(=O)(CC(=O)NCCCOCCN(C(=O)C(C)CSC)C)OC N1(C(C2CC(O)(CNC(c3sccc3F)=O)C2)=O)C2CCC1CC(O)C2 N1(C(c2c(-c3ccc(C)cc3I)cncc2)=O)CCc2nc(C)sc2C1 c1(OC)cccc(CC(=O)OCC(O)COCC(F)(F)C(F)F)c1F C=C(C)CCCC(=O)N1CCN(C2CCN(C(=O)C(C)C3CCCO3)C2)CC1 N1(C(CC2N(C(C#C)=O)CCOC2)=O)CCC2(CC1)CC(=O)N2 C(=O)(C(CCC1CC1)NC(c1csc(CO)n1)=O)NC(C1CC(F)(F)C1)C O=C(CCCCCc1ccc(F)cc1)NC1CC(NC(=O)Cc2ccccn2)C1 c1(CCC)ccc(Cl)cc1-c1nc(-c2ccn(C)n2)nn1CC1CCCOC1 C1(C(N(CC(=O)N(CC(CC)OC)C)C)=O)CCC1(F)F C1(NC(C2CCCCS2(=O)=O)=O)CC2CN(C(C3CCC4CC4C3)=O)CC12 CCCCCC(C)(C)C(=O)NC(CC)CCCC(=O)NC1CCC(C2CC2)C1 C1(NC(C(NOC)=O)=O)CC2CCC1C(NC(C1CC3COCC3C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CCC(NC(C2(O)CC2)=O)C1C N1(C(CC(=C)C)=O)CCC(NC(c2ncoc2-c2ccco2)=O)CC1C Cc1ccc(C(N2CCCC(C)(NC(=O)C(C)C#N)C2)=O)cc1Br C1(CNC(C2C(C)=C2)=O)CN(C(c2occ3c2CCC3)=O)CCC1(C)C c1(C(=O)NCCCNC(C(C(CC)CC)OC)=O)c(O)nnc2c1CCC2 C1(C(=O)N(C2CCC(O)CC2)C)(COC)C=CCN1C(c1csc(C)n1)=O c1(SC)nn(C)cc1C(=O)NC(C)CC1CCN(C(C2OCCOC2C)=O)CC1 N1(C(C)=O)CCc2ccc(NC(=O)C(C)Oc3ccc(CO)cc3)cc21 C1(OC(C(c2cc(C)no2)(C)C)=O)CCC(F)(F)C1 Cc1cc(=NC(=O)C(=O)NCC(C2CCCC2)NC(C2CC=CCO2)=O)[nH]o1 C1(C(=O)NC(C)CC(C)NC(=O)Cn2cc(N)cn2)(CC)CCNC1=O C(=O)(C(C)(C)C(=O)N1CC(NC(=O)C=CCN2CCC2)C(CO)C1)OCC N1(C(COCC=C)=O)CCN(C(c2ccc(N3CCCC(O)C3)cc2)=O)C(C)C1 c1(NC(C2CC(NC(c3cc(Cl)sc3Cl)=O)C2)=O)c(Cl)ccc2cccnc12 C1(C(=O)NCC2CCC(CNC(c3cc(C)oc3C)=O)CC2)CC2CC2CC1C Cc1ccc(C)c(NC(=O)C(Cn2cncn2)NC(=O)C(=O)CC(C)C)c1 c1(C(C)=O)cn(C)nc1C(=O)NC(C)CC(C)NC(C1CCC(C)O1)=O O(NC(=O)C(C)C(C)NC(c1coc(CC)n1)=O)CC C(C)(C)(C(C)CC(=O)NC1CN(C)CC1(F)F)NC(CCSCC)=O c1(CC(N2CCC(OCCNC(c3ncc(N)nc3)=O)C2)=O)csc2nccn12 Cn1cnc(C(=O)NCC23CC(NC(C4CCCN4C=O)=O)(CO2)C3)cc1=O C=CCC(C(=O)N(CCCCN(C)C(C1(CN(C)C)CCCC1)=O)C)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CCOC2(CNC(C2(N(C)C)CC2)=O)C1 N1(C(C2N(CC)CCC2)=O)CCN(C(c2cc(C(C)=O)cs2)=O)CC1C(C)(C)C Cc1noc2nc(C(=O)NC3CCC(CNC(c4cnco4)=O)C3)ccc12 C(=O)(C1CCc2ccccc21)NCC(C)(C)NC(=O)C(F)=CC1CC1 n1(C(C)C)ccc(C(=O)NC23CC2CN(C(C2(n4cccc4)CC2)=O)C3)cc1=O C(CCCC(C)(C)C(=O)NNC(=O)C1(F)CC1C)NC(C1C(=C)C1)=O c1(C(=O)NCCOCCCNC(CCC2C(C)=NOC2=O)=O)c(C)nc(C)n1O C1(CN(C(CC2(COC)CCCC2)=O)C)CCN(C(=O)C(C)N(C)C)CC1 CC(C)C(C)(C)C(=O)N1CC2C(CC(=O)NCC3CC34CCOCC4)C2C1 c1(C(N(CC(O)CN(C)C(C2(C(F)(F)F)CCCC2)=O)C)=O)cc(C#N)ccn1 C(=O)(C(C)(C)C(F)F)N(CC(CNC(C(c1ccc(C)cc1)C)=O)C)C c1(OCC(=O)OCC(=O)NCc2nc[nH]n2)c[nH]nc1C(F)F.C12CC(C1)CO2 C1(C(=O)NC(c2cn(C(C)C(=O)NC3CC3)nn2)CCC)CCCS1(=O)=O C(C(O)CN=c1[nH]nc(C(C)C)o1)NC(C1CCC(C(=O)OC)C1)=O C1(C(=O)NCC=CC(=O)N(CC(C)O)CC(C)O)CCCC(F)C1 c1(C(=O)NC2CCCN(C(c3n(CC)ccc3)=O)C2C)cccc2c[nH]nc12 N1(C2CCN(C(c3c(SC)ccs3)=O)C2)CCC(NC(=O)C2=CCC2)CC1 CN1N=CC(CC(=O)N(C2CCCC2)Cc2ccccc2)C1=O C1(OC)CC(C(=O)NC2CCC(C(N)=O)C2)N(C(=O)CCC2CCC2)C1 C#CCCCCC(=O)N1CC(=O)NCC1C(N1CCC(O)(C#C)C1)=O C1(C)(NC(C(C)OC2CCCC2)=O)CCN(C(=O)COCC2CCCCO2)CC1 C1(NC(c2nc(C3CC3)cs2)=O)CN(C(C2CCCCCC2)=O)C2CCCCC12 c1(CNC(=O)NC2(C3CCCCC3)CC2)c(Cl)oc2ccccc12 N1(C(C2(C#C)CN(C(=O)C(C)=C3CCCC3)C2)=O)CC(C)C(C)C1C C12(CC(=O)NC(C3CCN(C(C=CCN(C)CC)=O)C3)C)CCC(CC1)C2(C)C Cc1ccc(C=CC(N2CCC(C(C)NC(c3cc(O)nc(Cl)c3)=O)C2)=O)cn1 c1(N2C(COCC)CCC2)nnc(-c2ccccc2C)n1Cc1ccc(CC)s1 C(=O)(CC(F)(F)F)NCC(=O)N(CCNC(C1C(C)CC1)=O)CC1CC1 N1(C(C(C)(C)c2cccs2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C(=O)(CN(C(=O)CN(C)CCOCCOC)C)N(CCC)CCC N1(C(CC(=O)OC(C)(C)C)=O)CCN(C(c2cnnc(O)c2)=O)C(CC(F)F)C1 Cc1ccc(C(=O)NCCC2CN(C(C3(C(N)=O)CCC3)=O)CC(C)O2)c(Cl)c1 c1(C(=O)NCCOCCNC(c2c(C)ccnc2C)=O)sccc1S(N)(=O)=O N1(C(C(C)SCC)=O)CCN(C(=O)C(O)C2CCCC2)C(CCO)C1 CCCC(O)(CCC)CC(=O)N1CC(O)(C2(CNC(=O)CCNC(N)=O)CC2)C1 Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCCC(C)(C)C)CC3F)c2c1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(=O)NCC2CN(C(C(C(C)O)(F)F)=O)CC2(C)C)cncc2ccsc12 C(=O)(C1CCSc2ccccc21)Nc1c(C#N)cc(Br)cn1 c1(C(c2nnnn2C(C)C)NC2(CC=C)CCC2)ccc(Cl)cc1F Cc1cc(CC(=O)NC2CC(=O)N(c3cnn(C)c3)C2)ccc1O C(C)(C)(CC(=O)N1CC(O)(CNC(=O)Cc2ccccc2C(C)C)C1)OC c1(NC(C2CCCCN(c3cc(Cl)c(O)nn3)C2)=O)cccc(C2CC2)c1F CCCC(C)(O)C(=O)NC1CCC(CNC(c2ccc(Cl)o2)=O)CC1 C12CN(CCN1c1nnc(C3CC4(CCCC4)C3)n1C)C2.c1(CC)ccccc1 c1(C(=O)NCC2CN(C(COc3cn(C)nc3)=O)C2)cnc(O)nc1O c1(OCC(C)(C)NC(C2CCC(CC)C2)=O)ccc(F)cc1 c1(CC(=O)Nc2cccc(CNC(C3CCC(F)(F)C3)=O)c2)cc(Br)ccc1O N1(C(=O)NC(C2(C)CCCO2)c2cccs2)CCC(Oc2ccccc2)CC1 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1CCCCN(C(c2nc(CC)oc2)=O)C1 c1(C(N2C(CC(=O)Nc3cc(I)ccc3F)CCC2)=O)cnc2ccccc2n1 c1(CC)n[nH]c(=NCC2CN(C(c3ccc(OC(F)F)cc3)=O)C2)s1 Cc1cc(Cl)ncc1NC(C1(CNC(=O)CC2OCCC2(C)C)CC1)=O C1(NC(CC(N)CC2CCCCC2)=O)CCc2c(cnn2CCO)C1 N1(C(CCCC(=O)OC)=O)CCCC(C)(C)C1C(=O)NCCc1ocnc1CO CCC(C)C(C)C(=O)NC1CN(C(=O)CNS(=O)(=O)N(C)C)CCC1C c1(CC)ccc(C)c(C(N2CCC(C)(CCNC(C3CC(OC)C3)=O)C2)=O)c1 N1(C2C(c3cn(CCC)nc3)C2)CCCCC1c1cn(-c2ccccc2C)nn1 n12cc(cn1)C(=O)NCC2.n1(CCOC)cc(-c2csc(C)c2)nn1 c1(C(N(CCCN(C)C(c2cc(CO)n(C)n2)=O)C)=O)ccc2ccoc2c1 N1(C(=O)Cc2ccsc2)CC(C2CN(C(=O)CC3CCSC3)C2)C1 c1(CC(=O)NC2CCC(F)(F)C2)cnc2n1CCOC2.n12cc(nn1)CNCC2 c1(C(N(C2CN(C(c3[nH]c(=NC)sc3)=O)CC2(C)C)C)=O)cnc2[nH]ccc2n1 N1(C(C2C(C)C2C)=O)CC(NC(c2ccnc(N(C)C)c2)=O)C2(CCOCC2)C1 C1(C(=O)NCC)C2CC3C(C2)C13.n1(C)cc(CN=[N+]=[N-])cn1.C12CC(C1)NC(=O)C2 CC1CCCC(CC(=O)NC(CN2CCC2)C(C)(C)C)O1 N1(C(C)=O)C(CN)CC2CC12.C(=O)(C(C)(C)OCCCF)NC c1(C(=O)NCCC2CCCN(C(CC(COC)C)=O)C2)cn2cccnc2n1 n1(C2CCN(CCNC(N3CCC(OC)CC3)=O)CC2)cnc2ccccc12 c1(C(=O)NC2CCC(NC(C3N(C)CCCC3)=O)CC2)ccc(O)c(CO)c1 N1(C(C(C(C=C)C)C)=O)CC2(CCN(C(=O)CCCc3cccc(Cl)c3)CC2)C1 C1(NC(CC2(C=C)CC2)=O)CCC(O)CN(C(=O)C(F)C(F)(F)F)C1 N1(C(C2C(=C)CC2)=O)CCN(C(c2cccc3cncn23)=O)C2(CC2)C1 N1(C(CC(C)CF)=O)CC(NC(c2cncc(C(F)(F)F)n2)=O)CC(F)C1 c1(NC(C)CNC(c2cncc(Cl)n2)=O)ncnc2ccc([N+](=O)[O-])cc12 N1(C(c2cnccc2Cl)=O)CCC(N=c2[nH]c3cc(F)cc(F)c3o2)C1 N1(C(CCc2ccc(OC)nc2)=O)CC2CCC1CN2C(=O)C(C)NC(N)=O c1(C(N2CC3C(CN(C(C4C(=C)CC4)=O)C)C3C2)=O)csc2c(OC)cccc12 C1(CC(=O)NCC2(F)CC(CNC(c3cc(CC4CC4)on3)=O)C2)CCC2CC12 c1(CC)cc2c(N3CCN(C(C4CC4C4CC4C)=O)CC3C)ncnc2s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)C(C)NC(C2(O)CC2)=O)cc1 C1(CNC(CC=CC)=O)CN(C(c2nnn3c2COCC3)=O)CCC12CCOC2 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(C=CC)=O)(C)CC CC(O)(CC(=O)N1CCCC(F)(CNC(=O)Cc2ncc(Cl)s2)C1)C(F)(F)F C1(CNC(CCNS(C)(=O)=O)=O)CC2(CCC2)CN1C(C1CCOC(=O)CC1)=O C(=O)(C(F)(F)CCn1cccn1)N1CC2C(CNC(C(C)(C)SC)=O)(C2)C1 c1(CC)nc(C(=O)NC23CC(C(N4CCC(OCCN(C)C)C4)=O)(C2)C3)c(C)o1 c1(NC(C(c2cnn[nH]2)N(CCCCC)C)=O)ccc2c(c1)OCCO2 C(C)(CNC(c1n[nH]cc1Br)=O)(CO)NC(CC1CN(C)C1)=O N1(C(COCCOCC#C)=O)CCC(C(=O)NCC2C=CCCC2)C(C)(C)C1 C12(NC(c3c(C)nc(C(C)(C)C)s3)=O)CCN(C(C3(S(C)(=O)=O)CC3)=O)CC1C2 N1(C(=O)NC(c2ccc(SC(F)(F)F)cc2)C)CCN(C)C(C)C1C N1(C(c2ccnc(C)n2)=O)CC2CCC2(CC(N2CCC(OCC(N)=O)C2)=O)C1 Cc1c(C(N2CC3CCN(C(=O)CN4CC(=O)NC4=O)C3C2)=O)sc2nccn12 Cc1oc(CO)cc1C(=O)NCC(C)(F)CNC(C1(C)CCCC1C)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCC2C(CCN2C(=O)C(C)NS(C)(=O)=O)C1 C(CCCCCC(=O)N1CC(CNC(=O)C(=Cc2cccnc2)F)C(C)C1)SC c1(C(C)C)ccc(C(=O)OCC(C)CN(C)C(C2CCOC2)=O)o1 C1(NC(C(C)C(C)O)=O)CCN(C(=O)Cc2cccs2)CCC1CO C1(C(=O)NCCOCCN(C)C(c2cc(=N)[nH]c(=N)[nH]2)=O)Cc2cscc2C1 c1(CC(=O)NCC(C)NC(C2(F)CCOC2)=O)ccc(C(N)=O)nc1 N1(C(C2(CC#C)CCCO2)=O)CC2CC(NC(C3CCC(C)C(C)C3)=O)CC2C1 C1(C(N2CCC(=C)CC2)=O)CC(OCCNC(=O)COC)C12CCC2 c1(CC(=O)NC(C)C(C)NC(=O)CCF)nc(NC(=O)OC(C)(C)C)no1 CC(CN=c1ccc(S(=O)(=O)N2CCCSC2)c[nH]1)N1CCCC(C)C1 Cc1cc(C(N2CCCN(C3CC3)CC2)C(=O)NC(C)C)c2c(c1)CCC2 C=C(C)C(O)CC(=O)NCC1(CNC(=O)C(C(C)(C)C)SC)CCCC1 c1(C(=O)NCC2C(CNC(C(C)(C)C3CC3)=O)C2)cnc2c[nH]nc2c1 N1(C(C2C(COC)C2)=O)CCCC(C(=O)NCCc2ccc(C)s2)C1 N1(C(C(=O)NCC)=O)CC2CC2(NC(=O)CCC2CC(C)(C)CO2)C1 C#Cc1ccc(C(N2CC3C(NC(c4cccc(C(N)=O)c4F)=O)C3C2)=O)nc1 C1(NC(C(C)=C(C)C)=O)CCN(C(C2CCCCC2)=O)C1c1ccccc1 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCC(NC(c2cnc(C)o2)=O)C1 C1(C(=O)NC2C(C)CN(C(C34CCC(C)(CO3)C4)=O)C2)CNC(=O)CC1(C)C Cc1cccc(OC(C)C(N2CC(F)CC2CNC(C2(C#N)CCCO2)=O)=O)c1 C1(C(N2C(C)COCC2C)=O)CNC(=O)C12CCN(C(C1(C3CC3)CC1)=O)CC2 C1(CC)CCC(NC(=O)C(C2(O)CCC2)NC(=O)CCN(C)CCOC)CC1 C(=O)(CCCCC(=O)NC12CC(C1)N(C(c1nnc(O)nc1O)=O)C2)N(C)C N1(C(C(c2ccccc2Cl)C)=O)CC(N(C(=O)CCCC2CCC2)C)C(O)C1 C1(CC(=O)NCC(CNC(C(c2cccnc2)OC)=O)C)CCCC(F)(F)C1 CCCCC(C(=O)N1CCC(CCC(=O)NCCCn2ccnc2C)C1)N(C)C CCC(C)CC(=O)NCC1CCCN1C(=O)C(C)=C1CCCC1 N1(C(CC2(OC)CCCCC2)=O)CC2CCCC(CNC(=O)CP(C)(C)=O)C2C1 CCC(C(C)(F)F)NC(=O)COC1CN(C(=O)CC(F)(F)F)C1 c1(C(=O)NCC(C(C)C)(C)NC(c2ccnnc2)=O)cccc2c1OC(F)(F)O2 C#CCC(C)(CC)C(=O)NCCC1CC(NC(C2(C#N)CCSCC2)=O)C1 c1(C(=O)NC(C(=O)OC)(C)C)ccc(OC(F)(F)F)c(-c2ccccc2F)c1 Cc1sc2ccccc2c1C(N1CC(O)(C(C)NC(C2CC3CC3C2)=O)C1)=O N1(C(COCCC)=O)CC2CCCC(NC(=O)C(N3CCC(O)CC3)C)(C2)C1 c1(C(C)(C)NC(c2ccc(OC)cc2)=O)ccc(-c2nn[nH]n2)c(O)n1 C(c1cn(C)cn1)=CC(=O)NC1CCC(N(C)C(c2ccc(C(N)=O)o2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)NCC(c1ccccc1)N(C(=O)Cc1nnc(O)s1)C Cc1nc(NCCN(C(c2ccc(CO)o2)=O)C2CC2)c2cnn(C)c2n1 Cc1nccc(C(N2CC(C3CC3)(C(=O)NOCC(F)(F)F)C2)=O)c1N c1(CC)oc(C(N2CCCC(CNC(C3CCCC(CF)C3)=O)C2)=O)cc1C c1(C(C)C)nccc(C(=O)NC2CCC2NC(=O)CSc2ccc(O)cc2)n1 C1(NC(CC(C)(C)O)=O)CC2CCC1N(C(=O)CN1CCCC(C(=O)O)C1=O)C2 N1(CCC(=O)N(CC(C)NC(CNC(=O)OCC=C)=O)C)CCNC(=O)C1 c1(C(N(CC(=O)NCC2CCN(C(N)=O)C2)CCOC)=O)sccc1C#N C#CCCCCC(=O)Nc1cccc(CC(=O)NCCCN2CCC(O)C2)c1 c1(C(C(=O)N(C(C)CO)CC)C)cccc(Br)c1 N(C(=NCCC1OCCC1(C)C)NCC1CCOC1)Cc1c(Br)cn(CC)n1 C1(NC(C2C(C)(CC)C2)=O)CCC(C(=O)NCC2(N(C)C)CCCC2)CC1 Cc1ncc(C(N2CCC(O)(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)cc1N N1(C(CC2CCC(C)C2)=O)CCOCC(CNC(C23CC(CN2C2CC2)C3)=O)C1 C1(OC)(CNC(=O)C(C2CCCCC2)NC(=O)C(CO)N(C)C)CCCCC1 C1(C(=O)NCCCC(C)NC(=O)CCC(F)(F)F)CCCC(C)(C)C1 c1(C(N(CCN(C(=O)CCNC(=O)CO)C(C)C)C)=O)c[nH]c(Br)c1 C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(c3ccc(Cl)s3)=O)C2)=O)c1 N1(C(c2cnn(C3CC3)c2)C(=O)NCCCF)CCCC(c2cnco2)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCC(NC(=O)CC23CCC(CC2)C3)CC1C C1(O)(C(=O)NC2CCCC(NC(c3ccsc3Cl)=O)CC2)CC2(CCOCC2)C1 N1(C(C(C(C)OC)NC(C2CNC(=O)O2)=O)=O)CC2CCN(C)C2C1 C1(C(=O)NCC2N(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCC2)CCC(C#N)C1 Cc1ccc(OCC(=O)N(CC(O)CNC(c2ccc(O)c(N)c2)=O)C)c(C)c1 C1(NC(=O)Nc2cccc(C(N)CO)c2)CCn2nnnc2C1 C1(NC(C(CC)=CC)=O)CN(C(c2cnn(CCO)c2N)=O)CC2(CCC2)C1 N1(C(C2(NC(c3cc(C)on3)=O)CCCC2C)=O)CC2CC(C)C2C1 C1(O)(CC(N2C(C(CNC(Cc3c(C)ccs3)=O)(C)C)CCC2)=O)CCCCC1 C(=O)(CCCN=[N+]=[N-])N(C)CC1CCCN(C(C2(F)CC=CCC2)=O)C1 C1(c2n(C)cnc2)CN(C(=O)C2=CCC2)CC1NC(c1cc(Br)c[nH]1)=O Cc1ccc(Cl)c(O)c1C(=O)NCCNC(C1(C)C=CCCC1)=O Cc1cccc(S(=O)(=O)NCCC(C)C(=O)O)c1Cl C(=O)(C(F)CC)NC1CC(CCC(N2CC(CC)C2)=O)C1 c1(C(=O)NCCC2(NC(CCC#C)=O)CCCC2)c(OC)cccc1Cl CC(C)(O)CC(=O)NCC1CC(NC(c2ccnnc2NC2CC2)=O)C1 c1(C(=O)NC2CC(CNC(C(C)CC(F)F)=O)OCC2)cc2c(cn1)COCC2 N1(c2cc(NC(CCCN(CCO)CC)C)ncn2)CCC2(CCCCC2)C1 Cc1conc1CC(=O)NCC1CCN(C(=O)C(C)OC2COC2)C1 N1(C(C2(C#C)CC2)=O)CCCC(C2(NC(=O)C(C)NC(=O)NC)CC2)C1 C(=O)(CC(C(F)F)c1ccccc1)NC(CC(C)NC(c1cnc[nH]1)=O)C c1(C(C(=O)NCC(F)F)N(C(COC)(C)C)C)ccc2ccccc2c1C C(C(C)C)(C(O)C(=O)NCCN(C(C1(c2ccccc2)CC(C)C1)=O)CC)OC c1(CCNC(C2CN(CCN3CCCC3)CCC2O)=O)ccc2c(c1)OCO2 c1(CNC(=O)NCCN2CCC(C)(CSC)C2)nc2sccn2c1C C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1nccn2ccnc12)=O C1(NC(Cc2c(C)nco2)=O)CC2(C1)CC(NC(c1onc(C)c1C)=O)C2 CN1CC(C(=O)OC(C)(C)C)CC12CCC2.C12CCCN(C1)C(=O)Cn1cc2nn1 C1(C(N(CCC(=O)NCCCc2cc(C)no2)CC#C)=O)CC=C(C)CC1 N1(C(c2cc(OC)no2)=O)CCN(C(=O)C(F)(F)c2nccn2C)C(C)CC1C CC(C)C(CC(=O)Nc1cccc(C2CC2)c1)NC(=O)C#CC(C)(C)C CC(C)C(O)CC(=O)NC1CN(C(c2scnc2C(C)(C)C)=O)CC1CC1CC1 C1(F)(CNC(C=CCOC)=O)CC(NC(=O)C=Cc2cocn2)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)C(C)CC2CN(C(c3coc(C)n3)=O)CC12 C(CC(C)C(=O)N1CCC(C(C)C(=O)NC(CCOC)C(C)C)C1)=CC c1(-n2cc(CC(C(F)(F)F)N3CCOCC3)nn2)ccc2cccc(Cl)c2n1 CC(N=c1[nH]c(=NCc2nnc(CO)s2)[nH]c2c(F)cccc12)c1csnn1 c1(NC(C2(NC(CC=C)=O)CC(CO)C2)=O)cnc(Cl)c(C)c1 c1(C(N2CCCC(NC(c3cc[nH]n3)=O)(CO)C2)=O)cc(Br)ccc1[N+](=O)[O-] N1(C(CCC(C)(C)F)=O)CCC2(CC1)CCN(C(=O)CN1CC3C=CC1C3)CC2 c1(C(C)=O)ccc(C#N)c(N2CCCCC2)c1.c1(N2C(=O)CCC2)ccc(F)cc1 Nc1cc(F)c(F)cc1C(=O)NCC1CCCC1NC(=O)Cn1ccccc1=O C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(CNC(CCC#C)=O)=O)C(O)C1 C1(CC(=O)NC2COCCN(C(c3csc4nccn34)=O)C2)CC2(CCC2)CO1 C=CCC(C)(CC)C(=O)N1CSCC1C(N1CC2(C1)CC2(F)F)=O c1(CC)nc(N2CCCC(NC(c3c(C(F)(F)F)cnn3C)=O)CC2)[nH]c(=N)n1 c1(CNC(=O)CC2CC2)nnc2n1CCN(C(c1ccc3cccnc3n1)=O)C2 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C)c2C(F)F)=O)c(N)c1Cl N1(C(C2(C)CCN(C(c3c(C)cc(CC)o3)=O)C2)=O)CCC2(CCC(O)C2)C1 N1(C(C(CSC)(C)NC(=O)C#CC2CCC2)=O)CCc2nc[nH]c2C1 c1(NCC2CCC(CCCCC)O2)ccc(=N)[nH]n1 Cc1ccoc1C(=O)NCCC1CN(C(=O)C=CCN2CCCC2)C1 O=C(C#CC1CCOC1)NCC1(C(=O)NCC(F)C2CCC2)CC2(CC2)C1 N1(C(c2ccc(CCC)s2)=O)CCN(C(=O)CC2CC(COC)C2)C(CC)C1 C1(CC(=O)NC(CNC(c2cc(CCC)[nH]n2)=O)CC)CC(O)C12CCC2 N1(C(=O)Cc2ccc(Cl)cc2)CCCC2C1CCN2C(=O)Cc1ccncc1 N1(C(C=CC)=O)CC(C2CCCN(C(c3[nH]c(=N)sc3-c3ccccc3)=O)C2)C1 c1(C(=O)NC(C2CCCN2C(=O)CCc2ccccn2)C)nn(C(F)F)cc1Cl CC(C)C(O)CC(=O)N1CC(F)(F)CC1CNC(c1cnn(C(C)(C)C)c1)=O c1(SC)c(CNC(c2cnc(OCC(F)F)cn2)=O)cccc1C c1(CC)cccc(CC)c1CC(=O)NCC(C)CN(C)C(C12CC(F)(C1)C2)=O c1(CNC(C2CCC(NC(c3ncccc3Br)=O)C2)=O)ccnc(F)c1 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cccc2nonc12 C1(C(=O)NCCC(C)N2CCCC2)C=CC(NC(=O)CCc2cn(C)nn2)C1 c1(C(N2C(CNC(C3CCO3)=O)CCC2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C2CCNCC2)(C(=O)NCC(C(C)C)=O)CCOCC1 C#CC(C)(C)C(=O)NCC1CCCCN1C(c1c(C)noc1CCC)=O c1(C(=O)NCC2N(C(C(C)n3cccc3)=O)CCOC2)noc2ccc(Cl)cc12 c1(C(N(C(C2CCC2)C)C)C)cccc2ccccc12 C(CC(O)C(=O)NC1CN(C(C)C)CC1C)NC(c1c(C)con1)=O N1(C(CCOC)=O)CC(C)(C)CC1CC(N1C2CCC1COC2)=O c1(C(N2C3CCN(C(C(CCC)O)=O)CC3C2)=O)cc(=O)c2ccc(F)cc2o1 C1(CNC(c2n(C)nc(O)c2)=O)C(O)C(O)CN1C(=O)C=CCO c1(CCN(CC(C)NC(C2CC(OCC)C2)=O)C)cccc(Cl)c1 C(c1ccnn1C)=CC(=O)OC(CC(N(C(=O)C=CCN1CCCC1)C)C1CC1)=O CCC(C)(CC)NC(=O)C(C)CN(C(=O)C(F)F)C c1(OC)cc(CNC(C2OCCC2CNC(C2(C3CC3)CC2)=O)=O)n(C)n1 C=CC(C)(O)CC(=O)N1CC(F)CC1CC(=O)NC(c1cnn[nH]1)C c1(CC(N2C3(CN(C(c4ccc(=O)oc4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C)(C(=O)NC(CCCNC(C2C(C)=CCS2)=O)(C)C)CCCCNC1=O N1(C(CC(CCC)CC)=O)CCC2(CCCN2C(=O)C(C(C)C)SC)C1 CC(C)(CC(=O)N1CC(NC(c2sc(F)cc2Cl)=O)C(O)C1)CC(F)F c1(C(=O)NCCCCNC(=O)CC2CCCOC2)c(F)cc(Cl)cc1Cl c1(CC)cnccc1C(N1CC2C(C(N3CC(C)=C(C)C3)=O)C2C1)=O CC(CNC(=O)CC(=O)N(C)C)CC(=O)Nc1ccc(F)nc1 N1(C(C(C)NC(=O)OCC)=O)CCCC(C(C)NC(c2cccc(SC)n2)=O)C1 c1(CC(=O)NC(C2C(C(=O)NCC3(OC)CC3)C2)C)n[nH]c(C)n1 c1(C(C)=O)ccc(N(C)CCN(C)C(C23CCC(CC2)CC3)=O)c([N+](=O)[O-])c1 c1(NC(C=CC(CC)C)=O)nn(C)cc1N N1(C(C(C)=C(C)C)=O)CC(C2(NC(=O)COCc3ccccc3Cl)CC2)C1 C(CC1=CCOCC1)NC(c1c(CNC(C(COC)(C)C)=O)ccs1)=O C1(C(=O)Nc2cccc(NC(CCCCC(N)=O)=O)c2)Cc2c[nH]cc2S1(=O)=O N1(C(C2C(CC)C2)=O)CCCC(C2CCN(C(c3ncn(C(C)C)n3)=O)CC2)C1 C1(NC(CN(CCC)C)=O)CC2(CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 C1(CC(=O)NCc2cn(CC)nn2)CN(C(=O)C(C(C)O)N(C)C)CCO1 Cc1ncc(C(=O)NCc2ccc(C(=O)NCCc3ncc[nH]3)s2)s1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C23CC(F)(C2)C3)=O)CC1S(C)(=O)=O c1(CC)cnccc1C(N1CCC(CO)(NC(=O)Cc2ccoc2C)C1)=O N1(C(C2(C)CC2)=O)CC2OCCN(C(=O)C(O)Cc3cnc[nH]3)C2C1 C(=O)(C(CC)CC(F)F)NCC1C(NC(CC=C)=O)CCC1 c1(C(C(=O)NCCN(C(C2CCC(CC)C2)=O)CCOC)F)cccc(C)c1 N1(C(C(CC)OC2CCCC2)=O)CCC(C2(NC(=O)C3=CCCOC3)CC2)CC1 C(C(=O)N1CCCC1(C)C(N1CCC(CN=[N+]=[N-])C1)=O)(C(C)(C)C)OC Cc1cc(C(C)C)nc(=NCCNC(c2c(C)oc(C)c2C)=O)[nH]1 c1(CNC(C2C3CCC2(c2cccnc2)C3)=O)cncc2cnccc12 C(=O)(C(F)CC(C)(C)NC(=O)CC(C1CC1)C1CC1)NCC(CSC)OC C1(N(C(=O)COCC2CCCO2)C)CC2CC1N(C(C1CCCCCC1)=O)C2 C(=O)(C#CC1CCCO1)N1CC2C(Nc3nc(OC)nc(OC)n3)C2C1 N1(C(C=CC(C)(C)C)=O)CCCC(CCC(=O)N2CC(F)C2)C1 C1(C(=O)NCCC2(NC(C(CCSC)O)=O)CCCC2)CC(=O)N(C)C(=O)N1 Cc1ccc(-n2ccnc2SCC(=O)Nc2cnn(C)c2Cl)c(C)c1 C1(CN(C)C(C2CCC(C(N)=O)CC2)=O)COCCN1C(C1CC(F)(F)C1)=O C(=O)(C1=NOC(C)(C)C1)NC1C2(CCN(C(CCCN(C(=O)OCC)C)=O)C2)C1 C1(NC(=O)CCCc2nccs2)(CO)CCN(C(=O)CC2CCC=CCC2)C1 C1(C)(NC(CN2CCC(C)CC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(CC)CCCCC)N1C(CC=C)(C(=O)NC2CC3(C2)CC3(F)F)CCC1 C(=O)(C(C)(F)C(C)(C)F)NC1C=CC(C(=O)NCc2[nH]nc(C(C)C)n2)C1 C1(C(=O)NC2C(NC(CCC(C)(C)F)=O)COC2)CSC(c2ccccc2)=N1 Cc1cn2cc(C(=O)OC3CCC(C)CC(C)(C)C3)nc2c(C)n1 C#Cc1cnn(C)c1C(=O)NCC1CC(NC(c2c(C(=O)OC)n[nH]c2C)=O)C1 CC1CCCC(C)N1C(=O)C(N1CCOCC1CNC(=O)COCCN(C)C)=O c1(CN2CC(NC(Cc3ccc(OC)cc3)=O)C(C)C2)cc(Cl)c(O)cc1F N=c1[nH]nc(CC(=O)NCC2CCCN2C(=O)CCCOc2cccnc2)s1 C1(NC(C2CCC3C(C2)C3(F)F)CCl)CCSC12CN(CC1CCCCCC1)C2 Cc1cc(=NCc2c(F)ccc(F)c2F)[nH]c(NC2CC3(CCCC3)C2)n1 Cc1ncnc(C)c1C(=O)NC1CCN(C(c2cccc(C(F)F)n2)=O)CC1O c1(N(C)C)nc(C(N2CCC(CNC(C3CCCC(=O)O3)=O)C2)=O)cc(O)n1 C(C)(C)(C(O)CO)NC(C(CC)NC(N)=O)=O.C(=O)C(C)C C(=O)(C(O)Cc1cnc[nH]1)N(CC(CN(CC(C1CCC1)OC)C)O)C c1(C(=O)OC)cc(C(C(=O)NCc2nnn(C)n2)N(CCCN(C)C)C)c(C)o1 CC1CN(C(c2ccc(CF)cc2)=O)C(C)CN1C(=O)C(O)CC1CCCC1 CCCC(C)CC(=O)NCCC1CN(C(c2cccc(C)c2O)=O)CCO1 Cc1cc(Cl)cc(Br)c1NC(C1CCSC(C(C)C)C1)=O O=C(CC1OB(O)c2ccccc21)NC1(C2CCN(C(=O)C(F)OC(F)F)C2)CC1 C(=O)(C(F)(F)C(O)C(C)C)NCC1(C)CCCN(C(C2(CC#C)CCC2)=O)C1 c1(C(=O)NCCCNC(C(C)C(C)C2CCCCC2)=O)cccc2nc(O)oc12 c1(C(N2CC(NC(=O)CCOCc3ncc(C(=O)O)[nH]3)C2)=O)cccc2oncc12 C1(C(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)on2)=O)CN(C)C(=O)N1 Cn1cc2ccc(C(=O)NC3CN(C(C4(Cl)CC4(F)F)=O)CC3C3CC3)cc2n1 Cc1ccc(C)c(C(=O)NC(C2CCCCN2C(C2CC3(C2)CC(C)C3)=O)C)c1 C1(C(N(C)CC2CCCN(C(c3c(OC)noc3C)=O)C2)=O)CCCCN1N=O N1(C(C(C)(C)c2cccnc2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(-c2ccc(C(=O)Nc3c(C#N)cccc3)cc2)nc2ccccc2o1 CC1(C)C(CNC(c2nnn(C(C)(C)C)n2)=O)CCN1C(=O)CCC(N)=O N1(C(Cn2c(CCC)ncc2)=O)CC2CCC(C1)N(C(c1ncc(C)cn1)=O)C2 C(=O)(C1CCCc2nc[nH]c21)NCCC(CNC(Cc1c(C)cccn1)=O)O N1(C(CS(=O)(=O)NC)=O)CC(C)N(C(=O)CCc2cscn2)CC1C c1(C(=O)NC2(C3CN(C(C(C)OCC=C)=O)C3)CC2)cncc2nnn(C)c12 C(C1CCC(=O)O1)=CCN1CCC(C(C)C(=O)N(C)C)C1 CC1COC2(C1)CN(C(=O)CC1(NC(=O)OC(C)(C)C)CCOC1)C2 c1(C(=O)NCC2(O)CCN(C(C3CN(C)C(=O)C3)=O)C2)cc2sc(Cl)cc2[nH]1 C(=O)(C(C)CCCC(C)C)NC1(C(=O)NCCc2cc(CC)no2)CCCC1C CCC(C(=O)NC(C)(C)CCC(=O)NCC1CCCC1OC)C(C)C Cc1nc2cncc(C(N3CCC(CNC(=O)C4=CCSC4)C34CC4)=O)c2[nH]1 N1(C(CC(C)(F)F)=O)Cc2ccccc2C(NC(=O)C(c2ccc(F)cc2)F)C1 C(CN=c1[nH]nc(-c2ccccc2)o1)N(C(CC1N(CC)CCOC1)=O)C C(=O)(C(C)(C)Cc1cccc(Cl)c1)NC(CN(C(c1ccc(=O)oc1)=O)CC)C c1(COC(C2CCCC(C(F)(F)F)C2)=O)nc2cc(Br)c(F)cc2s1 c1(C(=O)NCC(C(C)C)NC(C(=Cc2cnc[nH]2)C)=O)cc(C(F)F)nn1C c1(C(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)cc2sccc2[nH]1 CCCCC(CC(=O)Nc1ccc(OC)cc1F)NC(=O)Cc1ccnc(C)c1 CC(CNC(C1CCCS1)=O)(C1CC1)NC(=O)C(=O)NCC(F)F C(=O)(C(CCC(N)=O)N(C)C)N1CCCCC(NC(CCCOC)=O)C1 c1(C(=O)NC(C)CNC(c2cn(CC(N)=O)nn2)=O)cc2cn[nH]c2cn1 C#CCC(C)(CC)C(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O Cc1cccc(C(=O)NC2C=CC(CNC(=O)Cc3csc(C)n3)C2)c1 N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)C(c2cccc(Cl)c2)O)CC(O)C1 c1(C(=O)OC)ccncc1C(=O)NCC1(NC(C2CC2(C)C(F)F)=O)CCC1 c1(C(=O)NCC(CNC(=O)CCc2ccncn2)F)c(O)cc(F)cc1F C1(CC)(NC(=O)CC2CCC2C)CCN(C(c2ccn(C)c2)=O)CC1 c1(OC)ccc(C)cc1C(N1CCCC(NC(c2ncc(F)cc2F)=O)CC1)=O C=CC1COCC1NC(=O)COC(C1CC2(CC2)C1)=O c1(-n2cc(CNC(C)C)nn2)ccc(CNC(C2CC2F)=O)cc1 N1(C(C(C)(C)O)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(C(=O)NC(C)C(c2c(F)cccc2Cl)O)cc2n(n1)CCCCC2=O N12CCCC(C)(CC1)C(=O)NC(CCC)C2=O.c1(OCCSC)ccncc1 CS(=O)(=O)c1coc(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)CC2F)c1 Cn1ncnc1NC(=O)NCCC1CCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NCCC(C)N(C(=O)CC(F)(F)Cl)C)cccn2cncc12 Cc1cc2c(Br)ccc(C(=O)NC3(CF)CCN(C(=O)C(C)O)C3)c2o1 N1(C(C2N(C(C3CCN(C)C3)=O)CSC2)=O)CCOCC12CC2 N1(C(C2C(C(C)C)CCC2)=O)CCC2(CC1)CC(NC(=O)CC(C)C(F)F)CO2 CC1(C(=O)O)CCN(C(C2(C3CCCCN3Cc3ccccc3)CCOCC2)=O)C1 C1(NC(C(N2CCSCC2)C)=O)CCCN(C(=O)CCC2CCC(=O)NC2)C1 N1(C(CSCc2ccc(C)cc2)=O)CC2(CC(NC(=O)CCC[N+](=O)[O-])CO2)C1 C1(NC(C2CCCCNC2=O)=O)CN(C(=O)C2=CCCSC2)Cc2ccnn2C1 CC1CCC(NC(=O)CCCn2cncn2)CN1C(=O)C=CC(C)(C)C c1(OC)ccc2c(C(=O)NC34CC(CNC(=O)CC(C)CF)(C3)C4)cnn2c1 C(C(O)CC(F)(F)F)C(=O)N(C(=O)C(O)CN1CCCC1)CC1(F)CCCC1 C(C1=CCCOC1)NC(CCN(C(C1(C)CC1)=O)CCO)=O C1(C(N2CCOCC2)=O)(CNC(=O)CCOC2CCCC2)CC2(CC2)C1 CC1CCN(C(c2cnc3n2CCC3)=O)CC1CNC(=O)Cc1cn[nH]c1 Cc1c(C(N2CCC(NC(=O)CSCC(=O)Nc3ccccc3)C2)=O)ncn1C C1(CNC(CC(C2CC2)NC(CCN(C)CCO)=O)=O)CCC2(CC1)CC2 N1(C(c2cc(C)nn2CC(F)F)=O)CC2CC(NC(c3sccc3C)=O)C2C1 Fc1ccc2c(c1)C1CCC1CN2Cc1ccc2nc[nH]c2n1 c12ccccc1NC2=O.n1(CC)ccc(CN2CCC(N(C)C)C2)n1 c1(C(=O)NC(CC=C)CNC(C)=O)ccc(OC)c(S(C)(=O)=O)c1 CC1CCN(c2nnc(C(F)F)n2CC2CCCCO2)CC1F c1(CC(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)C2)cc2cc(Cl)ccc2[nH]1 c1(NC(C2CN(Cc3ccc(OCCO)cc3)CCO2)=O)c(O)cccc1[N+](=O)[O-] c1(C(CN)(F)F)ccc(C(=O)NC2CC(N)C2N)cc1 c1(CC(N2CCCC(CNC(C3CC3F)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CCC(C)(F)F)NC(CNC(CC1N(C(C)=O)CCCC1)=O)(C)CO c1(CN(C)C(C2CC(NC(C)C)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(C(N2CCC(C(CC)CC)C2)=O)CC2CN(C(=O)C(C)(C)OC)CC2C1 N1(C(C(C(C)C)C#N)=O)CCC2(CCC2NC(c2ccc(CN(C)C)o2)=O)CC1 C(=O)(CCCC(F)(F)CO)N1CCCC(C)(NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(CC(C(=O)NC2C(CNC(C=C(COC)C)=O)C2)NC=O)ccc(C)cc1 CC1=C(C(=O)NC2CC3(NC(=O)CCCCc4cnn[nH]4)COC2C3)CCCO1 c1(C(=O)NC2C=CCN(C(CSCC(N)=O)=O)C2)sc2cc(F)ccc2c1Cl N1(C(C(CC)(C)O)=O)CC2CCCC2(NC(=O)C2=CCN(Cc3ccccc3)C2)C1 c1(C(=O)NC2CCCN(C(C3(C)CC=C(C)CC3)=O)CC2)cc2c[nH]cnc-2n1 CCC(C)(C)C(=O)N(CC(C)(C)NC(=O)CCc1ccc(SC)cc1)C N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C(C)CC#N)CC(O)C1 C(C)(C(C)CC)N(c1ccccc1)C(CSCC)=O C1(C(C)NC(=O)CCC2CNC(=O)N2)CCN(C(c2cn(C)cn2)=O)CC1 N1(C(C2CC(C)(C)N(C(c3ccc(C#N)cc3)=O)C2)=O)CCCN(C=O)CC1 c1(CC(N2CCC(N(C(C(CC)O)=O)C)C2)=O)coc2ccc3ccccc3c12 S(=O)(=O)(c1ccc(NCCN(C)C)nc1)NC1CCCC(NC(C)=O)C1 CCC(C)(CO)C(=O)N(C1CCC(n2cc(C(CC)N(C)C)nn2)CC1)C N1(C(CCC#C)=O)CC2(CCCCC2)C1NC(=O)OC(C)(C)C CC1CCCC1C(=O)NCc1c[nH]nc1C1CCN(C(=O)C(=O)NCC(F)F)C1 CC1CN(C(c2ccc(Br)o2)=O)CCC1NC(=O)C=CC(N)=O C(=O)(CC(C)C(=O)OC)N1C(CCC(N2C(C(=O)OC)CCC2C)=O)CCC1 C1(C(N2C(C#C)CC2)=O)CN(C)CCN1C(c1cscc1OC)=O N1(C(C2(C)CCOCC2)=O)CC2CN(C(C3CC4OC(=O)OC4C3)=O)CC2(C)C1 C(=O)(NNC(=O)CN1CCCC1)C12CC(NC(=O)OC(C)(C)C)(C1)C2 C(CC1=CCCCC1)N(C(C1(NC(C(c2ccn(C)c2)C)=O)CCSC1)=O)C N1(C(C#CC(C)C)=O)CCCC12CCN(C(c1ccn3ncccc13)=O)C2 c1(CNC(C2(CC)CCCC2)=O)ccc2c(c1)CN(C(=O)C1=CCOC1)C2 Cn1c(Cl)cnc1NC(=O)NC1(C(=O)O)CCN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC2CCN(C(c3cncc(SC)c3)=O)CC2)CC(C)(C)CN1C Cc1cc(C(=O)NCC2CCN(C(=O)C(C)SC(F)(F)F)C23CC3)cc(C)n1 C1(OC)CN(C(=O)Cc2cscn2)C(C)(CNC(=O)CNS(N)(=O)=O)C1 N1(C(CC=C)=O)CC2C3CCC(C(NC(=O)Cc4cc(C)cc(F)c4)C3)C2C1 C1(C(C(=O)OC)(C)C)CCN(CC(=O)N(CC(C)(O)C(=O)O)C)CC1 CCCC(C)(C)CC(=O)N1CCC2(CC2)CC1C(=O)N(C1CCN(C)C1=O)C Clc1ccc(-c2csc(CSc3cccc(Cl)c3)n2)cc1 N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(C1CCCN1C1CCCC1)=O)C2 c1(CNc2nc(C)nc(N(C)Cc3cc(O)ncn3)c2)ccc(N=S(C)(C)=O)s1 CC1=C(C(=O)NC2(CF)CN(C(c3cc(C)nc(O)c3)=O)C2)CCO1 C1(C(=O)NCCCC(C)NC(C=C(CCC)C)=O)CCC(C(=O)N(C)C)CC1 C1(C(=O)NC2C(C)CCN(C(C3C(C4C(C)C4)C3)=O)C2)CCc2nncn2CC1 C(C(C(C)C(C)C)NC(=O)CN1CCCC1=O)NC(CCc1c(C)cccn1)=O Cc1ccc(O)c(C(=O)NC(CNC(=O)CN2CCC(=O)NC2=O)C2CC2)n1 N1(C(C(CC)N(C)C)=O)CC2CC(C(=O)NCC3(SC)CCCC3)C(C2)C1 N1(C(CC(CC)(F)F)=O)CC2(C1)CN(C(c1cc3c(=O)[nH]ccn3c1)=O)CCO2 N1(C(C2CN(CC)C(=O)CC2)=O)CC2CCCN(C(c3cc(CO)[nH]n3)=O)C2C1 c1(C2(N(C)C(=O)NCC3(c4cc[nH]n4)CC3)CC2)ccc(F)c(F)c1Cl C1(NC(CCOc2cccc(C)c2)=O)CN(c2nnc(C)s2)CC(C)(C)C1 C1(C(N2C(CCCC)C=CC2)=O)CCN(c2nc[nH]n2)CC1 C(=O)(C(C)(CC)CC)NCC(CC(=O)N(C(CC#C)C)C)O CC1C(C(=O)N2CC(NC(c3ccc(O)nc3Cl)=O)CC2(C)C)=NOC1C C1(CNC(CP(C)(C)=O)=O)CCC2(CO1)CC(NC(C1CC(O)C1)=O)C2 c1(C(N(CCCOC)CCNC(=O)CSC2CCCO2)=O)ccccc1C C(C(O)C(=O)Nc1ncccn1)NC(=O)C1CC1.C12CCCC1N2 C1(C)(C(=O)NC2(CNC(C3C(C)CCCC3)=O)CC2)CCC2(CC1)OCCO2 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CN(C(=O)C=C3CCN(C)CC3)CC2(C)C1 N(C(=NCCc1ccccn1)NCc1ccc(CO)cc1F)C(COC)C1CC1 N1(C(c2cc(Cl)ccc2OC)C(=O)NC(CC)C)CCCN2CCCC2C1 N1(CC(C)SC)CCC(=O)N(Cc2cccc(Cl)c2)C1=O C(=O)(CC(CC)CC(C)C)N(C(C(=O)N1CC(CC)C1)CC(F)(F)F)C C(c1ccc(S(=O)(=O)NCc2ccccn2)cc1)=CC(=O)N(C1(CO)CCC1)C n1(CC)cc(C(=O)NC2CCC2CNC(=O)Cc2cc(C)nn2C)c(C2CC2)n1 c1(C(C(=O)NCCCSC)N(C2CC3CC3C2)C)ccc(C)cc1Cl.C1C(=O)N1 C(=O)(C(C)CC(C)CC)NCc1c(CNC(C(F)=CC)=O)cccc1 CCC(CC)(CO)C(=O)NC1CCN(C(c2cccc(C3CCC3)c2)=O)CC1F N1(C(C2(CCOC)CC2)=O)CCC(CCN(C)C(c2n[nH]c(C)c2F)=O)CC1 c1(C(N2CCN(C(c3c[nH]c(=NC)s3)=O)CC2)=O)cc(C(C)C)ccc1F c1(C(COC)NC(=O)C(c2sc(Br)nc2Cl)N2CC(O)CC2C)cccc(F)c1 N(C1CN(C(=O)CCC(F)F)CCc2ccccc21)C(C1(COC)CCCC1)=O N1(C(C2(CSC)CC2)=O)CCCC1CCCNC(=O)COc1cc(C)on1 N1(C(c2c(CC)nco2)=O)CC2CC(C1)N2C(C1COCC(C)O1)=O Cc1cc(=O)ccn1CC(=O)NC1CC2CC(NC(=O)Cn3ccnn3)C1C2 c1(C(=O)NC(c2cccc(OC)c2)C(=O)OC(C)C)c(Br)nc2n1CCOC2 N1(C(c2nc(OC)sc2)=O)CCCC(CC2CN(C(c3ccncc3Cl)=O)C2)C1 c1(C(=O)NC2CCCC(NC(Cc3cc(OC)no3)=O)C2)sc(F)cc1Cl C(=O)(CCN=[N+]=[N-])NCC(C(=O)N1CC(CC)C1)O Cc1ccc2nc(C(=O)NC3CCCC34CCN(C(=O)CC3CC3)C4)cn2c1 CC(CCC(C)(C)C)C(=O)N(C)CC1(NC(=O)C2=CSCS2)CC1 Cc1cnn2c(NCC(=O)Nc3ccc(O)cc3)cc(Cl)nc12 c1(C(N(C2CCN(C(c3c(C)cc(C)nc3)=O)C2)C)=O)ccc2c(c1)COC2=O CCC1=C(C(=O)N2CCC(NC(c3cnc(S)[nH]3)=O)C2(C)C)CCCO1 N1(C(CC2CC(=O)C2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C1C2 n1(CCC)cncc1CNC(C1(CNC(=O)C=Cc2cncs2)CC1)=O C1(NC(c2cnc(NC(C)=O)o2)=O)CN(C(C2CSC2)=O)CC1F N1(C(C(CC)C)=O)CC2(CCC(NC(=O)OC(C)(C)C)C2)C1 c1(C(N2CC(N(C)C(C3CCC(=C4CCC4)CC3)=O)C2)=O)ccc(N)c(CO)c1 N1(C(C(C(C)C)NC(C(CC)=CC)=O)=O)CC2(CC(N(C)C)C2)C1 N1(C(C2(CC)CCN(C(=O)Cc3csnn3)C2)=O)CC(C)CCCC1C C(=O)(C(CC(F)F)N(C(=O)CC(C)SC)C)NCC(CO)OC N1(CCNC(=O)Cc2cnc[nH]2)CCN(C(=O)C=C2CCC2)CC1 CC(CCNC(=O)C(c1ccccc1Br)(F)F)CCNC(=O)C=CC1CC1 C1(C(=O)NCC2CCN(C(CCc3cn(C)nc3)=O)C2)CCOC(=O)CC1 C1(NC(=O)CC2CC(F)(F)C2)CCN(C(C2CCCC(F)(F)C2)=O)C12CCC2 c1(C(N2CC(O)(CNC(=O)COCc3nc[nH]n3)C2)=O)cc(C(F)F)ccc1F C(=O)(C1CCCn2ncnc21)N1CC(CC(C)NC(C2CN(C(C)C)C2)=O)C1 C(CCS(=O)(=O)Nc1cccnc1OC(F)F)N(C)C1CC1 CCC1=NOC(CC(=O)NC2(CO)CCN(C(C3(OC)CC(C)(C)C3)=O)C2)C1 C1(CC(=O)NCCCNC(=O)CC2C=CCC2)Cc2cc(C(F)(F)F)ccc2O1 C1(CC#C)(C(=O)N(CCCNC(=O)CC2CC2(Cl)Cl)C2CC2)CCOC1 c1(CC(C)NC(c2nnc(CCCC)s2)=O)ccccc1C c1(C(=O)NC(CC2CCC2)C(=O)NCCCO)ccc(C(F)F)cc1 C12(CNC(C3N(CCC(C)C)CCC3)=O)CCC(C1)N(C(c1cccnc1)=O)C2 C(Cc1cnc[nH]1)(C(=O)NCCC(C)NC(=O)CCC1CC1)NC(C)=O CC1CC(NC(c2ncoc2-c2ccon2)=O)CN1C(=O)C=Cc1ccnn1C c1(C(=O)NCCN(C(c2csc(CO)n2)=O)C2CC2)ccc2ccnc(O)c2n1 c1(C(N2CC(Cn3cc(C4CC=CCC4)nn3)C2)=O)ccc(O)cc1 N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CN(CC(C)C)C2)=O)C(O)C1 N1(C(C(C)OCCC=C)=O)CCC(CCC(=O)N(CCC(=O)NC)COC)C1 CC(C)C(C)(CNC(C1OCCC1C)=O)NC(c1cn(C(F)(F)CO)nn1)=O c1(C(N2C(CNC(CC(=O)NCC)=O)CC3(CC3)C2)=O)cc(C)c2c(c1)CCC2 c1(C(N2C(C(=O)NCCCNC(=O)NC)C=CCC2)=O)ccc(C)nc1C c1(C(N2CC(N(C(CCCCSC)=O)C)C(F)C2)=O)cc(C)nc(O)n1 c1(C2(C)OCCO2)ccc(CNC(=O)NCCC2CCCCCC2)cc1 C1(OC)CC2CC(c3nnnn3CCCF)(NCC3CC4(CC4)C(=O)O3)C2C1 N1(C(c2n(C)ccn2)=O)CCc2nc(CNC(C3CC3C3CC3)=O)sc2C1 C(=O)(C1=CCCN(C(=O)CC2(CSC)CC2)C1)N(C(C=C)C1CC1)C c1(NC(C(c2cccnc2)NC(c2ccc(COC)s2)=O)=O)cc(C)ccc1C c1(C(=O)NC(C2CCN(C(c3cccc(OCCF)c3)=O)C2)C)cnnc(O)c1 N1(C(C2CC(NCc3c(C)cccc3)C2)=O)CCCC2CCCCC12 N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1cncnc1)=O)CCO2 c1(C(=O)NC2(CN(C)C(c3ccc(Br)nc3F)=O)CC2)c[nH]c2cccc(C#N)c12 C(=O)(C(COC)CC(C)C)N1CC(C(=O)NCC(F)C2CCC2)(COC)C1 CC1CN(C(c2ccco2)=O)CCC1CNC(=O)CCc1ccc(Cl)cc1 c1(C(N(CC(CC)NC(C2(CC#C)CCCO2)=O)C)=O)ccccc1C(C)=O C1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCC(=C)C)CC2CCC1CC2 CC1CCC(=CC(=O)NCCCC(C)NC(C2(c3ccno3)CC2)=O)CC1 C1(C=O)CC(C)=NO1.C1(=O)CCN1CC1CC1.C(C(C)N)SCC c1(NC(C2C=CC(NC(C3CC(O)CN3)=O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)(C)F)=O)CCC(F)(F)C(CNC(C2(CC3CCCC3)CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCCCC2)C1 C1(C(=O)NCCC2(CNC(c3cc(C(C)=O)on3)=O)CC2)CC=C(C(C)C)CC1 c1c(C)cnn1C.c1(CCN(C(=O)NCCOCCOCC)C)ccc(C)[nH]1 N(C1C(=O)Nc2c(Cl)cccc21)C(C1COCCN(C(C2(COC)CC2)=O)C1)=O N1(C(CNC(=O)NC)=O)CCN(C(=O)C=Cc2nc(C)co2)CC1C1CCC1 c1(C(C)C)ncc(C(=O)NCC2CCCC2NC(=O)Cc2ccoc2)cn1 c1(C(N2CC3CC2CN3Cc2c(O)cccc2F)=O)ccc(Cl)cc1Cl c1(SCC(N2CCCC(NC(C(C(=O)OC)C)=O)C2)=O)ccc(C)c(C)c1 C1(S(N)(=O)=O)(C(=O)NCC(CNC(Cc2c(OC)ccc(F)c2)=O)F)CCCC1 N1(C(CC)=O)CCC(O)(CNC(=O)Cc2cc(OC)no2)C1 N1(C(CNC(CCC)=O)=O)CCCC1CCNC(=O)C(C)(C)c1cncs1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC2(NC(=O)Cc3cc(C)on3)CCCC12 C1(N(C(Cn2ncc(C)c2)=O)C)CC2CC1N(C(C1CCC(=O)C1)=O)C2 CC(C)C(O)C(=O)N(C1CC(OCC)C1)CC1(Cc2ccccc2)CCCC1 c1(OC)cc(OC(F)(F)F)ccc1NC(c1nccn1C(C)C)=O C1(NC(CC2ON=C(C)C2)=O)CCC(F)(CNC(=O)Cn2ccc(C)c2)C1 c1(C(=O)Nc2c(CC)ccc(F)c2)cc([N+](=O)[O-])ccc1OC C=CC(C)(C)CC(=O)NCC(C(F)(F)F)N1CCN(C(=O)CC2CSC2)CC1 N1(C(c2n(CCC)ncc2)=O)CC(NC(c2coc(OCC)n2)=O)CC1C C(=O)(CS(=O)(=O)C(C)(C)C)N1CCN(C2CCC3C(C)(C)C2C3)CC1 C12(C(=O)NCC3(CCOC)CC3)CC(C)(CN1C(=O)Cc1ccns1)C2 c1(NCCc2cnc(C)o2)nccc(=NC(C)CS(C)=O)[nH]1 C1(COC)(NC(C2CC2(C)C(C)C)=O)CN(C(C2(C(=O)N(C)C)CC2)=O)C1 C(C1=CCN(C(C2CCC=CO2)=O)CC1)NC(CC1(OC)CCC1)=O c1(CC)ccc(C)cc1C(=O)NCCC(C)NC(C1(C)CCNC1=O)=O c1(C(N2CC(N(C(=O)CC3CCC4CC34)C)C2)=O)cc2c(s1)CCC2 c1(NCC2CN(C(CC(C)N(C)C)=O)C2)ncnc2cnccc12 NC(=O)CC(O)C(=O)N1CCCC(O)(CNC(=O)CNC(C2CCOCC2)=O)C1 C1(c2ccccc2)(NC(C(C=C)OC)=O)CS(=O)(=O)C1 N1(C(C(CCC)CC)=O)CCC(C2CC(NC(=O)Cc3scnc3C)C2)CC1 C12(C(=O)NC3CCC(NC(C(CCC)c4ccccc4)=O)C3)CCN(CC1)CC2 CC(CS(C)=O)C(=O)NC12CC(CNC(c3ncccc3C3CC3)=O)(C1)OC2C c1(CC)ccc(CCCNC(C)(CCI)c2nnnn2C2COC2)cc1 NC1CCCn2ncnc21.c1(-c2n(C)nnn2)ccccc1 C1(CNC(CNC(CCC)=O)=O)CCCN(C(=O)C(C)(CC2CCC2)OC)CC1 N1(C(CN(CCOC)C)=O)CC(CNC(=O)CN2CCOCC2)CC1C C1(CC)C(C(=O)NC2CCC2(C)C)CCN1C(=O)CN(C)C(=O)OC c1(C(N2CCC(NC(c3ccc(CC)cn3)=O)C(F)C2)=O)ccn2c1CCCC2 n1(CCCC)ccc(C(=O)NCC2CC(NC(=O)Cc3cnn(C)c3)C2)n1 CCC(CC(=O)NCC(C)(C)CN(C)C(C1(F)CCCCC1)=O)SC C(=O)(C1=CCOCC1)NC1C(CNC(CC2N(C(C)=O)CCC2)=O)C1 C(C)(C)(C(=O)N(CCNC(c1cn(CC2CCCOC2)nn1)=O)C1CC1)N(C)C Cc1ccc(Br)cc1C(=O)NCCCCCCN(C(=O)C(C)C1CCCO1)C N1(C(C2CCCNC2=O)C(=O)NC)CCC(C)=C(Br)C1 N1(C(CNC(CNC(C(C)N(C(C)=O)C)=O)=O)=O)CCCC2CNC(=O)C12 c1(C(=O)NCCCN(C)C(c2coc(Br)c2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C1=CCCSC1)NC1C(CCC)CN(C(c2c(SC)cnn2C)=O)C1 c1(CO)ccc(CNCCN(c2ccccc2Cl)C2CCCCC2)c(Cl)c1 c1(C(=O)NCC(CNC(=O)Cc2cnn(C3CC3)c2)OC)cc(F)c(N)cc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1CC(C)(C)N(C(=O)CC=C(Cl)Cl)CC1 C1(CNC(C(C(CC)C)=O)=O)CCC2CN(C(=O)C=Cc3cnn(C)c3)CC12 C1(O)(CNC(C2CC(C)N2C(=O)OC(C)(C)C)=O)COC2CC1C2 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C1(NC(COCCNCc2ccnc(O)c2)=O)CC(F)CN1C(=O)OC(C)(C)C c1(CS(=O)(=O)N(C(C#C)C2CCC2)C)ccc2ccccc2c1 C1(CC2CN(C(Cn3cc(CC(C)(C)C)nn3)=O)C2)CCCCC1 CN1C(=O)CCC1C(=O)N(C1CCCCC1)CCNC(=O)CC1(CO)CC1 c1(-c2n(-c3ccc(OC)cc3)nc(CO)n2)cc(F)ccc1O N1(C(c2cccc(Br)c2)C(=O)NC(C(=O)OC)C)CC(CN(C)C)CC(C)C1 c1(N2CC(C(C)NC(=O)CCc3cnn(C)n3)C2)ccnc(-c2nccs2)n1 n1(CCC)nc(C(=O)N(C2CCNCC2)CC)ccc1=O C1(NC(CC2(COC)CC2)=O)CN(C(=O)C(C)(C)CC2CC2)CC1C(F)(F)F C1(C)(CNC(c2cnn(CC)c2C2CC2)=O)CCN(C(=O)C2=CCOC2)CC1 Cc1cnc(NCC2CCCC2NC(=O)CSc2nc[nH]n2)nc1 Cc1cc(NC(c2nncs2)=O)ccc1NC(=O)C(C)n1cncn1 c1(CCN(C(=O)NC2C(C(C)NC(C)(C)C)C2)C(C)C)ccccc1 C1(NC(CS(CC)=O)=O)CC12CCN(C(=O)C=Cc1cccc(CO)c1)CC2 N1(C(CCc2cccc(C)c2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC12CC2 CCC(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CC1 CCCCCCCN(C)C(C1C(C)CCN1C(c1ncn(C)n1)=O)=O c1(N(C)C)ncc2c(n1)CCC(NC(=O)C(=O)NCc1c(F)cc(F)cc1F)C2 C1(C(=O)NC2C(NC(C3CCCN(C(=O)OC)C3)=O)CCC2)CC2C=CC1CC2 c1(CC)oc(C(=O)N(C)CCC2CCN(C(=O)C=CC=C(C)C)CC2)cc1C N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2ccc(I)c(O)c2)=O)CC(F)(F)C1 C1(NC(C2N(CCC(C)C)CCC2)=O)CC2CC1N(C(=O)COCC(C)(C)C)C2 c1(C(=O)NCC2(COC)CN(C(C3CC(O)CN3C)=O)C2)ccc(OC)c(C)c1 c1(OC(F)F)cc(C)ccc1C(N1CCCC(N(C)C(C2(OC)CC2)=O)CC1)=O CC1CN(C(c2cnc(CC3CC3)s2)=O)CCC1Nc1cc(C(N)=O)ncn1 C12(C(N3CCN(C(CCc4cc(C(C)=O)c(C)o4)=O)CC3)=O)CCN(CC1)CC2 C=C(C)C1CCC(C)(O)C(NC(=O)C(=O)NCC23CCCCC2NCC3)C1 c1(C(C)C(=O)NC2(C)CN(C(c3cnc(O)c(Cl)c3)=O)C2)ccc(C#N)cc1F CCCC(CC)C(=O)N1CCOCC1CN(C)C(c1cnncc1C)=O C1(NC(CCSCCC)=O)CC(CC(=O)NCc2ccc(SC)o2)C1(C)C N1(C(C(CC)=CC)=O)CCC(C)N(c2ccncn2)CC1 c1(C(N2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)=O)n[nH]c(C2CC2)c1Br Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(CC(=O)NC2CCC(CNC(C3(C(C)=O)CC3)=O)C2)ccc(C)nc1Cl Cc1ccc(C(N2CCN(C)C(CNC(C3(CC(C)C)COC3)=O)C2)=O)c(O)n1 CCC(C)C(C)CNC(=O)CC(C)(C)N(C)C(C1(CC)CCCCO1)=O c1(C2N(Cc3cccc(C(C)N)c3)CCC2)ccc(F)cc1Br C1(CNC(COCCC#C)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)N(C(CC(=O)NCCCC#C)(C)C)C c1(C(=O)Nc2cnncc2Br)cc(C(=O)NC2C=CCC2)cc(C)n1.CCSC Cc1coc(C(=O)NC2(CNC(=O)Cc3cccc(C(C)C)c3)CC2)c1C C(C1c2ccsc2CCN1C(=O)CC1CC1)NC(=O)CCOCC1CCOCC1 Cc1c[nH]c2ncc(C(=O)NCC3CCCCN3C(C3CC(C)(F)C3)=O)cc12 C(c1ccc2ccccc2n1)=CC(=O)NC12C(CN(C(c3c(OC)ccs3)=O)C1)C2 c1(CC)ccc(Br)cc1C(=O)NCC1(F)CCCN(C(c2nc[nH]n2)=O)C1 N1(C(CN(C)CC)=O)CCCCC1CC(C)(C)C.c12cc(on1)C(=O)N(CC)C2=O C(=O)(C1=NNC(=O)C1)NC1(C)CCN(C(C2CCCN(CC)C2)=O)C1 N(C1c2ccccc2CC1NC(=O)CCS(C)(=O)=O)C(Cn1nc(C)c(Cl)c1)=O c1(NC(C(C)NC(CNC(C2CCCC2)C)=O)=O)ccccc1C1CC1 Cc1cc(=O)n(C)cc1C(=O)NCc1nc(C(=O)NC2(C)CCCC2C)co1 Cc1ccc2[nH]c(C(N3CCC(C)C3CNC(=O)CC3C=CCC3)=O)cc2c1C c1(C(=O)NC2CC(NC(CC(C)C3CCCO3)=O)C2)csc2c1CCCC2 Nc1ccc(C(N2CC(CO)(NC(C34CC=CC(C3)OC4)=O)C2)=O)cc1Cl N1(C(C2CC(=C)C2)=O)CCCC2(CC(NC(=O)C(C)(C)OC)CO2)C1 C1(NC(Cc2ccc(CCC)cc2)=O)CC2CC(C1)N(C(C1(C)CC1(F)Cl)=O)C2 C1(C#N)(C(N2CCCN(C(C(=O)NC(C)C)=O)C(CO)C2)=O)CC2CCC1CC2 c1(C(=O)NCCC2CC(NC(CCOCCN(C)C)=O)C2)[nH]nc2ncccc12 c1(-c2n(C(C)C)ncc2)nc2c(s1)CC(C(=O)NCc1ccnc(F)c1)CC2 CC(c1cccs1)=CC(=O)NCC1CN(C(=O)CN2CCCNC2=O)CC1O Cc1cccnc1S(=O)(=O)C(N1CC(O)C(O)CC1(C)C)=O Cc1nc(C)n(CCC(=O)NC2CCN(C(=O)CSCCC(C)C)C2C2CC2)n1 c1(-c2scc(CCNC(C(n3cc(CCC(C)O)nn3)C)=O)n2)ccc(F)cc1 c1(C(N(C)CCC2CCN(C(C3CC3Cl)=O)CC2)=O)ccnc2ccccc12 CCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)NC(c1ccn(C)c1)=O c1(C(=O)NC2C(CNC(c3cc(C(C)=O)sc3)=O)C2)cc(C)nc(O)c1[N+](=O)[O-] N#Cc1ccc(C(N2CC3CCN(C(C4CC(C(F)F)C4)=O)C3C2)=O)cc1F C1(C(N(CC(CC)NC(=O)C(F)(F)CO)CC)=O)CC2CCCN2C(=O)N1 N1(C(=O)NC2CC(n3ccnc3)C2)CCCC(O)(Cn2cc(CO)nn2)CC1 Cc1ncnc(C)c1CC(N1CCC(NC(C2CC2(C)C(C)C)=O)CC1)=O N1(C(C(c2cn(CC)nc2)(F)F)=O)CCOC(CNC(=O)C(C)(C)CC2CC2)C1 C1(CC(N2CC(COC)(CNC(=O)C(C)CSC)C2)=O)CCC(F)(F)C1 N1(C(c2cc(C)sn2)=O)CCC2(CCC2NC(C2CNC(=O)CC2(C)C)=O)CC1 N1(C(C(C)CN(C)C)=O)CCN(C(=O)C=CC2(C)CCOCC2)CC1CO N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)C=Cc2cncnc2O)C(CO)C1 CC1CC(NC(=O)CCCCCF)CN(C(c2cccc(C(F)F)c2F)=O)C1 N#Cc1cccc(CC(N2CCC(CO)(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c1 C1(OC)(OC)CC(C)(C(=O)Nc2ccnc(-n3cc(N)cn3)c2)C1 Cn1ccc(C(=O)NC2CCOCC2NC(C2C3(CC3)C23CC3)=O)c1C1CCC1 C12CCCC(C1)CNC2=O.c1(NC(=O)NC(=O)C(Cl)(Cl)Cl)cncc(C)c1 c1(CC(=O)N(CCNC(=O)CC2CC=CC2)CC)ccc(O)cc1Cl c1(N2C3CN(C(c4cnc(CCC)s4)=O)CC2CC3)nc(O)c2c[nH]nc2n1 C(CCN=C1NCCO1)NS(=O)(=O)Cc1ccccc1 Cc1nc(Cl)ccc1C(=O)NC1(C)CCN(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CC2CC1(C(=O)NCc1scnc1C)C2 C1(NC(C2CCS(=O)(=O)N2)=O)CCC2(CCN(C(c3cc(=O)cc[nH]3)=O)CC2)C1 Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)c(N)c(F)c1 c1(N(CC(=O)NC(C)C)C)nc(=NCCC2CCCC23CC3)[nH]c2c1CCCC2 Cc1cnc2n1C(C(=O)NCC1CN(C(=O)CNS(=O)(=O)C3CC3)C1)CCC2 C1(C(=O)NCC(CN(C)C(C2(C(C)(F)F)CC2)=O)O)CCOC1(C)C c1(CC(=O)NC(CN(C(C2(CCF)CC2)=O)CC)C)cc(C)on1 c1(N2CC(CN(c3ccccc3)C(=O)C=CI)C2)nccnc1F c1(NC(C2C(C)C2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OCC(CN2CCC(C)(C(=O)Nc3cc(C)ncn3)C2)O)cccc(C)c1C N1(C(c2scc(C)c2)=O)CCN(C(=O)CCOc2ccccc2F)CC1C N1(C(c2cccc(C(C)C)c2)=O)CC(C)(CNC(=O)C2=CCCS2)CC1(C)C C12(C(N(CCN(C)C)CC)=O)CCN(C(c3cccc(CC#N)c3)=O)CCC1C2 N1(C(C2C(CC)CCO2)=O)CC(C)(C)CC1CC(=O)N(C)Cc1cnn(C)c1 C(=O)(CCCCC(=O)NC(C)(C)C(C)NC(c1csc(O)n1)=O)NC CCC(O)C(C)(C)C(=O)NCC(CC(=O)NC1(CO)CC(OC)C1)C1CCC1 Cc1cc(N2CCC(CC(C)(C)C)C2)nc(NCCCSC(F)(F)F)n1 c1(C(N(C)CC2N(c3cc(OC)nc(C)n3)CCC2)=O)cc2cccnc2[nH]1 C1(C(=O)NCC(C)NC(C2(C(=O)NC)CCC2)=O)CCC(C)(C)CO1 N1(C(CC(C)(C)O)=O)CCC2(CCCCC2NC(c2cc(O)nc(Cl)c2)=O)C1 C=Cc1ccccc1-c1cnc(CNc2cc(C#N)ncn2)nc1 CCC(C)C(C(=O)Nn1nnc2c1CCCC2)NC(=O)C=CC(C)(C)C N1(C(CCC(=O)NC)=O)CC2(COC(CNC(=O)CC34CCC(CC3)CC4)C2)C1 CC(C(=O)N1CCC(CNC(c2ccc(C3CCC(=O)N3)cc2)=O)C1)C(F)F C(=O)(C(C)(C)CCOC)NC1C2(CC(NC(C(C=C)(F)F)=O)C2)C1 c1(NC2(c3n(C4(C)CC4)nnn3)CCCSCC2)ccc(F)c(S(N)(=O)=O)c1 Cc1csc(-c2cn(CC3CCN3C(=O)C(O)Cc3ccccn3)nn2)n1 c1(OC)cc(C(=O)NCC(CC(C)O)c2ccccc2)cc(SC)c1OC N1(C(C2(CC#C)CCOC2)=O)CC2(CCC(Nc3cc(CC)ncn3)CC2)C1 O=C(CCCCCCCCCO)NC1CC2C1CCN2C(C1C2CNC(=O)C12)=O C1(CNC(CCC=C)=O)CN(C(c2noc(-c3ccccc3)c2C)=O)CCO1 C(=O)(CCS(=O)(=O)CC(C)C)NCC(CCNC(C1CC=C(C)CC1)=O)O CCC(CC(=O)N1CCC(CNC(c2cnsn2)=O)(COC)C1)CC(F)(F)F CC1(NC(c2ccc(O)c(Cl)n2)=O)CCC(NC(=O)CC2CCOCC2)CC1 C1(CNC(c2nc(COCC)sc2)=O)C(C)CCN1C(c1cnc(NC)cn1)=O CCC(CN(C)C)CC(=O)N1CCCC(NC(=O)C=Cc2cccnc2)C1C C1(C)(C(N2C3(CNC(C4=C(C)OCC4)=O)CC(C2)C3)=O)CCC(C)C1(C)C c1(C(=O)NC2CC(C)(NC(CC=C)=O)C2)cc(Cl)cnn1 CCN=C(NC1CC1(c1ccccc1)C)N1CCC(F)(C#N)CC1 S(=O)(=O)(c1c(Cl)cccc1Cl)N(C1CCNCC(OC)CC1)C1C(C=C)CNC1 N1(C(COCC(=C)C)=O)CCCN(C(=O)CSc2ccc(F)c(F)c2)CC1C C1(NC(CCC#CC)=O)COCCN(C(=O)CCCSC(C)(C)C)C1 C1(CNC(C(C(C)C)C2CCCC2)=O)CC2OC1C1CC21 N1(C(C(F)=CCC)=O)CCC(O)(C(C)NC(=O)Cc2ccc(C)nc2)C1 C1(C)(CNC(CS(CC)=O)=O)CC(F)(F)CN1C(C1CC2(CC(=O)N2)C1)=O c1(C(N2CCC(N(C(=O)CCC3CC3)CC)CC2)=O)ccc(N(C)C)cc1F N1(C(c2ccc(CC)o2)=O)CC2(CC2)CC1CNC(C12CC(CO)(C1)OC2C)=O N1(Cc2ccc(-c3ccc(C(=O)NC(C)(C)C)cc3)cn2)CCn2cncc2C1 Cc1ccc(Cl)c(N(C(COC(C)=O)=O)CC2CCCN(Cc3nn[nH]n3)C2)c1.CCO c1(N2CC(NC(C(=O)OCC)=O)C(F)(F)C2)ccn2ncc(I)c2n1 C=CCC(C(=O)NC(CO)C(C)NC(C1(C)C=CCC1)=O)C(C)C N1(C(C2(COC)CCOC2)=O)CCN(C(=O)CCCC(F)F)C(CCO)C1 C=Cn1nncc1C(N1CC(O)(CNC(=O)CC2CC2C)C1)=O Cn1ccc(C=CC(N2CCC(CCC(=O)NCC[Si](C)(C)C)C2)=O)c1 N1(C(COCCOCC)=O)CCCN(C(c2ccccc2-n2cncn2)=O)CC1 C(=O)(CN=c1[nH]c2c(c(=NC3CCCCC3C(=O)OC)[nH]1)CSC2)NCC N#Cc1ncn(CC(N2CC(F)(C(=O)NCCc3cn[nH]c3)C2)=O)n1 N1(C(CC(C)N2CCCC2=O)=O)CCC(NC(=O)CSCc2ncc[nH]2)CC1 Cc1cc(C(=O)NC2CC2NC(=O)CSCc2ccncc2)nn1C(F)F C1(N(C(c2c(C3CC3)cnn2C)C(=O)NC2CCC2)C)CNC(=O)C12CC2 Cc1nnc2n1CCN(C(C1COCCN(C(c3ccc(N)c(F)n3)=O)C1)=O)C2 c1(C(N2CC(=C(CNC(COCCC=C)=O)F)C2)=O)cc(F)ccc1Br c1(C(N2CC(CCc3cn(CC(CC)CC)nn3)C2)=O)cc(C)ccc1F CC(C)C(C)CC(=O)NC(C1CC(NC(C2CCC(C(N)=O)C2)=O)C1)C N1(C(CC2CC(CC)C2)=O)CCCOC(CCNC(=O)CCn2cncn2)C1 c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccc(Br)o1 C1(CC(=O)OCC)CCCCN1C(c1cnn(CC)c1)C(=O)NCC1CCC1 C1(CNC(c2cc(CC)nn2C)=O)C(C)CCCN1C(c1csc(COC)c1)=O Cc1nc(-c2ccccc2)ncc1C(N1CCCN(C(C2C(C)C2C)=O)CC1)=O c1(CC(=O)NC2CC(NC(c3c(CC)c[nH]n3)=O)C2)coc2c(F)c(F)ccc12 c1(C(=O)NC2CC(N(C(CNC(C(CC)C)=O)=O)C)C2)ccc(C)nc1N C(C)(C)(CCCC(=O)N(C1CCCC1C)C)NC(c1nc(C)sc1)=O C(=O)(C(C)CC(F)(F)F)NC(C1N(C(c2cc(C)n(C(C)(C)C)n2)=O)CCC1)C N1(C(C(C)(C)OCC)=O)CCCCC(CNC(C2(c3ccc(Cl)cc3)CC2)=O)C1 C1(C(N(C2CCN(C(=O)C(O)CC)C2)C(C)(C)C)=O)N(CC#C)CC1(C)C C(=O)(C1=C(C#N)CCC1)N1CCN(C(Cn2c(=O)sc(C)c2C)=O)CC1C(F)F CC(=O)CCCCCCC(=O)N1CCC2(CCOC2=O)C1 C1(C(=O)NC(c2nccn2C)CC)CCCCC1CNC(=O)CCC=CC(C)C N1(C(C=CC=CCC)=O)CC(F)CC1C(=O)Nc1cnn(C(F)(F)F)c1 C1(C(N2CC(OCC)C2)=O)CN(C(=O)CN2CCC(C)CC2)CC1C N1(C(C2CN(C(C(CC)NC(N)=O)=O)CC2C)=O)CC2CC1CN2C C1(NC(c2cnc[nH]2)=O)CC2(C1)CN(C(=O)CC1CC=CCC1)C2 C1(C(=O)NCC2CC(NC(=O)CC34CCCC3C4)C2)CCCN2CCCC12 N1(C(C(C)OCC(F)(F)F)=O)CCCCC(CNC(=O)Cc2cncs2)C1 C1(C(=O)NC2CC(NC(C3CC(OC(F)(F)F)C3)=O)C2)(OC(C)C)CCOC1 c1(C(N2C3CC(CC(C)O)CC2CC3)=O)cc2ccncc2c(O)n1 C1(COC)(NC(=O)CCCc2nc(C3CC3)no2)CC1(F)F c12ccc(cc1)SCCN(CC)C2=O.CCCC(CO)NC(C1(CC)COC1)=O C1(C(=O)NCCCCN(C)C)CCOCC1NC(c1nccnc1N)=O C1(C(=O)NCc2cc(OC)ncc2)CN(C)CCN1C(c1ccco1)=O N1(C(=O)C(c2ccccc2Cl)O)CC=C(CCNC(C2(n3nccn3)CC2)=O)CC1 CC(CF)CC(=O)NC(C)CC1CN(C(=O)C(F)(F)C2(O)CCC2)C1 C1(C(=O)NC2(CO)CCN(C(c3cccc(CSC)c3)=O)C2)CCC2(CCC2)C1 C(CNC(c1cccc(OC(F)F)n1)=O)(C(C)(C)C)NC(C(COC)O)=O n1(CCC(=O)NCC2CCC(CC)CC2)cnc2ccccc12 c1(OC)cc(C(=O)OC)cc(C)c1.N12CCC(CC1)C(=O)N1CC(C)(C1)C2=O C1(NC(C2CCC(SCC)CC2)=O)CCN(C(C2CC3CCC(C2)O3)=O)CC1O C(=O)(C#CC1CCC2(CC1)OCCO2)N(CCN(C(C(C(CC)C)OC)=O)C)C Cc1c(C(=O)NC2COCC2NC(c2cn(C)nc2Br)=O)nnn1C C1(C(=O)NCC(C)(CO)NC(c2c(C)cc(CC)o2)=O)CC2(C1)CS(=O)(=O)C2 N(C1CCc2cc(CNC(C3CC(O)C3)=O)ccc21)C(c1ccc(CC)cn1)=O Nc1ccc(F)c(F)c1C(N1CCC2(CC(NC(C3CCCN3N=O)=O)C2)C1)=O C(CC(C)(C)CC(=O)NCCOCCCNC(c1ccc(C)s1)=O)OC CCC(CC(C)C)C(=O)N1CCC(C(=O)NCC(n2ccnn2)C)(CC)C1 C1(CN(C)C)COCCN1C(=O)CCN(CCCO)C(=O)CC1CCSC1 CCCCCC(O)C(=O)NC1CN(C(c2nn(-c3ccc(C)cc3)cc2O)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CC2CN(C(=O)C=CS(C)(=O)=O)CC2C1 n1(CC)nc(C(C)C)cc1C(N1CC(NC(C2(C)CC=CCC2)=O)C(O)C1)=O c1(OC)cc([N+](=O)[O-])ccc1C(N1CCN(C(=O)CNC(=O)C(=O)N(C)C)CC1)=O Cc1nc(C(=O)N(C2C3CN(C(C4CCN(C)C4C)=O)CC23)C)n(C)n1 c1(C(N2CCC(CC)C2C(=O)NCc2nnn(C)n2)=O)cc(O)cc(F)c1 N1(C(c2cccs2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1c1cccc(F)c1 c1(C(N2CCCC(C(C(=O)NCCCOCC#C)C)C2)=O)ccc(C)cc1C c1(C(=O)NC(C2CCCCN2C(c2nnn(C)n2)=O)C)cc2ccccn2c1 Cn1cnc2c(CNC(c3ccc(N4CCC(CO)CC4)nc3)=O)cccc12 c1(C(N(CC(C)(C)CNC(C2CCCN2C2CC2)=O)C)=O)ccc(CO)cc1 C12CC(C)CN(C1)CC(=O)N2C.CCC(C)C(=O)NCC(N1CCCC1)=O c1(C(N2C(CNC(Cc3ccc(C)s3)=O)CCCC2)=O)cc(C)c(N)cc1F C(=O)(C1CCCn2nccc21)NCC1(OC)CN(C(=O)CC(C)(O)C2CC2)C1 CC(C(=O)NCC(C1CC1)N(C)C(C12CC(C)(CCO1)C2)=O)C(F)(F)F C1(C(=O)NC)CC(O)CN1C(c1c[nH]nc1CNC(=O)CC1CCC(=O)C1C)=O c1(OC)cnc(Cl)cc1C(=O)N(CCCNC(C1CC12CC2)=O)C(C)C C1(CC)CC(O)CN1C(=O)C(C)(C)NC(c1cn(C)nn1)=O c1(CCC(=O)NC(CCOC)CNC(c2ocnc2C2CC2)=O)ccccc1Cl N1(C(c2c(C)nc(C)c(C)n2)=O)CCCC2(CCN(C(=O)CCC(C)(C)F)C2)C1 C1(NC(Cc2n(C)ccc2)=O)CC(O)CN(C(c2cnc(O)cc2O)=O)C1 c1(C(=O)NC(COC)CC(=O)NC2(C)CC2(C)C)cc2cccnc2[nH]1 c1(C(N(C)CC2CCN(C(c3c(C)cc(F)cc3)=O)C2)=O)cc(N)cc(O)c1C c1(C(=O)NC(C2CCCN2C(C2CC2C2CC2)=O)C)cccc(-c2nc[nH]n2)c1 c1(OC)c(C(=O)N(C2CN(C(C34CCN(CC3)CC4)=O)CC2F)C)occc1=O C1(C(=O)NC(CNC(C(CSC)O)=O)(C)CO)CN2CCN1CC2C C1(CNC(c2ccn(CCCC)n2)=O)CN(C)CCN1C(=O)Cn1ncnn1 N1(C(C2(C)C(C)CN(C(COC(CC)C)=O)C2)=O)CCN(C)C2(CCC2)C1 N1(C(CCN(CCCCC)C)=O)CCN(C(=O)CC2CC(CC)=NO2)CC(O)C1 c1(C(=O)NC23CC(CNC(C4(C)CCCOC4)=O)(C2)C3)cc(O)cc(=O)o1 c1(SCC(=O)NCC(CNC(c2cnn(C(C)C)c2N)=O)OC)ccccc1F C1(CNC(C(C)c2ccsn2)=O)(NC(=O)CC2(C)CCC2)CCCC1 N1(C(C=CC(C)N(C2CCOC2)C(C2CC(N(C)C)C2)=O)=O)CC(C)(CCO)C1 c1(OC)cccnc1C(=O)NCC12CC1CN(C(C1C3COCC13)=O)C2 N1(C(CCCOC)=O)CCCCC(NC(=O)C=CC2CCCO2)C1 c1(CC)ccc(C)c(C(=O)NC2CCCCN(C(c3cscc3OC)=O)C2)c1 N1(C(c2ccn(CC)n2)=O)CC(NC(c2ncccc2OC)=O)CC2(CC2)C1 c1(C(=O)NCC(CN(C(C2CC(CC)C2)=O)C)O)cccc2[nH]ccc12 c1(C(=O)NC2CCCCCN(C(C(C)O)=O)C2)cn(C)c2ncccc12 C=CCC(C)(C)CC(=O)N1CCC(C(C)C(N2CCC2(C)CCO)=O)CC1 N1(C(c2nc(-c3c(OC)ccs3)sc2)=O)CCOC(c2ccccc2Cl)C1 c1(CC)ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)cn1 c1(SC)cc(C(=O)NC2CN(C(=O)CC3CCOC3=O)CC2F)cc(Cl)c1 C(N=c1[nH]nc2cccnn12)c1ccc(Nc2nc(C)nc(NC3CC3)c2)cc1 c1(NCc2c(C)nn[nH]2)nccc(=NCC2C(F)(F)C23CCCC3)[nH]1 C#CCC(CC#C)C(=O)N(CCCNC(C1(O)CN(C)C1)=O)CC C1(CC(=O)N(CCCOCCN(C(=O)CCF)C)C)(C(F)(F)F)CCC1 C(C(C)(C)CNC(C1(OC)CC1)=O)N(C(=O)COCC1CCCOC1)CC N1(C(C(c2cccnc2)NC(CCC(=O)N(C)C)=O)=O)CC2CCCC(C1)N2C C1(C2CC2)(C(=O)NCC2(F)CC(NC(CNC(C)=O)=O)C2)CCOCC1 CC(C)C(C(C)NC(=O)CC(C)(C)C)NC(c1ccnc(C(F)F)c1)=O C1(NC(c2cc(OC)no2)=O)C2CC1N(C(=O)CN(CCO)CCO)C2C c1(C(=O)NCC2CN(C(C3CC34CC4(F)F)=O)C2)cccc2c3c([nH]c12)CCC3 N1(C(C(C=C)(C)O)=O)CCN(C(c2cc(C3CC3)n(CC)n2)=O)C(CO)C1 c1(NC(C2CC(O)CN2C(=O)C2CC2)=O)cnc2cccc([N+](=O)[O-])c2c1 c1(C(N2CCC(O)(C(C)NC(c3nc(CCC)sc3)=O)C2)=O)cnc(O)c(F)c1 C1(C(N(C(C(=O)OC)C)C)=O)(NC(=O)CCc2nccs2)CCC(C)(C)C1 c1(OC)cccc(C=CC(N2CC(NC(c3scnc3C)=O)C(C)C2)=O)c1 C1(NC(C2C(C)N(C(=O)Cn3cccc3)CC2)=O)CCC(=O)NC1(C)C C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC(CCOC)COC C1(=O)CCCCOC1.N1(C(CCOCCCNC(=O)OCC)=O)CCCC(C)C1 CCCCC(C)CCC(=O)NC(C)CSC.C1C(C2CCC2)CC(=O)N1C C1(CNC(c2ccc(COC)cc2)=O)(NC(=O)CNC(C)=O)CC2CCC1C2 C1(=CC(=O)NCC(CCNC(C2CC=C(C)CC2)=O)O)CCOc2ccccc21 N1(C(CN(c2ncccn2)C)=O)CCCC(NC(C2CCCC(O)C2)=O)CCC1 CC(C)C1=NOC(C(N2CC(F)(F)CC2CCNC(=O)C=Cc2ccsc2)=O)C1 O=C(O)CC(CC1CC1)NC(=O)CNC(=O)COc1ccc(Cl)cc1.C1CCO1 c1(C(=O)NC2(C)CCN(CCCCCC)C2)cccc2occc12 C1(N(C)C(c2ccc[nH]2)=O)CN(C(c2cnn(C3CCC3)c2)=O)CCC1O CC1(C)CC(F)(F)CCC1C(=O)NC1(CNC(=O)Cn2cnc([N+](=O)[O-])c2)CC1 c1(OC)cc(C)c(C(N2CC3(CCCN3C(C3CC3C3CC3)=O)C2)=O)c(C)c1 c1(C(=O)NC(CC=C)CNC(C2C=CCCC2)=O)ccc(CO)cc1F c1(COC)cc(C(=O)NC(Cc2ccccn2)CC(=O)O)sc1C N(C1CCc2c(C)cccc21)C(c1n(C)nc(C)c1Br)c1nnnn1C C1(OC)CCCC(C(=O)NC2CC(CNC(c3cc(=N)[nH]n3C)=O)C2)C1 CC(O)C(C(N)=O)NC(c1ccc(CNC(c2ccc(N)cn2)=O)cn1)=O N1(C(C(C)NC(C)=O)=O)CCC2CN(Cc3ccnc(F)c3)CC12 CC1CC(c2cn(CC(F)(F)F)nn2)CCN1C(c1cc(Cl)sc1Br)=O CC1CN(C(c2ccccc2C(=O)NC(C2CCC2(C)C)=O)=O)CCC1SCCO.C C1(CCC)CCN(C(c2ncnn2CC)C(=O)N(CC(C)C)C2COC2)CC1 c1(C(N2CCN(C)CC2CNC(=O)C(C)(C)C)=O)nc2cncnc2nc1O C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1cc(C)cs1)=O N1(CC(C)NC(C2C(C)C2(F)F)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 C(C(=O)NC(CC1CCC1)C(=O)N(CC1=CCCOC1)C)(C(C)(C)C)OC Cc1ccc(C)c(OCCC(N2CC3(NC(=O)CC4CC(CF)C4)CC2C3)=O)c1 C1(C)(C(=O)NCC2CC(C(=O)NCC(CC)(O)CC)C2)CC2C=CC1C2 N1(C(c2ncn(CC)n2)=O)C2CCC1CC(NC(C1(C)CCC(OC)CC1)=O)C2 C12(CCC(=O)OCc3ccn(C)c3)CCC(CC1)C2 c1(NC(=O)CCNC(=O)NCc2ccccc2Br)cccc2c1NCC2 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2C)=O)nc(Br)n2ccccc12 C1(NC(C(CC)C(C)C)=O)CN(C(=O)C(C)(C)C2CCCC2)CC(F)(F)C1 C1(NC(C(C(C)C)N2CCCC2)=O)CCc2nnc(-c3ccccc3)n2C1 N1(C(CSCC=C)=O)CC2CC1CCC2NC(c1ccc(C(C)(C)C)c(Cl)c1)=O N1(C(C2(C#C)CC2)=O)CCC(N(C)Cc2ccn(C(C)C)n2)C1 Cn1cc(C(N2CC=CC2CNC(=O)CCN2CCOCC2)=O)cn1 C1(c2n(CCCSC)nnn2)(NC2CCC3(CC2)CSC3)CCCC(C2CC2)C1 c1(C(COCCCC)NC(=O)NNC(=O)c2conc2C)cccc(Cl)c1 N1(C(C2CC(CC)C2)=O)CCCCC(NC(c2cncc(OC)c2C)=O)C1 CN1C(=O)C(NC(=O)NCC(N2CCCC2C(N)=O)=O)CC1c1ccc(Br)cc1 C(c1cc(F)c(O)c(F)c1)=CC(=O)NC(CNC(c1cnnc(O)c1)=O)C1CC1 c1(CNC(COCC)=O)ccc(COC2CC(OC(C)(C)C)C2)nc1 N1(C(CCc2ccc(C)o2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C(O)C1 N1(C(C(=O)N(CC(CC)(C)OC)C)=O)Cc2ccc(O)cc2C1 N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1C(C)C C12(C(N3CC(NC(C(=O)NC(C)C)=O)C(F)CC3)=O)CC=CCN1CCC2 c1(C(N2CCCC(CCCCNC(C=CSC)=O)C2)=O)ccc2nn[nH]c2n1 c1(C(N(C)Cc2ncon2)=O)cn2c(n1)CCN(C1CCC(C)(C)C1)CC2 NS(=O)(=O)c1ccc(CC(=O)NCCCCC(CO)NC(=O)CC2CCCO2)s1 N1(c2ncc(C)cn2)CC2CCC(NC(C3CCCN3N=O)=O)CC2C1 c1(CC(=O)NCCOCCNC(=O)Cc2ccns2)ccc([N+](=O)[O-])cc1Cl C(=O)(CC(C(F)F)c1ccc(F)cc1)NC1C(NC(CCC(=C)Cl)=O)C1 C(=O)(C(C)(O)C(C)(C)C)NCC1CC2(CC(NC(c3c(CC)ocn3)=O)C2)C1 c1(OC)ccc(CN2CCC2C(=O)Nc2nc(Br)ccc2C)cc1C(F)(F)F C1(COC)(CNC(=O)CCC2CC2(Cl)Cl)CCCN1C(=O)Cc1c(C)noc1Cl C1(NC(c2ccc(C#C)cn2)=O)CC2CCCC(C1)N2C(=O)C(F)=C1CCCC1 Cc1ccncc1C(=O)NC1CC1C(=O)Nc1cnsc1 C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)C(C)NS(C)(=O)=O)C2)c(F)c1 CC1CN(C(=O)C(C)N(C)C)CC1CC(=O)NC(CO)C1(C)CC1 C1(C(=O)NC2CCN(CCOC)C2)CN(C(=O)C=CCN2CCCC2)CC12CC2 Cc1occ(C(F)(F)F)c1C(N1CC(CNC(c2cn[nH]c2)=O)C(C)C1)=O c1(N2CCCC(CCNC(c3ncc(C)c(C)c3)=O)CC2)ncnc(C)c1C#N N1(C(C(CC2CCC2)NC(Cc2c(C)n[nH]c2)=O)=O)CCOC(CN=[N+]=[N-])C1 c1(C(=O)NC(CNC(C2(COCC)CC2)=O)(C)C)nn(C)c(=O)cc1C N1(C(C(COC)(C)OC)=O)CCCCC(NC(C2CC(N3CCCC3)C2)=O)C1 C1(CNC(CC(=O)NCC#C)=O)CC2(CCN(C(c3nocc3C)=O)C2)CO1 Cc1c(C(=O)NC(C)CC(C)(C)c2ccccc2)cccc1Cl N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCCCC1CC(O)C(F)(F)F c1(C(=O)NC2(C)CN(C(C3(CO)CC(C)(C)C3)=O)C2)cc2ccsc2s1 S(=O)(=O)(CCC(=O)NCC1CCN1C(c1cnc(C(F)(F)F)c(F)c1)=O)NC c1(CNC2CCC(C(=O)NCc3c(OC)cccc3)OC2)ccc(Br)cc1O c1(C(=O)NC(CCNC(Cc2c(C)n[nH]c2C)=O)C(C)C)ncc2[nH]ncc2n1 c1(C(N2CC(N(C(c3c(CCC)occ3)=O)C)C2)=O)ccc(Cl)c(OC)c1F C1(NC(c2cnc(OC)c(C)n2)=O)CCC12CCN(C(=O)C1=C(Cl)CCC1)CC2 Cc1sccc1C(=O)NCC(F)CNC(=O)C(F)(F)C1CCOCC1 C1(CC)CN(C(=O)CC2CCN(C)C2=O)CCN1C(=O)Cc1ccc(OC)nc1 C1(CNC(COc2cc(C)on2)=O)CC12CCN(C(=O)Cc1ccc(Cl)s1)CC2 c1(OC)cc(C(N2CCC3C(NC(=O)Cc4cn[nH]c4)C3CC2)=O)ccc1C#N O=C1NC(C(=O)NCC2(CCNC(c3ccc(F)cc3CO)=O)CC2)C2CCC12 C12(CNC(C(c3cccnc3)C)=O)CC(CN1C(=O)CNC(c1cccnc1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)CCNS(=O)(=O)C(F)(F)F)OC c1(C(=O)NC2CCCC(NC(C=C(C)Cl)=O)C2)cnc2c(c1)C(=O)CCC2 C1(NC(c2nc(COC)sc2)=O)CN(C(c2cc(C3CCC3)[nH]n2)=O)C(C)(C)C1 N1(C(CNC(CC)=O)=O)CCC2(CCCCC2NC(c2cscc2C(F)F)=O)C1 N1(C(CN(C)C(C2(CS(N)(=O)=O)COC2)=O)=O)CCCCC1CO c1(CC2CCC2)cc(O)ncc1-c1nc(C2(C)CC2)nn1Cc1ccc(Cl)cc1 C1(C#N)(C(=O)NC2(C)CCN(C(C3CCCS3)=O)C2)CC2CCC1CC2 C(=O)(NNc1cccc2ccccc12)Nc1cc(SC)ncc1 C=CC1(C(=O)NC2CC(NC(=O)C(F)OC(F)(F)F)C2)CCCCC1 C1(NC(=O)Nc2c(OCC)ccs2)CCCCCC1c1ccccc1 CC1CN(C(c2cnc(C3CCCO3)s2)=O)CCN1C(c1cc[nH]n1)=O c1(C(=O)NCCC(Cn2cc(CC(COC)O)nn2)F)ccc(F)c(OC)c1 C1(CN(CC)CC)CCN(C(c2ccn(C3CC3)c2C)=O)CC1 c1(C(=O)NCCC2CCCN2C(=O)C(F)OC(F)(F)F)cnc2n1CCOC2 C=CCCC(C)(C)CNC(=N)NC(C(CC)CC)c1ccccc1 N1(CCC(=O)NCCNC(=O)CCc2cnc(O)[nH]2)Cc2ccccc2C1 N1(C(CC2N(C(C(C)OCC3CC3)=O)C3C2CCC3)=O)CCc2ccncc2C1 c1(NC(c2ccncc2F)C)cc(NCC(N2CCCCCC2)(C)C)ncn1 CC(C)CC(C)(CNC(=O)CCOC1CCCC1)NC(C1CCC1C(C)(C)C)=O Cc1nc(C(C(C)C)NC(=O)CC2CC3CC3C2)no1 C(=O)(CC1=NN(C)C(=O)C1)N(C)CC1(O)CCCN(C(C(C)SC(C)C)=O)C1 CC1CN(C(c2ccnc3ccnn23)=O)CCCN1C(C1CC=CCC1)=O N1(C(C2N(C(=O)OC)CCC2)=O)CC(NC(c2cccc[n+]2[O-])=O)C(O)C1 C1(NC(C(c2n(C)ccc2)=O)=O)CS(=O)(=O)CC1NC(C1CCC1)=O C(=O)(C(CC(C)C)C(C)C)NCC#CCNC(c1c(C)nc(N)cn1)=O N1(CC(=O)NC(C2CCCN2C(c2csnc2C2CC2)=O)C)CCC(C)(O)C1 C(C)(CC(=O)N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)(C(F)F)N(C)C Brc1ccc(CN2CCOCC2)c(N2CCOC(c3cccs3)C2)c1 N1(C(C(CCC)c2ccccc2)=O)CCCC(NC(=O)C(F)(F)COC)C1C C1(C(N2CCC(O)(CCNC(C(CC)C#N)=O)CC2)=O)CCC2(CCOCC2)O1 c1(C(=O)NC(CCCCC(=O)OC)C)ccc2nc(F)ccc2c1 c1(C(N2CCC(COC)(NC(=O)C=CC3CCCO3)C2)=O)ccc2nncn2c1 c1(CNC2C3CN(C(C4CCC(OC)CC4)=O)CC32)cc(C)c(Br)cc1F N1(C(CCCCC)=O)CC2CCN(C(c3c(C)ccc(Cl)c3F)=O)CCC2C1 CCC(CC(=O)NC(C)C(C)(C)CO)N(C(=O)C=CC1(C)COC1)C Cc1c(C(N2CC(O)CC2(C)C(=O)NC2CC(C)C2)=O)[nH]ccc1=O CCCC(O)CC(=O)NC1CN(C(C2(c3cccs3)CC2)=O)CC1C c1(C(=O)NC2CN(C(COC)=O)CC(C)(C)C2)cc2c(Br)c(F)ccc2[nH]1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC(C(C)NC(CCC(C)C)=O)C Cn1ncc2cc(C(=O)NC3(C)CCN(C(c4cc(N)cnc4Cl)=O)C3)sc12 c1(OC)cc(OC)cc(C(=O)NC2COCC2NC(C2CC2(F)F)=O)c1 C(N=c1[nH]c(=NC(C)c2ccc(Cl)cc2)[nH]c2c1COC2)C1CC(=C)C1 C(c1cccc(F)c1)=CCC(=O)NCC1CC1NC(C1CC(N2CCC2)C1)=O c1(C(N(CCN(C(CC=C=C)=O)C)C)=O)ccc(N2CCC(C)=N2)cc1 C1(NC(c2c(C)sc(Br)n2)=O)CN(C(=O)C=CCO)CCC1CO N1(C(C2CC2CNC(C2(NC(C)=O)CC2)=O)=O)CCCN(C=O)CC1 N1(C(C(C)C2CCCO2)=O)CC=C(C(=O)N2CCn3nccc32)CC1 C1(CNC(CCCC#C)=O)CN(C(=O)Cc2cc(F)cc(F)c2)C(C)(C)C1 N1(C(=O)CC(c2ccccc2)N2CCCC2=O)CCC2(CCN(C(=O)C(F)F)C2)C1 Cc1c(-n2nc(CCN(C)C)nc2Cc2nncn2C)cccc1Cl C(=O)(CC(C)C(F)F)N1CC(OC)C(C(=O)NCc2cccc(C)c2O)C1 C(CCC(=O)NCCN(C(c1occc1CC)=O)C(C)C)OCCC C(CCCC(=O)N(C)CC1CCCN(C(=O)CCSc2ccccn2)C1)OC N1(C(C2=NOC(C)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC(O)C1 c1(C(=O)NC2CCN(C(C(C)(C)Cc3ccccc3)=O)C2)nccc2[nH]ccc12 C(C(CNC(=O)C(Cc1ccco1)NC(=O)CSc1ccccn1)C(C)C)OC c1(OC)ccc(C(=O)C(=O)NCC2CCC(C)CN2C(c2cccs2)=O)cc1Cl c1(C(=O)NC2CC3(CN(C(CC(COC)COC)=O)C3)C2)ccn2nncc2c1 c1(NC(c2nnnn2Cc2ccccc2)(C2CCOCC2)COC)cncnc1C C1(CNC(C2CC=CCO2)=O)CCN(C(c2cnnc(O)c2)=O)CC1O N1(C(CCN(C)CC)=O)CCC(O)(C(C)Nc2nccc(-n3ccnc3)n2)C1 c1(OC)c(O)cc(C(N2CCCC2C(=O)Nc2cnc(C)c(Br)c2C)=O)cc1O C12(C(N3CCC(O)(CN(C(C(CCN(C)C)O)=O)C)C3)=O)CCC(O)(CC1)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(=C)CC1C(=O)NC1CCSC1 C(=O)(C1CCCc2sccc21)NCC(C)N(C(c1c(C)n2c(nc1)ncn2)=O)C N1(C(CC2(C=C)CC2)=O)CCC(O)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C(=O)(C#CC(C)(C)C)N1CC(ONC(c2c(C)nccn2)=O)C1 C1(C(=O)NCCn2ncc(C)c2)CN(C(=O)CC23CCCC2C3)C(C)(C)C1 c1(OC)cc(OC)c(Cl)c(C(N2CC(CNC(c3cc(OC)n(C)n3)=O)C2)=O)c1 CC1(C#N)CCN(C(C2CC3C=CC2N(C(c2c[nH]nc2C2CC2)=O)C3)=O)CC1 CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)NC1CCCCCC1CO)C2)=O c1(C(=O)NC)cc(S(=O)(=O)NCC2(O)CCOCC2)cn1C C=CC(C)C(=O)Nc1cn(CC(=O)NOCC=C(C)C)nn1 C(=O)(C(CO)C(F)(F)F)NC1CC(C(=O)NC(C2CCCO2)CC)C1 Cc1cc(O)c(C(=O)NCCCC(=O)N(C)C)cc1F Nc1c(C(=O)OCC(=O)NCC(C2CCOC2)O)ccc(Cl)c1Cl C(CC(C)C)(C(=O)NC(Cn1cncn1)C(=O)N1CCC(CC2CC2)C1)OC CC1CCCC(C)CN1C(=O)CC(C)(C)CNC(C1(C#N)CC1(C)C)=O C(c1cc(OC)cc(OC)c1)=CC(=O)NC(C(C)NC(C(CC)CC)=O)C C1(C)(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(=O)CCc1cc(C)on1 c1(CC(=O)N(CCN(C(c2c(NC)cnnc2)=O)C)C(C)C)csc2nccn12 C1(C)(NC(COC)(C)C(c2nnnn2C2CCC(C(=O)OC)C2)(C)C)CCCC1 C1(C(=O)NCC2(C(N3CCC3CO)=O)CC(=C)C2)CSCC(=O)N1 C1(NC(c2c(OC)nsc2)=O)(CO)CCCN(C(c2n[nH]cc2C)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)CC(C)(C)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CC(C(C(=O)N2CCC2CC2CC2)OC)C1 N1(C(CNC(CCC)=O)=O)C2CCCC1CN(C(c1cc(OC)ns1)=O)C2 c1(N2CC(C(C)NC(C(c3cccnc3)OC)=O)C2)nn2cc(C)nc2s1 N1(C(c2c(C)ocn2)=O)CC(N(C)C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 C1(C(=O)NCC2CCN(C(c3noc(CC)c3C)=O)C2)CC2COCC(C1)C2 N1(C(c2c(C)cc[nH]2)=O)CC2(CCN(C(C3CC3c3ccccn3)=O)CC2)C1 N1(C(C2CCSCC2)=O)CC2CCC1C(CNC(C13CCCN1CCC3)=O)C2 N1(C(CC(COC)C)=O)CCN(C)C(C(N2CC(CO)C2(C)C)=O)C1 C1(NC(c2cn(CC=C)nn2)=O)CC1C1CCCN(c2ncnc3c2CCO3)C1 Cc1cc(Cl)ccc1CNCC1CCCN1C(c1ccc(-c2ncc[nH]2)nc1)=O C1(NC(c2cnnc(Cl)c2)=O)CCCCC1NC(c1occc1Br)=O C1(C(=O)NCC(C)C)COCCN1C(c1cnc(Br)s1)=O C1(C(=O)NC(CC)CNC(c2nnsc2C)=O)CCCCC1O N1(C(CCC2CC(OC)C2)=O)CCCC(CCNC(=O)CCCN(C)C)C1 c1(Sc2n(C)ccn2)ccccc1NC(=O)NCC1(C)CNC(=O)O1 C1(C(C)NC(C2(CCOC)CCC2)=O)CCCN(c2nnc(C#N)s2)C1 C1(C(N2CCC(C)(CNC(c3ccc(C)s3)=O)CC2)=O)CCS(=O)(=O)C1(C)C N1(C(C=CCN(CC)CC)=O)CC=CC1(C)C(=O)NCCc1cn(CC)cn1 c1(CCC(N2CCN(C(C3CC3(F)F)=O)C3CC23)=O)c[nH]c2ccccc12 c1(C(=O)NCc2c(C(=O)NC3C(CN(C)C)CCC3)scc2)ccc(N)c(F)n1 N1(C(c2cc(OC)c(C)cc2)=O)CCCC(C2(NC(=O)C3=CCSC3)CC2)C1 C1(C)(NC(c2ccn(C)c2)=O)CCC(NC(=O)Cc2c(Cl)cccc2Cl)CC1 c1(C(=O)NCC(N(C)C(C2(Cl)CC2)=O)C2CC2)cc(Br)cc([N+](=O)[O-])c1 Cc1ncnc(O)c1CCC(=O)NCC(C)(CO)NC(C12COCC1C2)=O C1(F)(C(=O)NCCN(C)C(c2cc(OC(F)F)n(C)n2)=O)C2CCCCC12 O(C1CCc2cc(Br)cnc21)C(C(c1cccc(F)c1)C)=O C(=O)(C(C(C)O)NC(=O)C(C)(C)C)NC(Cc1cc(SCC)n[nH]1)=O N1(C(c2c(C)noc2)=O)CC(NC(=O)CCc2ccc(Br)c(F)c2)C2(CC2)C1 c1(C(C(=O)NC(C2C3CN(C(c4ccccc4F)=O)CC23)C)O)cccc(Cl)c1 C1(C(=O)NCC(c2ccncc2)O)(CC)CCCN(C(=O)C=Cc2ccoc2)C1 c1(C(N2CC(CNC(C(CC=C)OC)=O)(OC)C2)=O)ccc(N)cc1Br C1(CC)CCC(C(N2CCCC2(C(=O)N(CC(F)(F)CO)C)CC)=O)CC1 N1(C(CN2C(=O)CSC2)=O)CCN(C(c2cccc3cc[nH]c23)=O)C2CCC12 c1(CC)[nH]nc(C(N2CCCC2CN(C(C2C=CC=CC=C2)=O)C2CC2)=O)c1Cl N1(C(C2C(CC)C2)=O)CCC(CNC(=O)C2=CC(C)(C)C2)C(CC)C1 c1(CCCC(=O)NCC2C(NC(c3c(OC)c[nH]n3)=O)C2)ccc(Br)cc1 C1(C(=O)NC2(c3cn(C)nc3)CC2)CC(O)CN1C(=O)C(C)(F)c1ccon1 O=C(O)CC(CC(=O)Nc1cccc(CC(F)(F)F)c1)c1cccc(F)c1 Cn1nncc1C(c1cnc(CC(F)(F)F)s1)=O C1(CC)C(NC(=O)C=C(C)C2CC2)CCN1C(=O)CCCOc1ccc(C)cc1 Cc1cnc(C(=O)NC2(CO)CCN(C(=O)C(=O)NC3CC3)C2)c(C)c1 N1(CC=CC(=O)NCC(n2ccnn2)C)CCCC1 N(C(=NCCSc1nccn1C)NCC1CCCC(=O)N1)C(c1nncs1)C c1(C(=O)OCC)cnc2nc(NS(=O)(=O)C3CCC(N(C)C)C3)oc2c1 C1(CN(C(C2C(C)(C(=O)OCC)C2)=O)C)CCN(C(=O)Cn2ccc(C)c2)CC1 c1(C(C)C)nocc1C(=O)NCC(C1(O)CN(C(=O)CN2CC3CC3C2)C1)(C)C c1(OC)cccc(-c2cn(C(C)CNC(c3ncc(C)cc3C)=O)nn2)c1F C=C1COCCN(C(c2cnc(C(F)F)s2)C(=O)NC2(C)CC2)C1 N1(C(C2(CCC=C)CC2)=O)CC2(C(=O)NCc3cnn(C)c3C)CC1CO2 c1(CCC(=O)N(CCC(C)NC(=O)C(C)(C)CO)C)ccc(Cl)cc1Br C#Cc1ccc(C)c(NC(C2CC3CC3N2C(=O)C(C)(C)CC2CC2)=O)c1 c1(C(N2CCN(C(C(C(C)C)SCC)=O)C(C)C2)=O)ccc2c(C)noc2n1 C(=O)(C#CC1(C)COC1)NCC(C)NC(c1ccc(C(F)(F)F)[nH]1)=O CC1(C)C2CCC1(C)C2C(=O)NC1CCN(C(c2cc(Cl)cs2)=O)C12CC2 CC1C(=O)N(CC(=O)OCCC2CCC(C)C2)C(=O)C1C C(=O)(C(C)S(=O)(=O)C(C)C)N(CC(C)NC(c1c(NCC)ccc(Cl)c1)=O)C N1(C(C2CC(C(C)C)C2)=O)CCC(N(C)C(c2coc(CC3CC3)n2)=O)C1 N1(C(CCOCCCOC)=O)CCC(C2(NC(=O)CCNC(N)=O)CC2)C1 C1(CC)CC2CCC1(CNC1(c3nnnn3CC)CCCC(CC(=O)OC)C1)C2 CC1CC(C(=O)NCC2CCC(CNC(=O)COCC3CC3)CC2)CCS1 c1(CC)noc(CC)c1CC(N1CC(O)(C(C)NC(c2ncn(C)n2)=O)C1)=O N1(CCC)C(=O)CCC1C(=O)N(CCCNC(=O)CCCC#N)CC N1(C(CCC=C)=O)CCOCC(CNC(c2nn(C)nc2Br)=O)C1 C(CCO)(C(F)F)N(C(C(C1(O)CCC1)NC(CCC)=O)=O)C C1(NC(N2C(CC)CCCC2)=O)Cc2c[nH]nc2CC1C Cc1cc(C(=O)NC2C=CC(C(=O)NCC3CC(C(C)C)C3)C2)[nH]c1C c1(OC)ccc2c(N(C3CCNCC3F)C(c3ccc(Cl)c(O)c3)=O)ncnc2c1 Cc1c(C=CC(N2CC(NC(=O)CNC(=O)C3CC3)CC2(C)C)=O)cnn1C N1(C(c2ccc(OC)nc2)=O)CCC(C2CCN(C(=O)C(C)P(C)(C)=O)CC2)C1 c1(OC)ccc(C2CC2)cc1NC(C1CCN(C)CC1)=O N1(C(CCN(CCC)C)=O)CCN(C(c2ccccc2C(F)(F)F)=O)CC(O)C1 N(C(=NCC(C)C)N1CCC2(CC(C(F)F)=NO2)C1)Cc1ccc(CCC)cc1 c1(CC)ccc(N(C)C(C2CC(NC(=O)Cc3cccc(F)c3)C(O)C2)=O)cc1 c1(SCC)ccccc1C(=O)N(CC(C)CNC(C1CC1c1nccn1C)=O)C c12cccc(c1)S2.C1(NC(=O)C2CC2)CCN(C(=O)CC2CC2C(F)(F)F)C1 N=c1nnn(CC(=O)NC(c2ccccc2)CNC(c2nn[nH]c2Cl)=O)[nH]1 c1(OC)nn(C)cc1C(N1CCCC1(C(=O)NC1(CF)CC1)C(C)C)=O O=C(C#CC1CCCC1)NC1COCCN(C(=O)CN2CCSCC2)C1 CCCC(C)CC(=O)N1CC2(CNC(C3CN(C)C3)=O)CCC1C2 C(=O)(CCC(O)C(C)(C)C)N1CC=C(CNC(c2c(C)nc(C3CC3)nc2)=O)CC1 c1(CC)cccc(NC(C2(NC(=O)CC3CCCC3C)CC2)=O)c1 c1(C(N2CC(CS(C)(=O)=O)N(C(=O)C3=CCSC3)CC2)=O)cnc2n1CCOC2 CCC(C)C(C)(O)CNC(=O)CCC(C)(C)NC(c1cnc(C)nc1)=O CP(C)(=O)CC(=O)NCC1(O)CN(C(c2cc(CCCO)on2)=O)C1 c1(OC(C)C)cccnc1C(=O)NC1CCC1NC(=O)C=Cc1cscn1 O=C1NCC(C(=O)NCC#CCNC(=O)CCCn2cccn2)N1 C#Cc1ccc(CC(N2CCC(NC(=O)C=C3CCN(C)CC3)C(O)C2)=O)cc1 c1(NCC2(CNC(c3nnn4ccccc34)=O)CC2)c(Br)cccc1[N+](=O)[O-] C(C(=O)N1CC(O)CCO1)N(C(C)CC(N(C)C[Si](C)(C)C)=O)C C#Cc1cccc(C(N2CCOCC2CNC(C2CC2C=C)=O)=O)c1Cl c1(OC)c(C(N2CC(OC)C(NC(=O)Cn3ncn(C)c3=O)C2)=O)cccc1N C(=O)(CC(C(F)F)n1ccnc1)NCCC(C(C)C)NC(=O)CCCOC(C)(C)C O=C(C1=C(Cl)CCC1)NC1CC(NC(c2cccc(-n3cncn3)c2)=O)CC1O c1(OCC(=O)NCC(CC)NC(C2CCCC2(C)C)=O)ccc(F)cc1 N1(C(=O)NN(C)Cc2ccc(NC(C)=O)cc2)CC(N(C)C)CC(C)C1 C(C1=NOC2CN(C(c3scc(C)c3OC)=O)CC12)NC(COCC=C)=O c1(C(=O)NCC(C)NC(c2cc(OC(F)F)n(C)n2)=O)cccc([N+](=O)[O-])c1O c1(OC)noc(C)c1C(=O)NC(C)CCCCNC(c1cc(C(C)=O)c(C)o1)=O C(CC(C)C(=O)N1CCC(C)C1C(=O)NCCC(=O)NCC)=CCC c1(NC)cc(C(N2CCC(NC(C3CCN(CC(C)C)CC3)=O)C2)=O)cc(Cl)n1 C1(OCC)COCCC1NC(c1cncc(CNc2ccccn2)c1)=O C(C(C)CC(=O)NCCC1(C(=O)NC2CCC(F)(F)C2)CC1)NC(C)=O C1(C(=O)NC2CN(C(c3cc(CCC)n(C)n3)=O)CC2C)CN2CCN1CC2 C1(NC(C(C)SCCCC)=O)CC(C)CN(C(c2cncc3c2CCC3)=O)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCCC(NC(=O)CCc2ccc(Cl)s2)CC1 C(=O)(NNC(=O)C(=O)NC(C)CC1CCCCC1)NCC1CC(C)CC(C)C1 C1(NC(=O)CC2CCCC2)CN(C(C2CC2c2ccccc2)=O)C2CCCC12 c1(CCC)sc(C(=O)NC(C)(CNC(=O)C(C)c2ccsc2)CO)cc1CC C12(CC)CC(NC(c3cc(CNC(=O)C(C)=C4CC4)on3)=O)(CO1)C2 C1(C2CC2)(CNC(CN(C)C2CC2)=O)CCN(C(c2cnsc2)=O)C1 C(=O)(CCCC(=O)N(CC1C(NC(CSCCC)=O)CCCC1)CC)NCC O=C(C#CC1CCCCO1)NC1CCC2(CC1)CC(NC(=O)C(F)C1CCC1)C2 C1(CCNC(C2(CC)CC2(F)F)=O)CN(C(c2cncnc2C2CC2)=O)CCO1 C(CC(C)(c1nnnn1C1CCCC1)NCCCCO)(OC)OC c1(C(=O)OC)ccc(F)c(CN2CCC(F)(C(=O)NC3(CC#N)CCCC3)C2)c1 O=C(N=c1nc(O)[nH]c(O)n1)c1c[nH]c2ccc(-c3ccnc(O)c3)cc12 CN(NC(=O)Cn1cc(CCCC#N)nn1)c1ncccn1 C12(NC(c3c(Cl)ccc(OC)n3)=O)CCCC1N(c1nnco1)CCC2 c1(C(=O)NCC23C(CN(C(C4(NC(C)C)CC4)=O)C2)C3)nccn2ccnc12 N1(C(COC(C)(C)C)=O)CCC2CN(C(c3ncc(Cl)cc3Br)=O)CCC12 N1(C(c2c(C)onc2Br)=O)CCN(C(C2CC2F)=O)C(CO)C1 C(=O)(C(C)(C)CN1CCOCC1)NCC(C)N(C(CCN(CC)CC)=O)C C#Cc1ccc(C(N2CC3(CC3)CC2C(=O)Nc2cnccc2CC)=O)c(C)c1 C1(NC(c2ccc(Cl)cn2)=O)CC=CCC1C(=O)NCC(O)C(F)(F)F CC1(CNC(C2CC(=C3CCC3)C2)=O)CCC(NC(=O)Cn2ncccc2=O)C1 Cc1nn(C)cc1C1CCC(CO)N1C(=O)Cn1nnnc1C N1(C(CCOCC#C)=O)CCSCC1CCNC(c1cc(C)n(C)n1)=O C1(n2c(C(=O)NCCC(C)(C)NC(=O)C3=CCOC3)cnc2)CCCC(O)C1 N1(C(c2ncn(CC)c2)=O)CCCN(C(=O)Cc2ccc(C)cc2F)CC1 c1(C(=O)NCC(CNC(CC2C(CC)C2)=O)(C)O)cc(Cl)n[nH]c1=N.CC=O Cc1cc(CNC(c2n[nH]cc2CNC(C2(C#N)CCOC2)=O)=O)ccn1 CC(C)(C)C(O)C(=O)NCC(C)(C1CC1)NC(c1cc(Cl)cc(Cl)c1)=O C1(CNC(CCOC)(C)c2nnnn2C(C)(C)C)(CO)COCC2CCCCN12 c1(OC)cccc2c(C(N3CCCC(NC(=O)COC4CCOC4)C3)=O)coc12 C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CCC1C(NC(=O)CC1CC(C)=NO1)C2 C#CCC(CC(F)F)NC(=O)C1=CCC(NC(c2cc[nH]c(=NC)c2)=O)C1 C12(NC(CC(CC=C)NC(=O)Cc3cc(C)cs3)=O)CC3CC(CC1C3)C2 c1(OC)ccc(C2(NC(c3cnn(CC(C)C)c3)=O)CCOCC2)cc1Br C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC2C(CNC(CS(CC)(=O)=O)=O)(C2)C1 C1(C(=O)NC2C3CC2CN(C(=O)C=Cc2nccs2)C3)CC2C=CC1C21CC1 C(CN=c1[nH]c(C2CC2)nc2c1CCC2)NC(=O)NC1COC(=O)O1 C(=O)(C1=CCC(C)(C)CC1)NCC1(C(=O)Nc2c(Br)cn(C)n2)CC1 C1(CC)C(NC(C2CC(N(C)C)C2)=O)CCN1C(c1csc(C2CCCO2)n1)=O C(C1CCOCC1)=CC(=O)NCC(C(C)C)NC(=O)Cc1ccn(C)n1 c1(C2(NC(N(CCN(CC(F)(F)F)C)CC)=O)CC2)cccc(Cl)c1Cl C1(c2cn(Cc3nc(CC)sc3)nn2)CCCCN1C(=O)C(F)(F)CC C(C(C)CCCC(C)C)NC(CC1(C)N(C(c2c(CC)nns2)=O)CC1)=O C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(c2cc(OC)c(Cl)cc2)=O)C1 c1(C(N2CC3(C(C(=O)NC(c4cnccn4)C)C3)C2)=O)ncc(Cl)cc1Cl C1(C(N2CC(CC)C2)=O)CC(O)CN1C(=O)CCCCNC(=O)C1CC1 c1(OCC)cc(F)c(-c2ccc(NCc3ccc(NC(C)=O)cc3)nc2)cc1F c1(C(=O)NCC2CCN2C(=O)CCOC2CC2)c(C(F)(F)F)nc2n1CCCC2 N1(C(COCC(=O)NCCC(N(CCOC)C)=O)=O)CCOCC1.C12CC(C1)O2 c1(OC)cccc(O)c1C(N1CCCC(CO)(NC(=O)CC2CCCCC2)C1)=O c1(NC(C2(CNC(c3ncoc3C)=O)CC(=C)C2)=O)cn(CC)nc1C#N C(=O)(CCCCCF)OCC(c1ccc(C#N)cc1)C c1(C(=O)NCC(CC)NC(c2ccc(F)nc2F)=O)cc(C2CC2)cnc1Cl CC(CS(C)(=O)=O)C(=O)NC1CCC1NC(c1cc(O)nc(N(C)C)n1)=O C1(OC)CC(CNC(c2ccsc2)=O)N(C(C2CC(=O)CCO2)=O)C1 c1(C(=O)NC2(CO)CCN(C(=O)CCc3cncs3)C2)cc2ccccc2[nH]1 c1(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)cccc(C(C)(F)F)n1 C1(C2CCN(C(C3(CO)COC3)=O)C2)(NC(C(CC(C)C)OC)=O)CC1 n1(C(CC)(C)C)nnnc1C(c1cnsc1)NC(C)CCc1ccc(C)o1 C1(C(=O)OC)CCCN(C(=O)Cn2ccc(-c3ncccc3F)n2)C1C C1(NC(CC(CC)O)=O)CCN(C(C2(N3CCCCC3=O)CC2)=O)CC1C C1(OC)CN(C(=O)C(F)=CC2CC2)C(C)(CNC(=O)Cn2cccn2)C1 C(CCCC(=O)O)n1cc(CN(CC(c2ccccc2OCC(F)F)O)C)nn1 C(=O)(C1=NNC(=O)CC1)N(CC(C)NC(=O)C=CC1CCOCC1)CC C1(NC(Cc2cn(CC)nc2)=O)CC(F)CN(C(=O)CN2CCOCC2=O)C1 C1(C(N(CC(C)O)CCNC(c2[nH]c(=NC)sc2)=O)=O)COC2(CCC2)CO1 N1(C(C(N2CCSCC2)C)=O)CCCCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 c1(NC(c2ccc(OC(C)C)cc2)=O)cc(C2=CCC(O)CC2)ccn1 c1(CNCC2C(CC(F)(F)F)CCCC2)nnn2c1CCCC2 c1(OC)ncc(Cl)cc1C(=O)NCC1CCN(C(c2ccn(C)c2)=O)C12CC2 C1(OC)CC(CNC(=O)COCc2ncc(C)o2)N(C(=O)CC(C)F)C1 N1(CC(=O)N(C(c2occc2C)=O)C(C)C)Cc2ccccc2CC1CO.CN c1(NC(C)=O)ccc(C(=O)N(C(C)CCNC(=O)C2=CCCS2)C)nc1 C(=O)(CC(F)(F)F)N1C(C(=O)NCCCC(C)NC(=O)C2=CCC2)CSC1 O=C(N=c1ccnc(C(F)(F)F)[nH]1)C1CC1C(=O)N(c1ccc(F)nc1F)CC c1(C(N2CC(=O)NCC2C(N2CCCC2CF)=O)=O)cccc2[nH]ncc12 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(=O)CC2CCCCC2)CC1C N1(C(C#CC(=O)N(C)C)=O)CC2CCN(C(C3CCC4(CCC4)C3)=O)C2C1 c1(C(=O)NC(CNC(c2onc(CC)c2C)=O)C)ccc2c(c1)C(=O)OC2 c1(C(=O)NCCCCNC(C(C)(C)N(C)C)=O)ccc(S(C)(=O)=O)o1 C(c1ccc(Cl)cc1F)=CC(N1CC(CC(=O)NCC(O)C(F)(F)F)OCC1)=O CC(C)C(C(=O)NCCC(C)NC(c1cnccn1)=O)c1cnn(C)c1 N1(C(C(C)C2CCCO2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)C(C)CN2CCOCC2)cc1Cl C1(c2ccc(Br)cc2)(NC(=O)Nc2cnc(OC(C)C)s2)CC2(CC2)C1 c1(NC(C2CCN(Cc3ccc(OC)cc3Br)C2)=O)ccc2c(c1)c(Br)nn2C C(=O)(C(O)CC(C)(C)C)NC(C1CCCC1)CNC(C(C)(C)OC(C)C)=O c1(N2CCC(NC(C3N(C)CCC3)=O)C(O)C2)ccc([N+](=O)[O-])c(C(F)(F)F)c1 N1(C(c2cnc(Cl)cn2)=O)CC2CCN(C(=O)COCC(F)(F)F)C2C1 c1(CC)c(C(=O)N(CCCCN(C)C(C2CCCN(C)C2)=O)C)ccn1C CC1CCCC1(C)CNCC(=O)N(C(F)C(=O)O)C1CCCC1.C(C)(C)(C)O C(N=c1[nH]cc(Cl)c(C)c1C#N)C1CN(C(C(C(CC)C)C)=O)CC1C(F)(F)F CN(Cc1ccc(Cc2cccs2)cc1)N1CC2(CC=CC2)C1CO N1(C(c2c(CC)ocn2)=O)CCOC2(CCN(C(C3CCCC34CC4)=O)CC2)C1 c1(CC)c(C(=O)NCCC(O)CNC(C2CC3CCCCC23)=O)cccc1C C(CN=c1ncc(C(F)F)c[nH]1)NC(=O)CC1CC(C)OC(C)C1.CCOC C1(C(=O)NC2CC(NC(C(C3CCCC3)OC)=O)C2)CCC(=O)O1 C(=O)(CS(=O)(=O)CC(F)(F)F)NC(CN(C(c1c(CC)ccc(OC)c1)=O)C)C CC#CCC(C(=O)N(CC)CC1CCOCC1)NC(=O)C(C)C(C)(C)C C12(C(=O)OC)CC(CNC(c3nnnn3CCCF)C3CC3)(C1)OC2C.n1(C)cnnn1 N1(C(c2c(SC)ccs2)=O)CCCC(NC(=O)Cc2c(C)noc2C)C(F)C1 c1(C(N2CC(O)(C(C)NC(c3cn(C)nn3)=O)C2)=O)ccc(F)cc1 c1(-n2cc(C)nc2)cccc(C(=O)NC(C)C(C)NC(=O)Cn2nnc(=O)[nH]2)c1 C(C)(CC1CCC1)(C(=O)N1CC(=C(F)CNC(c2ccncn2)=O)C1)OC N1(C(c2c(CCC)n(C)nn2)=O)CCN(C(c2cccnc2O)=O)C(C2CC2)C1 n1(CC(=O)N(C2CCN(C(C(C)(C3CC3)OC)=O)C2)CC)nnc2c1CCCC2 C12(C(=O)NC(CCOC)C(=O)NC(C)Cc3nn[nH]n3)CCCC1OCC2 Cc1[nH]c(-c2ccccc2)c(C)c1CN1C(C(N2CCOCC2)=O)CCC1C N1(C(c2cccc(OCc3ccc(F)cc3)n2)=O)CCCC2(CCNC2)CC1 C1(OC)CC(CNC(=O)C(C(C)C)C2CCC2)N(C(c2ccnn2C(F)F)=O)C1 N(C(=NCCCCl)NCc1cc(F)cnc1Cl)C1C(CC(C)C)C1 C=CCC(C)C(=O)N(C1CCN(C(=O)CNC(=O)Cc2cccc(F)c2)CC1)C n1(CC)nc(C(=O)NC(CC2CC2)CC(=O)NC(c2ccc(C)s2)C)cc1C N1(C(C2(COC)CC2)=O)CC(NC(=O)C=C(C)c2ccccc2C)CCC(O)C1 Cc1ncccc1C=CC(=O)NC(C)CN(C(=O)C(c1cccc(O)c1)C)C c1(C(N2C(C(=O)OC)CC(O)C2)=O)nn(C)c2c1C(O)CCC2 N1(C(c2ccn(C)n2)=O)CC2CC(NC(C3(c4ccnn4C)CC3)=O)CC2C1 c1(C(N2CCC3(CN(C(C4(SC)CC4)=O)C3)C2)=O)cc(C)ccc1S(N)(=O)=O c1(-c2n(C(C)C(C)(C)C)nc(CC3CC3)n2)cc(F)cc(Br)c1F C(C(COC)CC(=O)NCC1CN(C(C2(C(C)(F)F)CC2)=O)CCCO1)OC c1(C(=O)NC2CCN(C(C3CN(C(C)=O)C3)=O)C(C)C2)ccc2ocnc2c1 c1(OC)ccccc1C1CCN(C(=O)C(N)Cc2ccc(C(F)(F)F)s2)CC1 c1(CC)ccc(F)c(C(=O)NCC(C)N(C)C(c2cnsc2C)=O)c1F C(=O)(C(Cc1ccccc1)CC(C)C)N1CCN(C(C(=O)OCC)C)CC1 C(CCC(=O)N(C1(CC(C)C)CC1)C)NC.C(C(=O)NC(C)C)=CC=CCO CCC(COC)(C(=O)O)NS(=O)(=O)CCCCOc1ccccc1 CC(CC(C)(C)C)C(=O)N(CC(Cc1ccccc1)NC(=O)CC(C)(C)C)C C(=O)(CC(CC)CC)NC1C(NC(COCCCC#C)=O)CCC1 C1(C(C)(C)C)(C(=O)NC2CN(c3cc(NCCSC)ncn3)C2)CNC(=O)C1 C(C1CCCc2ccccc21)N1CCC(C(=O)Nc2nc(C)n(-c3nc[nH]n3)n2)C1 C(=O)(C(CNC(=O)CC(F)(F)F)CC(C)C)N(CCCC)CC CC1CCN(C(=O)C=C2CCCCC2)CCN1C(C1CC=CCO1)=O N1(C(C2(c3cccs3)C(C)C2)=O)CCCC(CNC(=O)COC2CC2)CC1 Cc1nc(S)sc1CC(N1CCC(CCNC(c2ccc(Cl)nn2)=O)CC1)=O c1(OC)cc(C)[nH]c(=NCC2CCCC2NC(c2cc(C)oc2C)=O)n1 c1(CC(=O)NC2C(C)CCN(C(C3COC(C)C3)=O)C2)cc2ccccc2o1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(CNC(c3c(CC)nccc3)=O)C(C2)C1 C(CN=c1[nH]c(=NCc2cc[nH]n2)[nH]c2c1CSC2)n1c(C)ncc1 C1(CNC(=O)COC2COC2)CCCN(C(c2scnc2Cl)=O)C1 C1(NC(C(Cn2cccn2)NC(c2c(C)[nH]cc2)=O)=O)CCN(C)CC1C C1(C#N)(CNC(C(CNC(C2CC(C)C2)=O)O)=O)CCCCC1 C1(C(=O)NCC2CC(C)(C)CCO2)CCC2CC1C2(C)C.CC1C2CCN1C2=O C1(NC(C(=O)Nc2n(C)nc(C3CCCO3)c2)=O)CC(C2CCCC2)C1 Cc1cccc(C(=O)NC2(CNC(=O)CCC3CCCCO3)CC2)c1Cl Cc1sc(CNC(N2CCC(CCCCO)CC2)=O)c(C)c1Br c1(C(=O)NC23CC(NC(c4ncc(NC)nc4)=O)(C2)C3)cnc2cc(C)ccn12 C1(C(N2CCC(O)CC2)=O)(COC)C=CCN1C(=O)C(C(C)OC)N(C)C N1(C(C(C(C)C)N(C)C)=O)CCCC(C)(C(=O)NC2CN(NC=O)C2)C1 C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)CC2CCCC2)CC(=O)CC(=O)N1 c1(C(=O)NC2CC(CCNC(=O)C(F)n3cccn3)C2)cc(SC(F)F)ccc1Cl C(CC(C(=O)NCCC1CCCN1C(C1CC1F)=O)OC)OC C1(NC(C(CSC)C)=O)CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)CC1O c1(C(=O)NCCCNC(C2CC3(C2)CC(F)C3)=O)cc(F)c(F)c(O)c1F C1(C(=O)NC(C)C(O)C(F)F)CC2(CCN(C(c3cc(CO)on3)=O)C2)C1 Cc1cccc(=O)n1CCCC(=O)N(O)Cc1cn(CC2CCCO2)nn1 C1(CNC(c2cnc(C)n2C)=O)CN(C)CCN1C(=O)CCc1cccs1 N1(C(C(Cn2cccn2)NC(C2CC(SC)C2)=O)=O)C2COCC1C2 CN1CCc2ccc(C(N3CCC3CNC(=O)Cn3ccc(Br)n3)=O)cc21 CCCC(C(=O)NCC1CCC1NC(=O)C(c1ccccc1OC)=O)NC(C)=O C=CC(C)(CC)C(=O)NCCCN(C(c1cc(Cl)ns1)=O)C1CC1 C=Cc1cncc(C(=O)NC(C2CCN(C(c3snc(O)c3Cl)=O)CC2)C)c1 c1(OC)cc(CN2CC(O)CC2C(=O)Nc2cnc(C)s2)cc(C(F)(F)F)c1 c1(C(N(CCCCCNC(CC(C=C)C)=O)C)=O)c[nH]c2c(Br)cccc12 c1(CC(=O)NC2C(NC(C3(C)CC(F)(F)C3)=O)C2)n[nH]c2ccccc12 c1(C(=O)NCCOC2CCN(C(CCC(C)OCC)=O)C2)cc(F)cc(F)c1N c1(CN(C(c2cc(Cl)cs2)C(=O)NCC2CC2)CCN(C)C)cccc(Cl)c1 n1(CC)ncc2c(NCC(C(C)C)OC)nc(N(CC(C)NC3CC3)C)nc12 c1(OC)ccc(F)cc1-c1cn(C2CCCN(C(c3[nH]c(C)nc3C)=O)C2)nn1 CCC(C)(CO)CN=c1[nH]c(=NCC2COCCO2)c2sccc2[nH]1 c1(C(N2CCC(C(C(=O)NC(c3ccn(C)n3)CC)(C)C)C2)=O)cnc(C)nc1 c1(C(N(C(=O)C(O)CCOCC)CC(C)O)=O)cc2ncccc2[nH]1 C(=O)(C1=NOC(C)(C)C1)N1CCCC(Cn2cc(-c3ccc(C)cn3)nn2)C1 C1(C)(C(N2CC(COC)(NC(=O)CCn3cc(C)cn3)C2)=O)C=CCCC1 CCC(CC)(CO)C(=O)N1CC(CCNC(c2ccnc3c2CCO3)=O)C1 N1(C(C2CC3CCC2C3)C)CCC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)CC1 C1(NC(CN(C(C)=O)C)=O)CCCC(C(=O)NCCCOCCO)CC1 c1(C(=O)NCCCCC(C)NC(c2ccnc(CO)c2)=O)cn2cnnc2cn1 C1(C(=O)NCCN(CCOC)C(C2CCCC2OC)=O)CCCC(=O)N1C C12(NC(CCc3ccc(C)s3)=O)CC1CN(C(c1cc(CO)oc1C)=O)C2 Cc1noc(C(C)C)c1NC(C12CC(CN1C(C1C3CC(=O)CC13)=O)C2)=O c1(N2CCC(C)C(NC(c3cccc(OC)c3)=O)C2C)ccc([N+](=O)[O-])c(C)n1 C1(CNC(N)=O)CCC(C(=O)NC2C(NC(CCNC(=O)OCC)=O)C2)O1 c1(SCC(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)nc2ccccc2o1 C1(NC(C(C)OCCOC)=O)COCCC1C(=O)NCCc1ocnc1CO C(C(C)(C)CNC(c1nocc1C(C)(C)C)=O)N(C(C(C1CCC1)OC)=O)C C1(NC(C2CC=CCO2)=O)CC2CN(C(c3ccnc(Cl)c3)=O)CC12 C1(NC(c2c(OC)csc2)=O)CC(CNC(c2csc(=N)[nH]2)=O)C1(C)C c1(C(N2CC3C(CC(=O)NCC(C(CC)CC)O)C3C2)=O)cccn2ccnc12 CCCCC(C(=O)NCC1CN(C(=O)COC(C)C)CCO1)C(C)C N1(Cc2n(C)c3c(n2)c(Cl)ccc3)CCc2c(Cl)c(Br)cc(F)c2C1 N1(C(C(OC)OC)=O)CCCC1CCNC(c1nonc1C(C)C)=O C(=O)(C1=NOC2COCC12)NC1CCCC(CC(=O)NC(C)(C)CCCF)C1 C1(NS(CC)(=O)=O)CCCC(C(=O)NC(=O)C(N2CCC(C)CC2)=O)C1 CCCCC(C(=O)NC(CNC(=O)CC(=O)N(C)C)CC)C(C)C C1(C)(CC)COCCN1CC(=O)Nc1cn(C)nc1-c1cnccn1 c1(C(N2CCC(N3CCCC3)C2)C(=O)NC)cccc(C(N)=O)c1.C1CC1 C1(NC(C2CC(=C)C2)=O)CCCC2CN(C(C34CC(CO)(C3)C4)=O)CC12 Cn1cc(C=CC(=O)NC2(C(=O)NCCC(N)=O)CSC2)cn1 N1(C(C=Cc2nc(C)sc2)=O)CC(NC(=O)C(n2nccc2C)C)C2CCCC12 C1(C(N(C)CCOCCNC(C2(COCC)CC2)=O)=O)CC2CCC2C1 Cc1ncc2n1CC(C(=O)N(C)CCNC(=O)C(C1(O)CCOCC1)(F)F)CC2 CCCC(CC)CCC(=O)NC(c1nocc1C(=O)NCCCN1CCC1)C N(C(=NCC=C1CCOCC1)N1CCCC(n2ccnn2)C1)CC(=C)C C=Cn1nccc1C(N1CCCC1(CNC(=O)C(N)=O)COC)=O c1(CNC(=NC)NCc2csc(C)n2)sccc1S(C)(=O)=O N1(C(C=C(C)C)=O)CCC(c2cccc(F)c2)(NC(=O)C(=C2CCCCC2)F)C1 c1(CCN=C(NCCC(=O)N(C)C)NC2CCCC2)cc2ccccc2o1 C(=O)(CC(C)CCC)NC12CC(C(=O)NC(CCC)CCO)(C1)C2 N1(C(CCCCCC(C)O)=O)CCC2CCN(C(=O)CC3CCC3)CC12 O=C(C1=COCC1)NC1CCCC(NC(c2cc(C3CCOCC3)[nH]n2)=O)C1 NC(=O)CC(O)C(=O)NC1CN(C(=O)Cc2cccc(OCCN(C)C)c2)C1 CC1CN(C(=O)C(C)(C)c2ncco2)CC1CNC(=O)CN1CCOCC1=O c1(C(CC(=O)NC(CS(C)(=O)=O)c2ccccc2)(C)C)c[nH]c2c(Br)cccc12 c1(C(N2C(C(N3CC(C(CC)C)C3)=O)CC(F)CC2)=O)cc2ccccn2c1 c1(C(N(CC(C)NC(=O)CC2CCCCCCC2)C)=O)ccccc1S(C)(=O)=O c1(CC(N2C(CNC(C(F)=CCC)=O)CC(OC)C2)=O)ccc(C)nc1Cl C=CC1(CC(=O)NCCN(C(C2C3CCCCC23)=O)CC)CCCCC1 Nc1cc(F)c(C(N2CC(C3(NC(c4cccnn4)=O)CC3)C2)=O)cc1F C1(NC(C(C)(C)NC(Cc2c(C)n(C)cn2)=O)=O)CCCCCC1(C)C c1(N(C)C)ccccc1NC(=O)COC1CC(NC(=O)Cc2ccc(O)nc2)C1 C12(CCC(C)(C)C1)C(=O)N2.c1(CNC(CSCC)=O)nnc(C)o1 C1(n2cnnn2)(CC(=O)NC2C(NC(CC(=O)OC)=O)C2)CCOCC1 C1(CCNC(CC2N(C)CCC2)=O)COCCN1C(c1ccccc1CC#N)=O c1(C(=O)NCC(CCOC)NC(CCC(=O)NCCC)=O)cc(Cl)c(F)cc1Cl N1(C(c2cc(C)sn2)=O)CCC(NC(=O)CC2(C)CCCCCC2)CC1C c1(C(=O)NCC2(O)CCN(C(C3N(C)CCC3)=O)C2)cn(C)c2c(Cl)cccc12 Cc1ccc(C(=O)NC(C2CCN(C(=O)CCOC3CCC3)CC2)C)cc1F CC1CC=CCC1C(N1CCOC(CNC(=O)C=C2CCC2)C1)=O C1(NC(c2c(C)snn2)=O)CCN(C(c2nnc(S)n2C)=O)CCC1(F)F N1(C(C)C)CCOC(C(=O)NC2CCC(NC(=O)Cc3cccc(O)c3)CC2)C1 C(C(C)C(=O)NC1CCN(C(C2(N(C)C(=O)OC(C)(C)C)CCC2)=O)C1)OCC C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)NCCN(C(c1cnnc(O)c1)=O)CC C1(C(=O)NCC2(F)CN(C(CCSc3n(C)ccn3)=O)C2)CCCC2CCCN12 C1(CNC(c2cnon2)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 c1(CC=C)cccc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1 c1(CNC(C(=O)N(CC)C)=O)cc2c(s1)CCC2.C12CCCCN1C2=O CCCC(C(=O)NC(C)(C)CCCNC(=O)COc1cccc(Cl)c1Cl)C(C)C c1(CC)c(C(=O)NC2CCCC(NC(=O)CCn3nc(C)nc3C)C2)nnn1C c1(C(=O)NCCOCCC(=O)NCCc2ccc(F)nc2)c[nH]c(=S)cn1 CCC(CCCC(=O)NC1CC2(CCCC2)C1)NC(C1(C)CC(F)C1)=O C1(C(N2CC(C3(NC(CCC(=C)Br)=O)CC3)C2)=O)CCc2nncn2C1 O=C(C1=COCC1)NCCN(C1CCCCC1)C(C1CCC(F)C1)=O c1(NC)ccc(C(N2CC=CC2(C)C(=O)NC(C)Cc2ccncc2)=O)nc1 c1(C(=O)NC(CC)CNC(C2CCC(N(C)C)CC2)=O)ccc2oc(C)nc2c1 N1(C(C(C)C2CCCO2)=O)CCC(C2(O)CN(C(=O)C3=CCCCC3)C2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)ccc2c(O)n[nH]c2c1 N1(C(CC2CN(C(CC3(NC(C)=O)CC3)=O)C(C)C2)=O)CCCCC(F)(F)C1 C1(NC(C(C)=C2CCCC2)=O)CC=C(C(=O)N2CCCC(CO)CC2)C1 C1(C(=O)NCCC(C)NC(c2csnc2Cl)=O)CC2CC1CO2 N1(C(C2(OC)CC2)=O)CC2CC1CC2NC(=O)CCc1cccc(C(F)F)c1 Cc1ccn2cc(C(=O)NCCCCNC(c3cc4sccc4[nH]3)=O)nc2c1C N1(C(C=C2CCC(C)C2)=O)CC2(C)CN(C(C3CCC(C)C3)=O)CC2(C)C1 CC(C)CC(CC(=O)NCC1OCCC1(C)C)NC(c1c[nH]c2cnccc12)=O C(=O)(C1CCc2cccc(F)c21)NCC(C)(O)CNC(c1cncc(N)n1)=O c1(C(=O)NCC2=CCN(C(C(C(C)C)C)=O)CC2)c(F)ccc2ccncc12 C(N=c1[nH]cc2ccnc-2[nH]1)C1(C)CCN(C(c2cc(C(C)C)on2)=O)CC1 c1(N2CCC(C)(C(F)(F)F)CC2)nc(N2CC3CCC3(N)C2)nc2ccccc12 c1(C(=O)NC(C)CNC(=O)Cn2ccc(O)nc2=O)c(F)cccc1[N+](=O)[O-] C1(NC(c2c(C)nn(CC)c2Cl)=O)CCC2CC1CN2C(=O)C1=NNC(=O)C1 C(=O)(C1CCCc2cncn21)N(CCCN(C(C1N(C(C)=O)CCOC1)=O)C)C c1(C(=O)NC2(C3CN(C(C4(COC)CC4(F)F)=O)C3)CC2)nccn2nc(C)cc12 N1(C(C2CCCN(CC)C2)=O)CCC(C(=O)NCCCSC)(OC)CC1 N1(c2cc(NCC(C)CC(C)O)nc(COC)n2)CCc2sc(Br)cc2C1 c1(CC(C)(C)C)cc(=NC(=O)N(C2CCC2)CC2CC2)[nH]o1 O=C(C1=CCCN(C(c2ccc(F)cc2F)=O)C1)Nc1cc(Cl)c(F)c(Cl)c1 c1(C(=O)NC2CCCCC2NC(C2CCC(F)(F)CC2)=O)cc2scnc2[nH]1 C1(C(=O)NCC(O)C(F)F)(CC)CCCN1C(c1csc(CO)n1)=O Cn1cnc2[nH]c(=NCC3(C)CCOCC3)[nH]c(=NC3CCCN(CCO)C3)c12 N1(C(CC2(OC)CCC2)=O)CCC2(CC1)CN(C(=O)C(C)(C)c1csc(C)n1)C2 CC1(F)CCC(C(N2CCCC(C)(NC(c3cnn[nH]3)=O)C2)=O)CC1 c1(C(c2nnnn2CCCF)NCC2(CC)COC2)ccnc(Cl)c1 C#CCC(C)(CC)C(=O)N(C)CC1CCCN1C(=O)C(C)=CCC Cc1cccc(C=CC(=O)N(CCN(C(=O)C=Cc2cnccn2)C)C(C)C)c1 C1(NC(=O)NC(CC(C)C)Cc2ccccc2)N(C(C)(C)C)CCOC1(C)C N1(C(C(C)S)=O)C(C(=O)NC2COCCC2O)CC2CCCCC12 c1(C(N2CC(c3ccccc3)(NC(C3CCCCO3)=O)C2)=O)cn2ccsc2n1 N1(C(C(C=C)OC)=O)CC2CC2(CNC(C2(C)COC2)=O)C1 c1(C(=O)NCC(CNC(c2ccn(C)c2)=O)(C)O)cc(C2CCCCC2)n(C)n1 C1(NC(c2c(C)noc2C)=O)CCN(C(c2c(OC(C)C)ccs2)=O)CC1F C1(C(=O)NC23CC(NC(C=CCOC)=O)(C2)C3)CC=CCC1C(=O)O C(=O)(CC(CC)C(C)C)N1CCC(C(=O)Nc2cnc(CCC)nc2)C1C N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC(CNC(C23CCC(C2)C3)=O)C(C)(C)C1 CC(C)C(C#N)C(=O)N(C)CC1CCCN1C(=O)C(C)C=Cc1ccccc1 C(=O)(C1=CC2CCCCCCC12)NCCC1(NC(COCCCC)=O)CC1 c1(C(=O)NCC(CCC)NC(=O)CNC(=O)OC(C)(C)C)cncnc1C c1(COC)ncc(CNC(=O)CNC(C2(C#N)CC2)=O)[nH]1 Cc1c(NCCCSc2ccc(Cl)cc2)nc[nH]c1=NCc1cocn1 C(=O)(CCCCCn1cnnn1)NC1CN(C(c2cc(CCC)c(C)s2)=O)C1 c1(SC)cc(F)ccc1C(=O)NCC1CCCC(NC(C2(O)CCSCC2)=O)C1 Cc1csc(=NCC(=O)N2CCCC(C)(NC(C3CCCCC34CC4)=O)C2)[nH]1 C1(CC(=O)N(C(CNC(C2(C#N)CC2)=O)C2CC2)C)CC2(CCC2)C1 c1(CC2CC(C(N(CC(CN(C)C)O)C)=O)C2)nnc(O)n1C C12CCN(CC1)C(=O)C1CC1c1nc(no1)C2.NC1(C2CCCO2)CCC1 N1(C(c2n(COC)ncc2)=O)CCC(CC(C)NC(C2(C3CC3)CC2)=O)CC1 CCC(F)C(=O)NCCC(C)(C)NC(c1ccc(CC(C)C)s1)=O CN1CCC(C(N2CCC(NC(c3csc([N+](=O)[O-])c3)=O)CC2)=O)CC1=O c1(C(=O)NC2C3CN(C(C4C(COC)C4)=O)C2C3)c[nH]c2cc(Cl)ccc12 N1(C(c2ccc(OC)nn2)=O)CC(N(C(=O)CC2CC=CC2)C)C2(CC2)C1 C1(CCC#N)CC=CC(NC2(C3CC=CCC3)CC2)C1 C(CCS(=O)(=O)C(C)C)N(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)C C(=O)(C1OCCc2ccc(C)cc21)N(CCC)CCNC(=O)CCC1CC1C Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CC(N(C(=O)CC(O)C(C)C)C)C1 CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC1[N+](=O)[O-])C1CCC1 CC1CN(C)CCC1N(C)C(C1CCC(NC(c2ccnc(O)c2)=O)CC1)=O C(CN=c1ccc2c([nH]1)CCCC2=O)N(C(C1CCCC12CCC2)=O)CC C1(C2CC2)(NC(c2cccc(F)c2)=O)CCN(C(=O)CSCc2ccccc2)C1 c1(C(=O)OCC)ccc(OC)c(S(=O)(=O)N2CCN(C)C(CO)C2)c1 N1(c2c(C(=O)Nc3cc([N+](=O)[O-])ccn3)cccn2)CCc2cccnc2C1 C12(NC(CCC=CC)=O)CCCCC1CN(C(=O)CC(C)CC(=O)OC)C2 C1(NC(=O)CCN(C(c2ncoc2C(F)F)=O)CC2CC2)CC2CC2C1 c1(NC(c2n(CC(=C)C)nnn2)c2c[nH]nc2-c2cccs2)ccc(O)cc1C C1(NC(C(C)OCC#C)=O)CC2CC1CN(C(=O)C(C)SC(C)C)C2 c1(CC)n[nH]c(=NC2C(C)CN(C(=O)C3=C(C)OCC3)CC2C)s1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 CC(=O)CCCCC(=O)N1CC(OCC(=O)NCc2c(C)cccc2F)C1 c1(CC(=O)N(CCOC)CCNC(=O)C=C(C)I)nnccc1C Cc1cccc2c1CC(C(=O)NCC(O)CNC(c1ccc(CO)o1)=O)O2 N1(C(C(CCNC(Cn2nc(C)oc2=O)=O)O)=O)CCC2(CC1)CSC2 C#Cc1cccc(CNC(=O)C(C)CN(C(=O)Cc2csc(C)c2)C)c1 N1(C(CCCC=C)=O)CC(CCNC(c2cnn(C(C)C)n2)=O)OC(C)C1 C1(NC(CCCC)=O)CN(C(c2cc(C)n(CC3CCCO3)n2)=O)CCC1CO C#CCC(CC(=O)NCC(C)(O)CO)NC(=O)CS(C)(=O)=O C(=O)(C(C(C)(C)C)NC(C1C2COCC12)=O)NCc1ccc(OC)nc1 CCC(C)C(C(=O)N(C)Cc1ncco1)NC(C1COCOC1)=O CC1(C)COCC1C(=O)NC(c1cccnc1)C(=O)NCc1ccccc1F C1(NC(C(CCN(C)C)NC(=O)CC2CCC(=O)CC2)=O)CN(C)C(C)(C)C1 C(CC(O)C(=O)NCC=C1CCN(C(C2CCOC2=O)=O)CC1)SC N1(C(C2CNC(=O)N2)=O)CCC2(CCCC(CNC(C3(CF)CC3)=O)O2)CC1 C1(COC)CCCN1C(=O)CC(C)NC(c1cccs1)=O N1(C(COCC=C)=O)CCC(C)(NC(=O)CC2CCCCCC2)C1 c1(C(N2CCC(N(CCC)C(C3CCCC3OC)=O)C2)=O)cc(C)nc(OC)n1 c1(CC(=O)NC2CC(NC(C3(O)CCC3)=O)C(O)C2)cc2nc[nH]c2cc1Br c1(OC)ccc(C(=O)N(C2CCN(C(=O)C=CC(F)(F)F)C2)C)cc1[N+](=O)[O-] Cc1cn2cc(C(N3CCCC3CCCNC(C3CCCN(C)C3)=O)=O)nc2s1 C1(CC=C)(NC(=O)C=CC2CCCC2)CCN(C(C2CC2C(C)O)=O)C1 CCS(=O)(=O)CC(=O)N1C(C(=O)NC(CCO)C(C)C)CC2CC12 c1(OCC(=O)NCC2CCCC(NC(CC3(OC)CC3)=O)C2)cc(C)ccc1O C(=O)(CCC=O)NCC.C12(OCC)CN(C1)C(=O)c1ncoc1CNC2.NC c1(SCC)ccccc1C(=O)NC1CC1CNC(=O)CC1CCCC(=O)N1 CCCS(=O)(=O)CC(=O)N1CC(NC(=O)CCOc2ccc(Cl)cc2)CC1(C)C c1(SCC)cnccc1C(=O)N(CC(C)NC(=O)CCC1CCCCN1C)C CC(C)CCC(O)C(=O)N(C)CC1CCCN1C(c1cccc(C(C)(C)C)c1)=O N1(C(C(c2ccc(C)o2)C)=O)CCC2C(C1)CN2C(c1cn(C(C)C)nc1C)=O C(=O)(C(CO)C(C)(C)C)N1CCN(C(c2n(CC)ncc2)=O)C(C)C1 N1(C(C(c2n(C)ncc2)NC(=O)CCn2cnnn2)=O)CCCC2(CC2)C1 c1(-c2cn(C(CCC(=C)C)C(=O)OC(C)(C)C)nn2)cnc2cccnn12 c1(C(=O)NCC2CCN(C(C(CC)(C)F)=O)C2)ccc2c(c1)OCO2 c1(N(C)Cc2cnc(CC)s2)nc(N2CCCC3(CCCO3)C2)c2c(n1)CSC2 C1(C(=O)NC2CC(C(F)F)(NC(C3CCCO3)=O)C2)CCC2CC1CO2 N1(C(c2c(SC)cccn2)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 C(=O)(C(C)C(C)(C)C)N1C(CCNC(c2c(C)cn(C)c2)=O)COCC1 C1(CC(=O)N(CCN(C(=O)C(c2cnn(C)c2)C)CC)CC)CCC(=O)N1 c1(C(C)NCCS(CC(C)C)(=O)=O)ccc2c(c1)COC2(C)C O=C(C1=C(Cl)CCOC1)NC1CCCC1 C(=O)(CCCCC(F)(F)F)N(C1C2CN(C(c3cnc(N(C)C)nc3)=O)CC21)C N1(C(C2(CC#C)CCN(C(=O)Cc3cncc(C)c3)C2)=O)CCC(C)C(O)C1 C1(C(N2CCC(C)(N(C)C)C2)=O)CCc2ccnn2C1 C1(NC(COCCCCC)=O)CC2CC(C1)N(C(C1CCCC3(CC3)C1)=O)C2 CN=c1nc(C(N2CCOC(CNC(c3cnc(SC)s3)=O)C2)=O)cc(C)[nH]1 C12(C(=O)NCCC3(NC(=O)CSc4nc[nH]n4)CCC3)CCCCC1C2 S(=O)(=O)(CCC(=O)N1CCCC(N(C)C(c2sc(CO)nc2C)=O)C1)NC N#CC1CN(C(c2cc(O)nc(Cl)c2)=O)CCN1C(=O)CCc1ccoc1 C1(CNC(N(C)Cc2cccc(-n3cccn3)c2)=O)CCC(C)c2ccccc2C1 S(=O)(=O)(c1cccc(SCC)c1)NC(N1C(CCC)C(=O)NCCC1)=O N1(C(C(C(C)C)C2CCC2)=O)CCC2(CCC(NC(=O)CC3CCCC3)C2)C1 N1(C(CCC#CC)=O)CCCN(C(=O)C(c2ccc(C#N)cc2)O)CC1C CC(C)CC(C)CC(=O)N1CCCC(C)C1CNC(=O)CC1(C)CCCCC1 C1(NC(c2cccn2C2CC2)=O)CC2CC1N(C(C1CCC1)=O)C2 N1(C(CCCOCC)=O)CCN(C(c2cnc(OC)nc2)=O)C(CC)C1 Cc1cn2ccc(C(N3CC4CC(NC(=O)C(C)(O)C5CC5)CC3C4)=O)cc2n1 C1(COC)(NC(=O)CCc2nncs2)CCN(C(c2nccnc2C(N)=O)=O)C1 Cc1cc(C)n(CCCC(=O)NC2(C)CN(C(=O)C(C)c3ccon3)C2)n1 N1(CCCCOCCCN)CCN(C(c2cccc(Cl)c2)=O)CC1 c1(NC2(c3n(CCSC)nnn3)CCC2)cc2n(n1)CC(O)CO2 CCCC(C)CCCC(=O)NC1CCC(NC(c2c(C)nsc2N)=O)C1 c1(N(C)CC2CCCO2)nc2ccsc2c(=NC2CCCSCC2)[nH]1 Cc1ccc(C(=O)NC2CC(NC(=O)C(CC(C)C)c3ccccc3)C2)c(O)n1 c1(OC)ccc(OCC(F)F)c(NC(=O)C(=O)NCCCN(C)C(C)=O)c1 C12(CNC(c3cc(C)n(C(F)F)n3)=O)CCCC1CCN2C(=O)C=CCF c1(CCN(C)CCO)cn(CCCN(C)C(C2(F)CCCC2)=O)nn1 CC1OCCOC1C(=O)NC(C(=O)N(C(C)C(F)F)C)c1ccco1 C1(C(=O)NC(C23CCC(CO2)C3)C)CCOc2ccccc2O1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(c1ccnc(C(F)F)c1)=O N1(C(C(C)C2CC2)C(=O)NC(C)(C)C)CCCC(c2nncn2C)C1 Cc1cccn2nc(C(=O)NCCC3CC3C)cc12 C1(CC=C)(C(N2CCC(C(C)NC(c3ncsc3NCC)=O)C2)=O)CCCC1 CCC(C(=O)NCC(C1CCCCC1)NC(=O)CNc1nccs1)NC(C)=O CC1CN(C(c2cnc(C3CC3)[nH]2)C(=O)NCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(=O)CC2CCCCC2F)(CO)CCN(C(=O)CCOC2CC2)CC1 C(C(C)C)(C(O)C(=O)NCCC(C)NC(C1(C)CCN(C)C1=O)=O)OC C1(CC=C)(C(=O)N(CCC2CC2)CC)CCN(C(=O)Cc2ncccc2C)C1 C1(C(=O)NC2CN(C(COCC)=O)CC(C)C2)COc2ccccc2O1 CCCCC(CC(=O)NCCCO)NC(=O)C(C)(O)C(C)C c1(C(=O)NC2(C3N(C(CCN(c4ccncc4)C)=O)CCC3)CC2)ccc(F)cn1 c1(C(=O)NCC(CC=C)NC(C2CCS2(=O)=O)=O)cc(C(F)(F)F)cn1C N1(C(C(C)n2ccnc2)=O)CCSCC1C(=O)NCC(O)(CO)CO CN1CC2CN(C(c3c(Br)cc(Br)c(O)c3Br)=O)CCN2C1=O c1(N2CC(O)(C(C)NC(=O)CC3CCC(O)C3)C2)nc2c(cc1C#N)CCOC2 C1(C(N2CCCCC(NC(=O)COC3CCOC3)C2)=O)CCCC12CCOCC2 C1(C(=O)NCC(CNC(c2c(CCC)n[nH]c2)=O)F)CCCCN1S(N)(=O)=O C1(C(N2CC(OCC)C(CNC(=O)CC3(CO)CC3)C2)=O)CC(C(C)C)=NO1 CC1(CNC(c2csc(-c3ccsc3)n2)=O)CCCN1C(C1CC1F)=O CC(C)(O)CC(=O)N1CCC(C)(NC(c2cc(-c3ccccc3)ccn2)=O)C1 N1(C(CCN(CCCO)C(c2nc(CC)sc2)=O)=O)CCN2C(=O)OCC2C1 c1(C(c2n(CC(=C)C)nc(C3CCCO3)n2)C)ccc(F)c(F)c1 C1(C(=O)NC(CC=C)CNC(c2cccc(F)c2Cl)=O)CCc2nc[nH]c2C1 C1(C)(OC)CC2CC1CC2NC(=NCCSc1ccc(Cl)cc1)NC(C)CF C1(NC(C(CC)(F)F)=O)CN(C(C2(C3CCCCO3)CCC2)=O)CC2(CC2)C1 N1(C(C)C(=O)NC2(CN(C)C)CN(C(=O)CC(Cl)Cl)C2)CCC(O)CC1 N1(C(C(C)(Cl)Cl)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C(F)(F)C1 Cc1ccnc(C)c1CNC(=O)C1=CCC(NC(C2CCNC(=O)C2)=O)C1 c1(C(=O)NC2CC(NC(c3c(C)cc(C)o3)=O)C2)cc(Cl)ccc1-n1cccc1 C1(C)(C(N2CC(C(NOC)=O)C2)=O)CC(O)CN1C(=O)C(F)(F)F c1(N(C)C)ccc2c(-c3ccc(CN4CC(C(=O)O)C5(CNC5)C4)cc3)coc2c1 C1(C(=O)NC2(CO)CN(C(CS(C)(=O)=O)=O)C2)CC2CCC1CC2(F)F C(=O)(C(C)(C)C(F)F)NCCOC.N12CCC(CC1)OCCN1CCC(C1)C2=O C(C(C)(C)CNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)CCSC(F)(F)F C1(NC(CC=CC=C)=O)CC1C1CCCN(C(c2c(C)noc2C2CC2)=O)C1 N1(C(C(CC)O)=O)CCC(C)(CNC(=O)C(C)(C)OC(C)=O)CC1 C1(CCO)(NC(CNC(CCC)=O)=O)CN(C(=O)C(CC)n2cncn2)C1 Cc1c(NC(=O)C(=O)NC2CN(C(=O)CC3(C)CC3)C3CC23)cccc1F O=C(C1Cc2c(Cl)cccc21)NC1(CNC(C2Cc3nccn3C2)=O)CCC1 N1(C(C(CC#C)(C)C)=O)CC=C(CC(=O)NCC2(n3ccnn3)CC2)CC1 C=C(Cl)C(C)(C)C(=O)N1CC(N(C)C)C(O)C1.C12(CCN(C)CC1)CC(=O)N2 CC(CC1CC1)N=c1ccnc(NC2(c3cc(F)ccc3F)CC2)[nH]1 C1(C(=O)NC(C)CNC(c2ccccc2Cl)=O)CCCCC(=O)C1 C1(CC(=O)NCCCNC(C(C)CSC(F)(F)F)=O)CCC2CC1C2(C)C N1(C(CC=C)=O)CC2(COC(CNC(c3c(C4CC4)cccc3F)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)NC1C(C(=O)NC(C(=O)OC)C)CCC1 C1(CN(C(=O)Cc2cnc[nH]2)C)CSCCN1C(C1CC(N2CCOCC2)C1)=O C1(C(N2CC(CNC(=O)CC3CSCCS3)C2)=O)OCC2CCCCC12 N1(Cc2cccc(OC(C(=O)OC)C)c2)CCC(Cc2nnc(SC)o2)C(C)C1 CCCCC(C)C(=O)NCC=C1CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C1(C(=O)NC2CCC(CNC(C(C)C)=O)C2)CC2CCCCCCC12 N1(C(C(C)NC(CN(C(C)(C)C)C(C)=O)=O)=O)CCCC1(C)CCC(N)=O CC1(C)Nc2ccccc2C1NC(C1CCC(C)(CN)CC1)=O N1(CC(=O)NCC2C(OC)(OC)CC2)CCCC(C)(c2ccccc2)C1 C1(C#N)(C(=O)NCC2N(C(CCCSC)=O)CCC2)CC12CCC2 C1(c2cn(CC(C3CN(C(C(CC)n4cncn4)=O)C3)F)nn2)CCC(C)CC1 c1(SC(C)(C)C)cc(C(=O)NCc2cc(C(F)(F)F)co2)cs1 C(=O)(C#CC1(C)CC1)NCCCCC1(NC(CC(CC)SC)=O)CC1 Cc1cc(F)ncc1-c1cn(CC(C)NC2CCN2C)nn1 c1(CN2C(C(=O)Nc3cccc(CCC)n3)CSCC2)c(Cl)cncc1Cl N1(C(C(CC#C)(C)CC)=O)CCCCC2(CCN(C(C34CCC(CC3)C4)=O)C2)C1 C(C1=CCN(C(=O)Cn2cc(CO)nn2)CC1)NC(C=COOCC)=O C1(C)(C(=O)NCC(C=C)(C)C)CC(O)CN1C(c1cn(C)cn1)=O c1(C(=O)NC2CCCN(C(C(CC)OC3CCCC3)=O)C2)ccn2ccccc12 c1(C(N2CC(O)(C(C)NC(c3csc(CO)n3)=O)C2)=O)cc2ccccc2nn1 N1(C(c2cn(CCCC)nn2)=O)CCC(O)C(NC(c2csc(Cl)n2)=O)C1 n1(C(CC)C)ncc2c(C(=O)NOC(c3ccccc3C)C)cc(C)nc12 C1(C(C)N)CCCN(C(=O)C(=O)NC2CCC(n3ccnn3)C2)C1 c1(C(N(CC(F)(F)F)CC)=O)ccncc1C1=CCC(C(F)(F)F)CC1 C(=O)(CCC(C(=O)OCC)NC(c1n[nH]c(-c2cc(Cl)ccc2Cl)n1)=O)OC Cc1cccc(CC(N2CCC(NC(=O)CCC(F)F)C2C)=O)c1 n1(Cc2ccc(C(=O)NC3CNCC34CCC4)cc2)cnc2cccnc12 C1(C(=O)NC(C=CC(=O)NC(COC)C)(C)C)CCC(C)O1 c1(C(=O)NCC2N(C(C3(CC=C)CCC3)=O)CCCC2)nc(C)n(C)c1C c1(OC)ccc(C(N2CCN(C(c3cccc(Cl)c3OC)=O)C(C)C2)=O)c(F)c1 C#CCC(C)(C(=O)N1CCC(OCCF)C1)NC(C1CC2CCCC2C1)=O N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(C)(C)CC1CNC(C1CC(CC2CC2)C1)=O c1(C(=O)NCC2CC(NC(c3n(CC=C)ccc3)=O)C2)c(C)nc2ccccn12 C1(C)(N(CCCCC(=O)OC)C(=O)N)CCCCCC1.c1(-c2ccccc2)ccc(N2CCCC2)nc1 c1(CNC2CCC(CC(=O)Nc3cn(CC)nc3C)CC2)ccc(Cl)nc1Cl c1(OC)ccc2c(c1)CC(C(=O)NC(C)(C)CN(C(=O)Cn1cccn1)C)O2 Cc1oc(-c2cnn(C)c2)nc1C(=O)NC(C)C(C)F c1(Nc2c(-n3c(NC4CC(=C)C4)nnn3)cccc2)c(C(C)=O)ccc(Br)c1F N1(C(c2cnc(S)nc2)=O)CCC(F)(C(=O)N(C2CCOC2)CCO)C1 C1(NC(C2(C)CCCS2)=O)C=CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccn2)cc(C)c2c(c1)CCC2 N1(C(c2c(C(C)C)cco2)=O)CC2CCC2(NC(C2CC2(C)C(F)F)=O)C1 N1(C(c2cn(CCC)nc2)=O)C2CCC1CN(C(c1cn(C(F)F)c(C)n1)=O)C2 c1(C(=O)NC(C)C(C)NC(c2cc(O)ncn2)=O)cccc2c1nnn2C C1(CC)(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)C(C)OC)CC1 N1(C(CC2ON=C(C)C2)=O)CC(C(N2CCC(C3CC3)C2)=O)CC12CCC2 C12CCCCC1NC2=O.C1(C(N)=O)(NC(=O)CCCC2CCCO2)CCCCC1 C1(NC(c2scc(OC)c2)=O)CC(O)CN(C(C23CCC(CO)(CC2)C3)=O)C1 C12(CC(=O)NCC3(O)CCCN(C(=O)CC4CC5CC5C4)C3)CCC(CC1)OC2 c1(C(=O)NC2(C)CCCN(C(CC(C)F)=O)C2)cc2cc(Br)cn2cn1 C1(CNC(CN2CCC(OC)C2)=O)(CO)CCN(C(c2c(C)nsc2N)=O)C1 N1(C(CC(=C)Br)=O)CCOC(CN(C)C(C2CC(=O)N(CC(C)C)C2)=O)C1 N1(C(C(C)=CC=C)=O)CCC2(CC1)CC2C(=O)NC1(CO)CC2CCCC12 C1CN(CCC=C(F)C(=O)NCc2cc(C(N)=O)co2)C2(CCC2)C1.CCC=C C1(CC(N2CC(CN(C)C(c3cc(C(F)F)nn3C)=O)C2)=O)CN2CCC1CC2 CC1(C)COC(C(=O)NCC2CCN2C(=O)COC2CCCCCC2)CO1 n1(CCOC)nnnc1C(c1cncn1C(C)(C)C)NC(C1CCCCC1)C C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)C(C)OCC2CC2)CC1C1CC1 C(=O)(C(O)CCC(C)C)NCC(CN(C(C1CCCCS1(=O)=O)=O)CC)(C)C c1(CNC(C(C)C(C)O)=O)cccc2c1CN(C(C1(F)CC=CC1)=O)C2 c1(C(=O)CN2CCN(C(=O)C3CC3)CC2CC(F)(F)F)ccnc2[nH]ncc12 C1(CNC(c2ncoc2C2CCC2)=O)CN(C(C2CCCO2)=O)CC1O N1(C(C23N(C(c4cc(C)c(O)nn4)=O)CC(C)(C2)C3)=O)CCCC(C)(O)CC1 c1(C2(CNc3nccc(N(C)CC4CCC4)n3)CCC2)ccc(F)cc1F c1(OCC(=O)NCCC(C)N(C)C(C2CC2C)=O)ccc(F)cc1O c1(CN2CCC(CC(=O)NC3CCCN(C)C3)C2)c(F)cc(C(=O)O)cc1F C1(C(C)=O)CC(C(=O)NCC(C)CNC(=O)CC2(CSC)CC2)C1(C)C Cc1cn(C)cc1C(=O)N(C(C(=O)NCc1nccs1)C1CC1)C C(CC(C)C(=O)NC(C)CNC(=O)Cc1ccccc1OC(C)C)OC c1(CNC(C2N(C(C)C)CCC2)=O)cccc(C2CC2)c1Cl N1(C(C=CC=CC)=O)CCCC(C)(NC(c2ccc(Cl)nc2Cl)=O)C1 C1(CC(=O)NCCC(C(C)C)NC(c2ccco2)=O)SC2=NCCN2C1=O C1(CC(=O)NC2CC(CNC(CCc3cn(C)nc3)=O)C2)CCCC(=O)N1 c1(C(N2CCC(O)C(O)CC2)C(=O)NCCCSC)ccc2ccc(Br)cc2n1 c1(C(=O)NC2(CNC(C3CC(C(=O)OC)C3)=O)CCC2)sccc1Cl C1(C2CC2)(NC(CN(C(c2ccc(C)n2C)=O)C)=O)CCCC1 c1(C(=O)NC2CCC(C(=O)NCC3C(=O)OCC3)C2)cccc2nccn12 c1(C(C(=O)N(C2CCN(C(C3C=CC=CC=C3)=O)C2)CCC)C)ccc(F)cc1 C1(NC(CC2(C=C)CN(C(=O)COC)C2)=O)CCc2n[nH]cc2C1 c1(NCC(C)(C2CC2)NC(c2cc(C3CC3)on2)=O)ccc([N+](=O)[O-])cc1C#N C1(C)(CNC(C2N(CCCC)CCOC2)=O)CN(C(c2cnns2)=O)CC1C C1(CC(N2CC(CNC(C3C(=C)CC3)=O)C(C)C2)=O)CCCNC(=O)C1 c1(C(=O)NCC(N(C)C(c2coc(CC3CC3)n2)=O)C2CC2)ccn2ccsc12 N1(C(c2n(C)ncc2C2CC2)=O)CCN(C(c2ccnc(Cl)c2Cl)=O)CC(O)C1 C12CCCN(C1)CC(=O)N(CC1CC1)C2.c1(CC)ccon1 N#Cc1csc(C(=O)NCC(O)CNC(=O)CC2CC(C(F)F)C2)c1 N1(C(C2CC(OC)C2)=O)CC(C)CN(C(=O)C=CC=C(Cl)Cl)C(C)C1 Cc1cc(C(N2CCC(CO)(NC(=O)C=CC(=O)N(C)C)CC2)=O)cc(C)c1O C(N=c1[nH]c2c(c(=NCCC3CC(=O)N(C)C3)[nH]1)CSC2)C1N(CC)CCCC1 C(=O)(C(O)CCCCC)NCC1(F)CC(CNC(C2C(=C)C2)=O)C1 S(=O)(=O)(c1cccc(=NCCCn2ccnn2)[nH]1)NCC(C)(C)F c1(C2C(C(=O)NCC3(N(C)C)CC3)(COC)C2)ccccc1 S(=O)(=O)(c1[nH]c(=NCc2cncs2)ccc1Br)NCC(CC)(CN(C)C)CC C1(C(=O)NC(CSCC)CO)CN(C(C2CC(=O)CC(=O)N2)=O)CCN1C C(=O)(C(C)(C)C1CCN(C(=O)C(C)NC(=O)C(C)(C)C)C1)NCCOCC c1(C(=O)NC(CNC(C(C=C)(C)C)=O)(C)CO)nc(OC(C)C)ccc1Cl C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)(C)CCCC3)=O)C2)CCCC1 c1(NCC(CC)C)ccc(S(=O)(=O)NCC)cc1C#N.C(COC)(C1CC1)N C1(C(=O)OCC)CCC(c2nnnn2C2(C)CC2)(NCc2cnc(OC)s2)CC1 N1(C(=O)NC2(C(=O)O)CCCC(C)C2)CCC2(C1)CC2(F)F C(=O)(C1Cc2c(Cl)cccc21)NCC(C)NC(C(CC(=O)OC)(C)C)=O C1(C(C)C)CCCCC1N(C(C1CCCSC1)C(=O)NCc1cccc(Cl)c1)C CC1C(C(=O)NC2(CCF)CCC2)CCN1C(=O)Cc1ccsn1 N1(C(C(F)=CCC)=O)CCC(C2CC2)C1CNC(C1CCCCCC1)=O N1(C(=O)CC2CCCCCC2)CC2(CO)CC1(C(=O)NCc1cn(CCO)nn1)C2 C(CCCCC(=O)N1CCC(C(=O)NCc2ccc(C)nc2O)C1)OCC C1(C(C)NC(=O)CCc2nc(C3CC3)no2)CCC(c2ccccc2)CC1 C(=O)(CC(C)(C)CC(=O)NCCC(O)CNC(=O)CCC1CC(C)C1)OC CC(C)(CC(=O)N1CC2(CCN(C(=O)CC3CCC(=O)NC3)C2)C1)CC(F)(F)F N1(C(CC(C)F)=O)CC2(CO)CC1(C(=O)NCC(C)OCCO)C2 CON1CC(C(=O)NC(CC(=O)NC2(C(O)CO)CC2)C2CC2)CC1=O C1(CC(=O)NC2(COC)CC2)CN(C(=O)Cc2ccon2)CC12CC2 C(=O)(C(CCC(C)C)N1CCOCC1)NCC(CC)C#N C(=O)(C(F)(CNC(C1CNC(=O)N1)=O)C(C)C)N1CCC(C(CC)C)CC1 CC(C)C(CNC(=O)CN(C1CC(C#N)C1)C(C1CCC1)=O)C(C)C C1(C(=O)NCCCN(C(=O)C2=CCC(C)CC2)CCC)OCC2CCCCC12 c1(NC(C)=O)cnc(C)c(C(N2CCC(NC(=O)CC3(C)CC3(F)Cl)CC2)=O)c1 N1(C(CC2C(OC)CC2)=O)CCN(CCCNC(C2CCCN2C2CC2)=O)CC1 N1(C(C(COC)OC)=O)CCC(COC)(NC(C2Cc3nccn3C2)=O)CC1 c1(CC(=O)N)cc(Cl)ccc1C(=O)NC.N1(C(C2C(SCC)C2)=O)CCCC1CC c1(C(c2n(CC=C)nnn2)NCc2ccc(C3CCC3)cc2)ccc(I)c(C)c1 CC1(C)C(CNC(c2ccnc(F)c2)=O)CCN1C(c1ncc(Cl)cc1Cl)=O c1(C(=O)NCC(C(C)(C)C)NC(CCC=C=C)=O)nn2cccnc2c1Cl c1(C(=O)NCC=C2CCN(C(c3cc[nH]c3)=O)CC2)cc2c(Cl)cccc2s1 C(C)(CO)(C(=O)NCC1(CNC(=O)CCc2ccccc2C)CCC1)OC N1(C(C2C(C)CCO2)=O)CC2CN(C(c3occc3Br)=O)CC2C1 C1(NC(c2cn(CC=C)nn2)=O)CC(O)CN(C(=O)CCC=CC)C1 N1(C(C(F)=CCC)=O)CCC(C(C)CNC(=O)CCC23CCC(CC2)C3)CC1 C1(C(=O)NCC2(CCCNC(c3c(C)csc3)=O)CCCC2)CC2COCC2C1 N1(C(C2(C#N)CCCC2)=O)CC2CCC(CNC(C3C=CCCC3)=O)(C2)C1 O=C(NNc1cc(F)c(Br)cc1Cl)c1ccccc1S(=O)(=O)NC1CCCC1 c1(C(=O)NC2C(NC(COc3cccc(C)c3)=O)C2)cnc(Cl)c(N)c1 C1(CC(=O)NC(c2cnc[nH]2)C)COCCN1C(c1cncc(C(F)(F)F)c1)=O N1(C(CNC(C(C)N(C)C)=O)=O)CCOC(C#N)C1.N12CCC(C1)OCC2=O N1(C(C2(CC(C)C)COC2)=O)CCC(CO)(NC(c2cc(C(C)C)on2)=O)CC1 N1(C(CNS(CC)(=O)=O)=O)CC2CC(NC(=O)CCCCC(=O)NC)CC2C1 c1(C(N(CC)CC2CCCN2c2ncncc2OC)=O)cncc(OC)n1 C(C(C)CC(=O)Nn1cnc2ccccc12)NC(CCCCCNC(C)=O)=O c1(OC)ccc(CCC(N2CCC(CN(C)C(C3(C(F)F)CC3)=O)CC2)=O)cn1 c1(COC)nc(C)c(C(N2CCCC2C(C)NC(C2(O)CC2(C)C)=O)=O)s1 O=C1NC(=O)C2(CCCC23CN(C(c2cccc(-n4cnnc4O)c2)=O)C3)N1 c1(OC)ccc(Nc2ccc(Cl)nc2)cc1F.C12CC(C1)NC2=O C(=O)(C(C)(C)C(=O)NC)N1CCC(c2c(CNC(C(C)SCC)=O)c[nH]n2)C1 c1(C(N(C2CCCN(C(CC(CC)O)=O)C2)C)=O)cc(Br)c(C)cn1 c1(C(=O)NCCCCC(C)NC(C2(CC)CCOC2)=O)ccc2c(n1)CCC2=O N1(C(c2c(CC)c[nH]c2)=O)CCC2CCCC12C(=O)NC1(C)CC(O)C1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2C)C(C)C1 c1(C(N(C)CC2N(C(C(C)=CC)=O)CCOC2)=O)cc(O)nc(C2CC2)n1 c1(NC(C(c2c(C)cccn2)N2CCSCC2CCO)=O)ccc(Cl)cc1F CC1CN2CCN1C(C(=O)NCCC1CC(NC(=O)CC(C)(F)F)C1)C2 C1(F)(C(N2CC(C(C)NC(C(CC)C)=O)C2)=O)CC=CCC1 O=C(C(O)C(F)(F)F)N1CC2C(C(N3CC(O)C(O)C3CO)=O)C2C1 C(=O)(C1(O)CCCc2ccccc21)NCC(Cc1c(C)c(Br)ccc1)CO C1(NC(CN2CCC(n3c(C)n[nH]c3=N)CC2)=O)CC2(CC(=O)N2)C1 c1(OC)cc(Cl)c(Cl)cc1NC(=O)C(=O)NC(C1CCCOC1)CCO c1(N2CCC(CC)C2)nc(N2CCn3nc(C(C)(C)C)cc3C2)nc2c1COCC2 C(c1ccc(Cl)cc1)=CC(=O)NCC1C=CC(NC(C(C)c2ccon2)=O)C1 C(=O)(C(O)CCC(C)C)N1CC(C#C)(C(=O)NCc2nc(CO)n[nH]2)C1 c1(C(=O)NCC(CCC)C(=O)NCC(F)Br)ccc2n[nH]cc2c1 Cc1cccc(C2CCCN2C(=O)C(=O)NCc2cnc(C3CCC3)s2)c1C C(=O)(C(F)C(C)(C)O)N1CC(C(C(=O)N(CCC(N)=O)CC)OC)C1 C1(CCNC(C2CCCOCC2)=O)CCCN(C(c2cnc(Cl)cn2)=O)CC1 c1(N2C(C(=O)NCC3CCCOC3)CC3(CC3)C2)ncnc2ccc(F)cc12 c1(CN2C(COC)CN(C(C3CCCCN3C)=O)CC2)cc(Br)cc(C)c1O c1(C(N(C2(CC(=O)N(CC(C)O)CCO)CC2)C)=O)cscc1Cl Cc1ccc2c(N3CCN(C(=O)C(C)(O)CC(C)C)CC3)ncnc2c1 C1(NC(C2(C(N)=O)CC2)=O)CC=C(C(=O)N(CC(O)CO)C2CCC2)C1 CS(=O)C=CC(=O)NCCC1CCN(C(C2CCCN2C(=O)C(F)(F)F)=O)CC1 N1(C(C=CC(=O)N(C)C)=O)CCC2CCC(NC(c3cc(Cl)nnc3O)=O)C1C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(C(C)NC(c2cnn(C)c2N)=O)C1 O=C(CCCn1ccnn1)NCC(C1CCOC1)NC(=O)Cc1nc[nH]n1 N1(C(c2c(COC)cco2)=O)CC2CCCCN2CC1CNC(=O)C=CCOC C(=O)(C(CNC(=O)C(C)=CC(C)(C)C)C(C)(C)C)N1CCCC(C#C)C1 N1(C(c2c(C)csc2Cl)=O)CC2OCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 c1(CNC(C=CCN(C)C(C2CCSC2)=O)=O)ccc(Cl)cc1 N1(C(=O)OC(C)(C)C)CCC(C#N)(NC(c2cccc(OCC(F)F)c2)=O)C1 CC(CC(=O)N1CCCC1C1(NC(=O)C=CC(F)(F)F)CC1)CC(F)(F)F c1(C(N2CCC(CSCc3nnc(CC)o3)C2)=O)ccc2c(Br)cccc2n1 C1(C(=O)NC2(CF)CN(C(C(C)CN(C)C)=O)C2)CCCCN(C)C1=O N1(C(Cc2c(C)scc2)=O)CCOC(CCNC(=O)CC2CC(F)C2)C1 N1(C(CC=CCC)=O)CCCN(C(=O)CSc2nncn2C(C)C)CC1C N1(C(C(C(C)C)N(C)C)=O)CCCCC(NC(=O)CC2(C)CCC2)CC1 Cc1ccc(C(=O)N(CC(C)NC(=O)C2=CCOC2)C)c(F)c1F C1(C(N(CC(CC)(O)CC)C)=O)CN(C(=O)CN2CC3CC3C2)CC12CC2 c1(-c2cccc(OC)n2)cc(C(=O)Nc2ccc3cncn3c2)cc2cc[nH]c12 C(C(=O)NCCC1CN(C(c2ccccc2)=O)C1)(C(C)C)N(CC)CC c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)cc2)=O)cnn2c1N(C)CC2 N1(C(COCCCC#C)=O)CC(CC(=O)NCCn2cncn2)CC1C C1C(C)(C)CNC(=O)C(C)CC(C(=O)NC)N1CC1CC1.CCOC C12(CNC(=O)CC3CCOC3=O)CC(CN1C(=O)CCC1CCCO1)C2 O=C1NC(=O)C2(CCCN(C(=O)C(F)(F)c3cccnc3)C2)N1 C=C1COc2c(C(N3CC(C)CN(C(=O)CCCCC)CC3C)=O)cnn2C1 C1(N(C(=O)CC2CC3(CC3)C2)CCO)CCN(C(=O)Cc2nc[nH]n2)CC1 c1(C(=O)NCC2CC(NC(C3(OC(C)C)CCOC3)=O)C2)cnc[nH]c1=N n1(C(C)(C)C)nnnc1C(C1CC1c1cccs1)NCC1CCCO1 CC1CC=C(C(=O)N2CC3CN(C(c4cc(C#N)ccc4F)=O)CC3C2)CC1 Cc1nc(F)ccc1CN1CCCCC1C(=O)NCCC(C)C N1(C(=O)NC)CCCC1(C)C(=O)N(CCCNC(c1ccncc1C)=O)C C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccoc1C)NCc1c(C)cccc1 c1(C(=O)C)ccnc(CNC(=O)CO)c1.C1(OCC#C)CN(C2CCC2)C1 c1(OCC)ccc(NC(=O)NC(=O)COc2ccccc2C(N)=O)cc1OC O=C1CC(=O)NC(C(=O)NC2(CC(N3CCOCC3CO)=O)CCCCC2)C1 c1(C(N2CC(CC)C(NC(=O)C=CCO)C2)=O)ccc(S(=O)(=O)NC)o1 C1(O)(CCNC(CS(N)(=O)=O)=O)CCN(C(=O)Cn2ccnn2)CC1 C1(C(C)NC(COC(CC)CC)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(CC=CC)=O)CCC(N(C)C(C2CC(CC(C)(C)C)C2)=O)CC1 c1(C(N2C(CNC(C3(C)N(C)CC(OC)C3)=O)CC2)=O)c(O)ccc(Cl)c1F C(=O)(CCCCCC(C)O)NC(CC=C)CNC(c1cncc2ccsc12)=O C12CCN(C1)C2=O.c1(NC(C(c2ccccc2)NC(N)=O)=O)n[nH]cc1F C#Cc1ccc(OCC(=O)NCC2(C)CN(C(c3cnn[nH]3)=O)CCO2)cc1 CCCC(C)(C)CC(=O)N1CCC(C(F)C(=O)NCCCc2nnnn2C)C1 C(C1=CCN(C(=O)C2=CCCCO2)CC1)NC(C1CCC1c1nc[nH]n1)=O C=CCC(C)(C)C(=O)N1CC(CC(C)NC(C2(C(=O)OC(C)(C)C)COC2)=O)C1 C1(NC(c2csc(CNC(=O)C(O)C3CC3)c2)=O)CCCC(CO)C1 N1(C(c2c(C)con2)=O)CCN(C(=O)CCc2cccn2C)CC1CF C1(C(=O)Nc2cn(C)nc2)C2CCC(C2)C1NC(=O)Cc1ccco1 C1(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CCSC1(C)C C1(C(=O)NCC2CC(F)CN2C(c2cccnn2)=O)CC2(C1)CC(F)(F)C2 N1(C(Cc2ccc(OC)cc2)=O)CC2(C1)C(NC(=O)CC(C)F)CCS2(=O)=O C12(CCCC1)NC(=O)CSC2.C1CCCCO1.C12CC(C1)C(=O)NCC2.CS C(C(F)(F)CCC(=O)NC1C(C)CCC1C)n1cc(-c2cc(C)c(F)cc2)nn1 CC1(C)C(CNC(C2CCCN2S(C)(=O)=O)=O)CCN1C(=O)CC(F)(F)F C(C1=CCCSC1)(c1n(C2(C)CC2)nnn1)NC1CC1F c1(OC(C)C(=O)N(C)CC2(C(C)(C)O)CC2)cccc(F)c1.C1(=O)C=CCN1 c1(CC(=O)NCC(CC=C)NC(=O)C(CSCC)OC)ccc(O)c(Cl)c1 CC1CN(Cc2cccnc2)CCC1NC(c1cc2c([nH]1)CCC2)=O CN=C(NC(C)(C)C=Cc1ccccc1)N1CN(C)C(=O)C1C CC1(N(C(C2CCCCCCC2)=O)CONC(C2CC23CCCC3)=O)CCCC1(F)F c1(OC)ccn2cc(C(=O)NC3CCCC3NC(c3oncc3C)=O)nc2c1 C1(C(N2CC(C)(CC)C2)=O)CC(C)(C)CN1C(C1CC(=O)C1)=O C1(C(N2CC(NC(c3cc(CCC)[nH]n3)=O)C(C)C2)=O)CC2(CCC2OC)C1 c1(C(N2CCC(F)(CNC(Cc3nc(C)sc3C)=O)C2)=O)ccccc1[N+](=O)[O-] N1(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCCC2NC(=O)CC2CC=CCC2)C1 c1(CCCC(=O)N(C2CN(C(c3cnc(C)[nH]3)=O)C2)C)ccc(F)cc1Br C1(OC)(CNC(C2(C)CC2F)=O)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1 N1(C(C(CC)(C#N)CC)=O)CC2OCCN(C(C3CCCSC3C)=O)C2C1 O(NC(=O)C(CNC(=O)COC1CC(=O)C1)C(C)(C)C)CC(C)C CC(C)C(C)CC(=O)NCC12CC(NC(=O)CN3CC4CCC3C4)(C1)C(C)O2 c1(C(N(C2CCN(C(C(C)OC3CCCC3)=O)C2)C)=O)cc2cc[nH]c(=O)c2s1 S(=O)(=O)(c1ccccc1F)NCC(=O)N(CCCNC(C1(C#N)CCC1)=O)C C1(C(=O)NCC2CCN(C(Cc3cc(C)on3)=O)C2(C)C)CCOCC12CCC2 c1(C(C)NC(CC2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)nn(C)cc1O c1(C(=O)NCC(C)NC(=O)CC2(C(F)(F)F)CC2)nccnc1OC1CCCC1 C1(NC(=O)NCC(C)CN2CCCC2)CC12CCCCC2 N1(C(C2CCC(NCc3cn(C(C)C)nc3)C2)=O)CCC2SC(=O)C=C2C1 c1(SCCC(=O)NCCCCN(CCCNC(C(=O)NCC)=O)C)n[nH]c(C)n1 N1(C(c2ncnc(C)c2C)=O)CC2(CNC(c3cnc(C)n3C)=O)CCC1CC2 C=CCN=c1[nH]cc(C(N2CCN(C(c3cc(F)n(C)n3)=O)C(CCC)C2)=O)s1 C(=O)(C1=CC2CC=CCC12)N1CC(C(N)=O)(CNC(c2[nH]c(CC)c(Cl)n2)=O)C1 N1(C(CSCC#C)=O)CCC2(C=C(C(=O)N(C)CCOC(F)F)C2)C1 C1(NC(CCSCCC)=O)CC2CCC1(C(=O)NCc1cc(C)co1)C2 C(=O)(C1CCCc2sccc21)N1CC(O)(C(C)NC(C2COCC(C)(C)O2)=O)C1 c1(C(=O)NCC2OCCN(C(c3c(C)ccnc3Cl)=O)C2)cccc2cnnn12 C1(C(=O)NCCCN(C(C2CSCN2C(C)=O)=O)CC)OC2CCC1CC2 N1(C(CC)C)CCN(C(=O)CN2CCN(C(=O)C(C)(F)F)CC2)CC1 N12CC(F)CC1CN(C(C)=O)CC2=O.C(C=O)=CCOCC.OC C(CCCC(C)(C)C)NC(C(C(C)O)NC(=O)COCCF)=O C1(C(C)(C)O)(CO)CCN(C(C2(C3CCCCO3)CCOCC2)=O)C1 n1(C(C)CO)cc(C2CCN2NC(=O)C(c2cccn2C)=O)nn1 C(C#CC(C)n1cc(C(c2ccccc2)C)nn1)(OCC)OCC CC1CN(C(=O)Cc2cnco2)CCC1N(C(=O)CCCC(=O)N(C)C)C CC1(NC(c2cnc(S)[nH]2)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C1 C1(C(N(CC(=O)NCC(F)F)CC)=O)C(C)(C)C1(F)F c1(CC(=O)NC2(CCNC(=O)CC3CCC(=O)N3)CC2)csc(C(F)(F)F)n1 CC(CC(=O)NC(C(=O)NCc1ncco1)c1cccs1)n1cccc1 CC(C)S(=O)(=O)c1cccc(C(=O)N(CCCCN(C(=O)CC(C)(C)C)C)C)c1 CC(N=c1[nH]c2c(c(=NC3CCCS(=O)(=O)C3)[nH]1)CCCCCC2)c1cnc[nH]1 c1(C(=O)NCc2c(CNC(CNC(=O)OC)=O)cccn2)cc2n(n1)CCCN2 C(CC[Si](C)(C)C)NC(C1(SC)CN(C(C2CC(C)CO2)=O)C1)=O C1(CCCNC(c2c(C)nco2)=O)CN(C(c2cnccc2N(C)C)=O)CCO1 N1(CC(=O)NCC2CC3CCC2C3)Cc2ccc(NC(c3cnns3)=O)cc2C1 c1(C(N2CC(NC(c3cccc(NC(C=C)=O)c3)=O)C2)=O)cnc(Cl)c(C)c1 N1(C(C(CC#C)C)=O)CCC(CCOC)(NC(=O)CC(C)c2cnn(C)c2)CC1 c1(OC)cccc(C(C(=O)NCC(F)CNC(c2nc(C)sc2C)=O)OC)c1 c1(CC(=O)NCCc2csc(-c3cccc(F)c3)n2)ccccc1O C1(CN(C)C(C2CC2c2cncnc2O)=O)CCCN(C(c2ccsn2)=O)C1 O=C(C1Cc2ccc(Cl)cc21)NC1CN(C(c2ccc(Cl)o2)=O)CC(F)(F)C1 c1(C(=O)NCC(CO)NC(C2(CC)CCC2)=O)ccnc(OC2CC2)c1 N1(C(C(C(=O)OC)C)=O)CCC12CCN(Cc1cc(Br)cc(C)c1O)CC2 CC(CC(C)NC(=O)CCC1CC1)NC(c1n[nH]c(-c2ccccn2)n1)=O N1(C(CC(CCC)O)=O)CCC(C(=O)N2CC(C(N)=O)C(C)C2)=C(F)C1 C1(N(C)CCN2CCC(O)C2)CCN(c2nnnn2-c2ccccc2)CC1 C(c1ccccc1F)=CC(N1CC2CC1CC2NC(C1(F)CCCCC1)=O)=O N1(C(c2n(CCCC)ncc2)=O)C2CCC1C(NC(=O)COCC)C2 C(=O)(CC(C)COC)NCC1(C(=O)NCC(C)OCC#C)CC=CC1 CN1C(=O)CN(CC(N2CC(C3(Nc4ncnc5sccc45)CC3)C2)=O)C1=O C(=O)(CCCn1cncn1)N(C(C)C(=O)NC(C)CSC)CC C1(C(=O)NC(C2CCN(C(c3csc(-c4cnc[nH]4)n3)=O)C2)C)CC(F)(F)C1 C1(C(N(CCNC(C2(N(C)C)CCCC2)=O)C2CC2)=O)CC12CCC(F)(F)CC2 C(=O)(C#CC1CCOCC1)NCC1N(C(c2cc(S(=O)(=O)N(C)C)oc2)=O)CC1 c1(-c2cccc(CCNCCC)c2)c(C)ccc2ccccc12 C1(C(C)C)CCCN(C(=O)CN(C(c2ccnnc2)=O)CC2CC2)CC1 CC1(C)CC(C(=O)NCC(O)CCC(N2CC(c3cc(O)no3)C2)=O)=NO1 C(=O)(C1=NOC(CNC(c2c(C)oc(C)c2C)=O)C1)N1CC(CCC)OCC1 c1(C(C)C)cc(C(=O)NCCC(O)CNC(=O)CN(C2CCSC2)C)ccc1O c1(C(=O)NC2CC(N(C(C(C(C)C)SC)=O)C)C2)cc(Cl)c(F)c([N+](=O)[O-])c1N C1(=O)C(O)CCN1.C123CC(C1)(C2)CNC(=O)C3.C1(C(=O)OC(C)(C)C)(OC)CCC1 N1(C(c2ccc(OC)nc2OC)=O)CCC2CCC(NC(C3CCC(=O)O3)=O)C12 CCCS(=O)(=O)C(C)C(=O)NCC(C1CCCN1C(c1ccncc1O)=O)(C)C c1(C(=O)NCCOCCN(C)C(C2(F)CC=CCC2)=O)cccc2c1nc(O)n2C Cc1ccc(-c2cc(NC(=O)C(C)OC(c3cnn(C)c3C)=O)n[nH]2)cc1 N1(C(C=CCC)=O)CC(CC(=O)NC2CC2(C)C(F)F)CC1(C)C C(=O)(C1=C(Cl)CCC1)N1CCC(CN(C)Cc2nncn2C)C1 N1(C(COCCCN(C)C)=O)CC2(CC2)CC1CC(=O)NCC(F)(F)CO c1(C(=O)NC2CC(F)(CNC(c3ccn(C)c3)=O)C2)cc(N)c(Br)c(F)c1 N1(C(CC2(NC(C3CCSC3)=O)CCC2)=O)CC(O)(C2CC2)C1 c1(OC)ccc2cc(C(=O)NCC3(Br)C(C)C3C)[nH]c2n1 c1(C(N)=O)ccnc(C(=O)NC23CC2CN(C(C2CSCCS2)=O)C3)c1 c1(C(=O)NC2C3(CC(NC(C(COC)(C)OC)=O)C3)C2)cnc2c(C)cccn12 c1(Cc2onc(C(C)(C)NC(c3ccccc3)=O)n2)ccc(N)c(Cl)c1 C=CCC(C(=O)NC(CNC(=O)CCNS(C)(=O)=O)C(C)(C)C)NC(C)=O C1(CCC)CN(C(c2ccncc2Br)=O)CCN1C(C12CC(O)C1C2)=O c1(C(=O)NCC2N(C(CC3N(C(C)=O)CCC3)=O)CCCC2)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(N2CC(CNC(C3CC3(C)Br)=O)C2)=O)n1 Cc1cc(C)c(C(=O)NC2CC(NC(c3cc(C4CC4C)on3)=O)C2)cn1 CCCC(C(O)C(=O)N1CCOC(CC)C1)NC(C1C2CCC(C2)C1C)=O C1(C(=O)NC(c2cccnc2)CC)CC12CCN(C(=O)CC1CC=CC1)CC2 C#CC1CC2CCC1N(C(=O)C(CNC(=O)C1=C(Cl)CCCC1)CC=C)C2 CCC(CNC(C12COCC1C2)=O)(CC)NC(c1cncnc1)=O C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CCN(C(c3cnn(CCC)c3C)=O)C2)C1 CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(c1cccnc1NC)=O N1(C(CCN(C)C(c2nc(C#N)cs2)=O)=O)CCN(C(N)=O)CC1 C1(COC)(CNCc2ccc(C(C)(C)C)s2)CCCO1 C(N=c1ccc(C#N)c(C)[nH]1)C1C2CN(C(C(CC)CC(C)C)=O)CC21 C(CCC(C(=O)NOCC(C)C)NC(C1OCCOC1C)=O)OC CC1CCC(NC(c2ccc(C3CC3)cc2)=O)CN1C(=O)Cc1cccnc1 N1(C(c2cc(C)nnc2O)=O)CC2ON=C(CNC(=O)C3=CCCCC3)C2C1 c1(C(C)NC(C(Cc2cn[nH]c2)NC(COCCCOC)=O)=O)ccc(O)nc1 C1(C(N2C3CC(NC(COCC=C)=O)C3CC2)=O)COc2ccccc2C1 c1(C(N2CCC(C)(NC(CN(C3CCCC3)C)=O)C2)=O)cncc(O)c1Cl C1(C2CCN(C(C3CCC4(CC3)CC4)=O)CC2)(NC(CCOC(C)=O)=O)CCC1 Cc1cccc2cc(C(=O)NC3CC4(C3)CC(CNC(=O)CSC3CC3)C4)sc12 c1(C(N2C(COC)CCC2)=O)ccc2nccn2c1.c12cccc(c1)NC(=O)N2 c1(C(=O)NCC2(C)CCCC2NC(C2(CO)CC2)=O)cc(CO)ccc1Cl C1(C(N(CC(C)C#N)C)=O)CCN(C(=O)CC2CCOC2(C)C)O1 c1(CC)ccc(C=CC(=O)NC2CC2CNC(=O)Cn2ncc(Cl)c2C)cc1 CC(C)CC(CN(C(=O)Cc1ccnn1C1CCC1)CC)NC(c1ccc(F)s1)=O C1(CNC(C=CC)=O)CC(C)(C)CCC1NC(c1cncc(NS(C)(=O)=O)c1)=O c1(C(C)C)ccc(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)CC2)cc1 N1(C(C2CC(CC)C2)=O)CCC(OCCNC(=O)NCCC2CC2)C1 Cc1sncc1NC(=O)C(C)NC(=O)COC1CC=CC1 CCCCC(F)C(=O)N(CCCNC(=O)C(C)(C)C(F)F)C1CC1 C1(CC)CN(C(C2(CC(=O)OC)CC2)=O)CCN1Cn1c(CC)ccn1 c1(CNC(C(C)(O)C2CC2)=O)cncc(C(=O)NCCn2cnnn2)c1 C#Cc1cccc(C(=O)NCCOCCNC(=O)CC2(C)CCS(=O)(=O)N2)c1C N1(C(c2c(COC)noc2)=O)CCN(CCCNC(C2(C)CCOC2C)=O)CC1 N#CC1CCC(C(=O)NCCCCCCNC(=O)C(F)CC2CCC2)CC1 c1(CS(=O)(=O)N(C2(C(OC)OC)CC2)CC2CC2)cc(C)ccc1C c1(OC)ccc(CN(C(c2cccc(Cl)n2)C(=O)NCC2CCOC2)C)cc1F CC1(C)C(O)CCCN1C(C1(c2ccccc2F)CCC1)=O c1(N(CCOC)C)cncc(C(=O)NCCN(C)C(C2CC(C)(F)C2)=O)c1 N1(C(c2ccc(C(=O)NCC)nc2)=O)CCOC(C)(C(=O)OC(C)(C)C)C1 N1(CC)CCN(CCC(=O)NC2CC(NC(c3cn[nH]c3)=O)C2)CC1 C(CSC)(C(=O)N1CC(O)(C(C)NC(C2(C(F)F)CC2)=O)C1)OC C1(CC(N2CC(C#C)(F)C2)=O)CC2(C1)CN(C(=O)CC1CCCC(=O)N1)C2 C1(C(=O)NCC(C)CNC(=O)C(c2cccc(F)c2)C)CN(C)CCO1 C(=O)(CCC(C(=O)N1CCC(N(C)C(C2CCC2)=O)C1)N(C)C)OC N1(C(CCC=CC(C)C)=O)CCC(C)C(CNC(=O)CCCF)C1 C(=O)(C(C)CC1CCCC1)NCCOCC(=O)NCCCC(c1cccs1)C C(=O)(CC(CC(C)C)NC(c1cc2ccccn2c1)=O)N1C(CC=C)CCCC1 N1(C(C(CC)=CC)=O)CC=C(CNC(=O)C(C)NC(=O)OC(C)(C)C)CC1 C(CC(=O)Nn1ccnn1)N(C(=O)C(CC)C(F)(F)F)CC#C N1(C(Cn2nnc(C)n2)=O)CCCCC1Cn1cc(CCN2CCCCC2)nn1 c1(OC)ccc(Br)c(C(N2CC3(C2)CN(C(=O)Cn2ccc(C)n2)C3)=O)c1F c1(CC)ccc(C)cc1C(=O)NCC(n1cc(CN(C)C(C)C)nn1)C Cn1c(=O)ccn(CC(=O)NCC2CN(C(=O)CC3(O)CC3)CC2(C)C)c1=O CC1(C)CC(C(=O)NCCOCCNC(c2cn3cnnc3cn2)=O)CNC1=O c1(C(N2CC(NC(c3c(OC)cccc3)=O)C(C)C2)=O)cc(Cl)ccc1N Cc1ccc(C(N2CC(NC(=O)CC3CCCSC3)CC23CCC3)=O)cc1C#N CC(CC(F)(F)F)N(C(CC1CCCCO1)C(=O)NC1CCC1)C C1(NC(C2C(C#C)C2)=O)CC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 CC(CNC(=O)C=CCNC(c1ccc[nH]1)=O)CN1CCCC1 C=CC1(CC)COCCN1C(=O)CS(=O)(=O)CC1COCCO1 C(C(C)(C)CC(=O)NCC1CC(C)(C)CN1C(=O)C(C)c1ccco1)OC C1(NC(c2cncc(Cl)c2)=O)COC2CN(C(C3CCC34CCOCC4)=O)CC12 c1(C(N2CC(C(=O)NC3CCN(C(C)C)C3)C(F)C2)=O)ccc2cncn2c1 c1(N2CCC(CCOCC)(NC(c3csc(C)c3)=O)CC2)cc(O)nc(=O)n1C C(=O)(C1Cc2ccccc21)NC1CCN(C(c2c(OC)ccs2)=O)C(C2CC2)C1 Cc1cc(OCC(=O)NC2CCC(CNC(=O)C(O)C3CC3)C2)ccc1Cl c1(-c2c(CN3CCN(C(C(C(C)C)O)=O)CC3)cccc2)cc(O)c(F)c(F)c1 CC(=O)CCCCC(=O)NCc1nc(C(N2CCC3(CCO3)C2)=O)co1 Cn1nnnc1C(c1cnn(-c2ccccc2)c1)NC1CCSCC1 c1(C2N(C(C(C)(C)NC(C)=O)=O)CCC2)ccc(Cl)c(F)c1.C12CN(CCO1)C2 CC1CCCN(C(c2cccc3c[nH]nc23)=O)C1CNC(=O)COCC(F)(F)F C1(NC(c2cnc(N(C)C)o2)=O)CN(S(=O)(=O)Cc2ccccc2Cl)CC1O N1(C(C(CO)N(C)C)=O)CC2OCC(NC(c3ccc(-c4ccco4)o3)=O)C2C1 N1(C(C2C(CC)CCO2)=O)CC(NC(=O)CCn2cnccc2=O)CC12CCC2 CCCC(CNC(c1cc(CC)n(C)n1)=O)C(=O)NCC#CCC N1(C(CS(=O)(=O)NC)=O)CCC(NC(=O)CC2CCC(C)(C)C2)C(F)(F)CC1 C12(C(N(CCCCNC(CC3CCC(C)O3)=O)C)=O)CC3CC1(CO)CC3C2 C1(C(=O)NC2(c3ccccc3)CN(C(CCCOC)=O)C2)CS(=O)(=O)CC12CC2 c1(OC)cccc2c(CC(=O)NC3CCN(C(=O)C(O)CC(F)F)C3)coc12 c1(CC(=O)NCCC(C)NC(c2nccnc2C(N)=O)=O)ccc2c(c1)COC2 C=CC(CC)CC(=O)NCC(CO)NC(=O)C(F)=C(C)C1CC1 N1(C(C(C2(O)CCC2)NC(C(CCOC)C)=O)=O)CCCOCC1C c1(C(N2C(C(N3CCC(C(=O)NC)C3C)=O)CCC2)=O)cc(=O)n(C)cn1 CC1Cc2cc(S(=O)(=O)NC3COc4cc(Br)cc(F)c43)cc(Cl)c2O1 C1(CNC(=O)NCCc2c(C)ccnc2)CCC2(CCC2)CO1 n1(CCCOC)c(N2CCOC(C)C2)nnc1CC(C)(C)O Cc1nc(C(N2CCC(O)(C(C)CNC(=O)COC3CCCC3)C2)=O)c(C)s1 C=CC1OCCC1NC(C1(OC)CCN(C(=O)C=CC2CCCN2C)C1)=O C1(CCC)C(=O)NCCN1C(=O)C(CC)N(C)C(c1occc1C)=O C1(NC(C(=O)NC2(C)CC(N)C2)=O)C2CCCC(F)(F)C12 C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(N(C(c2cc(C)n(C3CC3)n2)=O)C)C(F)C1 c1(C(=O)NCCCC2(NC(C3ON=C(C)C3C)=O)CC2)sc2ncccc2c1Cl CC(=O)CCN=C(NCc1ccc(C(N)=O)nc1)NCC(C)(C)C1CC1 C(=O)(C1=CCCN(C(C2Cc3nccn3C2)=O)C1)N1CCC(C)(C)CC1 c1(C(N(CC(O)CNC(c2ccnc(C3CC3)n2)=O)C)=O)cccc2oc(O)nc12 C=C(C)CCC(=O)NC(CNC(c1ccncc1OCc1cccs1)=O)C(C)C c1(C(=O)NCC2(O)CCN(C(c3cc(F)ccc3F)=O)C2)ccc2cncn2c1 N1(C(=O)CCCC2CCC2)CCCC(F)(CNC(C23CC(CC(F)F)(C2)C3)=O)C1 C1(CCNC(c2cc(COC)on2)=O)COCCN1C(=O)CCC1CCCOC1 C(C(C)C#N)NC(CN(C(=O)C=C(C)C1CC1)CCOC)=O c1(C(=O)NCCCN(C)C(C2CCC2(F)F)=O)ccc2c[nH]nc2n1 c1(C(=O)NC2CC(C)(NC(CC34CC(C)(OC3)C4)=O)C2)ccc2oc(=N)[nH]c2c1 C(=O)(C#CC1(C)CCCO1)NCC1(O)CC(CNC(c2c(F)ccc(C)n2)=O)C1 c1(C(=O)NC2C3(CC(NC(C4(C)CNC(=O)C4)=O)C3)C2)nc2cccnc2s1 N1(C(C2C(C)CC2C)=O)CCC2(CC1)CCN(C(=O)CCC(=O)c1cccs1)C2 C=C(C)CN=C(NC1CC(O)C12CCOCC2)N1CCC(OCCNCC)CC1 C1(C(=O)NC2CCN(C(CCSC)=O)CC2)CCc2n[nH]cc2C1C C(CCC1CC1)(C(=O)NOC1CCOC1)NC(COCC)=O.c1nc[nH]n1 c1(C(=O)NC(CNC(c2cnc(C(C)=O)s2)=O)C)coc(S(=O)(=O)N(C)C)c1 C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cccc(N)n2)=O)CCN1C N1(C(CC(=C=C)C)=O)CC2(CC)CC1(CNC(=O)C(c1ccccc1)O)C2 c1(C(=O)NCCCOCCN(C)C(c2cc(CO)n(C)n2)=O)cnn2ccccc12 N1(C(=O)CSc2ccsc2)CCC2CN(C(C3CN(C4CCCC4)C3)=O)CC12 N1(C(C(CSC)OC)=O)CCC(O)(CCNC(c2cc(F)ccc2O)=O)CC1 c1(C(N(CCCCNC(C(CC=CCC)C)=O)C)=O)cc(C(F)(F)F)ccc1F C=C(Cl)CC(C(=O)NCC1(S(C)=O)CC1)NC(=O)CC1CCCNC1=O N1(C(C2C(C(=O)NCCc3ccccc3)C2)=O)CCCC1c1ccccc1 N1(C(CN(S(C)(=O)=O)C)=O)CCCC1CCNC(C1(CO)CCCO1)=O CC(CN)CC(=O)N.C(=O)(CS(N)(=O)=O)N1CC(N(C(=O)OC(C)(C)C)C)C1 c1(CCN2CC(CC(=O)NC(CCCN(C(C)=O)C)C)C2)cc(OC)ccn1 c1(NC(C)Cc2ccc(C3CCCC3)cc2)cccc2c(C(=O)O)nccc12 c1(OC)c(C(=O)NCC2(CC(=O)NCCc3nnc(C)s3)CC2)cnn1C N1(C(c2cc(OC)ncn2)=O)CCCC2CN(C(=O)CC3CC3)CCCC12 N1(C(C2CC(C(C)C)C2)=O)CC2CCN(C(=O)CCc3cccc(O)c3)C(C2)C1 c1(N(C)CC)nc(=N)[nH]c(=NCC2CC2NC(=O)CNc2ccccn2)[nH]1 C(=O)(CCCC(C)(F)F)NCCCC(C)(C)NC(C(C)NC(CC)(C)C)=O c1(C(=O)NCC(C)N(C(=O)CCc2cn(C)cn2)C)cc(O)nc(Cl)c1 CN1CCOc2c(C(=O)NC3CC4CC(NC(=O)C(C)(C)C)C4C3)cccc21 C1(NC(C2CC(N(C)CC)C2)=O)CN(C(=O)CC2CCCOCC2)CC1C1CC1 C1(SCc2ccc(C)cn2)CCNC2(CCC2)C1 C=CC(C)CC(=O)N1CC2CC1C2NC(=O)CNC(c1cc(C)oc1C)=O C(=O)(C1CCCc2nc[nH]c21)NC1CCN(C(c2c(N)nc(Cl)cc2)=O)C12CC2 N1(C(CNC(C(CC)C)=O)=O)CC2CC(C1)C2NC(C1CCCCO1)=O N1(C(C2CCCSC2)C(=O)NC(C)C)CCCCC2(CCC2)C1 N1(C(C(C(C)C)F)=O)CCCC(O)(CNC(c2ccnc(OC3CC3)c2)=O)CC1 c1(OCC(N2CCC(C)(NC(C(CC=CC)C)=O)C2)=O)c(C)cc(Cl)cc1C Cn1nc(C(=O)NCC2CCC(CN=c3[nH]nco3)CC2)c2c1CCCC2 C#CC1(C(N2CCC(N(C(=O)Cc3ccc(C)nc3)CC3CC3)CC2)=O)CCCC1 C1(F)(C(N2CCC(OCC#C)C2)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(OC)cccc(F)c1C(C)NC(=O)C(=O)NCC(c1ccc(C)cc1)(F)F c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C2CC2)ccccc1N1CCCC1=O Cc1coc(C(=O)NC(c2ccccc2)C(=O)NCC(O)CF)c1 C1(C(=O)NCCCNC(COc2c(C)cc(Cl)cc2)=O)CC2CCCCN2C1 C1(NC(c2ccc(C(F)F)o2)=O)CN(C(c2cc(Cl)ccn2)=O)CC12CC2 c1(OC)cc(F)ccc1NC(C1CCN(C(=O)c2c[nH]c(C#N)c2C)O1)=O S(=O)(=O)(c1ccc(C#N)c(N2CCC(=O)N(C)CC2)c1)NCC(CC)C(C)C n1(C(C)C)nc(C(=O)NCCCC(C)NC(C2(C)CCCO2)=O)c(Br)n1 c1(C(=O)NC(C)CCNC(c2cc(C3CC3)n(C)n2)=O)sc2cccnc2c1Cl C1(CNC(=O)C(O)c2ccco2)CCCC1NC(c1cncs1)=O C1(CCNC(C2C(OC)C2)=O)CSCCN1C(=O)C(=O)Cc1ccc(Cl)cc1 C#Cc1ccc(C(=O)NCCCN(C)C(c2ccn(CC(C)C)n2)=O)cn1 N1(C(CC(C)(F)F)=O)CCCC(C2CCN(C(=O)C3=COCCC3)C2)C1 CC1(c2nn[nH]n2)CCCN(CCS(C)=O)C1 CCC(C)(C(=O)N1CCC(N(C(=O)Cc2cc(-c3ccccc3)on2)C)C1)OC N1(C(c2cc(C(=O)OC)ncc2)=O)CC2CCC(C1)N2C(=O)C(C)=C(C)C N1(C(C=CCOC)=O)CCC(C)N(C(c2ccc(C(F)(F)F)c(F)c2Cl)=O)CC1 C1(NC(C(C)(C)c2ccno2)=O)CN(C(C2CC2c2cccc(O)c2)=O)CC1O C#CC1(C(=O)NC2(C)CC3(CC3)C2)CCN(C(=O)CCc2nccs2)CC1 c1(CNC(=O)NC2CCN(C)C2c2cccs2)cccc2c1OC(C)(C)CC2=O C(CN=[N+]=[N-])(C(=O)NCC=Cc1ccccc1)NC(C=C1CCC(C)CC1)=O C(c1cncc(C)c1)=CC(N1CCC(N(C(C2CC2(F)Cl)=O)CC)C1)=O C=CCC(CC=C)C(=O)NC(C)CCC(=O)N1CC(CC23CC(C2)C3)C1 c1(C(=O)NCC2C(C)CN(C(c3cccc(=O)o3)=O)C2)[nH]nc2c1CCC2(C)C N1(CC#C)CC2C(CNC(=O)CC(c3ccc(F)cc3)c3ccccc3)C2C1 C(=O)(C(=O)CCC(C)C)N1C(C(=O)NC(CC=C)(C)CC=C)C(C)CC1 c1(SC)ccc(O)c(C(=O)NCC2CC2CNC(=O)C(N2CCNC2=O)C)c1 c1(CNC(C2C(OC)C2)=O)nc2c(s1)CN(C(c1c(C)cccc1N)=O)CC2 c1(CCC)ccc(C(C(C)C)Nc2ncc(C3CC3)s2)cc1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CN(C(C23C=CC(CC2)C3)=O)CC(F)(F)C1 C(=O)(C(O)C(F)(F)F)N(C(CNC(c1coc(Br)n1)=O)C1CC1)C Cc1ccc(Br)c(C(=O)NCC2CCCC2NC(=O)CC(C)C)c1 CC1CC(CNC(c2cc(-c3cnn(C)c3)on2)=O)CN1C(=O)CN1CCC1 CS(=O)(=O)CC(=O)N1CCC(C2N(C(c3cnccn3)=O)CC2(C)C)CC1 C(N=c1[nH]c2ccc(O)cc2s1)C1(C)CCC(NC(Cc2scc(C)c2)=O)CC1 C1(C(=O)OCC2C(=C)C2)CCC2(C1)CC2(F)F N1(C(CS(=O)(=O)N(C)C)=O)CCC2CCC(NC(=O)Cc3cnn(C)n3)C1C2 CCC(O)C(C)C(=O)NCC1(NC(C2CN(S(C)(=O)=O)C2)=O)CC(F)(F)C1 C1(C)(CC)CC(NC(=O)CNC(=O)CN(C)C)CCO1.C(C(C)(C)C)N1C(=O)C1 C(=O)(C1(C)OCCc2ccccc21)NC1C(NC(C2(CC)CC2)=O)CC1 C(C(=O)NOCC1CCCO1)(c1cccs1)NC(c1cc(OC)n[nH]1)=O c1(C(=O)NC(C)CCCNC(C2(C)C(C)(C)C2(C)C)=O)ncc(Cl)c(N)c1Cl c1(C(C)C(=O)NCCN(C(C2CC(N(C)C)C2)=O)C2CC2)ccc(F)c(F)c1 n1(CC(=O)N(CCC)CCNC(c2csnc2C)=O)nc(C)n(C)c1=O C1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)Cc2ccccc2C1 C(=O)(CCCC(=O)OCC)N1CC(CNC(C2(CC=C)CCCC2)=O)C(C)C1.O Cn1nc2c(c1CNS(=O)(=O)c1cscc1C(F)(F)F)CCCC2 C1(CC=C)(NC(C2CCCC2CC)=O)CCCN(C(C2COC(C)(C)C2)=O)C1 C(=O)(CC(C(C)(C)C)NC(c1ccc(O)c(C)c1)=O)NCC(=O)OCC#C C1(C(=O)NCC2OCCN(C(C3C(C)OCCC3)=O)C2)CCc2nc(O)[nH]c2C1 n1(CC)cc(Cl)c(C(=O)NCC(C2CCCCC2)NC(C2CCC(C)(C)C2)=O)n1 Cc1ccc(-c2cncc(C(=O)N(CC(O)CNC(C3CC3F)=O)C)c2)cc1 C12(C(N3CCC(C(=O)OC)C3)=O)CCN(C(c3ccc(OC)cc3O)=O)CC1C2 c1(C(N2CC(NC(CN(C(=O)OC)C)=O)C(F)CC2)=O)cn2c(n1)CC(C)CC2 S(=O)(=O)(c1ccccc1Br)NCCC1CCCN(C(c2ccsn2)=O)C1 C1(CCCCCNC(C(C)OC2COC2)=O)CCN(C(c2nonc2N)=O)CC1 C=CC(C)(C)C(=O)NC1CCCN1C(C1COCCN1C(=O)NCCC)=O Cc1c(C(=O)NCC2(NC(=O)C=C(Cl)Cl)CCOC2)cnn1-c1ccccc1F Cc1cc(C(N2CC(CNC(C3(C)CCCN3C)=O)C2)=O)n(CC(F)F)n1 N1(CC(=O)N(CCNC(c2c(C)con2)=O)CCOCCO)CC(=O)NC1=O C1(NC(c2c(OC)cc(C)s2)=O)CC(NC(C2CN(CC(C)C)C2)=O)C12CCC2 CON(CCC(=O)NCCN1CCCCCC1)C(=O)C(C)OC(C)(C)C C(N=c1[nH]c2c(c(=NCCc3c[nH]nc3O)[nH]1)CCCCC2)C1(CO)CC1 c1(OC)ccc(Cl)c(CCNC(c2ccc(OCc3csc(C)n3)cc2)=O)c1F C1(CC)CC(C(=O)NC23CCCC(NC(=O)C=CCO)(C2)C3)CC(=O)N1 O=C1CCC2CCN(C(=O)Cc3cccc(C4CC4)c3)C1C2 CCC(CC)CC(F)C(=O)NC1CC2(C1)CC2C(=O)NCC1CC(C)CO1 C1(C(=O)NCCOCCNC(c2c(=N)[nH]c(C3CC3)nc2)=O)CCCCC12CCC2 c1(C(N(CC(C)NC(=O)C(=O)N(C)C)CC)=O)ccc2c(c1)N(C)CC2 c1(C(=O)OCC2(C)CCC(C(=O)OCC)C2)onc2c1CCCC2 c1(OC)nc(C)ccc1CN1CC(N2CC(NC(c3cnn(C)c3)=O)CC2=O)C1 c1(NC)c(C(=O)NCC2(C)CCN(C(c3cc(O)nc(O)c3)=O)C2)cccc1N Cc1cc(C(=O)NCc2ccc(CN(C(=O)C=CS(C)=O)C)cc2)c(C)nc1C c1(NC(=O)CO)cccc(C)c1.c1(CC)noc(CC)n1.C12CC(C)(C1)OCC(=O)N2 c1(C(N(CC(CC)NC(=O)C(F)Cc2ccccc2)C)=O)ccc(OC)c(C)c1 c1(C(=O)NCCOCCCN(C(=O)CCn2cnc(=N)[nH]2)C)ns[nH]c1=O c1(C(N(CC(C)NC(C(C(C)C)SCC)=O)C)=O)nn(C)c(Br)c1C c1(C2(C(=O)NCC(CO)NC(C3(C)CCC(=O)N3)=O)CC2)cccc(F)c1F C(=O)(CC(C)(C)N(C)C(C)C)NCCCCN(C(C1(CCC=C)CC1)=O)C CC(C)CC(CCO)NC(C1C2CCC(C2)N1C(=O)CCCC1CC1)=O Cc1c(NC(=O)NC2CCN(C(C)C)C2)cccc1F N(C(=NCC(O)c1cccc(F)c1)N1CC2C(C)C2C1)C(C)C c1(C(N2C(C(=O)OC)CN(C)CC2)=O)ccc2c(c1)CCCNC2 Cc1[nH]nc(C(=O)NC2CN(C(C3CCC=CCCC3)=O)CCC2F)c1[N+](=O)[O-] CCCCCCC(C(=O)N1CC(CC)CC(O)C1)NC(=O)CCCCC(=O)OC C(=O)(C1CCCn2ccnc21)NC1(C)CCN(C(CC2CCN(C)CC2)=O)CC1 C12(C(=O)NCCC3CCN(C)C3)CC(CO)(CN1C(=O)C#CC1CC1)C2 C#Cc1cccc(C(N2CCCC(C)(CNC(c3ncn(CC)n3)=O)C2)=O)c1Cl C1(NC(c2c(C(C)C)onc2)=O)CCc2onc(C(=O)N(C3CCCC3)CCO)c2C1 Cc1nc(N2CC3C(NC(=O)C(C)CC4CCCC4)C3C2)c2cnn(C)c2n1 Cc1cncc(CC(=O)NCc2ccc(C(=O)NC3C(C)CCC3C)nc2)c1 C1(NC(CCCCCSC)=O)CN(C(c2ccncc2F)=O)C2CCCC12 C1(C(=O)NCC(C(C)(C)O)F)C2CC(O)C(C2)N1C(C1CCCS1)=O c1(C(=O)NCC(CN(C)C(c2cn[nH]c2)=O)(C)C)cccc2c1CCCCC2 Cc1cc(-n2cc(CCN(C(=O)CC3OCCOC3(C)C)C)nn2)cc(F)c1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CNC(C2CC(CF)C2)=O)C(C)C1 CCC(CC(=O)N1CC(CNC(c2sc(=N)[nH]c2C)=O)CC1(C)C)C(C)C N1(C(C2(C)CC(=C)C2)=O)CC2(CC(NC(=O)C=Cc3cnccn3)CO2)C1 N1(C(C(C(C)C)SCC)=O)CCC2(CC2NC(c2ccnc(C)c2)=O)C1 CC1(C(=O)NCCC2CCCN(C(=O)CCOC3CCCC3)C2)CCOCC1 Cc1cc(C(=O)NCCN2CCN(C(=O)C(C)(C)C(N)=O)CC2)n2nccc2n1 N1(C(CC2CCCC(C)C2)=O)CCC2(CCCN(C(=O)CCCN=[N+]=[N-])C2)CC1 C=CCC(F)(F)C(=O)NCC1CC(CNC(C2CCC(CC)C2)=O)C1 c1(C(=O)NCCCOCCNC(c2cc3scnc3[nH]2)=O)cnc2[nH]cncc1-2 C1(NC(c2cscn2)=O)C=CCN(C(=O)CCC(F)F)C1 C(N=c1[nH]cnc2ccccc12)C1CN(C(c2c(OC)cccc2)=O)C(C)C1 C1(NC(CCCOCC)=O)CC2CCC1(C(=O)NCC(=O)OC(C)C)C2 N1(C(CNC(C(CC)C)=O)=O)CCCC12CCN(C(c1nnccc1C)=O)C2 CCCCC(=O)NCC1(C(=O)NC2COCC2CC)CC=CC1 c1(C(=O)NC2CCCC(NC(c3cc(C)no3)=O)C2)cc(O)ccc1Br N(C(=NCC1OCCCO1)NCC1CCC1)C(C#C)C C(C)(CN=c1nc2[nH]ncc2c[nH]1)NS(c1c(OC(C)C)ccc(OC)c1)(=O)=O CC1CCOCCN1C(=O)CCc1ccccc1 Cn1nc(C(N2CCC(NC(=O)CSC(C)(C)C)C(F)C2)=O)c2nc[nH]c(=O)c12 N1(CC(=O)NC)CCCCC1n1ccc(C)n1.c1(C2CN2)ccccc1Cl c1(C(=O)NC2C(NC(C(C)OC)=O)C2)cccc(C2(O)COC2)c1 c1(CCC(=O)NCC(C)CN(C(=O)CC2CCCC2)C)nc2ccccc2s1 C(N=c1nc2sccc2c(NC2CCCC2C#N)[nH]1)c1c(OC)c(C)cc(C)c1 c1(SC)ncc(C(=O)NC(C)CC(C)NC(=O)Cc2c(C)cccc2C)c(O)n1 C1(NC(c2c(C)n(CC(C)(C)O)nc2)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(c2nccc(Cl)c2O)=O)CC1C N1(C(C)=O)CCCC(NC(C2C3CC2N(C(C2CC(=O)CS2)=O)C3)=O)C1 CN(C)C(=NCC1CC(=C2CC2)C1)NCc1ccc(Br)c(N(C)C)c1 c1(OC)ccc(C2CCCCC2)cc1C.C(C1CONC(=O)N1)OC c1(C(N2C(C)(CNC(C3CC3C(F)F)=O)CCC2)=O)cc(O)c2ccoc2c1 C1(C)(CC)CC(NC(C2(C(=O)OC)CC2)=O)CN1C(=O)Cc1cnc(C)o1 C(=O)(CC(F)(F)C(=O)OC)NCCCCCN(C(C1CC(=C)C1)=O)C n1(CC)nc(C)c(CC(=O)NCC2CC(C)(C)CN2C(=O)C(C2CC2)OC)c1C C1(C(=O)NC(C)C(=O)NCC2CC3C=CC2CC3)CCc2nnnn2C1 CCC(CC(=O)N(CCNC(=O)C(=CC1CCCCC1)F)C1CC1)C(C)(C)C c1(C(=O)NCC=CCNC(c2cc(=O)cc(Cl)[nH]2)=O)ccn2ccnc2n1 N1(C(C2(C=C)CCC2)=O)CCC(CC)(NC(=O)Cc2c(C)cnn2C)CC1 C1(NC(C2N(C(C(C)C)=O)CCC2)=O)CCN(c2ccc(C(C)(C)C)cc2)CC1 c1(C(=O)NC(CCNC(C2C(C)(CC)C2)=O)(C)C)ccc(C=CC(=O)OC)cc1 CCC(CC)(CN=c1[nH]c(=NCC(C)S(C)=O)[nH]c2cc(OC)ccc12)OC C(CCC(C)C(=O)N1CC(CCNC(c2occ(C)c2C)=O)C(C)C1)OC Cc1nc2ccc(C(=O)NCC3CCCCN3C(c3cnco3)=O)cc2nc1C CCCCCCCCC(=O)N1CC2CCC2(CC(=O)NOc2ccccc2F)C1 C1(OC)CN(C(C2(C(C)(F)F)CC2)=O)CC1NC(c1cc(C2CCC2)no1)=O Cc1nnsc1C(C)NC(=O)CCCNC(=O)CC1CCOC1C C1(NC(CCCN=[N+]=[N-])=O)CC2CCC(C1)C2NC(C1CC(=O)NC(=O)C1)=O N1(C(c2cc(C)c(F)c(C)c2)=O)CC2CCN(C(c3cccnc3S)=O)CC2C1 C(=O)(CC(C)(C(F)F)N(C)C)NC1C2CN(C(C3CC(CC)NC(=O)C3)=O)C1C2 C1(CNC(c2c(C(C)C)cco2)=O)CN(C(=O)C(C)C(F)F)C2(CCOCC2)C1 Cc1cc(C(C)(C)C)ccc1CN(C)C(=NCC1CCCO1)NCC(C)(C)CO N1(C(C2CC(CC)C2)=O)CCOCC1CNC(c1sccc1C(=O)OC)=O C1(NC(CCc2n(C)ccn2)=O)CC2CC1CN(C(c1ccc(=O)n(C)c1)=O)C2 CC1(C)CN(C(=O)CCn2ccc(=N)[nH]2)CCC1NC(c1ccc(CO)cn1)=O Cc1cccc(C(C)C(=O)NCC(C)NC(c2cnc(S)n2C)=O)c1 c1(N(C(N2CC(F)C(F)C2)=O)Cc2cc(-c3ccccc3)cs2)ccc2cc[nH]c2c1 C(c1ccc(F)cc1F)=CCN1C(C(=O)NCCc2ccc(Br)s2)CCCC1 O=C(C1CS(=O)(=O)c2ccccc21)NC1C=CCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(=O)CCCn2cc(CC(O)C3CC3)nn2)CCC(S(=O)(=O)C(F)F)C1 Cc1c(Cl)c(C(N2CCC(N(C)C(c3cc(Cl)c(Cl)n3C)=O)CC2)=O)nn1C Oc1c(CN=C(NCC2CCCCO2)NC2CCCCC2F)cccc1Br c1(OCC)cccc2c1OCC(C(=O)N(C1CN(C(=O)C(CC)C(C)C)C1)C)=C2 CCC(CC)C(F)C(=O)NC1(CNC(c2cc(C)c(N)cn2)=O)CCCCC1C c1(C(N(CCOC)CCNC(C2CC(C)N(C)C2)=O)=O)cc(C)c(O)c([N+](=O)[O-])c1 c1(CNC(C2CCN2Cc2ccc3sccc3c2)=O)ccc(F)c([N+](=O)[O-])c1 CN1CCOCC1C(=O)NC1CC(CNC(=O)CCSc2ccccc2)C1 CCC(CCC(=O)NCC1(O)CCCC1(C)C)NC(C1(C)CCN(C)CC1)=O C1(NC(c2n(C)c(=O)ccc2)=O)CN(C(C2(C(F)F)CC2)=O)Cc2nccn2C1 Cc1nc(C2CCC2)oc1C(=O)NC(C1CN(C(c2c(Br)nnn2C)=O)C1)C Cc1ccc(C(N2CC(NC(=O)C(c3cn(C)nc3C)O)C(O)C2)=O)c(C)n1 c1(OC)ccc(C(N2CCC(NC(=O)CSS(C)(=O)=O)C2C(C)(C)C)=O)c(F)n1 N1(CC(NOCCC(C)O)=O)CCN(C(C2CCC(=O)CC2)=O)CC1 CC1CN(C(=O)CC2COCCN2C)CCN1C(=O)C=Cc1ncc[nH]1 N1(C(C2(CC(C)C)CC2)=O)CCC(CN(C(=O)CC2CSCCO2)C)CC1 c1(C(N2CCC(C)C2)C(=O)NC(C(=O)OC)C)cn(C)nc1Br C1(NC(C(CCC)OC)=O)CCC2(CC1)CN(C(=O)C=C1CCC1)CCO2 c1(CN(C(C2N(C(C=CCN(C)CC)=O)CC2)=O)C)ccccc1C c1(CN2CC(NC(c3c(C)n[nH]c3)=O)C(F)C2)ccc2cc(Br)ccc2c1 O(NC(=O)CCC1CCCN(C(C2CCC(CC)O2)=O)C1)CC(=O)OCC S(=O)(=O)(c1ccccc1S(C)(=O)=O)N1C(C(=O)Nc2ccc(OC)nc2)CCC1 C1(CCCC)CN(C(=O)CCC2CCCN2C)CCN1C(=O)Cc1sccc1Cl C1(NC(C2(C)COC(=O)N2)=O)CN(C(C2CC(C3CC3)C2)=O)C2(CCCCC2)C1 C1(NC(c2ccc(OC(C)C)nc2)=O)CCN(C(c2cnn(C)c2F)=O)CC1O C1(NC(C(C)CC#N)=O)CC(C(=O)NCC(=O)NC2CCC2)=CC1O C1(O)(CNC(C(CC=CCC)C)=O)CCN(C(C2CC(C(=O)OC)C2)=O)CC1 c1(C(=O)NC2CCC(NC(=O)C3=CCCS3)CC2)cnn2cc[nH]c(=O)c12 N1(C(c2cccc(F)c2)=O)CC2(CCN2C(=O)CC2CCS(=O)(=O)C2)C1 N#Cc1ccc(NC(c2coc(-c3ccccn3)n2)=O)cc1-c1ccncc1 CC(C)CC(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)NC(=O)CSc1nc[nH]n1 c1(SC)ncc(C(N2CC(F)CC2CNC(C2(C(N)=O)CC2)=O)=O)n1C C(CC(O)CC(=O)NC1CCN(C(=O)CCC(C)(C)c2ccccc2)CC1O)SC c1(C(=O)NC2CN(C(c3cnc(N)c(Cl)c3)=O)C3C2C3)ccc2c(c1)COC2 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2(C)C1 c1(OC)ccnc(C(=O)NCCCC(C)NC(c2cc(C3CC3)ncn2)=O)c1F C#CCC(C)(C(=O)N1CCCC(COC)CC1)NC(C1CCCCCCC1)=O c1(C(N2CCC(n3cc(CC(C(C)C)O)nn3)C(O)C2)=O)cc(I)cc(Br)c1C CC1Cc2ccccc2N(C(c2cc(F)c(N)c(F)c2)=O)C1C C1(C(CO)NC(=O)Cc2cc[nH]n2)CCN(C(=O)Cc2ccc(F)cc2)CC1 c1(CNc2cccc(C(=O)NC(C(C)C)CO)c2)sc2ccccc2c1Cl N(C1CCCc2occc21)C(C(CCSC)NC(C1CCN(C)CC1)=O)=O N1(C(C2(COC)COC2)=O)CC(NC(C2(OC(C)=O)CC2)=O)CC(O)C1 N1(C(c2cc(C)oc2)=O)CCCC(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(CC(=O)NC2CCC(NCc3c(C)ncs3)C2)ccc(Br)cc1Cl C(CC(C)C(=O)NCCN(CCOC)C(C1(c2ccc(F)cc2)CCC1)=O)=CC N1(C(C(CC=CC)NC(C2CCC(C)(C)OC2)=O)=O)CC2COCC2(C)C1 O=S(=O)(c1ccc(Br)cc1NC1(C2CCCO2)CCC1)NCC1(N2CCCC2)CC1 C1(CC)CN(C(C2COCCC2(F)F)=O)CCN1C(c1cncc(C(C)C)c1)=O C12(NC(C3C(SC)CCC3)=O)CCC(NC(c3oc(C)nc3C)=O)(CC1)C2 Cc1nc(C)c(-c2nc(C3CCCO3)nn2C2CCCC2O)nc1C N1(C(C2(CCNC(C3(F)C(C)(C)C3(C)C)=O)CC2)=O)CC2(CCNC2=O)C1 Cc1oc(C)c(C(=O)NCC2CC(C)CN(C(c3cc(F)c[nH]3)=O)C2)c1C c1(OC)nc(Nc2nc(Cl)ccc2C(N2CCCCC2CCO)=O)ncc1F c12ccc(c(F)c1)CO2.c1(CNCC(CCC)C)ccccc1OC Cc1cc(C(=O)N=c2cco[nH]2)cc2c1NC(=O)CC2 C1(NC(c2ccsc2)=O)CC2CN(C(C3CCS(=O)(=O)N3)=O)CC2C1 c1(CC)ncc(NC(=O)COC2CC(NC(c3ncncc3Cl)=O)C2)cn1 CC(C(=O)NCC1(CF)CCC1)N(C(=O)CCC1CCCO1)C1CC1 N1(CCCCC2(C)OCCO2)CC(C2=NOCC2)C1 C1(C(=O)OC)CN(Cc2cn(C(C)C(=O)NCc3ccccc3Br)nn2)CCO1 c1(C(=O)NCCOCCCN(C)C(c2coc(O)n2)=O)ccc2c(c1)OCCO2 N1(C(COCCOCC#C)=O)CCC2CC12C(=O)NC(CN(C)C)CO c1(C(CC(=O)OC2CC2C(=O)NCC=CCNCC)C)cccc(F)c1 N1(C(C(CC)=CCCC)=O)CCCC1(CNC(=O)CC(=O)OCC)CC C1(NC(c2cnsc2)=O)CCCCC1CNC(C1CCCC1(F)F)=O c1(OC)cc(Cl)c(C(N2CCC(c3cn(CCO)nn3)(N(C)C)C2)=O)cc1Cl c1(C(c2n(CCCC)nnn2)NCCCC(C)(F)F)ccc2cccc(C)c2n1 c1(C(N(CCCCNC(c2nc(CC)sc2)=O)C)=O)cc2n(n1)CCCC2=O C1(OC)(OC)CC(CNC(c2csnc2C)c2nnnn2CCCSC)C1 CCCC(CNC(C1CCCCC1OCC(F)(F)F)=O)C(=O)O C1(N(C)C(C2CC(C)(C)CN2C)=O)CCC2CN(C(=O)Cc3cnoc3)CC12 C#CC1(NC(=O)CCC2(C)CCCN2C(C2CS(=O)(=O)C2)=O)CC2CCCC12 C1(O)(C(C)NC(=O)CCc2cccs2)CCN(C(c2c(N)cccc2Cl)=O)CC1 N1(C(C(c2ccccc2)OC)=O)CC2(C1)CN(c1cc(O)ncn1)C2 c1(C(=O)NC2(CF)CCN(C(CC(CC)C)=O)C2)ccc(F)c2ccsc12 OC1CC2CC1CC2CN(c1cccc(C(F)(F)F)c1)C1CC2(CNC2)C1 C1(CC=C)(NC(=O)CCOCC)CCN(C(=O)CNC(=O)C(F)(F)F)C1 c1(C(N2CC(NC(C3CC(C)(CC)C3)=O)C2)=O)cncc(-n2cccc2)c1 c1(NC(C2C(C(=O)Nc3ncc(C)c(I)c3)C2)=O)ccc2c(c1)NC(=O)CCC2 c1(CN(C)Cc2cncc(C(N)=O)c2)cc(C#N)cs1 C1(NC(=O)CCCn2cccc2)CCCC(c2ccccc2)C1 N(C(=NCCc1cccs1)NCC1CCC1N(C)C)C(C)Cc1cnccn1 CCCC(C(=O)NCCC1CCOCC1)NC(c1ccc(F)cn1)=O c1(OCOC)ccccc1OC.C1(C(C)C)CNCCC(=O)N1.C1(C)C(=O)N1 N1(C(c2ccc(OCOCC)o2)C(=O)NCC2CCCO2)CCC(C2CC2)CC1 N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(n2nccc2C)C)CC12CC2 c1(C(N(CCN(C(CCC2C(C)C2)=O)C)C)=O)cn(C)nc1C1CCC1 C(C1CN(C(c2sccc2F)=O)Cc2ccccc21)NC(c1[nH]n(C)c(=O)n1)=O c1(C(=O)NC2CC2NC(c2ccc(-c3ccncc3)s2)=O)cc2cccnc2[nH]1 c1(NC(C2C3CN(C(=O)C=Cc4cnccn4)CC23)=O)ccc(F)c(F)c1F N1(C(c2ncc(-c3c(OCC)c(C)ccc3)cn2)=O)CC(O)C(O)C(O)C1CO C1(NC(c2c(C)ncn2O)=O)CC12CCN(C(=O)C(C)OCc1ccccc1)C2 C(=O)(C(O)CC(C)(C)C)N1C(C(C)C)CCC1C(=O)NCCC1COCC1O C1(C(=O)NCC(C(C)C)NC(C2CCCCS2)=O)CCCC(C)CC1 c12nc(ncc1F)N(c1cnn(-c3ccccn3)c1)O2.CC1(CO)CNC1 NS(=O)(=O)c1ccsc1C(N1CC(O)(CNC(=O)CC2CCSCC2)C1)=O C1(NC(C2(CNC(c3ccco3)=O)CC2)=O)CC2CCCCCC12 c1(C(=O)NC2C(NC(=O)C=Cc3cccc(O)c3)CC2)cc2n(n1)CCCC2O CCC(C(N)=O)NC(C1CCN1C(c1cnn[nH]1)=O)=O C1(C(=O)NC2CC(OC)CN(C(C=CCC)=O)C2)CCn2c(C)nnc2C1 c1(C(=O)NC(CC)CNC(c2cn(C)cc2C)=O)coc2ccc(O)cc12 c1(C(C)C)ccc(C(=O)N(C)CCOCCNC(=O)CCc2ccoc2)nc1 c1(-c2scc(NC(c3cncnc3)=O)n2)ccc(O)cc1F C12(C(N3C4C(NC(c5cc(F)ccc5Cl)=O)CC(C4)C3)=O)C3CC(CC13)C2(F)F c1(C(=O)NC2CC(C)N(C(c3ccccc3)=O)C2)ccc2nnn(C)c2n1 c1(C(N(CC(CC)NC(=O)CCC2CC2(C)C)C)=O)cc(Cl)c(F)cc1F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(C)C)NCC(CC=C)(C)CO C1(C(N(CCN(C(C)=O)C)C)=O)CCCN(C(=O)C=CC2CCC2)C1 C1(C(=O)OC)CCN(C(C2C(CNC(c3cc(CO)on3)=O)C2(C)C)=O)C1C FC1CCCCCN(c2cc(-c3cccc(Cl)c3)ncn2)C1 c1(C(N2CCCN(C(=O)OCC)CC2)=O)ccc(C)c(F)c1Br c1(C(=O)NC2CCC(NC(CC(c3cccc(F)c3)C)=O)C2)cccc(F)c1N Cc1ccc(O)cc1C(=O)NCc1cc(C(=O)NC2(C3CC3)CCCC2)ccn1 CCCC(C)CCCC(=O)NCC12CC1CN(C(c1cnc(C(F)F)cn1)=O)C2 C(C)(C(=O)N1CCC(NC(c2cc(CCO)on2)=O)C1)(C(C)C)OC c1(C(=O)NCC(F)CNC(C2(Br)CC2)=O)ocnc1-c1ccccc1 CCCCCCC(C)C(=O)NCCC(C)N(C(=O)C=Cc1cncc(OC)c1)C C12(C=O)CC1CCN2C(=O)CC1CC(OCC)C1.C(=O)(C(SC)NC1CC1)OCC C1(C(=O)NC2CCCC2c2ccccc2C(F)(F)F)CC2CCC1NC2 c1(C(=O)NCCC(C)N(CCC)C)c[nH]nc1CNC(=O)C(O)C1CCCC1 CON(C(=O)C1CCCCN1C(=O)Cc1cncc(C)c1)C1CCCC1 N1(C(c2cc(C)nnc2C)=O)CC2(C=C(C(=O)N3CCC(C)(O)C3)CO2)C1 N1(C(CCCC#C)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 n1(CC)ccnc1C(=O)NCC1C=CC(NC(=O)C=CC(F)F)C1 N1(C(CCC(=O)OC)=O)CCN(C(c2c(C(F)(F)F)n[nH]c2C(F)F)=O)CC1C C(=O)(C(F)CCC(C)(C)C)N1C(C(=O)NC(CC(C)C)C)CC2(CC2)C1 n1(CC(N2CCCCC2CCC2CCCC2)=O)nc2ccccn2c1=O Cc1ccc(C#N)cc1NC(C1CCCC(NC(C2(O)CCC2)=O)CC1)=O N1(C(C2CC(OC)C2)=O)CC2(CNC(=O)C(C(C)(C)C)SC)CC(F)(C1)C2 CC1(C)CCCC(c2cccc(CNC(=O)NC34CC3CNC4=O)c2)C1 C1(CC)CCCN(C(=O)CC(C)C(F)F)C1C(N1CC(C)(C(N)=O)C1)=O N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2n[nH]c(O)n2)=O)CC1C c1(OC)ccc(CC(=O)NCC(O)CNC(c2sccc2C2CC2)=O)cc1 C1(NC(C(C(C)OC)NC(C2CCC(=C)CC2)=O)=O)C2CCC(F)(F)C12 C(N=c1[nH]c2c(c(=NC3CCC3C3CCCC3)[nH]1)CCC2)c1cc(O)nc(O)n1 c1(OC)ncc(F)c(=NC(=O)c2cccc3c2CCN(S(=O)(=O)CCCl)C3)[nH]1 CCC(C)(CCNC(=O)CC1CCCC(C)C1)NC(c1cn(C)nn1)=O N1(CC)CCN(C(C2C3CN(C(C4CCCSC4)=O)CC23)=O)CC1 CCCCC(F)C(=O)NC(C(=O)NCCCCCF)C(C)OC c1(C(=O)NC2(C(=O)NC(c3onc(CC)n3)CC)CC2(C)C)oc(CC)nc1C C1(NC(=O)CC2(NC(C3CCCCO3)=O)CC2)CCCC(F)C1 C(CC(C(=O)NCC1(F)CC(CNC(=O)C=C(C)Cl)C1)NC(N)=O)SC C(N=c1cc(C(C)=O)nc[nH]1)C1N(C(C2(C=C)CCOCC2)=O)CCC1 C1(O)(CCNC(Cc2nc(CC)sc2)=O)CCN(C(=O)COC(C)(C)C)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(C2CC2(Cl)Cl)=O)C(C)C1 Cc1cccc(Cl)c1C(=O)NC1CC(NC(=O)CS(=O)(=O)N2CCN(C)CC2)C1 N1(C(c2c(CC)cncc2)=O)CC2(C=C(C(=O)N3CCC(CC)C3)CO2)C1 C1(NC(c2nccc(C)c2)=O)C2CC1CN(C(C1CCS(=O)(=O)N1)=O)C2 CC1(C)CN(C(=O)CCN2CCC(O)CC2)CC1NC(c1cc2ccsc2[nH]1)=O N1(C(C2(c3cn(C)nc3)CC2)=O)CCC(C)(NC(=O)Cc2nnc(O)s2)CC1 C=CC1(CC(=O)NC(C2CCCO2)CC)CN(C(=O)CCC(N)=O)C1 C(=O)(C(F)C(=O)N1CCC(N(CC(C)C)C(C2CC2(F)F)=O)CC1)OCC Cc1cc(N2CCC(F)(CF)C2)nc(=NCC2CCC(C(F)(F)F)O2)[nH]1 c1(CC(=O)NCC2CCN(C(C(C)O)=O)C2)ccc(C#N)nc1 CCC(C)(CCC(C)C)C(=O)NCCNC(=O)C(C1CCCCC1)N(C)C C1(CNC(C(C)CC2CCCC2)=O)C(C)CCCN1C(=O)CCCOC(C)(C)C c1(N2CCC(CC=C)(NC(c3cc(C)n(CC)n3)=O)C2)ncc2ccsc2n1 C(=O)(C(CC(C)C)ONC(c1oc(C)nc1C)=O)NC1C(CCOC)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(c2ccc(Cl)cc2)C)cc1N C1(NC(c2ccc(NC)cn2)=O)C2CC(O)C1N(C(=O)C(F)=C(C)C)C2 c1(C(C)=O)cc(C(N2CCC(O)(C(C)NC(C3CCOC3C)=O)C2)=O)ccc1C c1(C(=O)NCC(CNC(C(C)OCCCCCC)=O)C)ccc(SC2CC2)cc1 C1(C2(O)CN(C(=O)Cn3cnc(C(N)=O)n3)C2)(CNC(C(C)(C)SC)=O)CC1 C(=O)(CC(C(F)F)n1cccn1)N(C(CNC(c1n(C(C)C)ccn1)=O)C)C C1(C(N(C2CCCN(C(c3c(OC)cccc3)=O)C2)C)=O)COCCC1(F)F N1(C(CCOC)=O)CC2(CCC(NC(c3nc4ccccc4[nH]3)=O)C2)C1 c1(NCC(C)(C)CCCO)nc(N2CCC(C3CC3)CC2)nc2scnc12 CC1CN2CCN1C(C(=O)NC(CNC(=O)Cc1ccccc1CO)C1CC1)C2 C(=O)(C(F)CCC(C)(C)C)N1CC2C(C(N(C3CCC4CC34)C)=O)C2C1 C1(CNC(=O)Cc2cscn2)CCN(C(c2cc3cccnn3c2)=O)CC1(F)F c1(C(C)=O)cc(C(=O)NC2(CCNC(=O)Cc3csc(C)c3)CC2)oc1C c1(C(=O)NC(CN(C)C)C(=O)NCc2ccnc(F)c2F)ccc2cccnn12 CCC(C(=O)N1CC2C(C(N3CC4(C3)CN(C(C)=O)C4)=O)C2C1)C(F)(F)F N1(C2C(NC(C(C)NC(N)=O)=O)C2)CCCCC1 C1(OC)CC(NC(C2(SC)CC2)=O)CN(C(=O)C=Cc2ccc(C)s2)C1 C1(CC(=O)NC(C)(C)COC(F)F)CCCN(C(=O)CCCSC(C)(C)C)CC1 CCCC(CCC)C(=O)N1CCN(C(c2nc(C)ccc2OCC)=O)C(CC)C1 C12(C(N3CCN(C(c4c(CC)n(C)nc4)=O)C4C3C4)=O)CC(C)(C1)OC21CCC1 N1(C(C=NOC)=O)CC2CCCC2(CNC(C2C3CCCC23)=O)C1 c1(C(=O)NCCC(C)(C)NC(=O)COCC(F)(F)F)c(F)ccc(Cl)c1F C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(=O)COc2ccccc2O)CC1C CC1CN(CCSc2nc(C3CCN(C(=O)OC(C)(C)C)CC3)n[nH]2)CC(C)O1 c1(C(=O)NC(CNC(C2(COC)CCC2)=O)C)ccc(N)c(F)c1F C1(OC)C(NC(=O)CN(C(=O)C=CC2CCCC2)C(C)C)CC12CCC2 S(=O)(=O)(c1ccc(=NCC2(c3ccccc3F)CC2)[nH]c1)N1CCC(C)(CO)C1 C1(C(=O)NC2CC(N3CCCC3)C2)(NC(C2(C)C(C)C2)=O)CC(O)C1 C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(C(C(=O)Nc2ccc(C)cc2)C)CC1 N1(C(CC(=O)OC)=O)C2CCC1CC(CNC(c1cnc(-c3ccco3)s1)=O)C2 C1(C)(CNC(C(C)c2cccs2)=O)CCN(C(C2(c3cccnc3)CCC2)=O)C1 C1(N(C(CC(=C)I)=O)C)CC2CC1N(C(c1ccncc1)=O)C2 C1(C)(CNC(CCOC(C)=O)=O)CCC(NC(c2cc(CC3CC3)c[nH]2)=O)C1 C1(C(=O)NC2C(c3onc(C)n3)C2)CC1C1CN(C(=O)Cc2ccccn2)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)C2CCCC1N(C(=O)CSC)C2 c1(CC)cccc(NC(C2CC(C)CN(C(=O)CC3CCC(O)C3)C2)=O)c1F c1(Nc2scc(C(=O)Nc3ncc(Cl)cc3O)n2)ncnc2sccc12 Cn1ncc(S(C)(=O)=O)c1NC(=O)C(=O)NCCC1CCCN1 CCCC(C)C(=O)NCCC(O)CNC(=O)C=CI C1(C)(CNC(=NCC2CC(OC)C2)NC2CCS(=O)(=O)C2)CCS(=O)(=O)CC1 c1(CNC(c2cncc(O)c2)=O)ccc(CNC(C2CC3(CC3)C2)=O)cc1 CCCCC(C)CCC(=O)N1CCCC(C)(CNC(c2ncn(C(C)C)n2)=O)C1 C1(NC(C(C)C)=O)COC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 O=C(C1=CCOCC1)NC1(C(=O)NCC(O)CC2CCCC2)CC(O)C1 N1(C(C(C)SCC)=O)CC(OC)C(NC(c2ccc(-c3scnc3C)cc2)=O)C1 C1(C(N2CCC(CCNC(c3n(C)c(S)nc3)=O)CC2)=O)CC2(C1)CC2(F)F N1(C(C(C(C)C)N(C)C)=O)CCOC2(CCC(NC(c3nc(=N)[nH][nH]3)=O)CC2)C1 c1(CC)cscc1NC(=O)CN(C(=O)C(=Cc1cscn1)C)C1CCC1 C1(CNC(=O)C2CC2)CC2COCC2N1C(c1cc2ccoc2cn1)=O N1(C(c2c(C)ncs2)=O)CC(NC(c2cnn(C3CCCCC3)c2)=O)CC1C C(=O)(CCC(F)(F)F)N(CC(=O)NCCOCC=C)C N1(C(CN2C(C)CCCC2)=O)CCC(C(=O)N(C2CCC2)C2CC2)C1(C)C C1(C(=O)NCC#C)CC2CCC1N2C(C1CCC(C)(C)C1)=O c1(C(N2C(CNC(C(COC)OC)=O)CCC2)=O)cccnc1C N1(CCNC(c2cc(Cl)cnn2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 c1(C(=O)OCC)c[nH]cc1C(=O)NC(CNC(=O)CSc1cccnc1)C1CC1 C(C(=O)OC(=O)OC)(C1CC1)NC(CC)=O.C12(CCC1)CCC(=O)N2 N1(C(CCOCCC)=O)CCCC(C(=O)NCCC(O)(CC)CC)C1C C(=O)(C1CCCc2c[nH]nc21)NC1C=CCN(C(c2c(C)cc(=O)oc2C)=O)C1 C(=O)(CCc1cccs1)NC1(CCNC(COCCN(C)C)=O)CC1 C1(NC(=O)CCCNC(C2(F)CC=CC2)=O)CCC(F)(C(=O)Nc2ccco2)C1 Cc1ccccc1C=CC(=O)NCC12CC(CO1)N(C(=O)C(C)OCC1CC1)C2 C1(NC(C2CCC3(CC2)CC3)=O)CCC(=O)N(CC(F)(F)F)C1 C(CC(C(C)(C)C)NC(=O)OC(C)(C)C)N(C)C(C1CCCN(CC(F)(F)F)C1)=O c1(C(=O)NC2(CNC(C=CC3C(C)C3(Cl)Cl)=O)CC2)cccc([N+](=O)[O-])c1 c1(N2CCC(CCNC(C3(C)CCOCC3)=O)C2)ncnn2c(Br)ccc12 C1(C(=O)NCC23CC2CN(C(c2nnc(O)nc2O)=O)C3)CC(C2CC2)=NO1 c1(C(N2CCCC(OCC(C)C)C2)C(=O)NC2(C)CC2)ccc2ccccc2c1 c1(-c2n(Cc3ccc(OC)cc3)nc(C3CC34CC4)n2)cc2cc(C)ccc2[nH]1 N1(C(C(Cc2ccco2)NC(COCCOCC#C)=O)=O)CCC(N(C)C)C1 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(F)C1CCC1)C(C)C CCC(CNC(c1cc(C)c(CO)o1)=O)(CC)C(=O)NCC1CCCC1N(C)C C1(CNC(C2C(C)(CC)C2)=O)CN(C(=O)Cn2ncn(C)c2=O)CC1OCC Cc1cc(Cl)ccc1OC(C)C(=O)NC1CCCC1CNC(c1cnoc1C)=O c1(C(=O)NCCOCCN(C)C(C2CC(F)(F)CS2)=O)cccc(C2CC2)c1 C(=O)(C(C)CC(C)C(C)=O)N(CC(=O)N(C(CCO)C(F)F)C)C(=O)OCC CC1=C(C)CC(C(N2CCN(C(c3cncc(N)c3)=O)C(C3CCC3)C2)=O)CC1 S(=O)(=O)(c1cc(NCC(c2cccs2)O)ccc1C)NC C(C(C)C(F)C(=O)NCCCN1CCCC1)NC(c1cncc(OC)c1)=O c1(N2CCC(OCCNC(C3CCCSS3)=O)C2)cc(Cl)nc(C2CCCO2)n1 Cc1cc(CNC(C)(CC(C)C)c2cccc(Br)c2)ccc1P(C)(C)=O N1(C(c2cnc(COC)s2)=O)CCN(C(=O)C(F)F)CC1c1nccn1C C1(CNC(c2cccc(OC)n2)=O)CC2(C1)CN(C(C1CCOC1C)=O)C2 c1(CC(=O)NCC(C(C)(C)C)NC(C(CCC)C#N)=O)cncc2ccccc12 C(c1ccc(F)cc1)=CCC(=O)NCC(CC(C)C)NC(C1C(CCOC)C1)=O C1(NC(C(CC)CO)=O)CCN(C(c2cc(C#N)ccc2C)=O)CC1(C)C N1(CC)CCOC(CNC(c2cc(I)ccc2Cl)=O)C1c1cnn(C)c1 O=C(C1=CCCCCC1)NCCCN(C(c1cnc(Cl)s1)=O)CC1CCCC1 CC1CN(C(c2ccc(C3(F)COC3)cc2)=O)CC1NC(=O)C1CC1.NC=O CC(C)CC(O)C(C)C(=O)NCC(C)C(=O)NCC(C)C(C)C CC(C)CC(C)(O)CNCC(=O)NS(C)(=O)=O n1(CC)nc(C(=O)NC2CN(C(c3cnnn3CC)=O)C2)c(=O)c2ccccc12 C(=O)(CS(=O)(=O)CC)N1CCC(N(C(=O)CC2CCCCO2)CC#C)C1 N1(C(c2c(COC)n(C)nc2)=O)CCCN(C(=O)CCCc2ccsc2)CC1 c1(N(C)CC)ccc(S(=O)(=O)NC2CCC(NCCF)C2)c(Cl)c1 N1(C(C(C)(C)C2CCCO2)=O)CC2OCCN(C(=O)Cc3ccoc3)C2C1 c1(-n2cc(C(N(C(C(CC)NC(=O)CO)=O)C)C)nn2)ccccc1C Cc1ncc(NC(C23C(NC(C4CCN(C)C(=O)C4)=O)C4CC2C3C4)=O)c(C)n1 CC(C)C(CCc1ccccc1)C(=O)NCCN(C)C(c1ccc(N)c(O)c1)=O N1(C(CCNC(C)=O)=O)CCN(C(=O)C(C)(C)F)CC1c1ccnn1C CC(CNC(=O)CC1(O)CCC1)(CO)NC(=O)CCC1CCOCC1 CC1(C)OC2(CNC(c3cc(F)c(Cl)cc3F)=O)CC1(NC(=O)C1=CCOC1)C2 N1(C(CSCCC)=O)CCCC(N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CCF)C1 C=CC1(CNC(=O)CSCCNC(=O)COC(C)=O)CCC1 c1(CC(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(C(F)(F)F)n(C)n1 CC1CN(c2nc(=N)nc(N(C)Cc3ccc(=N)[nH]c3)[nH]2)CC(C)(F)O1 c1(CC(N2CCC(C)(CNC(C(CSC)C)=O)C2)=O)csc2cc(C)sc12 C1(F)(NC(c2ccc(OC)cc2C)=O)CS(=O)(=O)CC12CCC2 C12(CNC(C(CC)CCOC)=O)CCCC1N(C(c1ccccc1O)=O)CCC2 c1(CN(C)C)ccc(C(=O)NC2CCC(C)(CNC(=O)C(C)(C)C)C2)cc1 c1(OC)c[nH]c(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCCC2)cc1=O C1(NC(CCc2n(C)ncc2)=O)CCCC12CCN(C(=O)Cc1ccns1)C2 C1(CC)CC(C(N2CC(=C(F)CNC(=O)CC3COC(C)(C)C3)C2)=O)CCC1=O O(C=C(C#N)C(=O)N1CCCC1CCCNC(c1cc(CC(C)C)c[nH]1)=O)CC CCCCCCN(C)C(C1CCOC1CNC(=O)CNC(C1CC1C)=O)=O N1(C(c2nc(C)sc2)=O)CCC(O)C1C(N1CCC(C(F)(F)F)C1)=O N1(C(c2n(CC)nnc2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1Cl)=O C1(NC(c2ccc(O)cn2)=O)CN(C(c2csc(S)n2)=O)CC2(CCC2)C1 C1(CN(C(C(C)=C(C)C)=O)C)CCCN1C(c1cc(Cl)no1)=O c1(-c2nnc(C)o2)cccc(CNC(C2CC(=O)N(c3ccccc3F)C2)=O)c1 C12(C(N(CCCC#C)C)=O)CCN(C(c3cnc(CC)nc3)=O)CCC1C2 C1(N(C(C2CC3CC3C2)=O)CC)CCCN(C(=O)C=Cc2ncc(C)[nH]2)C1 CN1CCC(C(=O)NCCN(C(c2csc(C(C)(C)C)c2)=O)C2CC2)CC1 C12(C(=O)NCc3cc(C)no3)C(NC(C3CC3C(C)C)=O)C3CC1C2C3 Cc1ccc(O)c(CC(N2CCCC2(C)CNC(c2cc(C)nn2C(F)F)=O)=O)c1 n1(CC(=O)NCC(C)CNC(C2(C)CCC2)=O)nc(-c2cccs2)oc1=O N#Cc1cccc(Br)c1CNC1CC(NC(=O)Cc2cc(F)c(F)cc2Br)C1 C(=O)(C1CCCc2nnn(C)c21)NC(C)C(C)NC(=O)CC(=O)NC1CC1 CC(C(C)(C)C)=CC(N1CC(F)(CN(C(=O)CCCOc2ccccc2)C2CC2)C1)=O Cc1c(C(C)(C)C)o[nH]c1=NC(=O)NC(C)CN(c1cccc(Cl)c1)C c1(C(N2CCC(C)(NC(C3CC(OCC)C3)=O)C2)=O)c(F)ccc(OC)c1OC CCC(CC(C)C)C(=O)NCCC(C(C)C)NC(C1CNC(=O)CC1(C)C)=O n1(CC=C)cccc1C(=O)NC1CCCC1CNC(c1scnc1C1CC1)=O C(C)(C)(C(C)NC(c1ccnn1CC1CCC1)=O)NC(COCCC)=O c1(OC)nc(C)c(C(=O)NC2CCC(N(C)C(C3CC(CCO)C3)=O)C2)s1 CC1(n2cc(CCCCNC(=O)COc3cccc(CO)c3)nn2)CCOCC1 c1(C(C(=O)NCCC#C)NC(=O)C(C)NC(N)=O)cnn(C)c1 N1(C(CCOCCN(C)C(C2CC2(C)C(F)F)=O)=O)CCc2ccc(O)cc21 Cn1cc(-n2cncc2C(=O)NCCCNC(=O)CNc2nccs2)cn1 c1(NC(c2ccc(-c3cn[nH]c3)cn2)=O)ncc(F)cc1O C1(NC(=O)C=Cc2cscn2)COC2(CCN(C(c3ccccc3CO)=O)C2)C1 C=C(C)CCC(c1nnnn1CCOC)NCC1CCN(C2CCCC2)CC1 c1(C(=O)NCC(=O)NCC2CCC2NC(=O)CC2CC=CC2)cc(O)cc(=O)o1 c1(C(=O)NC(CNC(C(C)=C(CC)C)=O)(C)C)cncc2c[nH]nc12 C#CCCC(O)C(=O)N1CCN(C(C2SCCS2)=O)C(C)C1 CC1(C(N2CC3CCC3(NC(c3csc4nnsc34)=O)C2)=O)CCC12CCC2 c1(CNC(=O)CCC2(NC(=O)CCC3CCCOC3)CCC2)cnn(CCO)c1 N1(C(C=CC(C)(C)NC(c2c(CC)nn[nH]2)=O)=O)CCCCC(C)C1 C1(CNC(c2cnc(C)s2)=O)CC12CCN(C(=O)CCn1cc(Cl)cn1)CC2 c1(CNC(Cc2cc(C)on2)=O)ccc(CNC(C2CCC(C(N)=O)O2)=O)cn1 c1(OCC(=O)NC2CCCCC2NC(=O)CCC2CCC2)cc(F)cc(Cl)c1 C12(CC)CN(C(c3sc(SC)cc3C)=O)C(CNC(C3CNC(=O)C3)=O)(C1)C2 c1(NC(=O)C(=O)NC2COC3(CCCC3)C2)ccc2sccc2c1 C(=O)(CC1=CCCCC1)NC1CCC(N(C(c2c(Cl)cncc2Cl)=O)CC)CC1 C(=O)(CCCC(=O)NC1CC(O)CN(C(c2cnoc2C2CC2)=O)C1)OCC Cc1nc(C(=O)NC2(C)CCN(C(=O)CCN3CCCCCC3)C2)ccc1C#N N1(C(c2cncc(OC)c2C)=O)CCC2CN(C(c3ccncc3O)=O)CC2C1 C(=O)(CC(C)(O)COC)N1CC(CCC)C(C(=O)NC(CCC)c2ccco2)C1 N1(C(C(C#C)(C)C)=O)CCN(C)C(C(=O)NCc2ccccc2C)C1 CC1(C(=O)NCC2(CF)CCN(C(=O)CCC[N+](=O)[O-])C2)CCc2ccccc21 CCCC(C)(CC)N(c1nnnn1Cc1cn(C)nc1C1CCC1)CC C1(C(=O)NCCC(=C)CNC(C)=O)CCN(C(=O)C(CC)CC)CC1 c1(CN2CC(OC)C(C(=O)O)CC2)ccc(F)c(F)c1Cl N1(C(C(CNC(C)=O)(C)C)=O)CCC2(CCCC2CNC(C2CC23CC3)=O)CC1 C(C(C(=O)NCC(N1CCCCC1)C)C(C)(C)C)NC(C(c1ccc(C)o1)C)=O N1(C(C(=O)NC(=O)NC)C)CC2CN(C(=O)CC3C(C)(C)C3(C)C)CC2C1 CC(C)C(C)(CNC(=O)C(O)Cc1cn(C)cn1)NC(=O)CCCn1ccnn1 C1(C(C)(C)C)CCC(C(=O)NCCOCCNC(=O)CCCC2CCOCC2)C1 N1(C(c2nncn2C)C(=O)NC(C(=O)OC)C)Cc2nccn2CC(CO)C1 c1(C(=O)NC(C(C)NC(c2cc(CC)nc(O)c2)=O)C)cnc2ccnn2c1C N1(C(C#CCNC(CC2N(C)C(=O)CC2)=O)=O)CCC2(C1)CC2(F)F N1(C(C)=O)CC2(CCN(C(=O)CCc3nnc(-c4ccccn4)o3)CC2)C1 CC1CN2CCN1CC=CC2=O.C1(CCC(=O)N(C)C)CC(C)(C)CO1 N1(C(c2cnn(C3CCCC3)c2)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1 c1(C(C)(O)C(=O)NC2CN(C(=O)C(O)C3CC3)C2)ccc(Cl)cc1 C(=O)(C(C)CC(C)C)NCc1occ(C(=O)Nc2c(OC)nn(C)c2)c1 Cc1cc(C)c(C(=O)NC(CNC(=O)Cn2ccc(C)n2)CC(C)C)cn1 c1(C(N2CC(CCCCNC(COCC(=O)NC)=O)C2)=O)cc(N)cc(F)c1 C1(NC(C(C)SC)=O)C2CC3CN(C(=O)CCc4cnc(C5CC5)o4)C1C3C2 C(c1ccc(SC(F)F)cc1)=CC(=O)NC1CN(C(c2cc(C)sc2)=O)C(C)C1 CC(C)C(C)CC(=O)NCc1csc(CNC(C2C3CCC(F)(F)C23)=O)n1 C1(C(=O)Nc2c(C#N)ccs2)Cc2c([nH]c3ccccc23)CN1C(=O)C=CCBr C1(C(N2CCC(NC(c3ccc(Cl)cc3Cl)=O)(CO)C2)=O)Cc2cccnc2C1 C#CCC(CC(F)F)C(=O)NCC(CC)N(C(=O)Cn1nnnc1C(C)C)C N1(N2CC(N(C(CCc3cc(C(C)=O)c(C)o3)=O)C)C2)CCC2(C1)CC2(F)F N1(C(c2cccnn2)=O)CCC2(CC1)CC(NCc1ncccc1F)C2 c1(C(=O)NCC2N(C(C3(CC(C)=O)CCCC3)=O)CC2)cnc2n1CC(C)CC2 Cc1cccc(-c2nc(C(N3CC(C#N)C3)=O)cs2)c1C N1(C(CC2CC(C)C2)=O)CCN(C(=O)CCCn2cncn2)CC1CC1CC1 N1(C(c2nc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(C(c1occc1C)=O)C3 C(=O)(C(C)Cc1ccco1)N(CCOCCC(=O)N(CC(=C)C)CC)C c1(C(=O)NCC(C(C)C)(C)NC(=O)CC2CCCO2)cnc2ccccn2c1=O c1(NC(C(c2cn(C)nn2)NC(=O)C(=O)C2CCCC2)=O)ccc2c(c1)OCC2 C1(NC(C(C2CCCC2)OCC)=O)CCCC2CN(C(C3COC(C)C3)=O)CC12 CC(C(=O)NC1CCN(C(=O)COC(F)(F)F)CC1F)C(F)(F)F C1(NC(c2n(CC)nc(C)c2)=O)CN(C(=O)CC(C)(C)C2CC2)CC2CCCC12 CCC(CC)(CO)C(=O)NC1CCN(C(c2cc(OC)c(OC)cc2O)=O)CC1 c1(-c2c(C(=O)NCc3cc(C)on3)ncs2)ccccc1C CCC(C(=O)NCc1ccon1)N(C)C(C1CC(C)(F)C1)=O c1(COC)nc(C(=O)N(CCCCCNC(=O)CC2C=CCC2)C)co1 C12CCN(C1)C2=O.c1(NCCNC(C(=O)NC)=O)ccn(C)n1 N1(C(C(C(CC)C)NC(C)=O)=O)C2CCCC1CN(C(=O)C(CO)N(C)C)C2 CCC(C)(C)CC(=O)NCC1CCCN1C(c1[nH]c(C)cc1C)=O C1(O)(CCNC(c2cnn(C(C)C)n2)=O)CCN(C(=O)CC2(O)CCCOC2)C1 C1(NC(CCc2cc(OC)no2)=O)CCCN(C(c2ccncc2)=O)C1C C1(OC)CCC2(C(=O)NCC(CC(C)C)NC(=O)Cn3cncn3)CC12 N1(C(C#C)=O)CCCC2(CNC(c3cc(F)cc(Br)c3C)=O)CCCC12 Cc1[nH]nc2c(C(=O)NC3(CNC(=O)CC=C(Cl)Cl)CCCCC3)cccc12 c1(C(N2CC(c3ccccc3)(NC(C3C(C)(C)COC3)=O)C2)=O)ccc(O)c(F)c1 C1(C(=O)NCC2(C(=O)N(C3CC(O)CC3O)CC)CC(=C)C2)CCC(=O)NC1 Cc1ccc(C(N2CCC2CNC(c2cscc2C(N)=O)=O)=O)c(=O)n1C N1(C(C(C)(C)OCCC)=O)CC2CC(C(N3CC(C(N)=O)C4(CC4)C3)=O)CC2C1 Cc1cnc(C(N2C3CC2CN(C(=O)C(c2cnn(C)c2)O)C3)=O)cc1Cl Cc1cc(CNC(=O)C(=O)NC(C)(C)C2CC2)cc(Cl)n1.C12CC(C)N(C1)N2 c1(C(=O)Nc2c(C)nc(Br)cc2)cn2c(n1)CN(C(=O)C=Cc1cnc[nH]1)CC2 C(=O)(CCCCC(C)C)N1C2CN(C(CCCCCOCC)=O)CC1C2 c1(OC)cccc(I)c1C(=O)Nc1ncc(CCNC(=O)CCC(C)C)s1 CCC(C)(C(N)=O)NC(C1CCCC(NC(=O)CCc2ncccn2)C1)=O C1(OC)CC(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C(C)C)SC)C1 N1(C(C2OCCC(=O)C2)=O)CC2(C1)CN(C(c1cnsc1)=O)CCO2 c1(CC)ccc(C=CC(c2ncc(I)cc2Br)=O)cc1 C1(C)(CC)CC(NC(=O)C(F)F)CN1C(=O)CCCCCc1ccccc1 CCCC(C)CC(=O)NCC1(O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 c1(C(C)(C)CNC(=O)Nc2ccccc2)ccc([N+](=O)[O-])cc1 C(=O)(CC(C)(C)C(=O)NC1CCCCC1NC(C1CCCCS1)=O)OCC C1(C(=O)Nc2cn(CC(N3CCCC3)=O)nn2)CCc2ccccc2C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)cc(N)cc(F)c1 CCCCCC(F)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)C1 c1(C(N2CC(COC)(NC(C3CC(C)=NO3)=O)C2)=O)cc2sc(C)nc2[nH]1 c1(COC(C2NC(=O)CC2c2cccc(Cl)c2)=O)ccc(OCC2CC2)cc1F c1(CC(N2CCC(CCOC)(NC(C(CC#C)C)=O)C2)=O)cccc(C)c1C Cn1nc(O)cc1C(N1CCC(CCn2cc(CCc3nn[nH]n3)nn2)CC1)=O c1(C(N2CCC(NC(CCSCC(C)C)=O)C(F)C2)=O)ccc2nc[nH]c2c1 C1(NC(C(c2cccs2)SC)=O)CC(F)(F)CC1NC(c1cnccc1Cl)=O C12(C(N3CC(CCNC(CS(=O)(=O)N(C)C)=O)C3)=O)CCCCC1NC(=O)CC2 c1(C(N2CC3CC2C3NC(C2(F)CCC2)=O)=O)cnn2c1CCCC2 c1(C(=O)NC(C2CCN(C(C3CC(c4ccccc4)C3)=O)C2)C)nn(C)cc1Br n1(CC)ccc(CC(=O)NC(CN(C)C)C(=O)NC2CC(c3ncc[nH]3)C2)n1 C1(C(=O)NC2CC(CCC(=O)NCc3ccc(C)o3)C2)(CC)CCNC1=O N1(C(c2c(NC)cnnc2)=O)CCC(C(=O)N(C2CN(C)C2)C)CC1C c1(NCC23CC(C(=O)NC4COC(n5cccc5)C4)(C2)C3)ccc(OCF)c(Cl)c1 Cn1nc(C(N2CCC(CNC(c3ccc(Cl)nn3)=O)CC2)=O)c2ccccc12 CN(C)S(=O)(=O)N(C)CC(=O)NC1CCCC1NC(c1cc(Cl)ccc1O)=O c1(CC(=O)NCC(C(C)C)NC(c2ccnn2CF)=O)cnccc1C(F)(F)F c1(C(=O)NCC(c2ccccc2)CNC(C2CC(=C)C2)=O)sccc1Br C1(CNC(=O)CC(F)F)CC2CC2N1C(C1CC(=O)N(C2CC2)C1)=O C=C(Cl)C(C)(C)C(=O)NC1CC2(C1)CC2NC(C1(C)CC2CCC1O2)=O c1(OC)ncccc1CC(=O)NC(C1CCCN1C(c1ccncc1Cl)=O)C N1(C(C(SC)SC)=O)CC2CCCC(N(C)C(C3CCS(=O)(=O)C3)=O)C2C1 C=CC(CCC)CC(=O)NCC1CC(C(=O)NCCN(C)CCF)=NO1 c1(NC(C2CC(C)CN2Cc2csc(Br)n2)=O)cc([N+](=O)[O-])ccc1Br C#CCCN=C(NCC12CCC(CC1)CC2)NC1CCN(S(C)(=O)=O)C1 C12(C(N3CC(CC)SCC3)=O)CC(C)(CN1C(=O)CCCC(C)C)C2 N1(C(c2c(CC=C)cccc2)=O)CCCN(C(c2c[nH]cc2CC)=O)CC1C Cc1conc1C(=O)NC1(CCCCNC(=O)Cn2ccc(Br)n2)CC1 N1(C(=O)NC(c2ccc(OC)c(C)c2)C)CCC(C2CC(F)(F)C2)C1 C(=O)(C(C)(O)CC(F)F)N(CCCNC(=O)COCC1CC1)C N1(CCC)CC(C(N2CC(NC(c3nocc3C3CC3)=O)C(F)C2)=O)CC1=O N12CCC(C(O)C1)C2=O.Cc1ccsc1C1CC1NC(=O)C(F)=CCCF N1(C(C(CC(=C)C)OC)=O)CCN(C(c2nocc2Cl)=O)CC(O)C1 C1(C(N(CCCCN(C(c2c(SC)n(C)nc2)=O)C)C)=O)CC(S(C)(=O)=O)C1 c1(NC(N2CCOCC2)=O)cc(C2=CCN(c3ccccc3[N+](=O)[O-])CC2)cs1 c1(C(=O)NCCC2CCC(NC(c3scc(C)c3)=O)C2)cc(C)cc2c[nH]nc12 N1(C(C(C)OCC#C)=O)CCCC(C(=O)NC(C)C)C1 c1(N(C)Cc2cc(C)no2)ncc(N)c2ccccc12 CC1(C)CCN(C(c2ccncc2)=O)CC1C(=O)NCC1(C)CCC(=O)N1 c1(-n2c(=O)c2=O)c(C)cccc1C.c1(S)cccnc1OC.CO C1(C(N(CCC(=O)OCC)C)=O)C2CCN(C(=O)C(c3cncn3C)O)CC12 N1(C(Cn2c(C)nnn2)=O)CCC(CNC(c2ncccc2OCF)=O)C(C)C1 c1(C(N2CC3(CN(C(C(c4ccc(O)cc4)C)=O)C3)C2)=O)cc(Br)cc(Cl)c1O C(C(=O)NCC1CN(C(=O)CC(=O)N(C)C)CC12CC2)(C(C)(C)C)SC c1(C(N2CCCC(N(C(c3nc(C)n(C)n3)=O)CC)C2)=O)c(C)oc(C)c1Br C1(F)(CNC(C2(C)CC2(Cl)Cl)=O)CCCN(C(=O)C(O)c2ccco2)CC1 C(=O)(CCCCCn1cc(C2(C)CCCN2C(=O)C(C)(C)SC)nn1)OCC C1(C(N(C(C)C(=O)NCCCN(C)C)CC)=O)C2CCCCC12 N1(C(CNc2c(OC)cccc2)=O)CCN(Cc2cn(C)nc2C)C(C2CC2)C1 C1(NC(c2cc(C)ns2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC2(CCC2)C1 C1(O)(CN(C(Cc2c(CC)con2)=O)C)CCN(C(c2ccc(CO)nc2)=O)C1 C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(=O)C(O)c1ccsc1 C(C(C)(C)C(=O)N1CCCC(OC(F)F)C1)NC(=O)NC(CCC)COC CC(C)(CCF)C(=O)NCC(O)CC(=O)NCCCC1CCOC1=O c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCOCCC(C)C)c(Br)noc1C c1(OCC)sccc1C(=O)NC(C)CNC(c1ccc(Cc2ccccc2)s1)=O c1(N(C)Cc2c(COC)cccc2)nccc(=NCC2CCCN2C)[nH]1 c1(OC)ccc(CN2CC3C(Nc4ncnc5occc45)C3C2)cc1C#N c1(OC)ccc([N+](=O)[O-])c(NCC2CN(C(C3(CO)CC3)=O)CCCO2)n1 c1(C(N2CC(C(C)NC(c3cn(-c4ccccc4)nn3)=O)C2)C)cnccc1Cl c1(C(=O)NC(CNC(C(CC)CC)=O)CO)c[nH]c2nc(Br)ccc12 C(CC(O)CC(=O)N1CCC(F)(CNC(=O)C(C)NC(c2cccs2)=O)C1)SC C=CCC(C)C(=O)NC(C1CCCN1C(c1cc(C2CCC2)nn1C)=O)C C1(CC(=O)NCC2(C(C)(C)O)CN(C(C3(CO)CCCO3)=O)C2)CCS(=O)(=O)CC1 CC(CCCc1ccccc1)C(=O)NCCCN(C)C(C1CC1OC(C)(C)C)=O CCC(C(=O)NC(C1CN(C(=O)C(C)n2cncn2)C1)C)OC1CCCCC1 c1(CN(C)Cc2cn(CC3(Cl)CC3(F)F)nn2)ccc(C(F)(F)F)cn1 c1(CC)ccc(Cl)c(C(=O)NC2CC(F)CN(C(=O)Cc3ccoc3)C2)c1 c1(CCCC)nc(C(N2CC(O)(CCNC(=O)CC(C)SC)C2)=O)cs1 C1(OC)(CNC(=O)CN2CCC2)CN(C(C2(C)CC(=O)C2)=O)C1 C1(NC(C2CN(C(N)=O)C2)=O)CCOCC1NC(=O)Cc1cc[nH]c1 c1(C(=O)NCC(CO)NC(C2C(F)(F)C23CC3)=O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(Cc2cccnc2)CCCO)C2Cc3c(Cl)cccc3C12 c1(CC2(C(=O)NCC3OCCN(C(C(N)=O)=O)C3)CC2)cccc(F)c1F C1(CC(=O)NC(C(=O)NOCCO)C2CC=CCC2)CCCC(O)C1 C1(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)O)CNC(=O)C(C)(C)C1 N1(C(CCC=C)=O)CCC2CN(C(=O)CCc3nccn3C)CC12 c1(C(N2CCN(C(CC(CCC)C)=O)CC2COC)=O)c(F)ccc(Cl)c1F C(=O)(C(COC)CC(C)C)NCC(C)(C(C)C)NC(CCOC)=O c1(NC(C2CC(N(C)C)C2)=O)cc(C(=O)NC2CC2)ccc1OC(F)F C1(C(N2CC(CC(CNC(C3C(C(C)C)C3)=O)(C)C)C2)=O)(N(C)C)CCCSC1 c1(C(=O)NCC(CNC(CCCNC(C)=O)=O)(C)O)cccc(Br)c1O CN1CCc2cc(C(=O)NC3CC(NC(c4ccc(F)cc4F)=O)C3)sc2C1 N1(C(c2cccc(NC(C)=O)n2)=O)CC(F)(F)CC1C(N1CC(=O)NC(C)C1)=O N#Cc1ccccc1C(N1CCC1C(N1CCC(O)(CC2CC2)C1)=O)=O CCC(F)(F)C(=O)N1CC(CCNC(c2ccncc2C(F)F)=O)(OC)C1 C1(F)(C(=O)NC(CNC(C2N(CC)CC2)=O)C2CC2)C(C)(C)C1(C)C N1(C(C23CCCC2C3)=O)CC2(CCN(NC(c3[nH]cc(CC)c3)=O)CC2)C1 C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2F)(F)F)Cc2nnsc2S1 C(=O)(C(C)(C)c1cnco1)NC(CC1CN(C(CNC(CCC)=O)=O)C1)C CC(C)(C)C(CNC(c1c[nH]c(Br)c1)=O)NC(C1(C)CC2CC2C1)=O C1(C(=O)NC2CC(OCC)C2)CN(C(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(CNc2cccc(-n3cc(C)c(-c4nn[nH]n4)n3)c2)CCC2(CO1)CC(O)C2 C(=O)(C(C(C)CC)NC(N)=O)NC1(C)CN(C(COCC(=O)NC)=O)C1 C(N=c1cc(C)nc(-c2ccccn2)[nH]1)C1CCN(C(C(CC)C)=O)C1 C1(CC(=O)N(CCOCCNC(CNC(=O)OCC)=O)C)C=NN(C)C1=O C1(C(N2C(CN(C(=O)Cc3ccc(N)cc3)CC)CCC2)=O)CCCC(C)(C)C1 Cc1cc(-c2nc(C3CC(O)C(F)C3)n(Cc3ccccc3)n2)c(C)o1 Cc1ccc(CNC(C2CCN(C(c3nn(C)c(C)c3Br)=O)CC2O)=O)c(F)c1 N1(C(C(CC)O)=O)C(C(=O)Nc2cnc(Br)cn2)CCC1C C12(CNC(CC(=O)N(C)C)=O)CC(NC(c3cc(F)c[nH]3)=O)(C1)C(C)(C)O2 C(=O)(CC(C)CC(C)C)N1C(CC(=O)NCC2(OC)CC2)CCCC1 N1(C(c2ccc(OC)nc2NCc2ccccc2)=O)CCc2n[nH]cc2C1 CC(C)(C)C(C#N)C(=O)NC1(CNC(=O)C=Cc2cccc(Cl)c2)CCCCC1 N1(C(c2nc(OCC)sn2)=O)CCCCC1C(C)NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C2(O)CCN(C(C34CCCCC3NC(=O)C4)=O)CC2)(NC(CCSC)=O)CC1 c1(OC)cccc(Cl)c1C(=O)Nc1ccsc1C(=O)Nc1ccc(C)nc1 C1(NC(=O)CSc2ccccn2)CCCCN(C(C2(CO)CCCC2)=O)C1 c1(C(=O)OC)c(NC(C2CCC(NC(C3CCCN3C)=O)C2)=O)ccnc1Cl c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)C(CC)C2)=O)c(F)cc(N)cc1F c1(OCC(=O)NCCC(C(C)C)NC(c2ccon2)=O)cc(F)cc(Cl)c1 C1(NC(C(C)=C2CC2)=O)CN(C(=O)CCC2CCC2)C2(CCCOC2)C1 C1(CNC(C=C(C)C(F)F)=O)CCCCCN1C(=O)CC1COC(C)(C)C1 c1(OC(C)C(=O)NC2CCCC2NC(=O)C(C)CF)cccc(Cl)c1 C1(O)(C(=O)NCC2(C#C)CCC2)CCN(C(c2nccc(C)n2)=O)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NC(CNC(C(C)C1CCC1)=O)C1CC1 CCC(CCC(=O)N1CCCC(F)C1)NC(C1CC2(CC2)CO1)=O C1(C)(C(N2CC(N(C)C(C3CC(F)C3)=O)C2)=O)C=CCC1 N1(C(COCCC=C)=O)CCN(C(=O)Cc2ccsn2)C2CCCC12 N1(C(CC)=O)CC(Nc2nc(OC)cc(OC)n2)C2(CCOCC2)C1 C1(NC(C2CCS(=O)CC2)=O)CCCN(C(C2CC(OC(F)(F)F)C2)=O)CC1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(NC(c2cc(=O)cc[nH]2)=O)C12CC2 CC(C)C(C)(O)C(=O)N(C)CC1CCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC(C)(O)CNC(=O)COc2ccsn2)cnc2ccccn12 CCC(CNC(=O)CCOCCNC(=O)C(O)CN(C)C)CC c1(NC(c2n(CCCOC)nnn2)(C)C2COC2)cc(-c2cccs2)n(C)n1 c1(-c2c(C(N(CC(CNC(C3C(OC)CC3)=O)O)C)=O)c[nH]c2)ccccc1F C1(C(N2CC3(CCN(C(Cc4nc(C)sc4)=O)C3)C2)=O)CC2CS(=O)(=O)CC2C1 C1(CNC(CCC(CC)OC)=O)CC12CCN(C(C1CCCN(CC)C1)=O)CC2 c1(OC)cnc(C(=O)NCC2CCCN(C(C3CC4CCC3C4)=O)C2)nc1 c1(C(=O)NC2(C)CCN(C(CCCCCN(C)C)=O)C2)noc2ccc(Cl)cc12 C(CC(C(C)(C)C)N(C)C(=O)NC)OC.c1(C(C23COCC2C3)O)ccc(F)cc1 c1(CC(N2CCC(NC(c3cc(CO)[nH]n3)=O)C(O)C2)=O)nc2c([nH]1)CCCC2 Cc1nsc(C(=O)NC(C)CN(C(=O)CC2CC(O)C2(C)C)C)c1N CC1(C)C2CC1CN(C(=O)COC1CN(C(C3CC(C)(O)C3)=O)C1)C2 c1(CC)c(C(=O)NC2CC(C)(CNC(=O)CCC(=O)N(C)CC)C2)cccc1F c1(C(N2CC(C)C(CNC(c3cccc(F)c3F)=O)C2)=O)cc(O)cc(O)n1 CCCC(C(O)C(=O)N1CC(N2CCCCC2)C1)NC(=O)C=CC(F)F Cc1c(Br)ccc(F)c1C(N1CCC1C(N1CC(F)(C(=O)N(C)C)C1)=O)=O Cc1oc2nc(Cl)ccc2c1C(=O)N(CC(O)CNC(C1OCCO1)=O)C C(=O)(C1=CC2CCCCC12)NC1(C)CC(NC(c2ccc([N+](=O)[O-])c(O)c2)=O)C1 c1(C(N2CCC(CNC(CC3(C)CC3)=O)C2)=O)ccc(Cl)c2occc12 c1(C(=O)NCC(=O)NCC(C)NC(c2ccno2)=O)cccc(O)c1 CON(CCC(=O)NCC1CC12CCOCC2)C(=O)C1(C)CC(C)(C)C1 O=C(N=c1cc(Oc2ncc(Br)cn2)[nH][nH]1)c1cc(F)ccc1OCC(F)(F)F c1(C(N(CCC2N(C(c3cc(C)no3)=O)CCCC2)C)=O)c(C)cc(Cl)cc1N C1(CC(C)NC(c2cc(C)sc2)=O)CCN(C(=O)CC(C)O)CC1 N1(C(CCNC(CC2CCC(C)C2)=O)=O)CCNC(=O)CC1 Cc1ccc(C(=O)C(=O)NCC(C)NC(=O)CCC2CCCO2)cc1 C1(C(N2CCN(C(C(=O)OC)=O)CC2)=O)COCCN(Cc2cccn2C)C1 c1(CC(=O)NC2CN(C(C3C(c4cn(C)nc4)CCO3)=O)C2)cnccc1Cl C1(C)(CC)C=C(C(=O)NCC(=O)NCC(=O)NC(Cc2ccco2)CO)C1 CCCC(CC)CCC(=O)N1CCCCC1CCNC(=O)CCCN(C)C Cc1cc(F)c(C(N2CCC3C(C2)CN3C(=O)Cc2cc[nH]n2)=O)cc1Br c1(CC)oc(C(=O)NC(C2CCN(C(C3CC3CC(C)C)=O)C2)(C)C)cc1C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCCC(NC(=O)Cn2nccc2C)C1 c1(OC)ccc(NC(=O)OC(C)(C)C)cc1SC.n12cc(nn1)CC(=O)N2 c1(C(=O)NCC=CCNC(CCCCSC)=O)nc2c(Br)cccn2n1 c1(C(N2CC3(CC(C(N4CCC(F)C4)=O)C3)C2)=O)cccc2ccncc12 C(=O)(C1=CCSC1)N1CC(OCC)(CNC(C2CCC(OC)C2)=O)C1 C12(NC(C(F)=CC)=O)CN(C(c3ccn(C)n3)=O)CC1CS(=O)(=O)C2 c1(OC)cncc(C=CC(=O)NC2C=CCN(C(c3ccoc3Br)=O)C2)c1 c1(OC(C)C)ccccc1C(=O)N(C)CC1(O)CCN(C(=O)CC(F)(F)F)C1 C12=CC=C(C=C1)C2.c1(C(C(=O)NC)N(CCF)C2CC2)c[nH]nc1C c1(C(=O)NCC(CC(C)C)NC(c2c(Cl)cnn2C)=O)ncc(C(N)=O)cc1Cl N1(C(CC(CCC)NC(c2c(CO)n[nH]c2C)=O)=O)CCN(C)C(C)(C)C1 c1(C(=O)NCC2(NC(C=CC(C)(C)SC)=O)CCOC2)cc(C#N)c(N)cc1O N1(C(CC(CC)C2CCC2)=O)CC2CCC1C2NC(c1ccc(OC)cc1N)=O C1(CC(=O)NCC(CNC(C(CCOC)C)=O)(C)OC)CCC(C)(C)CO1 C(CC(C)P(C)(C)=O)NC(c1cncc(-c2cnn(CC)c2C)c1)=O N1(C(C2(CC=C)CCN(C(c3cc(CC)no3)=O)C2)=O)CCC2(CC(OC)C2)C1 n1(CCC)nccc1C(=O)NCC1(NC(=O)CC2CC2(Cl)Cl)CCOC1 CC1(C(=O)NCc2cn(C3CN(C(C4CC(O)C4)=O)C3)nn2)CC2CCC1O2 CN1C(=O)CCCC1C(N1CCOCC1CNC(C12CC(CO1)C2)=O)=O C=CCC(C)C(=O)N1CC(CC=C)(NC(=O)CCCn2ccccc2=O)C1 c1(C(N2C3CC(CN(C(C(C(C)O)N(C)C)=O)C3)C2)=O)cn(C)c(=O)n(C)c1=O C(=O)(C1CCCc2n[nH]cc21)N(C1CCN(C(c2cnc(C)nc2)=O)CC1)C n1(CCC)nnnc1C(C1CCCCC1)NCC1(CCC)CCC1 C1(C(N2CCC(C(N(C3CCN(C)C3)CC#C)=O)C2)=O)CCN(C)C(=O)C1 c1(C(C(=O)NCCCSC)N(C)Cc2sccc2Br)cn2cccc(F)c2n1 c1(C(C)(C)Nc2c(C)cccc2)cccc(C#N)c1 c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C)C1CNC(=O)CC1(O)CC1)=O C(CO)(C(=O)N1CC2COCC2O1)NC(C(COC)C)=O CC1CN(C(C2(O)CCOCC2)=O)CCC1C(=O)N(C)OC1CCCC1 N1(C(C2CCCN(C)C2)=O)CC2CC(NC(C34CC(C)(C3)C4)=O)CC1C2 N1(C(C=CC(CC)=CC)=O)CCN(C(c2nccnc2N)=O)C(C)CC1C C(N=c1[nH]c(N2CCc3ccnc(N(C)C)c3C2)nc2c1CSC2)c1c(C)ccs1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1(C)N(C(c2cncc(C)n2)=O)CCC1 c1(OC)ncccc1C(=O)NCCC(Cc1ccccc1)NC(=O)C1=CCCS1 N1(C(c2c(OC)cc(C)s2)=O)CC2(CCCCN2C(c2cc(C)c(C)nn2)=O)C1 C1(NC(C2(OCC)CCC2)=O)C2CN(C(=O)CCCCC3CC3)CC12 C(=O)(C(C)C(=O)N(C)CC1CCCN1C(c1ncc(F)cn1)=O)OC Cc1cnn(CC(=O)N(C2CCC(NC(c3ocnc3C(C)C)=O)C2)C)c1 c1(OC)ccc(O)c(C(=O)NCC(N2CCN(C(c3ccco3)=O)CC2)C)c1 C(C(CO)N=c1nc[nH]n2c(Br)ccc12)NC(=O)C=C1CCC1 C(=O)(C(F)CC(CC)CC)N1CCC(CNC(CCC=C)=O)(CO)CC1 c1(C2C(C(=O)NCC(CNC(c3cc(C4CC4)on3)=O)OC)C2)ccc(C)cc1 c1(NC(C2N(c3nccc(OC)n3)CCOC2)=O)nc(Cl)ccc1O c1(C(=O)NCC(CNC(C2CCS(=O)(=O)CC2)=O)OC)nn(C)c(N)c1C Cc1c2c(-c3cnc(C(=O)Nc4cccc(CCO)c4)nc3)cccc2nn1C c1(C(=O)NCC2CC(NC(C(CC=C)C)=O)C2)cc(O)nc(CC)n1 CCS(=O)(=O)CC(=O)N1CCC(C2CCCN2C(c2cc(Br)n[nH]2)=O)C1 CN1CCCC1C=CC(=O)NCC(C)(C)NC(C1C=CCCC1)=O N1(C(C2CC2C(F)F)=O)CCN(C(c2snc3ccccc23)=O)C2(CCC2)C1 C1(NC(=O)Cn2cccn2)CC12CCN(C(=O)CC1CCOC1)C2 N1(C(CCCC(=O)NC)=O)CCC(F)(F)C(CNC(C2CCN2C(C)(C)C)=O)C1 c1(C(=O)OC)cc(C(=O)O)cc(S(=O)(=O)NC2(CC(F)F)CC2)c1 c1(OCCCC)ccc(C(=O)NCC2(O)CN(Cc3csnn3)C2)cc1 Cc1occc1C(=O)NCC1CCN1C(=O)C(C)c1cc[nH]n1 C1(NC(C(CN(C)C)O)=O)CC2CCC1(NC(=O)CNC(c1cccnc1)=O)C2 c1(C(N2C(CNC(c3cccnc3O)=O)COCC2)=O)ccc2c(c1)CCCO2 N1(C(C(=O)NC2COC(C(F)(F)F)C2)=O)CCCc2ncccc21 C1(C)(C(N2CC(NC(c3cc(C)ncn3)=O)C3(C2)CC3)=O)CCCCNC1=O C1(NC(CC=C)=O)CN(C(c2cc(N(C)C)nc(Cl)c2)=O)CCC1O C1(NC(c2c(C)occ2)=O)CCN(C(c2ccc(-n3ccnc3O)cc2)=O)C1C C1(CNC(c2cc(C)[nH]n2)=O)CCCCN1C(=O)CCC1(C)CCC(=O)N1 c1(N2CC(OC)(CNC(c3c(C)ncn3C)=O)C2)c(C)cncc1[N+](=O)[O-] C=CCC(CC(=O)N1CCOCC1CCO)NC(=O)Cc1cccc(O)c1 CCC(C)(CO)C(=O)N1CCCC(CCNC(=O)Cc2cnc[nH]2)CC1 C1(CC)CCN(C(c2cnccc2C)=O)C(C(=O)NC(C)CN=[N+]=[N-])C1 Cc1ccc(NC(=O)Cc2ccc(Cl)cc2C#N)c(Cl)c1O C(CC(=O)N1CC(NC(=O)C2=CSCS2)C1)(C(F)(F)F)OC C(=O)(C(C)=Cn1ccnn1)NCC12CN(C(CC(=C=C)C)=O)C(C1)CO2 c1(C(=O)NCC2C(NC(c3cc(-c4ccncc4)on3)=O)C2)ncccc1F C(=O)(C(C)C(C)NC(c1sc(F)cc1C)=O)NC(C1CCCCC1)CCC C(C#Cc1cccnc1)NC(N(c1ccc(F)cc1)C(C(C)C)C)=O CCC(CCOC)C(=O)NC(C)(CNC(=O)Cc1cc(C)nn1C)C(C)C C(CC)(CS(=O)(=O)c1ccccc1)Cc1[nH]c(=NC(C)C(C)C)cc(CC)n1.N C1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CC2)COC(=O)N1C c1(C(N(C2CCN(C(c3ccc(C#C)cc3)=O)C2)C)=O)cccc(F)c1C#N N1(C(C2CC(C)OC2)=O)CCC(C(O)CNC(=O)CCCN(C)C)CC1 N1(CC(=O)NCCc2nc(C)sc2C)CCS(=O)(=O)CC1c1cnn(C)c1 c1(NC(=O)CSc2cc(F)c(C(=O)O)c(F)c2)ccc2c(c1)OC(F)(F)O2 c1(CC)cc(NC(C2COCC2NC(c2cc([N+](=O)[O-])n[nH]2)=O)=O)cc(F)c1 CC1CN(C(=O)Cn2cnnn2)CCC1NC(c1cc(Cl)n(C)n1)=O CC1(C)CC(NC(=O)COc2cnn(C(C)(C)C)c2)CN1C(=O)CCF N1(C(Cc2c(C)cccc2C)=O)CCN(C(=O)C2=CC(C)C2)C(C)C1C c1(CNC(c2[nH]cc(C)c2)=O)cc(C(=O)NC2(C)CCSCC2)n(C)n1 c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)[nH]nc2ncnc(O)c12 c1(C(=O)NCC2(F)CN(C(C3N(CCC)CCC3)=O)C2)cnn2c1CCCC2C C1(C(N(CCC)CCNC(=O)C(C)(C)N(C)C)=O)CC12CCOC2 c1(CCC)cc(C(=O)NCC2COCCN2C(=O)Cc2ccccc2C)ccn1 c1(OC(C)C)cnc(N(C2CCCN(C(=O)C=CI)C2)CCO)nc1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)COc2ccccc2Cl)c(C)cn1 c1(CC(N2CC3C(NC(c4c(C)nsc4)=O)C(C3)C2)=O)c(C)oc2ccccc12 C(=O)(NN=c1[nH][nH]c(=Nc2ccccc2Cl)s1)c1ccc(C(N)=O)nc1 C#CC1(O)CCCN(C(=O)CC2CCN2C(=O)CN(C)C(=O)OC)C1 CCCC(C(=O)OC)C(=O)N1CC=CC1C(=O)NOCCCCC1CC1 c1(OC)ccc2cc(N(C(=O)NCC3CCSC(C)C3)CC#N)[nH]c2c1 c1(OCCN(C)C)c(C(N2CCCC(C3CC(N)CCO3)C2)=O)cccc1N c1(C(=O)NCC(C)(CNC(C2CCCN2C2CC2)=O)OC)ncc(C)cn1 c1(C(N2C(CCNC(C3OCC(C)(C)C3)=O)COCC2)=O)cnc2ccccn12 C1(C(=O)NC(C2CCN(C(c3cn(C(F)F)cn3)=O)CC2)C)SC2C=CC1CC2 N1(C(C(C)(C)C#N)=O)CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC(CO)C1 c1(C(CNC(C=C(COC)C)=O)NC(=O)CC2CSC2)ccc(OC)cc1.C(COC)=C C(C(C)CC(=O)NCCCC1CCOCC1)NC(c1ccn(CCC)n1)=O c1(NC(C23C(CN(Cc4cc(OC)cc(C)c4)C2)C3)=O)ccc(I)c([N+](=O)[O-])c1 C1(NC(Cc2c(OC)cccc2)=O)CN(C(C2COCCN2C)=O)CCC1O Cc1nc(C(C)(C)C)sc1C(=O)NCC(O)CN(C(=O)CCCN(C)C)C C(N=c1nc(O)c2ccccc2[nH]1)C12CCC(NC(C3C(=C)C3)=O)(C1)CO2 CS(=O)CCC(=O)N1CCN(CC(=O)Nc2cccnc2Cl)CC1 C1(C(N(C)Cc2nncn2C)=O)(NC(=O)C=CC2CCCN2C)CCC(C)(C)C1 c1(C(=O)NCC23C(CN(C(C4N(C)C(=O)CCC4)=O)C2)C3)ccc([N+](=O)[O-])cc1 FC1CCCCCC1N=c1nc(N2CCOC3(CCCC3)C2)c2c([nH]1)CCC2 N1(C(C2(C#C)CCC2)=O)CCC(N(C(=O)CSC2CCCC2)C)C(C)C1 C1(CCC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CCCC(O)C1 C=CCC(C(=O)NCCC1CCN(C(c2c(NC)c[nH]c2C)=O)C1)NC(C)=O N1(C(c2c(C)nn(C3CC3)c2)=O)CCCC(NC(=O)CC2CCCC2)C(F)C1 CC1COc2c(C(=O)NC3CCCCC3CNC(=O)CS(C)(=O)=O)cccc21 C1(CCC)CCN(C(C2(NC(=O)C(C)COC(C)=O)CC(O)C2)=O)C1 Cc1ccc2c(c1)CC(C(=O)NC1CN(C(c3ccc(=N)[nH]n3)=O)CCC1F)S2 C1(NC(CNC(=O)NC)=O)CCCC(CNC(=O)CCNC(c2ccsc2)=O)C1 c1(SC)nc(Cl)cc(=NC2CCCC(NC(c3cc(N(C)C)ccc3F)=O)C2)[nH]1 C1(=CCNC(Cn2ccc(C)n2)=O)CCN(C(C2(C#N)CC2C)=O)CC1 N1(C(c2nc(CNC(c3n(CC)cnn3)=O)oc2C)=O)CCOC(C)(C2CC2)C1 CC(C)CC(C(=O)N(C)Cc1cocn1)ONC(C1CCCCC1)=O CC1(C)CC(CC(=O)Nc2cccc(CNC(c3ccsc3)=O)c2)CCO1 C1(CNC(C=C(C)Cl)=O)C2CC1N(C(c1cccnn1)=O)C2 c1(CC(CNS(=O)(=O)CC2CCCOC2)CO)ccc(Cl)cc1 c1(C(N2CCC(CC=C)(NC(=O)C(C)C(C)C)C2)=O)cc(C#N)c(F)cc1F C1(CC)CN(C(=O)C2CC2)CC1NCC1(c2ccc(OC)cc2)CNC1 CC1(F)CC2(CN(C(C34CCN(C(=O)C(=O)NCC5CC5)CCC3C4)=O)C2)C1 C(CC)(CCCC(=O)NCc1cc(C)cnc1F)NC(C1(CCC)CC1)=O C1(CNC(C(P(C)(C)=O)O)=O)CC12CCN(C(c1cc(C(N)=O)cs1)=O)CC2 c1(OC)c(C(=O)NCC2CCN2C(c2cc(C(C)(C)C)n(C)n2)=O)cccc1Cl CC1=C(C(=O)NCc2cc(C(=O)NCC(c3ccccn3)O)on2)SCCO1 c1(-c2c(OC)cccc2)nc(=NC(=O)C2=NN(C(C)C)C(=O)CC2)s[nH]1 c1(OC)c(Cl)nc[nH]c1=NCC1CN(C(=O)CCCCF)CCO1 c1(C(N2CC(C(C)NC(=O)C(O)CCc3ccccc3)C2)=O)cc(O)nc(O)c1 C1(C)(C(N2CC(F)(CNC(Cc3cc(C)sc3)=O)C2)=O)CCC(=O)C1 c1(CS(Cc2cc(C)no2)=O)sc2ccccc2c1C C#CCCC(C(=O)N1CCC(C(N)=O)CC1)NC(=O)CCC1CCC(=O)C1 c1(C(=O)NC2CC(NC(C3CCC3(F)F)=O)C2)cnc(CC2CC2)nc1O c1(-c2cn(CC(N3CC4(CCC(N(C)C)C4)C3)=O)nn2)cccc(P(C)(C)=O)c1 c1(C(=O)NC2CC(CC)(CC)N(C(C34COCC3C4)=O)C2)cc[nH]c2nccc1-2 CC(CC(=O)c1ccccc1F)C(=O)NC(Cc1ccccc1)CO C1(CNC(C(C)C)CCO)CC2(CCC(F)(F)CC2)CO1 c1(C(N2CCC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)cccc(F)c1C(F)F N#CC12C3C4C1C1C2C3C41C(=O)NCC(C1CCC1)NC(=O)CCNS(C)(=O)=O N1(C2CCN(C(C(C)C)=O)C2)CCC(NC(C2(c3nccn3C)CC2)=O)CC1 C=CCCC(C)(C)C(=O)N1CC(O)(CN(C(=O)C(CCCC)NC(N)=O)C)C1 N1(C(=O)CCNS(=O)(=O)c2cccc(Br)c2)CCc2c(O)ccc(F)c2C1 C1(C(=O)NCC(C)NC(c2cnc(C3CC3)[nH]2)=O)CCCC2C1C2(F)F CCC(CC(=O)NC(c1ccnn1C)C(N1CCCOCC1)=O)C1CC1 C(=O)(C1=C(Cl)CCOC1)NCCCOCCN(C)C(C1(C2CC2)CCCCO1)=O CC1=C(C(=O)NC2(CO)CN(C(=O)C(C)(O)C(C)C)C2)CCC(C)(C)C1 Cc1c(C(=O)NC2COCCN(C(=O)C(C)n3ccnn3)C2)sc2nnc(S)n12 C(c1cnn(C)c1C)=CC(=O)N(CCOCCNC(C(n1ccc(C)n1)C)=O)C N1(C(COCN2C(=O)COCC2)=O)CC2(CNC(=O)C(F)(F)CO)CC1CO2 C(CCC(C)(F)F)N(C)C(C1CN(C(c2cccnc2)=O)CCO1)=O C(=O)(C(C)(C)CCF)NCC(C)CC(N1CC2CC2C2CC12)=O S(=O)(=O)(c1cccc(NCc2nc(C#N)cs2)n1)N(CCF)CC C1(C)(C(=O)NC(C)CCN(C(=O)C(C)CF)C)Cc2ccccc2C1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2NC(=O)CCc2cncnc2O)C1 C(=O)(C(C)CCC(C)(C)C)NC(CN(C(c1cc(N(C)C)nc(Cl)c1)=O)CC)C C1(NC(c2cc(C)ncn2)=O)COCCN(C(=O)CCc2ccc(F)cc2Cl)C1 c1(CCC(=O)NCCCN(C(=O)C(Cl)=CCl)C)nc2ccccc2s1 n1(CCN(C)C)cc(C(=O)NC2(CNC(C3CC(CCO)C3)=O)CC2)nn1 N1(C(=O)C2=COCCO2)CC2C3CCC(C2C1)N(C(=O)Cc1ccnc(O)c1)C3 CC1(NC(C2CCCC2N2CCOCC2)=O)CCCN(C(c2cccnc2)=O)C1 CCCCC(O)C(=O)NC1(CO)CCN(C(=O)CC2COCC(C)(C)O2)CC1 CCCCC(CC)NC(C1C=CCCN1C(C1C2CC(=O)CC12)=O)=O C(=O)(C(CNC(=O)CC(C)OC)N(C)C)NCCOC C1(CNC(c2[nH]cc(C)c2)=O)COCCN(C(=O)C(C(C)O)N(C)C)C1 C(=O)(CCCC(C)(C)C)N1C(C(=O)NCCSCCOC)C=CCC1 C1(NC(C=CCN(C)CC)=O)CC2CC1N(C(C1(COC)CCC1)=O)C2 c1(C(=O)NC2CC(CC(N3CCCC(=C)C3)=O)C2(C)C)cc(F)ccc1C C#Cc1cncc(C(=O)N(C2(C(=O)NOCC=CCl)CC2)C)c1 S(=O)(=O)(c1cccc(F)c1C)N1CC2CCN(Cc3nc(OC)c(C)nc3)C2C1 c1(C(N2C(c3c(C)noc3C)CCC2)=O)cc(Br)cc(=N)[nH]1 N#Cc1ccc(C(=O)NCC2CC(C(=O)NCCCN3CCCC3)CO2)cc1 C(=O)(CC1NC(=O)c2ccccc21)N1C(C)CCN(C(COC)=O)CC1 C1(CNC(C(COC)C)=O)CCC(F)(CNC(c2cc(Cl)c[nH]2)=O)CC1 c1(C(=O)NCC2CCC(NC(Cc3c(C)cnn3C)=O)C2)ccn(C)c(=O)c1 C1(CC(=O)NCC(C(=O)NC)O)N(C(=O)C=CC(F)(F)F)CCC1(C)C C1(C(N(C)C)=O)(NC(=O)C(F)=CCCF)CCC1 c1(CNC(C(c2cccc(Br)n2)C)=O)ccccc1OC(F)(F)F N1(C(c2c(C)cc(C)n2C)=O)CCC2(CC1)CC2c1cn(CC2C3CCCC23)nn1 c1(C(=O)NC(CC(C)NC(CCOCCCOC)=O)C)cc(C)cc2c1CCC2 C1(NC(C(c2cn(C)nc2)=O)=O)CN(C(=O)C(N2CCCC2)C2CC2)CC1F c1(CC(=O)NC2CC(NC(C(CC)(C)C)=O)C2)c[nH]c2cccc(Cl)c12 Cn1ccc(C(=O)NC2(C(=O)NCC3(C)CC=CCC3)CC(CO)C2)cc1=O c1(CC(=O)NC2CN(C(C3(CC=C)CC3)=O)CC3C2C3)cccc([N+](=O)[O-])c1C N1(C(c2sc(C)c(C3CCOCC3)n2)=O)CCC(C)(SC(F)F)CC1 CC(C)(O)CC(=O)NC1CCOC(CNC(c2cn(CC(F)(F)F)cn2)=O)C1 C#CCC(CC(F)F)NC(c1coc(CNC(=O)C2=NOC(C)C2)c1)=O c1(C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc2ccoc2c1 Cc1ccc(C(CNC(=O)Cc2cc(C)on2)NC(=O)Cn2ccc(C)n2)cc1 CC(=O)CCCC(C)C(=O)NC(CCSCOC1CCCC1)C(N1C2CCC1C(C)C(O)C2)=O CCCCC(O)C(C)C(=O)NC(C(=O)NCC1CC2(CCC2)CO1)c1ccco1 C1(CNC(C2(OC)CCOCC2)=O)CC2CCCC2N1C(=O)C(C)C1CC1 N1(C(CCC(C)SC)=O)CCC(C(=O)NC2CC2CN(C)C)C12CC2 C1(NC(CC=C=C)=O)CCC2CCN(C(c3ccc(N4CCCC4)nc3)=O)C12 N1(C(c2cnc(C)o2)=O)CC(NC(=O)CN2CC(C)C2)CCC1C C1(C(N(C2CCN(C(C=CCOC)=O)CC2)C)=O)CC(COC)C12CCC2 N1(CC)CCN(C(=O)C(n2cc(COc3ccc(O)cc3)nn2)C)CC1C Cn1c(C(=O)NCC2CC(C(=O)NCc3cncc(Cl)c3)=NO2)ccc1C#N N1(C(Cc2cn(CC)nn2)=O)CCC(C)C1CNC(c1ccc(C)n1C)=O C1(NC(c2n[nH]cc2C2CCC2)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1C(F)(F)F C1(C(N2CCC(C(=O)NCC(F)F)CC2)=O)CCC(=O)N2CCOCC12 c1(OC(C)C(N2CCN(C(=O)CCC#N)CC2)=O)ccccc1Br CC1CCN(C(=O)CCC(C)(C)NC(=O)CSC2CC2)CC(C)O1 CC1OCCOC1C(N1CCOC(CCCNC(c2ccc[n+]([O-])c2)=O)C1)=O c1(CC)ccsc1C(=O)NCc1ncoc1CCNC(c1ccc(C(C)C)s1)=O C1(CC#C)(C(=O)NC(c2cccc(C)n2)C)CCN(C(C2CC23CC3)=O)C1 C(N=c1cc(C)nc(N2CC3C(CO)C3C2)[nH]1)c1c(C)ccs1 Cc1cc(CCC(N2CCOCC2CCNC(=O)CCC(C)N(C)C)=O)nn1C c1(C(=O)NC(CCC)CNC(C2C=CCS2)=O)cccn(C)c1=O CCC(C)C(O)C(=O)N1CC(OCC(=O)NCC2CCC(C)(C)CC2)C1 C=C1CC2(C1)CN(C(C1CCCC(NC(c3ncccc3F)=O)CC1)=O)C2 N1(C(=O)NC2C(NC(=O)Nc3ccccn3)CCC2)CCCc2ccccc21 c1(C(N2CC3CC2C3NC(C2(Cl)CC2(F)F)=O)=O)nc2ccccc2s1 N1(C(C(CSC)(C)C)=O)CCN(C(c2ccc(CCN(C)C)[nH]2)=O)C(COC)C1 CC(C)C(C)CN(C)Cc1ccc(COC)s1 C1(N(C(C=CC=CC)=O)C)CS(=O)(=O)C12CCN(C(=O)C(C)CCC)CC2 c1(NC(c2cnc(C)nc2C(C)C)=O)sc(C)c(C)c1C#N C(=O)(CCC(C)(C)C#N)N1C(C(N2CCC(OC(C)=O)C2)=O)CSC1 C(CCN=C(NCC(C)(C)C(C)(C)O)NC1CCCN(c2cc(C)nn2C)C1)OC N1(C(C2(OC)CC(CF)C2)=O)CCC(CCNC(C2(C3CCCO3)CC2)=O)CC1 CC1CC(C(N2CCC(C(C)C(=O)NC3CCC(CO)C3)CC2)=O)CN1C N1(c2c(C)c(NC(C)Cc3cnc[nH]3)ncn2)CCC(C2CCCOC2)CC1 c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)OC)=O)cc(C)ncc1Br c1(C(N(C(C)CCNC(C2CCCCC2(F)F)=O)C)=O)ccc2c(ccn2C)c1 N1(C(C2CCC3(CC3)N2C(c2ccc(CO)cn2)=O)=O)CCC2(C1)CC2(F)F CCC(CC)(CO)C(=O)NCC1(NC(c2cc(CO)n(C)n2)=O)CC1 C12(C(=O)OC)C3C4C1C1C2C3C41C(N1CC(CO)C(O)C1)=O N1(CC(C)C)CCCC1(c1ccccc1)C(N1CC1)=O C1(C)(CN(C(=O)C=Cc2cocn2)C)CCCC1NC(=O)CN1CCSCC1 c1(C(=O)NCC2CC(NC(CCOCCCOC)=O)C2(C)C)ncc(F)cc1F c1(CC)nc(C)c(C(=O)N(C2C3CN(C(C4OCCC4C)=O)CC23)C)o1 N1(C(=O)CCc2ccc(F)nc2)CCC2(CCN(C(=O)CCc3cocn3)C2)C1 C1(CNC(c2ccc(CC)s2)=O)CCC(C)N(C(C2CCC(O)C2)=O)C1 c1(CCNC(=O)NC2CCC(CCCCC)O2)nc(C)c(C)s1 C(CC(C(=O)NCc1cn(CC(N2CCC(O)(C(F)F)C2)=O)nn1)OC)OC C(c1ccccc1)=C(CC)C(=O)NC1CCCC1CNC(=O)Cn1cncc1C c1(C(N2CCC3C(NC(C4CC4CF)=O)C23)=O)ncc(F)c(N2CCOCC2)n1 Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)Cn1nnnc1C1CC1 c1(C(=O)NCC2N(C(C(CC)C(F)(F)F)=O)CCOC2)ccc2nnn(C)c2n1 c1(C(N(CCN(C(C(CC=C)(C)C)=O)C)C)=O)c[nH]c2ncnc(O)c12 N1(C(C(CCC)(C)C)=O)CCC(C2CCN(C(=O)CCc3ccc(Cl)nc3)C2)C1 c1(C(=O)NCC2(F)CCN(C(c3cncc(OC)c3)=O)C2)cc2c(s1)CCSC2 C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)COc2cccc(F)c2)C(CO)C1 N1(C(CN(C)C(N)=O)=O)CCC(C2(NC(C3CCS3(=O)=O)=O)CC2)CC1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC1(C)C Cn1nc(C(=O)NC2CCC(CNC(=O)CC3CC(C)(C)CO3)CC2)cc1O CN1CCC(N(CCC#N)C(C2CCC(=O)C2)=O)CC1 C1(CNC(C=C(CC)CC)=O)CCCCC1NC(=O)COC1CC(F)(F)C1 c1(C(=O)NCC(CCC)NC(C23CC=CCN2CCC3)=O)cnc2[nH]ccc2n1 C1(CC(=O)NC2(CNC(C=CCN(C)C)=O)CCCC2)OCCC1(C)C Cn1ncc2c1CC(NCC(=O)Nc1ccc(F)c(F)c1F)CC2 C1(N(CC#C)C(C2(C)CC2Br)=O)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 C(CCN(C(=O)CCOCC)C)(C(C)C)NC(C12CC(CCC)(C1)C2)=O c1(C(=O)NC2CC(CC(=O)NCc3c(CC)n[nH]c3)C2(C)C)cc2occc2[nH]1 C1(N(C(Cc2cc(C(C)=O)sc2)=O)CCO)CCCN(C(C2CC(C)=NO2)=O)C1 c1(C(N2CC(C)(F)CN(C(C3CCSC3)=O)CC2)=O)cc2ccccc2c(O)n1 C1(CCNC(=O)CCOC2CCOC2)CCN(C(c2ccco2)=O)C1 C(C)(C)(CCC(=O)NC(C1(O)CCN(C(c2ccc(CO)cn2)=O)CC1)C)OC c1(C(=O)NCc2c(C)c(F)ccc2)ccc2nc(C3=CCCC3)cn2c1 c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cn(C)nc2SC)=O)cc(N)c1 C1(C(=O)NCC#CCNC(Cc2n(C)ccc2)=O)CN2CCN1CC2 C1(C2(NC(CN(CC)CC)=O)CC2)CCCCN1C(c1ccc(C(C)=O)[nH]1)=O c1(C(N2CC3C(NC(CC(COC)C)=O)(CC3)C2)=O)cccc2c1CCC2 Cc1ccc(CC(C)C(=O)NCCC(O)CNC(=O)CC2CC(F)(F)C2)cc1 N1(CCN=C(NCC(=O)NCC=C)NC2CC(=C)C2)CCn2nccc2C1 C1(NC(C(C)=CC=C)=O)CCC(C(=O)NCCSCC)C1 c1(NC(NC2CCCn3nccc32)=O)cc2ccc(OC(F)F)cc2o1 N1(C(CCc2scc(C)n2)=O)CCC(F)(CNC(c2cc(Cl)cn2C)=O)C1 C=C(C)CCCC(=O)NC1(c2ccccc2)CCN(c2ncncc2C#N)C1 N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)CC(C)F)C1 C(=O)(CCC(C)(C)N(C)C)NC(C(=O)NC(C(CO)SC)C)COC c1(C(=O)NCCCNC(c2c[nH]nc2C(F)F)=O)cc(C2(O)COC2)on1 c1(C(=O)NCC2C(C)(C)CCN(C(C(C)SCC)=O)C2)coc2c(Cl)cccc12 Cc1ccc(F)c(CNC(=O)C=CC(C)NC(c2occ3c2CCC3)=O)c1 C1(CC)CN(C(c2ccc(OC)cc2)=O)CCC1NC(=O)CCCC(C)C N12CC(CC(O)C1)C2=O.Cc1ccccc1C1(NC(C2(NC(N)=O)CC2)=O)CC1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCC(C)C1C(=O)NCC#CC1CC1 CC12CCOC(C(N3CCC(NC(c4ncnc(O)c4Cl)=O)CC3)=O)(C1)C2 c1(C(N2C(CCNC(c3c(C#N)scc3)=O)CCCC2)=O)cc2n(n1)CC(F)C2 N1(C(c2n(CC=C)ccn2)=O)CC(NC(C2CCCC2OC)=O)C(C)C1 CCC(C)(CC)C(=O)N1CC(CNC(c2cncs2)=O)OC(C(F)(F)F)C1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C(=CC2CCCC2)C)=O)CC(O)CC1(C)C(=O)NOCCC(C)O C(=O)(C1CCc2ccccc21)NC(COC)CC(=O)N(CC(O)CF)C CC(C)C(C(C)NC(c1ccnn1CC(F)(F)F)=O)NC(=O)CSCC(N)=O C1(C(=O)NCCCN(C(c2cncc(C)n2)=O)CC)CC2CCC1CC2OC C1(C(=O)NCC2C(NC(C3CCC(C)(CC)O3)=O)CCCC2)CN2CCN1CC2 N1(C(C(C)NC(C2CC(N=[N+]=[N-])C2)=O)=O)CC(C)C12CCOCC2 c1(CC(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)cc(Br)ccc1C C12(C(=O)N(c3ccccc3)C3COC3)CCCN(CC1)C2 CCCC(C)(O)C(=O)N1CC(NC(c2cn(C)nc2I)=O)C1 Cc1c(C(=O)NC2CCN(C(=O)CC3OCCO3)CC2O)sc2[nH]cnc(=O)c12 C(=O)(C1=NOC(CNC(=O)CCCC2CCC2)C1)NCCOCC(=C)C N1(C(CCCN2CCCC(C)C2)=O)CCC2(CC1)CC2C(=O)N(C)C N1(C(C(C(CC)CC)C)=O)CCC2(CC1)OC1(CO)CC2(NC(=O)C(C)CF)C1 C(=O)(C#CC1CCOCC1)N1CCC(C(N2CC(C)=C(C)C2)=O)C(C)C1 C1(NC(COCCOC)=O)CCN(C(=O)CC2CCOC(C)(C)C2)CC1F N1(CC(=O)NCC(CCNC(=O)C(C)C2CCOC2)OC)CCC(C)(C)C1 N1(C(COCCC#C)=O)CCC(CN(C)C(C2C(c3ccccc3)C2(C)C)=O)C1 c1(C(c2ccccc2OC2CCC2)N(C)C(c2ccccn2)=O)cccc(Cl)c1F C(CC(C)(C)C(=O)NCC1(C)CCC(NC(C2(C(C)(F)F)CCC2)=O)C1)OC c1(C(=O)NC2C(C(N(CCOC)C)=O)CCOC2)ccc(O)nc1C c1(C(=O)NCC(CC)NC(=O)Cc2ccc(O)cn2)ccc(C)c(Cl)c1F C1(CCOC)(NC(CCC#C)=O)CCN(C(c2nc(Br)c[nH]2)=O)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC12CCC2 n1(CCC(=O)NCC2(O)CC(NC(C3CCSC3)=O)C2)nc(O)c2c1CCCC2 C(C(C)C(F)C(=O)N(CC(C)O)C(C)C)NC(C1C(C(=O)OC)CC1)=O C(=O)(C(C)(C)C(C)NC(=O)CCCN(C)C(C)C)NCCn1c(C)nc(C)n1 c1(C(=O)NCC2C3CN(C(c4on(C)c(=O)c4)=O)CC32)ccc(Cl)nc1N C1(C(N2C(C(=O)OC)C2)=O)CCCN(C2CCSC2C)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC(NC(c2cccc(F)n2)=O)C2(CCC2)C1 c1(C(N(C2CCCC(NC(C(C)=C(C)C)=O)C2)C)=O)cc(F)c(O)c(F)c1 C1(C(N(C2CN(C(C(C)Cc3ccccc3)=O)C2)C)=O)CCCCCN1C C=CCCC(F)(F)C(=O)NCC1CN(C(=O)C(C)CO)CC1(C)C Cc1cccc2cc(C(=O)NCCCNC(c3c(Br)noc3C3CC3)=O)nn12 C#CCC(C)(C)C(=O)N1CCC(NC(=O)CCCCCc2ccccc2)C(F)C1 c1(NC(=O)NC(C2CCCOC2)C(=O)NC)ccc(C(F)(F)F)nc1 N1(C(c2c(C)n[nH]c2)=O)CCC2(NC(C3CCCC(C)CC3)=O)CCCCCC12 c1(CC=C)cccc(C(=O)N(C(C)CNC(=O)CC(c2ccc(F)cc2)C)C)c1 c1(C(=O)NCC(N(C)C(C2(C(C)(F)F)CC2)=O)C2CC2)c(N)cccc1[N+](=O)[O-] c1(N(C)Cc2ccc(C)cc2)nc2c(c(=NCC(C)CC(C)O)[nH]1)COC2 C(C(=O)N1CCN(C(c2ccc(OC(F)F)c(Cl)n2)=O)CC1C)(C(C)(C)C)SC C(CC(C(=O)NCCC1CC(C)=NO1)NC(c1cscn1)=O)=CC C(CCCCCC(=O)N(CC(O)CNC(C1(CCCF)CC1)=O)C)SC C(=O)(C(C)(F)C(F)(F)F)N1CC(COC)N(C(c2oc(CO)cc2C)=O)CC1 CCC(O)C(=O)NC1(CNC(C2CC2C#N)=O)CCCC1 C1(CC(=O)NC(C2N(C(C3(C(=O)OC)CC3)=O)CC2)(C)C)CC(C)(C)CO1 C1(C(N2C(C=C)CCC2)=O)CCN(C(=O)c2cc(C(C)C)nn2C)O1 CC1CN(C(c2ncc(Cl)cc2F)=O)CCCN1C(C1CCC(C(F)(F)F)O1)=O c1(C(N(C)CC2CN(C(c3cnc(O)o3)=O)CCO2)=O)[nH]cc2c1CCS2(=O)=O c1(COC)nccc(=NC2CS(=O)(=O)CC2NC(c2ccc(O)nc2)=O)[nH]1 CCC(C(=O)NC)NC(C1(NC(=O)CC2CCC3CC23)CC1)=O C#CC1(F)CN(C(=O)CC2CCCCN2C(C2CCC2C(=O)OC)=O)C1 CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CCC(=O)N(C)C C(C(COC)C(=O)N1CCC(N2CCN(C(c3cccnc3N)=O)CC2)C1)OC Cc1nc(F)ccc1NC(=O)CC1C=CC(NC(C2CC2OC(C)(C)C)=O)C1 c1(CC)cnnc(O)c1Cl.c12ccc(cc1)NC(=O)C(C)OC(=O)COC(=O)C2 C(CC(C)(C)NC(=O)CC1CC1C(F)(F)F)NC(C1C(C=C)C1)=O C1(C(F)(F)F)(COC(C(CC)F)=O)CCOCC1 C1(C(=O)NCCCS(C)=O)CN(C(c2cnn(CCF)c2)=O)CCO1 C1(C2CCCC2)(NC(C2CC(C)CN(C(=O)C=CCF)C2)=O)CCC1 C1(NC(c2cccnc2F)=O)CC2(C1)CC(NCc1ccc(F)nc1F)C2 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CC(C(F)(F)F)(OC)C2)sc(C)c(C)c1C c1(OC)cccc(CC(=O)NC(C)CC(C)NC(C2CCC(C)C2)=O)c1 C(N=c1[nH]c(=NCC(CO)OC)c2sccc2[nH]1)c1ncc(CC)s1 c1(C(=O)NCc2ccc(C(=O)NC3CCCNC3=O)cc2)cccc2ccnn12 C1(NC(C(C)C2CCC2)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCOCC2 N1(C(C(CCCC)O)=O)CCC2C1CCCN2C(=O)Cn1ncc2cccnc12 CC(C)(C#N)CCC(=O)NC1(C2CC2)CCN(C(=O)Cn2cc(Br)cn2)C1 c1(NC(C2OCCN(C(c3cc(OCC)n[nH]3)=O)CC2)=O)ccc(N=[N+]=[N-])cc1 Cc1ccc2[nH]nc(C(N3CC4(CNC(=O)C=CCO)CCC3C4)=O)c2c1 N1(C(C(CC)=CC)=O)CCOCC1CCNC(=O)C(O)C(C)C CC1CN(C(=O)CCC2CC2)CC(C)C1NC(c1cc(Br)ccc1F)=O CCS(=O)CC(=O)NCC1(OC)CN(c2ccc(COC)cn2)C1 C(=O)(CC(C)C(F)F)NC1(F)CC(CNC(C(C)ON2CCOCC2)=O)C1 c1(C(=O)NCCC2CCN(C(c3sc(F)cc3Cl)=O)C2)ccn2ccnc2c1 c1(C(N(C)CC2(NC(C34CCC3CC4)=O)CC2)=O)nccc2[nH]ccc12 C1(C(N(C)CC2CCCN2C(C2(C)CCCS2)=O)=O)CN2CCN1CC2 S(=O)(=O)(c1cc(C)cnc1N1CCCCC(N2CCCC2)C1)N1CC=C(C)CC1 C1(SCCC(=O)OC)(CNC(=O)C=Cc2ccccc2)CCN(CCOC)CC1 CC1(C)CCCC(C(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)CC1 c1(CN2C(C(=O)Nc3c(OCC)cc(F)cc3)CC3CC32)cc(F)c(Br)cc1Cl c1(-c2cn(C(C)(C)CCN3CCOCC3)nn2)ccnc(CO)c1 CC(CN(C)C)CCC(=O)N(C)CC1CN(C(=O)Cc2c[nH]ccc2=O)CCO1 c1(C(N2C(C(=O)NCc3cn(CC#C)nc3)CCCC2)=O)cccc(C#C)c1C C(=O)(C1=CC2CC(C1)CC2O)N(CC(=O)O)Cc1ccc(Cl)c(Cl)c1 C(N=c1[nH]cnc2[nH]ccc12)C1N(C(C2CCCN2C2CCCC2)=O)CCC1 c1(SC)nc(N2CCC(O)C(C(N3CCOC4(CC4)C3)=O)C2)ncc1F C1(NC(CCCCN(C)C)=O)CC12CCN(C(=O)CC(C)(F)F)C2 c1(OC)cccc2cnc(NC(C3CC3NC(=O)Cc3cccnc3Cl)=O)nc12 c1(C2(O)CC(C(=O)NC(C)CNC(=O)C(=O)NC3CC3)C2)cccc(Cl)c1 c1(Cc2c(F)ccc(C#N)c2)cc2nc(C(=O)O)ccc2o1 N1(C(C(=O)NCC2(NC(=O)OC(C)(C)C)CCOC2)=O)CC2(CCN2C)C1 S(=O)(=O)(c1ccc(NC(c2nnc(Br)n2C)C)nc1)NC(C=C)(C)CC c1(C(=O)NCC2(OC)CCN(C(=O)C(C)NC(C)(C)C)C2)cc2n(n1)CC(F)C2 CCC(C)(C)C(=O)C(=O)NC1(C(=O)NCC2CC(O)C23CCC3)CCN(C)C1 N1(C(c2cccc(-c3cc[nH]n3)c2)=O)CCC2CC1CN(C(C1(O)CCC1)=O)C2 C(C)(CCCNC(=O)C(O)CNC(c1cc(COC2CCC2)on1)=O)OC(C)C N1(C(CCn2c(C)ncc2)=O)CC2CC1CN2C(C12CCC1CC2)=O Cc1ccn(C(C)C(N2CCC(C(=O)NC(c3scnc3C)C)C2)=O)n1 C1(C(=O)NCC(CC)C#N)CN(C(=O)C(C)(C)C(C)(C)C)CC(C)(C)C1 C1(NC(CC(CC)(F)F)=O)CN(C(c2cc3cccnc3[nH]2)=O)CC1C1CC1 N#Cc1ccc(Cl)c(C(=O)NC(Cc2cn(-c3ccccn3)nn2)C(=O)O)c1 Cc1ccc(C(=O)NC2CC(CNC(=O)CC3CC4C=CC3C4)C(O)C2)c(N)c1 N1(C(CC(C=C)CC)=O)CCC2(CC1)CC2CNC(c1conc1C1CCC1)=O O(NC(=O)CC(C)C(C)(C)NC(C1CCCCO1)=O)CCCOCC C1(NC(CCCc2scc(C)n2)=O)C2CC1CN(C(C1CC13CC3)=O)C2 C1(CC(N2C(CNC(C=CC(CC)=CC)=O)CC2)=O)CC2(CCC2)C1 c1(CC)cccc(CC)c1CC(=O)NCC1CC(O)CN1C(=O)CC1(C)CCC1 c1(N2CCC(C(C)(C)NC(=O)COCC3CCCO3)C2)ccc(C#N)nn1 C=C(C)CCC(=O)NC1(CO)CN(C(C2CC3CC2CO3)=O)C1 C1(CC(=O)NCC(CNC(=O)OC)F)CCC(NC(c2ncsc2C(C)C)=O)C1 C1(F)(CNC(c2ccc(C)o2)=O)COCCN(C(c2ccc(CO)c(F)c2)=O)C1 C1(NC(CC(CC)OC)=O)CC2CC(NC(=O)CCCCN3CCCC3)CC12 C1(C(=O)NCC(C)N(C(=O)C(=O)C2CCCC2)C)CCC2(CCOCC2)O1 C1(C(N2CC(O)(C3CCCN3C(C3CC(=C4CC4)C3)=O)C2)=O)CC12CCOCC2 c1(CC(C)NC(C(C2CN(C(C)=O)C2)OC)=O)c[nH]nc1C N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(=O)Cn2nc(C)n(CO)c2=O)C(F)C1 C1(C(=O)NCCC2(O)CN(C(c3cc(Cl)ncc3N)=O)C2)(OC)CCCC(C)C1 CCC(C)C(C)C(=O)N(C)CCN(C)C(c1cnnc(Cl)c1)=O c1(N(C)C)ccc(C23CCC(C2)C3C(=O)NCc2cn(CC(=O)O)nn2)cc1 C12(CCCC1)C(=O)N1CC(C1)OCCNC2=O.C1(C=O)(CO)CC1C.C#CCN C1(CC)CC(C(=O)NC2CC(N(C(=O)CC=CC(C)(C)C)C)C2)C1 CC(CCCC(=O)NCc1cn(C2CC2)nn1)NC(=O)C(C1CC1)N(C)C c1(N(C)C)ncc(C(N2CCC(c3ccccc3[N+](=O)[O-])C2)=O)cc1C#N C1(NC(C(CC)C(F)(F)F)=O)CCC12CCN(C(C1CN(S(C)(=O)=O)C1)=O)CC2 C1(N(C(C(C=CC)O)=O)CCF)CCCN(C(=O)COC(C)=O)C1.CCCCCC C1(F)(C(=O)NC(C=CC(=O)NC(CCSC)CO)C)CC=CCC1 C(=O)(CCCCCN=[N+]=[N-])NCCC(C(=O)N(CC(=C)C)CC(=C)C)O N1(C(c2n(C=C)nnc2)=O)CCC(NC(C2CC23CC(O)C3)=O)C(F)(F)CC1 N1(C(Cn2c(C)cnc2)=O)CC(O)CC1(C)C(=O)NCCC(F)(F)CO c1(C(N2CCC(N(C(=O)C(CO)N(C)C)CCC)C2)=O)ccc(=O)n(CCF)n1 c1(CNC(=N)NC2CCCCC2)ccc(CN2CCCC2)cc1 O=S(=O)(c1ccc(NC2CC3CC(O)C2C3)c(Br)c1)NCC1CC=CC1 c1(C(N(CCCn2cc(C3CC3)nn2)CCC)=O)ccc(-c2cnco2)cc1 c1(C(N2CC(O)(C(C)NC(c3c(CC)nc[nH]3)=O)C2)=O)ccc(N)c(N)n1 C1(CNC(C2N(C)CCC2)=O)COCCN1C(c1ccc(OCCOC)cc1)=O C(=O)(CCS(N)(=O)=O)N1CCC(N2CCC(NC(C3C(OC)CC3)=O)CC2)CC1 C1(NC(=O)C=Cc2ncco2)CC2(CCN(C(c3cc(C(F)F)ccn3)=O)C2)C1 C(C)(C)(CCC(=O)NC(c1nc(C(=O)NC2CN(C(C)=O)CC2C)co1)C)OC c1(OC)ccc(C)nc1C(N1CC2CC1CC2NC(=O)CCOCC(F)(F)F)=O c1(C(N2CCN(C3CCC3)CC2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(C)c1 C1(C(=O)NC2CC3(C(NC(c4c(CC)n(CC)nc4)=O)C3)C2)CN2CCN1CC2 N#CC1CCN(C(=O)CCOCCNC(=O)C(c2ccccc2)F)CC1 C1(C(=O)NCCOCCN(C(=O)C(F)CC2CCC2)C)CC2COCC2C1 C(=O)(C1CSc2ccccc21)NCCC1=CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(N(C(C2(C(N)=O)CC2)=O)CC)CCN(C(=O)C=Cc2c[nH]nc2C)CC1 N1(C(C(C)OC)=O)CC2CN(C(c3ccccc3CCN(C)C)=O)CC2(C)C1 N1(C(C(CCC)CC)=O)CCC2(CCCN2C(c2cnc(C(F)F)cc2C)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCSCC1CCNC(c1ncccc1C(C)(C)C)=O C(=O)(C1CS(=O)(=O)c2ccccc21)N1CC(NC(CC2C(C)(C)C2)=O)C1 C(c1nc2ccccc2o1)=CC(=O)N(CCNC(c1c(C)cnnc1O)=O)CC C1(C(N2CC(CNC(CC(C(CC)C)O)=O)C2)=O)(OC)Cc2ccccc2C1 C(=O)(C1CCc2nccn21)N1CC(NC(c2c(CCC)nco2)=O)CC12CCC2 C1(NC(c2cncc(OC)c2)=O)CC2CN(C(=O)CC(=O)NC3CC3)CC2C1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC(C1)N(C(c1cnc(C3CCOC3)s1)=O)C2 C1(NC(c2cn(C)c(=O)n2C)=O)CC12CCN(C(=O)C#CC1CCOC1)CC2 c1(C(=O)NC2COCCN(C(C(C)(F)F)=O)C2)occ2c1CCCC2 N1(C(C(CC)(C)OC)=O)CC(NC(=O)Cn2ccc3ccccc23)CC(C)(C)C1 c1(-c2ncc(CNC(c3ccsc3)C)s2)ccccc1F N1(C(c2[nH]cc(CC)c2)=O)CCN(C(=O)CSc2ccccc2Cl)CC1 CCC(CC(=O)NCC1(C)CCN(C(=O)C(COC)C(F)(F)F)C1)C(F)F C1(OC)CC2CCC(C1)N2N1C(C=O)C2CC2C1.n1(CC=O)cnnc1 n1(C(C)C)ccnc1C.c1(NC(N(CCN2CCCC2)C2CC2)=O)ccccn1 CC(C)C(C)CN=c1[nH]c(=NCCOC(=N)O)[nH]c2ccc(Cl)cc12 c1(C(=O)NCCCCNC(CCOCC(C)C)=O)cc2c(s1)CCS(=O)(=O)C2 N1(C(C2(C)CC=CCO2)=O)CC2CCCC2(CNC(=O)Cn2cc(CO)nn2)C1 CCC(CC(=O)NCCCCCSC)NC(=O)CC1CC=CCN1C N1(C(C2N(C(C=CCCC)=O)CC(F)C2)=O)CCS(=O)C(C)C1 C1(CC)CCN(C(=O)COC2CN(C(C3CC=CCC3)=O)C2)CCO1 CN1CCOC(C(=O)NCC2(C)CN(C(c3ccns3)=O)CCO2)C1=O c1(CSC)cccc(C(=O)N(CCNC(=O)C(C)CO)CC2CC2)c1 CC(CC(=O)NC1(C2CCCN2C(=O)CO)CC1)C1CCCO1 Cc1nc(CC(=O)NC2CC(NC(c3ocnc3-c3ccccc3)=O)C2)c(C)s1 C=C(C)CC(C(=O)NC(C)Cc1cn[nH]c1)NC(=O)C(C(C)C)SC n1(CC(=O)N(C2CCC(CNC(C(CCSC)O)=O)CC2)C)cccc(C)c1=O C(C(C)(C(=O)NCCOC1CN(C(C2CCN(C)C2=O)=O)C1)OC)OC Cc1nc2c(o1)CCN(C(C1CCCCCN1C(C1CCC=CCCC1)=O)=O)C2 N1(C(C2C(C)(C)C2)=O)CCC(O)(CCNC(=O)C2=CCCCC2)CC1 C12(NC(c3ccc(O)cc3)=O)CCCC1CN(C(c1cc(=O)cc(Cl)[nH]1)=O)C2 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)NC(c1cc(OC)ccc1O)=O)CC c1(OC)ccc(N)c(C(=O)NCCC(C)NC(=O)CCOC2CCCOC2)c1 CCC(N=c1[nH]c(N2CC3CC3(CC)C2)nc2cc[nH]c12)c1cccc(OC)c1 c1(C(=O)NC2C(NC(=O)CCOCC(F)F)CCC2)cn2c(n1)CCCC2 Cc1ccc(C(=O)NCC(O)CNC(=O)C(C)S(N)(=O)=O)c2cccnc12 C1(NC(C2(CNC(c3cn(CC)nn3)=O)CC2)=O)CCCC(C(N)=O)C1 c1(CN(C(C)CN2CCOCC2)C(C)C)cccc(NC(c2ccco2)=O)c1 C1(C)(C(N2CC(NC(C3C=CCC3)=O)CC(C)C2)=O)Cc2ccccc2N1 c1(C(N2CC(NC(CC=C)=O)C(C)CC2)=O)ccc2nc(O)n(C)c2c1 C1(C)(C(=O)OCC=CCCC)C2CC3CC(C2)CC1C3 CCCCC(CC)n1cc(NC(c2cnn(C3CC3)c2)=O)nn1 c1(CC(N2C(CN(C(c3nc(OCC)oc3)=O)C)CCC2)=O)cccc(C)c1Cl C1(NC(c2c(CC)n(C)nn2)=O)CCCCN(C(=O)Cc2cc(C(C)C)no2)C1 C1(CNC(Cn2c(C)cc(C(=O)O)n2)=O)CN(C)CCN1C(=O)Cn1cnnc1O c1(CNC(C2N(C(C)C)C(C)(C)OC2)=O)cc(Br)cc2c1OCC2 C(=O)(C1=CCC(C)CC1)N(C(C)CN(C)C(c1ccc(-n2cnnn2)cc1)=O)C C1(C(C)(C)C)(CNC(CCC=CC)=O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)C1 c1(OC)c(N)c(C(=O)N(CC(C)NC(C2CC2CF)=O)C)cc(Cl)c1Br N1(C(CCN(CCCCC)C)=O)CC2CC2(CNC(c2cc(C(C)C)c[nH]2)=O)C1 C1(C(C)NC(c2ncc(Br)cn2)=O)CCCN(C(=O)COC2CCCC2)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CCOCC1CNC(C1(F)CCCOC1)=O)=O c1(C(c2n(CCOC)nnn2)NCCCC(F)(F)F)noc2c1CCC2 CC1CCC(O)CN1CC(c1ccc(Cl)cc1O)=O O=S(=O)(c1cnc(NCCOc2ccc(F)cc2)c(Cl)c1)NC1CCC2CC12 c1(C(=O)NC2CCCN(C(c3ccn(C)c(=O)c3)=O)C2)c(F)cc(F)c(F)c1F N1(C(=O)Cc2nc(F)c(F)cc2F)CCCC2C1CCCN2C(=O)CC1CCC1 N1(Cc2ncc(OCC)cn2)CCC(NC(=O)Cc2ccc(Cl)c(F)c2)C(C)C1 c1(C(=O)NCC(C(C)C)NC(=O)C=Cc2nnn(C)n2)c(Cl)c([N+](=O)[O-])nn1C C1(NC(c2sccc2Br)=O)CC2(C1)CC(NC(=O)C(c1ccccc1)O)C2 C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CC(C)c1ccncc1 N1(C(C2(C)CCC2)=O)Cc2ccc(C(=O)Nc3cc(Cl)ncc3[N+](=O)[O-])cc2C1 C(=O)(CCCN(C(=O)C(C1CC1)NC(=O)CCCN(C)C)C)OC CC1CC=C(C(=O)N(C(C)(C)CC(N2CC(=O)NCC2C(N)=O)=O)C)CC1 N1(C(C(CSC)(C)C)=O)CCOC2(CCN(C(=O)Cc3sc(C)cc3C)C2)C1 C1(C)(C(=O)NCC(C)(C)NC(C2(F)CCOC2)=O)CC(c2ccccc2)=NO1 CC(CCCC(=O)NCC1C=CCCC1)NC(C1CCN(C)C1)=O c1(C(=O)NC(CNC(C2(c3cc[nH]n3)CC2)=O)CO)cc2ncccc2[nH]1 c1(C(c2n(C3(C)CC3)nnn2)(C2CC2)Nc2cnc(F)nc2)cc(Cl)ncc1F Cn1cc(Cl)c(C(=O)NC2CC3C(NC(C4CCS(=O)CC4)=O)C3C2)n1 c1(C(=O)NCC2C(NC(CCC(CC)CC)=O)C2)cc2cccc(OC)c2o1 c1(C(=O)NC2CCCCN(C(c3n(CC)nc(C)c3)=O)C2)ccc(F)cc1C#N N1(C(COCCN(C)C)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(F)C1 c1(C(N(C)CCOCCNC(=O)Cc2cnccn2)=O)cncc(Cl)c1Cl N1(C(c2ncc(C)cc2C)=O)CC(NC(C2CC3CCC3C2)=O)C2CCCC2C1 C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1snc(Cl)c1Cl)=O C1(NC(CC(C)NC(=O)Cc2ccccn2)=O)CC2CCC(C1)C2O c1(C(N2C(CNC(C3(OC)CC3)=O)CC(C(C)C)CC2)=O)cn2cc(Cl)cnc2n1 N1(C(C2N(C(C)C)CCCC2)=O)C2CCC1CN(C(=O)C(O)C1CCC1)C2 N1(C(CSCC(=O)OC)=O)CCn2c(CNC(=O)C(F)n3cccn3)nnc2C1 C(CCCCCN=[N+]=[N-])NC(C(C)(CO)NC(c1cc(F)cnc1O)=O)=O N1(CC(=O)NC2CCC(NC(C(C)(C)C)=O)C2)CCCS1(=O)=O N1(C(c2n(C)nc3c2CCC3)=O)CCC2C1CCCN2c1ncncc1F c1(-c2cn(CCCC(N3CCOC4CC34)=O)nn2)cccc2[nH]ccc12 C1(C(N(CCOCC=C)C)=O)CN(C)CCN1C(=O)CC(C)(O)C=C C12(CNC(CCOC)=O)CC(NC(=O)CC(C)C(C)C)(C1)C(C)O2 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2)C1C(=O)N(C)Cc1ccns1 c1(OC)cccc2[nH]cc(CC(N3CC(NC(C4CSC4)=O)CC3C)=O)c12 C(c1cccc(O)c1)=CC(N1CCC(NC(c2c(CC)nc(C)o2)=O)C1)=O c1(C(=O)NCC#CC(=O)NCC(F)C2CCC2)cncc2[nH]ccc12 C1(NC(=O)NCC2C(c3ccc(Br)cc3)(C)C2)CCCC2OCCC12 C1(OC)CN(C(=O)Cc2ccc(C)o2)CC1NC(C1CCCN1C(=O)C1CC1)=O O=C1CC(C(=O)NCC(C2CCC2)NCC2(c3cn(CCF)nn3)CC2)=NN1 c1(OCC(=O)N(C2CC(NC(=O)C(C)(C)C(F)F)C2)C)cccc(C2CC2)c1F c1(C(=O)NCC(=O)NCc2ccco2)cccc(-n2cncn2)n1 c1(C(N(C2CCN(C(=O)COc3cccc(C(N)=O)c3)C2)C)=O)coc(C#N)c1 c1(OCC)cccc2[nH]cc(C(=O)NC3CCC(NC(c4ccccc4I)=O)C3)c12 N1(C(c2n(CC=C)ccn2)=O)CCCC(C2CCCN(C(=O)C(F)OC)C2)C1 Cc1ccc(-c2cnc(NCc3cccc(OC(F)(F)F)c3)c(O)c2)c(C)n1 C(=O)(C(O)CC(C)(C)C)N(C(=O)Cn1nc(C(F)(F)F)cc1Cl)C(C1CSC1)C c1(C(=O)NC(CNC(C2CCC(CC)O2)=O)C)nc(C)c(C)[nH]1 c1(C(=O)NC2(C)CC(NC(C3(CCC)CCNC3=O)=O)C2)ccc(C#N)cc1C C(=O)(C(C)(C)C(F)(F)F)N1C2CC(C(=O)NC(C(C)C)C3CC3)C1CC2 C1(NC(CSCC)=O)CN(C(c2cc(OC)cc(Cl)c2F)=O)CC12CCC2 c1(C(=O)NC(CC)CNC(c2cccnc2S)=O)c(C)nn2c(C)cc(C)nc12 C1(C(=O)NC2CC(C)(NC(CC3CCC(C)CC3)=O)C2)C2C3CCC(C3)C12 C1(CC(=O)N(CC(=O)N(CC(C)(O)C2CC2)C)C)COC(=O)C1 C(=O)(CC1CS(=O)(=O)c2ccccc21)N(C1CCN(C(C)=O)CC1)CCO C1(NC(c2c(C(F)(F)F)ncn2O)=O)CN(C(=O)C2=COCC2)C2(CCOC2)C1 C1(NC(=O)OC(C)(C)C)CC12CCC(C(=O)NCc1n[nH]cc1C1CC1)CC2 N=c1cc(C(=O)NC2CCC(NC(=O)Cn3cccn3)C2)c(Br)c[nH]1 C1(NC(CN(CCOC)C)=O)CC12CCN(C(c1csc(C(C)C)n1)=O)CC2 c1(C(=O)NCC(=O)N(CCNC(C(CC)N2CCCC2=O)=O)C)ccccc1C N(C1CCCc2cc(CNC(=O)CC(C)c3cccnc3)ccc21)C(CC(=C)C)=O c1(OC)cc(CC(=O)NC(CNC(=O)C(C)SC)CC(F)(F)F)ccc1Cl C1(C(=O)NC2CC(F)(F)C2)CN(Cc2cccc(F)c2O)CCC1O c1(C(C)C)ncoc1C(=O)NC(C)(C)CCNC(=O)C(F)OC(F)(F)F C1(NC(COC)=O)CCCC(CNC(=O)C(CCSC)OC)C1 C1(NC(c2cnc(C3CC3)nc2)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 C(=O)(C(C)CN(C)N1CCOC2c3ccccc3OCC12)Nc1c(C)cccc1 C1(O)(CNC(c2ccsc2)=O)CCCN(C(C2CCCOC2c2cc[nH]n2)=O)C1 C1(CNC(CCCOCCC)=O)CC2(CCOCC2)CN1C(=O)C(F)(F)CO N1(C(C(CCC)C)=O)CCN(C(c2ccc(Cl)cc2NCCN)=O)CC1C Cc1cccc(O)c1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)n1)=O N1(C(c2scc(COC)c2)=O)CC(CNC(=O)Cc2cnn(C(F)F)c2)C(O)C1 c1(C(=O)NCC(CC)NC(C2CCCN2C2CC2)=O)cc(OC)cc(OC)c1 c1(C(=O)OC)cc(C(=O)NCCNC(=O)COCC2CCOC2)c[nH]1 C1(CNC(c2cc(Cl)c(Cl)c(Cl)c2)=O)CC12CCN(C(C1CSC1)=O)CC2 N1(C(C2C=CC(NC(C(C=C)C)=O)C2)=O)CCC2OCCC2C1 c1(C(=O)NCC2C(CNC(c3nc(C)nc(O)c3)=O)C2)nc2nccc(C)n2n1 CC1(C)CCC(CC(=O)NCC(C(C)(C)C)NC(=O)C2=COCC2)C1 c1(OC)cc(OC)c(-c2cccc(O)c2)cc1CN(CC(=O)N1CCCO1)C C12(C(=O)NCCN(CC(C)O)C(c3c(C=C)cnn3C)=O)CCCC1CC(=O)C2 C1(O)(CCNC(=O)CCC2CC2)CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C(=O)(C(COC(C)=O)CC(C)C)NCC(=C)CCNC(=O)C(C)COC C1(N(C(C(COC)C)=O)C)CCC2CN(C(c3cc([N+](=O)[O-])ccn3)=O)CC12 N1(C(C2(CCN(C)C)CC2)=O)CC2CCC1C1CN(c3nnco3)CC21 CCC1=NOC(C(=O)NCc2cccc(NC(c3scnc3C3CC3)=O)c2)C1 C=CC1(CC(N2CCCC(N(C(=O)CNC(=O)NC3CC3)C)C2)=O)CCCCC1 c1(C(=O)NCCC(C)N(C)C(c2ccns2)=O)csc(-c2ncc[nH]2)n1 N1(C(C2(CC)CCN(C(=O)CC3CC4CC4C3)CC2)=O)CCCC2CC1C2(C)C C(C1=NOC2CN(C(c3c[nH]c(CN4CCCC4)c3)=O)CC12)NC(CCC(=C)Cl)=O c1(N2CCC3(CCN(C)C3)C2)nc2c(c(=NCC3(CCO)CC3)[nH]1)COC2 N1(S(CCC)(=O)=O)CC(C(=O)NC(COCc2ccccc2)CO)CC(F)C1 Brc1ccc2c(c1)OCCN2Cc1cnc2n1CCC2 C1(CN(C(=O)C(F)OC(F)(F)F)CC)CCCN1C(=O)CCN(C)C(C)=O C1(C(N2CC(C)N(c3nc(-c4ccccc4)ns3)CC2)=O)CCOCC12CCC2 C1(C(N(CCOCCC(=O)NC(C(=O)OC)C)C)=O)COC(C)C1 C1(C(=O)NC2CC(C(N)=O)C2)CC2C=CC1C2.c12cccc(c1)NC(=O)CC2 O=C(C(O)C(F)F)NCC1(NC(=O)C(F)(F)Cc2ccc(F)cc2)CCC1 C(C(C)(C)C#CC(=O)NC1(CO)CC2CCCC12)NC(c1nc(C)oc1)=O C(CCC(C)(C)C(=O)N1CCCC(CCF)C1)NC(C(CC)CC)=O C1(C(=O)NC(CCC)C(=O)NC)CCCCCN1C(=O)CC1(C)CCOC1 C1(CC(C)C)CCN(C(=O)C(C2(O)CCCCC2)NC(=O)CSC(C)C)CC1 N1(C(C2CCC(CCC)CC2)=O)CCCCC2(C1)CN(C(c1ccoc1Br)=O)C2 c1(C(=O)NCC(CC)NC(C2(O)CCCCCC2)=O)cc(C)cc(Br)c1 Cc1ncn(C)c(=O)c1C(=O)NCC#CCNC(C1CC2CCC1O2)=O c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2O)ccc(F)c2ccccc12 c1(CC)cc(C(=O)NCC2C3CN(C(=O)C(C)(CC)CC)CC23)ccc1O C1(OC(c2ccc(Cl)cc2)CC)CCC(C)(C)CC1.N12CCCC1C2 c1(C(=O)NC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)cnc2c(c1)CCC2 N1(c2nc(C)nc(C)c2C)CCc2ccccc2C(NC(=O)Cn2ncnn2)C1 N#Cc1ccc(N)c(C(N2CCCN(C(=O)CCS(N)(=O)=O)CC2)=O)c1 C=CC1(C(N2CCC(C(C)C)CC2)=O)CCN(C(=O)Cc2cc(Cl)cs2)C1 C(=O)(C1CCc2snnc21)NC(CCCNC(CCNS(C)(=O)=O)=O)(C)C C(=O)(CCCCC(=O)N1CCCC1CCNC(C1(C)CC1(Cl)Cl)=O)OC C1(NC(c2n(CCOC)nnn2)c2n[nH]cc2Br)CCN(C(=O)OC(C)C)CC1 N1(C(c2ncn(C(C)C)c2)=O)CCCC12CCN(C(c1cccn(O)c1=O)=O)C2 CC(CNC(c1cc(C(F)F)[nH]n1)=O)C(F)C(=O)NC1(C)CCCC1O C1(NC(CCCCC)CNC(=O)OC(C)(C)C)CC2C=CCC(C1)C2 c1(C(=O)NCC(CNC(c2ccnnc2S)=O)OC)ccc(S(C)(=O)=O)cc1 C1(NC(c2ccn(CC)n2)=O)CC2CC1N(C(c1cnn(CCN(C)C)c1)=O)C2 N1(C(C=CC(C)C)=O)CCC1CNC(C1(C2CCCO2)CC1)=O C=CCC(C)(C)C(=O)N1CCC(C(=O)NCc2cc(O)ccc2O)C1 c1(-c2cn(C3CN(C(CC4(N(C)C)CCCC4)=O)C3)nn2)nnc2n1CCCC2 CC(C(=O)N(C)CCOCCN(C(=O)C=CCO)C)C1CCCO1 c1(C(=O)NC(C2CN(C(c3cc(O)ccc3O)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC23CCN(C(C=Cc4nc(C)sc4)=O)CC2C3)cc(N)c(Cl)c(O)c1 C1(F)(NC(CN(CCOC)C(=O)OCCCNC(=O)NC(C)(C)C)=O)COC1 N1(C(C(CC=CC)CC)=O)CC(O)(C2(CNC(=O)CC3C=CCCC3)CC2)C1 c1(COC(C(C)C(C)c2ccccc2Cl)=O)cn2ccccc2n1 c1(C(C)C)ncc(C(=O)N(C(C)CNC(=O)C(C)C2CC2)C)s1 n1(CC(=O)NCCC2CC(NC(C3CN(C(C)C)C3)=O)C2)ncc(O)nc1=O N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)CCc2nccs2)CC(C)(C)C1 Nc1c(C(=O)NC2CCC(NC(c3n[nH]c4c3CCC4)=O)C2)sc2ncccc12 C1(C(=O)NC(C2CCC2)C)CCC2(CN(C(c3ccn(-c4ccccc4)n3)=O)C2)O1 CCC(C)C(C)N=c1[nH]c(CC(N2CCOC(c3n[nH]c(CO)n3)C2)=O)cs1 C1(CNC(C=CC(CC)=CC)=O)CN(C(=O)CN(C)C(c2ccoc2)=O)CC1C C1(C2CCN(C(=O)C(C)(C)C(C)(C)O)CC2)(NC(C(C=CCCC)O)=O)CC1 N1(C(C(C)OCC)=O)CCN(C(C2CC(F)(F)C2)=O)C(CC)C1 c1(C(=O)NC2C3CN(C(CCSCCCC)=O)C(C3)C2)cc(F)c(F)c(F)c1 c1(C(N2C3C(CNC(CC4(OC)CCC4)=O)C(C3)C2)=O)cnc2[nH]cnc2c1 CC1COC(CO)CN1C(=O)Nc1ccc(-c2ccsc2)nc1 c1(C(=O)NCC2COCCN(C(c3cc(C)ns3)=O)C2)ccnn2ccnc12 CC(C)C(C(=O)N1CCC(N(C(=O)C(O)C2CCCC2)C)CC1)n1cccc1 S(=O)(=O)(c1cccnc1NCC1(OC)CCS(=O)(=O)C1)NC1CC2(CC(OC)C2)C1 N1(C(c2nc(CC)oc2)=O)CCC(CC(N2CCOCC2)=O)CC1 C=CC(CC)CC(=O)NCC1(NC(c2ccnc(N(C)C)c2)=O)CCCC1 c1(OC)cc(C(=O)NCC(C)(C)CN(C(=O)Cc2ccc(F)cn2)C)ccn1 CC1(C)COCC(C(N2CC(CNC(c3nn[nH]c3Cl)=O)C(F)(F)C2)=O)O1 c1(C(C)(C)C)nc2cc(NC(=O)N(CCC(=O)O)CCCN(C)C)ccc2o1 C1(C2CC2)(NC(=O)CCc2ccsc2)CCN(C(C2CCNC2=O)=O)C1 c1(OCC)cccc(OCCC(C)C)c1N(C)C(=O)NCc1cc(C)on1 C12CCCC(C1)N(CC)C(=O)C2.C1(NC(CSCC(=O)OC)=O)CC(=C2CC2)C1 Cc1cn(C)cc1C(=O)NC(C)CN1CCN(C(C2(CN(C)C)CC2)=O)CC1 C(C(=O)NC1CCC1NC(=O)CCOCC(C)C)(C(C)C)n1ncc(C)c1 N1(C(c2cc(CCC)ncc2)=O)CCCCCC1CNC(=O)COC1(C)CCC1 O=C(CN1CCCC(O)(c2cnn[nH]2)C1)C1Cc2ccccc21 Cc1ccc([N+](=O)[O-])cc1C(N1CCCC(NC(c2ccc(Br)c(F)c2)=O)C1)=O CS(=O)(=O)c1ccc(N2CCN(C(C3CCCNS3(=O)=O)=O)CC(O)C2)nc1 CC1(C)OCc2cc(C(N3CCOCC3CNC(=O)Cc3ccon3)=O)ccc21 C(C(F)(F)CCC(=O)NC12CCN(CC1)C2)n1cc(-c2ccc(C(C)=O)s2)nn1 c1(CNC(CC(C)NC(N)=O)=O)cccc(NC(=O)Cc2ccccc2Cl)c1 N1(C(C2CCN(C(CC(C)C3CC3)=O)CC2)=O)CCC12CCC(O)CC2 C=CC1(CC(N2CC3CC2CO3)=O)CN(C(c2ccnc(CO)c2)=O)C1 Cc1ccc(NC(C2CC(CNC(=O)CC(C)c3ccncc3)C2)=O)o1 C(CC(O)C(=O)NCC(=C1CN(C(C2CN(C)C(=O)N2)=O)C1)F)N(C)C C1(OC)CC2CC(OC(=O)NC(C)C)C2C1 CC1N(C(C2C3CCC(C3)N2C(C2CCC2C#N)=O)=O)CCC1(C)C CC1CN(C(C2(c3cccc(F)c3)CC2)=O)CC1CNC(c1ncn(C)n1)=O c1(NC(C2CCCN2C(C2CCCN2C(c2cccs2)=O)=O)=O)cccc(I)n1 C(=O)(C1=NOC2COCC12)NCCCCC1CN(C(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C2COCCO2)=O)CC2(CCCCN2C(c2ccco2)=O)C1 C(C)(CCC(=O)NCC(c1ccccc1)NC(c1cc(C)nn1CCO)=O)OC C1(N(C(CCCN(C)C)=O)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC12CC2 c1(C(=O)NOCC(C)NC2CCC2)cc(O)sc1C.C(CCOC(C)(C)C)OC NS(=O)(=O)c1ccc(CC(=O)NC2CCN(C(=O)Cc3ccno3)CC2F)cc1 C1(NC(=O)Cc2ccccc2F)CCC12CN(C(C1SCCCS1)=O)C2 CC(C)C(O)CC(=O)NC1CC(C)N(C(=O)Cc2csc(-c3cccnc3)n2)C1 c1(C(=O)NCC=C(CCC)CCNC(=O)OC(C)(C)C)ccc2c(n1)CCC2 N1(C(CC(C)n2cccc2)=O)CC2CCN(C(C3CCC4(CCCC4)C3)=O)CC12 Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)COCC3(F)CC3)C2)c1C c1(C(N2CC(C)(NC(c3ccc(-n4cccc4)nc3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 C1(NC(COC(CC)C)=O)CCN(C(c2ccc(NC(C)=O)cn2)=O)CC1F CCC1=C(C(=O)NCC2CC(C)N(C(=O)C3=CC(C)C3)C2)SCCO1 N1(C(c2cccc(C#N)c2Br)C(=O)NCCCC)CCN2CC(F)(F)CC2C1 CC1(C)CC(CC(=O)NCCC(F)(F)F)CN1C(=O)C=CC(F)F C1(NC(C2(OCC)CC2)=O)CC1C1CCN(C(C2CCCCN2CC)=O)CC1 C(CC(C(=O)N1CCC(CNC(N)=O)CC1)NC(=O)CC1CCC(=O)CC1)OC O=C1CCN(CC(=O)NC2CCCCC2NC(c2cc(Cl)ccc2Cl)=O)C(=O)N1 C=C(Cl)CCCN=c1cccc(S(=O)(=O)NC2(C)CCC(C)(C)C2)[nH]1 N1(C(CN2CCC(OC)CC2)=O)CC2CC(NC(=O)C(C)(C)NS(C)(=O)=O)C1C2 C1(O)(CN(C(=O)C(F)n2ccnc2)C)CN(C(=O)CCc2cncs2)C1 N1(C(CCCCCCNC(C2CCC3(CC3)C2)=O)=O)CCC2CCC(O)C1C2 c1(C(=O)NC(CNC(c2c(OC)cncn2)=O)C)cc(Br)cc2c1OCC2 c1(C(N2CCN(Cc3c(OC)c(Br)ccc3)C3C2C3)=O)ccc(F)c(F)c1O C(c1ccccc1F)=CC(=O)N(C)CC1(O)CCN(C(=O)Cc2ccc(Cl)s2)C1 N1(C(CNC(CC)=O)=O)CCC(O)(C(C)CNC(c2cnnc(C)c2)=O)C1 C1(NC(=O)CCn2ccnn2)CN(C(=O)Cn2ncnn2)CC12CCC2 c1(OCC(=O)NCCN(C(c2cc(Cc3ccco3)on2)=O)CC)ccn(C)n1 c1(C2C(C(=O)NCc3cn(CC)nc3C(F)(F)Cl)C2)ccc(C)cc1C c1(OC)nc(C(=O)NCC2CN(C(=O)C=CC(C)C)C3CC23)cc(O)n1 c1(C(=O)NCCC2(O)CN(C(C3(CC)CC3(F)F)=O)C2)cc2[nH]nc(C)c2cn1 C1(O)(C(C)NC(=O)COCCN(C)C)CCN(C(C2COC(=O)C2)=O)C1 Cc1nc(C)c(CCC(=O)NCC(C)(C)CC2CC2)c(O)n1.C(=O)(CCCC(F)F)N N1(C(C2CC(C)=C(C)CC2)=O)CCC(NC(c2n[nH]cc2Br)=O)C(C)(C)C1 N1(C(c2c(SC)snn2)=O)CCCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 c12ccc(C)cc1CC(=O)N2.N1(C(CCN(CCC)C)=O)CCCC(C(=O)OC)C1 N1(C(C2(C)C(C)C2)=O)CCCC2CN(C(=O)C=CCN3CCOCC3)CCC12 c1(C(=O)NCC2(O)CC(NC(C3CC(=C)C3)=O)C2)sc2ccc(C)cc2c1C c1(C(=O)NC2CCOC(C(N3CCC(F)(F)CC3)=O)C2)nnc(O)nc1O C1(C(=O)NC2CCC(NC(c3ccc(NC(C)=O)cn3)=O)C2)Cc2nncn2C1 C1(COC(Cc2cccc(OC)c2)=O)CC(C)(C)CC(C)(C)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC2CCC1CN2C(C1CCCC12CC2)=O)=O N1(C(=O)C(C2CCOCC2)O)CC2CCC2(CC(=O)NC2CCC=CCCC2)C1 CC(C)(C(c1nnnn1CC(F)F)NCCC(Cl)Cl)c1ccccc1 c1(OC)cnccc1C(=O)NCCCCNC(C1CCC2(CC2)C1)=O c1ccc2oc3c(c2c1)CCCC3.O=CN=c1ccc(Cl)c(Cl)[nH]1 C1(C)(C(=O)NC2CC(CNC(Cc3c(C)cccn3)=O)C2)COC(C)(C)CO1 C1(CC(N2CC(c3cn(CCOC)nn3)(O)C2)=O)CCN(C)CC1 N#Cc1ccc(C(N2CC(C(F)(F)F)CC2=O)=O)cc1-c1cccnc1 c1(C(=O)NC2CN(C(C(C)CF)=O)CC(C)(C)C2)c2c(nn1C)CCSC2 C1(C(=O)NCC(CO)OC)CN(C(=O)CC2CSCCO2)CC1C(C)C C1(OC)CN(C(c2cnncc2C)=O)CC1C(N1CC(O)C1(C)C)=O c1(C(=O)NCC(n2cc(-c3c[nH]c(C(=O)O)c3)nn2)C)cnn(C)c1S(N)(=O)=O n1(CCC(N2CCN(C(C=CCC)=O)CC(C)C2)=O)nnc2ccccc2c1=O C=CC1(NC(=O)CC2CCCN(C(=O)CC3CCOC3C)C2)CCCC1 c1(CN2CCC(C(=O)OC(C)(C)C)(OC)CC2)c[nH]c(=O)c2ccnn12 C1(NC(c2c(OC)scc2)=O)CC2(CCCN(C(c3ccc(O)nc3Cl)=O)C2)C1 CC1(CCNC(=O)CC2(CNC(c3c[nH]cc3C3CC3)=O)CC2)CCCO1 C1(NC(CCC(=O)Nc2ccccn2)=O)CC2CC(C1)N(C(=O)OC(C)(C)C)C2 N1(C(c2cc(CC)oc2C)=O)CCCN(C(=O)CN2CCCC2C)CCC1 c1(OC)ccc(C(=O)NC2CC(C)N(C(C3CCCC(N(C)C)C3)=O)C2)nc1Cl N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(c2ccc3ncsc3c2)=O)CC(CO)C1 c1(OC)cc(C)c(C(=O)NC2CN(C(c3ccc(=N)[nH]n3)=O)C2)cc1Cl C1(C)(C(=O)NCC2(O)CN(C(c3c(COC)nn(C)c3)=O)C2)CCCCNC1=O C1(C)(NC(COCCC)=O)CCN(C(C2(OC)CCCC2)=O)C1.C(=O)OCC CC1(C)CC(CNC(C2CC(F)(CF)C2)=O)N(C(C2CCOC2(C)C)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCCNC(N)=O)N1CCN(CC)CC1C c1(NC(C)=O)ccc(C(=O)Nc2ccccc2N(C)C)cc1 N1(C(CCC(=C)C)=O)CCC(NC(=O)C(C)OCCc2ccccc2)CC(O)C1 O=C1OCC2CN(CC(c3ccc(Cc4ccccc4)cc3)=O)CCC12 CC1(C)CCCOC1C(=O)NCCCC(=O)NCC1C2CCCCC12 C(=O)(CCC(=O)NC1CCCCC1CNC(c1ncc(OC)cn1)=O)OC C1(NC(C=C(C)c2cccs2)=O)CN(C(=O)CC2C=CCC2)Cc2ccnn2C1 C(=O)(CCCS(C)(=O)=O)NC(C)C(CO)NC(C1CC(n2cnnc2)C1)=O c1(NC(C(N2CCC(C)(CCN)C2)=O)=O)cc(Br)c(F)cc1Cl CC1CCCCCCN1C(c1coc2c1CN(C(c1cn(C3CC3)nn1)=O)C2)=O C(=O)(C(C)(C)C(C)O)N1CCC(C)(NC(C(C)Oc2cnccn2)=O)C1 N(C(=NCC(F)(F)C(C)(C)O)NCC(C)(C)S(C)(=O)=O)C(c1cccs1)C c1(C(N2CCC(NC(COCCCC#C)=O)C(CC)C2)=O)ncnc2ccsc12 C1(NC(CCc2cccc(C)c2)=O)CN(C(c2ccc(Cl)c(O)c2)=O)CC1(F)F N(C1CN(C(=O)Cc2cccc(Cl)c2Cl)Cc2ccccc21)C(CSC)=O C(=O)(C#CC1CCCCC1)NC(c1c(C(N(CCC)CC2CC2)=O)con1)C C1(CC(=O)NC(C)(CNC(c2snnc2C)=O)C2CC2)(CN(C)C)CCCCC1 CCC(C)C(=O)N(C)CCOCCN(C)C(c1cc(Br)no1)=O CC1CCC(CNC(=O)C=C2CCN(C)C2)N(C(=O)Cc2ccc(F)c(F)c2)C1 N1(C(c2c(CNC(c3ccc(CC)[nH]3)=O)nnn2C)=O)CC23CCC2(COC3)C1 C1(F)(CNC(C(Br)=C(C)C)=O)CCC(NC(=O)Cn2cc(C(C)O)nn2)C1 C1(C)(CNC(Cc2n(C)ncc2)=O)COCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 c1(C(=O)NC2C=CCN(C(C(C)C)=O)C2)nc(C(F)(F)F)ccc1F N12CCC(C)(C1)C2=O.c1(C(=O)NC(CC)CSC)ccsc1C(F)F c1(C(=O)NC2(CO)CN(C(c3cnc(C(C)(C)C)o3)=O)C2)ccc(CCO)cc1 c1(C(=O)NC2CCN(C(C3CC4C=CC3C4)=O)CC2)ccn2ncnc2c1 C(C1CCOC1)=CC(=O)NCC1(O)CC(CNC(C2CNC(=O)N2)=O)C1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(=O)COCCO)CCC1(C)C)C2 O=C1CN(Cc2nc(F)ccc2Br)C(=O)N1CCOCCO.C1CC1 Cc1nc(CSCC(=O)N(C)CCNC(c2cn(-c3ccccc3)nn2)=O)cs1 CC1CC(NC(c2c(C3CCC3)cnn2C)=O)CN1C(=O)C(C1CCC(=O)N1)C N1(C(CCOCCOCC)=O)CCC(CNC(=O)C(F)OC(F)(F)F)C(CC)C1 c1(C(N2CC(CC)N(C(C3C(F)(F)C34CC4)=O)CC2)=O)cn2ccc(C)cc2n1 C1(O)(COC)CCN(C(=O)C(C2CCCO2)NC(=O)CC2(N(C)C)CC2)C1 Nc1cc(C(N2CC3CC3(NC(C34COCC3C4)=O)C2)=O)cc(O)c1Cl c1(C(N2CC(CN(C)C(C3CCCC3O)=O)C2)=O)cc(C(C)(C)C)no1 Cc1ccc2c(=NCCN(C)C(C)C)[nH]c(N3C4CNC(=O)C34CCC)nc2c1 N1(C(C(CC)(C)F)=O)CCC(F)C(NC(c2cnc(C3CC3)nc2)=O)C1 C1(CNC(C2C3CC4C(C3)C24)=O)CN2CCCCC2CN1C(=O)CC1CC1 N1(C(C(C)N2CCCC2)=O)CCC(NC(C2(C)CCSCC2)=O)C(C)C1 n1(CC(=O)NC(C2CCCN(C(c3cc(CO)on3)=O)C2)C)ncccc1=O C=CCC(CNC(=O)C(C)=C(C)CC)C(=O)N(CC(C)(CO)CO)C C1(COC(=O)CC2(NC(C(=O)NC3CC3)=O)CCC2)C=CCOC1 C1(C(N(C(C)CNC(c2cccc(C(C)(C)C)c2)=O)C)=O)CCC2(C1)CC2(F)F N1(C(C(c2cncnc2)NC(CCC2CCC(=O)C2)=O)=O)CC=CC(O)C1 c1(C(C)NC(C)C#N)cccc(C(F)(F)F)c1.C12CC(C1)CC(=O)NC2 n1(CC)cnc2[nH]c(=NCC(C)CCCO)nc(N3CCc4nc[nH]c(=N)c4C3)c12 c1(NC(C2C(C(=O)NCC(C)(C)CO)C2)=O)cc2sccc2s1 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2C(F)(F)F)=O)cccc(C2CCC2)c1 N1(C(CCOCC)=O)CCN(C(=O)C(CC#N)c2ccccc2)CCC1C C=CCC(C(=O)Nc1cnn(Cc2cncc(OC)n2)c1)NC(C)=O Cc1c(C(=O)NCC(C)(O)CNC(=O)C(F)F)sc(Cl)c1Cl C1(CNC(c2n(C(C)C)ccc2)=O)CCCN(c2ncnc(O)c2Br)CC1 N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(=O)C(Cl)=CCl)CC1 C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(c1c[nH]nc1CC)=O Cc1cc(F)cc(CN2CCC(F)(CO)CC2)c1O.c12cc(ccc1F)C(=O)N2 N1(C(C2N(CC)CC2)=O)CCC2CCC(NC(c3cccc4[nH]ncc34)=O)C1C2 c1(NC(c2ccoc2)C)ccc(S(=O)(=O)NC(C)C(C)(C)OC)cc1Br C1(CCNCc2nnc(C(C)(F)F)s2)COCC(C)O1 Cc1ccc(C(=O)NC2CCN(C(C3CCCCC3(F)F)=O)C2)cc1C C(=O)(C1=CCCOCC1)N1CCC2C(C(N3C(C)CC(O)CC3)=O)C2C1 c1(CC)cc(C(=O)NC(C2CN(C(=O)CC(C)C(F)F)C2)C)cc(F)c1 CCC(C)(C)C(O)C(=O)NC1(C(N2CCN(CC(C)O)CC2)=O)CCCC1 N1(C(=O)CCc2nccs2)CCN(C(C2(C3CCC3)CC2)=O)C(CC(F)(F)F)C1 C(=O)(C(F)C(=O)NCC1(O)CCN(C(c2coc(O)n2)=O)C1)OCC C1(NC(CN(CC)CC)=O)CC(CO)N(C(C2CCC(=O)O2)=O)C1 CCC(C)CC(C(=O)NCCc1cnn(C)c1)NC(=O)CCCCN=[N+]=[N-] Cc1cn2cccc(C(=O)NC3(C)CN(c4nc5ccc(N)cc5s4)C3)c2n1 c1(OC)c(Cl)ccc(C(=O)NCC2CC(NC(=O)C(C)C(F)(F)F)C2)c1F c1(NC(=O)Nc2c(C)cc(N3CCN(C)CC3)cc2)noc2cc(Cl)ccc12 CCC(CO)C(=O)N1CC(=C(F)CNC(C2CCCS2)=O)C1 C=C(C)C(C)(C)C(=O)NC(CNC(c1cnc(C2CC2)s1)=O)CC(C)C c1(C(N2CCCC(N(C(=O)CN3CCCC3C)CC)C2)=O)cc2c(ccn2C)[nH]1 N1(C(CN(C(COC)=O)C)=O)CCN(C(c2snnc2C)=O)CC(C)(F)C1 C(=O)(C#CC1CCOCC1)N1CC(O)(C(C)NC(C2(C)CCCC2(F)F)=O)C1 c1(C(=O)NC(C(C)NC(c2c(C)nc(CCC)s2)=O)C)c(N)cccc1F c1(CC(=O)NCC(C)CN(C)C(C2CC2C(C)O)=O)ncc(Cl)s1 CCC(CC(=O)NC1(CCCC(=O)N(CCCOC)C)CCC1)SC Cc1nc(N2CCC(C3CCCCN3C(c3cc(C4CCC4)no3)=O)C2)sc1C Cc1cccc(Br)c1C(C(=O)NC1CC2CC1CC2=O)NC(=O)COC(C)C C1(NC(CSCCC)=O)CCOC12CCN(C(=O)Cc1cnc(C3CC3)[nH]1)CC2 c1(C(=O)NCC2CC(NC(C(C(C)(C)C)N(C)C)=O)C2)cc(F)c(C#N)c(F)c1 c1(OC)cc(C(=O)NCC2(C)C3CCCC23)c(C(F)F)cc1OC(=O)C(C)(C)C C1(C)(C(N(C2CCN(C(=O)CCc3ccc(N)cn3)CC2)C)=O)CCC(=O)N1 C(CC(=O)N(C(C)C(=O)OC)C(C)C)(CC(C)C)NC(C(COCC)C)=O C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(=O)C(CC2CC2)OC)C1 n1(CC(OC)OCC)ccc2c(NCC)cccc12.C1C(=O)N1 n1(CC=CC)nc(C)c(=NCCN2CCN(S(C)(=O)=O)CC2)[nH]1 N1(C(c2c(C)[nH]nc2Cl)=O)CC2(C1)CN(C(C1CCCC1CF)=O)CCO2 c1(N(CC(Cl)Cl)C)nc(N2CCC(Cc3ccccc3)C2)c2sccc2n1 CCCCN=C(NCC1CCOC1)N1CCC(c2c(C)[nH]c3ccccc23)C1 c1(C(=O)NC2CN(C(=O)C=CBr)CC23CC3)cccc2[nH]cc(Cl)c12 c1(C(=O)NCC2N(C(c3c(C)nc(C)o3)=O)CCCC2)cncc(C)c1Cl C=CCC(CC(=O)NC1(C)CCCC1O)NC(c1cnnn1C=C)=O C1(C(=O)NCCN(C)C)CC12CCN(C(=O)C(c1ccccc1)O)CC2 C1(CNC(C(C)OC)=O)C2CN(c3ccnc(-c4nccs4)n3)CC12 c1(C(=O)NC2CCCC(NC(c3ncc(N(C)C)cn3)=O)C2)ncnc(O)c1F N1(C(CC2(COC)CCCC2)=O)CC2CCC1C1CN(C(=O)C(F)OC)CC21 N1(CC(=O)NCCC(CNC(=O)C(C)C(F)F)OC)CCCCC1C c1(NC(C(=O)NCC2(OC)CCCS(=O)(=O)C2)=O)ncnc2c1COC2 C(C(=O)NC1CCC(F)(F)CC1)(C(C)CC(C)(C)C)N(CCC=C)CC S(=O)(=O)(c1ccc(=NCCNS(=O)(=O)CC)[nH]c1)N1CC(C=C)OCC1 c1(C(C(=O)NC2CCOC2)N(CCF)CC)cccc(C(F)(F)F)c1F c1(C(=O)NCC(CNC(C2C(C(C)C)C2)=O)(C)C)ccccc1CCC(F)(F)F C1(NC(=O)C=Cc2ccc(F)cc2)CCN(C(C2(F)CCOC2)=O)CC12CCC2 C(=O)(CCCCC(F)F)N1CCC(CNC(C(C2CCCCC2)OC)=O)C1(C)C N1(C(CCC(=O)NCCC)=O)CCC(C(=O)NCCCc2cncnc2)C1(C)C c1(C(N2C(C)(C(=O)NCCC(CCC)O)CCC2)=O)cc(C)cc(O)n1 C(CC(=O)NCc1cnn(C)c1C)(C(F)(F)F)NC(c1cc(CC)sn1)=O CS(=O)(=O)c1nccc(N2CCC(O)(C(=O)Nc3c(Cl)ccnc3Br)C2)n1 Cc1cn2cc(C(=O)NC(C3CN(C(C4CC(=O)N(C)C4)=O)C3)C)cc(C)c2n1 c1(N(C)C)ccccc1C(N1CC(OCC(=O)NC2CC(NC(N)=O)C2)C1)=O Cc1cnc2cccc(C(N3CCN(CCNC(=O)CNS(C)(=O)=O)CC3)=O)n12 C1(CCC)CCCCN1C(c1n[nH]cc1-c1ccc(OC2CC2)cn1)=O N1(C(CC2CCC(=O)C2)=O)CC2CCCC(NC(C34CCC(CC3)OC4)=O)C2C1 N1(C(C(C)NC(C)=O)=O)CCC(F)(CNC(=O)C(C)NC(=O)C2CC2)C1 c1(SC)cccc(Br)c1CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)O CC1(C)NC(=O)OC12CCN(c1ncnc3c1CCCC3)C2 CCCCC(O)C(=O)NC1CN(C(c2cc(N)ccc2SC)=O)CC1F c1(C(CNC(=O)C(C)(N(C)C)N(C)C)NC(CC2CC(C)C2)=O)cccc(Cl)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCC(CNC(c2cnsc2)=O)CO)c1C CCCCC(C)CCC(=O)N1CCC(CCC(=O)N(C2CC(O)C2OC)CC)C1 CC1(C)CC(C)(C(N2CCCCC(F)(F)C2)=O)CN1C(=O)C1=NOCC1 Cc1nccc(CCCNc2cc(N(CC(C)C(F)(F)F)C)ncn2)n1 C12(C(N3CCN(CCN(C)C(C4CC(C)(O)C4)=O)CC3)=O)CCCN1CC(O)C2 C(C)(CC(C)(C)CO)NC(CC1N(C(C(=Cc2cn[nH]c2)C)=O)CC(O)C1)=O N1(C(c2cc(C)nc(O)n2)=O)CCC2CCCN(C(=O)CCN3CCCC3)C2C1 C1(=O)CCCC(=O)N2CC3CC3(C2)NC(=O)C(C)ONC1=O.CCCNOCC N1(c2nnc(CNC(CC)=O)n2CC2CCCCO2)CCC2(C1)CC(F)(F)C2 c1(SC)cc(C(F)(F)F)ccc1CN1CCN(C(=O)CC2(C)CCCO2)CC1C c1(CNc2c(OC)cccc2C(=O)OC)cc(C)c(F)c(F)c1 CCS(=O)c1ccccc1C(=O)NC(CCN(C)C(c1cc(Cl)cs1)=O)C(C)C N1(CCC(=O)N(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)CC)CCCCC1C Cc1nc(Br)c(C(N2CCC(CO)(NC(=O)C(C)C3CC3)C2)=O)s1 N1(C(c2c(OC)oc(C)n2)=O)CCC(O)(CNC(c2cnc(SC)n2C)=O)CC1 CC1CN(C(=O)COCC2CC2)CC(CCNC(c2nn(C)nc2Br)=O)O1 Cc1cnc(F)cc1C(=O)NC(C)CCCCN C(CCCCC(=O)NCc1cnc(C)o1)NC(C(CC)CN(C)C)=O c1(NC(C2N(C(c3nc(COCC)sc3)=O)CCC2)=O)ccccc1C c12ccc(cc1C)[nH]c2=O.CCCCC(=O)NC1(CC(=O)C2CC2)CC1 S(=O)(=O)(c1ccc(NCC2CCC3(CCCC3)C2)c2cnccc12)NCC(=C)Br C=CC1CC(N(C(c2cc(CC)on2)C(=O)NCC(C)C)C)C1 C1(NC(c2cc(OC)ncn2)=O)CCN(C(=O)CNC(=O)CN(C)C)C1(C)C C=CC1CN(C(C2CCC(NC(c3coc(CO)c3)=O)CC2)=O)CC1O c1(C(N2CCC(O)(CNC(C3C(OCC)C3)=O)C2)=O)cc(-n2cccc2)ccn1 c1(SC)ccc2cc(C(=O)NCC3CC3CNC(c3csc(C#N)c3)=O)[nH]c2c1 CCC(C)C(O)C(C)C(=O)N1CCOC(C(C)NC(c2[nH]cnc2C#N)=O)C1 Cc1cccn(CC(N2CCC(NC(c3ccc(C(C)C)o3)=O)C(O)C2)=O)c1=O c1(C(c2nnnn2CCCF)NC2CC(=C)C2)ccc(Br)cc1Oc1cnsc1 CC#CC1CCN(C(=O)CCCN(C)C(c2ccsc2C)=O)C1 c1(C(=O)NCC(C2CCN(C(C=CSC)=O)CC2)(C)O)cc(Cl)c(C)cn1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2C(C)C)=O)cccc(COC)c1C CC(C)CCCCC(=O)N1CC(CC(=O)NC2C3CCCOC23)C(C)C1 c1(CO)cc(F)cc(F)c1.c12ccc(cc1)NCc1cccn1-2.c1ccccc1 C(CNC(=O)CC1CC2(CC2)CO1)(CC(=O)NC1(C(N)=O)CCCCC1)OC N1(C(C2CC(=O)NCC2)=O)C2CCC1C(CNC(c1ccc(F)s1)=O)C2 c1(C(COC(C(C)SSC2CC(c3ccccc3)C2)=O)=O)sccc1C#N CC1C(NC(c2cncc(N=[N+]=[N-])c2)=O)CC2CCC1N2C(c1nccn1C)=O C(=O)(CC(CNC(=O)CC(C)SC)C1CCC1)N1CC(C)(CC=C)C1 C1(C(N2CC(C)C(C(N3CCOCC(O)C3)=O)C2)=O)CC2CC(=O)C1O2 N1(C(CC=C)=O)CC(NC(=O)C(C)CC)C(O)C1 c1(CC)ncc(Cl)c(C(=O)NC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2O)n1 C1(C(=O)NC(CNC(c2n(CCC)nc(C)c2)=O)C(C)(C)C)CC2(C1)CC(C)C2 c1(C(N2C(CNC(C(C=C)OC)=O)CC(COC)C2)=O)ccc2c(c1)NCC2 C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)CSCC(N)=O)CC2C)s1 C1(CC(=O)NCCCCNC(C(C)OC(C)(C)C)=O)CCC(=O)N1C c1(OC)nc(N2CCC(OCCNC(C3(C)CCCNC3)=O)C2)ncc1C CCC(CNC(C1CCN(C(=O)OC(C)(C)C)C1(C)C)=O)(CC)C(=O)OC C1(C(N(CCCCNC(CSCC=C)=O)C)=O)CCCN(C(C2CCC2)=O)C1 C1(C(N2CCCC(C(C)(C)NC(CC(=O)N(C)C)=O)C2)=O)CCCN2CCCC12 C(=O)(CCCC(C)(F)F)N1C(C(C)C)CN(C(C2CC=CCC2)=O)CC1 C1(NCC(C)=C2CC2)(CO)CC2(CCCCC2)C1.C(C)(C)C C1(C)(C(N(CC(C)(C)CNC(c2csc3cncn23)=O)C)=O)CCCNS1(=O)=O C1(C(=O)NCCC2(NC(COCc3cc(C)no3)=O)CCC2)CCCC(=O)N1C c1(C(N2CC(CNC(C(=O)NCC)=O)CC23CCC3)=O)cccc2ncc(C)n12 N1(C(C2N(C(CN3CCC(=O)CC3)=O)CCCCCC2)=O)CCOCC(C2CC2)C1 C=CCC(F)(F)CNC(C1(CC)CCCN1C(=O)Cn1cc(Cl)cn1)=O c1(C(=O)NC2(COC)CCN(C(=O)CC(C)SC)C2)ccc(Cl)c(Br)c1 C=CC1(NC(=O)C(CNC(c2cnoc2C(C)C)=O)N(C)C)CCC1 C1(N(CC(=O)N(C)Cc2ccccc2)CC2COC(=O)N2)CS(=O)(=O)CC1C C1(N(C(=O)C(=O)NCC2CC2)CC)CCCN(C(=O)Cn2ncn(C)c2=O)C1 C12(C(=O)NCC3N(C(C(N4CCSCC4)C)=O)CC3)CCCC1(C(N)=O)C2 N1(C(CCCN(C(C)=O)C)=O)CCC(CO)(CNC(=O)CCS(C)=O)CC1 c1(OC(C)C)ccc(CN2CCSC(C(N3CCCCC3C#N)=O)C2)cc1Cl Cn1c(C(=O)NCC(C2CCCCC2)NC(=O)C(F)C2CC2)cc(Cl)c1Cl N1(C(=O)CCn2cc(COC3CCOC3)nn2)CC2CC(C1)C1CCCCN1C2 C1(C(C)C)CN(C(=O)CCF)CCC1NC(c1nocc1Cl)=O C1(Cc2ccc(C)cc2)CCCCC1N=c1[nH]c(=NCC(C)F)[nH]c2ccsc12 n1(CCC)nc(C)c(C(=O)NCCCN(C)C(c2nnn(C)c2C(F)F)=O)c1C N1(C(c2nc(-c3cc(NC)n[nH]3)n(CCn3ccnc3)n2)CC)CC(C)CC(C)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCC3(F)F)C2)sccc1C#N c1(C(=O)NC2CCC(N(C(CCC(=O)N(C)C)=O)C)CC2)c(F)cc(N)cc1F c1(CNC(=O)C(O)C2CN(C(=O)CC3CCCSC3)C2)ncccn1 C1(CCNC(c2ccsc2)=O)CCCN(C(=O)COC2CCCC2)CC1 C(CCN=C(NCC(O)Cn1ccnn1)NC1CC(=O)N(CC)C1)OCC C(=O)(C1CNC(=O)c2ccnn21)N1CC(C(C)NC(c2ccc(Br)o2)=O)C1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(O)C1C2NC(c1snc(O)c1Cl)=O CCCC(C)CC(=O)N1CCCC(N(C(=O)CCOC2CC2)CC2CC2)C1 N1(C(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CC1(C)Br)=O)C2 O=C(C1=COCCC1)NC1CC(F)CN(C(c2cc(O)nc(Cl)c2)=O)C1 N1(C(C=C(C)C)=O)CC(NC(=O)C(C(C)C)OCC(C)C)C2(CC2)C1 c1(CCC)nc(C)c(NC(C2CCCC(C)C2)=O)o1 N(C(=NCCF)NCc1cc(F)cc(Cl)c1)CC1CC(C(C)(C)C)C1 Cc1c(Cl)cnn1CC(=O)NC1CC1CNC(=O)CCCc1cncs1 N1(C(C(CC(=C)C)OC)=O)CC2CC(C(=O)NC(CO)C(F)(F)F)C(C2)C1 C1(CNC(C2CCC(N(C)C)CC2)=O)COCCN(C(C2(C)CCNC2=O)=O)C1 c1(C(C(=O)NCC(C)OC)NC(=O)CN(CC(C)(C)C)C)cn(C)nn1 C1(OC)CC(NC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2occc2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NC1(CN(C(CSCCCC)=O)C)CC1 C1(=O)C(CN)C1=O.c1(CC)snnc1C(C)N.CC(C)C c1(C(N(CC(=O)NCC=C(C)C)C2CC2)=O)cc2ccccc2[nH]1 N1(C(COCCOC)=O)CCN(Cc2c(OC)ccnc2Cl)C(CO)C1 N1(C(C(c2cccc(C)c2)=O)=O)CCc2ccccc2C(NC(C2(F)CC2)=O)C1 C(c1ccncc1)=C(C)C(=O)NCC(C1CCCN1C(=O)CN1CCCC1C)(C)C c1(C(N2CC(NC(C(CSC)O)=O)C(C)(C)C2)=O)cc(N)c(C)c([N+](=O)[O-])c1 C=CCCCCC(=O)N1CCCC1(C(=O)NC)CCc1ccccc1 N1(CCC(=O)NCC#CCNC(C2C3CCC(=O)C23)=O)CCCCC1=O CCS(=O)(=O)c1cccc(CC(N2CCNCC2c2cccc(Cl)c2)=O)c1 C(=O)(C(O)CC(N)=O)NC1C(C(=O)NC2C(OC)C(O)C2)CCC1 N1(c2cc(NC(NOC(C(C)(C)C)(C)C)=O)ncn2)CCCC2(CC=CCO2)C1 c1(C(N2CCC(C(C)NC(C3(N(C)C)CCC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1F N1(C(CC(C=C)C)=O)CCN(C(=O)CN2CCCCCC2)CC(C)(C)C1 C(CN(C)N1CC(O)(C(C)C)C1)Oc1cccc(C)c1 c1(C(=O)NC(CCNC(C(CC(C)(C)C)OC)=O)C)cccc2nn(C)cc12 c1(CC(=O)N(CCN(C(=O)CCc2cccn2C)CC)CC)cc(F)ccc1Cl c1(C(=O)NC(CNC(CC=CCCCCC)=O)CCOC)cc(O)ncc1F CCCCC(C)C(=O)NC12CC(C(=O)NC3CCCCN3c3ncccn3)(C1)C2 c1(C(=O)NCCC2N(C(C3CCC(=O)NC3)=O)CCC2)c(F)cc(F)cc1Cl C=CCC(CNC(=O)CC1CC(F)(F)C1)C(=O)NC1CCCCCCC1 CN1C(=O)CCc2cc(C(N3CCCC(C(N)=O)C3)C(=O)NC(C)(C)C)ccc21 CCC(CCCC(=O)N1CCC(CCN(C)C)C1)NC(=O)CC(=O)OC(C)(C)C c1(CC(C)NCC2(OCC)CS(=O)(=O)C2)ccc(Cl)cc1Cl N1(C(C(CC=C)C)=O)CCC(C2CC2)(CNC(C23CCCN2CC(OC)C3)=O)C1 C1(NC(Cn2ncc(CC)c2)=O)CCN(C(=O)CCc2ccsc2)CC1CC O=C1C=C(c2ccnc(NC(=O)NCCNc3cccc4ccccc34)c2)CCC1 CCCCCCCCCC(=O)N1CCN(C(=O)CCCF)CC1CCC CC1CC(C(=O)NC(C)(C)CNC(c2cc(-c3cnn(C)c3)[nH]n2)=O)=NO1 c1(C(N2CCC(CCCO)C2)C(=O)NCCC#N)ccc(C2CCC2)nc1 c1(C(N2CC(F)CC(NC(CC3CCN(C)C3)=O)C2)=O)cnn2ccccc12 c1(C(N)=O)cscc1C(=O)NC1CCC(CCNC(=O)CSc2nc[nH]n2)C1 N1(C(C2CCC(CC(C)C)CC2)=O)CC2CN(C(=O)CCF)CC2C(F)(F)C1 c1(C(C(=O)NCCCN(C)C(C2CCCC2CF)=O)(C)C)ccc(Cl)cn1 c1(C(=O)NC(=O)C(C)Cn2cccn2)cn(CCCCNC(CCOC)=O)nn1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC(CC=C)NC(c1ccn(C)c1)=O Cc1nc2c(F)cccc2cc1C(=O)NC1(C2CN(C(=O)CNC=O)C2)CC1 N1(C(CC2(CC=C)CCCC2)=O)CCCCC(CNC(=O)CC2CC=CCC2)C1 Cc1ccn2ncc(C(N3CC4=C(C3)CN(C(=O)C(C)C3CCOC3)C4)=O)c2n1 c1(C(C)C)cc(C(=O)NC2CCCC2NC(=O)CCC2CCC(O)CC2)nn1C C(=O)(C1=NOC(CC2(O)COC2)C1)N1C2(CNC(C#CC(C)C)=O)CC(C1)C2 c12ccc(cc1)CCCN(C)C2.CC(F)CCN(C)C CC(C)(C)C(CC(=O)NCC1OC(=O)CC1(C)C)NC(=O)CSCC(N)=O N1(C(c2c(=O)ccn(C)c2)=O)CC(CNC(C2CC3CCC2C3)=O)CC12CCC2 CCC(C)C(CC(=O)NCCN1CCC(O)C1)NC(c1ccnc(C2CC2)c1)=O c1(COC)cc(C(N2CCCCC2CCNC(c2ccnnc2O)=O)=O)n(C)c1 c1(CNC(CC(CC)NC(c2ccc(Cl)s2)=O)=O)cc(F)ccc1F C(N=c1[nH]c(=NCCCn2cc(Br)cn2)[nH]c2c1CSC2)C1(SC)CCCCC1 c1(C(=O)NCC2C3CN(C(C(CCC)C)=O)CC32)cc(O)cc(Br)c1 CN1N=C(C(=O)N2CCC(F)(CNC(c3cccc4c3OCC4)=O)C2)CCC1=O CS(C)(=O)=NCC(=O)NC1CC(c2ccc(C(=O)O)cc2)C1 O=C(N=c1cc[nH]cc1O)C1CCCC2C1CCN2C(=O)CSc1ccccc1 C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2 c1(C(=O)NCC2CC(O)(CNC(C(CC)=CC)=O)C2)cccc(NC(C)C)c1 c1(CC)ncc(C(=O)NCC(c2ccccc2)CNC(=O)C(O)CSC)o1 Cc1c(C(N2CC(CNC(c3ccc(C(N)=O)cn3)=O)C(C)C2)=O)nnn1C c1(CCC(N2CCC(F)(CNC(C3(N(C)C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 CC(C(C)C(=O)N(C)Cc1nccs1)NC(=O)CCC1CCCOC1 CCCCCC(C)CC(=O)NCC1(O)CC(NC(=O)CCCCC(=O)OC)C1 C12(NC(Cc3nc(C)[nH]n3)=O)CCN(C(c3ccc(F)cc3Cl)=O)CCC1C2 Cc1cc(O)ccc1N(C(=O)CC=CCNC(=O)C=CC(C)(C)C)C CC1CCc2sc(C(N3CCCCC3CNC(=O)CCCC3CCC3)=O)cc2C1 N1(C(c2ccoc2)=O)CCOC(CC2CC2)C1.c12cc(co1)C(=O)NCC(=O)N2 C1(C(=O)NCCOC(C)(C)CNC(c2coc(Cl)n2)=O)CCCCC1O N1(C(CC(C=C)C)=O)CCC2CCC(NC(c3cc(CC)cc(Cl)c3)=O)C1C2 N1(C(=O)Cc2cc(Br)ccc2F)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 C(F)(F)(C(F)(F)F)c1scc(C(c2n(CCOC)nnn2)NCCCF)c1 c1(COc2cc(CCC)[nH]c(=O)c2)cc(Br)cc2c1OCC2 N1(C(C2CC(SC)C2)=O)CCCC(C)C1CNC(c1cc(C)ccc1C)=O c1(C(=O)NC2CC(CCNC(CC=C)=O)C2)cnn(C(C)C)n1 N1(C(C2(OC)CCC2)=O)CC(N(C(=O)C=Cc2ccc(SC)cc2)C)C(C)(C)C1 c1(C(N2CCC(C(=O)Nc3c(OC)c(F)ccc3)C2)=O)cc(C)cc2[nH]ccc12 C1(NC(Cc2cccc(C)c2Cl)=O)COC2(C1)CN(C(C1CC3C=CC1O3)=O)C2 c1(CC)cc(CN2CC3(CNCCO3)C2)c2sc3ccccc3n12 C12(NC(C(C)C3CC3)=O)CCCN(C(c3ccccn3)=O)C1C2 c1(CC)ccc(C(=O)NCCC2CC(NC(c3cnccc3CC)=O)C2)cc1 c1(C2(CN3CC(O)(CSCC(C)C)C3)CC2)ccc(Br)cn1 c1(C(=O)NC2C3(CN(C(C(COC)(C)O)=O)C3)CCC2)ccc2[nH]c(=N)[nH]c2c1 C1(C(N(CCNC(C(C)OCC#C)=O)CCOCCO)=O)CCC(C(F)(F)F)CC1 c1(C(=O)NC2CCCN(C(CC(COC)C)=O)CC2)[nH]c2cc(F)ccc2c1C N1(C(C2(N(C(C(CC)CN(C)C)=O)C)CC2)=O)CCn2nccc2C1 CC1CCN(C(c2c(F)cncc2Cl)=O)CC1CNC(=O)CSc1cccs1 C1(C(=O)NC(C)C=CC(=O)NC2(CO)CCC2)CNC(=O)CC12CCC2 C1(CNC(CCNC(C)=O)=O)CC2CC2N1C(c1ccsc1C)=O CN1CCC(C(=O)NCC2CCCN(C(=O)C(C)(C)F)C2)S1(=O)=O C1(C)(NC(C(N2CCC(O)CC2)C)=O)CCN(C(=O)CCc2cncn2C)CC1 N1(C(C(C=C)O)=O)CC2CC1C2C(=O)NC(CO)CCC1CC1 C(C)(CNC(C1(NC(=O)C(F)OC(F)(F)F)CCCC1)=O)(CO)OC c1(C(N2CCCC(CC=C)(NC(c3coc(Br)c3)=O)C2)=O)cccc2nncn12 N1(C(=O)OC(C)(C)C)CCC(C2CC2(F)F)C1.c12cc(ncn1)C(=O)O2 c1(OCC)ccc(CCC(=O)NC2CC(CNC(C3(C)CC(F)(F)C3)=O)C2)cc1 C1(CNC(C2CCC2)=O)CC2(CCN(C(C3OC4CCC3CC4)=O)CC2)CO1 C(=O)(C1=C(C)OCC1)NCCCN(C(C1C(C)(CC)C1)=O)C1CC1 c1(CNC(C(C2CC2)OCC)=O)nc(C)c(C(=O)NCCN2CC3CC3C2)o1 N1(C(c2cc(CC)[nH]n2)=O)CC(C2CCN(C(C3C4COCC34)=O)CC2)C1 c1(C(=O)NC2C=CC(CNC(COC)=O)C2)c(OC)ccc2ncccc12 c1(C(=O)NC(C)(C)CNC(C2(O)CCCCCC2)=O)ccc(P(C)(C)=O)s1 C(=O)(CCCCC(=O)OC(C)(C)C)N1CC(NC(c2ccc(C(C)=O)cc2)=O)C1 c1(C2CCN(C(C(C(=O)OCC)(CC)CC)=O)CC2)cc(S(N)(=O)=O)c(Cl)cc1Cl C1(NC(c2ccc(F)o2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CC1F c1(-c2ccc(C(=O)NCCNC(CCC3(C)CC3)=O)s2)ccc(F)cc1 Cc1cc(CNC(=O)C(C2CCCCC2)O)oc1C(=O)NC1(CCF)CCC1 c1(C(=O)NC(C)CN(C)C(C2CCC(=O)C2)=O)cc(F)cc2ccncc12 C(=O)(CC(O)C(C)C)N1CC(OC)C(NC(CC2(NC(C)=O)CCC2)=O)C1 N1(C(c2ccc(SC)s2)=O)CCC2(CC1)OCCCC2NC(=O)C(C)C(C)C c1(C(=O)NC(CCCCNC(C2CC(SC)C2)=O)C)cncc2ncn(C)c12 N1(C(C(C(C)C)C)=O)CCC2(CC(NC(C3(C(=O)OC(C)(C)C)CCC3)=O)C2)C1 N1(C(C=CCCC=C(C)C)=O)CC2CCN(C(C3CN(C)CCO3)=O)CC2C1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)C(C)(O)CCC)CCC12CCC2 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)Cc2csc(=N)[nH]2)C(CO)C1 Cc1ccc(S(=O)(=O)NCCC(=O)Nc2cccc(Nc3nccs3)c2)c(F)c1 CC1(CNC(C2CCCS(=O)(=O)C2)=O)COCCN(C(c2cccnc2N)=O)C1 c1(C(=O)NCC2(O)CCN(C(C(C)S)=O)C2)ccc(Cl)c(Cl)n1 C1(CNC(=O)CC2CCC(=O)O2)CC2CCC1N(C(c1c[nH]cc1Br)=O)C2 CN1CCCC1CCC(=O)N(C1CCN(C(C2(CN(C)C)CC2)=O)C1)C N1(C(C(C(=O)OC)C)=O)CCCC(O)(C(=O)NCC2(CSC)CCC2)C1 O=C(C1=CCOCC1)NC1COCC1CNC(c1ccc(Cl)c(Cl)c1)=O C(=O)(C(CC(C)SC)N1CCCC(CCO)CC1)NC(c1ccccc1)C C(=O)(C(F)(CNC(=O)C1=CCCCCC1)C(C)C)N(C)Cc1onc(CC)n1 c1(C(N2CCC(NC(C=Cc3cn(C)nc3)=O)C2)=O)cc2c(s1)C(C)(C)CCC2 c1(SCC(C(=O)NC2C(CNC(CNC=O)=O)COC2)O)ccc(F)cc1 C1(COC(C2(C(C)=O)CC2)=O)CCCC2(CCC2)O1 C1(F)(CNC(c2cnc(SC)[nH]2)=O)CCC(NC(C2CCCCS2)=O)C1 C(=O)(C1(C)CCn2ccnc21)NC(COC)CC(=O)N1CCC1CF C(C)(N=c1nc2sccc2c(N2CCC(C(F)F)CC2)[nH]1)c1c(C)cccc1 N1(C(CC2(OC)CCC2)=O)CCCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 CC1CSCCN1C(C1CCC1NC(C1OCCC1(C)C)=O)=O N1(C(C2(CCOC)CC2)=O)CCCC(O)(CCNC(c2cccc(N)c2F)=O)C1 c1(NC(c2c(CNC(CC(OC)OCC)=O)occ2)=O)ccc(CN(C)C)c(F)c1 C(=O)(CCC(N)=O)NC(c1cccc(Cl)c1)CNC(c1c(OC)n[nH]c1)=O CC1(C#CC(=O)NCCC2(C)CCN(C(c3cccc(F)c3O)=O)C2)CCCO1 C(=O)(C(C)C(=O)N(C1CCN(C(=O)CN(C)C(N)=O)CC1)CCO)OC C1(C(=O)NC(C#C)CO)CCn2cncc2C1 c1(CC(=O)NCC2CN(C(CC(=C)Br)=O)C(C)C2)ccccc1[N+](=O)[O-] C=C(Cl)CCC(=O)N1CC2CC1C2NC(=O)Cc1csc(C2CC2)n1 c1(NCC2N(C)CCN(c3ccc(C(F)(F)F)cn3)C2)csc2ccc(Cl)cc12 c1(CC(N2CC3(CCN(C(C4CC4CF)=O)CC3)C2)=O)c(Cl)cccc1[N+](=O)[O-] C1(N(C(CCCC)C)C)CCN(C(=O)CCC2CCOC2)CC1C Cc1cc(N)cc(C(N2CCC(NCCO)CC2)=O)c1F c1(C(=O)NCCOC)[nH]c(C)c(C(N2CC(C)SC(C)C2)=O)c1C N1(C(CCCn2cc(C3N(C)CCC3)nn2)=O)CCC12CCN(C)C2 C(C1=CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1)NC(C(C(C)C)SC)=O N1(C(C)=O)CCCC1CNC(C12CC(C)(C1)C2)=O C(=O)(C1=COCCC1)NCC1CC(NC(=O)CSC2CCCCO2)C1 c1(C(N2CC(CCCNC(COCC)=O)OCC2)=O)cnc2[nH]c(C)nc2c1 C(CC(CNC(c1cccn1C)=O)NC(=O)CCOC1CCOC1)OC C1(NC(c2ccc(C(N)=O)cn2)=O)CCCCN(C(c2ccnn2C2CC2)=O)C1 N1(C(c2c(C)scc2)=O)CCC(N(C)C(c2ccc(C(F)(F)F)[nH]2)=O)C(C)C1 C(=O)(C(CC(C)(C)C)NC(=O)C=CC1CCCCC1)N(C1C(C)COCC1)C C1(NC(C2(C(C)C)CCCO2)=O)CC2CC(NC(c3ccc(O)nn3)=O)CC12 CN=S(C)(=O)c1ccc(C(=O)NCC(C)N(C)C(c2ocnc2C)=O)cc1 C1(CNC(CCN(C)C)=O)CCCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OC)ccc(F)nc1NC(C1CC1C(=O)Nc1cccc(C#N)c1)=O C1(COC)(NC(c2ccn(CO)c2C)=O)CCCN(C(=O)CN2CC3CC3C2)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCN(CC(C)O)CC1.C12CC(C1)C(=O)N2 C1(C)(CC(=O)NCCc2nc(C)[nH]n2)CCCN1C(=O)CC1CCCCC1 Cc1nc(C(=O)N(C(C)CNC(c2c(-c3ccccn3)noc2C)=O)C)c(C)o1 C1(NC(CSC)=O)CCSC12CN(C(=O)C(C)Cc1ccc(F)cc1)C2 C=CCCC(C(=O)OC)NC(=O)C(CC)NC(c1nscc1C)=O c1(C(=O)NCCC2OCCN(C(C3C(C)(C)CCC3)=O)C2)cc(Cl)cc(Cl)c1F FC1(F)CC12CCC(CN1CCC(C3NCC34CCC4)CC1)CC2 N1(Cc2c(C)cc(C)[nH]2)Cc2ccc(O)cc2CC1C(N1CCC(F)C1)=O c1(OC)c(Cl)cc(NC(=O)Nc2cn(C)nc2C(F)(F)F)cc1Cl c1(COC)cc(NC(=O)NC(C)Cc2cccc(O)c2)ccc1F c1(NC=O)ccc(C(=O)NC2CC(CO)N(C(=O)CC3CCOC3=O)C2)cc1 N1(C(C(C)CC2CCC2)=O)CC2(CCCC2)C1C(N1CCN(CCO)C(=O)C1)=O C(C(O)C(=O)NCC1CC1CO)NC(c1cc(Cl)ns1)=O C1(CNC(c2c(C)ccnn2)=O)CN(C(c2coc(C(F)(F)F)c2)=O)CCC1C C1(C(=O)NC(c2c(C)c(Cl)ccc2)c2ccc(Cl)cc2)CCCC(F)(F)C1O C1(CNC(C(c2cnn(C)c2)C)=O)CCCN(C(C2CC3C=CC2C3)=O)CC1 c1(CC(=O)NCCC2(O)CN(C(CCC(C)OC)=O)C2)coc2ccc(C)cc12 c1(C(=O)NC2CN(c3cc(NC(C)=O)ncn3)C2CO)c(Cl)nc(SC)nc1Cl C1(C(N2C(C(=O)NCC(N(C)C)C3CC3)CCC2)=O)CCCC(=O)C1 N1(C(Cc2ccc(OC)c(OC)c2)=O)CCN(C(=O)CCNC(N)=O)C(C)C1 Cc1csc(CC(=O)C(CC2C3CCOC3C(=O)N(C)C2)=O)c1.c1(CCN)cc(C)on1 N1(C(C=CC=CC)=O)CC2CCN(C(c3ccc(Br)c(OC)c3)=O)CC2C1 CCC(O)C(F)(F)C(=O)N1CC(CNC(c2cc(Br)nn2C)=O)C(O)C1 N1(C(c2cc(Cl)nn2C)C(=O)NCCOC)CCN(C)C2CC12 N1(c2ncnc(C)c2Br)CCC12CCN(C(=O)C(C)c1cccs1)CC2 N1(C(CC=CC=C)=O)CC(C)(C)CC1C(N1CC(C(=O)OC)(OC)C1)=O N1(C(CNS(NC)(=O)=O)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC2(C)CCCC12 CCC(CNC(C1CC1(F)Cl)=O)(CC)NC(c1cncn1C)=O C1(NC(Cc2cc(OC)no2)=O)CC12CCN(C(C1CC1F)=O)CC2 c1(NC(=O)NC(C)CCCOc2cccnc2)cnc2ccnn2c1 Cn1cc(S(F)(F)CNC(=O)NC23CC(Cc4ccccc4)(C2)C3)cn1 CC(C)(CC(=O)NC1CCC1NC(c1c[nH]nc1C(C)(F)F)=O)CC(F)F C=C(C)CC(C)C(=O)N1CCCC(CCNC(=O)CCOc2ccccc2F)C1 c1(CN2CC(C(=O)Nc3ncncc3Cl)C(O)CC2)c(O)ccc2ccccc12 C1(C(C)(C)C)CC(CNC(=O)CP(C)(C)=O)CN(C(c2cncn2C)=O)C1 c1(N2CCC2)cc(C2CC2)nc(Cl)n1.C1(CC(=O)N(C)C2CC2)CCC(=O)N1C N1(C(c2cccc(OC)c2)=O)CCCC(F)(CNC(=O)CN(C)S(N)(=O)=O)C1 c1(OCC)c(OC)cc(C(=O)NCCCNC(C23CC(C)(C2)C3)=O)cc1Cl C(C(C)(C)C(=O)NC1CCOCC1NC(=O)CC1CNC(=O)O1)SC N1(C(c2c(CCC)n(C)nc2)=O)CC2CCN(C(c3cc(C)nn3CC)=O)C2C1 CCN=C(NCC12CC(C1)C(C)O2)NCC1(C(F)(F)F)CC1 N1(C(c2c(C)nsc2)=O)CCC(O)(CNC(=O)CC2CCC(=O)N2)C1 c1(Cn2c(C(CC)(COC)NC(C(C)C)c3cn[nH]c3)nnn2)ccc(C#N)cc1 C1(CNc2ncc(C)c(SC(C)C)n2)CC2CCC1N(C(=O)CSCCC#N)C2 c1(C(N2CCC(O)(C(C)C)C2)C(=O)NC2COC2)cccc2sccc12 c1(C(=O)NCC(CN(C(CC(=O)OCC)=O)C)C)cc2n(n1)CCN(C)C2 C1(CC(=O)N(C(C)CNC(=O)Cc2ccnn2C)C)CCCCC1C C(=O)(C(C)(CNC(=O)C(C)SC(C)C)CC)NC(CCC)CO C(c1ccncc1)=CC(=O)NC(CC(=O)NCC1(O)CN(C)C1)C1CC1 c1(CNCC2N(C(c3cocn3)=O)CCOC2)ccc2c(c1)Cc1ccccc1-2 C(=O)(CCCCCCNC(C1(C(C)(C)OC)CC1)=O)NCC(=O)NCC Cc1cn(CC(=O)NC2CCN(C(c3cnc(S)[nH]3)=O)C2(C)C)c2ccccc12 c1(C(=O)NCCCCN(C)C(C2CC=CCC2)=O)cncnc1-c1ccccc1 C1(NC(c2c(COC)ccs2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)C1(C)C C(=O)(C1=CCC(C)CC1)NCCOCCCNC(c1c(C)cccc1)=O c1(C(=O)NCC=CCC(=O)NCC(CSC)OC)c[nH]nc1C1CC1 c1(OC)cc(C(=O)NCC2(NC(C3CCC(O)C3)=O)CCCC2)ccc1F Cc1c(OCC(=O)N(C)CC2CCCN2C(C2(C#N)CCOC2)=O)cccc1Cl N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(C)C)=O)C(C)(C)C1 CCCC(Cl)C(=O)N1CCC(=CCNC(=O)C(=O)Nc2cccc(Cl)c2)CC1 C1(S(C)(=O)=O)(C(N2CCC(NC(C(CC=C)OC)=O)CC2)=O)CCC1 Nc1nc(C(=O)NC2CC(NC(=O)CC3CCCOCC3)C2)ccc1O N1(C(C2(C)C3CCNCC23)=O)CC2(CC(CN(CCO)C3CC3)CO2)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C1CNC(c1coc(C)c1)=O Cc1ccnc(C(=O)NC2CCC2CNC(c2c(C)c[nH]c2CC(N)=O)=O)n1 c1(C(N2CC(C)C(NC(C3(c4cccnc4)CCC3)=O)C2)=O)cnc2n1CCC2 C1(CC(=O)NCC(CC)(CC)NC(C(CC)F)=O)CCCCC1(F)F Cc1cc(F)c(NC(=O)NCC(=O)Nc2ccccc2)c(I)c1 CCC1=NOC(CC(N2CCN(C3CN(C(=O)Cn4nnc(=O)[nH]4)C3)CC2)=O)C1 C1(C#N)(C(=O)NC2(c3cn(C(CC)C)nn3)CCC(C)C2)CCOCC1 Cc1c(NC(C2CC2c2cccnc2)=O)n[nH]c1C1CC1 C1(C(=O)Nc2c(C)c(F)ccc2)COC2(CCN(C(C3(F)CCC3)=O)CC2)C1 C(=O)(CC1=NN(C)C(=O)C1)NC1C(C=C)CN(C(c2cnn3ccsc23)=O)C1 CC#CCCC(=O)NC1CCC(NC(c2cc(Cl)sc2NC(C)=O)=O)CC1 C#CCCCCCCC(=O)NCC(O)CN(C)C(c1ccc(P(C)(C)=O)s1)=O C1(NC(C=CC(CC)=CC)=O)CC2(C1)CC(NC(=O)C(N1CCSCC1)C)C2 C1(C(F)(F)F)(C(=O)NC2(C)CN(C(C3C(=C)CC3)=O)C2)CC2CCC1C2 Cc1ccc(F)nc1NC(=O)NCCCc1nc(-c2cccnc2)cs1 N1(C(=O)CC2(NC(=O)CCc3ncco3)CCC2)CCC2(CC(OC)C2)C1 C(=O)(CS(=O)(=O)CC(C)C)N1CCC(OCCNC(c2n[nH]c(C)c2C)=O)C1 Cc1csc2c(C(N3CC(C)(NC(=O)CC4CCCC45CC5)C3)=O)ncnc12 C1(NC(=O)CC2CC2)CCN(C(c2cnc(C3CC3)nc2O)=O)CCC1CO Cc1cc(C)c(C(N2CCC(NC(c3nncn3C)=O)C(F)C2)=O)c(=O)o1 C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(c1cc(C(F)(F)F)n[nH]1)=O N1(C(=O)CCc2cccnc2Cl)CC(CNC(=O)C(O)CC2CC2)C2(CC2)C1 c1(OC)ccccc1C(N1CCC(C)(NC(C2CC2(Cl)Cl)=O)C1)=O N1(C(C(C)C2CCCO2)=O)CCC2(CC1)CCN(Cc1ccn(C)n1)C2 N1(C(CCCC)=O)CCN(C(C2(N3CCCC3)CCC2)=O)CC1COC Cc1nc(N)cnc1C(=O)NCC1CCCCN1C(c1cc(C(C)C)n(C)n1)=O c1(SC)cc(C(N2CC3(CCN(C(=O)C(=O)NC4CC4)C3)C2)=O)c(Cl)cc1Cl CCC(CC(=O)NCCN1CCN(C(C2CCCCNC2=O)=O)CC1)C(C)C N1(C(C2CN(C(COCCCC)=O)CC23CC3)=O)CCN2CCCCC1C2 CC1(C)CC(CNC(c2ccc[n+]([O-])c2)=O)CN1C(c1cnn2c1SCC2)=O Cc1ccc(C(N2CCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)nc1 C1(CC(N2CCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)CCC2(CC1)CC2 c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)C2)=O)ncsc1S(N)(=O)=O n1(CCOC)nc(-c2cccc(C(F)F)n2)nc1C1CC(C)=NO1 c1(C(N(C2CC(NC(Cc3ccc(C)o3)=O)C2)C)=O)cnn(C)c1N C1(C(=O)NCC2(O)CCN(C(C3(O)C(C)(C)C3)=O)C2)CCC(F)(F)CC1 CN1N=C(C(=O)NCC=CCC(N2CC(C)(C)CCC2CO)=O)CCC1=O C(=O)(CCCCCN1CC(C(=O)OC)CC1=O)NC(CC)CNc1cc(C)ncn1 C1(NC(CCC=CC)=O)CS(=O)(=O)CC1NC(c1cccc(Cl)c1)=O c1(Cc2cc(C(=O)NCC3(NCC4CCC4)CCCC3)[nH]c2)ccc(CO)nn1 c1(C(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCC2)ncn2ccccc12 Cc1cc(Cl)ccc1C(=O)NC1CN(C(c2cc(Cl)on2)=O)CCC1C c1(C(=O)NC2CCN(C(C3C(COC)C3)=O)C2)cccc2c1OCC2 C(CNC(C1CCCC(O)C1)=O)(C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O C(=O)(CN=c1[nH]c(=NCC2CC(O)C23CCC3)[nH]c2c1SCC2)N(C)C C(=O)(C(C)(C)CC(=O)NCC1CCN1C(=O)CCCCc1cnc[nH]1)OC c1(N(C(C2CCOC2)CNC(=O)CC(=O)OC(C)(C)C)C(C)=O)ccc(F)cc1Cl CON1CCC(C(N2CCC(O)(C(C)NC(=O)C(=CC3CCCC3)C)C2)=O)CC1 Cc1cc(C=CC(=O)NC2CC2NC(C2CCC3(CC2)CC3)=O)c[nH]c1=N c1(OC)cc(=O)n(C)cc1C(=O)N(C)CC1CCN(C(=O)C=C(C)C(C)(C)C)C1 N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CN(C(=O)CC(C)(C)O)CC2(C)C1 C(C)(C)(CC(=O)NCc1nc(CNC(=O)C(C2CCOCC2)OC)cs1)OC c1(NC(CC)CNC(=O)C=Cc2cnc[nH]2)nc(Cl)nc2c1ncn2CC C1(C(=O)NCC2C(OC)CC2)CC2CCC(C1)N2C(=O)CCc1cccc(C)c1 CC(O)(CNC(c1coc(CNC(=O)C(F)OC(F)(F)F)n1)=O)C(F)F c1(C(=O)NC2C3CN(C(CCc4ccn(C)c4)=O)C2C3)ccc(F)c(CO)c1 C1(NC(c2[nH]c(=N)sc2)=O)CCCOC1C1CCN(C(N2CC3CC3C2)=O)CC1 C=Cn1nccc1C(=O)NC1CCN(C(=O)CCCOCCC)C1C(C)(C)C Cc1cccnc1C(F)(F)C(N1CCOC(CF)C1)=O c1(OC)cc(C)c(COC(=O)Nc2ccc3n[nH]cc3c2)cc1OC C=C(Cl)C(C)(C)C(=O)N1CCCC(NC(=O)C(F)(F)C(C)O)C1 c1(OC)cc(Br)ccc1C(=O)NC1CN(Cc2ccccn2)CC1C#N C1(Nc2c(C(N(C)C)=O)cccc2)CCC2CN(C)CC12 Cc1ccc(C(=O)NCCOC2CCN(C(C3CC(=O)CO3)=O)C2)n1C c1(C(=O)NCCN(C(CC=C)=O)CCCN(C)C)cc(Cl)cc([N+](=O)[O-])c1O c1(OCC(=O)NCCCN(C(c2c(C(C)C)cnn2C)=O)C)nc(O)nc(O)n1 C1(NC(=O)CCc2cccs2)CC2CC(C1)N(C(=O)C(O)Cc1ccccc1)C2 Cc1cc(C#N)cnc1C(N1CCC(C2CCCN2C(=O)C=C2CCC2)CC1)=O N1(C(C2CCC(CC)O2)=O)CCCC(C)C1CCNc1ncc(F)cn1 CC(CS(C)=O)C(=O)NCCC1(CNC(=O)CCNc2ccccc2)CC1 Cc1nc(C(C)(C)C)sc1C(=O)NC1CCN(c2ncc(Cl)cn2)C1C c1(C(=O)NCC2CCC(F)(CNC(C3(C)CCC(=O)C3)=O)C2)cnn2c1CCC2 N1(C(C)C(=O)NC(CC(=O)Nc2cccs2)c2cccs2)CCC(O)CC1 c1(C(c2nnnn2C)NCCNC(C(C)C)=O)cccc(C(F)(F)F)c1F c1(C(N(C2CC(C(=O)NCC(C(C)C)SC)C2)C(C)C)=O)ccc2c[nH]nc2n1 N1(C(c2c(NC)cnnc2)=O)CCCC(NC(=O)CCS(=O)(=O)N(C)C)CCC1 CN1C(=O)CCC1C(=O)NCC1(F)CC(CNC(=O)Cc2ccccc2Cl)C1 C(CC(C)CCCC(C)C)NC(c1cc(Cl)ccn1)c1n(C(CC)(C)C)nnn1 C(C(CC(C)C)C(=O)NCC12CC(C)(CCO1)C2)NC(C(C)=C1CCCC1)=O C1(CC(=O)N(CCC(C)NC(=O)Cc2cccc(Cl)c2)C)CCCCCO1 C12(NC(CC=C)=O)CCCC1(F)CN(C(c1cc(OC)cc(OC)c1N)=O)C2 Cc1occc1CC(=O)NC1CCN(C(=O)C(C2CCOCC2)O)C1 C(=O)(C(C(C)C)NC(=O)CC(C)NC(=O)CCC1CC1C)NCC c1(NC(=O)CN2CCCOC(c3ccccc3)C2)ccc2cnccc2c1[N+](=O)[O-] c1(C(N2CCCC(NC(C(CC)C(C)(F)F)=O)C2)=O)nc2sc(C)cn2c1C CC1(NC(C2CC2c2ccncc2F)=O)CCC(NC(c2nn[nH]c2Cl)=O)CC1 Cc1c(F)ccc(N)c1C(=O)NCC1(NC(C2CC3CC2C3)=O)CCC1 C1(C(=O)NCCc2c(C)nc[nH]2)CSCCN1C(=O)C(C)n1ccnn1 N1(C(C(C)OCC2CC2)=O)CCC(O)(CCNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(=O)NC(C2CCCN2C(=O)CCn2ccnc2C(C)C)C)CC(F)C(=O)N1 c1(C(N2C3C(NC(CNC(=O)OC)=O)C(CC3)C2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(C=CCOC)=O)CCC2(NC(=O)Cc3cc(F)c(C)cc3F)CCCCCC12 c1(C(N(C(C)CNC(c2cnoc2-c2ccc(Cl)s2)=O)CC)=O)cccnc1 C(=O)(C1CCCn2ccnc21)N1C(C(=O)Nc2nccc(C(N)=O)c2)CCCC1 c1(C(=O)NCCCCC(C)NC(C2CC(C)(C)CO2)=O)ncnc2c1CCC2 N1(C(C=CCCC)=O)CCOC(CCNC(=O)C(C)(C)c2cnn(C)c2)C1 c1(C(C)C)cccc(CNC(=O)NCC(C2CC(F)(F)C2)O)n1 C1(C(=O)OC)C2CCC(CC2)C1NC(C1CCN(Cc2ccccn2)CC1)=O Cc1ccc(F)cc1C(N1CCC(O)C(NC(=O)CC2CN3CCC2CC3)C1)=O c1(SC)cc(C(N2CC(O)(CNC(=O)CC3CCCC3C)C2)=O)ccc1[N+](=O)[O-] C(CCC(C)C)(C(=O)N1CCNC(=O)CC1C)NC(c1cc(C)no1)=O C(CCC(O)C(=O)NCC(C)Cn1ccnc1)NC(CC)=O C(CC1=CCCCC1)N(c1ccccc1)CC1CC(=O)NCC1 C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(c2ccncn2)C)C1C Cc1cnc2n1CCN(C(c1cccc(NCCOc3ccc(F)cc3)c1)=O)C2 c1(C(=O)NC(CCNC(C(c2scc(C)n2)C)=O)C)cccc(-n2cnnn2)c1 C1(C)(CNC(c2c(CC(C)C)onc2)=O)CCN(C(c2ccc[nH]2)=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCN(C)CC1CNC(C1CCCCC12CC2)=O C1(NC(CCN(C(CC)CC)C)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1C N1(C(C(C2CC2)OC)=O)CCC(C(C)NC(C2(OC)CCCOC2)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)Cn2cccn2)CC)CC(O)(c2ccccc2)C1 c1(C(=O)NC(CNC(CC=CC)=O)CC(F)(F)F)n[nH]c2c1CC(C)CC2 C#CC1CCN1C(=O)C(c1cn(C)nn1)NC(C1COC(C2CC2)C1)=O c1(C(C)=O)cnc(C(=O)NCC2(C)CCC(NC(=O)C=Cc3cccs3)C2)cn1 N1(C(C2C(CC)C2)=O)CC(NC(c2ccc(-c3ccncc3)cc2)=O)CCC1C Cc1noc(C)c1CCC(=O)N1CC(N(S(=O)(=O)CCCl)C)C1 c1(CCCC)noc(CCC(=O)N(C2CCN(C(=O)CCSCC)C2)CC)n1 N1(C(CC(CC)CC)=O)CC(C)CN(C(=O)CSc2ccc(C)c(C)c2)CC1C C1(C)(C(NOCC(=O)N(C)CC2CCN(CC)C2)=O)CNC(=O)N1 c1(C(N2CCC(NC(c3c(CC)nccc3)=O)C2)=O)ccc2c(c1)N(C)CC2 C1(CCCCNC(C=C(CC)C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 C1(C(N2C(CN(C)C(c3nn(C)cc3N)=O)CCC2)=O)CC12CC(F)(F)C2 c1(C(N2CC(OC)C(NC(c3ncoc3C)=O)C2)=O)cccc2c1CC(C)(C)C2 c1(C(N2CCC(C(N(CC(=O)N(C)C)CC)=O)C2)=O)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3c(CC)c[nH]c3)=O)CC2CC)cc(C)c(F)cc1F c1(C(N(CC(C)NC(c2c(CC)occ2)=O)C)=O)ccc2cccc(O)c2c1 N1(C(c2ccn(CCCC)n2)=O)CC2CC1C2NC(c1nc(C(C)C)oc1C)=O C(=O)(C(C)(C)CNC(c1ccns1)=O)NC(C)C1CC1 C(=O)(C(C)(C)C)NC(C)C(=O)N(C)CC1CN(C(=O)CC2CCCCC2)C1 c1(C(N2C(C)(CC)CC(NC(=O)CCC3CCC3)C2)=O)cc(=O)c(OC)cn1C C1(NC(CC(C)c2cnn(C)c2)=O)CCC(N(C)C(c2cc(Cl)cn2C)=O)CC1 c1(C(N2CCC2CC2CC(NC(C3CC3)=O)C2)=O)cnn(Cc2ccccc2)c1 N1(C(COCCC=C)=O)CCCC(C(=O)NCc2cnc(C(C)C)[nH]2)C1CC C1(C(=O)NCC=C=C)CC2CC1CN(C(c1ncc(F)cn1)=O)C2 c1(OCC)cccc(CNC(C)C(=O)NC2CCC(C)C2)c1 C1(C(=O)NC(CCOC)C(C)C)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(N2CCN(CC3CN(C(CC(C)F)=O)C3)CC2)=O)cc(C2CC2)nc(O)c1 N1(C(C(CC)F)=O)CCCCC1C1(CNC(=O)C(C)OC)CCC1 C12(NC(CCC=CC)=O)CC1CN(C(=O)COc1ccccc1O)C2 CCCC(C)CCCC(=O)N1CCN(C(=O)C2=CCOCC2)CC1 C(CC1=CCN(C(C23CC(C)(C2)OC3C)=O)CC1)NC(c1cc(SC)ncc1)=O N1(CC(=O)NCCOCCCNC(C2(C(=O)NCC)CCC2)=O)C(=O)CNC1=O CC1=C(C(=O)N2CC3C(CNC(=O)CCC(C)(F)F)C3C2)C=C2CCCN=C2N1 C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN(C(=O)C(F)C(C)(F)F)C2)C1 C1(N(CCc2ccc(OC)cc2)C(c2cnc(C)s2)=O)CCNCC12CC2 N1(C(CCOC)=O)CC(C(=O)NCC2CC(C(=O)OC)C2)C2(CC2)C1 C=C(Cl)CC(C(=O)NCCC1(COC)CC1)NC(=O)CCc1nc(C)no1 CC1CCN(C(c2ccoc2)=O)CCN1C(=O)CCN1C(=O)NC(C)(C)C1=O C(=O)(C(=O)NCC(C)NC(=O)Cn1cncn1)NCCCOC C1(CNC(C(SC)SC)=O)CCN(C(c2cc3c(s2)CCC3)=O)C12CCC2 c1(C(=O)OC)cc(Br)c(NC(C23CC2CN(C(c2nccn2C)=O)C3)=O)c(I)c1 C(=O)(CC(=O)NCCSC(C)(C)C)NC(C)CCNC(=O)CC1(C(F)F)CC1 N1(C(C=C(C)C)=O)CCC2(CC1)CC(C)N(C(c1ncoc1C)=O)C2 N1(C(C2N(C(C)C)CCC2)=O)CCC(N(C)C(c2cc(O)nn2C)=O)C(C)C1 Cc1nc2nccc(NCC3(O)CN(C(c4cc(C)oc4C)=O)C3)n2n1 C(CC(C(C)(C)C)NC(=O)COC1CCC(C)CC1)N(C(c1cnc(C)s1)=O)C C1(NC(C2(OC)CCOCC2)=O)CC2CN(C(=O)CCc3cccc(O)n3)CC12 S(=O)(=O)(c1ccc(Oc2ccccc2)cc1C)N1CC(OC)C2(C1)CC2 N1(C(C2(CCOC)CC2)=O)CCC2(CCC(NC(=O)Cc3cncs3)CC2)C1 Cc1ccc2cc(C(N3CC(C)(NC(=O)CNC(=O)OC(C)(C)C)C3)=O)ccc2c1 N1(C(C2C(CC)CCC2)=O)CC=CC(NC(=O)C(C)(C)Cc2cnn[nH]2)C1 C(=O)(C(=O)N=c1ccn(CC(N)=O)[nH]1)NC1C(c2cccc(OC)c2)C1 c1(C(=O)OC)ccncc1S(=O)(=O)NC1(c2ccc(Cl)cc2)CCCC1 C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CCCC(C)(C)C1 c1(C(=O)NCC(CC(=O)N(C(C)CS(C)=O)C)(C)C)cncc2[nH]ccc12 Cc1ccc(Br)nc1C(N1CCN(Cc2cnc[nH]2)CC1)C(=O)NCCC#N c1(C(C2CC2)NC(C2CCN(C(=O)Cc3cncnc3)CC2)=O)cccc(Cl)c1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CC2NC(C1(C(F)(F)F)CC1)=O C(=O)(C(CC(C)(C)C)NC(=O)CC1CC1(C)C)Nc1c(OC)ncc(C)c1 C1(C(N(CCn2ncc(C)c2)C)=O)C2CCC(C2)C1NC(=O)C=CC(=O)N(C)C N(C1CC2CCCc3cccc1c32)C(c1ccc([N+](=O)[O-])c(F)c1)=O CCCCCS(=O)(=O)CC(=O)NCCC1CN(C(=O)C(O)COC)CCS1(=O)=O C1(CC)C(C(=O)NC2CC(CNC(=O)CC(C)C)C2)CCN1C(=O)OC(C)(C)C c1(C(=O)NC23CC2CN(C(C24CC2CCC4(F)F)=O)C3)nccc2[nH]ccc12 C1(C(N(CCSC)CC)=O)CCCC(NC(=O)C=CC2CC2)CC1 C1(C2CC2)(NC(C(C)NC(C2CNC(=O)C2)=O)=O)CCOC1 N1(C(C(CC(F)F)N(C)C(=O)OC(C)(C)C)=O)CCC2(CC(C(F)F)=NO2)C1 C1(NC(C2C(NC(C(CN(C)C)N(C)C)=O)CCOC2)=O)CCC(=O)N(C)C1 c1(C(N2CCC(C(C)NC(c3cnsn3)=O)C2)=O)ccc(S(C)(=O)=O)o1 c1(OC)ccnc(CN2CC(c3cccc(C)c3)(F)C2)n1 N1(C(C=C(CCC)C)=O)CCCCC1CN(C(=O)CCc1ccon1)C CC(C)CC(C)C(=O)NC1CCCC1CNC(c1cc(C(F)(F)F)c(F)cn1)=O C1(CNC(C(CC)CO)=O)CN(C)CCN1C(=O)Cc1cccnc1OC N1(C(C(C)N(C)C)=O)CCC2(CNC(=O)C(C)(C)c3ccno3)CCCC12 c1(C(=O)Nc2c(OC)ccc(F)n2)nc2ccccc2[nH]1 C(=O)(C(=O)C(C)CC)N1CCC(CC#C)(C(=O)Nc2cnc(SC)nc2)C1 C1(C(N(C)Cc2onc(C)n2)=O)CCCCCC1NC(=O)CC1C=NN(C)C1=O n1(CC(=O)NCC#CCNC(CN(C(C)=O)C)=O)nnc(C)n1 C1(NC(=O)CSC(F)F)CC2CCC1CN2C(C1CCCC2(CC2)C1)=O Cc1cncc(C=CC(=O)NC2CN(C(=O)CC(C)c3ccncc3)CC2C)c1 C1(CNC(Cc2c(C)scc2)=O)CC(NC(=O)CNC2CCOCC2)C(O)C1 c1(OC)cccc2cc(C(=O)NC3CCCCNC3=O)c(=O)oc12 Cc1cc(=O)n(C)cc1C(N1CCC(N2CCN(C(=O)C(F)F)CC2=O)CC1)=O CS(=O)(=O)CCCCCCCC(=O)NC(c1ccc(Cl)s1)C(=O)O c1(C(=O)NC2CN(C(=O)CSc3nc[nH]n3)C2)c(Cl)oc2ccccc12 c1(C(=O)NC(CC#C)C(=O)NCCCN2CCOCC2)ccnc(C)c1N N1(C(C(C=C=C)C)=O)CC(C2CCCN(C(=O)C=Cc3cccc(Cl)c3Cl)C2)C1 C1(NC(c2c(C)n(C)nn2)=O)CC2CC1CN(C(=O)CCCN=[N+]=[N-])C2 C12(NC(C3CCN(CC(C)C)C3)=O)CC(CNC(=O)C(F)F)(C1)OC2(C)C N#Cc1cccc(-c2cc(CN3CCC(CC(N)=O)C3)ccc2OC(F)F)c1 N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(Br)s2)=O)C1 CCC(C)(C)C(C)CC(=O)N1CC2(C1)CN(C(c1cnnc(C3CC3)c1)=O)C2 C#CC1CCC(NC(=O)C#CCNC(c2ncccc2F)=O)C1 C1(C(NOCC(=C)C)=O)CN(C(C23CC(C#N)(C2)C3)=O)CC1(F)F CC(C)(CC1CCCO1)C(=O)N1CC(OCCNC(c2cnc(NC)cn2)=O)C1 c1(NC)cncc(C(N2CC(C(N3CCC(CCO)CC3)=O)(SC)C2)=O)c1 c1(C(=O)NC2CCC(CNC(c3cc(C#N)no3)=O)C2)cnc2ccccc2n1 N1(C(C(C)N(C(CCCOC)=O)CCOCCC)=O)CCC(N(C)C)C(C)C1 c1(C(=O)NCC2C(NC(CCc3ccn(C)c3)=O)C2)c(C2CC2)cccc1F c1(CC)cc(NC(c2[nH]ccc2CNC(=O)C(=O)NC2CC2)=O)cc(O)c1 Cn1nnc(C=CC(=O)NCCC2CCCN2C(c2ccc(F)cn2)=O)n1 c1(C(C(=O)NCC2C3CN(C(C4N(CC)CC4)=O)CC32)=O)ccc(F)cc1F c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)C)ccc(CO)cn1 Cc1c(F)ccn2c(NC(c3ccc(Cl)c(N4CCNC4=O)c3)=O)cnc12 CCCCC(C(=O)NC(C(C)C)c1ncc[nH]1)NC(=O)C=Cc1ccoc1 C(=O)(C(F)(F)C(C)O)NCC(C(C)(C)C)NC(C=CC(=O)OCC(C)C)=O c1(C(N2CC3CCN(C(=O)C=CC4CCCO4)C3C2)=O)ccn2c(O)nnc2c1 N1(c2n(CCCOCC)c(CCc3cccs3)nn2)CCC2(CCCO2)CC1 C1(NC(C(C)CC2CCCC2)=O)CCCC(CNC(=O)CSc2ccccn2)C1 CC(C)CCN=C(NCc1ccc(CO)cc1)NCC1CN(S(C)(=O)=O)CCO1 N1(C(C)C(=O)NCCC2(O)CN(C(c3scnc3Cl)=O)C2)C(=O)CCC1=O C(=O)(C1=CCC(C)CC1)NCC1OCCCN(C(C2(COC)CC2)=O)C1 C1(F)(CNC(C(F)=CC)=O)CN(C(=O)Cc2csc(Cl)n2)C1 CC1CCC(CNC(=O)CCCNC(N)=O)N(C(=O)CCc2ccccn2)C1 C1(N(C)C(C2CC2(C)Br)=O)CCN(C(C2(CC3CC3)CC2)=O)CC1 N1(C(C(C)(C)OC(C)=O)=O)CCC(CNC(=O)CN2CC(=O)N(C)C2=O)C(C)C1 CC1CCC2(CC1)CCN2C(=O)CCC1CCN(C(C2(CO)CCC2)=O)C1 c1(Cc2ccc(C3CCC(c4ccc(Cl)cc4)C3)s2)ccc(Br)cc1[N+](=O)[O-] c1(OC)ccc(C(C(=O)NC2(C)CC2)N(C)CCc2cc[nH]n2)cc1C N1(C(C2CCN(C(C3C(C)(C)C3)=O)CC2O)=O)CCC2(CC1)COC(=O)N2 Cc1cc(C#N)ccc1C(=O)NC1CC1CNC(C1CS(=O)(=O)CC(=O)N1)=O CC1C(NC(=O)CCc2ccncc2)CC2CCC1N2C(c1ccnc(Cl)c1)=O N1(C(c2c(C(C)C)noc2)=O)CC2CCCC2(CNC(=O)CSCC(F)(F)F)C1 c1(CC(N2C(C)CC(NC(C(C)CO)=O)C2)=O)c(O)ncnc1O N1(C(=O)C(Cl)=CCl)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)CCO2 CC1(O)CCCN(C(C2(F)CN(Cc3cncc(OC(F)(F)F)c3)C2)=O)CC1 c1(C(N(CC(C)(C)NC(c2ccc(CN(C)C)o2)=O)C)=O)cnc2n1CCOC2 c1(C(=O)NC(c2cn(C(c3cccnc3)C)nn2)(C)C)cc2scc(Cl)c2[nH]1 N1(C(C2(Oc3ccccc3)CC2)=O)CCC(O)C(c2ccccc2)C1 N1(CC(N2CC(O)CC(NC(Cc3ccc(C)o3)=O)C2)=O)Cc2ccccc2C1 C1(CNC(c2ccsn2)=O)CCCCCN1C(c1ccc(O)cc1)=O n1(CC(C)C)cc(S(=O)(=O)NCc2nc3cnccc3s2)cn1 Cc1ccccc1C(C)CC(=O)NCC1CCN1C(c1cccnc1)C(=O)N.C(C)C c1(OC(CC)C(=O)NC2(C)CCN(C(C3CC(C(C)C)C3)=O)C2)ccccc1C c1(CCOCC)nc(C(=O)NCCCN(C)C(C2CCCN2C(N)=O)=O)co1 CCCCC(O)C(=O)N1CCCC(N(C)C(c2ccc(O)cc2F)=O)CC1 C1(CC(=O)NC(c2ccccc2)CNC(C(C)SCCCC)=O)CCCC1(F)F CCC(C)C(O)CC(=O)NC(COC)CC(=O)NC1CCC(=O)NC1(C)C N1(C(CC2CN(C)C2)=O)CCC(CO)C(NC(c2ncccc2NC(N)=O)=O)C1 c1(N(C2CCN(C(C)C)C2)C(c2nn(CC)nc2C)C)nc[nH]c2nccc1-2 Cc1cc(C)c2nc(N3CCC(NC(c4ccnn4CCF)=O)C(F)C3)sc2c1 CC(C)CC(C)(C)C(=O)N1CCC(C)C(NC(c2ccccn2)=O)C1 Cc1cccc(N(C)C(C23CC(CN2C(=O)Cc2cccnc2)C3)=O)c1C c1(C(N2CCC(C)(OC)C2)=O)ccc2c(c1)CCCC2=O Cc1cc(C(N2CCOC(CC(=O)NC3CC3c3ccn(C)n3)C2)=O)ccn1 C1(C(=O)N(C2CC(NC(C3CCOCC3)=O)C2)C)(CC)CCOC1 N1(C(C=CCNC(C(CCCC)=O)=O)=O)CCCC2NC(=O)CC12 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1(F)CC(NC(=O)C=CCF)C1 N1(C(c2c(N)n(CCO)nc2)=O)CCOCC(CNC(=O)Cn2nccn2)C1 c1(C(C(=O)NC(CN(C(C2CC3(CC3)C2)=O)CC)C)C)ccc(C)s1 C(C(CC(C)C)NC(=O)CC1CC(n2cnnc2)C1)NC(Cc1cc(C)on1)=O c1(C(CC(=O)NC2(C(=O)OC)CC2C)N)ccc(F)c(F)c1 CC(C)C(CNC(C1(Br)CC1)=O)NC(=O)COc1cn[nH]c1 O(NC(=O)C(CCSC)NC(c1cc(C)c(C)o1)=O)CCCC#C C1(CC)CCC(C(N2CCC(CNC(=O)CCCC3CCCCC3)C2)=O)O1 c1(OC)cccc(CNC(C2C(N)C3CCCCC23)=O)c1Br Cc1cnc(C(=O)NCC2C3CC2N(C(c2ccc(C4CC4)cn2)=O)C3)c(F)c1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(c2ccc(F)cc2)=O)c1 N1(c2cc(OCC)nc(C)n2)CCC(C2CCCN(C(=O)CC3CC3C)C2)CC1 c1(C(=O)NC2CN(Cc3cccc(Cl)c3)CC2F)ccc2cccc(Cl)c2n1 CC(C)C(CNC(C1CCN1C)=O)N=c1nc(Cl)[nH]c(C)c1C#N N1(C(C2C(CC)N(C(c3cc(C)nc(O)n3)=O)CC2)=O)CC2CCC1CC2 CC1CN(C)C(C)CN1C(C1CN(CC#N)CCC1(F)F)=O Cc1cc(C(=O)NC(C)CCNC(c2ccsc2Cl)=O)c(N)c(Cl)n1 c1(OCC(=O)NCC(CN(C)C(C2COCCO2)=O)O)ccc(C#N)cc1Cl n1(CC)nnnc1C(C1CCCC1O)(C)NCCC(C)F C12(NC(CC)=O)CC3CCC(C1C2)N3C(c1nn(-c2ccccc2)cc1OC)=O c1(C(C(N2CC(N(C(CC3(OC)CCC3)=O)C)C2)=O)O)ccc(Br)cc1F C(=O)(C(C)C(O)C(C)C)NC(CCNC(CC1(C=C)CCC1)=O)(C)C N1(C(=O)CC2COCCO2)CC2CCCC2(C(=O)NC2C3CCC4C(C3)CC24)C1 c1(C(CC(=O)NCC(CNC(C(C2CCC2)OC)=O)(C)OC)C)ccc(C)cc1 C1(NC(=O)NC(C(O)C(F)(F)F)C2CC2)CCC2(CCOCC2)C1 N1(C(c2ccc(OCc3c(CC)cccc3)cc2)=O)CCS(=O)(=O)C2CCCC12 N1(C(C(C)(C)CO)=O)CC(N=c2ncc3ccccc3[nH]2)C(C)(C)C1 Cc1c(C(N2CC(N(C(=O)C3CCc4c[nH]nc43)C)C2)=O)[nH]c2c(C)cccc12 C(CC(=O)NCCCCC1CN(C(=O)COC2CCC2)C1)NC(C1C(C)C1)=O CC(C)CCCCCC(=O)N(CCC(N1CCCC1CCC(C)C)=O)C c1(C(=O)NC(C(C)NC(=O)CC2CCC=CCCC2)(C)C)cc(O)cc(F)c1F Cc1ccncc1C(C)NC(c1cn(C(C)(C)C)nn1)c1nnnn1C C1(NC(C2CCC(OC)CC2)=O)CC2(C1)CN(C(c1cnc(Cl)cc1I)=O)C2 N1(C(C(C)(C)CC2CC2)=O)CCC2CN(C(=O)CC(F)(F)Br)CC2C1 C1(CNC(C2(C(C)C)CCC2)=O)CC2CCC1N(C(=O)CCc1cccs1)C2 CC1CCC(CO)N(N(CCN2CCN(C)CC2)CCO)C1 c1(C(N(CCCN(C(CSCCC)=O)C)C)=O)cc2c(=O)n(C)c(=O)n(C)c2s1 N1(c2n(CCC#C)c(-c3cccn3C)nn2)Cc2ncnc(O)c2C1 CON(C)C(=O)C(C)(C)NC(=O)C(=O)NC1CC2(C1)CC(N)C2 Cc1ccc2snc(C(=O)NCC(C3CC3)NC(C3CC(N(C)C)C3)=O)c2c1 N1(C(C(CC=CCC)C)=O)CCCC2C(NC(c3cc(C)sc3N)=O)C(C)(C)C12 C=CCC(C(=O)OCC)NC(=O)C(COC)NC(c1ccn(C)c1C)=O C(=O)(C(O)CC(C)(C)C)N1CC(CC(C)NC(=O)CCNC(=O)C(C)(C)C)C1 N1(C(Cc2cccc(C)c2)=O)CCC=C(C(=O)Nn2nnc(C)c2C)C1 c1(C(N2CC=CC(NC(c3c(CC)nn(C)c3Cl)=O)C2)=O)coc2c1CCCC2 C12(NC(=O)Nc3cc(OCC)ncc3)CCC(C)(C1)OC2 n1(C(C)C)cc(C(c2nnnn2C(C)(C)C)NCCC2CCCC2)cn1 N1(C(CC(C=C)C)=O)CCN(C(c2cc(Cl)n[nH]c2=N)=O)C2CCC12 c1(CCC(=O)NCCN(C(C2(OC)CCC(C)C2)=O)C)c[nH]c2cc(C)ccc12 N1(CC(N2CCCC(C)(CNC(C3CC(O)C3)=O)C2)=O)CCc2sccc2C1 CCCCS(=O)(=O)NCC(=O)N(CCCN(C)CC1CCC(O)CC1)C N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2sc(O)nc2O)C(CCO)C1 c1(C(=O)NCCOCCN(C(c2cccc(C)c2)=O)C)cccc(Cl)c1Cl C(=O)(C(C)(O)CC(F)(F)F)N(CCCNC(C(C1CC1)OC)=O)C1CC1 c1(C(=O)NCC2C(C)CCN(C(=O)CS(C)(=O)=O)C2)cnc2c(Cl)cccn12 Nc1cc(C(=O)NCC2CCN2C(C23COCC2C3)=O)ccc1-n1cncn1 Cc1cncc([N+](=O)[O-])c1N1CCC(CN(c2ccnc(C(C)(C)C)c2)C)C1 N1(C(CC(C)C)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1F C(=O)(C1=CCC(C)(C)CC1)NCCCN(C(C1CC1(C)C(F)F)=O)CC n1(CC(=O)NC2CCN(C(COCCCCC)=O)C2C(C)C)cc(F)ccc1=O CC(F)(F)CC(=O)NC(Cc1cnc[nH]1)C(=O)NC(CO)CCF c1(C(N2CCC(N(C(C(CC)NC(N)=O)=O)C)C2)=O)nnc(C)cc1O C(CO)(C(=O)NCc1cnn[nH]1)NC(C(c1ccn(C)c1)C)=O n1(CC(=O)NCC(CC)(CC)NC(=O)C(C)NS(C)(=O)=O)ccc(=O)cc1C c1(C(=O)NC(CN(C(=O)C(c2ccc(O)cc2)=O)CC)C)cc(C2CC2)ccn1 c1(C(CNC(=O)C(F)=C(C)C)NC(c2nnc(CC)s2)=O)ccccc1OC N1(C(COCC(=O)OC(C)(C)C)=O)CCCC(CCNC(c2cc(F)cs2)=O)C1 N1(C(C)=O)CCc2cccc(C(=O)NC3(c4ccc(Br)c(Cl)c4)CCC3)c2C1 C1(C(=O)N)CC(C2CC2)=NO1.c1(CC)cc(CCCN(C2CC2)CC)sc1C c1(C(=O)NC2CCCCN(C(c3cncc(C)c3C)=O)C2)cc2ccncc2[nH]1 C(c1cccc(Br)c1)=CC(=O)NC(CNC(C=COCC)=O)CO CC1(C)COC1C(=O)NC(CNC(c1occc1Br)=O)C1CC1 Cc1cc(C(=O)NC2CC(CC(=O)NCc3cccnc3Cl)C2(C)C)c(C)s1 N1(C(C2C(C)N(C(c3nc[nH]n3)=O)CC2)=O)Cc2cccnc2C1 c1(C(=O)NC23CC(NC(CSC)=O)(C2)C3)ccc(Br)cc1O c1(C(=O)Nc2scc(C3C(C(=O)OC)C3)n2)c(Br)cnn1C C(=O)(C#CC1CCCC1)NC1CC(NC(C2CC(C)NC(=O)C2)=O)CC1O C1(CN(C)C(c2ccncc2)=O)CN(C(c2cn(C3CC3)nn2)=O)CCO1.ON c1(CC(=O)NC2(CCNC(CNC=O)=O)CCC2)cnc(C2CC2)[nH]1 c1(NC(C(N2C(NC(=O)OC(C)(C)C)CC2)=O)=O)cn(C(F)F)c2ccccc12 C1(C(=O)NCC=CC(=O)NC(c2ccco2)c2cccs2)CCCCN1C1CC1 C1(OC)CN(C(c2cnc(C(C)C)o2)=O)CC1NC(C1(c2cc[nH]n2)CC1)=O N1(C(=O)CCc2cncnc2)CCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(C3(CCN(C)C)CC3)=O)C2)cc1C C1(NC(c2ccc(C)o2)=O)CCN(C(c2ccccc2SCCO)=O)CC1C c1(C(N2CC(NC(CC(=C)C)=O)C(C)C2)=O)cn2c(n1)CC(C)CC2 C1(C2CC2)(CNC(=O)C2=C(Cl)CCC2)CCN(C(c2nc[nH]c3nccc2-3)=O)C1 CC1CN(C(=O)CC(C)(C)C)CCN1C(=O)C(c1ccc(Cl)s1)C C1(C(=O)NC2CN(C(=O)Cc3ccc(O)cc3)C2)CCCN(c2ccncc2)C1 C(C(CC)CC)(c1oncn1)NC(COC)=O.c1ccccc1 N1(C(C(C(CC)CC)F)=O)CCC2CN(C(=O)C(C)C(CC)CC)CCC2C1 CCC(C#N)(CC)C(=O)N1CCCC(CN(C(=O)CCc2ncccc2C)C)C1 c1(C(=O)Nc2nc(-c3ccsc3)cs2)ccc(S(=O)(=O)Cc2ccc(Br)cc2)cc1 Cc1ccc(NC(C2CC(F)CN2C(=O)Cc2ccccc2)=O)c(C)c1C C1(CNC(c2c(C)onc2C2CC2)=O)N(C(c2cncs2)=O)CCC1(C)C c1(OCC)cccc(C(=O)NCC2(CO)CCN(C(C3CNC(=O)N3)=O)C2)c1N S(=O)(=O)(c1ccc(NCCCN2CCN(C)CC2)cc1Cl)N1CC(C)=C(C)C1 N1(C(CC(CC)(F)F)=O)CC2(CCC2)CC1C(=O)NC1CN(C)CC1C C(CCO)(C(F)(F)F)NC(N1CCN(c2cc(C3CC3)[nH]n2)CC1)=O c1(OC)ccc(Cl)cc1C=CC(=O)NCC(O)CNC(c1cnc(Cl)[nH]1)=O C(c1c(Cl)cccc1Cl)=CCNC(CCCCNC(=O)OC(C)(C)C)=O N1(C(COCc2c(C)cccc2)=O)CC(C)N(C(=O)CCC2OCCO2)CC1C c1(C(=O)NCCC(=C)CNC(c2ccc(C3(C)CCO3)cc2)=O)cc(=O)cc[nH]1 C(CCc1cn[nH]c1)(C(=O)NCC(O)CF)NC(=O)OC(C)(C)C C1(NC(C(C=C)CC)=O)CCC2CCN(C(=O)C3=CCOCC3)C1C2 c1(C(=O)NCCC23CCC2CN(C(=O)C(Cl)=CCl)C3)cc2ccccn2n1 CC(C)(C)CC(O)C(=O)N1CC(F)(F)CC1C(=O)NC1CCNC1=O N1(C(c2cccc(OC)c2)=O)CCC2(NC(=O)CCC3CC3(C)C)CCCC12 Cc1nc(C2CC2)ncc1NC(=O)CCCNC(=O)CN1CCCCCC1 C(=O)(C(C)(C)C(N)=O)NC(CCOC)CNC(=O)C(c1ccccc1)SC CC1(C)CC(CC(=O)NC2C3CCCC23)N(C(c2ncncc2Cl)=O)C1 CC1(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)CCc2ccccc2C1 C1(C(N2C(CNC(CCCCCSC)=O)CCC2)=O)Cc2ccncc2C1 c1(C(=O)NCC2CN(C(CCC(=C)C)=O)C2)ncn2c1COCC2 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)c[nH]c2cccnc12 C1(NC(c2c(CCNC(C(C)(C)N=[N+]=[N-])=O)n[nH]c2)=O)CCc2nncn2C1 c1(C(=O)OC)ccncc1C(=O)NC1CC(NS(=O)(=O)CCCOC)C1 N1(Cc2c(OC)cc(O)cc2)CC2OCCN(C(c3nc(C)cs3)=O)C2C1 C12(CNC(CCCNC(N)=O)=O)CCC(CC1)N2C(c1cc2n(c1)CCC2)=O C(CCC1CC1)(C(=O)N1CCCCCC1)NC(c1ncncc1Cl)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCCCC1)CNC(c1n(CC)nnc1C)=O N1(C(c2nc(COC)oc2)=O)CCCC(NC(C2CCCC2C(F)F)=O)C1 N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CC2C3C=CC(O3)C2C1 c1(C(N2CCN(C3C(NC(C(CCC)C)=O)CCC3)CC2)=O)cc(O)ccc1C C1(CC=C)(NC(c2[nH]nnc2C)=O)CCN(C(c2nnc(C)s2)=O)C1 c1(C(=O)NC2CCCC(CNC(C(C)(C)SC)=O)C2)ccc(O)c(CO)c1 C1(C)(C(N(CC(CN(C)C(C2CC3CCC2O3)=O)O)C)=O)CCC(=O)C1 c1(C(N2CCC(N(C(C(=O)NC(CC)C)C)CC)C2)=O)cccc(C(F)F)c1 c1(SCC(N2CC(O)(CNC(C3(C(C)C)CCCO3)=O)C2)=O)cc(F)ccc1F n1(CCN(CC)CC)nc(-c2cc[nH]n2)nc1C(C)Sc1nccn1C N1(C(Cc2c(C)noc2Cl)=O)CCCC2(NC(=O)Cc3cccs3)CC2C1 C1(C#N)(C(=O)NC2CC3(CN(C(C4N(CC)CCC4)=O)C3)C2)CC2CCC1CC2 N1(C(C2(C#N)CC2)=O)CC(C(=O)NCCC2CCCC23CC3)C2(CCC2)C1 Cc1cc(=NCC(C)C#N)[nH]c(N(C)Cc2sccc2C)n1 c1(C(N(CC(C)NC(c2cc(C)nc(O)n2)=O)C)=O)oc2ccccc2c1CO C1(C(N(CC(C)CNC(c2cc[nH]c2)=O)C)=O)CCC(=O)C1 c1(C(=O)NC(CNC(c2ccc(COC)cc2)=O)C)cc(C)cc(Br)c1 Cc1[nH]nc(C(=O)NC2(C(N3CC(n4cnnc4)C3)=O)CC2(C)C)c1Cl C1(CN(C(=O)C(C)SC)CC)CCN(C(=O)C=C(C)C2CC2)CC1 CCS(=O)(=O)CC(=O)N1CCCC1CCN(C(C1CCN(C(C)=O)CC1)=O)CC C=Cn1nccc1C(=O)NC1CCN(C(=O)CC2CNC(=O)O2)CC1 n1(CCOC)ccc2cc(C(=O)NCCN(C(C3C(C)C3C)=O)CC3CC3)ccc12 c1(SCC)cnc(O)c(C(=O)NCCC(C)(C)NC(c2nc(O)c(C)s2)=O)c1 c1(CC(=O)NCC2CC(NC(C(C)O)=O)C2)csc2nccn12 CC(C)CCN(CC(=O)NC1(CCC(=O)NC2CC2c2ccoc2)CCC1)CC C(=O)(C1=NN(C)C(=O)CC1)N1CC2C(CNC(CC(C)N(C)C)=O)(C2)C1 N1(CCNC(C(C(C)OC)O)=O)CCCN(C(c2nonc2N)=O)CC1 Cc1ncc(C(=O)NC2CCCCN(C(c3ccnc(O)c3)=O)C2)c(C(C)C)n1 N1(C(C(=O)NCC(F)F)=O)CC(C(=O)NOCC2CCCC2)CC12CCC2 c1(NC(C(n2cc(C3CCC3)nn2)C)=O)ccc([N+](=O)[O-])cc1F N1(C(CC(=O)NCC#C)=O)CCC(C)C1CNC(=O)CSc1ccc(C)cc1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CCNC2=O)=O)ccnc2ccsc12 C(=O)(C(C)CS(C)(=O)=O)NCC12OC(C)C(NC(=O)C=Cc3cn(C)cn3)(C1)C2 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(N(C)C(C1CCCC(C)C1)=O)C2 c1(C(N(CCCNC(C2CC3CC2C3)=O)C(C)C)=O)cc2n(n1)CCCO2 Cn1ncc2cc(C(=O)NCC3C4CN(C(C5CCS(=O)(=O)N5)=O)CC34)cnc12 Cc1c(C(=O)NC2CCC2CNC(=O)CCC(C)(C)N(C)C)ccc(F)c1F c1(CCC(=O)NC2C(NC(c3c(C)ccnn3)=O)CCCC2)ccccc1C#N C12(C(=O)OCC)CCC(C(=O)NCCN(C(=O)C(C)CCOC)C)(CC1)CC2 Cc1cc(C(N2CCC(C)(CNC(=O)CC(O)C3CCCC3)C2)=O)nn1C1CC1 C1(C(CNC(CN(S(CC)(=O)=O)C)=O)C)CCN(C(C2C(C)C2C)=O)CC1 CC1CC(N=c2[nH]c(N3CCC(C(F)(F)F)CC3)nc3c(F)cccc23)CCO1 c1(COC)ncc(C(=O)NCC(C2CC2)NC(c2cc(-c3ccco3)c[nH]2)=O)s1 c1(OC)ccc(CN2CC3CC3(C(=O)Nc3ccccc3)C2)c(Br)c1OC CCCCC(O)C(=O)N1CCCC(O)(CNC(=O)C=C2CCC2)C1 Cc1nc(O)nc(O)c1CC(=O)NC1CCCC1NC(=O)C(C(C)(C)C)C1CC1 N1(C(Cc2c(C)ocn2)=O)CCCC12CCN(C(C1C(C)(C)C1(F)F)=O)C2 C1(C2CC2)(CNC(CNC(CC)=O)=O)CCN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(CC(CC)(F)F)=O)CC2OCCN(C(c3cnc4[nH]nnc4c3)=O)C2C1 C1(C(=O)NCC(CN(C(=O)CSCC2CCCO2)C)(C)C)C2CCCOC12 N1(C(CCCOCC)=O)CC2CC(NC(c3cc4cnn(C)c4s3)=O)CC2C1 C(=O)(C(F)C(C)CNC(c1cnc(O)cc1C)=O)NCc1cn(CC)nc1 C(=O)(C(CC)CC(F)(F)F)N(C1CCN(C(c2c[nH]cc2CC)=O)CC1)CC#C CN1C(=O)OCC1NC(=O)NCCCCCCn1cc(-c2cnccc2Cl)nn1 C1(CNC(c2c(OC)cnnc2)=O)(CO)CCCN(C(C2(C)CCCCC2)=O)C1 c1(CC(=O)NCCN(C)C(c2ncccc2C(F)(F)F)=O)c(F)cccc1C#N N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NC2CCC3(CCC3)C2)CC(C)(C)C1 C1(OC)CCC(C)(C(=O)NC2CCCN(C(C3CCC(C)O3)=O)C2C)CC1 c1(C(C(=O)NCc2ccccc2Cl)N(C)Cc2ncco2)ccc(F)cc1F c1(OC)ccccc1C(c1ccc(Br)s1)N(CCC(N)=O)CC(C)C N=c1[nH]c(NC(CC2CCCO2)CO)ncc1C(F)(F)F C1(C(=O)O)CC2CCCCC2N(C(=O)CCn2ccnc2)C1 c1(NC(C)=O)ccc(C(=O)NCC#CCNC(=O)CN(C)CCOCCO)o1 CCC(C)CCCC(=O)N1CC(C)C1C(N1CC2(C1)CN(CC)C2)=O CCCS(=O)(=O)CC(=O)NC12CCN(C(c3c(C)cc[nH]c3=N)=O)CCC1C2 C12(C(N3CCC(C(C)NC(c4cc(=O)cc[nH]4)=O)C3)=O)CCCCC1OCC2 C(=O)(C#CC1CCCOC1)N1CCCCC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 c1(-c2n(CC=C)c(N3CCNC(=O)C3)nn2)ncc(C)cc1F c1(C(=O)NCCNC(c2cc(C3CC3)no2)=O)n[nH]c2c1CCOC2 N1(C(C2CC(C)C2)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC(C)(C)C1 c1(CCC(=O)NCC#CCNC(=O)C2=CCSC2)cc(F)cc(Br)c1 C1(CC)CCCCC1C(=O)NC1(CO)CN(C(c2cc(C3(O)COC3)on2)=O)C1 C1(CNC(Cc2cnc(C)s2)=O)(CO)CCN(C(c2sccc2C)=O)C1 c1(C(=O)NC2C(C(=O)Nc3ncc(C)nc3)C2)ncc(Cl)cc1C c1(CN2CC(NC(c3cnc4ncccn34)=O)C(O)C2)c[nH]c2ccc(F)cc12 C1(CNC(COC2CCN(C)CC2)=O)CCCCCN1C(=O)CCc1cccs1 N1(C(c2c(C)onc2)=O)CCCC2(C1)CN(C(C1CCCN1C=O)=O)CCO2 C(CCCCCNC(=O)Cc1cc[nH]c1)N(C(=O)CC1CC1(C)C)C O=C1NCC2(CCN(C(CC3CCOC3)C(=O)NC3CCCCC3)CC2)N1 c1(NC)ccc(C(N2CCC(C(=O)NCC34CCC(CC3)O4)C2C(C)C)=O)cc1 c1(OC)cc(OC)nc(Cc2nc(CCCO)nn2-c2ccnc(Cl)c2)n1 c1(CC)ccc(F)c(C(=O)NC2(CF)CCN(C(=O)CCCNC(=O)OC)C2)c1 CCCCS(=O)(=O)NC(C)C(=O)N(CC(C)NC(=O)COCCOCC)C c1(N2CC(CN(C(c3c(C)cn(C)n3)=O)C)OCC2)cc(C(N)=O)nc(Cl)n1 C1(CC)CCCC(N=c2[nH]c3c(c(=NCc4nnc(C(C)C)n4C)[nH]2)SCC3)C1 C(=O)(C1=NOC(C)C1)N1CCC(C)(CC(=O)NCc2nnc(C)n2C)C1 N1(C(C2C(C(=O)OC)C2)=O)CC2C(NC(=O)Cc3cnc[nH]3)CS(=O)(=O)C2C1 CS(=O)(=O)C1CC(C(=O)NC2CCC(CNC(=O)CCc3cc(Cl)no3)C2)C1 c1(C(=O)NCC2CN(C(C3CN(CCC)C(=O)C3)=O)C(C)C2)cc(Cl)ccc1F c1(CNC(C(C)N(C(COCC(=O)OC)=O)C2CC2)=O)cccc(F)c1F CC(C)CS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1NC(=O)CC1CCCC(=O)C1 CC(C)(C)C(CNC(c1csc(O)n1)=O)C(=O)NCC12CCC(CO1)C2 N=c1ccc(C(N2CCCC2CCCNC(C2CC3C=CC2CC3)=O)=O)c(Cl)[nH]1 C(N=c1nc(N2CCC(OCCO)C2)c2c([nH]1)CCCCC2)c1nnn(C)n1 CCCC(C)(O)C(=O)N1CCC(C(=O)NCCc2cccc(O)n2)C1 c1(C(=O)NCCCNC(C2CC(c3ccc(F)cc3)C2)=O)nnn2c1CSCC2 C(=O)(CCCC(=O)OC)NCC1C(NC(CN(CC)CC)=O)CCCC1 C1(NC(=O)CCc2cccs2)CC2(C1)CN(C(=O)Cn1ccc(C3CC3)n1)C2 c1(C(=O)NC2CC(N(C(C(CC)O)=O)C)C2)cc(OC)cc2c1CCC2 C1(C#N)(NC(N(C(C)C)CC2CCC(C)C2)=O)CC1C(F)(F)F c1(C(=O)NCC(C)NC(Cc2c(C)noc2Cl)=O)nc2c(s1)CCCC2 c1(C(=O)NC2CCCC2CNC(C2(c3ccno3)CCC2)=O)cc[n+]([O-])cc1 c1(C(=O)NC(c2ccccc2)C(C)NC(C=C(CC)CC)=O)ncc[nH]c1=O N1(C(c2ccc(OC)cc2)C(=O)NC2CC(F)(F)C2)CCCC(C)(O)CC1 N1(C(Cc2onc(C)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)C)CC1 C1(F)(CNC(=O)Cn2ncnn2)CCC(NC(c2cc[nH]c2C(F)F)=O)C1 N1(C(=O)CCC2CCOC2)CCN(C(C2CCCCS2)=O)C(c2ncc[nH]2)C1 N1(C(C(CC=CC)NC(=O)CN(C)C(=O)C2CC2)=O)CCOC(C)(CC)C1 c1(C(=O)NCc2ccc(CNC(C(C)(C)SC)=O)cc2)cncc(Cl)c1C c1(OC)ccc(C(=O)NC(C2CCN(C(c3cccnn3)=O)C2)C)nc1Cl C1(NC(c2c(C)cco2)=O)CCC2CCN(C(C3CCCC34CC4)=O)C1C2 N1(C(C2C3(CC(NC(COCC=C)=O)C3)C2)=O)CCC2(CC1)CC2CO C1(NC(C2COC(C)(C)O2)=O)CCC2CN(c3cnc4ccccc4n3)CC2C1 C(C(C)(C(=O)NC1CCC(C(=O)N(C)CC2CCCC2(C)C)C1)OC)OC N1(C(c2c(C)noc2N)=O)CC(CNC(=O)C(C)OC2CCCC2)CC(C)(C)C1 Cc1nc2ccnn2c(C)c1C(=O)N(CCCCCNC(=O)CN(C)CCO)C C(=O)(C(F)(F)C(C)(C)O)N1CCC(C)C(NC(=O)C(O)C(C)(C)C)C1 c1(C(=O)NC(C)Cc2ccccn2)c(CNC(C2(C)CS(=O)(=O)C2)=O)nnn1C C#CC1CCN(C(=O)Cn2cc(CCNC(=O)OC(C)(C)C)nn2)CC1 c1(C(=O)OCC(N2CCC(C)C(C(=O)NCC(F)(F)F)C2)=O)cnn2ccncc12 Cc1oc(CNC(C2(O)CC(=O)C2)=O)nc1C(=O)NC1CCOC1(C)C C1(NC(C(C=C)(C)C)=O)CC(C(=O)NCCNS(N)(=O)=O)=CC1O N1(CCC(C)C)CCCC1C(=O)NC1CCC1CNC(c1ncnn1C1CC1)=O O(N(C)C(=O)CN=c1nc2c(cnn2C)c(N2CC3CCOC3C2)[nH]1)CC N1(C(CCSC)C)CCC(C)C(C)(C)C1.C1(N)CCc2cncn2C1 N1(C(c2ccc(C)c(C)c2)C(=O)NC(C(=O)OC)C)CC(C)Cc2ccccc21 CC1CCC(CC(=O)N(CC(=O)NCc2ccnn2CC(F)F)C)O1 N1(C(C(N2CCOCC2)C)=O)CC2CCC2(CNC(C2(F)CC3(CCC3)C2)=O)C1 c1(NC(C2(C)CCN(C(Cn3ncn(C)c3=O)=O)C2)=O)ccc(O)c(F)c1 N1(C(CC=C=C)=O)CC(NC(C2CC2(Cl)Cl)=O)CC2(CC2)C1 C=C1CC2(C1)CC(C(=O)NCCCOCCNC(=O)C(C1CCOCC1)C)C2 C1(C2CCN(C(=O)Cc3ccc(Cl)cc3)C2)(NC(C2CCC2(F)F)=O)CC1 C1(C(=O)NCC2C(C(NOCCC=C)=O)C2)CC=C(C)CC1 C1(NC(c2c(C)nns2)=O)CC(CNC(c2ccc(=O)oc2)=O)C1(C)C CCCCC(O)C(=O)NC1CCCC1CNC(=O)COc1ccc(Cl)c(CC)c1 c1(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)cccc(Br)c1F C(=O)(C1CCCn2cnnc21)NCC(C)CNC(=O)Cc1cccnc1Cl c1(CC(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(Cl)cc1C C1(NC(C2CCCCN(C(c3ccc(C)s3)=O)C2)=O)CCCC(C2CC2)C1 Cc1c(CNC(C2CC(C)(F)C2)=O)sc2cncn12 N1(CCSC)C(=O)NC(c2ccc(C)nc2F)C2=C1CN(c1ccccc1)C2=O C1(C(F)(F)F)(C(=O)NCC2N(C(=O)Cc3ccns3)CC=C2)CC=CCO1 O=[N+]([O-])c1cnn(C2CCCC2)c1NCc1ccc(C(F)(F)F)cc1F c1(C(N2CC(C(=O)NCCCCN(C)C)C(O)CC2)=O)cc(Cl)c(F)c(Cl)c1 c1(C(=O)OC)ncc(NC(C23CCC2CN(C(c2cccnc2)=O)C3)=O)cc1Cl C1(C)(COC(=O)CNCC(=O)NC(C(CCC=C)C)C)CCS(=O)(=O)CC1 c1(NCN2C(=O)CC(CCOC)C2)[nH]c(=NCC(CO)C2CC2)nc2sccc12 C1(NC(c2scc(COC)c2)=O)CCC2CCC1OC2 c1(NC(c2c(NC(c3c(C)cn(C)n3)=O)cccc2)=O)ccc(O)c(C(C)C)c1 C=C1CC2(C1)CC(C(=O)NC(c1ccc(CNC(=O)COC(C)C)cc1)C)C2 C(CCCC(C)(C)C(=O)NNC(=O)c1ccc(C)s1)NC(C(CC)C)=O C(C#Cc1cn(Cc2ccno2)nn1)NC(C(C)CC1CCCCC1)=O N1(C(C(C)C2(O)CCC2)=O)CCC=C(CNC(c2ccon2)=O)C1 N1(C(CC(CC)(C)C)=O)CC2CC1CCN2C(c1cnc(C(C)C)s1)=O N1(C(C(N2CCOCC2)C)=O)C2CCC1CC(C(=O)N(C)CC1CC(F)(F)C1)C2 C1(CNC(c2nc(CCCCC)sc2)=O)CN(C(=O)CCC(C)SC)CCO1 C(CS(=O)(=O)CC(=O)OCc1cccc(C)c1)Nc1c(C)ccc(C(=O)OC)c1 N1(C(c2n(C=C)ncc2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCC(C)OC)C2 Cc1nc2cc(C(N3CC(CCc4cn(CC5CC5)nn4)C3)=O)c(F)cc2[nH]1 Cc1cc(N)n(CC(=O)NC2(CNC(C3CC4C=CC3C4)=O)CC2)n1 Cc1scc(C(=O)NCC(O)C(=O)NCC2CCCOC2)c1C C1(=O)N=C2NNC=C2C(=O)N2C1CCC2.n1(CC)nc(C)cc1N(C)C C1(C(=O)NCCCCNC(CCC(C)(C)OC)=O)CC2CCCCN2C1 c1(OC)cnc(CNCc2ccccc2C(C)(F)F)nc1 N1(C(c2cccc(C(=O)OC)n2)=O)CCCC(N(C)C(C2(Cl)CC2(F)F)=O)CC1 c1(OC)c(N(C2CCN(C(=O)Cc3ccc(Cl)nc3C)C2)C)ncnc1C Cc1nn(C)c(N)c1C(=O)NCC1CCN1C(=O)C(C)CO c1(C(=O)NCC(CO)NC(c2c(C(C)C)onc2)=O)ccc2c(c1)OCC(=O)N2 N1(C(C2(C)CCCN(C(C3CCCCC3(F)F)=O)C2)=O)CCC2(C1)CC2(F)F C#Cc1cc(C(=O)NCC2CN(C(=O)Cn3ccccc3=O)CCO2)ccc1C C1(C)(C(N2CCN(CCN(C(=O)C(=O)C(C)(C)C)C)CC2)=O)CCCNS1(=O)=O CCC(CC)(CC)C(=O)N1CCC(N2CCC(NC(=O)C(C)C(C)C)CC2)C1 C1(c2cn(C3(C(=O)OC)CN(C(C4(CO)CCO4)=O)C3)nn2)CC2(CC(=O)C2)C1 C#CCC(CC(F)F)C(=O)N1CCC2(CC1)CC2NC(=O)CCC1CCCCO1 Cc1ccc(OCC(=O)Nc2cccc(NC(=O)C(n3ccc(C)n3)C)c2)cc1 C1(CCC)(NC(=O)COC2CCCCCC2)CCCN(C(c2nonc2N)=O)C1 S(=O)(=O)(c1cnc2ccccc2c1)N1CCC(c2ccc(C)cc2)(C)C1 c1(C(=O)NCC(C)CNC(=O)CC(C)n2cccn2)ccc(Cn2cccn2)o1 CC1C(NC(c2cnn(C3CC3)c2)=O)CCN1C(C1CCCSC1)=O C1(F)(C(=O)NC2CC(CNC(c3c(OC)nsc3)=O)C2)C2CCCCC12 N1(C(C(CSC)C)=O)CC=CC1(C)C(N1CCC(CC2CC2)CC1)=O C1(C(=O)NC23CC(CNC(CC4C(C)OCC4)=O)(C2)C3)CN2CCC1CC2 Cc1cc(NC(C2CCC(=O)N(C(=O)C(F)C(C)(C)O)CC2)=O)cc(C)c1C C1(CC)(CNC(=O)C(C2(O)CN(C(=O)C(C3CC3)OC)C2)F)CCCC1 C1(C(N(C2CC(NC(c3n[nH]cc3C3CC3)=O)C2)C)=O)Cc2ccc(F)cc2O1 CC(CCNC(c1cc(CNC(C2CC3(CCCO3)C2)=O)no1)=O)C(F)(F)F C1(C)(C(=O)NCCC(CNC(c2cc(CO)oc2C)=O)OC)CCC(C)=C(C)C1 N1(C(C(C=CC)O)=O)CC2(CC(NC(C3CCCC(F)(F)C3)=O)CO2)C1 CC1(NC(c2cnc[nH]2)=O)CCCN(C(c2c[nH]c(C#N)c2)=O)C1 c1(C(=O)NCCN(C)C(c2cc(N3CCCCC3)ncn2)=O)cc2n(n1)CC(F)C2 C(=O)(C1=NOC2COCC12)N1CC2(CN(C(CCCN(C(=O)OC)C)=O)C2)C1 C1(N(C)C(c2nn(C)cc2Cl)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CC12 c1(N2C(CN(C(C(C)(C)SC)=O)C)CCC2)ccc([N+](=O)[O-])cc1Br CCC(C)C(C(=O)NC(C)(C)CC)N1CCN(CC(F)(F)CO)CC1 c1(C(N2C3C(NC(C4C(C(=O)OC)C4)=O)C(CC3)C2)=O)ccc(=O)n(C(C)C)c1 C1(NC(Cc2cc(C)nn2C)=O)CC(F)CN(C(c2cncn2C(F)(F)F)=O)C1 C1(CCNC(c2ccoc2)=O)CCN(C(c2csc(-c3cccnc3)n2)=O)CC1 C=CC(C)CC(=O)N(C(C)C(=O)NC1CC(N(C)C)C1)C C1(NC(c2cnc(OCC)nc2)=O)CN(C(C23CC(CC(C)O2)C3)=O)CC1(C)C c1(CNC(CONC(c2cc(CCC)[nH]n2)=O)=O)c(C)cccc1Br C1(NC(CC2CC(C)(C)C2)=O)C2CC1N(C(c1ccccc1F)=O)C2 CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)COc2cccc(C)c2)C(C)(C)C1 C=CCC(C(=O)NC1CCN(C(=O)Cc2cncs2)C1CC)C(C)C c1(C(=O)NC2CC(NC(CN(S(C)(=O)=O)C)=O)C2)cc(C(F)(F)F)ccc1Cl c1(C(=O)NC2CCC(C)N(C(=O)Cc3ccc(Cl)s3)C2)ncc2c(F)cccn12 c1(C2(C)CC2)nnc(SCc2cnn(-c3ccc(F)cc3)c2)n1N c1(OC)ccc(-c2nc(C3CCCN(C(C)=O)C3)n(CCS(C)(=O)=O)n2)nc1 c1(C(N2CCC(c3nncn3C)C2)C(=O)NC(C(=O)OC)C)ccc(F)cc1 c1(-c2cn(CCCC(=O)NCC3(c4ccnc(F)c4)CC3)nn2)ccc(F)cn1 C1(C(=O)NC2(CO)CN(C(C3(CO)CC(C)(C)C3)=O)C2)CC12CCCCC2 c1(NC)nn(C)cc1C(=O)NCCNC(c1cc(C(=O)OC)no1)=O CC1CCCCC1(CNC(=O)COc1ccsc1)NC(C1CC(CC2CC2)C1)=O Cc1nc(Cl)[nH]c(=NC2CCC3CN(C(c4cc(CC(C)C)[nH]n4)=O)CC23)c1F c1(C(C(=O)N(CC)Cc2nnc(C(C)C)o2)F)ccc(C)cc1 N1(C(c2cnc(SC)n2C)=O)CCN(C(c2coc(C(N)=O)c2)=O)C(C)C1C C(C(=O)NCCC(C)N(C)C(C1CC=CC1)=O)(C(C)C)c1cc(C)no1 N(S(=O)(=O)N1CCC(C)(C)CC1)CC(CCN(C)C)(C)O C(=O)(C(F)C(F)(F)F)NCC1C(NC(c2cnc(=N)[nH]c2)=O)CC1 c1(C(C(=O)NCC(=O)NCCCNC(C(CC)C)=O)CC2CC2)ccc(F)cc1 C(C(=O)NOC1CCOCC1)(c1ccoc1)NC(=O)C(O)CC1CCCC1 c1(CC(=O)OC)ccc([N+](=O)[O-])cc1Br.C1(=O)C(=O)CCO1 c1(C(CNC(=O)C(C)O)NC(C2(C#C)CCCC2)=O)ccc(OC)cc1OC N1(C(c2cc(C)cc(Cl)n2)=O)CC(F)C(N=c2ncnc3[nH][nH]c(I)c2-3)C1 c1(C(C)(C)C)ccc(C(=O)NC2CCC(CNC(c3c[nH]c(=N)o3)=O)CC2)nc1 N1(C(CC(c2scc(C)c2)O)=O)CCC(CNC(C2CC(O)C2)=O)CC1 C1(C(N2C(Cn3cc(C(C)(C)NC(N)=O)nn3)CCCC2)=O)CC(S(C)(=O)=O)C1 C(C(=O)NC(c1nc(C(=O)NC2CCCN(O)C2=O)co1)C)(C(C)(C)C)OC C=CCCC(C)(C)C(=O)N1CC(CN(C)C(c2csc(C(C)=O)n2)=O)C2(CC2)C1 C1(C(=O)NCC(CN(C)C(C2CCC3(CCC3)O2)=O)(C)C)CCN2CCCC2C1 c1(CC)ccc(NC(C2(F)CN(C(c3cc(OC)ccn3)=O)C2)=O)cc1 C(=O)(CCS(=O)(=O)NC1CC1)N(C)CC1CCCN(C(C2CCCN2C=O)=O)C1 c1(C(=O)NCC2C(C)CN(C(C3CCC(=O)N3)=O)C2)ncnc(O)c1Br C(=O)(CCCCCNC(C1(n2cnnn2)CC1)=O)NCc1ccc(C)o1 c1(C(N2CCN(C(CN(C(CSC)=O)C)=O)CC2)=O)ccc(O)c(F)c1 N1(C(C2OCCC(=O)C2)=O)CCOC2(CCN(C(C3CCCO3)=O)C2)C1 c1(C(=O)Nc2cccc(NC(CN(CCC)C)=O)c2)cc(F)c(CSC)c(F)c1 c1(CNC(c2cc(-c3ccccc3)cs2)=O)cccc2c1CNC2 N1(C(c2ccc(OC)cn2)=O)CCC(C2CCN(C(c3snc(O)c3Cl)=O)C2)C1 c1(C(=O)OC)ccc(Oc2ccccc2NC(c2ccn(C)n2)=O)cc1 C1(C(N(CC(C(C)C)OC)C)=O)(OC)CCN(C(=O)C(C)Cn2ccnc2)C1 C(=O)(C1CCCCc2ccccc21)NC1(C(C)NC(=O)C2=CCCCC2C)CC1 C1(C2CCN(C(=O)C(F)C3=CCCCC3)C2)(NC(C=C(C)C(C)(C)C)=O)CC1 C1(C(=O)O)(CNC(=O)OC(C)(C)C)CN(C2CCC(C(F)(F)F)CC2)CCO1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)CCc1ccc(F)nc1)C2 N1(C(CC(CCC)NC(=O)C=Cc2cscn2)=O)CCN2CCC1CC2 Cc1sncc1C(N1CCC(N(C)C(c2cc(C3CC3)no2)=O)C1)=O C1(NC(c2cccc3c2CCCN3)=O)CC1C1CCN(C(=O)CC2CCC2)CC1 N1(C(c2cc(CC(C)C)nn2C)=O)CCCC(O)(CNC(C2(C)CCOC2)=O)C1 c1(C(c2n(CC(C)C)nc(-c3nc[nH]n3)n2)C(C)C)ccc(F)c(C(F)(F)F)c1 c1(C(N2CC(CNC(C=C(C)C)=O)C3C2C3)=O)cc2ncccc2[nH]1 C1(NC(C(F)=CC)=O)CCCN(C(c2ccc(C)c(N)c2)=O)C1C c1(C(=O)NCc2cccc(C(=O)NC(C#C)CC3CCC3)n2)c(C)cnnc1O N1(CC(=O)N(CC(C)NC(C2CC(C(=O)OC)C2)=O)CC)CCCCCC1=O C1(CNC(CSCCOC)=O)COCC2(CCN(C(=O)C(C)(C)CCC#N)C2)O1 c1(C(N2CC3(CN(C(C(C)OCC#C)=O)C3)C2)=O)cnn2c(C)ccnc12 C1(NC(CCOC)=O)COC2(CCN(C(=O)CNC(c3cccc(C)c3)=O)C2)C1 C1(C(=O)NCCC(F)(F)Cl)(CNC(=O)C2CC2)CCCCO1 CC(O)C(C)(C)C(=O)NCCC(CNC(=O)CC1CC2(CC2)CO1)[NH2+]C c1(OC)ccccc1NC(=O)C(N1CCCC1CC(N)=O)C1CC1(C)Br C(C(=O)O)(C1=CCC=CC1)Nc1c(OC)ncc(Br)c1C Cc1ccc(C#N)cc1NC(C1C2CCC(C2)C1NC(C1CCCCC1)=O)=O c1(C(=O)NCC(C)(C)NC(c2cncc(-c3cc[nH]n3)c2)=O)cc(F)cnc1O C12(CNC(c3ccc(C)nc3N)=O)CCC(CC1)N(C(C1CSCCS1)=O)C2 c1(C(=O)NC(C2(CNC(C(C)NC(CC)=O)=O)CC2)C)cc(C)ns1 Cc1cccc2ncc(C(c3nnnn3C)NCCCC3CCCC3)n12 Cc1[nH]nc2c1CCC(C(N1CCN(C(c3ccc4c(c3)OCC4)=O)CC1)=O)C2 C1(O)(CNC(=O)COCC2CCCC2)CCCN(C(C2CC3CC2CO3)=O)CC1 c1(C(=O)NC2C(NC(CSCC(=O)OC)=O)C2)cccc2nc(C)cnc12 N1(C(c2cc(CC)[nH]n2)=O)CCC(O)(C(C)CNC(c2ocnc2C)=O)C1 C1(CNC(C(C2(O)CCC2)NC(C2CC3CC(=O)C2O3)=O)=O)CC2(CC2)C(=O)O1 c1(NC(C2C3(CC(NC(C(=O)NCC)=O)C3)C2)=O)ccc(O)c(F)c1 Cc1cc(O)ccc1CN(CCc1nn[nH]n1)C(C)C N1(C(C=CC(C)(C)NC(=O)OCC)=O)CCC(N(C)C(c2nscc2C)=O)CC1 c1(CC(N2C(C)(C)CC(C(=O)O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 N1(C(c2n(CC(C)C)ncc2)=O)CCN(C(=O)C(C)O)C(CC(F)(F)F)C1 C(=O)(CC(F)(F)C(F)(F)F)NC(CC=C)CNC(c1cccc(C)c1N)=O C(C(CC1CC1)C(=O)NCc1cccc(C2CC2)c1)NC(C(C)C)=O CC1CN(C(=O)C(F)(F)c2csc(Cl)n2)CC1NC(=O)C(C)(Cl)Cl N1(C(c2c(C)cnnc2)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccnn1C)O Cc1cc(C(F)(F)C(=O)N(CC(C)N(C(=O)C(C)N(C)C)C)C)cnc1Cl N1(CCC)C(=O)NC(c2ccc(F)c(F)c2)C(C(=O)N(CC)CC)=C1C c1(CC)cnccc1NC(=O)NCC=CCOC N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(c2ccnc(C(F)F)c2)=O)CC1 CCCC(C(O)C(=O)NCC(C)(C)OC)NC(c1cc(C)c(N)cn1)=O c1(C(=O)OC)sc(=NCC2(O)CCCN(C(C3CCCN(CC)C3)=O)C2)[nH]c1Cl C(CN=c1[nH]c(=NCCC2CC2)[nH]c2cc[nH]c12)=CCOC c1(C(=O)NCCNC(C23OC(C)C(CC2)C3)=O)cc2nnn(C)c2s1 C12(C(=O)NC(C)(C)CCF)CCC(NC(=O)CC(Cl)Cl)(CC1)C2 N1(C(CC(C)C2CC2)=O)CC2(CCC(NC(C3CCC(C)(C)O3)=O)CC2)C1 O=C(CN=c1cc[nH]cc1)N1CC2CCCC12 c1(C(=O)NCC2(C(N)=O)CN(C(CNC(=O)NC)=O)C2)cccc2nn[nH]c12 c1(OCC)cc(C(N2CC(OC(C)=O)C2)=O)[nH]n1.C(=O)C(CC)c1cccnc1 c1(C(=O)NC2CCC(NC(Cc3onc(C)n3)=O)C2)cccn(C(C)(C)C)c1=O Cc1nc(C(=O)NCC2CN(C(=O)C(C)(C)C3CC3)CC2C)cc(O)n1 C#CC1(Nc2nccc(=NCC3CCN(C(C)=O)CC3)[nH]2)CCCCCC1 CC1CCN(C(c2cn(C)nc2C2CC2)=O)CC1C Cc1ccnc(C(N2CCOC(CN(C(=O)C(C)C(F)F)C)C2)=O)c1F C1(NC(=O)CCCF)CCC2(CC1)CCN(C(C13CC1COC31CCC1)=O)CC2 c1(C(=O)NC2CCCN(C(C(C(C)C)SC)=O)C2)cc2ccc(Cl)cc2c(=O)o1 C1(C(=O)NCCCNC(C2CC(=C)C2)=O)(C(=O)OC(C)(C)C)C2CCC12 c1(CC(=O)NCC2CCN(C(C3(C)CCOCC3)=O)CC2)cc(Cl)ccc1O n1(CC)nc(C(=O)NC2CC(C)(CNC(c3csc(C)n3)=O)C2)cc1C(F)(F)F N1(C(C2CC3(CC(NC(CC4CC(C)C4)=O)C3)C2)=O)CCCC(N=[N+]=[N-])C1 CCCCCC(O)C(=O)NCC(C)CNC(=O)CCCCO N1(C(C23C(CN(C(C(C(C)C)C)=O)C2)C3)=O)CCS(=N)(=O)CC1 C1(O)(CN(C(CNC(CC(C)C)=O)=O)C)CCN(C(C2CC2(Cl)Cl)=O)C1 N1(C(C(N2CCC(C)(N)CC2)=O)=O)CCCc2cc(OC(F)F)ccc21 N1(C(Cc2cc(C)[nH]n2)=O)CC(C2CN(C(C3(F)CCCC3)=O)C2)C1 c1(NC(C=CC(C)NC(=O)C(=O)N(C)C)=O)cc(F)ccc1N1CCOCC1 CCCC(C)CC(=O)NCC(c1cccc(OC)c1)NC(C1(O)CCC1)=O c1(C2C(C(N(C3CCC(NC(=O)COC4CC=CC4)C3)C)=O)C2)ccccc1F CCCCC(CC)CCC(=O)NCC(C1CCCC1)NC(=O)CCn1ccnn1 O=C(CCCCCNC(c1cccs1)=O)NCCc1ccc(O)nc1 c1(C(N2CC(NC(c3cc(C(C)(C)C)ncc3)=O)C2)=O)cc2ccc(Cl)cc2s1 c1(CCNC(CN(c2ccccc2)C(C=C)C)=O)snnc1C C1(CNC(=O)Nc2c(C(=O)OC)ncc(Br)c2)CCCCC(F)(F)C1 CC1(C)CC(N(CCN2CCCC2)C(=O)Nc2ccccc2)CC(C)(C)N1 c1(CNC(c2ccc(F)c(I)c2)=O)ccc(C(F)F)c(Br)c1 C1(NC(CC(C)c2ccco2)=O)CN(C(=O)CC2CC=CC2)CC12CC2 CCC(C)(C(=O)N1C(C)C2CC1C2NC(c1csc2nnsc12)=O)C(N)=O CC1C(C(=O)N(CCC(O)CO)C)CCCN1C(=O)C1=CCCOC1 Cc1c(N(C)CC2CC2)ncnc1N1CCN(CCOc2ccc(Cl)cc2)CC1 C(N=c1[nH]c(=NCC2CCOCC2(C)C)c2[nH]ccc2[nH]1)c1c(C)ccnc1 N1(C(c2c(C(C)C)nc(Br)s2)=O)CCC(C2CCCC2C(=O)O)CC1 c1(NC(C2(F)CCN(C(c3cc4sccn4c3)=O)CC2)=O)cc2ccccc2[nH]1 C1(NC(C2CCN(C(CC)=O)C2)=O)CCC2(CC1)CC2NC(=O)COC1CCC1 O=C(C1=NOC2(CCN(C(c3ccc(F)nc3)=O)C2)C1)NCCc1ncon1 C1(NC(CCC)=O)(CC)CCCN(C(C2CCC(F)(F)CO2)=O)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCC2(CC1)CCN(C(C1CCOCC1)=O)C2 c1(C(N(C)CC2N(C(CCc3ccc(C)o3)=O)CCC2)=O)nnc2n1CCCC2 CCCC(CCCNC(=O)C(C1CCCC1)OC)N=c1[nH]nc(CC)o1 C1(CC(=O)NCc2cc(C(C)C)no2)CC(NC(=O)C(F)C2CCCC2)C1(C)C C1(NC(C2(CC)CCC2)=O)CC2CC1CN(C(C1(C(=O)N(C)C)CC1)=O)C2 N1(C(=O)NCC2CC(CO)CO2)CCC2(CCCNC2=O)CC1 N1(C(C2(C(=O)OC)CCCC2)=O)CC(CNC(C2(c3ncco3)CC2)=O)C(C)C1 S(=O)(=O)(c1cc(-c2ccccc2)[nH]n1)NC(CC)CSC CCC(CC)(CCNC(c1cnc(C(F)(F)F)s1)=O)NC(=O)C(CO)NC(N)=O Cc1ccc(F)cc1CC(=O)NC1CC2CCC1N2C(=O)Cc1ccon1 c1(NC(=O)COCCC2CCC2)cc(Br)cc(I)c1 C1(NC(C2CCCS2(=O)=O)=O)CC1C1CCCN(C(=O)C=CC2CCOCC2)C1 c1(CN(C(C(=O)N2CC(OC)C2)C2CCCO2)C(CC)=O)ccc(Cl)c(C)c1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1(O)CCN(C(C2C(C=C)CC2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CCCC2)C1)NCC1CCC(=O)NC1 C1(c2nc(Cc3csc(C4CC4)n3)no2)(C(c2ccco2)=O)CCSC1 N1(C(CCn2c(C)cc(C)n2)=O)CCC(NC(=O)C#CC2CCC2)C(CO)CC1 C1(C(N(CCNC(c2cccc(CF)c2)=O)CC)=O)CCC2C(C1)C2(F)F C1(N(C(C(C)SC(F)(F)F)=O)C)CCCCN(C(=O)CCCCc2cnc[nH]2)C1 c1(SCC(=O)NC(CC)CN(C)C(C2CC(C)(F)C2)=O)ccc(Cl)cc1 c1(C(=O)NCC2(CNC(CC(CC)OC)=O)CCCC2)ccc2nn[nH]c2n1 C(=O)(CCCCCNC(C1CC2CC1CC2O)=O)NCc1nc(C)c(C)o1 C1(C(=O)NC(C2(OC)CCC2)C)C2CCN(C(c3cc(O)cc(F)c3)=O)CC12 C1(OCCCNC(C(CC)n2ccnc2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(C(N2CCN(C(C(C)NC=O)=O)CC2C#N)=O)cccc2ccncc12 C1(OC)CN(C(c2ccc(C)n2C)=O)CC1NC(=O)C(C)NC(N)=O C(CC(=O)N1CCN(C(=O)CNS(=O)(=O)C2CC2)C(CCO)C1)(C(F)(F)F)OC C1(CC(=O)NC2CC(OCC(=O)NCCCOCCC)C2)CSCCO1 C1(NC(C2C(C=C)C2)=O)CCC(NC(=O)COCC)C1 c1(C(N(CCC)CCNC(=O)C(CC)CC)=O)cc(NC(=O)N(C)C)ccc1Cl O=S(=O)(c1c[nH]ccc1=NC1COc2ccccc2C1)N1CCOC(CO)CC1 c1(CCNC(NC(C#C)CCC)=NCC)c[nH]c2cc(Cl)cc(Cl)c12 c1(NC(C2C(OC)CCN(C(=O)OC(C)(C)C)C2)=O)cc(I)c(F)cc1F CCCC(C#N)C(=O)N1CC2CC2(CNC(c2cc(Br)ncc2OC)=O)C1 N1(C(CCCCOC)=O)C2CCC1(CNC(=O)C(C)Oc1ccccc1F)CC2 c1(C(=O)NCC(CN(C(=O)Cc2ccoc2)C)O)ccc(OC(F)(F)F)cc1F N1(C(c2c(C)con2)=O)CCCN(C(c2cccc(CN(C)C)c2)=O)CC1C N1(C(CCc2ccc(C)nc2)=O)CC2(CC(NC(c3ccsc3C#N)=O)C2)C1 C1(O)(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CN2CCC1CC2 Cc1ccc(O)c(CN2CCC(F)(C(N3CCOC(C(N)=O)C3)=O)C2)c1 CC1=C(C(=O)NCc2nc(C(=O)NCC3(CO)CCCCC3)c(C)o2)COCC1 C1(C(N2CCC(C3N(C(C(C)CO)=O)CCCC3)C2)=O)CC2(CCC2O)C1 c1(CNC(C(C=C)O)=O)ccc(CC(C)NC(c2csc(CO)n2)=O)cc1 C1(NC(C2(OC)CCSC2)=O)CC(F)CN(C(C2CCCC(F)(F)C2)=O)C1 c1(N2CCC(CNC(=O)C(c3ccc(Cl)c(Cl)c3)CO)CC2)nc(Cl)ncc1Cl Cc1nc(C(=O)NC2CCC(CCNC(c3ccccc3N(C)C)=O)C2)c(C)o1 N1(C(C(N)=O)=O)CC2(CNC(=O)CC3COC(=O)C3)CC1CCO2 c1(OCCCN(CC(O)COCC2(CC(C)C)CC2)C)ccc(S(C)(=O)=O)cc1 C1(C(N(CC(CC)NC(=O)C(S(C)(=O)=O)C2CC2)CC)=O)CCC(O)CN1C Cc1nn(CC(=O)NCC2(C)CCCN(C(C34C=CC(CC3)C4)=O)C2)c(C)c1C C1(C(=O)NCCC(C)NC(C23COC(CCO2)C3)=O)C2(CCC2)C12CCC2 C1(NC(CC(C)OC)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 N#Cc1ccc(Cc2noc(C3CC(OC(F)F)C3)n2)cc1 C1(CC(=O)N(C)CC2CCCC2)CCCN1C(=O)CCc1cnn(C)c1 c1(C(N(CC(O)CNC(=O)CCC2CC2CC2CC2)C)=O)ncn2ccccc12 CC(C)(C(=O)NC1CCC1NC(=O)CC1COC(=O)N1)c1ccsc1 C(CCS(C)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C1CC1C(C)(F)F)=O)OC N1(C(c2c(C)nc(CC)o2)=O)CCCC(C(N2CCCC(CCO)CC2)=O)C1C C1(NC(C(C)O)=O)CS(=O)(=O)C12CCN(C(C1Cc3cncn3C(=O)N1)=O)CC2 c1(C(CC(C)NC(=O)NCC2(F)CC(C(=O)OC)C2)=O)ccc(F)cc1 N1(C(C2CN(C(N)=O)C2)=O)CC2(COCCC(=O)NCC(F)(F)F)CC2(CO)C1 C1(NCc2c(C)nn(-c3ccccc3)c2Cl)CCCNCCC1(F)F CC1(C)CC(CC(=O)NCC2([Si](C)(C)C)CC2)CN1C(C1CC(=O)CC(=O)C1)=O c1(C(N2CCC(N(C)C(c3cc4sccc4[nH]3)=O)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(C(F)(CNC(c1nonc1CC)=O)C(C)C)NCC(CCC)(C)O C1(NC2CC(C(=O)OCC)CC2O)CCC2C3C=CC(C3)C12 C(CC)(C(=O)NCCN(C(=O)Cn1cnc(Br)n1)CCOCCO)OCC C1(NC(C23OCC(C)(C2)C3)=O)CCCCN(C(c2ccnc(O)c2)=O)C1 c1(NC(c2cccc(OC)c2Br)c2nnnn2C2CCC2)ccc(Br)c(C)c1C C1(c2scc(CC(=O)OCC)n2)CCCN(C(=O)NC(C)C)C1 C(=O)(CS(N)(=O)=O)N(C(C)CNC(=O)C(c1cscn1)N(C)C)C c1(CC)nc[nH]c1C(N1CC(F)(CNC(=O)C(C)Cc2cnc[nH]2)C1)=O C1(NC(C2CCN(C)C2=O)=O)CC2CCC1N(C(=O)CCn1ccccc1=O)C2 c1(C(=O)NC2CCCC(NC(Cn3nc(C)oc3=O)=O)C2)cc([N+](=O)[O-])oc1C CCC(C)C(O)C(C)C(=O)NC(CC(=O)N(C(C)CCO)C)C(F)F CC(C)C(C(=O)NCc1ccc(C#N)o1)C(C)NC(C1CS(=O)C1)=O Cc1ccc(NC(=O)C(=O)N(c2cn(C)nc2Cl)Cc2ccccc2)c(F)c1Cl n1(CC)nc(C(N2CCC(NC(N)=O)C2)=O)cc1O.C12CCCC(C1)CC(=O)N2 Cc1cccc(N(C)C(=O)Nc2cn(C(C)(C)C)nc2C)c1C Cc1cc(NC(=O)C(CC2CCOCC2)NC(=O)CC2CSCCO2)cnc1Cl c1(NC(c2cccc(C)n2)C)ncccc1S(=O)(=O)N1CC2CCC2(C)C1 Cc1ccc(N2CCN(C(=O)C(=O)NC3CCCCCC3)CC2)cc1N N1(C(C(=O)NCC23CC(F)(CO2)C3)=O)CCC(C2CC2)C1 c1(C(=O)NCC(CN(C(=O)CC2(C)CCCO2)C)O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(=O)NC2CN(C(=O)CC(C)C)C3CC23)c(=O)n1 CCCCCCCC(=O)N(CC(CC)NC(c1c(F)ccc(F)c1Cl)=O)C C1(C(=O)NC(C)CC2CCC2)CN(C(C2CCN2C)=O)CC12CC2 C1(C(N(C)CC2C(NC(c3c(C)onc3)=O)CCC2)=O)OCC2CCCC12 C12CCCN(CC1)C2=O.C1(C(=O)N=CCc2cccs2)CCN(C2CCOC2)C1 N1(S(CC2(COC)CCOCC2)(=O)=O)CCC12CCOC(C)(C)C2 C1(NC(C(c2cn(C)nn2)NC(c2csc(O)n2)=O)=O)COCC1(C)C CCCC(O)CC(=O)NCCCC(C)NC(c1ccc(C#N)o1)=O c1(C(=O)OC)ccc(Br)nc1NC(c1ccc(-c2ccoc2)nc1)=O C1(C(N(C2CCN(C(=O)C=C(C)C)C2)CCC)=O)CC2(CCCCO2)C1 Cc1cnc(N)c(C(=O)NCC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C)c1 C(=O)(C1CCCc2nnn(C)c21)NCCOc1cc(CC)c(Cl)cc1 C(=O)(CC(C(F)F)NC(=O)C(F)C(C)(F)F)NC(C(=O)N(CC)CC)C N1(C(C(CC)C#N)=O)CCC2(CC1)CC(CNC(C1(OC(C)C)CCC1)=O)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1CCN(C(C)=O)C1)N(CCCCCC=C)C CC1CC(C(=O)NC2(C)CCCN(C(c3cc(Cl)nc(Cl)c3)=O)C2)CCS1(=O)=O N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)C(=O)Nc2ccc(C)cc2)CC1 c1(C(N(CCC(=O)NCCCCCN(C)C(C)C)C(C)C)=O)cc(F)ccc1O C(=O)(CC(O)C(C)CC)NCC(=C)CCNC(c1ccccc1CO)=O c1(-c2[nH]c(C)c(C(=O)O)c2C(=O)N=c2cc(C)n(C)[nH]2)ncnc2cccc(F)c12 c1(C(=O)NC(C)(CNC(=O)COCCc2ccccc2)C2CC2)cc(Cl)c(Cl)[nH]1 c1(C(N2CCN(C(c3cc(C=C)cc(F)c3)=O)CC2)=O)cc2ccc(O)nc2s1 c1(NC2CC(C)CN(Cc3ccccc3)C2)cccc2cccc(Br)c12 c1(C(=O)NCC2C3CN(C(C4C(C)CCS4)=O)C2C3)ccc(S(=O)(=O)N(C)C)o1 C(=O)(CCN1CCCCO1)N1CC2C(N=c3n(CCOC)[nH]nn3)CC(C2)C1 N1(C(CC(CC)C(F)F)=O)CCCC2(C1)CN(C(=O)C=Cc1cc[nH]n1)CCO2 C1(NC(C(C)OCC#C)=O)CN(C(c2cccc(CN(C)C)c2)=O)CCC1F N1(C(COCCOC)=O)CCC(C(C)(C)CNC(C2CNC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(Br)s1)N1CC2N(C(C3C(C)(C(C)C)C3)=O)C(C2)C1 C1(CC)CCCN(C(c2cnccn2)=O)C1C(=O)NCCOc1ccccc1 C=CCC(CC)C(=O)NC12CCC(C1)N(C(=O)Cc1cccc(OC(F)F)n1)C2 O=C(C1=CC2CC=CCC12)NCC1(NC(c2csc(O)n2)=O)CCC1 c1(C(=O)NC(CN(C(CNC(CCCCC)=O)=O)C)C)nc(OC)ccc1OC CCC(CC(=O)OC(C)(C)C)NC(c1ccnc(-n2cccn2)c1)=O C1(NC(C(C)=CC(C)(C)C)=O)C=CCCC1C(=O)NCCC=CCCC Cc1[nH]c(C(=O)N(CC(C)NC(=O)CC(C)n2cccn2)C)c(C)c1C CCC(C)CC(=O)NC1CCC1CNC(C1CC(CC(C)(C)C)C1)=O C1(CNC(Cn2nnc(C)n2)=O)CC(C(F)(F)F)CN1C(C1CCNC1=O)=O C12(NC(c3c(C)snc3)=O)COCCC1CN(C(=O)CSCc1cccnc1)C2 N1(C(C=C(C)C(F)F)=O)CC(NC(c2coc(O)n2)=O)CC12CCOC2 C1(C(N2C(C)CN(C(=O)CN3CCS(=O)(=O)CC3)CC2)=O)CC2C=CCC(C1)C2 C(c1cc(F)cc(F)c1)=C(C(=O)Nc1cnn(-c2c(C)ccc(C)c2)c1C)C#N C1(c2n(-c3ccn(CC)n3)nc(COC)n2)CNC(=O)CC12CCC2 C(=O)(C(C)CC(C)C)NC12CC(CNC(c3c(C)oc(-c4ccsc4)n3)=O)(C1)C2 C1(c2scc(C(=O)OC)n2)CCN(C(=O)NC2CC23CCC3)CC1 C1(O)(C(=O)NCC2(CNC(=O)C(F)n3ccnc3)CCOCC2)CCCCCC1 N1(C(CCC=C(C)C)=O)CC2CC1CN(C(=O)CCC(C)O)C2 c1(OCC)ccc(CNC(c2ncc(Cl)n2C)C2CCCCC2)cc1 C(=O)(C1=NNC(=O)CC1)N1CCC(C(C)NC(c2cc(C(=O)OC)[nH]c2)=O)C1 c1(C(=O)NC(C)CNC(c2cnc3ccsc3c2)=O)ccc2c(c1)C(=O)NC2=O C(C(C)(C)CCNC(C1(CCNC(c2ccco2)=O)CC1)=O)OC N1(C(C2CCC(C)(CC)O2)=O)CCCC(NC(c2cc(Br)co2)=O)CC1 c1(SC)ccc(Cl)c(C(N2CC=CC(NC(C3CC(C(F)F)C3)=O)C2)=O)c1 CCC(CCOC)N=c1[nH]c(N2CC3CCC(OC)C3C2)nc2c1CSC2 C=CCC(C(=O)NC(C)(C)C(C)NC(c1cnc[nH]1)=O)c1ccccc1 c1(OC)ncc(Br)cc1C(=O)NCC12CC1CN(C(=O)C(C)S)C2 Cc1ccc2cccc(C(=O)NCCC3CC(NC(c4sncc4C)=O)C3)c2n1 C(CCCC(C)(C)C)(C(=O)NCSc1ccccc1)N1CCC(n2ncc(C)c2)CC1 CC(N=c1[nH]c(=NCC(C)c2cccc(O)n2)c2cccc(F)c2[nH]1)c1cccs1 N1(C(c2occ(C)c2)=O)CC2(CCC2NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CCN(C(CC(=C)C)=O)C)C(C)(C)C c1(C(N(C(C)CCNC(=O)CC2C=CCCC2)C)=O)ccc(N)c(O)c1 c1(C(N2C(CNC(c3c(C)nco3)=O)C(C)CC2)=O)ccc(Br)c2cn[nH]c12 C#CC1(C(=O)NC(c2cn(C)cn2)C)CN(C(=O)C(O)C2CCCC2)C1 c1(C(=O)NCc2ccc(CNC(C(C)SCCCC)=O)cc2)ncc(F)cc1C C1(NC(COC(CC)C)=O)C2CC3CN(C(=O)Cc4nncn4C(C)C)C1C3C2 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)nnn2c1CCCC2 N1(C(C2(OC)CCCC2)=O)CCCC(O)(CCNC(=O)C(O)CSC)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2cccc(OCC)c2)cncn(C)c1=O CCCC(C)(C)C(=O)NC1CC1CNC(c1ccnc(OC(F)(F)F)c1)=O c1(CCC(=O)NCC(CCCCC)CO)nc(O)c2ccccc2n1 c1(CN2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(F)C2)cccc2cc[nH]c12 N1(C(C(Cn2ccc(C)n2)C)=O)CC(NC(c2csnc2C)=O)CC(C)C1 c1(SC2(C(N)=O)CN(C(C3(C(=O)OCC)CCC3)=O)C2)ccc(Cl)cc1 Cc1nc2cc(-c3nnc(SC4CSc5ccccc5C4=O)o3)cc(O)c2o1 c1(NC(C(C(C)C)NC(c2cocn2)=O)=O)ccc2c(c1)CCO2 C12(C(N3CC(NC(c4cc(C(N)=O)cc(C)c4)=O)C3)=O)CCOC1CCOC2 N1(C(CCCCSC)=O)CCCC1C1CCCCN1C(=O)Cc1cc(C)on1 C12(C(N(CC(CC)(C)OC)C)=O)CCN(C(c3c(Cl)cnn3C)=O)CCC1C2 C1(NC(Cc2c(C)ccc(C)c2)=O)CCC(O)CN(C(C2CC(C)(C)CO2)=O)C1 c1(NC(=O)C(C)OC(c2c(C)occ2C(F)(F)F)=O)cc(F)ccc1C(F)(F)F Cc1c(C(=O)NCC(C)(C)CNC(=O)C(c2ccc(F)cc2)F)cnn1C1CC1 N1(C(C(C)SCC)=O)CCN(C(=O)CCc2ccoc2)CC1C1CCC1 c1(C(=O)C2CC2)[nH]c(O)nc1C.C1(COC)(CN)CN(C(c2ccc(C)s2)=O)C1.NCC Cc1nccc(C(=O)NC2CC2C(=O)NC(c2cn(C)nc2C)C)n1 c1(CC(N2CCC(N(C(C(CCC)OCC)=O)CC)C2)=O)cccc(F)c1O Cc1nccn1C(C)C(=O)NCC1CC1CNC(=O)CCc1cnc(O)[nH]1 c1(C(=O)NC2(C)CCN(C(C3C4CCCC34)=O)CC2)ccc(N=S(C)(C)=O)s1 CC(F)(C(=O)NC1CCCC(CNC(c2cnc(Cl)c(N)c2)=O)C1)C(F)(F)F N1(C(=O)C=Cc2cnco2)CCC2(CCCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N1(C(CCSC)=O)CCCC2CN(C(C3(C)COCCO3)=O)CCC12 N1(C(c2nn(CC)c(C)c2)=O)CC2CCC2(CNC(=O)CCC(=O)NC)C1 C(=O)(C(C)C(=O)c1ccc(Cl)cc1)N(C(c1c(C)ocn1)=O)C C1(C)(C(=O)NCC=CCNC(C2CC(C)C2(C)C)=O)C(C)(C)C1(C)C Cc1nc2cc(C(=O)NCCC(C)N(C(=O)CC3CCCO3)C)ccc2n1C CC1(C)CCC(C(N2C3CCC2C(CNC(C2CCCSC2)=O)C3)=O)CO1 N1(C(C(C=CC)O)=O)CC(NC(c2cnn(CCC(C)C)c2C)=O)CC(F)C1 c1(C(=O)NCC(C)N(c2nnc(C3CCCC3)s2)C)csc(C(N)=O)n1 Nc1c(C(F)(F)F)nn(C2CC2)c1C(=O)NCC12CC(CSC)(CCO1)C2 N1(C(=O)C(O)Cc2ccc(Cl)cc2)CC2CCCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(C)C)CCNC(c1cc2c(ncn2C)s1)=O CCCCC(CC(=O)N(CCCF)CC)NC(c1ccnc2cc[nH]c12)=O C1(O)(C(C(=O)N(CC(C)OC)CC)F)CN(C(=O)COC(C)=O)C1 C1(C(N2CCC(C)(NC(c3cnc(Cl)[nH]3)=O)C2)=O)CC2CCCCCC12 c1(SCC#C)cccc(C(=O)NC(C)CCCCNC(=O)CC2(C)CC2)c1 CC(C(=O)NCCN1CCC(NC(=O)CCS(C)=O)CC1)C(C)(C)O C(=O)(C1Cc2ccccc21)NCCN(C(=O)CC1(C2CC2)CC1)CCC Cc1cc(C(=O)NCCCCNC(C2(N3CCOCC3=O)CC2)=O)c(C)n1C c1(SC)nc(C(N2CCC(F)(CNC(=O)C=CC3CCC3)C2)=O)c2ccccn12 c1(C(=O)NC(C)(CNC(c2ccsn2)=O)C2CC2)sc2cccc(F)c2c1Cl CC(C)(C)C(CNC(C1(n2ccnn2)CC1)=O)NC(C1(C)CNC(=O)C1)=O c1(C(C(=O)NCC)N(C2CCOC2)C)cnc(OC(C)(C)C)cc1OC.C(COC)S CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CCN(C(=O)COCCCF)C1 N1(C(C(CC)F)=O)CC(NC(c2cnc(S)[nH]2)=O)CC12CCC2 c1(C(=O)NCCC(C)(C)CO)c(C(F)(F)F)cccc1C(F)(F)F c1(C(=O)NC2C(NC(CC3CCC(C)CO3)=O)C2)ccc(F)cc1Cl CC1(C(=O)NC2CC2CNC(=O)COc2ccc([N+](=O)[O-])cc2)CCS(=O)(=O)CC1 c1(C(=O)NCC(CC)(C)NC(c2ccc(CO)o2)=O)ccc2c(c1F)CCC2 C(C#Cc1cn(-n2cnnc2)nn1)NC(=O)NC1CCS(=O)(=O)C1 N1(C(C2CCC(C(N)=O)C2)=O)CCCC(C)C1CNC(c1[nH]c(=NC)sc1)=O C1(C(=O)NCCOCC(=O)NC(C2CCCO2)(C)C)CCCC(C#N)C1 N1(C(C=C(C)c2cccnc2)=O)CCC2(CC1)CC2NC(C1CC1(C)C(F)F)=O c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C1CN(C)C(=O)N1)=O CC12CSCC1CN(C(c1ccc(CNC(c3cc[nH]n3)=O)cc1)=O)C2 C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CC2)CCCCN1N=O Nc1ccc(OCC(=O)NC(CNC(C2CC23CCOC3)=O)C2CC2)cc1 C(C)(CCC(=O)N(C1CCCN(C(C2CC2c2cccc(C)c2)=O)C1)CC)OC C12(CNC(c3c(C)nn(C)c3)=O)CCCC1CCN2C(c1nccn1C)=O c1(C2(C(N3CC(NC(c4csnn4)=O)(CO)C3)=O)CCC2)ccccc1F N1(c2cn(CCOCCCNC(=O)CC3CSCCO3)nn2)CC(=O)CCC1=O Cn1cc(Cl)cc1-c1nnc(N2CCOC(CF)C2)n1CC1CC1 CCCCC(C(=O)NC1(CNC(=O)C(F)=CC2CC2)CCC1)C(C)C Cn1ccc(S(=O)(=O)N2CC3CCN(C(=O)Cc4ccccc4Br)C3C2)n1 Cc1ncc(C(=O)N(C)CC2CCCN2C(C23CCCC2C3(F)F)=O)cc1C#N C(=O)(CCCC(=O)OCC)NC(C=CC(=O)NCC(C(=O)NCC)C)C C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(CC)SC)CC12CC2 c1(NC(C(C(=O)OCC)CC(=O)C2CC2)=O)ccc(OCC)c(OC)c1.C(C)(C)O S(=O)(=O)(c1cc(C(F)(F)F)cc(O)c1)N1CC(c2nc(C(C)C)[nH]n2)OCC1 Cc1cc(Cl)c(C(=O)NC2CCC(N(C)C(c3nccnc3Cl)=O)CC2)s1 CC1(NC(=O)CC2CCCCO2)CC(C(=O)NCC2C3COCC23)C1 CCC(CO)C(=O)NC(C)CC1CCN(C(C23CCC(C2)OC3)=O)CC1 c1(C(C)NC(c2nnnn2C)C2CC(OCOC)C2)cccc(F)c1C N1(C(CCNC(=O)NC)=O)CCC(NC(=O)Cc2cccs2)C1C(C)(C)C N1(C(CN(C)C)=O)CC(NC(c2cc(Cl)nc(Cl)c2)=O)CC2(CC2)C1 N1(C(c2ccc(COC)[nH]2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CC2(F)Cl)C1 c1(C(=O)NC(C2CCN(C(C3(CC=C)CC3)=O)C2)C)cc([N+](=O)[O-])cc(C)c1Cl CCCC(O)C(=O)N1CCC(C(=O)NCc2ccc(C(F)(F)F)cc2)C1 C1(NC(CC(CNC(c2c(OC)nn(C)c2)=O)C)=O)CCN(CC)CC1C C1(C)(CNC(c2c(C)coc2C(C)C)=O)CC(F)(F)CN1C(=O)CC1CCCC1 c1(SCC)ccc(CNC(=O)C(=O)NCCc2cc(Cl)c(Cl)s2)cc1 Cn1cc(C(=O)NC(COC(=N)O)Cc2ccccc2)c(C(F)(F)F)n1 CN1CCCCC1C(N1CC(NC(=O)C=Cc2ccsc2Br)C(O)C1)=O C1(CC(=O)NC(CC=C)C(=O)OC)C2CCCC2N1C(c1csc(C)c1)=O c1(C(C(=O)NC(CC)CNC(=O)C(C)O)O)cccc(OC)c1 N1(C(c2ccc(CC)s2)=O)CC(C)N(C(=O)C(C)CC(N)=O)CC1C Cc1[nH]ccc1C(=O)N(C1CCN(C(=O)CN2CC3CC3C2)C1)CCO N1(C(C=COCC)=O)CC2CCCC2(NC(c2c[nH]c(=N)cc2C)=O)C1 Cc1ccc(-c2ccccc2)c(NC(=O)Cc2cc(C)nn2C)c1 C1(C(=O)NC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)C2CC2)CC(C(C)C)=NO1 N1(C(c2cc(C)nnc2)=O)CCC(C2CC2)(NC(C2CC(F)(F)C2)=O)C1 c1(CN2CCC(CNC(c3cccc(CCC)c3)=O)C2)c[nH]c2cc(C)ccc12 C1(NC(c2scc(C)c2)=O)CCN(C(=O)C(N2CCOCC2)C)C12CC2 N1(C(CSCC#C)=O)CCCC2(CCC(NC(=O)C(C)(C)C3CCCCC3)C2)C1 C1(CNC(c2cc(OC)ns2)=O)CCC(C)CN1C(=O)CCSC1CCCC1 c1(C(N2CC3(N(C(C(C)CO)=O)CC3)C2)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 c1(C(=O)NC2CC(C(C(N3CC(N(CC=C)C)C3)=O)F)C2)cccc(O)n1 c1(C(=O)NCCC(C)(C)NC(CCC)=O)cncc2c1CCNC2=O c1(NC(C2CC(=C)C2)=O)nnc2ccccn12 c1(CC(=O)NC(C(C)C)CNC(C2(C)CCCS2)=O)cccc2c1OCCO2 CC1CC(C(=O)NCC2(O)CC(NC(=O)CCCn3ccnc3)C2)CC(C)O1 c1(OCC)ncc(NC(C2(CNC(c3cnc(Cl)n3C)=O)CCCO2)=O)cn1 N1(Cc2ncc(OC)nc2)CCC2(CC2C(=O)Nc2cnn(CCO)c2)C1 c1(CCNC(C2(C)CC(NC(C(CSC(C)=O)C)=O)C2)=O)cccnc1Cl Cc1ccc(CN=C(NCC(C2CCCC2)F)NC(c2cccs2)CC)c(C)c1 c1(C(=O)NCC(=O)NCC(=O)N(C2(C(=O)OC)CC2)C)cc(C)n(C)n1 C1(F)(C(N(C2(CCO)CC2)C)=O)CCCN(C(=O)C(F)=CC2CC2)C1 CC(C)(CC(=O)NC1(CNC(=O)C(c2cc(F)cc(F)c2)O)CCC1)C(F)(F)F c1(OC)nc(CC2CCCCN2C(C2CCCN(C(C)=O)C2)=O)ncc1Cl CCC(C)CC(=O)C(=O)NC(C(=O)NC1(c2cc[nH]n2)CC1)C1CCC1 N1(C(c2c(C)n(C)cc2)=O)CCC2(CC2)CC1C(=O)NC1(C(N)=O)CC1 c1(NCC=CCNC(CCCC)=O)c(C(=O)OCC)cc([N+](=O)[O-])cc1F C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(CS(CC)=O)=O)C2CC2)CCC1 N1(C(c2cc(CC)on2)=O)CCc2ccccc2C(NC(=O)C(C)C2CCC2)C1 N1(C(CC2CCN(OC)CC2)=O)CC2CC(C)N(C(=O)Cc3csc(S)n3)C2C1 CC(O)C(=O)NNC(=O)C(C1C(C)(C)C1(C)C)n1cccn1.n12cc(nn1)CNC1CCC2CC1 C(=O)(CC1CCOc2ccccc21)NCCCN(C(C1C(C)C1)=O)CCO N1(C(c2cccc(OCCC)c2)=O)CCC2CCC(NC(c3cnoc3)=O)C1C2 C1(C(=O)NCc2scc(CNC(C3(C#N)C(C)C3)=O)n2)CC2(C1)CC1(CC1)C2 c1(OC)cc(C)sc1C(N1CC(CCCCNC(=O)C(C)=CC2CC2)C1)=O N1(C(CC(CCC)CC)=O)CCCC2CN(C(C3CC4(CCOC4)C3)=O)CC12 C12(NC(CC(CC)(C)C)=O)CCN(C(c3cc[nH]c4nccc3-4)=O)CCC1C2 c1(C(=O)NCC(C)N(C(c2cc(OC)ncc2F)=O)C)ccc2c(c1O)CCC2 C1(C(=O)NCCOC2CCN(C(CSCCN(C)C)=O)C2)OCC2CCCC1C2 N1(S(C)(=O)=O)CCCC(NCc2cnc(C3CCNCC3)[nH]2)C1 N1(C(CCCCC(C)C)=O)CCCCC12CC(NC(C1CCCCC1(C)C)=O)C2 N1(C(C=C(CC)C)=O)CC(NC(c2cnoc2-c2ccccc2)=O)C(O)C1 C#CCC(CC(F)F)C(=O)NC1CCCCC1NC(=O)C(N1CCOCC1)C CC1OCCN(C(=O)CCN2CCC2)C1C(N1CCCC(C)CC1)=O Cc1cnc(C(C(=O)NCc2ccccc2)NCC(c2cnn(C(C)C)c2)C)o1 C1(NC(=O)CCCc2cccc(Cl)n2)CN(C(c2cnc[nH]2)=O)CCC12CCC2 C1(C)(OC)CCN(C(C2CC(O)(CNC(=O)Cn3cnccc3=O)C2)=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCC3CCCOC3)C(F)C2)=O)ncn1 C1(CNC(c2cc(C)no2)=O)CCCC2CN(C(=O)CC3CC(F)C3)CC12 c1(C(N2CC3(N(C(C4(CC)CC4)=O)CC3)C2)=O)[nH]nc2ccncc12 Cc1cc(C(=O)NC(C)(C)CN(C)C(C2CCCC(C)C2)=O)cc(Cl)c1 S(=O)(=O)(c1ccc(NCC2CSC2)c(C#N)c1)NC(C(C1CCCCC1)C)C c1(CCC(=O)N(C2(CNC(=O)C=CCN3CCCC3)CC2)C)ccc(F)nc1 S(=O)(=O)(c1c[nH]c(=NCCCNC2CCCC2)cc1C)NC(c1cnc(C)s1)C N1(C(C(C)(C)CCC#N)=O)CCOC2CN(C(C3CC4C=CC3C4)=O)CC12 C1(F)(C(=O)NCCCNC(CNC(=O)NCC2CCCC2)=O)C2CCCCC12 C1(CNC(C2ON=C(C)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CCC1(F)F C1(NC(c2cnc(O)o2)=O)CC2(C1)CC(CNC(C1CC3CCC1O3)=O)C2 C1(CCOC)(NC(c2cc(C)sc2C)=O)CCN(C(=O)Cc2csc(C)n2)C1 c1(NC(C)=O)cccc(F)c1C(=O)NCC(O)CNC(=O)C(C)n1ccnc1 C1(N(C(c2cc(CNC(c3cc(OCC)n[nH]3)=O)no2)=O)C)CC(C)CC(C)C1 C(=O)(CC(C)CC(C)C)N(C1CC(C#N)C1)CC(=O)NC(CCCC)(C)C C(=O)(CC1COc2ccccc21)NC1CC(NC(C(C)C#N)=O)C1 N1(C(C2CCN(C)CC2)=O)CCOC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1 C1(C(=O)NC(CC)CN(C)C(C2CCCCN2C)=O)CCC([N+](=O)[O-])CC1 c1(C(N(C2CCN(C(=O)CCCC(C)(F)F)C2)CCC)=O)cnc([N+](=O)[O-])n1C c1(OC(C)C(=O)NC2CCC(NC(=O)C(C)O)CC2)ccc(Cl)cc1Cl N1(Cc2cnc(C)o2)CC2CCN(C(C34CC5CC(C(=O)N3)C4C5)=O)CCC2C1 C#CC1(C(N2CCCN(C(C3CC=CC3)=O)CC2)=O)CCCCC1 N1(C(C(CC=CC)C)=O)CCC2(CC1)CC2C(N1CCC(C)C1(C)C)=O NS(=O)(=O)C1(c2cn(CCNC(c3ccc(C4CC4)cc3)=O)nn2)CCC1 CSC1=C(C(=O)N2CCC3(NC(=O)CN4CCCC4)CC3C2)CCCC1 C1(NC(c2c(F)cccc2F)=O)CN(C(C2CC(C(F)F)C2)=O)CCC1CO c1(CC(=O)NCC2(CCNC(CC3CC(=C)C3)=O)CC2)coc2cc(C)ccc12 C1(C(N(C)CC2(NC(c3csc(=N)[nH]3)=O)CC2)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NCCOC2CCN(C(C(C)N(C(C)=O)C)=O)C2)nn(C)c2c1CCC2 C1(CNC(C(c2cnn(C)c2)OC)=O)CCN(Cc2ccc(Br)s2)C1 N1(C(C2(CCNC(C34C(=O)C5CC3C4C5)=O)CC2)=O)CC2CCC2(CC2CC2)C1 C(C(O)CC(=O)NCCCN1CCCC1=O)NC(=O)COc1ccsc1Cl c1(COC)n[nH]c(=NCC2(F)CCN(C(=O)CC3CS(=O)(=O)C3)CC2)s1 c1(C(C(=O)NCC)N(C)C(C2CCCCC2)C)ccccc1OCC c1(C(N(C2C(C)CCN(C(=O)CNC(C3CC3)=O)C2)C)=O)ncn2cccnc12 Cc1cn2c(n1)CC(C(=O)N(C1CCCCC1N(C(=O)C(O)CN(C)C)C)C)C2 c1(C(=O)NC(C)CCNC(=O)CN2CCC(C)(O)C2)cc2cccn2cn1 N1(C(c2ccc(OC)c(N)c2)=O)CC2CCC1C1CN(C(C3CC3C)=O)CC21 C1(C(N(CCC)C)=O)CCC2(CCN(C(C3CCc4nc[nH]c4C3)=O)CC2)O1 N1(C(c2cc(CCCC)on2)=O)CCC(NC(c2ccnc(SCC)n2)=O)CC1 C(C)(C(CO)NC(c1cc(-c2ccco2)c[nH]1)=O)NC(C1C(OCC)C1)=O CCC(C)CC(C(=O)NC1CC(O)C1OC)NC(c1nnc(S)n1C)=O Cc1c(C(=O)NC(C)C(C)NC(c2ccn(CCF)n2)=O)c(C(F)F)nn1C c1(OCC(=O)NC2(C)CC(NC(C(c3cccnc3)C)=O)C2)ccc(F)cn1 c1(CC)n[nH]c(CC)c1CC(=O)NC1CC1NC(=O)Cc1cc(C)[nH]n1 n1(CC(=O)NCC(CNC(c2ccc(O)cn2)=O)OC)nc(C)ccc1=O N1(C2CCC(NC(C3(CC)CC3)=O)C2)CCN(C(=O)C=Cc2ccoc2)CC1 C1(CC)(NC(C(CNC(=O)C(C)(C)c2cscn2)C2CC2)=O)CCCC1 c1(C(=O)NC(c2cccc(OC)c2)C(=O)O)c(Br)cc(Cl)c2[nH]ncc12 C1(CC=C)(NC(c2cccc(Oc3ccccc3)c2)=O)CCN(C(=O)C(C)C)C1 C1(C)(C(=O)NCC(C)C(=O)NCCN2CCC(C)C2)CCN(C)CC1 N1(CC)CCCCC1C(=O)NC(COC)C(=O)NC(C)COCC1CC1.C1CC1 C1(NC(C(C2CCCC2)OC)=O)COC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 N1(C(c2cnc(C)s2)=O)CC(C(=O)NC(C(O)CO)C2CC2)C(C2CC2)C1 N1(C(c2c(C)cnnc2)=O)CC2C(C1C(=O)Nc1c(Cl)cnc(Cl)c1Cl)C2(C)C CCCCC(C(=O)OC)N1CCC(C(=O)NC2CCCCC2)(OCC)CC1 c1(NC(=O)NCC2(CNC(=O)OC(C)(C)C)CC23CCC3)ccc2n[nH]cc2n1 C(=O)(CS(=O)(=O)CC)N1CCC(C(CNC(C(C)(C)OCCC)=O)C)CC1 Cc1cc(C(N2CC3CC(C2)N3C(C2CC=CC(O)C2)=O)=O)cc(Cl)c1 c1(C(N2CC(C)(CNC(c3c(C)nc(C)s3)=O)OCC2)=O)cc(C#N)ccc1O c1(CCC(=O)NC2CCN(C(c3ccc(OC)nn3)=O)C2)ccc(Br)c(C)c1 c1(CC2(C)C(NC(=NC)NCCn3ccnc3)C2)ccc(F)cc1 n1(CC)ncc2cc(C(=O)N(CC(C)(C)NC(=O)C(C)C(C)(C)C)C)c(C)nc12 C1(C(N2CC(C)C(NC(=O)CCc3ccc(Cl)nc3)C2)=O)CC12CCOCC2 c1(OC)cc(C#N)c(NC(C2CC2NC(c2ccc(Cl)c(F)c2F)=O)=O)cc1OC CC(C)C(C(=O)N(C)C)NC(=O)COCC(=O)NC(C1CCCC1)C1CCC1 C1(CNC(CC)=O)CCC(COC(C)(C)C)CC1.C12CC(C1)NC(=O)C2 c1(C(N(C2CC(NC(C(C)Cc3cccnc3)=O)C2)C)=O)nccnc1C(N)=O C(=O)(C(CO)C(C)(C)C)Nc1c(F)ccc(C(=O)OC)c1 C1(C)(CNC(CCCCN(C)C)=O)CC(F)(F)CN1C(=O)CC(O)CN(C)C C#CCC(C)C(=O)N(CCCCN(C)C(c1cn(C)nc1SC)=O)C CCC(CC)(C(=O)N1CC(CNC(C2CCN(OC)CC2)=O)C(F)(CO)C1)OC CC1CN(C(c2coc(C(N)=O)c2)=O)CC(CCNC(c2cnc(S)n2C)=O)O1 N1(C(CNS(CC)(=O)=O)=O)CC2CC2(CNC(C23CCC(OC)C2C3)=O)C1 N1(Cc2nnc(C(=O)O)n2-c2cccc3nsnc23)CCc2ccc(Cl)c(Cl)c2C1 N1(C(C(C)Sc2ccc(C(=O)OC)cc2)=O)CCC2(C1)CN(C(=O)CCOC)C2 C1(C)(C(=O)NC(C2CCOC2C)C)CCCN1C(=O)CCc1csnn1 C1(C)(C(=O)Nc2cn(CC(=O)N(C)C)nc2)CC(F)(F)CN1 Cc1ccc2nsnc2c1C(=O)NCCC(C)CCNC(=O)C(=O)NC1CC1 C1(C(=O)NC(CNC(c2cc(C)cc(C)c2)=O)CO)CC2CCC1C21CC1 Cc1cnc(Cl)cc1NC(C1CCN1Cc1ccc(-n2cccn2)cc1)=O C1(C(=O)NCC2N(C(CC=CCC)=O)CCC2)CCCC12CCC2 N1(Cc2cccc(C)c2)CCC(O)(C(=O)NCc2ccc(C)c(F)c2)CC1 C1(CNC(c2scc(C(=O)OC)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)CCC1C C1(C)(C(N(C(CC)C(=O)NCC(=O)N(C)C2CC2)C)=O)CC(C)=NO1 C1(C)(NC(C(F)=CCC)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(C(=O)NCC2CCN(C(C3CSCCS3)=O)CC2)CCCCCS1(=O)=O c1(C(N(CCCN(C(=O)C(F)(F)C(F)F)C)C)=O)ccc2nc(CO)[nH]c2c1 c1(-c2cc(-c3nc(CCC(CN(C(C)=O)C)O)on3)no2)ccc(Cl)cc1 c1(C(C(=O)NCC(C)NC(C(C2CCOC2)OCC)=O)=O)ccc(Cl)s1 c1(C(=O)NCC2C(C)CCCN2C(c2cc(Cl)cn2C)=O)cc(F)c(N)cc1F C1(NC(c2cncc(Cl)c2Cl)=O)CC(C(F)(F)F)CN(Cc2ccccc2I)C1 C1(CNC(=O)C2=NOCC2)CCN(C(=O)CN2C(=O)CNC2=O)CCC1(F)F c1(OC)ccccc1OC(C)C(=O)NC1(C)CC(NC(c2ccc(Cl)cc2)=O)C1 Cc1cc(C(=O)NCC2(F)CC(NC(c3ncccc3Cl)=O)C2)cc(F)c1 CN1CCC(C)(C(N2CC3CC(CNC(=O)CCc4ccsc4)C3C2)=O)CC1 C(=O)(CCS(=O)(=O)NC)NC(C(C(C)C)NC(CC=CC=C)=O)c1ccccc1 CCCCC(CC)C(=O)N1CCC(CO)C(NC(=O)CCOC)C1 N1(C(c2ccc(S(C)=O)cc2)=O)CC(C2CCCN(C(=O)C3=CCOCC3)C2)C1 c1(NC(C(=O)NC(CN(C(c2cc(C(C)=O)on2)=O)C)C)=O)ccc(F)cc1 c1(C(N2C(C(N(CC(C3CC3)OC)C)=O)CCCC2)=O)cnc2n1CCC2 c1(C(=O)NCCC2CSCCN2C(=O)CC2COCCO2)cnccc1Br C(CCCCCCO)NC(C1N(C(Cc2cccc(C)c2)=O)CSC1)=O N1(C(C=CCOCCOC)=O)C2CCC1C(F)C(NC(c1[nH]nc(OC)c1Cl)=O)C2 C(=O)(C1COc2ccccc21)N(CCC(C)(C)NC(c1cccc(C)c1F)=O)C C1(NC(C(CC(N)=O)NC(C2CCC(O)C2)=O)=O)CC2CC1CC21CC1 CC1CC(CNC(C2CSCCS2)=O)CN(C(=O)CC2CC(=O)NC(=O)C2)C1 c1(NC(C(CCNC(c2cn(C(C)C)nc2)=O)O)=O)cccc(Cl)c1O c1(N(C2CCN(C(C)=O)C2)C)nc(=NCC2C=CCC2)[nH]c2c1CCCCC2 C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(C(CCC)=O)ccc(S(=O)(=O)NCC(O)CC=CCOC)cc1 c1(NC(C2C(C(C)O)C2)=O)cccc(NC(=O)NCC2C3COCC23)c1 C1(C(N2CCC(CNC(c3c(CCC)occ3)=O)C2)=O)Cc2cc(C)ccc2S1 N1(C(c2c(C)nsc2C)=O)CCC2CN(C(=O)C(C)OCc3ccncc3)C2C1 c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)cccc(-c2nnc(C)o2)c1 c1(NC)ccc(C(=O)NC(CCC2CC2)C(=O)NCC2CC2)nc1 C(CCSC)(C(=O)N1CCCC1CNC(N)=O)NC(c1c(CCC)nco1)=O C1(NC(c2ccc(CC)c(F)c2)=O)CC1C1CCN(C(=O)C(C)(O)C2CC2)CC1 CC1CCN(C(C2CC(CF)C2)=O)C1c1cn(CC(F)(F)F)nn1 C#CCC(C)(C)C(=O)N1CCN(CC(=O)NC(C2(O)CCCCC2)C)CC1 CCCC(C)C(=O)NCCC(C)CCNC(c1onc(Br)c1C)=O N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)CC(NC(C1CCNC1=O)=O)C2 CC1CCCn2c(C(N3CC(CNC(c4cccc(F)c4)=O)C(C)C3)=O)cnc21 c1(OC)cc(C(C(=O)NCC2CCCO2)N(CCN=[N+]=[N-])C)cc(C(F)(F)F)c1 C12(NC(C(C)OCCOCC)=O)CC(NC(C3(OCC)CC3)=O)(C1)C2 C1(O)(CCn2cc(C3CCN(C(C(CC)(C)O)=O)C3)nn2)CC2CCC1C2 c1(CS(C)(=O)=O)nc(C(=O)NCCN(C(C2CC2C(N)=O)=O)C2CC2)cs1 C(CC1CC1)(CC(=O)N1CCOC(CCF)C1)NC(C(CC)=CC)=O N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC2(CC1)CC2CNC(c1cnc[nH]1)=O c1(C(C(=O)NC(CC(N)=O)c2ccccc2)N(C)C)cccc(F)c1 Cc1ccc(C)c(NC(C2(F)CCCN(C(c3cnc(C(N)=O)cn3)=O)C2)=O)n1 C1(CNC(COC)=O)CN(C(=O)CSc2nnnn2C2CC2)CCC1C(F)(F)F C1(C2CN(C(=O)C=CC(=O)NC3CC3)C2)(NC(C(CC=C)C)=O)CC1 C1(OC)CC2CC(c3nnnn3C3(C)CC3)(NCc3cc(Cl)ccn3)C(C2)C1 C1(NC(COCCSC)=O)CC2CC1N(C(=O)Cc1ncc(F)cc1F)C2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(c3cc(Br)c(Cl)s3)=O)CC2C1 C=Cc1cnn(C)c1C(=O)N(CCCNC(=O)CCc1cnn(C)c1C)C1CC1 c1(C(C(=O)NCC2CC(CNC(C3C=CCC3)=O)C2)(F)F)cccc(Cl)c1 C(=O)(C(C)C(O)CCCCC)NC1CC2CN(C(C=CCC)=O)CC1C2 C1(C(N2CC(NC(CCC=C(C)C)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(O)(C(C)NC(=O)C(F)=CCCF)CN(C(c2coc(C3CCC3)n2)=O)C1 CC1CCN(C(c2ccc(O)nc2)=O)C(C(=O)N(CCCF)C)C1 N1(C(C2(CO)CCN(C(CC(CC)SC)=O)C2)=O)CCC(C2(C)CC2)CC1 Cc1cnc2cccc(C(=O)NC(CO)C(C)(C)F)c2c1 CCCCCC(O)CC(=O)NC(C)(CNC(=O)CCCS(N)(=O)=O)CO N1(C(C(=O)NCCCC2CC2)C2CCCC2)CCC(c2ncccn2)CC1 C#CCCCCCC(=O)NCc1cccc(CNC(=O)CC2CCCCC2O)c1 N1(C(=O)Nc2c(C#N)cnn2CCc2ccccc2)CCCCNCC(F)(F)C1 C(=O)(C(CCC(C)(C)C)NC(=O)C(C12CCC(CC1)CC2)F)OCC N1(C(c2cc(C)c(C)nc2)=O)CCN(C(=O)CC2CCCCC2O)CCC1C CC(O)CCCCCC(=O)N1CC(C)(NC(c2ccc(NC(N)=O)cc2)=O)C1 C1(NC(C2=NNC(=O)C2)=O)COC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 N(C1c2ccccc2CC1NC(=O)C=C(C)Cl)C(C(CC=C)(F)F)=O C1(CCNC(COC(CC)C)=O)CN(C(c2cccc(C(C)(F)F)n2)=O)CCO1 c1(OC)nn(C)cc1C(=O)NC(C)CC(C)NC(C1CC(=O)N(C(C)(C)C)C1)=O C1(CC(N)=O)CCCCN1C(=O)N(c1cccc(C2CCCC2)c1)C1CCCC1 c1(C(N2CC(CN(C(C(CC)C)=O)C)C3(C2)CC3)=O)nc2nccc(C)n2n1 c1(CCOC(C)C)nc(-c2cnn(C)c2)n(-c2ccnc(Cl)c2)n1 CC1(C)OCCc2cc(C(=O)Nc3ccc(Oc4ccncc4)cc3)ccc21 N1(C(Cn2nc(C)oc2=O)=O)CCC(CNc2nccc(C)n2)C(C)C1 Cc1cc(C(N2CC=CC2C(=O)NCc2cc(C3CC3)on2)=O)nc(O)n1 C1(CC(=O)NCC(CCCC)O)N(C(=O)C(F)CC2CCOC2)CCC1(C)C c1(C(=O)NCCOCC(=O)N(C(CCC)C)C)cccc(CC#N)c1 S(=O)(=O)(c1ccc(N2CCC3(CCCC(C(=O)O)O3)CC2)c([N+](=O)[O-])c1)N(C)C C1(C(N2CC(C)(CCC(=O)NC3(CCC)CC3)C2)=O)CC2(C1)CC(C)C2 N1(C(COC2CCN(C(C(=O)N(C)C)=O)C2)=O)CCCC(C)(O)C1 O=C1COc2ccc(S(=O)(=O)NC3CCC(NC(c4ccno4)=O)C3)cc2N1 O=C1CC(=O)CC(C(=O)NC2CCCCC2CC(=O)NCCC2CCCCC2)C1 CCCCC(CNC(=O)CN(C)C(c1ccsc1C)=O)CCC C1(C(N(C2CCCCC2)CC=C)=O)CC(=O)NC(c2cnn(C)c2)C1 c1(C(N(C(CNC(C2C(C=C)C2)=O)C)C)=O)csc(C2CCCCC2)n1 C(CC(=O)N1CC(C)CC1CC)(C(F)F)NC(CCC=CCC=C)=O Cc1cc(N)cnc1C(N1CCC1(C)CC(=O)Nc1ccc(O)cc1)=O c1(C(=O)NCC(CC=C)NC(C2(C)CCCS2(=O)=O)=O)nccc2ccncc12 C12(C(N(CC(CN(C(=O)CCCc3ccncc3)C)O)C)=O)CCC(F)(CC1)C2 c1(C(=O)NCC(C)(C)CNC(C2(CC3CC3)CC2)=O)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2nn[nH]c21)NC1(CC)CCN(C(C2(CC#C)CCC2)=O)CC1 N1(CC(=O)NC2(CCNC(c3cc(C)sn3)=O)CC2)CC(=O)NC1=O Cc1cc(C(N2CC(NC(C3CCCCS3)=O)CC2CO)=O)cc(N)c1O C12(C(N3C(C)C(NC(c4cccc(CO)c4)=O)CC3)=O)C3C4C1C1C2C3C41C C1(=O)C(C)(C)N1.n1(C(C)C(=O)N(CCCN(C)C)C2CC2)ccc(NC(N)=O)n1 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)Cn2ccc(C)cc2=O)C(CF)C1 c1(OC)cccc(C(N2CCCC2(C)CNC(=O)CC2CSCCS2)=O)c1 C(=O)(C(C)C(O)C(C)CC)NCC1C(C(N2CCC(C(=O)NC)CC2)=O)CCO1 C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)N(CC(N2CCCC2)C)C)c1 Cc1cc(-n2nc(CSC3CCCCC3)nc2C23CC(C)(C2)C3)cc(C)c1 C1(OC)Cc2cc(Br)ccc2N(C(=O)C=CC(F)C(C)=O)C1.C(C(=O)O)C1C2CC21 c1(C(=O)NCC(CC)NC(c2sc(OC)nc2Cl)=O)cncc(C(=O)OCC)c1 C1(N(C(C(C)OCC2CC2)=O)C)CCCCN(C(=O)C=Cc2ccccc2)C1 Cc1ccc(CNC2CC(C(=O)Nc3nn(C)cc3C(F)(F)F)C2)cc1Cl N1(C(CC2C(C)CCCC2)=O)Cc2occ(C(N3C(CO)CC3C)=O)c2C1 C(c1cccc(Cl)c1Cl)=CC(N1CCC(NC(c2ccccc2)=O)C1)=O c1(C(N2CCC(C)(NC(c3c(C)n(C4CC4)nc3)=O)C2)=O)nnn2c1CSCC2 N1(C(CCCC2C(C)C2)=O)CCC2(CC2)CC1C(N1CC2CCOC2C1)=O CC(C)C(CO)C(=O)NC(C)CC(C)NC(=O)C(C)CCNC(=O)OC(C)(C)C C(=O)(CCCC(F)(F)F)N(C1CCCN(C(=O)CC2CCCOCC2)C1)CC c1(NC(=O)NC(C2CCOC2)CO)cccc(Cl)c1C(F)F C#CCC(C)(CC)C(=O)NCC1CCC1NC(c1nc(C)sc1C)=O C1(C(N(CCCCCNC(=O)CSCc2cccs2)C)=O)CC2CCC1C2 CC1(C)CC(NC(=O)C(S(C)(=O)=O)C2CC2)CN1C(=O)CCNS(C)(=O)=O c1(OC)cc(OC)c(CN2CCOCC2CC(=O)NCC2CCCN2C)cc1Br N1(C(CCN(C(C)=O)C)=O)CC(NC(=O)CC2CCC(C)(C)O2)CC12CCCC2 C1(C(=O)NCCN(C(=O)Cc2cncnc2O)C)OCC2CCCC12 N1(C(C2C(CC)C2)=O)CCN(C(c2cccc(F)c2F)=O)CCC1C c1(OC)cc(C(N2C(C(=O)OC)CC3OCCC23)=O)cc([N+](=O)[O-])c1N N1(C(C2C(CNC(C(C)C)=O)CCO2)=O)CCS(=O)CC1C N1(C(Cc2n(C)ccc2)=O)CC2ON=C(CNC(=O)Cc3ccc(Cl)cc3)C2C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)C2)=O)c(N)sc(C)c1C c1(OC)cc(C(N2CCC(CNC(c3ccoc3)=O)(OC)C2)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCCO1)N(C)CC1CCN(C(Cc2cnc(C)[nH]2)=O)C1 N1(C(C2C(C)=C2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CC2CO N1(C(C=CCOC)=O)CC(NC(c2cccc(-n3cncn3)n2)=O)C2(CCC2)C1 c1(CC(N2C(CN(c3cc(O)nc(C)n3)CC)CCC2)=O)nnc2n1CCCC2 Cc1ccc(C(=O)NCC2(C)CN(C(=O)C(c3cncn3C)O)CC2C)c(N)n1 CC1=CC(NC(=O)C(CC2CCOCC2)NC(=O)C(C)C#N)CCC1 c1(OC)cc(C(=O)NC2(CO)CN(C(C3(C4CCCO4)CCC3)=O)C2)cnc1O C1(CNC(N2CC(C(=O)NC)C2)=O)(Cc2ccccc2)CCOCC1 S(=O)(=O)(c1ccc(Cl)cc1)N1CCC(NC2CCS(=O)(=O)C2)CC1 N1(C(=O)CCc2ccoc2)CCN(CC2CN(C(C3(O)COC3)=O)C2)CC1 c1(-c2cc(C(=O)N(CC3N(C(CCC=CC)=O)CCC3)CC)on2)ccc(F)cc1 C(CO)(C(=O)NC)N(C)C.c1(C(=O)NC2CC2)cn(CCC2CC(O)C2)nn1 c1(NC(C2COCCN(c3c(C)cncn3)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1CCCCN(C(CCC=C)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C(=O)NC2CN(C(N)=O)C2)CC1 C1(C)(CNC(Cc2c(C)n[nH]c2)=O)CN(C(=O)Cn2cccc2)CCO1 N1(C(CN(CCOC)C)=O)CCC2CCN(C(=O)C(=O)NC(C)C)C2C1 CCC(CNC(=O)C(C)Cc1ccco1)(CC)NC(c1ccc(CC(C)C)s1)=O c1(C(N2CC(N(C)C)C2)=O)cc(CN(C)C(C2(c3cccnc3)CC2)=O)nn1C c1(C(=O)NCC(CC=C)NC(C2(C(=O)NC)CC2)=O)ccc2cc(Cl)ccc2n1 N1(C(c2ccc(N)c(F)c2)=O)CCCC(O)(CNC(c2ccoc2)=O)CC1 CC1(CNC(=O)Cc2cc(F)ccc2F)CN(C(=O)C(F)CC2CCC2)CCO1 N1(C(c2nccc(C3(C)CC3)n2)=O)CCCC2(CCO2)C1 c1(C(=O)NC(CCNC(c2c(C)cccc2C)=O)C)ccc(C#N)cc1O O=S(=O)(c1cncc(Br)c1Cl)NCc1csc2c(F)cccc12 C12CN(CC(C)(C)C1)C(=O)N2.C(=O)(C(C)(C)OC(=O)OC)OCC C=C(C)CCC(=O)NC(C)CCN(C)C(c1ccccc1C1CCC1)=O CN1CCN(c2cc(C(=O)NCC3(SC)CC(F)(F)C3)ccn2)CC1 CC#CCCCC(=O)N1CCC(NC(c2ccncc2SCC)=O)C(CO)C1 N1(C(C)C)CC(CNC(N2CCC(O)(Cc3cccc(F)c3)C2)=O)CC1=O c1(C(=O)NCC(CN(C(C2(C(=O)NC)CCC2)=O)C)C)ccc2cc[nH]c2n1 C1(C(=O)NCCC(=O)NC2CC2)CC2(CCN(C(=O)NCCCCl)CC2)CO1 Cc1[nH]c(C)c(C(=O)NCC2(O)CC(C(=O)NCC3(O)CCC3)C2)c1C c1(C(=O)Nc2cccc(NC(c3cccc(C#C)c3)=O)c2)ccc(F)c(C)c1Cl C1(C(=O)NCC2(OC)CCN(C(C3CCC3)=O)C2)CCn2c(C)cnc2C1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)COCc2nc(C)no2)C2CC12 C(=O)(C(F)C(=O)NC1CCN(CCNC(=O)C(C)n2cnnn2)CC1)OCC C(=O)(C1=C(C(C)(C)C)N(C2CC2C)C(=S)NC1c1c[nH]c2cccnc12)OC Cc1sc(C(=O)NCCCCCNC(c2cnn(C)c2CC(C)C)=O)nc1O c1(OCC(=O)NC2C(NC(c3cc(C)no3)=O)C2)c(F)cccc1F N1(C(c2cc(C(N)=O)oc2)=O)CC(NC(=O)CN2CCSCC2)CC(F)(F)C1 C1(N(C(C(C)OCC=C)=O)CC2CC2)CCCN(C(c2cnsn2)=O)C1 CC(C)C(O)C(=O)NC1CC(CCC(N2CCC(n3cnnn3)C2)=O)C1 N1(C(C2CN(CC)C(=O)CC2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 C1(C(=O)NCC(C)CC(=O)N(C)Cc2ccccn2)Cc2nccn2C1 C1(N(C(c2nnn(C)n2)=O)CCN2CCC2c2ccccc2)CC2CCC1O2 N12CCN(CC1)C(=O)CC1CCN(C1)CC2.C1(C(=O)OCC)CCCN(CC)C1 CC1(C(N2CC(NC(=O)CCn3c(O)nnc3O)C2)=O)CC=CCC1 N1(C(c2nn(C)c(O)c2)=O)CCCC2C(NC(c3ncccc3Cl)=O)C(C)(C)C12 c1(-n2cc(C3(C)CN(C(C(F)(F)C4(C)N=N4)=O)C3)nn2)cccc(C#N)n1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C(CO)C1 N(C1CC(C)n2ccnc21)C(COCc1c(C)cccc1)=O c1(OCCC(=O)NC2CC(NC(=O)Cc3cscc3Br)C2)cccnc1 CC1CC(C)N(C(c2ccoc2)=O)CCN1C(=O)C=C1CCSCC1 C=CC(C)C(=O)NC1CCN(CCCNC(=O)CCCn2cccn2)C1 N#Cc1ccc(C(N2CCCCCC2NC(c2cn(C3CC3)nn2)=O)=O)cc1O C1(CNC(c2nnc(C)s2)=O)CC(F)CN1C(c1cc(C)n(C(F)F)n1)=O C1(C(F)F)(CNC(=O)C=CC2CCOCC2)CCN(C(c2ccc(F)cn2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CC(C2CN(C(=O)C=Cc3cccc(CO)c3)C2)C1 C(=O)(C1=NOC2COCC12)NC1C(C(=O)NC2CC(C)(C)C2)COC1 C1(CNC(C2(P(C)(C)=O)CC2)=O)CC2CCC1N(C(=O)CN1CCCC1=O)C2 C1(C(=O)NC2C(NC(=O)C=Cc3ccccc3)COC2)CCn2c(O)nnc2C1 CC1(F)CN(C(=O)C(c2ccc(Cl)c(Cl)c2)O)CCN(C(C2CC(O)C2)=O)C1 c1(COC(C2CCCN(Cc3ccccc3)C2)=O)ccc(C(F)(F)F)cn1 C1(OCCOC)CCN(C(=NCC2(OC)CCOCC2)NC2CCCC2)C1 N1(C(=O)CSc2ccc([N+](=O)[O-])cc2)CCC2(CC1)COCCO2 N1(C(c2c(C)noc2)=O)CCN(C(=O)CCS(N)(=O)=O)C(CCO)C1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CCn4ccnn4)CC23)c(O)n1 C#CCC(C(=O)NCC(C)(O)CNC(c1sc(C(C)C)nc1C)=O)C1CC1 C(=O)(C1=CCN(C(=O)CCNC(=O)C(C)(C)C)C1)N(CC(CC)O)C CC1CN(C(=O)CCCc2ccccc2Cl)CCC1NC(=O)C(F)F Oc1cc(Cl)ccc1-n1cc(CO)nn1.C1(OCCCN)CCNCC1 O=C1NC(CNC(=O)C(=O)NC(C2CCCCC2)C2CCCO2)CO1 CCC(CC(C)C)C(=O)N1CCC(F)(C(=O)NCc2cnco2)C1 Cc1ccc(C(=O)NC(C)CNC(c2ccc(-c3cnc[nH]3)cc2)=O)c(Cl)c1 c1(C(=O)NCCCCNC(C2CCC(F)C2)=O)ccc2nnn(O)c2c1 N1(C(c2ccc(C#N)[nH]2)=O)CCN(C(c2csc(CO)n2)=O)C2CCCCC12 N1(C(C(C)(C)c2nccs2)=O)CCC(C2CCN(C(=O)Cc3cc[nH]c3)CC2)C1 N=c1[nH]ccc(C(=O)NC2CCCC2NC(C2CC3CCC2C3)=O)c1[N+](=O)[O-] C1(NC(c2ccc3cc[nH]c3n2)=O)COC2(CCN(C(=O)COCC(F)F)C2)C1 CC12CN(C(c3cscn3)=O)CC1CN(C(C1CCCCC13OCCO3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CNC(C2CN(C)C2)=O)CC1 C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2cccc(O)n2)=O)C1 c1(C(=O)NC2(C)CC(NC(=O)CN3CC4CCC3C4)C2)cccc(O)c1Cl C1(CNC(CCN(C)CCO)=O)CC2(C1)CN(C(=O)C(F)C1CCOC1)C2 c1(C(=O)NCCOCCN(C(=O)CC2COC(=O)N2)C)ccc(Cl)c(O)c1 N1(C(CNC(C)=O)=O)C2CCC(C2)C1CC(=O)NC1C(O)C2CCCC12 C1(NC(c2n(C=C)nnc2)=O)CCSC12CN(C(=O)C=Cc1ncc[nH]1)C2 c1(C(=O)NCCSCC(=O)NCCC2CCCC3CC23)cc(O)cc(F)c1 c1(CC)nnc2cc(N3CC(NC(C4CC4(C)Br)=O)CC4(CCC4)C3)ncn12 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C c1(C(=O)NC(CCCCNC(CC)=O)CO)cc2c(ccc3ccccc23)[nH]1 CC1CC=C(C(=O)NCC2CC3CC3N2C(C2CN(C(N)=O)C2)=O)CC1 CCCC(C)(O)CC(=O)N1CC(CCC(=O)NOCCO)(C)C1 C(=O)(C1(C)OC(=O)c2ccccc21)NCC(n1cc(Cn2ccnc2)nn1)C C(CC(C(=O)NC(C)CO)NC(=O)CCc1csnn1)=CC C1(=CC(=O)NCC2(O)CN(C(C(OC)OC)=O)C2)CCC(C(C)(C)C)CC1 CC1OC2(C(=O)NCC=CCNC(c3cnccc3Cl)=O)CCC1C2 C=CCC(CC=C)C(=O)NCC1(C)CN(C(C2(C)CC=C(C)CC2)=O)CCO1 N(C1CN(C(=O)Cc2cnn(C)c2)Cc2ccccc21)C(C(CCCC)F)=O n1(CC(=O)N(C)CC2CC(OC)C2)cncc1C c1(C(=O)NC2(CC=C)CN(C(=O)C(F)(F)c3ccccc3)C2)cc(C)ccc1F C1(NC(c2cc(-c3cccs3)on2)=O)CC2(C1)CN(Cc1csc(Br)c1)C2 c1(C(=O)NCC2CC(C)N(C(C3CC(=C4CCC4)C3)=O)C2)ncc(C#N)cc1Cl N1(C(CC(CC(=O)OC)C)=O)CCC2C1CCCN2C(c1cc(Cl)ccn1)=O c1(CC(=O)N(CCCN(C(C(C2CC2)OC)=O)C)C)ccc(Cl)cc1Cl Cc1ccnc(C(N2CCC(NC(c3cnc(-c4ccsc4)s3)=O)C2)=O)c1 c1(OC)cc(C)ccc1N(c1cc(C)nc(-c2cnccn2)n1)Cc1cccs1 N1(C(C2CCSCC2)=O)CCC2CCN(C(=O)Cc3ccc(F)cc3)C2C1 c1(C2(CCC(N(CCCNC(=O)CCc3nc[nH]n3)C)=O)CC2)ccc(O)cc1 CC(O)C(C(=O)N1CCN(C2CC(CNC(=O)CC3CC3)C2)CC1)NC(N)=O C(=O)(C1=CCCN(C(C2CC2(F)F)=O)C1)NC(C)C(C)F C1(C(=O)NCC(=C)Br)CNC(=O)CN1C(C1COCC(C)O1)=O N1(C(C2CCC(C(=O)OC)CC2)=O)C2CCCC1CC(NC(c1ccoc1)=O)C2 N1(C(C(CC)CNC(=O)OC(C)(C)C)=O)CCCC(C)(NC(=O)C=CBr)C1 N1(C(C(C)(C)C(N)=O)=O)CC2C3CCC(C2C1)N(C(c1ccnnc1)=O)C3 N1(C(c2cc(C)n(C)c2)=O)CCN(C(=O)COc2ccc(F)cn2)C2CC12 c1(-c2nc(C(C)C)nn2-c2ccnc3cccnc23)cc2cc(Cl)ccc2o1 C(=O)(CC(C(F)F)C(C)(C)C)NC(CNC(C1N(C(C)=O)CC(O)C1)=O)CO C1(C(=O)OC)N(C(c2cc(C(F)(F)F)ccc2F)=O)CC12CCC2 CC1CC(n2nc(C3CCCO3)nc2-c2cc(-c3ccoc3)[nH]n2)CCO1 c1(C(N(CC(CC)O)C)=O)cn2c(n1)CCN(C(c1cccc(F)c1C)=O)CC2 CC(C)(C)CCC(=O)NC1(CCCNC(=O)CC2CCC3(CCC3)O2)CC1 c1(OC)cc(Cl)ccc1CNc1cc(NC23CCC(C2)C3)ncn1 N1(C(c2cc(C(=O)OC)sn2)=O)CCC2(NC(c3cccc(SC)c3)=O)CC2C1 c1(C(=O)NC2(C)CN(C(C34CCC(C(F)F)(CC3)C4)=O)C2)ccc(Cl)c(O)c1N c1(C(=O)NC2CN(C(C3CCO3)=O)CC2F)c[nH]c2c(Cl)cccc12 CCCC(C(C)CC)NCC(C)(C)CC C(=O)(C(C)(C)C1=CCSCC1)NCC(C(C)C)NC(C(=O)NCCOC)=O C1(NC(CSCCCC)=O)CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1C1CC1 C1(CC(=O)NC2CCN(C(c3cnn(C(F)F)c3)=O)CC2)CCCOCC1 CC1=NOC(C(N2CC(C(N)=O)(CNC(C3CC(C)(O)C3)=O)C2)=O)C1 c1(C(N2C(CNC(CNC(=O)OC)=O)CCC2)=O)cncc(C(C)(C)C)c1 c1(C(N2CCCC(N(C(=O)CCC3CC3)CC)C2)=O)cc(N)nc(Cl)c1 S(=O)(=O)(c1cccc(N2CCC(C)(N3CCCC3)C2)n1)N1CCC(C(C)O)CC1 Cn1cnnc1C1CCCC1C(=O)NCCN1CCC(NC(C2(CF)CC2)=O)C1 c1(C(N(C)CC2CCN(C(C(C)(C)SC)=O)C2)=O)ccc2cnoc2c1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NCC(F)C(C)(C)O)C2)=O)C1 c1(C(=O)NC(C)CCCNC(c2cc(CN(C)C)c[nH]2)=O)c(F)ccc(F)c1Cl CC1=C(C(=O)N(C(C)CN(C)C(C2CC3(CC3)CO2)=O)C)CCS1(=O)=O c1(COC)cc(C(=O)OC)cc(S(=O)(=O)NC(C)(CC)C2=CCCC2)c1 c1(OC)ccc(CC(=O)NCC2CN(C(=O)Cc3ccc(C)s3)C3CC23)cn1 C=CC1(C(=O)NC2(C(O)CO)CC2)CCN(C(c2c[nH][nH]c2=N)=O)C1 C(=O)(C(CCF)NC(C1CC(COC)C1)=O)NC1C(CCOC)C1 c1(C(=O)NC2CCC(CNC(CC3CC(=C)C3)=O)C2)c[nH]c(=O)c2ccncc12 N1(C(c2c(OC)ccs2)=O)CCN(C(c2ncc(C3CC3)cc2F)=O)C(CF)C1 C1(C(N2CC3C(NC(=O)Cc4ccns4)(CCC3)C2)=O)CC12CCC(F)(F)CC2 C1(OC)(CNC(=O)CCC2(C)CC2)CCN(C(c2cnn(C)c2Cl)=O)C1 C1(CN(C2CC(NC(C(C(CC)C)NC(C)=O)=O)C2)C)CCCCCCC1O N1(C(C2CN(S(N)(=O)=O)C2)=O)CC2CC1CCC2NC(c1ccncn1)=O CC1CCC(Nc2cccc(NC(N)=O)c2)CS1(=O)=O c1(C(=O)NCC(COC)NC(=O)C(C)CN(C)C)cc(C)c[nH]1 c1(N(C)CC2CC3CC3C2)cc(NCCCO)nc(C(F)(F)F)n1 C1(NC(=O)OCC)CCCN(C(=O)CC(=O)N(c2nc(C)nn2C)C)C1 N1(C(C(C2(O)CCC2)NC(C(C(C)C)C#N)=O)=O)CCC2CN(C)CC2C1 c1(C(C(N2CC(N(C(=O)CCOC3CCCOC3)C)C2)=O)O)ccc(F)cc1 c1(C(N2CCC(C)N(C(=O)CC3CCCC3)CC2)=O)cncc2c(F)cccc12 C1(NC(Cc2c(C)n(C)nc2)=O)CN(C(=O)Cc2nc[nH]n2)CC(F)(F)C1 n1(CCSC)nnnc1C(c1csc(-c2ccsc2)n1)NCC(C)OC C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(CN(C)C)cco2)=O)C1 CC1(C)CN(C(=O)CCCc2cccnc2)C(CNC(=O)CC2C=CCC2)CO1 C1(CNC(C(C)=CC)=O)COCC1n1cc(CNC(=O)CC2(C)CCCC2)nn1 C1(C(=O)NC(CCNC(C(C2CCCCC2)OC)=O)C)CN(S(N)(=O)=O)C1 C12(C(N3CCC(CCNC(Cc4nc(C)oc4)=O)C3)=O)CCC(C1)OC2 c1(-n2c(SC)ncc2)ccc(C(=O)NCCCN(C(=O)Cc2ncco2)C)cc1 C(=O)(C(C)(C)CNC(C12CCCC1(C(N)=O)C2)=O)OC N1(C(CC(=C)C)=O)CCC2CC2(NC(c2sc(-c3ccsc3)nc2C)=O)CC1 c1(CNC(C2(F)CCN(Cc3cncc(C)c3)C2)=O)cccc2cnccc12 C(=O)(CCC(C)NC(c1ccc[nH]1)=O)NCC(CC1CC1)OC N1(C(C2CC3CCC3C2)=O)CCC2OCCN(C(=O)Cc3cn[nH]c3)C2C1 c1(C(C)C)cccc(NC(=O)C(C2CCCC2)NC(=O)C#CC2CC2)c1 N1(C(C)=O)CCCc2cc(NC(C3(Cl)CC3(F)F)=O)ccc21 C1(NC(=O)C(N2CCC(C(F)F)C2)=O)CCC(CO)CC1 N1(C(C(C2(C)CC2)NC(c2cc(C)c(F)cn2)=O)=O)CCN(C)CC(C)C1 C1(C)(N(C)C)CCN(C(c2ccncc2)=O)CC1.C12CCN(C1)CC(=O)NC2 C(=O)(C(C)CC(N)=O)N1CC(CC=C)(C(=O)NC(c2ncccn2)CC)C1 C(=O)(C(CNC(c1cc(C)c(C)s1)=O)(CC)CC)NCC(=O)NCC=C C1(C(=O)OCC)C2COC(C(=O)N(CCCN(C)C(C3(CC)CC3)=O)C)CC12 CC1CC(=O)CCC1C(=O)NC1CC(CC(=O)NCc2cnccc2Cl)C1 C1(C(=O)NCC2N(C(CCOCCOCC)=O)CC3CC32)CCC=CCCC1 c1(OC)ccc(C(=O)NC2CCCCC2CNC(=O)C=CC(C)C)cc1N Nc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C(F)=C2CCCC2)nc1N C1(NC(CC2(NC=O)CCC2)=O)COCC1C(N1CCC(c2nn[nH]n2)C1)=O Cc1cnc(C(N2CCCC(NC(=O)CC3(C(F)(F)F)CC3)C2C)=O)c(F)c1 C1(n2cc(CN)nn2)CCCN(C(c2cc(N)ccn2)=O)C1.CC1(C)CC(CO)O1 Cc1cc(C(=O)NCC2CN(C(c3nn[nH]c3Cl)=O)C3(CCC3)C2)cc(=O)n1C Cc1c(C(=O)N(C)CC2CCCN2C(c2nncn2C2CC2)=O)cccc1C#N N1(C(c2cnc(OC)nc2C)=O)CC2(CCN(C(=O)CCCC(F)F)C2)C1 c1(C(=O)NC2(CNC(C3C(C)SCCC3)=O)CCCC2)cnn(C)c1C#N c1(C(=O)NCC2CCN2C(=O)CCOc2ccccc2)ncccc1Br C=CCC(C(=O)NCC(C1CCN(C(=O)C(C)O)CC1)O)NC(C)=O C1(C(=O)NCCOC(C)(C)CNC(c2nc(C3CC3)cs2)=O)OC2CCC1C2 N1(C(C(C)NC(C)=O)=O)CC(F)(F)CC1(C)CNC(c1cc(S(N)(=O)=O)c[nH]1)=O c1(NC2C(C(F)F)CCC2)cc(NCc2cncc(Br)c2)ncn1 N1(C(CC(=C)C)=O)CCC2(CO)CN(C(c3cnn(C)c3)=O)CC2C1 N1(CCN(C(Cn2ncc(C)c2)=O)C)CCN(C(=O)C(F)C2CCCC2)CC1 CC(C)C(C)(O)C(=O)N1CC(CNC(c2ccc(Cl)s2)=O)C(F)(F)C1 CC(CCO)N(C(=O)CC1(NC(=O)CSC2CC2)CCC1)C C1(COC)(CNCc2cn(C)nc2Br)CCCN1C(=O)OC(C)(C)C C(=O)(C(C)(C)CCNC(c1cnn(C)c1)=O)NCC(=O)N(C)C NC(=O)CCCCC(=O)NCC1(O)CCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 CC1(CNC(C2CC3(CC3)C2)=O)CN(C(c2ccnc(Cl)c2O)=O)CCO1 CC(C)CC(C)C(=O)NCC1CN(C(C2CSCC(=O)N2)=O)CCN1C CC#CCCC(=O)NCC1CCCC(NC(c2cnn(CC(F)F)c2)=O)C1 N#CCS(=O)c1ccc(C(N2CCC2CNC(=O)C(=O)NCC2CC2)=O)cc1 Cc1ccc(O)c(NC(=O)CC2CCN2C(c2ccc(=N)[nH]n2)=O)c1 C1(CNC(CCC)=O)CC2CN(C(=O)Cc3ncc(C)s3)CC12 CCC(CO)(C(=O)NCC1(C(=O)NCc2cccnc2)CC=CC1)OC C1(NC(C(c2ccccc2F)C)=O)COC2(CCN(C(c3ccoc3I)=O)C2)C1 c1(C(N2C(CNC(c3c(CC)occ3)=O)CC2)=O)cc2c(cc1N)OCO2 Cc1cnccc1-n1nc(CO)nc1CCN(C)C c1(OCC(=O)N(C2CC2)CC2CCCN2C(=O)C(O)C2CCC2)cnc(Cl)cn1 C(C)(C(=O)N(CC(C)N(C(=O)CSC(C)C)C)C)(C1CC1)OC N1(C(c2n(CCOC)ncc2)=O)CCC2(CCCN2C(C2CCN(C)C2)=O)C1 c1(CCC(=O)NCCC(CN(C(=O)COc2ccon2)C)O)cccc(F)c1F C1(CCC)(C(N2CC(O)(C(C)NC(c3cncc(F)c3)=O)C2)=O)CCNC1=O c1(OC)ccc(F)c(C(=O)N(C)CCNC(C2(CSC)CC2)=O)c1Cl C1(OC2CCN(C(C(C)O)=O)C2)CCN(C(=O)COCC2CCCC2)CC1 CC(CC1CC1)C(=O)NCC1(C(=O)NCCSC(F)F)CCCO1 C(=O)(N=S1(=O)CCNC(C)CC1)N1C(C)c2n(cc(C(C)C)n2)CC1 N1(C(C2(C)CC2)=O)CCC2(C1)CN(C(=O)C=C1CCOc3ccccc31)CCO2 C1(C(=O)NCCN(CCOC)C(c2cscc2C(N)=O)=O)CS(=O)(=O)C1 c1(CC)n[nH]cc1C(=O)NC1(CNC(=O)CN(C)CCOC)CC(F)(F)C1 C#CCC(CC(=O)N(CCCCO)C)NC(c1cc(C)c(N)cn1)=O Cc1cnnc(O)c1C(=O)NCC1CC(F)CN1C(C1CC2(C1)CC(F)C2)=O CN1N=C(C(=O)N2CC(NC(=O)Cn3ncc4cccnc34)C(F)C2)CCC1=O c1(C(N2CC(C=C)(CC(=O)NC3CCS(=O)(=O)C3)C2)=O)cc(O)ccc1F C12CCC(CC1)OC2=O.C1(C(=O)OCC)(NC(=O)C(C)NC(C)=O)CCOCC1 c1(C(=O)NCC2CCC(NC(C3(CC4CC4)CC3)=O)C2)ccc(O)nc1 N1(CC)CC(C)N(C(C2CCN2C(=O)Cn2nc(C)cc2C)=O)CC1C c1(C(=O)NCC(N2CCC(O)CC2)C)ncc(Oc2ccc(F)cc2)cn1 c1(OC)nc2ccc(C(N3CC(NC(c4cc(CO)ccc4Cl)=O)C3)=O)cc2[nH]1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)[nH]cc2c1CCCC2 c1(C2CN(C(c3nc(-c4cccnc4)cs3)=O)C2)cccc(Br)n1 c1(C(=O)NCCC2(C)CNC(=O)C2)ccc2cccc(F)c2n1 N1(C(c2n(C(C)C)ncc2)=O)Cc2ccccc2C1C(=O)N1CC2CC2C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NC1C(F)CCN(C(C(C)(C)O)=O)C1 Cc1cccnc1CC(=O)NCCC1CCN(C(C2CCC(O)C2)=O)CC1 c1(N2C(CNC(CC3C(C)=NOC3=O)=O)CCC2)nc(C)cc(C)c1C#N N1(C(C2(CC)CCN(C(c3cccnn3)=O)C2)=O)CC2CCC(C1)O2 n1(CC)nnc(C)c1CNC(=O)CC=CCNC(C1(O)CCCC1)=O C(C(=O)NCC(O)C(C)C)(C(C)C)NC(C1(CC=C)CC=CC1)=O N1(C(c2cn(CCC=C)nn2)=O)CCC(F)C(NC(c2ccc(Cl)cc2F)=O)C1 N1(C(Cc2scc(C)c2)=O)CCN(C(c2nnc(O)cc2O)=O)CC1CC(F)F c1(C(=O)NC(C2CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)C)cn(C)c(=O)n1C Cc1sc2ccccc2c1NC(=O)NC1(C)CN2CCC1CC2 c1(NS(CC)(=O)=O)ccc(C(=O)NCC(C)CNC(=O)CC(O)CSC)cc1F C1(C(=O)NCC2CCCN(C(c3cnn(C4CC4)c3)=O)CC2)CCCS(=O)(=O)C1 N1(C(CN(C(Cc2n(C)ccn2)=O)CC2CC2)=O)CCC(NC(=O)C2CC2)CC1 N1(C(CCC=CC)=O)CCN(C(=O)CC(C)NC(N)=O)CC2(CC2)C1 CC(C)CCCCC(=O)NC1CC2(C1)CC2C(=O)NCC1CCCN1C c1(C(=O)NC2CC3N(C(C4CC(OC)C4)=O)C(CC3)C2)cnn2c1C(C)CCC2 C(=O)(CC(C)(C(F)(F)F)N(C)C)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C C1(C(=O)NCc2cncc(C)n2)C2CCC(C2)N1C(=O)C(c1ccccc1Cl)O C1(NC(C2CC3C=CC2O3)=O)CCN(C(c2ccc(Br)s2)=O)C12CC2 C1(NC(C2C(C)CCO2)=O)CCCC(C(=O)NC2CC3CCC2C3)C1 C1(COCC(=O)NOc2ccccc2)CCCCCN1C(C(C(C)O)=O)=O c1(C(=O)NC(CC2CCN(C(c3ccn(CC)n3)=O)CC2)C)cc(Cl)ccc1N CCCCCC(CC)C(=O)N1CCC2(CC(NC(=O)C(F)C(C)C)C2)C1 c1(CN2CC3(CCC(C(=O)N(S(CC=C)(=O)=O)C)O3)C2)sc2ccccc2c1Cl CCCC(C)CC(=O)NCC(C1CCN(C(=O)Cc2cc(F)ccc2O)CC1)C C1(N(C(c2csc(-c3ccccc3)n2)C(=O)NCCCF)CC)CCN(C)CC1 c1(C(=O)NC2(CN(C(CCCOCC)=O)C)CC2)cc(Cl)c(Cl)[nH]1 N1(C(C2CCC(CC)O2)=O)CCC(NC(c2ccc(CO)s2)=O)C(CO)CC1 C1(CNC(C23CCC(OC)C2C3)=O)CN(C(c2cnn(C)c2N)=O)C2(CCC2)C1 c1(C(=O)NC2CCC(CCNC(CC(=C)C)=O)C2)c[nH]c2cc(OC)ccc12 Cc1cc(C(=O)NC(c2ccccc2)CNC(C2CC(C#N)C2)=O)ccc1O O=C1NCc2ccc(NC(C3CC3NC(C3(C(F)(F)F)CC3)=O)=O)cc21 CC1CC(CCNC(C2(C(N)=O)CC2)=O)CCN1C(c1ccc(Cl)o1)=O c1(C(=O)NCC2(F)CCN(C(C(CC)COC)=O)C2)coc2cc(OC)ccc12 CCS(=O)(=O)CC(=O)N1CCC(N(C(C2CCCN2C(C)C)=O)CC2CC2)C1 Cc1cccc(C(=O)NCC2(NC(c3cccn3Cc3ccccc3)=O)CC2)n1 c1(CC(=O)NC2C=CCN(C(=O)CC3C=CCC3)C2)cccc(-c2ccsc2)c1 CC1CN(C(C2CCS(=O)CC2)=O)CC1CNC(C1CN(S(C)(=O)=O)C1)=O C=CC1(C(=O)NC(C)C(=O)NC(C)C)CCN(C(c2cc(O)nc(O)n2)=O)CC1 C(=O)(C1=NOC(C)C1)NC1(CF)CN(C(Cc2c(C)nn(C)c2)=O)C1 CCCC(CC(C)C)C(=O)NC(C)(C)CCCNC(=O)COCC(F)(F)F N1(C(c2ccc(SC)s2)=O)CC2CC2(CNC(C2CC(C)(C(C)=O)C2)=O)C1 c1(CNC(C2(C(C)NC(C3CC(OC)C3)=O)CC2)=O)cnn(CC)c1 C1(C(=O)NC(CC)C(N)=O)CCC2(CCN(C(=O)CCc3cccnc3)CC2)C1 c1(CC(C(=O)NCc2conc2C2CC2)NC(N)=O)ccc(O)cc1 O=C(C1=C(Cl)CCCC1)NC12CCCC1CN(C(c1ncccc1F)=O)C2 N1(C(c2cc(Br)ncc2F)C(=O)NC)CCc2cc(OC)cc(OC)c2C1 c1(CC(=O)OCC2C(C(=O)OCC)(C(=O)OCC)C2)cncnc1O c1(C(C)NC(=O)CC2CCCN(C)C2)ccc(CNC(c2cnn(C)c2)=O)cc1 CCCCCC(=O)NC1CC(NC(=O)COCP(C)(C)=O)C(O)C1 CN1C(=O)C(O)C(C(=O)Nc2ccc(Cl)cc2C(=O)O)C1c1ccccc1 C1(CC#C)(C(N2CC(C)(N(C)C)C2)=O)CCN(C(=O)C(C)COC(C)=O)C1 Cc1cc(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)C2)nn1C1CCOCC1 C(=O)(C(C)N=c1cncc[nH]1)N1C2(CCN(C(c3ncc(CC)s3)=O)C2)CCC1 c1(N(CC)CC2CCN(C(c3csc(O)n3)=O)CC2)ncc([N+](=O)[O-])cc1C#N S(=O)(=O)(c1cncc(Br)c1)N1CC(NC(c2cc(Br)c(Cl)cc2F)=O)C2(C1)CC2 c1(CC)[nH]nc(C(=O)NCC=CCNC(=O)C(C)Cc2ccco2)c1[N+](=O)[O-] O=C(CC1OCc2cc(Cl)ccc21)NC1CC(CNC(C23CC(CO2)C3)=O)C1 N1(C(c2ccc(COC)o2)=O)CC(NC(c2cc(C#N)oc2C)=O)CC12CCC2 c1(CC)cccc(C(=O)NCCN(C)C(C2(C3CCCO3)CC2)=O)c1C c1(C(C(=O)NCCCNC(C(CC=CCC)C)=O)C)ccccc1S(N)(=O)=O N1(CC)CCOC(C(=O)N(CCC(=O)NCC(N2CCCC2)C)C(C)C)C1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 C1(CC#C)(NC(C2CCCC(NC(=O)C(C)c3cc[nH]n3)C2)=O)CCOCC1 CC(C)CC(CC(=O)NCCCC(C)NC(=O)CC1(N2CCCC2)CC1)CC(N)=O CC(C)C(O)C(=O)NC1(CCNC(=O)C(C(C)C)NS(C)(=O)=O)CCCC1 c1(N2C(C)CC(NC(C3CCC(=O)N3C)=O)CC2)nc2cccnc2s1 N1(C(C=Cc2cn(C)nc2)=O)CCC2CCNC2C1 C(CC)(C(=O)NCC(CNC(=O)Cc1c[nH]nc1C)OC)OCC c1(C(C)NC(C(COCC)NC(=O)Cc2nccn2C)=O)cccc(C)c1 c1(C(N2CCOCC(C3CC3)C2)C(=O)NCC(=C)C)noc2ccc(Br)cc12 CC1(C)C(CNC(=O)CC2CCC(O)C2)CCN1C(=O)Cc1ccc(O)c(Cl)c1 C1(C(=O)NCC(C)N(C)C(c2ncoc2-c2ccco2)=O)CC12CC(C)(C)C2 C(=O)(C1=C(Cl)CCOC1)NCC1N(C(c2ccc(C#C)cc2)=O)CCC1CC N1(C(c2c(SCC)cccn2)=O)CC2=C(C1)CN(C(C1(C)CCCC1C)=O)C2 N1(C(COCCSC)=O)CCC(C=C)(C(=O)NC2CCCC(C)(C)C2)C1 c1(OCCCC)ccc(C(=O)NCC(CC(C)C)NC(=O)COC)cc1OC(C)=O C(C)(CO)(C(=O)N1CC(N(C)CCO)C1)NC(C(C)=CC=C)=O c1(CCNC(CN(C(C)C(N)=O)C)=O)nc(-c2ncccn2)no1 C1(CNC(C=C(C)Cl)=O)CCN(C(c2cc(C3CCOCC3)on2)=O)C12CCC2 C(=O)(C(C(C)C)OC)N1CC(CC=C)(NC(=O)C(C)C)C1 Cc1nc(O)ccc1C(=O)N(CC(O)CN(C(=O)C(CO)c1ccccc1)C)C c1(OC)ccc(C(N)=O)cc1C(=O)N(C1CN(C(C2CCN(OC)CC2)=O)C1)C C1(C(=O)NC2CN(C(CCOC)=O)CC2C(F)(F)F)CC(c2cnn(C)c2)=NO1 C(=O)(C#CC1CCOCC1)NCC(N(C)C(c1scc(F)c1Cl)=O)C1CC1 N1(C(c2c(CC)noc2)=O)CC2CC(NC(c3cnn(C(C)C)c3C)=O)C2C1 C1(C(=O)NC(c2ccc(OC(C)C)cc2)C)CC(C)SC(C)C1.C1CO1 Cc1ncc(C(N2CCC(CNC(c3cc(C(F)F)cs3)=O)C(C)C2)=O)c(C)n1 C(=O)(C(C(=O)OC)C(C)NC(=O)C(=O)NCc1ccc(C(C)=O)cc1)OC C(C(CC(C)C)C(=O)NCC(C)CC(=O)N1CC(c2ccccc2)C1)OC Nc1ccc(Cl)c(C(=O)NC(CNC(=O)C=CBr)CC(F)(F)F)c1 n1(CC)cc(C(=O)NC2(CN(C)C(c3cscc3OC)=O)CC2)c(C)n1 CCC(C)CCCC(=O)N(CCCNC(C1CC2CCCC(C1)C2)=O)C1CC1 N1(C(c2ncn(CC)c2)=O)CC(F)(F)CC1CCNC(C1COCC(C)(C)O1)=O S(=O)(=O)(c1cnc(NCC(O)CF)c(Cl)c1)N(CC(C)C)CCCN(C)C(C)C CCS(=O)(=O)c1cccnc1CNC(=O)C(C)NC(C1CCC1)=O C1(NC(c2cc(C)c(O)cc2)=O)COC2C(NC(C3COC(=O)N3)=O)COC12 N1(C(c2c(CC)ncnc2)=O)CCN(C)CC1C(N1CC2CC1(CO)C2)=O Cc1cc(CCC(N2CC(c3cn(CC(C)(C)C)nn3)C(C)C2)=O)c(C)s1 C1(C(=O)NCC(N(C)C(c2cc(Cl)c(Cl)s2)=O)C2CC2)CCN2CCOCC12 c1(OC)ncc(Cl)cc1C(=O)NC(c1ccc(Br)nc1)(C)C N1(C(c2ncnn2CC(F)F)C(=O)NCCOCC)CCC(C)(CO)C1 C1(C(N(CC(C)N(C(CC(C)C)=O)C)C)=O)CCC(F)CC1 N1(C(CSCC(C)C)=O)CCC(C(C)CNC(=O)CN2CC=CC2)CC1 C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)N1CC(NC(C=C(C)C)=O)C(C2CC2)C1 c1(C(=O)NC(CNC(c2n(CCC)ncc2)=O)(C)C)cn2nc(C)cc2[nH]c1=O C1(CC)(NC(=O)C=CS(C)=O)CCCN(C(=O)C(c2cncc(F)c2)(C)C)C1 C1(C=O)CCCCC1O.C(C(=O)N(CC(O)CO)C)(C1CC1)OC c1(NC(c2cncc(NC(c3cncc(O)c3)=O)c2)=O)cc(Br)c(O)c(Br)c1 c1(NC(CCC2N(C(c3cc(C)on3)=O)CCC2)=O)cccc(Cl)c1F Cc1cncc(CNC(=O)NC2CCCN(C(=O)OC(C)(C)C)CC2)c1C N1(C(C2(CC=C)CCOC2)=O)C2CCC(C(=O)NCc3ccc(C)o3)C1CC2 CCCCCC(CC)C(=O)NCC(C(=O)NCCOC1CC1)C(C)C CC#CCCCC(=O)NC12CCN(C(=O)COc3ccccc3Cl)CC1C2 N1(C(c2nc(CCC)oc2)=O)CCC(NC(c2cc(C)c(C)[nH]2)=O)C(F)C1 N1(C(CN(C(=O)CCc2nccs2)C)=O)CCN(C(=O)CC(F)(F)F)CC1 N1(C(C=CCN(C)CC)=O)C2CCC1C1CC1(NC(=O)CCc1ccccc1)C2 C#Cc1cccc(C(N2CCCC(N(C(=O)C3=CCCC3C)CCF)C2)=O)c1C CCC(CC(=O)NC(c1cnc[nH]1)C)N(C)C(c1ccc(NC)cc1)=O N1(C(C(C)CNC(C2CCCC2)=O)=O)CC(=O)NC(=O)C1C Cc1nn(C)c(NC(C23CC2CN(C(c2ccsc2)=O)C3)=O)c1C(N)=O N1(C(CCCC)=O)CCCN(CCNC(c2cnnc(O)c2)=O)CC1 CCC(C(=O)N(C)CC1CN(C(C2CC23CC3)=O)C1)c1cccnc1 N1(C(c2c(C#N)ccs2)=O)CC2(CCCC2)C1C(=O)NCC(=O)NC(N)=O c1(NC(=O)NC(C)CC2CCCCN2C)cc(Cl)ccc1Cl.C12C=CCN1C2=O S(=O)(=O)(c1c[nH]c(C(=O)NC(C)C)c1)C(N1CC(=O)NC(C)C1)=O C1(CN(C(=O)C(C)NC(CNC(=O)OCC=C)=O)C2(CC)CC2)CCCC1.SC CCCC(C(O)C(=O)N1CCC(F)(C#N)C1)NC(=O)CC(C)CC N1(CCC(C)SC)CCCC(C(=O)NN2CCC(C(F)(F)F)CC2)CC1 C1(C)(NC(CNS(CCOCC)(=O)=O)=O)CCCN(C(c2[nH]cnc2C)=O)C1 c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ncsc1S(N)(=O)=O OC1CCC2(CCCN(Cc3ccc(Br)nc3)C2)CC1 Cc1c(Cl)ccc(Cl)c1NC(=O)CN1CCN(C(=O)C(=O)C2CC2)CC1=O c1(NCC(CC)(C)CC)cc(Br)ccc1S(=O)(=O)N1CCn2nc(C)cc2C1 N1(C(CC=C=C)=O)CC(NC(c2cc(O)cc(Cl)c2)=O)C2CC2C1 C(c1ccnn1C)=CC(=O)N(C)CC1CCN(C(COCC(=O)NC)=O)C1 c1(C(N2CC(NC(CCCCCSC)=O)C(C)C2)=O)cc(F)cc2cnccc12 C#Cc1cc(C(=O)NC(CC(C)CC)C(=O)NC2CCC3(CC2)N=N3)ccc1C C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Br)n2)=O)CC12CCOC2 C(=O)(C1=C(C)CCC1)N1CC(C(=O)NCC(C(CC)C)C)OCC1 C12(NC(=O)Cc3ccc(Cl)cc3Br)CCC(CN(C(=O)CC3CCC3)C1)C2 CC(C)CCCCC(=O)N1CC2CCC(C1)N2C(=O)Cn1ncn(C)c1=O Cc1cnc(N2CC3(CCN(C(=O)Cc4cc(C)on4)C3)C2)c([N+](=O)[O-])c1 N1(C(c2cc(CC)no2)=O)CCC(C2CC2NC(=O)C2=C(Cl)CC2)CC1 C1(NC(c2n(CCC)ccc2)=O)CCCCCN(C(C2CCCNS2(=O)=O)=O)C1 c1(C(=O)NC(C)CNC(c2ccccc2)=O)cc(-n2cnnc2)ccc1F C(=O)(C(CC)CC)NC1C(C(N(CCC#C)CCO)=O)CC1 Cc1cnc2n1CCC(C(=O)NCC1(O)CCN(C(c3cc(=O)cc[nH]3)=O)C1)C2 C1(NC(CCC(=O)NCC)=O)CC1C1CCCN(C(c2c[nH]nc2C)=O)C1 C12(NC(C(C)n3cccn3)=O)CC(CNC(C3CC3c3cnn(C)c3)=O)(C1)C2 N1(C(CC2N(C)CCC2)=O)CCC2(CC(NC(=O)CCCc3cccnc3)C2)C1 C1(C(C)(C)C)(Cc2ccccc2)CCN(CCOCC(N)=O)C1 C12(CN(C3CCN(c4ncc(C(F)(F)F)cc4Cl)C3)CCC)CC=CC(C1)OC2 Cc1cnc(C(=O)NCC2CCC(NC(C3(C(F)F)CCCO3)=O)C2)[nH]1 N1(C(CSCCCC)=O)CC(N(C(=O)CCC2C(=O)ON=C2C)C)C2(CC2)C1 CC(C)C1=NOC(C(=O)N(C)CCNC(=O)C(C(C)(C)C)OC(C)(C)C)C1 N1(C(c2n(C)ncc2)=O)CC(NC(=O)Cc2csc(-c3ccco3)n2)C(F)C1 C#CC1(C(N2CCC(OCCCCC)C2)=O)CCCC1 C1(CNC(c2n(C(CC)C)nnn2)c2ccn(CC)n2)CCC(C)(C)CC1 c1(OC(C)C(=O)NC(C)CN(C(=O)CCC2CCCO2)C)cccc(C(N)=O)c1 Cc1cc(F)cc([N+](=O)[O-])c1NC(c1nc(NC(C2CCCS2)=O)cn1C)=O CN(CCCC(=O)N1CCC(CCNC(=O)C#CC2CCOC2)C1)N=O c1(C(=O)NC)cccc(C(N2CCC(O)(CNC(=O)CCC3CCOC3)C2)=O)c1 C(N=c1nc(O)c(Br)c[nH]1)C1(O)CCCN(C(c2ccc(C)nc2O)=O)C1 c1(ONC(n2cc(CN3CCCC3c3nc[nH]n3)nn2)=O)cccc(F)c1 CC(C)(CCNC(=O)Cc1csnn1)C(=O)Nc1ccc(O)c(F)c1 c1(CNC(=O)CC(Cl)Cl)cccc(C(N2CC(c3nc(=O)o[nH]3)C2)=O)n1 c1(C(N2CCC(C)C(NC(C3(CC4CC4)CCC3)=O)C2)=O)ccc(N)c(F)c1F Cc1nn(CC(=O)NC(CO)C(C)NC(C2(C)CNC(=O)C2)=O)c(C)c1Cl Cc1cc(NCC(C2CC2)NC(=O)CC(O)C(C)C)c(Br)cc1[N+](=O)[O-] CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(C1SCCS1)=O CC(=O)CCCC(=O)NC1C2CC3C1C3C2C(=O)NCC1(C)CCC1 N1(C(C(C)N(C)C)=O)CC2CC1CC2CNC(=O)CCCc1csc(=N)[nH]1 c1(CC(CNC(=O)CC2CCCNCC2)OC)cccc(Cl)c1 Cc1n[nH]c(C)c1CN(C(C)C)Cc1ccccc1-c1ccccc1 N1(C(c2cc(COC)cn2C)=O)CCC2CCN(C(c3cccnc3N)=O)CC12 C1(C(=O)NCC2C(CNC(CC3(COC)CC3)=O)C2)CC2CC2C1 CS(=O)(=O)c1ccc(CNC(C2CCN(C(=O)CC(O)C3CC3)CC2O)=O)cc1 C1(NC(CCC(=C)C)=O)CCC(C)(CNC(=O)CCc2cncc(OC)c2)CC1 C12(C(N(CC(C)NC(c3ccccc3CC#N)=O)C)=O)CC(C1)C(C)(C)O2 c1(OC)cc(C)ccc1C(=O)NC1CCN(C(=O)CCCC(C)=O)C1C c1(C(=O)NCC2CCCN(C(CC(CC)SC)=O)C2)cccn2c(CO)nnc12 c1(C(=O)NCC(=O)NC(C)CNC(c2coc(Cl)n2)=O)ccccc1CC#N C1(CNC(CCC)=O)CCN(C(=O)C(C(C)(C)C)N2CCNC2=O)CC1O c1(C(=O)NC(C(C)C)CCNC(c2nc(Cl)c(Cl)s2)=O)ccc(O)c(Cl)c1 C1(C(N(C)CCOCCNC(C2CCCC(=O)N2)=O)=O)Cc2ccccc2O1 Cc1nn[nH]c1C(=O)N(Cc1cc[nH]n1)CC1CC1 c1(C(=O)NC(C(C)C)C)cc(CNC(=O)C=Cc2cncs2)on1 N1(C(c2nc(OC)oc2)=O)CCCC12CCN(C(=O)CSc1nncn1C1CC1)C2 N1(C(CNC(CC)=O)=O)CC(NC(C2CS(=O)(=O)CC(=O)N2)=O)CC2(CC2)C1 N1(C(C(CC)C(C)O)=O)CC2CC(NC(=O)C(F)CC3CC3)CC2C1 Cc1cnc(C(N2CCOCC2CC(=O)N(C2CC(F)(F)C2)C)=O)c(C)c1 c1(C(=O)NCC2(CCNC(C3C(C)(C(C)C)C3)=O)CC2)ccc(C(C)(C)C)[nH]1 C1(N(C)C)CCCC1OC(c1cc(-c2ccccc2)on1)=O C1(CNC(=O)Cn2cccn2)C(C2CC2)CCN1C(c1ncc(C(F)(F)F)s1)=O N12CCC(C3CC3)C1C2=O.C(=O)(CCC(=O)NC)NCCC.N12CCC1C2=O c1(C(N(CC(C)(C)NC(=O)CCc2ccncc2)C)=O)ccc(C#N)cc1F N1(C(c2c(NC(c3c(Br)ccc(F)c3F)=O)ccs2)=O)CCC2(CCOCC2)C1 c1(C(N2CC(F)(C(=O)NC(C3CCOC3)C)C2)=O)cc(C#N)ccc1Br N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(N(C)C(c2ccncc2Br)=O)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2(C=C(C(=O)N3CC(NC(N)=O)C3)C2)C1 N1(C(c2c(C)n(C3CC3)cc2)=O)CC2CCN(C(=O)C3=C(Cl)CC3)CC12 CN1CC(C(N2CC(C3CN(C(C4CCC5(CC5)C4)=O)CCO3)C2)=O)CCC1=O c1(C(N(CCNC(COC2(C)CCC2)=O)CCOC)=O)cc(F)cnc1O c1(CSC)c(C(=O)NC2CC2NC(c2ccccc2C2CCCC2)=O)cnn1C S(=O)(=O)(c1cccc(F)c1)NCC(N1CCN(C(c2ncn(C)n2)=O)C2C1C2)=O N1(CC(=O)NC(CCCCC)C)CC2(CC(NC(=O)CCn3cncn3)CO2)C1 C(=O)(C#CC1CCCC1)N1C(C2(NC(CSC)=O)CC2)CCC1 C(=O)(C1CCc2c(Br)cccc21)NC(c1cccnc1)C(C)C CC(C)C(CO)CCNC(=O)CC1CC(C)N(C(=O)COC2CCCC2)C1 N1(C(=O)Cc2ccc(O)c(O)c2)CCC2CN(c3ncnc4cc[nH]c34)CCC12 C12(C(=O)NCC3(CCNC(C4CCC(=O)NC4)=O)CC3)CCC(CC1=O)C2 C1(C)(C(=O)NCC(C)(C)NC(C(CC)n2ccnc2)=O)CCC(=O)N(C)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC=CC(NC(C2(C)CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CC(F)(CNC(C2CC(C)C2)=O)C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCCN(C(C2CC(CF)C2)=O)C(C)C1 c1(CNC(c2cc(CNC(c3c(OCC)ccs3)=O)on2)=O)cc2nc[nH]c2cn1 c1(CCNC(C(C2CCN(C(c3c(COC)ncs3)=O)C2)C)=O)c(C)noc1C c1(C(N2C(C(=O)NCC3(OC)CCC3)COCC2)=O)cc(C)c2ccccc2n1 C1(C(=O)NCC(C)CN(C(=O)Cn2ncn(C)c2=O)C)CCC2(CCC2)CC1 C(=O)(C(C)CC(N)=O)N1CCC(CN(C(C(=O)NC)C)C)C1 C1(C(=O)NCC(O)CO)CSCCN1Cc1ccc(Cl)o1 CC1(C)COC(CC(=O)N(CCCNC(=O)CC2(CO)CC2)CCO)C1 N1(C(c2c(COC)noc2)=O)CC(C)C(NC(c2cc(O)ccc2F)=O)C(C)C1 C(=O)(C(C)(C)C(O)C(C)C)NC1(CC=C)CCN(C(=O)C(C)CS(C)=O)CC1 c1(C(C)C)cc(F)ccc1NC(=O)NC(C)CN=[N+]=[N-] CC(C)C(CCN(C)C(c1nccnc1N)=O)NC(=O)C(c1cccn1C)=O N#Cc1cccc(C(N2CC3C(NC(=O)CC45COCC(C4)C5)C3C2)=O)c1 Cc1coc2c(C(N3CCCC(CCNC(=O)C(C)CC(F)F)C3)=O)cccc12 C1(C(N(CCN(C(=O)CC2OCCC2C)C(C)C)C)=O)OCCC1C N1(C(C(C)(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 CCC(CC(=O)N1CCCC1(C(=O)NC1CC(C)(O)C1)CC)CC(C)C c1(C(=O)NC(CNC(C2ON=C(C)C2)=O)(C)C)cccnc1CN1CCOCC1 c1(C(N2C(CCNC(C3CC3C3CC3)=O)COCC2)=O)cccn(C2CC2)c1=O N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1CC(F)(F)F C(=O)(C(C)N1CC(C)C1)N(CCCNC(C=C(CC)C)=O)CCO C12(CNC(C3CCN3C3CCCCC3c3ccc(F)cc3)=O)C(=O)C3CC1C2C3 C1(O)(C(=O)NCC(C)NC(=O)Cn2cnnc2O)CC(F)(F)C1 C1(NC(C=C(CCC)C)=O)CC2(C1)CC2NC(c1ccc(C2CC2)nc1)=O C12(CC(=O)NCCCc3ncco3)CCC1CN(C(=O)C(C1CCOCC1)O)C2 N1(C(c2cc(CC)c(C)s2)=O)CCC(O)(CNC(=O)C(F)CC2CC2)CC1 c1(C(=O)NCC(C)(C)NC(c2ccncc2)=O)csc(-c2ncccn2)n1 CC1CN(CCN2CC(=O)N(CC3CCC3)C2=O)CC(C)O1 C(=O)(C(C(C)C)NC(C)=O)NCC(CCC)NC(c1ccsc1)=O C(=O)(CCC(C)(C)NC(=O)C=Cc1ccco1)N1C(C)CC1CO N1(C(Cc2c(C)noc2)=O)CCN(CCCCCNC(=O)C(Cl)=CCl)CC1 c1(C(=O)NCCNC(c2cc(C(CC)C)no2)=O)cc(S(N)(=O)=O)c(C)o1 C1(CCC)CN(C(c2cncc(NC)c2)=O)CCN1C(=O)CC1CC(C)(C)CO1 c1(CNC(C2(CC)CCCC2)c2nnnn2C2CC2)ccc(C(F)(F)F)nc1C c1(C(C)C)ccc(CC(=O)NCC2CCC(NC(=O)CC(F)(F)F)C2)cc1 c1(C(=O)NCC2CC(O)C(O)C2)cc([N+](=O)[O-])n[nH]1.C12(C(N)=O)CN(C1)C2 c1(N2C(CCNC(C(C)(C)C)=O)CCCC2)ncnc2c(Br)c[nH]c12 CC(C)CC(C)CNC(=O)NC(C(F)(F)F)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)cnc(O)nc1O Cc1ccc(C(=O)NCC2CC(NC(c3ccc(O)nc3Cl)=O)C2(C)C)c(F)c1 CN1CCC(C)(C(N2CCC(C(N3CC(C)(CF)C3)=O)C2)=O)C1 CC1CCC(CC(=O)NCC(O)CN(C(=O)C(F)=CCCF)C)OC1 N1(C(C2(SC)CC(=O)C2)=O)CCCC(C(=O)NCC2(O)CC(C)(C)C2)C1 C1(CC(=O)NC)CN(C(=O)CCc2cc[nH]n2)CCN1C(=O)C=C(C)C O=C(C1=COCCC1)NC(Cc1cc[nH]n1)C(=O)NCc1nncs1 N1(CCCCCC)CCC(CNc2cn(C(C)(C)C)nc2Br)C(F)(F)C1 CC1(C#N)CCN(C(=O)C(CC2CCCC2)NC(C2C3CCC(F)C23)=O)C1 N1(C(C2(C#N)CCOC2)=O)C2CCCC1CN(C(C1CCn3nnnc3C1)=O)C2 C=CC(CC)C(=O)N(C1(C(N2CC(N3CC(O)C3)C2)=O)CCC1)C1CC1 Cc1nn(CC(N2CC(F)(CNC(=O)C(N3CCOC3=O)C)C2)=O)c(=O)o1 C1(CNC(c2n(CC)nnn2)c2ccc(-c3cc[nH]n3)o2)CC2(C1)CC(F)(F)C2 n1(CC)cnc2nc(N3CC4COCC(C4)C3)nc(N(CCCC(F)(F)F)C)c12 C1(NC(C(CC)C)=O)CCN(C(=O)COc2ccc(F)c(Br)c2)C12CC2 C1(CN(C(C2CC(C3CC3)C2)=O)CC)CCN(C(=O)CCC2=NC=CSO2)CC1 c1(C(=O)NCC2(C)N(C(CN3CC(C)(C)C3)=O)CCC2)ccc2nc[nH]c2c1 c1(OC)ccc(-c2noc(C3(C(=O)NC4CCCCC4C)CC3)n2)cc1OC c1(C(N2CCN(C3CC(C)(C)OC3=O)CC2)=O)cnc2c(c1)CCCO2 C1(CNC(C2C(C#N)C2)=O)CC(O)CN1C(c1cc(-c2ccc(Cl)s2)on1)=O Cc1ncc(Br)cc1NC(=O)NC1CCC(Cc2ccccc2)CC1 c1(C(=O)NCC2C(NC(C(c3cscn3)N(C)C)=O)CC2)ccc2nonc2c1 C(=O)(C(C1=C(C)CCCC1(C)C)N1CCCC1C1CCCCO1)NCC C1(CNC(C2CCC(COC)C2)=O)CC2(C1)CN(C(=O)C=C(C)Cl)C2 N1(CC(=O)N(CCC)CCC)CC(NC(c2c(C)cccc2F)=O)CCC1C c1ccc(NC2(c3nnnn3CC3CCOCC3)CSC2)cc1 N1(C(C=CS(C)(=O)=O)=O)CC(NC(=O)Cc2ccc(Cl)s2)CC2(CC2)C1 CC(C)(C(=O)N1CCC(C(F)C(=O)NCCC(C)(C)N2CCCC2)C1)C1CCC1 N1(C(CC=CC=C)=O)CC(NC(C2CC23CCOC(C)C3)=O)C2CCCCC12 C1(S(N)(=O)=O)(C(=O)NC2CC(C)(NC(CSc3n(C(C)(C)C)ccn3)=O)C2)CC1 N1(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CCO)CC1 c1(C(N2CC3CCC(O)CC3C2)C(=O)NC(C)(C)C)ccc2ccccc2c1 N1(C(C(CCCCC)O)=O)CCn2ncc(CNC(=O)CC(C)C(F)F)c2C1 c1(CC(=O)NCC2C(NC(C3(C)ON=C(C)C3)=O)COC2)cccc2nsnc12 c1(C(N2CC(OCCNC(=O)CCCCC3CC3)C2)=O)cc[nH]c2nccc1-2 C1(CC(=O)N(CCOCCNC(C=CC=CC)=O)C)C=CC(OC)C1 N1(C(CCC(C)(C)SC)=O)CC(C)N(C(=O)CC(C)C2CC2)CC1C N1(C(c2cc(CC)oc2C)=O)CC2CCN(C(C3CC34CCOC4)=O)CCC2C1 c1(C(=O)NC2(CC=C)CCN(C(C3CCCC(CF)C3)=O)C2)cc(O)nc(C)n1 CCC(CC)C(C(=O)N1CC(C)(OCC(=O)NCC=CC(C)(C)C)C1)OC CCCCC(O)CC(=O)NC1CCCC1CNC(c1ccc(CO)c(F)c1)=O C1(CC(=O)NCC2CCCN(C(C3(CNC(C)=O)CC3)=O)C2)CCCC(C)(C)O1 c1(C(=O)NCc2nc(C)c(C(=O)N(CCCN(C)C)C)o2)cn(C)c(=O)cn1 N1(C(CC2ON=C(C)C2)=O)CC2(CCN(C(=O)COc3ccc(C)cc3)CC2)C1 CCCC(O)(CCC)CC(=O)NC(C)CC(C)NC(c1ccn(C(C)C)n1)=O N1(C(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)C(N)=O)CCC1 C=C=CCCC(=O)NCC(C)(C)CNC(c1nonc1CC)=O c1(OC)ccc(C)nc1NC(C1CCN(C(C2CCC3(CC2)CC3)=O)CC1O)=O C(=O)(C1CCCc2scnc21)N1CCOCC(CNC(C=CSC)=O)C1 C(CC(=O)Nn1cncn1)N(C(C1(C)CCC1)=O)C(=O)OC(C)(C)C c1(C(N(CCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)scc(C)c1Cl Cc1ccc(C=CC(=O)NC(CNC(=O)CCC(=O)c2ccc(Cl)cn2)CO)s1 C1(C(N2CC(NC(c3coc(C(N)=O)c3)=O)C(O)C2)=O)CCOCC12CCCCC2 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2C1CCCN2C(=O)CC1CC1 C(=O)(C(C)CNC(=O)C(Cn1cccn1)NC(=O)CCC1CC(C)C1)OC C1(C(=O)NCC(CNC(c2c[nH]nc2-c2ccco2)=O)O)CCCCC12CC2 C#Cc1c[nH]nc1C(=O)NC1(C(N2CC(C#CC)C2)=O)CCSC1 c1(CC2(C(=O)NC(CC(C)=O)C)CCOC2)ccc(OC)cc1F c1(C(=O)NC(C2CN(C(C3CCC3(C)C)=O)CCO2)C)cccc2cncn12 N1(SCCNCCCC(C(=O)OCC)O)C(=O)NC(C)(C)C1=O Cc1cc(Cl)cc(C(C)NCC(C(C)(F)F)c2ccccc2)c1O C#CC1CCCCN(C(=O)NC(Cc2ccc(C)cc2)CC)C1 Cc1cccc(Br)c1C(=O)NC1CCOC(C(N2CC(Cc3ccco3)C2)=O)C1 C(=O)(CN=c1cc[nH]cc1)NC1(C)CCCN(C(=O)CCOCC2CCC2)C1 N1(C(C2(C(C)NC(=O)CC3CCC3)CC2)=O)CCN(C)C(C2CC2)C1 Cc1ccc(F)nc1NC(=O)Cn1cc(CC2(CN(C)C)CCC2)nn1 C(=O)(C(C)CCC(C)(C)C)NC(C)CCNC(c1nnn(C)c1N)=O Cc1cnc(C(=O)NCc2ccnc(C(=O)NC3(C(F)F)CCCC3)c2)cn1 c1(C(=O)NC(C)(C)CNC(=O)C=Cc2cnc[nH]2)c[nH]c2ccncc12 C(=O)(C(CNC(=O)CNc1cncn1C)CCC)NC(C#C)C(C)OC C1(CNC(C(c2ccc(F)cc2)C)=O)CN(c2ccnc(Cl)n2)CC(C)(C)O1 Cc1ccc(C(=O)C(=O)NC(C)CC(C)NC(=O)C(F)n2cccn2)cc1 c1(C(N(C(C)CCNC(c2ccc(Cl)nc2O)=O)C)=O)ccc2oc(O)nc2n1 N1(C(C(C)CF)=O)CCC2(CC1)CC2NC(c1ccc(C(C)(C)C)cn1)=O c1(C(N(CC(C)NC(C2CC2C2CC2)=O)C)=O)cc2ccc(F)cc2o1 C1(O)(CNC(C(C)(Cl)Cl)=O)CCCN(C(=O)C(O)c2ccco2)C1 C1(CC(=O)NCCCOCCNC(c2c(CC)nc[nH]2)=O)CC2CCC1O2 C=C(C)C(C)(C)C(=O)NC(CNC(C1C2CCC1(c1nccs1)C2)=O)C(C)C c1(C(N2CC(C)C(CC(=O)Nc3nc(O)[nH]c(=O)n3)C2)=O)cn(C)c(=O)nc1O N1(C(C(C=C)O)=O)CCCC(CCC)(NC(=O)Cc2ccc(CCC)cc2)C1 C(CC1=CCN(C(c2csc(-c3cccs3)n2)=O)CC1)NC(C(C)CC(N)=O)=O c1(OC)cc(C(=O)N(C2CN(C(=O)C(F)(F)COC)C2)C)cnc1O c12ccc(F)c(F)c1C(=O)N1CCC1C(=O)N2.N1(CC)CCN(CCCO)CC1 c1(NCC2C(C)N(C(=O)OC(C)(C)C)CCC2)ncc(Br)cc1C#N CC(C)C(C(=O)NCC(C)(C)OCCNC(=O)CCc1nc(=N)[nH][nH]1)C1CCC1 C1(C(N2CC3(CC(NC(C4OCCC(=O)C4)=O)C3)C2)=O)CCc2nccn2C1 N1(C(=O)COc2cccc(F)c2)CC2CCN(C(=O)COC3CCOCC3)C2C1 C1(CC)(NC(C2COC3(CCC3)C2)=O)CCCN(C(=O)CCNC(C)=O)C1 Cc1ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=COCC2)cc1C CCC(O)C(C)(C)C(=O)N1CCN(CC2(NC(=O)C(C)c3ccco3)CC2)CC1 c1(CCC(=O)NC(C)CCNC(=O)CC2CSC2)ccc2c(c1)OCO2 N1(C(=O)C=Cc2cnccn2)CC2(C(N3CC(O)(C4CC4)C3)=O)CC1CCO2 C(c1ccccc1C#N)=CC(N1C2CC(CNC(C(OC)OC)=O)(OC2)C1)=O c1(OC)cc(OC)c(C(c2nnnn2CC(F)F)NCc2sccc2Cl)c(C)c1 c1(CC)cccc(C)c1-n1nc(C(C)CC)nc1-c1cccc(-c2ccoc2)c1 c1(C(N(CC(CNC(C(c2cccnc2)OC)=O)O)C)=O)nccnc1N c1(C(=O)NC(CN(C(=O)CCC2CCOCC2)CC)C)coc2c1COC2 c1(C(N2C(CC)CN(C(=O)C(C)CC#N)CC2)=O)ccc2cnc(C)n2c1 S(=O)(=O)(c1cnc(NC2(CC(C)(C)C)CC2)cc1C)NC1CCN(CC(C)C)C1 c1(CC(N2C(CNC(CC(C)C(F)F)=O)C(C)CC2)=O)ccc2c(c1)CCCO2 N1(C(C(CCC)OCC)=O)CC2CC(NC(c3cccc(CO)c3C)=O)C(C2)C1 C1(C(=O)NCC2CCN(C(C=CC(CC)=CC)=O)CC2)CC2(CCC2OC)C1 C1(C(=O)NCC2C(NC(c3cc4cscc4s3)=O)C2)COc2ccc(F)cc2C1 C1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)nc2)CC2CCCCN2C1 N1(C(CC(=C)C)=O)Cc2ccnn2CC(NC(c2nc(C(C)(F)F)cs2)=O)C1 C1(NC(C=CC2N(C(c3cccc(CC)n3)=O)CCC2)=O)CCCCCC1CO S(=O)(=O)(c1cnc2ccsc2c1)NC(c1n(C)nc2c1CS(=O)(=O)CC2)=O C1(NC(C(C)SC(C)C)=O)C=CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 c1(NC(C(CN(C2CN(C(c3ccccc3)=O)C2)C)(C)C)=O)cnn(C)c1C#N c1(N2CCCC(CCC)CC2)nc(=N)[nH]c(=NC2CCC(C)(C)C2)[nH]1 CCCC(C(=O)NCC(CC(C)C)NC(=O)C=CCN1CCOCC1)N(C)C C1(C(C)NC(c2ccc(CSC)o2)=O)CCN(C(=O)CC2CCCN2C)CC1 N1(C(C2(CC#C)CCOC2)=O)CCCCC1CCNC(c1cncnc1)=O CCC(C)CC(C)(c1nnnn1C1COC1)NCc1ccc(CCO)cc1 C(=O)(C(F)C(C)(C)O)N1CC(CNC(C(c2ccnn2C)C)=O)OCC1 N1(C(CN(CCOC)C)=O)CCCC(CNC(=O)CC2CCC(OC)CC2)CC1 N1(C(c2cnc(CC)o2)=O)CCN(C(=O)CC(F)(F)F)CC1C1CCC1 Cc1ccc2cc(C(N3CCNCC3c3ccncc3)=O)nn2c1 Cc1cnc(C(=O)NCC(CNC(c2cc(=O)cc[nH]2)=O)CO)c(F)c1 N1(C(C2CCC(C)N(C(=O)CSC(F)F)C2)=O)CCCC2OCCC2C1 N1(C(C2N(C(C(CC)C)=O)CC2)=O)CCn2nc(C)cc2C1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC(C)C)CNC(c1n[nH]cc1Br)=O c1(CC)occ(C)c1C(=O)NCC(C)NC(C1CCOC(C)C1)=O c1(CC(=O)NCCCC2CCCN2C(=O)C(C2CC2)C2CC2)cccc(Br)c1 Cc1c(C(=O)NC(C)C(CO)NC(C2CC3CCC2C3)=O)sc2nccn12 c1(-c2nc(C(C)C)nn2C2CCSCC2)cn2cc[nH]c(=O)c2n1 Cc1cc2c(cc1C)OC(C(=O)NC(CC1CCCCC1)CC(=O)O)C2 CC1(C)C(NC(c2ccoc2CN2CCCC2)=O)C2CCCOC12 CCCCC(C(=O)NC(C)C(C)N(C(=O)C=CC1CCC1)CC)ON=C(C)C C1(C(N2C(CNC(c3ccnn(C)c3=O)=O)CCC2)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC(C)(CO)NC(C2N(CCC)CCC2)=O)c(C)cnnc1O N1(C(c2n(C)nc(C)c2Cl)=O)CCCC(C2CCN(C(=O)Cc3nc[nH]n3)C2)C1 c1(NC(C(N2CCCCC2CO)CC)=O)ccccc1C(C)C C12(C(=O)NCCCC(C)O)CC(CN(C(C3(C)COC3)=O)C1)C2 c1(N2CCC(NC(C3C(OC)CCC3)=O)C(O)C2)ncnc2c1nnn2C(C)C S(=O)(=O)(c1ccc(NC2COC(C)(C)OC2)c(F)c1)NCC1C(C)CCC1 c1(OC)c(CC(=O)NCC2CCN2C(=O)C2CC2)cccc1Br N1(CCNC(c2cc(CNC(C3CC(=C4CC4)C3)=O)on2)=O)CCCCCC1 CC(C)C#CC(=O)NC1COCC1NC(c1cccnc1N(C)C)=O c1(SC(C(=O)NCCN(C(=O)CCOCC2CC2)CCOC)C)ccc(F)cc1 c1(C(N2CCC(NC(C(CC)N(C)C)=O)CC2)=O)ccc(Cl)c2c1OCCO2 N1(C(C2(CCNC(C=CCC)=O)CC2)=O)CCS(=O)C(C)C1 C1(OC)(CNC(C2CCCN2C(c2cc(Cl)ns2)=O)=O)CCC(C)C1 C(=O)(C1SCCc2sccc21)N1CCN(C(C2CC3(CC3)C2)=O)CC(C)(F)C1 N1(C(c2nnn(CC)c2C)=O)CCc2sc(CNC(=O)CCCC(C)C)nc2C1 C1(NC(c2[nH]nnc2C2CC2)=O)CN(C(c2ccccc2O)=O)CCC1CO C(=O)(C(CC)c1cccnc1)N1CC(C(C)NC(CN(C2CC2)CC)=O)C1 c1(N(C(=O)CCCn2ccnc2)CC2(CN)CC23CCC3)nc2ccccc2o1 Cc1cc(O)ncc1NC(=O)C(CNC(c1cccc(O)n1)=O)CC1CC1 Cc1c(C(=O)NCCOCC(=O)N(C(C)C)CC2CCCCO2)cncc1F CC(C)(C)CC(O)C(=O)NC1CCCN(C(=O)Cc2ccc3c(c2)COC3)CC1 c1(C(c2nnnn2CCCF)NCC2(C)COCCO2)cc(S(C)(=O)=O)co1 n1(CC)cc(Cl)c(C(=O)NCCNC(C2CN(C)C2)=O)n1 C1(CNC(c2n(C)cc(Cl)c2)=O)CN(C(=O)C(C)(C)c2cnsc2)CCC1(F)F C(=O)(CCC(F)(F)CN=[N+]=[N-])N1C(C)(C)CC(NC(=O)COCC(F)(F)F)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(C(C)(C)OC(C)=O)=O)(C)C CC(C)(C)C(C(=O)N1CC(CO)(NC(=O)CNC(C2CCCCC2)=O)C1)C1CC1 N1(C(C(c2ccc(C)cc2)F)=O)CCC(NC(=O)CO)C12CC2 C(=O)(CC(N(C(C1CC1(F)Cl)=O)C1CC1)C1CC1)NC1(C(N)=O)CCC1 C1(NC(CN2CCC(OC)C2)=O)CCN(C(=O)Cn2nccc2C)CC1F c1(OC)ncc(Cl)cc1C(=O)NCCC1CCN(C(=O)C(C)(C)N(C)C)CC1 N1(C(c2scc(C)c2)=O)CCC2CCN(C(=O)CS(=O)(=O)NC(C)(C)C)C2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(C2CC(F)(CO)C2)=O)CC1C C(=O)(CC(CC)N(C(=O)CCN1CCOC1=O)C)N(CC(CCC)O)C c12ccc(C)c(c1)C(=O)N2.CC(=O)CCC(=O)NC1CC(CC(=O)N(C)C)C1 N1(C(CCCCCNC(C)=O)=O)CC2CCOC2(CNC(c2ccncc2)=O)C1 N1(C(c2c(-c3cn(C)nc3)onc2)=O)CCCC1C1CCCN1C(=O)COC1CC1 C1(F)(C(=O)NCC2(O)CC(C(=O)NCC3(OCC)CCC3)C2)CCCCCC1 CCCC(C(=O)OC)C(=O)N1CC(OC)CC1C(=O)Nc1ccc(CC)nc1 Cc1cnc(C(=O)NC2CCC(NC(=O)Cn3nc(C)oc3=O)C2)cn1 S(=O)(=O)(c1ccccc1C(=O)NC(C)CNC(=O)C(C)N)N(CCC)C.C(C)(=O)O N1(CC(=O)NCCC2CC(NC(C(F)OC)=O)C2)CC2CC2C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)Cc2cccc(Cl)c2F)CCCO1 C(=O)(CCS(N)(=O)=O)NC1(CC(=O)NC(c2nnc(C)o2)C)CCCCC1 C=CCC(CC=C)C(=O)N1CCCN(C(=O)Cc2nnc(O)s2)C(C)C1 C(CC(C)C)(C(=O)N1CCOCC(NC(=O)CCCc2cc[nH]n2)C1)OC C(=O)(C1=CCCN(C(=O)CC(CC)C(F)F)C1)N1CCC(OCC=C)CC1 C(=O)(CC(O)CC(C)(C)C)N(C1CCCN(C(c2sc3cc(C)sc3c2)=O)C1)C C1(CNC(CCN(C(C)C)C(c2cccc(=O)o2)=O)=O)CC(O)C12CCC2 C1(C(=O)NC2CC(NC(c3c(C)nn[nH]3)=O)C2)CC(=O)N(c2ccccc2)C1 Fc1ccc(C2CN(CC=CCOc3ccccc3)CCO2)cc1 c1(C(N2CCC(CNC(C3CC(F)(F)CS3)=O)C23CC3)=O)cnc2ccnn2c1 CC1(C(=O)NCC(C)(CO)NC(=O)COc2ccc(C(N)=O)cc2)CC=CCC1 N1(C(CC2(C)CC2)=O)CCC2CCCC12CNC(c1nc[nH]c2ncnc1-2)=O N1(C(c2c(C)oc(C3CC3)n2)=O)CCN(C(c2ccc(O)nc2)=O)C(CO)C1 N1(C(C)=O)CCN(NC(C2CC2NCc2ccccc2I)=O)CC1 C(C(C)C(C)C(=O)N1CCCC1CCNC(=O)C(F)(F)CCn1ccnn1)OC CCC(CC)C(C(=O)NC1CC(C)CN(C(c2ccccc2O)=O)C1)OC C(CCC(C)(C)NC(C1CCCCN1S(C)(=O)=O)=O)NC(Cc1nc(C)sc1)=O C#CC1(NC(C2(C(C)NC(C3CCN(OC)CC3)=O)CC2)=O)CCCOC1 Cc1cc(CCC(=O)NC23COC(CNC(C4CCC(C)C4)=O)(C2)C3)c(C)s1 C1(c2n(CC(=C)C)nnn2)(NC(c2ccccc2Br)CF)CCCSCC1 C1(C(=O)NC(CCC)(C)CC)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 c1(CNC(C=CC(CC)=CC)=O)cc(C(=O)Nc2cccc(C(C)C)c2)ccn1 N1(C(C(CNC(C2CC3(CSC3)C2)=O)O)=O)CCC2(CCC2)CC1 c1(N(S(=O)(=O)CCC2CCCC2)C(=O)Cn2ccnc2)cccc(Cl)c1 C1(NC(=O)CCF)CCCCC1NC(c1csc(C2CCCO2)n1)=O c1(CN(C(=O)C(c2ccccc2)c2cccs2)c2nn[nH]n2)ccccc1I Cc1ccnc(C)c1NCc1nccnc1CC(N1CCCC(COC(C)C)C1)=O Cc1occ(C(F)(F)F)c1CN(N1CCCC1)C=O.CC(F)F N1(C(C2(C)C(C)C2)=O)CCC(C(N2CCC(OCC3CC3)C2)=O)CC1 C1(NC(Cc2cccc(OC)c2)=O)C2CC3CN(C(C4CCCN4C)=O)C1C3C2 C(=O)(C1CCc2cccnc21)N(CCCNC(c1n[nH]c(C)c1O)=O)C1CC1 CCC(C)(CNC(=O)CCc1ncccn1)NC(=O)COC1CCC1 n1(CC(N2CCC(O)(CCNC(CC(C)(C)OC)=O)C2)=O)cnc([N+](=O)[O-])n1 C(=O)(CCCC(C)=O)N1CC(CC=C)(C(=O)NC(C)CC(N)=O)C1 c1(OC)c(CNC(=O)C(N2CCN(C(c3cccs3)=O)CC2)C)c(C)nn1C C(=O)(C1=CCCC(C)(C)C1)NC(C(C)C)(C)CNC(=O)C#CC1(C)COC1 c1(CC2N(C(c3nc(CSC)cs3)C(=O)NCC)CCCC2)ccc(C#N)cc1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)Nc2csnc2C)CC(C)C1 c1(C(=O)NCC(CC)NC(=O)C(c2ccccc2)O)nn(C)cc1[N+](=O)[O-] CC(C)(C)C(=O)NCC(O)C(=O)NCC1CCC(C=O)O1.C(N)=O O=C(C1=CS(=O)CCC1)NCC1CCCC1NC(c1ccnnc1Cl)=O C1(O)(CNC(c2c[nH]nc2-c2ccc(Br)cc2)=O)CCCCCC1 c1(COC)nc(C)c(C(N2CCC(COC)(NC(C3CCCOC3C)=O)C2)=O)s1 c1(C(N2CCCC(NC(C3(F)CC3)=O)C2)=O)ccc(Cl)c(N2CCCC2)n1 CC1CCC(Cl)=C(C(=O)NC2(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)CC2)C1 CC1CCN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)CCSCC(N)=O N1(C(C2C(C)C2)=O)CC(CNC(c2cnn(-c3ccccc3)c2)=O)C(C)C1 c1(CN(C2CCCN(C(c3c(SC)cccc3)=O)C2)C)ccncc1[N+](=O)[O-] C1(NC(c2c(F)ccc(OC)c2)=O)CCCCN(C(=O)CCCC2CC2)CC1 C1(NC(CCC=C)=O)CCCCC12CCCN(C(=O)C(C)n1cnnn1)C2 C=CCCCCCCC(=O)N1CC2(C1)CN(C(=O)CC(CC)C1CCC1)C2 C1(CC=C)(C(=O)NCC2(CC)CCOC2)CCCN1C(=O)CN1CCCNC1=O CC(CC(F)F)C(=O)N1CC=CC1CNC(=O)CCc1ccccn1 c1(OC)ccc(F)c(C(N2CCN(C(c3cc(Br)c(C)s3)=O)C(CO)C2)=O)c1 Cc1ncc(N)cc1C(N1CC=CC1CNC(=O)CCc1cnco1)=O Cc1ccnc2nc(C(=O)NC3CC(C)N(c4nnc(O)s4)C3)nn12 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)N(CCCCO)C2CCCC2)C2(CC2)C1 C1(C(NOC(CC)C)=O)(NC(c2cnsc2)=O)CC(CO)C1 N1(C(C(=O)NC2CCCC(N)C2)=O)CCC(O)(c2cccc(F)c2)CC1 C(C(CO)(CO)NC(C1CNC(=O)N1)=O)N(C)C(c1cncc(-n2ccnc2)n1)=O CN1N=C(C(=O)N2CCOC(C(=O)NCCc3cccc(Cl)c3)C2)CCC1=O CCC(C)C(CC(=O)N1CCCC1CNC(=O)C(O)CCC(C)C)NC(N)=O c1(C(C)(C)C)n[nH]c(=NCC2CC(NC(C34CC3COC4(C)C)=O)C2)o1 C(=O)(C1Cc2ccc(F)cc21)N1CCOCC(F)(CNC(c2c(C)c[nH]n2)=O)C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C2CC2)(NC(c2cncc(Br)c2)=O)C1 c1(NC(C)=O)cccc(CNCC(C2(C)CCNCC2)C)c1 C(CC(C)(C)C)(C(=O)NC(C1CCN(C(C2(C(C)C)CCC2)=O)C1)(C)C)OC c1(N2CCCN(C)CCC2)nc(=NCC2CC3CCC(C2)C3)[nH]c2ccccc12 c1(NC(CC)=O)ccc(NC(=O)NCC2CCC(C(F)F)O2)cc1 C1(NC(C2C(C)(C)OCC2)=O)C2CC3C(C2)C13C(=O)NOCC1(F)CCC1 C12(C(=O)NC(C(=O)OCC)C3CC3)CCC(C)(C1)OC2.C1(=O)CC2(CC2)CN1 CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1cnco1 N1(C(C=C(CC)C)=O)CC(C)(C(=O)NC2CN(C3CCC3)C2)C1 c1(OC)ccc2c(c1)CC(C(=O)NC1CC3(C1)CN(C(=O)CC1(OC)CC1)C3)O2 c1(C(N2CC3C(NC(CCC)=O)C3C2)=O)sc2ccccc2c1CC c1(CN2C(CNC(C(C)(C)C)=O)CCC2)c(F)c(F)cc(F)c1F O=C(CCCCCNC(C1(CO)CCOC1)=O)NCC1=CCCCCC1 C1(C#CC(=O)N(C(C)CCNC(=O)C(c2cccc(F)c2)C)C)(CC)CC1 c1(C(c2n(CC3CC3)nnn2)NC(=O)NC(C)(C)C)cc(Br)c(Cl)s1 C(=O)(CCCCC(C)C)N(CCC1CC(C)(C)NC1=O)CC c1(C(=O)NCC2(C(C)NC(c3c(C)cno3)=O)CC2)ccc(OC(F)F)cc1 C1(N(C(CN(CC(C)(C)C)C)=O)C)CCCC(NC(c2nnn(C)n2)=O)C1 C1(NC(C(n2nnnc2C(C)(C)C)C)=O)CC12CCN(C(=O)CC1CSC1)CC2 CCCCCCN(C(=O)CC1SCCS1)CCNC(C1CC1C(C)C)=O C(CC(C)(C)C(=O)NCC1CC1NC(=O)OC(C)(C)C)NC(C1C(OC)CC1)=O C(=O)(C(O)C(C)c1ccccc1F)OCCOCCOCCOC CCC(CC(=O)N(C)C(c1ccc(C)cc1)C)C(C)(C)C CS(C)(=O)=Nc1cccc(C(=O)NC2CC3(C2)C(F)(F)C32CCC2)c1 C1(NC(CC=C)=O)CC2CCC1N2C(C1CC(=O)N(c2ccc(Br)cc2)C1)=O c1(C(N2C(C)CC(NC(Cn3c(C)ccn3)=O)C2)=O)c[nH]c(C#N)c1C c1(-c2cc(C(=O)NC(CN(C(C(C=C)O)=O)C)(C)C)n[nH]2)ccccc1Cl C#CCCCCCCC(=O)N1CCC(N(CC#C)C(c2conc2CC)=O)C1 Cc1cn(C)c2nc(N3CCC4(CCCC4Nc4ncncc4F)C3)ncc12 c1(OC)ccc2nc(N3C4CCC3CC(O)(C(Cl)(Cl)Cl)C4)sc2n1 C1(C(=O)NCC2CN(C(Cc3nc(C(C)C)sc3)=O)CC2O)CCCC(=O)N1C N=c1[nH][nH]c(C(=O)NCC2CCN(C(=O)C=Cc3ccccn3)C2)c1Br Cc1cc(OC2CCN(CC3CCCCN3)C2)ccc1N(C)C C1(C(N2C(C)CC(CC(=O)NCCCN3CC=CC3)C2)=O)CN(C)CCN1C c1(OC)ccc(F)cc1C(N1CCC2(CC2NC(=O)C(F)C(F)(F)F)C1)=O c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CCC2)cc2nccc(Cl)c2s1 C1(NC(C(CSC)C)=O)COCCC1C(=O)N(CC(F)F)CCO CCCC(C)C(C(=O)Nc1ccccc1Cl)N1CCC(C(C)(C)OC)CC1 C1(C(=O)NC2C3CN(C(C(COCC)C)=O)C2C3)CC2(CCC(F)(F)CC2)CO1 n1(CC)c(N2CCN(C(=O)NC3CC3)CC2)nnc1C1CC1C(=O)OC c1(C(N2CCCN(C(C=CC)=O)CC2C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NC2CC(N(C(=O)CCCN3CCCC3)C)C2)occc1Br c1(C(=O)NCC)ccc(C)c(Cl)c1Cl.C1C(C)(OC)CNC(=O)C2(CC2)C(=O)N1 N1(C(c2n(C)ncc2)=O)CC2CS(=O)(=O)CC2(NC(=O)CCC2(C)CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NC(C)CC1CN(C(C2(C(=O)NC)CC2(F)F)=O)C1 c1(C(=O)NC)cccc(C(=O)NCCC(C)N(C(=O)C(C(C)C)N(C)C)C)c1 N1(C(C2CC(SC)C2)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)(C)C)CC(C)C1 C(N=c1[nH]c(C)nc2[nH]ccc12)C1(C(=O)Nc2ccc(OC)c(C)n2)CC1 C#Cc1cncc(NC(=O)C(CC2CC2)NC(=O)CC(CC)CC)c1 CON=CC(=O)N1CCC(NC(=O)CCN2CCOCC2)C1 C(C)(C(=O)N(CC(O)CN(C)C(C1CC(C(C)C)C1)=O)C)NC(CC)=O c1(C(=O)NCCN(CC(C)O)C(C2C(C=C)C2)=O)cc2n(n1)CCC2 C1(C(=O)NCC(C)C(C)O)(SC)CN(C(=O)CCc2ccc[nH]2)C1 n1(CCC(=O)NC2CC3(C2)CC3NC(C23CC(O)C2C3)=O)cnc2ccccc12 c1(C(N2C(CCC3N(C(CCC)=O)CCCC3)CCC2)=O)cnc(C)cc1Cl c1(C(=O)NC2(CCNC(CC(C)CN(C)C)=O)CC2)ccc(F)c(F)c1 N1(C(CC2C(C)CCO2)=O)CCCCC12CC(NC(=O)CCc1nc(=N)[nH][nH]1)C2 N1(C(CS(=O)(=O)NC)=O)CC2CCCC2(C(=O)NOC2CC2)C1 C(=O)(C(C)(C#N)CC)NCC1CC(NC(CC2ON=C(CC)C2)=O)C1 c1(NC(C2(CC(C)=O)CCC2)=O)ccc(C(=O)NCC(=O)O)nc1 C1(CC#C)CN(C(=O)CN(C(=O)C(C)COC)C(C)C)CCO1 N1(C(c2c(CC)nco2)=O)CCC2(CCC2)C(NC(c2cc(CO)n(C)n2)=O)C1 N1(C(N(CC)CC)=O)CC(C2(Sc3ccc(NC(=O)C(C)C(C)CC)o3)CC2)C1 C1(C(=O)NC(c2ccc(F)cn2)C)CC2(CCN(c3ncc(F)cn3)CC2)CO1 C1(C)(NC(c2cc(C(=O)OC(C)(C)C)on2)=O)CCOCC1CO N1(C(CCCOC(C)C)=O)CC2CCCC(CNC(C3(C(F)(F)F)CC3)=O)C2C1 N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)CC3CCC4(CCC4)CO3)CC2)C1 C1(NC(C2CCSC2)=O)CCC12CCN(C(C1CC1c1ccccc1)=O)CC2 C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2ccc(O)nn2)=O)C1)NC c1(CNC(c2c(C)nns2)=O)ccc2c(c1)CN(C(=O)C(C)O)C2 CC(C)(C#N)C(=O)NCC1CCCC1NC(c1sccc1C(C)(C)C)=O c1(C(N2CCC(CF)C2)=O)cnc(-c2ccncc2)cn1 CC1CN(C(C2CC2C2CCC2)=O)CCN1C(=O)CC(F)(F)F Cc1ccc(Cl)c(C(=O)NC2CCC(CNC(=O)C(N3CCSCC3)C)C2)c1N N1(C(CC2ON=C(CC)C2)=O)CCOCC(F)(CNC(c2ccc(C)o2)=O)C1 CCC(CC)C(F)C(=O)NC(C1(O)CCCCC1)C(=O)NC(C(C)C)C1CC1 c1(C(CNC(c2cnc[nH]2)=O)NC(c2cc(Br)n[nH]2)=O)ccccc1F c1(C(=O)NC2(c3nn[nH]n3)C(C)C2)cnc(O)[nH]1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(N(C)C)C2)=O)CC1C C12(C(=O)NC(CC=C)C(=O)Nc3cnc(F)nc3)CCCC1CCC2 C1(N(C)C(C2CCN(C)CC2)=O)CN(C(=O)C(c2cccn2C)=O)CCC1O Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CCCCCc1cccs1 C=CCC(C(=O)N1CCCC1CNC(C1(S(C)(=O)=O)CCOCC1)=O)C(C)(C)C c1(C(N2C(CNC(CN(CCC)C)=O)CC2)=O)csc(-c2cccs2)n1 c1(OC)cc(Cl)c(C)cc1C(=O)NC(CNC(c1occ2c1CCC2)=O)C(C)C c1(C(=O)NC2C(OC)CN(C(=O)C(C(C)C)SC)C2)c(C)nn(CCO)c1C c1(C(=O)NCC2N(C(c3cccc(CC)c3)=O)CCOC2)cccc2ncsc12 Cc1cc(C(N2CCC(NC(=O)CSC(F)(F)F)CC=C(Cl)C2)=O)cc(N)c1Cl c1(C(=O)OC)ccc2c(c1)C(C(=O)N(C(C)CNC(c1cnc(Cl)s1)=O)C)CO2 C1(C(=O)NCC2CC(C)OCC2)CC(C)(C)CCN1C(C1OC2CCC1C2)=O c1(C(C(=O)NCC(CNC(c2nnn(C(C)(C)C)n2)=O)F)O)ccc(F)cc1F C1(NC(C(CCC)N(C)C)=O)CC2C1CCN2C(=O)CC(=O)N(C)C C#CCC(C)(C)C(=O)NC(C)CNC(C1C=CCCC1)=O N1(C(C2CN(c3nc4ccccc4s3)C2)=O)CC2(CCCCC2)CC1C(F)(F)F Cc1cc(N(C)C)ccc1CNC(=O)C(CO)c1ccccc1.N12CC(C1)C2=O C1(NC(C=C(C)C)=O)Cc2ccccc2C1NC(c1cnc2c(n1)CCCC2)=O C(C(F)(F)CNC(c1ccccc1-n1cccn1)=O)(C1CC1)OC c1(C(C(=O)NCCCCCC)N(C)C(C)C)cc(F)c(F)c(F)c1 C(=O)(C1=CCCOC1)N1C(CCNC(=O)CCOCC(F)F)CCC1 N1(C(CS(C)(=O)=O)=O)CCC2(CC1)CC2NC(C1CCCC1CF)=O CC(C)C(C(=O)N(C1CCN(C(=O)CCc2cscn2)CC1)C)c1cnn(C)c1 C1(C(=O)NCC(CNC(=O)Cc2cnccc2C(F)(F)F)O)CCCC1C1CC1 N1(C(C2CN(C(CC3CC(=C)C3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 CC1(C)CCN(C(=O)Cc2ccon2)C(C(=O)NC2CCN3CCC2C3)C1 c1(SC)ccc(Cl)c(C(N2CC3CCC3(CNC(=O)CC3CCCN3C)C2)=O)c1 C1(CC)CN(C(=O)CCC(=O)N(C)CC)CCC1NC(=O)COC1CCOCC1 C1(C(=O)NC2C(O)C3CCOC23)CN(C(C2(CCCF)CC2)=O)CC12CC2 N1(C(c2nc(C)cn2C)C(=O)NC)CCN(C(C)C)CC1C c1(C(N(CC(C)NC(=O)C(O)C(F)F)CC)=O)cc(S(C)(=O)=O)cnc1O C1(CC)C(NC(=O)CNC(=O)CN(C)C)CCCN1C(=O)C(C)OCCOC C12(NC(CC3CC(OC)C3)=O)COC(CNC(C3CCC(C)C3)=O)(C1)C2 c1(OC)ccc(OC(=O)C(c2cccc(F)c2)OC)c(C)n1 C1(CNC(C2C(C(C)C)C2)=O)CCN1C(=O)C(C)n1cncn1 c1(CN2C(C(=O)N=c3[nH][nH]cc3Br)CC3CC32)cccc2ccncc12 C(=O)(C#CC(C)(C)O)NC1(CC=C)CN(C(=O)CC2CCC(F)(F)CC2)C1 C1(CN(C)C(c2cnc[nH]2)=O)CCCCN1C(C1(C)CCC1)=O Cc1cc2c(cc(C(=O)NCC(C)(C)CNC(C3(O)COC3)=O)n2CC2CC2)s1 C1(CC=C)(NC(=O)C(C)c2cccs2)CCN(c2nc(C(F)(F)F)ns2)CC1 C(C)(CNC(c1cc(Cl)cs1)=O)(CO)NC(CSCC(C)C)=O C(C)(C)(CC(F)C(=O)N1CCC(OCC(N)=O)C1)NC(c1c(C)nc(C)o1)=O c1(NC(C(=O)N(CC)Cc2cnn(CC(C)C)c2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(N)CC(=O)NCCn2cc(C3(O)COC3)nn2)cc(F)c(F)c(F)c1 C1(CCC)CN(C(=O)C(c2ccccc2Cl)OC)CCN1C(=O)CC(C)(C)OC c1(C(=O)NCC(C)N(C(c2c(C)cc[nH]2)=O)C)c(C)nc2ccccn12 C1(CNC(c2coc3c2COC3)=O)CC2COCC2N1C(=O)C=C1CCCC1 c1(CC)c(C(N2CC=CC(NC(=O)CNC(=O)CC(F)(F)F)C2)=O)nnn1CC C(=O)(CC(C(F)F)n1ccnc1)NC1C2CN(C(C(CC)O)=O)C1C2 C1(C(=O)NCC2CCC(N(C)C(C3(C)CCOCC3)=O)CC2)CCC2(CCC2)C1 C1(CNC(CC=C=C)=O)CCC2(CO1)CC(NC(=O)Cn1cc(C)cn1)C2 C1(C(C)(C)C)OCCC1CNCC1(F)CCNC1 CC1CCN(C(c2cccnc2Cl)=O)C(C)C1NC(C1CCCS1)=O N1(C(C(CCSC)(C)C)=O)CC(C)C(NC(C2COCCOC2)=O)C(C)C1 N1(C(CCc2onc(C)n2)=O)CCCCC(C(=O)NCCCCC(C)(F)F)C1 Cc1nn(CC(=O)N(CC(C)(C)CNC(C2SCCC2C)=O)C)c(C)c1C Cc1noc(C)c1C=CC(N1CCCCC1CCN(C(=O)CC1C=CCC1)C)=O Cn1cccc(C(=O)NCC(CC2CC2)C(=O)NCC2CCCC2(C)C)c1=O C12(C(N3C(COC)C=CCC3)=O)CCN(C(=O)C=Cc3cncn3C)CCC1C2 n1(CC)nc(C(=O)NC(C)C(C)NC(c2coc(CS(C)(=O)=O)n2)=O)cc1O c1(N(C(=O)NCCN(CCCC)Cc2cccc(Br)n2)C)ccc(F)cc1 Cc1cc(C)c(CC(N2CCC(N(C(=O)C(F)=CCCF)CCO)CC2)=O)s1 CC(C)(CC(F)F)C(=O)N1CCC(F)(CNC(C2CC(OC(F)F)C2)=O)CC1 c1(C(=O)NCC(CO)NC(CCC2CCCN(C)C2)=O)c(O)ccc(Cl)c1F CC1CC(NC(=O)C=CC2CCCO2)CCN1C(C1CC2CCC1C2)=O N1(C(CCOC(C)C)=O)CCC2(C1)CN(C(=O)CCC(C)N(C)C)CCO2 Cc1cncc(C)c1C(N1CCCC(c2cn(-c3ncc(Cl)cc3Cl)nn2)C1)=O N1(C(CCC(C)OC)=O)CC(NC(=O)CCCc2cccnc2)C2CCCCC12 CC(C)C(C(C)NC(c1cc(Cl)ns1)=O)NC(=O)CNC(=O)CC1CCCC1 N1(C(c2ccc(OC)s2)=O)CCCCC1C(N1CCOC(C2CC2)C1)=O Cc1nn(C)nc1C(=O)NC(C)(C)CNC(=O)C(C1CC1)C1CC1 C1(NC(=O)CN2CCC2)CCCCC1N=c1cc(Cl)nc(-c2ccccn2)[nH]1 c1(C(=O)NC2CCC(CC(=O)NCCC(COC)O)CC2)ncc(F)cc1N c1(CNC(C2CCC(=O)C2)=O)ccc(CNC(C2CCCC(=O)C2)=O)c(F)c1 C1(C(N(C2CCN(C(C(C)OCC(C)C)=O)CC2)C)=O)C2CCCCCCC12 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)CC1 C1(CC(C)NC(C2CC3(CC3)CO2)=O)CCN(C(C2CC3C=CC2O3)=O)CC1 Cc1cn2c(CC(=O)NCC(CO)NC(c3c[nH]cc(Cl)c3=O)=O)csc2n1 c1(OC)c(-c2nc(CN=[N+]=[N-])no2)ccc(C)c1F N1(C(C(c2ccccc2)OC)=O)CCC(NC(C2CC2[N+](=O)[O-])=O)C(F)(F)CC1 c1(C(N2CCC(NC(C(C)=C(CC)C)=O)C2C(C)C)=O)cccc2c1OCC2C C(=O)(CC(O)CNC(C1CCCCC1O)=O)NCc1c(CC)nns1 S(=O)(=O)(c1ccc(NCCN=S(C)(C)=O)cc1Br)NC1CC(CC)(CC)C1 C1(C(N(C(C)C(C)(C)C)C)=O)CC2CC1CC2NC(=O)COCC(C)(C)C C(=O)(C1=CC2CCCCC12)N1C(CN(C(C2CC=CC2)=O)CC)CCC1 C1(NC(CCN(CC=C)C(c2cn(COC)cn2)=O)=O)CC(=O)NC1=O C1(C(=O)NC(CCCNC(C2C(C)SCCC2)=O)CO)CC2CCC(C1)O2 N1(C(c2c(C3CC3)[nH]c(=N)s2)=O)CC2CC(NC(c3ccc(Cl)nc3)=O)CC2C1 c1(C(=O)NC2(COC)CN(C(C3C4CCC(=O)C34)=O)C2)ccc(CO)nn1 c1(CC(=O)NC2(CN(C(=O)CCS(C)(=O)=O)C)CC2)cccs1 C1(NC(CCN(C(C(CC)(C)OC)=O)C)=O)CC2COCC2C1 N1(C(CCC2(C)CC2)=O)CC=CC1CNC(C1CCC(C(N)=O)C1)=O CC1(C)C(C(N2CC=CC2CNC(=O)CCCc2nccs2)=O)C1C(F)F C1(C(=O)NCC(C(=O)OC)O)(NC(=O)C(F)C(C)C)CCC(C)(C)C1 c1(C(=O)OCC)cnc(Nc2nc(C)ncc2COC)nc1C(F)(F)F c1(CNCC)cccc(CNc2nc(C)ns2)c1 c1(CCC(=O)NC(CNC(C2(CCCC)CC2)=O)(C)CO)cccc(OC)c1F c1(C(N2CCC(CNC(c3c(C)ccn3C)=O)C2)=O)nc(C2CC2)ncc1Cl N1(C(C2(OC)CC(C)C2)=O)CCCC(NC(c2nnsc2SC)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCC(NC(c2cc(C(C)(C)C)ccn2)=O)C12CC2 CC1CN(C(c2cnccn2)=O)CC1NC(=O)CCOCCOCCCO c1(C(=O)NC23CC(C(=O)OC)(C2)C3)cc(C(F)(F)F)c(C)o1.c1(C(=O)N)ccon1 Cc1cnncc1C(=O)NCC(=O)NCC1(C#N)CC1 c1(NC(=O)NCC(=C)CCNC(=O)CC2CCCC(O)C2)cc[nH]c2nccc1-2 CC1OCCC1CC(=O)NC(C1CCCC1)CNC(C1CCCC1)=O c1(C(N2C(CCCNC(c3n(C)nnc3)=O)CCC2)=O)cc2ccc(F)cc2[nH]1 C1(C(N2CC(CC)N(C(C34CSCC3C4)=O)CC2)=O)CN=C2N=CNN2C1 C(=O)(CCCCCN(C)C)N(Cc1c(C)n[nH]c1C)CC1CC1 c1(C(N2C(C)CC(NC(c3ccccc3OC(F)F)=O)C2)=O)ccnn(C)c1=O C1(NC(C2CC(F)(F)C2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)C2(CCOC2)C1 c1(C(N2CCC3CCC(NC(C4(C)CCOC4)=O)C32)=O)n[nH]c2ccc(F)cc12 C1(CNC(CC2N(C(CC3(N(C)C)CCC3)=O)CC2)=O)CCCC2(CC2)C1 CCC(C)(O)C(=O)NC1C2CN(C(c3ccc(C4CCC4)nc3)=O)CC12 c1(N(CC)CC)ccc(C(=O)NCC2(NC(=O)C(C)C(C)n3cccn3)CC2)cc1 C12(C(N3CC(OCCNC(C(C(C)C)O)=O)C3)=O)C(=O)C3CCC1C2C3 C(=O)(C(C)CC(C)C(C)=O)N1C(CCNC(c2cc(CCC)[nH]n2)=O)CCCC1 C1(C(=O)OC)CCC(=O)N1C(=O)Sc1ccc(CCN)cc1 C1(C(=O)NCCCNC(COCCC#C)=O)(C(F)F)CCOCC1 C1(N(CC)Cc2ccoc2C)CCN(C(=O)OC(C)(C)C)C2(CC2)C1 CC1(C#CC(=O)N2CCC(Nc3ncc([N+](=O)[O-])cn3)C(F)(F)CC2)CCCO1 S(=O)(=O)(CCCCCl)NC1CC(N(CC(=O)N(CC)Cc2cccc(Cl)c2)C)C1 O=C1CC2(CO1)CN(C(=O)C(Cn1cccn1)NC(c1cccs1)=O)C2 C(=O)(CC(O)CC(C)(C)C)NCCCN(C(c1c(CCC)cccc1)=O)C1CC1 N1(C(C(C(=O)OC)(C)F)=O)CC2OCC(NC(=O)Cc3ccno3)C2C1 Cc1nc2cncc(C(N3CCC(C)C(CNC(=O)CC(F)F)C3)=O)c2[nH]1 c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Br)cnc1C(F)(F)F CCCCCC(=O)N1CCN(C(c2ncc(-c3ccc(F)cc3)o2)C)CC1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CCC2(CCCN2C(c2cccc(Cl)c2)=O)C1 N1(C(C(C)n2cccn2)=O)C2CCC1CC(N(C(=O)CCCC1CC1)C)C2 c1(C(=O)NC2CN(C(c3cscc3F)=O)CC2O)cccc2nc(O)ccc12 N1(C(C2CCN(C(CNC(=O)NC)=O)C2C)=O)CCCCCCC1C c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CNC(=O)C1(C)C)=O C(=O)(C(O)C(C)(C)C)NCc1cccc(CC(C)NC(c2ccccn2)=O)c1 c1(C(=O)NC2CC(CNC(=O)CCCF)CC2O)cc(Cl)cc(Cl)c1 CC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CC(C)N(C(c2cc(O)ncn2)=O)C1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(OC)CN1C(c1ccncc1NC)=O c1(OC)cc(C(=O)NCCCN(C)C(c2cnc(S)nc2)=O)sc1Cl N1(C(C(CC(C)(C)C)OC)=O)CCCC12CCCN(C(=O)C=C(C)C(C)(C)C)C2 C1(NC(c2c(OCC)scc2)=O)CN(C(C2CN3CCC2CC3)=O)C(C)(C)C1 c1(CC2(C(N3CC(C(C(=O)OC)O)C3)=O)CC2)cc(Cl)ccc1OC C1(CNC(C2CCSC2)=O)CC2(CCN(C(C3CCN3C3CCCC3)=O)C2)CO1 c1(NC(c2c(C)nc(NC(c3ccc(Cl)o3)=O)s2)=O)cccc2c[nH]nc12 N1(C(C(C)=C(C)C)=O)CCN(C(=O)CCc2ccoc2)CC1CO C1(C(=O)NCC(CC(C)C)NC(=O)C(c2ccncc2)C)CCCCN1N=O c1(CC)nn(C)c(CC(=O)NC2(CNC(C3(OC)CC3)=O)CCCCC2C)c1Cl C(=O)(C(C1=CCCCC1)N1CCCC(c2ccccc2F)C1)Nc1nnn(C)n1 C12(NC(=O)CCF)CCCC1N(C(C1CCC(C(F)(F)F)O1)=O)CC2 CC1CCC(C(=O)N(CC(C)CO)C)N1C(C1CCOC1(C)C)=O c1(C(N2CCCCC(NC(C3N(CC)CCCC3)=O)C2)=O)cc(F)c(Cl)cc1Cl N1(C(C(CC)OCC)=O)C2CCC1C(C)C(NC(=O)Cc1cnccn1)C2 Cn1cc(Cl)cc1C(=O)NCCOCCC(=O)N(CCF)C1CC1 c1(OC(C(=O)N(C2CCCN(C(=O)C3CC3)C2)CC)C)ccc(Br)cc1 C1(NC(Cc2c(C)n(C)cn2)=O)CN(C(c2ncoc2C(C)C)=O)CC1N=[N+]=[N-] Cc1cc(C(=O)NC2C3CC2N(C(c2ccnc(O)c2)=O)C3C)ncc1F c1(C(C)C)ncc(C(=O)N(CCC(C)NC(=O)CC(=O)NC2CC2)C)s1 Cn1nnnc1SCC(N1CCC1N(C(=O)C=C1CCCCC1)C(C)(C)C)=O C1(CNC(c2ccc(OC)s2)=O)CC2CC2N1C(=O)Cc1ccccc1Br CC(C)(C)S(=O)(=O)CC(=O)NCC1CC(O)CN1C(c1cccc2c1OCC2)=O c1(C(=O)NC(CC)CNC(c2cnn3c2NCCC3)=O)cncc2ncn(C)c12 Cc1sc(C)c(C(=O)NCC2CC(O)CN2C(C2CCCN2C=O)=O)c1C#N c1(C(N2CC(COC)N(C(=O)C=CC(=O)OC)CC2)=O)cccc2scnc12 C=C(CNC(C1CC1(F)F)=O)CCNC(c1nocc1C)=O S(=O)(=O)(c1ccc(NC2CCC(O)CC2)c(Br)c1)N(CC)Cc1ccnn1C c1(C(N(CCN(C(c2cnnn2CC)=O)CC)CC)=O)cccc(C(C)C)c1F C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C(=O)Nc2cc(F)ccc2F)C(O)CC1 C1(COC)(NC(c2csc(O)n2)=O)CCN(C(C2COC(C)C2)=O)CC1 O=C1CC(C(N2CCC(N(C(=O)Cc3cnoc3)CCO)C2)=O)CC(=O)N1 c1(C(C(=O)NCC(C)C)N(C)Cc2ccc(F)cc2)cccc(OCCCC)c1 c1(N2CCC(CC)(CO)C2)nc(N2CCCC(CC3CC3)C2)nc2c1ncn2C c1(C(N(C)CC2N(C(C(C)SC(F)(F)F)=O)CCC2)=O)cc(N)c(F)c(F)c1F C1(CC)(CC)C(OC)CC1N(C)C(=O)NC1CCN(C)CC1 Cc1nn(C)c(C(N2CCN(C(c3nn(C)cc3Cl)=O)C(CC3CC3)C2)=O)c1Cl C1(CC(=O)NCC(N2CCN(C(C3(C)CCC(=O)C3)=O)CC2)C)CCC2(CCC2)O1 N1(C(C2(C(=O)OC)CC2)=O)CCC2CN(C(c3cnc(Cl)cc3C)=O)CC2C1 n1(CC(=O)NC(C(=O)N(CC(C)SC)C)Cc2cn[nH]c2)cnc(C#N)n1 C1(CC(=O)NCC2C(NC(C(C)(C)OC)=O)CC2)CCCC(C2CC2)O1 c1(OCC(=O)NCCCN(C(C(C2CCCC2)OC)=O)C)cc(Cl)ccc1C C1(NC(CC=C(C)C)=O)CCCC12CN(C(C1CC3(CCCC3)CO1)=O)C2 C1(NC(CN(C(=O)Cc2cnn(C)c2)CC#C)=O)COC2(CCC2)C1 C1(C)(C(=O)Nc2c(CC)n(CC)nc2)CC(O)CN1C(=O)CC1CCCC2CC12 C(CCN=c1[nH]nc(O)s1)N(C(c1c(C)cno1)=O)CC1CCCCC1 C(=O)(C(F)C(F)(F)F)N1CC(n2cc(CNC(c3n(C(C)CO)ccn3)=O)nn2)C(C)C1 c1(NC(c2n(CC)nnn2)c2nscc2Br)ccc(C(=O)OC)c(F)c1 C1(C(=O)NCC2OCCN(C(c3cc(C)ns3)=O)C2)OCC2CCCCC12 N(C(=NCCSC)NCC(c1cccc(Cl)c1)OC)CC1(COC)CC1 C1(C(=O)NC(CC=C)CNC(C2CN(S(=O)(=O)CC)C2)=O)CN(C)C(=O)CCO1 C(=O)(CC(C)P(C)(C)=O)NC1C(C)CN(C(C2(C(C)(C)O)CC2)=O)C1 c1(SC2CC(NC(C3(COC(C)(C)C)CCC3)=O)C2)ccc(Br)cc1 C1(C(N2CCN(C(=O)CCC[N+](=O)[O-])C(CCO)C2)=O)CCN2CCOCC12 c1(C(N2CC=CC(NC(C(C)CC3CCCCC3)=O)C2)=O)nc(Cl)cc(N)c1Cl C1(CNC(CSCC#C)=O)COCC1NC(=O)CCC1(C#N)CCC1 c1(CC(=O)N(CCNC(C(C(COC)C)C)=O)CCOC)cnc2cccnn12 c1(C(=O)NC2(CC=C)CCNC2)cc(F)c(F)cc1NC(=O)N(C)C N1(C(c2c(C)n(CC(C)C)nc2)=O)CCN(C(=O)CCC2CC2)CC1CC1CC1 C(=O)(CP(=O)(C(C)C)C(C)C)N(CCC(C(C)C)NC(C(C1CC1)OC)=O)C C(CC(C)(C)C)(C(=O)NC1CCC(OC)CC1)NC(c1n(C=C)ncc1)=O C(=O)(C(C)(C)CCC#N)N1CCCC(C(N2CC(C)C2(C)C)=O)CC1 c1(C(CNC(C2SCCS2)=O)=O)cc(F)ccc1Br c1(CNC(=O)COC2CCC2)csc(CNC(c2ncoc2C2CCC2)=O)n1 CC(C)(CNC(=O)CC1CC2(C1)CN(C(=O)C1=COCC1)C2)C1=CCCC1 c1(C2N(C(C(C)=O)=O)CCCC2)cn(C2CCCc3c(F)cc(F)cc32)nn1 c1(C(=O)NCC(C)NC(CCc2c(OCC)cccc2)=O)ccc(C)n(C)c1=O C(=O)(C(C)(COC)OC)NC(COC)CNC(=O)CCSCC(C)C C(CCN=c1[nH]c(=N)[nH]c(=NCC23COCCN2C(=O)OC3)[nH]1)OCC c1(C(N2CCC(C(N(C)Cc3c(C)n[nH]c3)=O)(CF)C2)=O)ncn2c1CCC2 Cc1ccc(F)c(C(=O)NC(C)CNC(c2ccc(OCC(F)(F)F)o2)=O)c1 CC1(C(=O)NCc2nc(CNC(=O)COCC3CC3)cs2)CC1(Cl)Cl C1(C(=O)NCC(C)(C)OC(C)C)CN(C(C2CCCC(C)CC2)=O)CCC1(C)C N1(C(C2(CCCC)CCC2)=O)CCOCC(C(=O)NCCNS(C)(=O)=O)C1 C1(C(=O)NCC2CC2(Cl)Cl)CCCCN(C(=O)C=CC2CCCC2)C1 c1(C(=O)NC2CCC(N(C(CN(c3cnccn3)C)=O)C)C2)cncc(O)c1 C1(C(N(CC(=O)OC)C)=O)(CC)CCCN(C(C2(OC)CCOC2)=O)C1 CC1CCC(C(=O)NCC2CC(O)C(O)C2)CN1C(C1CC1(F)Cl)=O N1(C(C(CC)CC)=O)CCN(C)CC1CNC(=O)C(c1ccc(Cl)cc1)CO C1(C(=O)NC(c2noc(C)n2)CC)CC(NC(=O)C(C#N)CC)CCO1 c1(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)cc2cc(F)ccc2s1 C(CCS(=O)(=O)C(C)C)N(CCCNC1CCCN(C(COCCC=C)=O)C1)C N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(CCc2ccccc2F)CC1C c1(NC(C2CC3CC3N2C(c2ccc(Cl)o2)=O)=O)cc(F)c(F)cc1Br C1(C(=O)NC(CC(C)NC(c2ccc(CO)cn2)=O)C)CCS(=O)(=O)N1 c1(SC(C2(C)CC2(F)Cl)=O)ccc(Cc2cn(CCN3CCSCC3)nn2)cc1 Cc1ncccc1C(=O)NCCOCCN(C(=O)C(C)OCCN(C)C)C N1(C(c2ccc(C(C)=O)cn2)=O)CCCC(O)(CNC(c2csnc2C)=O)CC1 Cc1cc(C(=O)NC2CCN(C(C3COC(=O)N3C)=O)C2(C)C)cc(F)c1 N1(C(C2(CCC)CCC2)=O)CCC(C(F)CNC(=O)Cn2cc(C)cn2)CC1 c1(C(N(C)CC2CCCN(C(C(C)C)=O)C2)=O)c2c(cc3c1CCC3)CCC2 C1(C(=O)NCC2(NC(c3ncsc3Br)=O)CCC2)CC2CCC1O2 N1(C(CC(C)(C)C)=O)CCC(NC(C2(CCF)CCC2)=O)C(CO)CC1 C=C(C)CC(C(=O)NC1CCOC1C(=O)Nc1cnn(C2CC2)c1C)OC C(=O)(C1=CC(C)(CC)C1)NCCCC1N(C(CC)=O)CCCC1 c1(NCCCc2nnc(C)s2)[nH]c(=NCCCC(F)F)nc2ncn(C)c12 c1(C(N2CCOCC2CNCc2cn[nH]c2)=O)ccc(N2CCCCC2)cc1.C C=CC(C)(O)CC(=O)NCC1CC(C)CCN1C(=O)Cc1sc(S)nc1C C1(CC(=O)N(C(C)CCNC(c2cnn[nH]2)=O)C)(CO)CCCCC1 c1(CC(=O)NC2CC(N(C)C(c3ncccc3Cl)=O)C2)cnn2c1OCCC2 c1(C(N2CC(C)N(C(c3cc[nH]c3)=O)CC2)=O)ccc2nnn(C(C)(C)C)c2c1 Cc1ccccc1C(C)C(=O)NCC1C2CN(C(c3csc(C(C)C)n3)=O)CC12 N1(C(c2nc(N(C)C)oc2)=O)CCN(C(c2csnn2)=O)C(c2cn[nH]c2)C1 c1(C(N2C(C)CCC(CNC(C3CC(C)(F)C3)=O)C2)=O)cccc2cncn12 N1(C(CCC#C)=O)CC(OC)C(NC(=O)CC2CCCCC2O)C1 Cc1cc(C(=O)N(CCC(C)NC(c2ncn(C(C)C)n2)=O)C)n(C)n1 Cc1cccc(-c2cn(CC3CCN3C(c3coc(Br)n3)=O)nn2)c1 C(=O)(C1=CCCCO1)N1C(CC(=O)NCC(C)C2CCC2)CCCC1 N1(C(C(C)Cn2ccnc2)=O)CCC2(CCC2NC(C2CCC(=O)O2)=O)CC1 c1(C(=O)OC(C)=O)cccc(-c2cnc(NC(c3ccc(Cl)cc3)C)nc2)c1 N1(C(c2c(CC)n(CC)nc2)=O)CC(CNC(C2(C)CCCC2)=O)CC12CCC2 c1(C(N2CC(CC(C)NC(c3cc(OCC)n[nH]3)=O)C2)=O)nccc(Cl)c1O c1(C(=O)NCC(C)(C2CC2)NC(COCC=C)=O)c(C)nsc1NC1CC1 C(CNC(=O)C(c1cnn(C)c1)O)(CCCC)NC(COCCC=C)=O c1(CC(=O)NC2CC(C(N3CCC(c4ccccc4)C3)=O)C2)ccc(O)c(O)c1 C1(CC(=O)NCCCCCN(C)C(c2cn(C3CC3)nn2)=O)CCCCC1(F)F C(CC)(CC(C)O)NC(CCN(C(C(CC)OCC)=O)C1CC1)=O C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C(C)C)NC=O)CC(C)(C)C1 N1(C(C(CC#C)O)=O)CCN(C(c2cnn(C)c2Cl)=O)CC1CCOC c1(C(c2n(CC(=C)C)nnn2)NC2(C(=O)NC(C)C)CC2)ccc2occc2c1 c1(N(C(=O)CC2CC3COCC23)C)cccc2cccnc12 C1(NC(C(C)=C2CCCC2)=O)CN(CC2CCN(CC(C)C)C2)CC1C c1(CC(=O)NC(C2(CNC(C3(OC)CCSC3)=O)CC2)C)nc(C)sc1C N1(C(COC)=O)CCCC(C(C)(C)C(=O)NCC2(N(C)C)CCC2)C1 c1(CC(=O)OCC)cc(Cl)ccc1Cl.N1(C(CCCOC)=O)CC2C(C1)CO2 N1(C(C2C=CCC2)=O)CC23CCCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C3 C(=O)(C(CN(C)C)NC(=O)C(F)C1CCC1)N(CC=C)CCOC CCC(C)(C(=O)NCC1CCC(C)(C)CN1C(c1cc(C)nn1CC)=O)C(N)=O c1(C(C)(C)C)ccc(C=CC(=O)NCC(CO)NC(C2(C)C=CCCC2)=O)cc1 c1(C2N(CC3CC3CNC(C3N(CC)CCC3)=O)CCC2)ccc(OC)cc1Cl N1(C(CCC=CC(C)C)=O)CC(NC(=O)C(Cc2ccccc2)OC)CC(F)C1 c1(C(N2CC(C)C(NC(c3cc(CN(C)C)c[nH]3)=O)C2)=O)cc(Cl)c(F)cc1Cl CC1(C)CC(C)(CNC(=O)C2=CCCCO2)CN1C(c1ccc(C(F)(F)F)s1)=O N1(C(c2cccnn2)=O)CCCC2(C1)CN(C(c1cc(Cl)ccc1O)=O)C2 Cc1[nH]c2ncccc2c1C(N1CC(N(C)C(C2CC(N(C)C)CCO2)=O)C1)=O C1(CNC(CCN(C)CCO)=O)CC(NC(=O)CNc2ncccn2)C12CCC2 N#Cc1nnc2ccccc2c1N1CCC(O)(CNC(=O)C2=COCCO2)C1 Cc1nc(CN2CC(=O)N(CCCC3CCCCO3)C2=O)ccc1Br Cc1ccnc(C(C)(C)C(=O)NCC2CCC(NC(c3cn(C)c(O)n3)=O)C2)c1 C=CCCC(C(=O)NCc1noc(C(N)=O)n1)NC(C1CC1C1(C)COC1)=O c1(C(=O)OCC(C)NC(=O)OC2CCC2)coc(COC(C)(C)C)n1 c1(C(N2CCC(CCNC(CSCCC)=O)CC2C)=O)ccc(Cl)c(OC)c1F N1(C(c2cc(C)cc(O)c2)=O)CC(C)(C)OCC1CNC(=O)CCC1CCOC1 c1(N(C)Cc2nncn2C)nc2cc[nH]c2c(=NCC2CC23CCOCC3)[nH]1 n1(CC)nc(C)cc1C(=O)NC(C(=O)N(C1CC1(C)C)C)C1(C)CC1 Cc1nc2ccc(C(N3CC4(CCCCN4C(=O)C4=CCCC4)C3)=O)cc2s1 c1(SC)cc(C(=O)NCC2CCCN(C(C34CCC3C4)=O)C2)ccc1NC(C)=O c1(C(=O)NCC2(CNC(C=C(CSC)C)=O)CC23CCC3)ccc(N=[N+]=[N-])cn1 N1(C(c2cn(C(C)C)nn2)=O)CC2CC1CCN2C(=O)CCCCCF N1(C(c2ccc(NC(CCCCCOC)=O)cn2)=O)CCCC(C2CCC2)C1 C1(C(=O)NC2CC(C)CN(C(c3csc(O)n3)=O)C2)CC2COCC(C1)C2 N1(C(CCN(C)CC)=O)CCCCC1C1CCCN(C(c2cocc2C)=O)C1 C1(C(=O)NC(C(C)SC)C)CC=CC(NC(=O)CCn2ccnc2)C1 C(C1CCCC1)=CC(=O)NC(C1CC=CCC1)C(=O)NCC1CC(=C)C1 C(=O)(CCC(=O)N1CCC(CNC(c2cn(C(C)(C)C)nn2)=O)C1)OC CC(C(=O)NCC(C)(Cn1cccn1)NC(c1n[nH]c(C(C)C)n1)=O)S(C)(=O)=O C(=O)(C1CCCc2ccnn21)N1CC(CNC(=O)CCN2CCC2)C2(C1)CCC2 C1(NC(c2ccc([N+](=O)[O-])cc2)=O)CN(C(c2cnc[nH]2)=O)C2(CCOC2)C1 Fc1ccc(Br)cc1CNc1nc(-c2cccc(I)c2)cs1 C(CCCCCF)N(C1(C(=O)O)CCOC1)C C(=O)(C1CCc2cccc(=O)n21)N1CCC(C)(NC(C2CCCC2O)=O)CC1 C1(CNC(c2cc(C)n(C)n2)=O)CC(C)CCN1C(=O)C(C)Cc1ccnn1C c1(NC2C(NC(C(C(C)O)N(C)C)=O)CS(=O)(=O)C2)ncc([N+](=O)[O-])cc1Br c1(OC)ncc(C(=O)NC2CCN(C(=O)CC3CC3)CC2C)cc1C(F)(F)F C1(Cn2cc(C(C)(C)SC)nn2)CCN(C(c2cccc(C)n2)=O)CC1(F)F C1(C(C)(C)O)(CNC(C23CCCC2C3)=O)CN(C(C2(Br)CC2(F)F)=O)C1 c1(NC(C2(O)CCN(C(CCc3cccc(C)n3)=O)C2)=O)cc(Cl)ccc1I n1(CC(=O)N(C(CCNC(c2cn(C(C)C)nc2)=O)C)C)cccc(N)c1=O C(CC(C)C)(C(=O)NCC(C(C)C)NC(c1cc(Cl)ccc1O)=O)OC C1(C(=O)NC2CCCN(CC#N)C2)C2Cc3ccc(Cl)cc3C12 CC1(C)CCCN(C(C2CC(=O)CO2)=O)C1CNC(c1cccn2ncnc12)=O C(C(CC1CC1)C(=O)NCCCC1CCC1)NC(C1N(C(C)(C)C)CC1)=O n1(CC#C)cnnc1C(=O)NCC1(CC(=O)NC2CNC(=O)C2)CC1 N1(C(C(CC)CC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C(O)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2COCC(C1)C2NC(=O)CNC(=O)C(C)CC N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCN(C)CC1CNC(c1cc(C(N)=O)co1)=O C(CCCC(=O)N(C1CCCC12CC2)C1CC1)N(C(CC1ON=C(C)C1)=O)C C(CSC)(C(=O)NC(C)(CNC(c1csc(-c2cnc[nH]2)n1)=O)CO)OC C(=O)(C1=Cc2ccccc2C1C)NC(CNC(CCCOC(C)=O)=O)(C)C C1(C(N2CCC(N(C(=O)CNC=O)CC)C2)=O)CCC(F)(F)CC1(C)C C(=O)(C(CC)CCCC)N1C(Cn2cc(C(=C)C)nn2)CC(COC)C1 C1(NC(C(C)(C)CC2CC2)=O)COC2(CCN(C(c3cc(C#N)cs3)=O)C2)C1 C1(CC(=O)N(C2CCN(C(=O)C=Cc3ccc(C)s3)C2)CCC)CCCCC1O N#Cc1ccc(C(=O)NC(C2CCCCC2)CNC(C2CC2F)=O)s1 Cn1[nH]c(C(=O)NCC2(F)CCN(C(c3ccnc(C(N)=O)c3)=O)C2)nc1=O N1(C(c2cccc(N)c2N)=O)CCCC(C2CC2NC(c2cccnc2F)=O)C1 N(C1CCc2ccccc21)(C(CCC=C)(C)c1nnnn1C1(OC)CC1)C1CCC1 C#CCCCCCC(=O)NC(C)CN(C)C(C12CCC(CF)(C1)OC2)=O C12(CC(OCC)OC)CCCCC1N(C(=O)CCCCCl)CC2.C1CCCC(=O)O1 C1(NC(Cn2ncc(C)cc2=O)=O)CCCC12CN(C(c1n[nH]c(C)c1O)=O)C2 C1(C)(NC(c2ncn(C(C)C)c2)=O)CCCN(C(=O)Cn2cc(C(C)O)nn2)C1 N1(C(CN(CC)CC)=O)CCC(CCN(C)C(c2cnc(C(C)C)[nH]2)=O)CC1 C12(C(=O)NC(CN(C(=O)CC3(COC)CC3)CC)C)CC1COC2(C)C c1(C(N2CC(O)(C(C)NC(CS(CC)=O)=O)C2)=O)ccc(OC)c(N)n1 N1(C(C(c2cccs2)SC)=O)CCS(=O)(=O)C(CCNc2ccncn2)C1 C1(C(N(CCCCCCC)C)=O)CC2CCC1N2C(=O)C(C)CCN(C)C c1(C(N)=O)ccccc1C(N1C(CNC(C2CCCSC2)=O)CC2CC12)=O C1(C(N2CC(NS(CC(=O)OCC)(=O)=O)(CF)C2)=O)CCCC12CCC2 C(C(=O)NCCC(Cl)Cl)(C(C)(C)C)NC(CC(C)c1ccco1)=O N1(C(C(C)C2CC2)=O)CCC(O)(CN(C(=O)Cn2ccc(Br)n2)C)C1 c1(C(N2CCCC(O)(CNC(c3nccs3)=O)C2)=O)c(F)cc(Br)cc1F c1(CC(=O)NCC(C)(C)OCCNC(=O)COC(F)F)cccnc1Cl N1(C(COc2cn(C)nc2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C N1(C(c2cc(C)nn2C)=O)CCC2(CC1)COC(C)C2NC(=O)C(Cl)Cl c1(CCC)nc(C)c(C(=O)NC2CCCCC2NC(c2ccc(F)cn2)=O)o1 Cc1c(C(=O)NC(C)(CNC(=O)C(C)Sc2ccccc2)CO)cccc1Cl c1(C(=O)NC2CN(C(c3cc(I)ccc3Br)=O)CC2F)ccnc(Cl)c1Cl C(=O)(C(C)C(F)(F)F)N1CC(OC2CCN(C(c3c(C)cc(COC)o3)=O)CC2)C1 Fc1cccc2nc(NCCSc3cccc(Cl)c3)cn12 N1(C(c2cc(F)ccc2Cl)=O)CCC(N=c2ccc3nccn3[nH]2)C1 C1(CNC(C2(CCOC)CCCC2)=O)C2CCC(C2)N1C(c1cc(C)[nH]n1)=O C1(C#N)(C(N(CCCCNC(=O)CSC(C)(C)C)C)=O)CCCOC1 c1(SC)ccc(Cl)c(C(=O)N(C(C)CNC(=O)CNC(c2ccncc2)=O)C)c1 C1(CN(C(=O)C(C)(O)C2CCC2)C)CCCN1C(=O)CC1CCNC1=O C1(CNC(=O)Nc2n(CC)nnc2)CCC(F)(F)C(=O)N1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2c(N)cn(C)n2)=O)CC1 c1(C(=O)NCCCN2CCN(C(C(C(C)C)F)=O)CC2)cc2ccnn2cn1 N1(C(C(N2CCC(C)C2)=O)=O)CC(C(=O)OC(C)CO)CCC1=O Cc1cc(CNC(c2cc(F)c[nH]2)=O)oc1C(=O)NCC1CC1Cl NC1CCc2cc(C(=O)Nc3ccc(C#N)cn3)ccc2C1 CCC(CC(C)C)C(=O)NC1COCC1NC(=O)CSc1nnc(C2CC2)o1 C1(C2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)(NC(c2c(CC)nco2)=O)CC1 c1(CC)cccc(C)c1NCc1ccc(N2CCC(C)CC2)c(F)c1 Cc1cc(C(N2CCCC2C=CC(N2CC(O)(C(F)(F)F)C2)=O)=O)cc(F)c1 C1(C)(C(=O)NC2CCN(C(c3ccc(C(C)=O)s3)=O)C2(C)C)CCCCNC1=O C(=O)(CC(C)C(C)(C)C)NCCCCCNC(c1ccn(C(C)C)n1)=O CC1(C)CCC(NC(=O)CC(F)(F)F)C(CNc2ccnc(C3CCC3)n2)C1 c1(NCc2n(CCC)ccn2)cc(NCc2cnn(C)c2Br)nc(C)n1 c1(C(N2CC(CCCNC(C3N(CC)CC3)=O)OCC2)=O)cc([N+](=O)[O-])cn1C C#CC1CN(C(c2ccc(CO)o2)=O)CCN1C(c1n[nH]c(CO)c1C)=O C(=O)(C1=CC2CCC=CCCC12)NCCCN(C(=O)CCF)C1CC1 c1(C(=O)NCC2N(C(CC(COC)C)=O)CCC2)cc(F)ccc1O c1(C(=O)NCC2CCC(NC(c3ccc(Cl)nn3)=O)CC2)ccc2sncc2c1 Cc1ccc2c(c1)NC(C(=O)NCC(O)CC(F)(F)CO)NS2(=O)=O c1(C(N(C)CC2(CNC(c3ccn(C(F)F)n3)=O)CC2)=O)cc(O)nn1C c1(C(=O)NC)cc(C)nc(NCCCCCNC(C2COCCO2)=O)n1 CC1C(CNC(N2CC(N(c3n[nH]c(-c4ccccc4)n3)C)C2)=O)CCN1C c1(C(N2CC(C(NOCC(=O)OC)=O)OCC2)=O)ccc(C)c(OC)c1 N1(C(COCC)=O)CCCC2(NC(C3COCCC3(F)F)=O)CCCC12 C1(CC)CC(O)CN1C(C1COCC1NC(=O)Cn1ccc(C)n1)=O c1(C(=O)NC2CC(F)(CNC(C(C(C)(C)C)OC)=O)C2)cncc2nc(O)[nH]c12 Cc1cc(CC(N2CCCC(C)C2CNC(=O)C(O)C(C)C)=O)cc(C)c1 Cn1ncc(C(=O)NC2C3CC4CN(C(C5CC(O)C5)=O)C2C4C3)c1S(C)(=O)=O N1(C(C2CCN(C(CC)=O)C2)=O)CC(NC(=O)C(CC)CC)CC1(C)C.C(CN)O C1(C)(CC)CC(NC(=O)C(C)(C)NC(c2cnc(C)o2)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CC(C2CCN(C(c3ccc(C)s3)=O)C2)C1 C=CC1(C(N2CCCC(C(N3CC(N(C)C)C(C)C3)=O)C2)=O)CCOCC1 C12(C(=O)NCCN(C(CSCC(=O)OC)=O)C(C)C)CCC(C(F)(F)F)(CC1)C2 Cc1cc(=NCCOc2ncccc2Cl)[nH]c(=NCC2COCCO2)[nH]1 c1(OC(C(CC=C)(F)F)=O)ccc2cc(O[Si](C)(C)C(C)(C)C)ccc2c1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2nc(C)cs2)c1O c1(CC(=O)NC2CN(C(CCNS(CC)(=O)=O)=O)C(C)C2)nnc2n1CCCC2 c1(NC(C)=O)ccc(C(N2CCCC(NC(c3ccc(C)nc3)=O)C2)=O)c(Cl)c1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)(C)C)ccc([N+](=O)[O-])cc1Br CC1(CO)CC1(C)OC1CCCCC1 N1(C(c2cc(C(C)(C)C)[nH]n2)C(=O)Nc2ccccc2Cl)CC(CO)C(C)(C)C1 N1(C(C(CC)F)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(c2cn[nH]c2)C1 N1(C(CC2(C(=C)F)CCC2)=O)CCC2(CCC2)CC1CO C1(O)(C(=O)NCCC(CCNC(C(CC=C)CC)=O)C)CN2CCC1CC2 Cc1ccc(C(N2CC(F)(C(=O)N(C)Cc3ccncc3F)C2)=O)cc1C#N N1(C(C2OCC(C)C2)=O)CCn2ncc(CNC(C3CCSC(C)C3)=O)c2C1 C1(N(C(c2ccc(C)s2)=O)CCO)CCN(C(c2nccn2C(C)(C)C)=O)CC1 Cc1nc(CC(N2CCCCC2CCCNC(=O)C=Cc2cncs2)=O)[nH]c1C c1(CC(N2CC(C)CC(CNC(C(CC)=CC)=O)C2)=O)coc2ccc(C)cc12 c1(N(c2c(C(C)=O)cccn2)Cc2ccncc2)ccc(COC)c(F)c1 C=CCC(CNC(c1cnnc(C)c1C)=O)C(=O)NCC1(C(C)(F)F)CC1 N=c1nc2c(C(=O)NCCNC(c3cncc([N+](=O)[O-])c3)=O)cccn2[nH]1 c1(C(N2C3CCC2CC(NC(C24CC5CC2C4C5)=O)C3)=O)cccc2occc12 C1(C(=O)OC2CC(C)OC2=O)COC2COCC2O1 C1(CC(=O)NCCCNC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCCOC1 c1(C(=O)OC)[nH]c2nccnc2c1NC(=O)NC(C)(C)Cc1ccc(C)cn1 CC(C)CC(C)C(=O)C(C)(C)C.c12ccc(Br)c(n1)NS2 CC1C(C(N2CCN(C(c3n[nH]cc3C(F)(F)F)=O)CC2)=O)CCN1C Cc1cn2ccc(C(=O)NCC(C(C)C)NC(=O)CNC(=O)C(F)(F)F)cc2n1 n1(CC(=O)NC(C)CCCCNC(c2cnns2)=O)nnc2ccccc2c1=O c1(CC)ccc(-c2nc(C(N3CCC3C)=O)cs2)cc1 Cc1nc(CC(N2CCC2CNC(=O)C(N2CCOC2=O)C)=O)n[nH]1 C1(CCC)(NC(=O)C(CC)N(C)C)CCCN(C(=O)CSCC(F)(F)F)C1 CN(NC(=O)Oc1ccccc1)C(=O)c1coc(C(F)(F)F)n1 c1(CC)nc(O)c(C(=O)N(C)CCNC(c2csc(C(C)OC)n2)=O)cc1C#N CC(C)CC(C)CC(C)OC(c1cccc(N2CCCC2=O)c1)=O C#CC1CN(C(C2CC2C2CCCC2)=O)CCN1C(c1cnn(C)c(=O)c1)=O c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(C)(O)C2CC2)C(C)(C)C)c1 c1(CC)c(C(=O)NC(C)C(C)NC(c2cnc(SC)s2)=O)[nH]c(C)c1C(C)=O N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCC2)C(CNC(c2cc(C)c[nH]2)=O)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2c(C)cc(C)oc2=O)=O)CC(O)C1 c1(C(CC(=O)OC)NC(=O)C(C)(C)OC)ccc(OC(F)F)c(OC)c1 C1(CCCC)CN(C(=O)CC2CCCC(C)(C)O2)CCN1C(=O)CCSCC c1(N2C(C(C)C)CN(C(C3CNCCC3O)=O)CC2)nccc(S(C)(=O)=O)n1 C(=O)(CCC1=CCCCC1)N(C)CC1(O)CCN(C(CS(=O)(=O)NC)=O)C1 CCC(C)CCCC(=O)NC1CCCC(NC(c2cnn(C3CC3)c2)=O)C1 c1(CCC(=O)NC(CC=C)CNC(C2(n3ccnn3)CC2)=O)ncccc1C n1(CCC)nc(C)cc1C(=O)NCC(C)(C)NC(=O)C(c1cncc(F)c1)C CC1CN(C(=O)C2=CC(C)(C)C2)CC(CCNC(c2cccc(C#N)c2)=O)O1 c1(C(N2CC(CC=C)(NC(=O)CC3(C)CC3)C2)=O)ccc(Cl)cc1Cl CC#CCC(C(=O)NC(CO)CCO)NC(=O)CC1CCOCC1 CCC(F)(F)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC1C CC(C(C)(C)CN(C)C)NC(=O)NCc1ccco1.c12ccc(nc1)[nH]c2=O C1(C(=O)NC2CC(C(C)NC(=O)Cn3cccc3)C2)CC2(C1)OCCO2 Cc1c(C(=O)NC2(C)CC(NC(C3CCC=CCCC3)=O)C2)cccc1O c1(NC(C2N(C(Cc3scc(C)c3)=O)CCC2(C)C)=O)ccc2ncccc2c1 c1(OCC(N2CC(CNC(C3CC(=C)C3)=O)C(O)C2)=O)cc(Br)ccc1F CC1=C(C)CC(C(=O)NCC(O)CC(=O)NCC2(CO)CCCO2)CC1 C1(CC=C)(NC(c2cc(C3CC3)oc2C2CC2)=O)CCN(C(C2CC2C)=O)CC1 c1(C(N2C(C(=O)Nc3cccc(OC)c3I)CC(C)C2)=O)cc(F)c(C)c(F)c1 c1(SC)ccc(C(=O)NCC(C2CCC2)NC(c2ccnn2CCF)=O)s1 CCC(C)C(O)C(=O)NC1(C(=O)NCC(=O)N2CCCO2)CC(F)C1 C1(C(N2CCN(C(C(c3ccccc3)C)=O)CC2)=O)CCC(=C(F)F)CC1 N1(C(C(C)N(C)C(c2cccnn2)=O)=O)CC(O)(C(F)F)C1 C(CN=c1[nH]c(N(CC(C)CO)C)nc2c1CSC2)(C(F)(F)F)OC C1(C(N(CCNC(C2(C(CC)=O)CC2)=O)C)=O)CC=CCC1 CS(=O)(=O)C1CC(NC(C2CCC(NC(c3ccncc3O)=O)CC2)=O)C1 C1(NC(=O)CC2CCOCC2)CN(C(=O)CC2CCCC2)CCC12CCC2 c1(C(=O)NCC(CNC(C2(C(N)=O)CC2)=O)F)ccc(C#CC2CC2)cc1 Cc1cc(C)n(C)c(=O)c1CNC(=O)NCC1CCC(C(N)=O)O1 Cc1cc(C(N2CCN(CC3CN(C(=O)C(C#N)C4CC4)C3)CC2)=O)oc1Br C1(C(N2CCC(C(F)F)(CNC(C3(Cl)CC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2(C3N(C(C(CC)SC)=O)CCCC3)CC2)cc(N)ccc1C CN1CCOC(C(=O)NCC(CO)NC(=O)CCc2cncnc2)C1 Cc1cc(CNC(c2cn(C3CC3)cn2)=O)oc1C(=O)NCCC1CCCO1 N1(C(C=C(C)Cl)=O)CCC2CN(C(C34CCCN(CCC3)C4)=O)CC12 c1(C(=O)NCC2C(NC(C(CC)NC(N)=O)=O)C2)oc(C)nc1C C(=O)(CC1=CCN(C)CC1)N1CCC(NC(c2c(C)cccc2O)=O)CC1C C(=O)(C1=C(Cl)CCCC1)NC(CC(=C)Cl)C(=O)NC1CCCCCC1C C1(NC(c2nccc(C)c2N)=O)CN(C(=O)CCC2(C)CC2)CC12CCOCC2 N12CCC3CC13CC(=O)OCCC(CCn1cncn1)OC2=O.CC(C)(C)O c1(NC(C(CCC)OC)=O)ccc(NC(c2ccncc2N)=O)cc1C N1(C(=O)CC2CSC2)CCN(C(c2cccc3c[nH]nc23)=O)C2CCCCC2C1 C=C1CCCN(C(CC2CCC3CC23)C(=O)NCCSC)CC1 n1(CC(=O)NC(CCCCOCCOC(C)=O)C)nc(C(F)F)c2c1CCC2 C(=O)(CC(C(C)C)NC(c1cccc(C)c1C)=O)NCc1n(CC)cnc1 C(=O)(C1CCCc2nncn21)N1C(C)(C)C(NC(=O)CC2CC2)CC1 Cc1cccc(C(=O)NCC2CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)c1 C(=O)(C(F)C(C)CNC(C1CC2(CC(=O)C2)C1)=O)NC(CCC)CO Cc1cncc(C)c1C(=O)NC1CCC1NC(=O)Cc1cccc(Cl)c1Cl CCS(=O)(=O)c1ccccc1C(N1CCC(CO)C(NC(C)=O)C1)=O CC1(C)CCC(CNC(C2CC=CCC2NC(C2(CO)CC(C)(C)C2)=O)=O)O1 C1(C(=O)NCC2CCN(C(C)C)C2)C(C2CC2)CCN1C(=O)C1=CCCOC1 CCCC(CC)CCC(=O)N1CCC(C(N2CCCNC(=O)C2)=O)(CF)C1 c1(OC)ccccc1OC1CN(C(=O)CC(C)(C)C)C1 N1(C(CCC(=O)OC)=O)CC(F)(F)CC1C(=O)NCc1ccc(F)cc1C N1(C(c2c(OCCC)nccc2)=O)CC2CC1CC2NC(=O)C=C(C)C(=O)O Cc1cc(Cl)cc2[nH]c(C(N3CCC(N(C(=O)C4=CCCS4)C)C3)=O)cc12 N1(C(c2sc(CC)c(C)c2)=O)C2CCC1CN(C(C1CCC(COC)C1)=O)C2 N1(C(C2(C)CCOCC2)=O)CC(C2CCCCN(C(C3(C)CC3(F)Cl)=O)C2)C1 C1(NC(C2(CN(C)C)CC2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1F c1(C(=O)NCCC2(CNC(C3(Cl)C(C)(C)C3)=O)CC2)ncn2c1CCC2 c1(C(C(=O)NCC(C)C)N(C)Cc2csc(C(C)C)n2)cc2c(s1)CCOC2 C1(NC(c2n(CC(=C)C)nnn2)c2cncn2C)CC2CC3C(C2)C13 C1(NC(=O)Nc2cnc(Sc3n[nH]c(=NC)s3)nc2)CC2(CCC(CO)CC2)C1 CC1(C)CN(C(C2CC3(CC3)CO2)=O)CC1CC(=O)NOCC1CCCO1 C1(CC=C(C)C)CCCN(C(=O)CCC2CCCC2=O)C1 C(=O)(CC(C(C)C)C(C)C)NC1CCN(C(c2c(C(C)=O)cncc2)=O)CC1 C=CC(C)CC(=O)NCCCC(C)NC(c1cn(-c2cccc(Cl)c2)nn1)=O C1(NC(c2ccccc2)CC)CCN(c2ccncn2)C1 Cn1cnc(N2CCC(CCNC(=O)CSC3CC3)CC2)cc1=O C1(CNC(Cc2c(C)ocn2)=O)CCCC2CN(C(=O)CCCS(C)(=O)=O)CC12 C(=O)(N=c1cc(COC)n(C)[nH]1)C1CCCN(C(CC(CC)O)=O)C1 c1(NC(=O)NC(c2cccc(OC)c2F)C)nccn2c(C)nnc12 Cc1cc(F)sc1C(N1CCC(N(C)C(C2CC(C(F)(F)F)C2)=O)C1)=O C1(CNC(C(C)N(C)C(c2ccnnc2)=O)=O)CCCC2CC12 C(CCCCCC(=O)N1CCC(CC2CC2)C1)n1cc(-c2cc(OC)ns2)nn1 CCCC(C(=O)N1CCCC1CSC)NC(=O)C(=Cc1ccco1)C N1(C(CN(CCOC)C)=O)CC2CCC(NC(c3cc4ncccc4[nH]3)=O)(C2)C1 c1(C(N2CCC(N(CCC)C(C3CCC(C)CC3)=O)C2)=O)cccc(=O)n1C N1(CCCC(=O)NCC(CNC(C2(C=C)CCC2)=O)F)Cc2ccccc2C1=O C(=O)(CS(=O)C(F)(F)F)NCC(C)(F)CNC(=O)C1=NOCC1 N1(C(C(C)=C(C)OC)=O)CC2(COC(CNC(=O)C(N3CCOCC3)C3CC3)C2)C1 c1(OC)ncnc(NC(c2cc(-c3cncc(C(C)=O)c3)cnc2Cl)=O)c1OC c1(-c2c(C(N3C(C)CCC3C)=O)cc(Cl)cn2)nc2c(s1)CCC2 N1(C(CCCn2cc(CSC)nn2)=O)CC(C)C(O)C1 NS(=O)(=O)CCCCCC(=O)NC1CN(C(=O)CCCc2cnn[nH]2)C1 c1(C(=O)NCC2C(NC(C(CC)O)=O)CCCC2)csc2ncnc(O)c12 FC1(F)CC1C1CCN(c2ncnc(C3CC3)c2Br)CC1 C(=O)(C(F)(CNC(=O)C(C)(C)C(F)(F)F)C(C)C)N1C(CC(C)C)CC1 C(=O)(C(C)(CC)C(F)F)NCC1CCC(NC(CCCC(=O)NCCC)=O)CC1 c1(C(c2n(CCCSCC)nnn2)NC2CCCSC2)ccc(C2CC2)cc1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(c2cnn(C)c2C)=O)C1C c1(CC)ccsc1C(=O)NC1CC1NC(=O)CC(C)C N1(C(Cn2cc(C(C)(C)SC)nn2)=O)CCCC(Cn2cc(CC(C)O)nn2)C1 CC(CC(C)(C)C)C(=O)NC1CC12CCN(C(c1ccc(Cl)cn1)=O)C2 C(CCCCCCCC1CC1)(c1n(C(CC)(C)C)nnn1)NCCCC(C)(F)F CCCCC(C)C(=O)N1CCOC(CN(C)C(c2sc(C)nc2C(C)(C)C)=O)C1 c1(OC)ccc2ccc(=NCCOCc3nn[nH]n3)[nH]c2c1 N1(C(c2n(C(C)C)ccc2)=O)CC(NC(c2c(Cl)csc2Cl)=O)CC(C)(C)C1 N1(C(C2(SC)CC2)=O)CC2(CCC(NC(=O)C(N)=O)CC2)C1 CCCCCC(=O)NC1CC1CNC(=O)C(C)C(=O)OC(C)(C)C C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccccn2)=O)C1 c1(OC)ncccc1C(N1CCCC(C(C)C(=O)NOCCCC2CC2)C1)=O N1(CC(=O)N(C(CC)=O)C2CC2)CC2CC(C1)C2(C)C C=CCC(C(=O)NC1(C)CCCC1NC(C1CC=CC1)=O)NC(C)=O CC1CCCN(CC(=O)NCc2cn(C)nc2-c2ccc(Cl)cc2)CC1 C(=O)(C(C(C)C)C(C)C)NCC(CNC(c1nc(C(=O)OC)sc1)=O)OC Cc1cnccc1C(N1CC2C(CNC(c3cnc[nH]3)=O)C2C1)=O C1(C(=O)NCC(C(=O)NCC2CCC3(CC3)CO2)N(C)C)CCC2CC1C2(C)C N1(C(C(C(C)C)SC)=O)CC2(CCCC(CNC(=O)C(C)Cc3ccco3)O2)C1 c1(NC(CC(CC)NC(=O)COCC2CCCO2)=O)cc(OC)cc(F)c1 c1(OC)ccc(C(N2CCCN(C(C3CCCS3)=O)CC2)=O)cc1[N+](=O)[O-] C1(CCOC)(NC(C=CC=CCC)=O)CCN(C(C2(O)CC(C)(C)C2)=O)C1 N1(C(CC)=O)CCCC(C(=O)NCC2C3CN(C(c4c(C)ncn4O)=O)CC23)C1 CCC(CC(=O)N(C)CCN(C)C(c1cnn(CC(F)(F)F)n1)=O)CC(C)C N1(C(C(CC#C)O)=O)CC2CC(NC(c3cc(C(N)=O)ccn3)=O)C1C2 c1(OCC(=O)NC(CNC(C2CCC(CC)O2)=O)CC)cccc(C)c1C N1(C(c2noc(CC)c2C)=O)CCN(C(=O)C(c2ccccc2Cl)(C)C)CC1C Cc1cc(F)ccc1C(N1CC(N(C)C(C2CC2C)=O)C(C)(C)C1)=O C(=O)(CCCCCCCCCO)N1CCN(C(C(C(C)C)C(F)(F)F)=O)C(C)C1 N1(C(C(C)=CC2CC2)=O)CCCC2(NC(=O)COc3cc(C)ccc3F)CC2C1 CCCCCC(CCCCC)C(=O)NC1CCN(C(=O)CC2=CCN(C)CC2)C1 C1(NC(c2ccc(C#C)o2)=O)CC2(C1)CC(C(=O)NCC1(O)CCC1)C2 C(N=c1cc(C)[nH]c(=NCC2(C)CCOC2)[nH]1)c1c(CC)noc1CC c1(C(C)C)nnc(CCC(=O)NC2(C3CCCN3C(c3cnn[nH]3)=O)CC2)o1 N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CC(NC(c1cc(Cl)sc1Cl)=O)C2 CC1CC(C(=O)N(C2CCN(C(=O)C(c3ccccc3)F)CC2)C)=NO1 c1(C(=O)NCC2CN(C(c3c(CC)n(C)nc3)=O)CC2C)cc(C)c(F)c(C)c1 c1(NC(C2CCCN2CCNC(c2c(CCC)nco2)=O)=O)cccc(C)c1 N1(C(C2C(C)CCC2)=O)CCCN(CCNC(C2(S(C)(=O)=O)CCC2)=O)CC1 N1(CCNC(c2c(CC)cno2)=O)CCCN(C(=O)CC2(C)CCCO2)CC1 C1(NC(C23CC(NC(c4cnn(CC)c4C)=O)(C2)C3)=O)CCCC(O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3CNC(=O)C3)C2)=O)cc(F)cc2nc[nH]c12 Cc1nc(C=CC(=O)NCC(CC(C)C)NC(c2ncn(C)c2C)=O)[nH]c1C N1(CCC(=O)N(C(C)CNC(C2CCC2C(=O)OC(C)(C)C)=O)CC)CCOCC1 N1(C(c2ccc(Br)cc2OC(F)(F)F)=O)CC2(CCCN2C(=O)C#CC2CC2)C1 C1(Nc2c(C)c(NC3CCC(C)(C)C3)ncn2)CCN(CP(C)(C)=O)CC1 N1(CC)CCC(C#N)(CN2Cc3cccc(c3)C2)CC1.C(C)(C1CC1)NC C1(NC(c2nc(Cl)sc2)c2nnnn2Cc2cccs2)CC2CC3C(C2)C13 Cc1ccc(Cl)cc1C(=O)N(C1CN(C(C2(c3ccc(Cl)cc3)CCC2)=O)C1)C CN1CCC(C(=O)NCCc2ocnc2CNC(C2(C(N)=O)CCC2)=O)C1 C1(NC(C2C(C(=O)NCC#C)C2)=O)CCOCC1NC(=O)CC1(C)CCCCC1 Cc1ccc2oc(C(N3CC4(CCN(C(C5CC(F)CN5C)=O)C4)C3)=O)cc2n1 C(=O)(C(F)(F)C(C)O)N(CCC(C(C)C)NC(=O)C(N1CCSCC1)C)C C1(C(N(CC(O)CNC(C2(c3ccccc3)CCC2)=O)C)=O)CC2C=CC1CC2 c1(C(=O)NC(CN(C(COCC(=O)OC)=O)C)C)c(C)cc(C)nc1S N1(C(c2ccn(CC)c2C)=O)CC2(CC(NC(C3CCS(=O)CC3)=O)CO2)C1 CCN=C(NCc1ccc(S(=O)(=O)N2CCCC2)s1)N1CCC2C(C1)C2(F)F C(=O)(CC(C(F)(F)F)NC(c1cccc(OC)n1)=O)NCC(CC(=O)OC)O Cc1cccc(C)c1C1(C(N2CCC(N(C(=O)CC(C)(C)O)C)C2)=O)CC1 Cc1cc2sc(C(=O)NCC(C)CN(C(=O)Cc3c(C)cccc3Cl)C)cc2s1 N1(C(c2ccc(OC)cn2)=O)CCN(C(c2cncc(N)n2)=O)C2CCC12 N1(C(C(F)=CC)=O)CC(C)(C)CC1CNC(C1(c2cccc(Cl)c2F)CC1)=O C1(CNC(C(CC)OC)=O)CCN(C(=O)C(c2c(C)nn(C)c2C)=O)C12CCC2 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CCC(NC(C2(C=C)CCC2)=O)C1 Cc1ccc(Br)c(C(N2CCC(NC(=O)C(F)(F)C3CC3)C(O)C2)=O)c1F c1(-c2nc(COC)nn2-c2ccccc2)cc2scc(Br)c2[nH]1 N1(C(CCCCSC)=O)CC2CCC(C2)c2ccccc21 C1(C)(CNC(c2c(CC)csc2)=O)CN(C(c2cc(OC)nn2C)=O)C(C)(C)C1 C1(CC(=O)OC)COC(C)(C)CN1N(Cc1ccccc1)CCc1ccccc1 C1(COC)(NC(c2cnncc2C)=O)CCN(C(=O)CNC=O)C1 C(=O)(CCCCC(F)F)N1CC2(CC(NC(c3cn(CCOC)nc3C)=O)C2)C1 c1(N2C(C(=O)NC(C(=O)OC)C(C)O)CCC2)nc(C(F)(F)F)c2sccc2n1 C(=O)(CC(C)CNC(=O)CN(C)C(=O)C1CC1)NC1(CC)CCC1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(c3n[nH]cc3Cl)=O)CC1O)C2 C12(NC(Cc3c(C)ncs3)=O)CCOC(CNC(C3CCCS3)=O)(C1)C2 Cc1ncncc1C(N1CC(CNC(c2cc(Br)sn2)=O)CC1C)=O N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC(NC(=O)CCn2cc(Cl)cn2)C1 C(=O)(C(C(C)C)NC(C1CC(O)(CNC(c2ccc(C(N)=O)o2)=O)C1)=O)OC N1(C(C2C(CC)CCCC2)=O)CC2=C(C1)CN(C(=O)CC1CCN(OC)CC1)C2 CC(C)(C)C(C)(C)C(=O)N1CCC(F)(CNC(c2cn3ccnc3s2)=O)CC1 c1(C(C(=O)OC)NC(C2C(C(CC)=O)CCCC2)=O)cc(F)c(F)c(F)c1 c1(OC)ccc2ccccc2c1CCNC(c1cc(CN(C)C)on1)=O N1(C(c2cc(CCC)[nH]n2)=O)CCCC(NC(C2CC23CC3(F)F)=O)C1 C1(NC(C(CCC)C)=O)CN(C(c2cnncc2O)=O)CCC12CCOCC2 Cc1cc(CC(=O)NC2CC(CNC(C3CCSCC3)=O)C2)n[nH]1 CC1(C)C(CNC(c2nccnc2N)=O)CCN1C(c1ccncc1Br)=O C1(N(C(C2(N3CCCC3C(=O)OC)CC2)=O)CCO)CCCCCC1 c1(C(=O)NC(C2CCN(C(CC(C)O)=O)CC2)C)ccn(CC(F)(F)F)c(=O)c1 c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(O)C2)=O)ccnc2cc(F)cnc12 c1(CNC(c2ccc(Cl)c(Cl)c2)c2cn(C)nc2C2CCC2)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CCN(C(CCC(=C)C)=O)CC2CC)c(O)nnc2c1CCCC2 c1(CC(N2CC(C(C)NC(C=C)=O)C2)=O)nc(-c2ccccc2)oc1C C1(F)(C(=O)NC2CC(CCNC(C=CCCC=C(C)C)=O)C2)CC2(CCC2)C1 C1(CC)C(C(N2CC(C=C)(CO)C2)=O)CCN1C(=O)CNC(=O)C(C)CC N(C(=NCCCCl)NCCc1ccccc1)C1CCCC(CC)C1 Cc1nc2c(-c3cn(-c4cc5n(n4)CCC5)nn3)cccc2o1 C(=O)(C(C)CCC(C)(C)C)N1CC2(N(C(CC3(COC)CC3)=O)CCC2)C1 c1(C(N2C(CN(C)C(c3coc(Cl)c3)=O)CCC2)=O)nn(C)cc1Cl N1(C(C(CC)(F)F)=O)CCC(CO)(CNC(=O)CC2(O)CCCCCC2)CC1 C1(CC(=O)NC(C2CCOCC2)C#C)CC(NC(=O)C=CCCC)C1(C)C N1(C(c2c(CC)scc2)=O)CC2CCC1C2NC(=O)C(C)SC(F)(F)F C(C(CC(C)C)C(=O)N1CC(F)(C(=O)NCC2(CO)CCCCC2)C1)OC c1(C(N2CC3C(NC(C4C5COCC45)=O)C3C2)=O)cccc(S(=O)(=O)C(F)F)c1 c1(C(=O)NCC2(C(=O)OCC)CCCC2)ccc(=O)n(C)n1.c1csc(C=O)n1 C1(O)(CNC(C=Cc2ccc(C(N(C)C)=O)cc2)=O)CCC(F)(F)CC1 C1(CC(=O)NC)CCN(C(=O)NCC(O)CN2CCOCC2)C1 N1(C(c2cnc(CC)s2)=O)CCN(C(C2CC(C(C)C)C2)=O)C2(CCC2)C1 N1(C(c2c(SC)snn2)=O)CCCC(O)(CNC(=O)C(F)C(C)C)C1 c1(CCC(=O)NCC(C)NC(c2c(Cl)cc(C)nc2)=O)n[nH]c2c1CCCC2 N1(C(CCCC#C)=O)CC(CC(=O)N(C2CCN(C)C2)C)CC1(C)C c1(-c2cc(C(=O)NCC(C)NC(=O)C(O)C3CCCC3)no2)ccccc1Br N1(C(CC(C)(C)C)=O)CC2CCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2C1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(=O)C1=CCN(C)C1 c1(C(N2C(C)CC(CNC(c3scnc3Cl)=O)C2)=O)cc(OC(F)F)cc(F)c1 C#CCC(C)(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cccc(C)c2)C1 c1(C(N2CCC(C(CNC(C=C(CC)C)=O)F)CC2)=O)cccc2c1ccn2C N1(C(C(CCN(C)C)O)=O)CCC2CN(C(c3nocc3Cl)=O)CCC12 C1(NC(C(CC)Cc2ccc(N)cc2)=O)CCCN(C(=O)C(CC)N(C)C)C1C CC(C)C(CCNC(=O)Cc1csc(CCC(F)(F)F)n1)NC(=O)CC(C)(C)C C1(CC(=O)NCCc2cccc(C)c2)CN(C(=O)C(C)C(F)F)C(C)(C)C1 N1(C(C(CC)COC)=O)CCN(C(=O)C2=NOCC2)C(C(C)(C)C)C1 N1(CC(=O)NCCC)CCC(CC(=O)NCC(c2cnn(C)c2)(C)O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCN(C)CC1CNC(=O)CCc1nc(C)cs1 N1(C(c2c(C)cccc2C)=O)CC(CNC(C2(C#N)CCCC2)=O)C2(CCC2)C1 N1(C(CC)=O)CCc2cc(C(N3CCC3CNC(=O)CC(C)SC)=O)ccc21 C(=O)(C1CCCc2ncccc21)N1C(CNC(C(C)CCO)=O)CC(F)(F)C1 Cc1[nH]nc2c1CCC(C(=O)NCC=C1CCN(C(=O)C(C)(C)C3CC3)CC1)C2 N1(C(C2N=C(C)SC2)=O)CCC2(CCN(C(=O)CC3CCCC(=O)N3)C2)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCN(C(=O)CC2CCN(C)C2)CC1 CCCS(=O)(=O)CC(=O)N1CCCC1CN(C)C(c1cnc(C2CC2)s1)=O n1(CC(=O)NC(CC)CNC(C2COC(=O)N2)=O)cc(S(N)(=O)=O)cn1 C1(NC(c2[nH]cc(CC)c2)=O)CCC(C)(CNC(=O)C=Cc2sccc2C)CC1 c1(NC(=O)OCC)ccc(C(=O)NC(CNC(=O)CNC(N)=O)CC(C)C)c(F)c1 c1(N(C)CCF)nc(N(C)Cc2csc(C(F)(F)F)n2)c2c(n1)COC2 N1(C(Cc2ccc(C)s2)=O)CC2CC2(NC(c2cnnn2C)=O)C1 c1(C(=O)NCC(C)(CNC(C2CCCOC2C)=O)OC)nccc2ncccc12 C(=O)(CC(C(F)(F)F)OC)NCC1CC(NC(C(C=C)OC)=O)CC1O c1(C(N2CC(CNC(CSCC#C)=O)C(O)C2)=O)ccc(N)c(Cl)c1 C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O N1(c2nc(OCC)c(C)cn2)CCC2(CCCN(C(c3cnns3)=O)C2)C1 C12(C(=O)NCCN(C(C)(C)C(=O)OC)CCC)CCC(C#N)(CC1)CC2 CC(C)CCCC(C)C(=O)NCC1(CC(=O)N(C)CC2CC2C)CC1 c1(C(=O)NC2CCCN(c3nc(SC)nc(C)c3)C2C)sc2cncn2c1C C1(CC)CCN(C(=O)CC2CCCNC2=O)C(CNCc2ccc(OC)nc2)C1 C1(=CC(=O)NC2CN(C(=O)COC3C#CCCCCC3)C2)CN2CCC1CC2 C1(CNC(CCN(CCC)C)=O)CC(C(C)C)CCN1C(=O)C(CC)NC(C)=O O=S(CCNc1nccc(=NCc2cnn[nH]2)[nH]1)CC(F)(F)F c1(CC(=O)OC)nc(CNCC2CCCC2O)cs1 CC1(C)CCCOC1C(N1CCCC(CCNC(C2CCC=CCCC2)=O)C1)=O c1(C(N2CCCC(O)(CNC(c3c(C)nncc3)=O)C2)=O)cc(C#N)ccc1O c1(-c2ccc(CNS(CC(=O)OCC)(=O)=O)cn2)cc2c(F)cccc2o1 C1(C(N2CCC(CC(=O)NC(C3CCOC3)C)CC2)=O)CCC(C2CC2)C1 C12(Cn3cc(C4CN(C(C5CCC(=O)NC5)=O)C4)nn3)CCC(CC1)OC2 Cc1coc(C(=O)N(C)CC2CCCN2C(=O)Cc2cccc(C(N)=O)c2)c1C N1(C(C(CC)C)=O)CCCC(CCCCNC(=O)Cc2ccc(C(C)=O)cc2)C1 C(=O)(C(O)C(C(C)C)OC(C)=O)N1CC2C(C(=O)NC3CCCC(OC)C3)C2C1 Cc1cnc(NC2CCC(NC(=O)CC3CCCC3(F)F)CC2)nc1C c1(C(N2CC(O)(C(C(=O)NC(CCC)CC)F)C2)=O)cncc2[nH]ccc12 C(=O)(CC1CC(=O)c2ccccc21)N1CCN(C(CCC(=C)C)=O)CC1CCO c1(N(C2(C#N)CCNC2)C(C=CC(C)C)=O)ncnc2cccc(F)c12 c1(C(=O)NC(C2CCCN(C(=O)CNC(=O)C(C)(C)C)C2)C)cccc(Cl)c1Cl n1(CC)ccnc1C(=O)NCc1ccoc1C(=O)NC(C)CSC N1(C(C2CCCN(C(C3CC(O)(CC#C)C3)=O)C2)=O)CCOC(C)(C)C1C N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(O)CCC1C(=O)NCC1(CCCCO)CC1 C1(CNC(C2N(CC)CCC2)=O)CCC(C)(C)CN1C(c1cc(O)cc(O)n1)=O C(=O)(CCCCc1ccccc1)OCCC(=O)NCC(=C)C(=O)OC CCCCN=C(NCC1CC(F)C1)N1CCC2(CC(C(F)F)=NO2)C1 CC(F)(F)CCCC(=O)Nc1ccc(N)c(OCC(=O)NC2CCCC2)c1 N1(C(c2c(C)coc2)=O)CC(OC)C(CNC(=O)CC2(n3ccnc3)CC2)C1 c1(C(=C2CCN(C)C2)C(=O)NC2CC(F)(CNC(CCOC)=O)C2)ccccc1 Nc1nc(Br)ccc1C(=O)NCC1CCN(C(=O)CN2CC=CC2)CC1O C(CN=c1[nH]ncs1)C(=O)N1CC(n2cc(C3CCCC3)nn2)CO1 N1(C(COC2(C#C)COC2)=O)CC2CCC2(CC(N2CC(C(=O)N(C)C)C2)=O)C1 N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2cc(CC)no2)=O)C(C)C1 c1(C(=O)OCC(C(=O)OCC)C)ccc(F)c(F)c1N c1(OC)ccc(S(=O)(=O)N(C)C)c(NC(C2CC(=O)C2C(C)(C)C)=O)c1 N1(C(C=CC)=O)CC2(CCCCN(C(C3CCOC(C)(C)C3)=O)C2)C1 N1(C(C(C2CCN(C(C3CCCN(C)C3)=O)CC2)C)=O)CCC2COCC2C1 N1(C(C2N(C(CNC(CCC)=O)=O)CC(C)C2)=O)CCC(O)C(O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCCC2(NC(C3CCCC(C)O3)=O)CC2C1 c1(N2CCN(C(c3ccc(C)cc3O)=O)C3C2C3)ncc2[nH]ccc2n1 CCC(CC)(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1c1ccccc1F)OC C(=O)(C1CC(=O)Nc2ccccc21)NCC(C)NC(c1ccc(CCO)cc1)=O CN1CC(C(=O)NCCOCCNC(c2cnc(O)n2C)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1cc2sc(=NC(C)CC(C)C(F)F)[nH]c2cc1Cl)N1CCC(CC)C1 c1(C(=O)NC2C(C)N(C(C3CCC3(F)F)=O)CC2)cc2c(s1)CCOC2 c1(-c2cc(C(N3CCC(CCC(=O)OC)C3)=O)sc2)cncc(F)c1 C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CCN2CCCCC2=O)C1(C)C Cc1nc2cccc(C(=O)NC(C)CC(C)NC(=O)CN3CC(C)(C)C3)n2n1 C1(C(=O)NCC(C)OC(F)F)CCC(C)N(C(=O)C(C)c2ccco2)C1 n1(CC)cc(CCNC(=O)C(c2cccs2)NC(C2CCC(=O)O2)=O)cn1 Cc1cc(CN(C)C(C2CC(CCNC(=O)C(C)CN(C)C)C2)=O)nn1C c1(C(N2CC3CC(NC(C(COC)(C)O)=O)C3C2)=O)ccc(C)c2ncccc12 N1(C(C(CCC)(C)O)=O)CCCC2(NC(C3CCc4ccccc4C3)=O)CC2C1 c1(OC)ccnc(C(N2CC(NC(C3(C)CCN(C)C3=O)=O)C(C)C2)=O)c1OC Cc1cc(C=CC(N2CCOC(c3ncno3)C2)=O)ccc1F CCCCCCC(=O)NC1CCN(C(=O)C(C2CCCCC2)OC)CC1O c1(N2CCC(CCC)C2)cc(C(=O)OC)nc(C)c1 CC1(C)C2CCC1(CS(N1CC3C(C1)N3c1cc(C3CC3)ncn1)(=O)=O)C(=O)C2 c1(C(N(C(CCNC(C2(CCOC)CCC2)=O)C)C)=O)csc(C(F)F)n1 N1(C(C2C(C)OCC2)Cn2cnnc2)CCc2nnc(-c3ccncc3)cc2C1 C1(CCCNC(N(CCC)C)=O)CNCCO1 N1(C(c2ccc(CC)cn2)=O)CC(C)CCC1CNC(=O)CC1(CO)CC1 C(=O)(C(C)(C)C(N)=O)NCC(CC)NC(=O)C(CC(C)C)N(C)C Cc1ncc(C(N2CC3C(NC(=O)C(C)N(C)C)C3C2)=O)cn1 Cn1ncc2cc(C(N3CCC(CNC(=O)COCC(F)F)C34CCC4)=O)sc12 c1(C(=O)NC2CC(C(=O)NCC3CCC(C)C3)CC2O)cnn(C)c1C#N C1(C(=O)NC(CC2CCN(C(C(COC)C)=O)CC2)C)CCCC12CCOCC2 C1(NC(C(C=CC)O)=O)C2CC3C1C3C2C(=O)NCC=CC=CC C1(C(=O)NC(CC(C)NC(C2CCCOCC2)=O)C)CC2CCC1CC2 c1(C(C)NC(N2CC(c3ccc(C)cc3)(O)C2)=O)ccc(F)c(F)c1 C(=O)(C(CC(C)C)C(C)C)N1CCC(CC#C)(C(N2CCC(C3CC3)C2)=O)C1 N1(C(C(c2cncnc2)C)=O)CC2CCC1C(CNC(c1cnc(N)cn1)=O)C2 C1(NC(C2COCCOC2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 N1CC2CCCC(C(=O)O)(C1)C2(F)F.c1(OC(C)C(=O)O)ccccc1CCC c1(OC)cc(S(C)(=O)=O)ccc1NC(C1CSCCN1C(c1cscc1C)=O)=O N1(C(C(C)OC)=O)CCC(NC(c2cnn(-c3ccccc3)c2)=O)C1C(C)C N1(C(C(CN(C)C)(F)F)=O)CCC2(CCCN2C(=O)CC2CCNC(=O)C2)C1 C(C(CO)(CO)NC(=O)CN1CCCC1C)N(C(c1cn(CC=C)nc1)=O)C Cc1nc(C(N2CCSCC2CCNC(C2OCC2(C)C)=O)=O)nn1C c1(CCC(=O)NC2CN(C(C=CCC)=O)CC(O)C2)c[nH]c2cc(C)ccc12 N1(CC(C2CCCC2)OC)CCC(C(=O)NC2CCCCC2)C1 C1(O)(CNC(C2(C#N)CC2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)C1 CC1CC2CN(C(C3CCCCN3C(c3cnn(C)c3)=O)=O)CC2N1S(C)(=O)=O c1(CC)ccccc1C(N1CCC(O)C1CN1CCC(CC2CCC2)C1)=O N1(C(C2C(C=C)OCCC2)=O)CC(CNC(=O)CCOCC2CC2)CC(C)(C)C1 N1(C(c2c(C)c(C#N)[nH]c2)=O)CC2(CCCC2)C1C(=O)NCc1cnns1 CC1CCCN1CC(=O)NCCNC(C1CN(C(C2CCN2C(N)=O)=O)C1)=O CN1CCC(C(F)(F)F)(NC(C2CCN2C(=O)CCc2ccccc2)=O)C1 n1(CC)c(CSc2cnc(C(c3ccccc3)O)s2)nc2cc(Cl)ccc12 N1(C(C(C)C#N)=O)CCN(CCNC(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCC(=C)CCNC(=O)C(C)(C)C#N)cc2cc(OC)ccc2n1C N1(C(=O)CSc2nncs2)CCCC1C1(NC(=O)C(O)Cc2ccccc2)CC1 N1(C(CC2CC(N(C)C)C2)=O)CCCCC(C(=O)NCC(N2CC=CC2)=O)C1 CC1(C#CC(=O)NC2CN(C(=O)Cn3ccc(C(F)(F)F)n3)C(C)(C)C2)COC1 C1(CNC(c2cn(CCO)nn2)=O)CCC2CN(C(=O)C=Cc3cc[nH]n3)CC12 CCC(C)(C(=O)NCC1CN(C(=O)Cc2ccn(C(F)F)n2)CCN1C)C(N)=O c1(C(N(C(C)C)CCNC(C2CCCCNC2=O)=O)=O)nccc2c1CNC2=O C1(NC(CSC)=O)CN(C(c2cccnc2-n2nccn2)=O)CC1N=[N+]=[N-] N1(C(c2cc(OC)no2)=O)CCN(C(=O)C(C)NC(N)=O)C(C)C1C c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)cccc2nn[nH]c12 C1(CNC(C(C)Sc2nnnn2C2CC2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 c1(C(N2CCC(CC=C)(NC(=O)C(C)O)C2)=O)nc(Br)c2c(F)cccn12 C1(NC(C2CCC(NC(C=C3CCC(C)CC3)=O)CC2)=O)CCCCC12CC2 C1(N(C(CCNC(COC)=O)=O)C)CN(C(c2cnc(C(C)C)s2)=O)CC1F N1(C(Cn2ccc(C)c2)=O)CC(NC(C2CCC(=O)NC2)=O)C(C(F)F)C1 O=Cc1cccc(CN2C(C(=O)Nc3cccc(C(F)(F)F)c3)CC3CC23)c1Br C1(F)(CNC(CC2CCC(=O)N2)=O)CCCN(C(=O)Cc2ccncc2Cl)C1 N1(C(C2C(C)(C)CCN2C(=O)CC#N)=O)CCC(C)(O)C(O)C1 Cc1nc(C(C)C)oc1C(=O)NC12COC(CNC(c3coc(Cl)n3)=O)(C1)C2 N1(C(c2c(CC)ncs2)=O)CCN(C(=O)CCCC2CCCC(=O)N2)C(CC)C1 C12(C(=O)NC3CC(N(C)C)C3)CC(n3cc(C4CCCC4O)nn3)C1C2 Cc1cn2ccc(C(=O)NC3(CO)CN(C(C4CC5CCC5C4)=O)C3)cc2n1 c1(CC)onc(C(=O)NC2(C)CN(C(c3cc(C4CC4)ccn3)=O)C2)c1C c1(CN(C(C=CC(C)NC(c2ncoc2C2CC2)=O)=O)C)cccnc1O c1(C(c2n(CC=C)nnn2)NCc2cnc(CC)s2)ccc2c(n1)CCC2 c1(C(=O)NC(C(C)(C)NC(CCCc2scc(C)n2)=O)C)cc(Cl)cc(C)c1C C1(CC(=O)OCC)CCC(C(N2CCC(NCCCN(C)C(C)C)C2)=O)CC1 c1(CNC(C(c2cnn(C)c2)NC(c2c(C)cccc2)C)=O)ncc(F)cc1F c1(C(=O)NC(CNC(CCCOCC=C)=O)CCOC)ccc(C)c([N+](=O)[O-])c1 c1(CNC(C23CC(n4cc(CN5CCCC5)nn4)C2C3)=O)cccc(C(=O)O)c1 Cc1cccc(C(C)C(=O)NCCOCCN(C)C(c2nc(Cl)c(Cl)s2)=O)c1 C1(C(=O)NC(C=C)C2CCC2)CC1C1CN(C(=O)CN=[N+]=[N-])C1 C(=O)(C1Cc2c(Cl)cccc21)NCCN(C(CC(CC)C1CC1)=O)CCOC c1(C2(C(=O)NCCC(=O)NCC=CCSC)CC2)ccncc1 Cn1nc2c(c1C(=O)NCc1ccc(Br)c(F)n1)CCCC2 CC1CN(C(c2cnccc2C(F)F)=O)CCC1CNC(=O)C=CCN1CCC1 c1(-c2c(C(=O)OCc3n(C)ncc3)csc2)ccc(Cl)cc1 Cc1nn(CC(=O)NC2CC3CCC2N3C(=O)C(C#N)C(C)(C)C)cc1[N+](=O)[O-] Cc1ccc2c[nH]nc2c1NC(C1CCCN(C(=O)Cc2cc(Br)cs2)C1)=O C1(O)(CNC(C2C(C=C)C2)=O)CCCN(C(c2ccc(N)cc2OC)=O)C1 C1(N(C)C(c2ccnn2CC#N)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(C(CC(F)F)Nc1nccnc1N)NCC(C)C CCC(C#N)C(=O)NC1C=CCC(C(=O)NC2(C(C)O)CC2)C1 c1(C(=O)NCCCNC(C(CC(=O)OC)(C)C)=O)cncc2c1CCNC2=O S(=O)(=O)(c1ccc(NCC2CCC(C(C)(C)C)CC2)c(Br)c1)N1CC(C)C(O)C1 Cc1cc(C(=O)NCC2CCN2CC=C(Cl)Cl)sc1C C1(NC(C(C)=C2CCCC2)=O)CC(F)CN(C(c2cnc(S)n2C)=O)C1 C(C(C(=O)N1CC(F)(CF)C1)n1cc(C2CC2)nn1)OCC.c12cc(no1)OC2 N1(C(c2c(CNC(=O)CCC3CC3(F)F)n[nH]c2)=O)CC23CCC2(COC3)C1 c1(CC(=O)NC2CC3(C2)CC3NC(c2cnn(C3CCC3)c2)=O)ncncc1Cl CC(C)CC(C)C(=O)NC1CN(C(=O)C(O)CCc2ccccc2)CC1C N1(C(C)=O)CC(C)CN(C(c2coc(S(C)(=O)=O)c2)=O)C(C)C1 CCC(CCC(=O)NCCC[Si](C)(C)C)NC(C1C2CCC(F)C12)=O Cc1nn(C)cc1CC(C(=O)O)NC(c1ccc(OC(F)(F)CF)cc1)=O c1(C(=O)NC2(CC(=O)NCc3ccc(Cl)o3)CC2)cnc(CO)cn1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(c2c[nH]nc2C2CC2)=O)CC1 c1(OC)ccc(F)cc1CC(=O)N(CC(O)CNC(C1CCCN1C(C)=O)=O)C c1(C(=O)NC2C(C)CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)ccc2oc(=O)oc2c1 c1(C(=O)NC2CN(C(c3ncsc3C(F)(F)F)=O)C2)ncc2n1CCCC2 c1(C(N2CCN(C(C(C=C=C)C)=O)CC2)=O)ccnc2ccccc12 c1(CC(=O)NC(CC)CNC(=O)CN2CCC(C)C2)cc[nH]c(=N)c1 c1(OC)cc2c(C(=O)N(CCNC(C34CC(C)C3C4)=O)C3CC3)c[nH]c2cc1Cl Cn1cc(C=CC(=O)NCC(C)(C)C(=O)NCCn2ccnn2)cn1 c1(C(=O)NCC2(CCNC(CC(C)C)=O)CC2)cc(F)cc([N+](=O)[O-])c1Br Cc1sc(C(N2CC3CC2(CNC(C2CC(=O)NC2=O)=O)C3)=O)cc1[N+](=O)[O-] C(=O)(C(C)C(=O)OC(C)(C)C)N1CC(OC)(CNC(c2ccc(C(F)F)s2)=O)C1 C1(CC)CN(C(c2ncoc2-c2ccon2)=O)CCC1NC(C1COC(C)C1)=O c1(OC)ccccc1C(=O)NCC1(O)CCN(C(=O)CC2(C)CCOC2)C1 CC1(C)Oc2cc(C(N3CCC(CO)(Cc4ccccc4)CC3)=O)cnc2NC1=O C(CC(CC)C(=O)NC1CC(C)(NC(=O)CCN(C)CC)C1)=CC c1(C(N2CCC(C(C)NC(=O)C(F)=CCCF)CC2)=O)ccc(C#N)cc1F N1(C(C(C)C)=O)CC(O)C(O)C1CNC(C1(CN2CCCC2=O)CCCC1)=O C(=O)(C(Cc1ccccc1)C(C)C)NCCC(C)(C)NC(C1ON=C(CC)C1)=O C(N=c1[nH]c(=N)[nH]c(=NCc2nc(CO)n[nH]2)[nH]1)c1ccc(F)c(C)c1F Cc1cncc(C(=O)NC2CCN(C(c3ccsn3)=O)CC2F)c1C C(=O)(CCS(=O)(=O)CC(C)C)N1CC2(CN(C(C(COC)OC)=O)C2)C(CO)C1 Cc1c(C(N2CCN(CCCNC(C3CCO3)=O)CC2)=O)cnn1CCO c1(OC)ccc(CNC(C2(C)CCCN2Cc2ccc(F)cc2O)=O)c(C)c1C N1(C(c2c(C)ccnc2)=O)CC2(CCC2)CC1C(=O)NC(CO)C(C)(C)CO C(=O)(C1CCCc2nccn21)N(CCCCN(C)C(C1(n2nccn2)CC1)=O)C C1(NC(C(C)OCC)=O)CC2CCCC(C1)N2C(=O)CC(=O)NCC1CC1 Cc1ccc(C(=O)NCC2CCN(CCCN3CCCCC3)C2)cc1 c1(C(=O)NC(C2CCCN2C(c2cnc(C(F)F)s2)=O)C)ccc(CO)o1 c1(CN2CCCC(CCNC(c3cc(C)nn3C)=O)C2)cccc2cc[nH]c12 c1(OC)cc(C(N2CCC(CNC(c3cccc(C)c3)=O)C23CC3)=O)ccc1F c1(C(N2CCC(C)(NC(C(C)NCCCCCC)=O)C2)=O)ccc(C)cc1SC Cc1cc(C(=O)NC(C)CC(C)NC(c2nnn3c2CSCC3)=O)cc(=O)n1C c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ccc(O)c(Br)c3)=O)C2)ccc1Br C#CCCCCCC(=O)NC1CCCC1NC(=O)C(c1ccccc1Cl)(F)F O=C(CC(C(F)F)NC(=O)COCC1(O)CC(O)C1)NC1CCOC1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1)NC C1(C(N2CCC(C(=O)OC)(OC)C2)=O)CC2(CCC2)CN1Cc1ccccc1 c1(CC)cccc2sc(C(N3CCC34CC(NC(=O)OC)C4)=O)nc12 c1(C(=O)NC(CNC(c2cn(C)nn2)=O)CO)cccn(C2CCC2)c1=O c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2)ccc2ccsc2c1 c1(CCCC(=O)NCCN(C(C2C(SC)CCC2)=O)C)cccc(Br)c1 Cn1nc(C(N2CC3CC2C3C(=O)NCC#CC2CC2)=O)cc1C#N c1(N(C(CC(C)C)c2nn[nH]n2)C(N2CCN(C)CC2)=O)ncccc1F CCCCCC(C)(C)C(=O)NC1CCOC(C(=O)N(CCC)CCC)C1 c1(CC(=O)NCC(CC=C)NC(C2CCC3(CCC3)C2)=O)cccc(F)c1OC c1(C(=O)OCC)oc2ccccc2c1CC(c1cc(Cl)ccc1F)(C)C(=O)O C1(C(N(C)CC2CN(C(C3CCC(CO)CC3)=O)CCO2)=O)CCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)NCC3(NC(C45CC(C)C4C5)=O)CC3)ncc2c1 c1(CNC(=O)NC(c2ccc(OCCCC)cc2)C)cc2ccncc2s1 CC1(C)C(NC(=O)COCC2CCCOC2)CCN1C(=O)C=Cc1ccccn1 CC1CCC2N(C1)C2.C12CCC(=O)N1C(=O)C(CC)N(C)c1cc(ncn1)N2 c1(C(N2CC(C(N)=O)(CNC(=O)C(c3cncn3C)O)C2)=O)cccn(O)c1=O N1(C(=O)CSc2cccc(O)c2)CCCN(C(C2CC2c2ccccc2)=O)CC1 c1(NC2CCCN(CCCO)C2)[nH]c(=NCc2ccsc2)nc2sccc12 C1(C(N(CC(C)(C)NC(=O)CCn2cnnn2)C)=O)CCC2(CC2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(C2C=CCC2)=O)C(C)C1 Cc1ccc(N2CCCC2)c(C(=O)NC(C)CNC(c2ccc(=O)oc2)=O)c1 CCCC(C)(O)C(=O)N1CCC(c2ccccc2)(NC(=O)CSC(F)F)C1 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)CCCC)C12CCC2 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(CO)C2(C1)CN(C(=O)CCNC(N)=O)C2 C(C(F)(F)C(=O)NC(C1CCN(C(=O)C(=C2CCCCC2)F)C1)C)OC c1(C(N2CCC(O)(CNC(=O)Cn3cnnn3)C2)=O)cccc2nc(O)ccc12 c1(C(=O)NCC2CCCN(C(C(CCC)CC)=O)C2)cc(C)c(N)cc1Cl c1(CNC(CN(C(=O)CCC(CC)OC)CC#C)=O)cnc(F)cc1C c1(CC(=O)NC2(CNC(C(COC)O)=O)CC2)cccc(C)c1 C=CC(C)(CCOC)C(=O)NCC1CN(C(=O)Cc2cccs2)C2(CCC2)C1 C(C)(CNC(c1ncc(Br)cc1F)=O)(CC(C)C)NC(CSC)=O N1(C(c2cc(C)c(C)s2)=O)CC(CC(=O)NCC(C)(O)C(C)(C)C)CC1(C)C CCC(O)C(F)(F)C(=O)NCC1CCCN1C(C1CC1C(N)=O)=O C(=O)(C1=C(C)CCCC1(C)C)NCC1N(C(C(CC)SC)=O)CCCC1C C(=O)(C1CCCc2ccccc21)NC(C1CN(C(C(F)OC)=O)C1)C c1(C(C)C)ccc(C(=O)NCC2CCN(C(C3(C)CCN(C)C3)=O)C2)nc1 N1(C(C)C(=O)NCC2(NC(c3csc(Cl)c3)=O)CCCC2)CCCC(O)C1 c1(NCC(=O)NCC2(c3ccccc3)CC(NC(C3C(C)=C3)=O)C2)ccc(C)cc1 c1(CC)c(C(=O)NC2CCCC2NC(=O)CCc2ccc(O)nn2)cnn1CC C1(N(C(c2nnc(C)s2)=O)C)CN(C(c2cc(C(C)C)oc2C(C)C)=O)CC1F CCCC(C)(C)CC(=O)N1CCC(C(F)C(=O)N(c2cccc(CC)c2)C)C1 C(=O)(C1=C(Cl)CCOC1)NC1COCCN(C(COCc2c(C)ncs2)=O)C1 c1(C(=O)NCCN(C(=O)CCn2ccnc2C(C)C)CC)ncn(C(C)C)n1 C1(OC(C)(C)C)CC(OCC(=O)NC2CC(Cc3ccccc3)C2(C)C)C1(C)C CCCCC(C)C(=O)N1CCC(C(C)NC(c2cc(CN(C)C)c[nH]2)=O)C1 C(=O)(C1CCc2cccc(=O)n21)NCC=CCNC(CC1(C)OCCO1)=O N1(C(CC(CC)OC)=O)CCC2(NC(c3ccc(SC)cc3Cl)=O)CCCC12 CC1CCc2[nH]c(=NCCCOc3ccccc3F)[nH]c(=NCC(Cl)=CCl)c2C1 CC1(C)CCCc2c1nc(Cl)[nH]c2=NCC1CC(NC(=O)CCS(C)(=O)=O)C1 C1(C(=O)NC(CNC(C2N(C)CCC2)=O)C2CC2)COc2cc(O)ccc2C1 Cc1ncc(CC(=O)NC23CC(NC(=O)COCc4nccn4C)(C2)C3)s1.CC C1(C(=O)NC(C)CCCNC(=O)C(=Cc2c[nH]cn2)F)CC1C1CCOCC1 c1(CNC(N(C2CCCC2(C)C)C)=O)nnc2c(=O)[nH]ccn12 C1(N(C(CSC)=O)CC2CC2)CCCN(C(=O)C(C(C)C)NC(N)=O)C1 n1(CC(=O)NCC(C)(CNC(c2cncc(C)c2)=O)OC)ccccc1=O c1(CC(N2CC(NC(C(n3cnc(C#N)n3)C)=O)C2)=O)ccc(CO)cc1 CC1CC(CNC(c2csc(CO)n2)=O)CN1C(c1nn[nH]c1Cl)=O c1(C(N2C(C(=O)Nc3c(OCC)ncnc3)CC(F)C2)=O)cc(C)ccc1O C1(NC(c2c(C)cncn2)=O)CN(C(c2ccc(C(N)=O)o2)=O)CCC1O c1(-c2n(C(C(C)C)C)nc(CS(C)(=O)=O)n2)cn2c(n1)CCC(C)C2 c1(C(=O)NCC2N(C(c3c(C(C)C)cccc3)=O)CC2)cc2ccccc2n1C Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(C2CC3CCC(C2)C3)=O)C1 CC(C)C(=O)C(=O)N(CC(=O)NC1CC1(C)C)C(C)C S(=O)(=O)(c1ccc(NCCc2ccccn2)cc1Cl)N(CCCCO)C C=C1CCC(C(N2CC(C(C)NC(=O)CC(C)(C3CCC3)N(C)C)C2)=O)CC1 C#Cc1ccc(CC(=O)NCCC(C)(C)CNC(c2c[nH]ccc2=O)=O)c(F)c1 Cc1cccc2oc(N3CC4CC(NC(C5(S(C)(=O)=O)CC5)=O)CC4C3)nc12 N1(C(C2CNC(=O)N2)=O)CCCCC(CNC(c2n[nH]cc2C2CCC2)=O)C1 O=C1CC(C(=O)N2CC(NC(c3ccccc3Cl)=O)CC2CO)=NN1 C1(C(=O)NCCc2c(C(=O)Nc3cc(C)no3)c[nH]n2)CCCCC(=O)N1 c1(C(=O)NC(CNC(C(C)NC(c2cccs2)=O)=O)C)cc2ccccc2[nH]1 C1(C(=O)NCC2N(CC)CC2)(C(C)C)CCCN1C(=O)C=Cc1cscn1 CC1(Cn2cc(CC3CN(C(C4CCCCC4)=O)C3)nn2)CCCC1(F)F N1(C(c2nn(CC)c(O)c2)=O)CCN(C)C(C(=O)NCC2CC23CCC3)C1 c1(OCC)cc(C)c(C(=O)NC2CC(C)N(c3ccnc(CC(C)C)n3)C2)cn1 C1(NC(C(C)OCC=C)=O)CCCC1CNC(=O)CC1CCCN1C(C)C C1(C(N(C(c2ccccn2)C)C2CC2)=O)OCCC1NC(=O)OC(C)(C)C C1(c2ccc(C(=O)OC)cc2)C(n2cc(OCCCN)nn2)CCC(=O)N1C CCCCCS(=O)(=O)CC(=O)NC12CCCC1N(C(=O)Cc1cnc(C)s1)CC2 N1(C(CCN(C(C)=O)C)=O)CCCC(NC(=O)Cc2cccc(F)c2O)CC1 C(=O)(CS(=O)(=O)CCO)NCCC1(O)CCN(C(CCSC)=O)C1 c1(C(N2CC(CCNC(c3cnc(N(C)C)s3)=O)C2)=O)cccc2cncn12 c1(C(N2CCCC2Cc2ccccn2)=O)cnc(-c2ccsc2)s1 CN1CCC(C(=O)NCC2CN(C(N)=O)C2)(NC(=O)CCC2CCOC2)C1 C1(C(=O)NC2COCC2NC(C2CCCN2c2ncccn2)=O)C2CCC1CC2 N1(C(c2nc(-c3cc(OC)ncn3)sc2)=O)CC(OC)CC(c2ccccc2)C1 Cc1c(C(=O)NCCCC2CCCN2C(=O)CC(C)F)sc2ccc(Cl)cc12 c1(CC(=O)NC2C3CN(C(CCCCC)=O)C2C3)cnc2c(C)cccn12 c1(C(=O)NC(C(C)(C)NC(CSCC=C)=O)C)ccc(-c2cccs2)nc1C C1(C2CN(C(C3N=C(C)SC3)=O)C2)CN(C(C2(F)CCCC2)=O)CCO1 C1(C(N2CCCN(C(C=Cc3c(C)n(C)nc3)=O)CC2)=O)CNC(=O)CC1(C)C C(CCCCCN(C)C(c1ncsc1Br)=O)NC(C1CCC(C)S1)=O Cc1cc(C(N2CC(=C(F)CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)nc1C C=CC(O)(C(=O)NCC(CNC(c1ccc(Cl)cc1)=O)CO)C(F)(F)F C1(CNC(c2cnc(CC)o2)=O)(CO)CCN(C(=O)C(C2CCCCC2)C)C1 C1(C(N(CC)Cc2ccccn2)=O)CCCC1NC(c1cnsc1C)=O c1(SC)cccnc1C(=O)NCC(C)CN(C)C(C1(c2cc[nH]n2)CC1)=O c1(CC(=O)NCC(CN(C(C2SCCS2)=O)CC)(C)C)ccccc1OC(F)F c1(SCC(N2CCCC(N(C(=O)CN(C)C(C)C)CC)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1nc[nH]c1Br)NC(CCC)(N)C(=O)O N1(C(C2(C)CCCC2)=O)C(C(=O)NCCCCN2CCC2)CCC12CC2 CC1CCCC1(C(N1CCC1CN=[N+]=[N-])=O)NC(C1CC(=O)C1)=O c1(OC)ccc(CNC2(c3ccccc3)CC2(F)F)cc1OCC(F)(F)F c1(C(=O)NC2C(NC(C3C(C=C)OCC3)=O)CCC2)nccc2[nH]ccc12 CC#CC1CCN(CCNC(=O)Cc2scnc2C)CC1 Cc1onc(CC(=O)NCCSCC(=O)NC2(C)CCCC2C)c1C#N Cc1cc(Cl)c(Cl)cc1CN1CC2C(NC(c3cc[nH]n3)=O)C2C1 c1(C(C)NC(=O)NC(c2cc(Br)ccn2)CC)ccc(F)c(C)c1 C=CC(CCC)CC(=O)NC(C(=O)NOCCCN(C)C)C1CCCC1 C1(CNC(CCOCCCOC)=O)CC2C=CC1CC2.C12(CC1)C(=O)N2 c1(NCCc2ncn(CC)c2)cc(Cl)c(Br)cc1[N+](=O)[O-] C=CC(C)(O)C(=O)NC1CC(OCC(N2CC(C(C)CC)C2)=O)C1 C1(NC(c2c(CNC(C(C)Cn3cccn3)=O)noc2)=O)CC12CC(O)C2 C12(C(=O)NCc3c(C(=O)OC)n[nH]c3)CCC(C(=O)NCC=CCSC)(CC1)C2 C1(O)(CC(=O)NCC(C)C(=O)NC2CCNC2)COC(C)(C)C1.C1(C2CC2)CC1 C(C(C(=O)NC(C)CCC1CC1)C(C)(C)C)NC(c1n(CC)ccc1)=O CCCCCC(O)C(=O)NCC1CCN(C(c2ccc3c(c2)NCC3)=O)C(C)C1 c1(C(N2CCCC(N(C)C(c3cc4c(s3)CCC4)=O)C2)=O)cc2cccnc2s1 Cc1ccc(C(=O)NCC2(CN(C)C(C3(CCC4CC4)CC3)=O)CC2)c(O)c1 C(CC(O)CNC(=O)CCOCCCNC(C1CN(C)C1)=O)OC C1(NC(C(C2CC(C)(C)C2)OC)=O)CC(C)(CNC(=O)C=C(C)C(C)C)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1C(C)(C)C1(F)F)NCc1c(C)occ1 c1(C(N2CC3C(C(=O)NC(C#C)C)(C3)C2)=O)ccc(Br)c(OC)c1F c1(CN2CCCC(CCNC(c3c(C)cc(Br)cn3)=O)C2)cccc([N+](=O)[O-])c1 C1(C(N(C)Cc2ncn(C)n2)=O)CN(C(C23C(=O)C4CC2C3C4)=O)CC1(C)C c1(C(C)(C)N(C(=O)CN2CCC(N3CC=CC3)C2)CCC)cc(C)c(C)cc1C C(=O)(CC(C)C(F)F)NCC(CCCC)NC(C1CCCN(CC)C1)=O c1(NC(C2(CCC=C)CN(C(=O)CC3CCC(=O)C3)C2)=O)ccc(OC)cc1C C12(C(=O)NC3CN(C(C(C)CN4CCOCC4)=O)C3)CCCCC1NC(=O)C2 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)(C)CCNC(=O)C=C1CC1 C(=O)(C(COC)C(F)(F)F)NC(C1CC(NC(C(CCC)O)=O)C1)C N1(C(C2(C)CN(C(C=CC3(C)COC3)=O)C2)=O)CCCCC(CC2CC2)C1 Cc1cccc(C(C)(C)C(=O)NC2C3CN(C(C4CC=CCC4)=O)CC23)c1 N1(C(CSC(C)C)=O)CCN(C(C2CCCSC2C)=O)CC(C)C1 c1(C(=O)NCC2(CC(=O)OCC)CCCCC2)ccc2c(n1)OCC(=O)N2 c1(C(=O)NC2CC(F)(CNC(C3(C=C)CCCCC3)=O)C2)c(F)ccc(O)c1F C(=O)(CS(=O)(=O)c1ccccc1F)N(CCNC(C(C)C)=O)Cc1ccccc1 c1(CNC(C=C(CC)C)=O)ccc(C(=O)NCc2cnco2)nc1 c1(OCC)ccc(=NCCOC2CCN(CC)CC2O)[nH]c1 N1(C(=O)C=CSCC2CC2)CCC2C(CCCN2C(=O)C(O)Cc2ccccc2)C1 C1(C)(NC(Cc2nc(COC)sc2)=O)CCN(C(=O)CN2CC=CC2)C1 O=C(C1OCCn2ccnc21)NCC1CCCCN1C(=O)COCC1CCCC1 c1(C(=O)NCC2C3CN(C(c4n(C)nc(Cl)c4)=O)CC32)cnn2ccncc12 C(CCNC(C1(C)CCC(=O)C1)=O)(C(=O)NCCNS(=O)(=O)CC)OC C1(NC(CC(=O)NCC)=O)CCOC12CCN(C(c1cc(Cl)ncc1F)=O)CC2 C1(CNC(CC(CC)O)=O)CCCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(C)NCC2(C)CC2NC(=O)OC(C)(C)C)c(Cl)c([N+](=O)[O-])nn1C N1(C(=O)C=Cc2cn[nH]c2)CCC2(CNC(C3(Br)CC3)=O)CCCCC12 N1(CC(=O)N(CCC)CC2CC2)CCCCC1c1nc(C(C)(C)C)cs1 C(C(C)(O)CC(=O)N1CCC(C(=O)NC2CCCC2C#N)C1C(C)C)OC C1(NC(c2ccn(C)n2)=O)CN(C(c2c(Cl)csc2Cl)=O)CCC1CO CN1CCN(CC(N2CC3(CC(NC(=O)COCc4nccs4)C3)C2)=O)CC1=O c1(C(N(CCNC(C2C(CC)CCN2C(C)=O)=O)C(C)C)=O)ccc(C)cc1F C12(CNC(C3N(C)CCOC3)=O)CC(C1)C(NC(=O)CN1C(=O)CNC1=O)CO2 Cc1cccn2c(C(N3CCN(C(=O)Cc4cnoc4)CC3C(C)C)=O)cnc12 c1(C(=O)NC2CC(C)(CC)N(C(=O)Cc3cc(C)no3)C2)ccc(F)c(N)c1F C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(C(C)SCC)=O)C1 CN1CCCC(CN(C)C(c2c(CNC(=O)CCn3ccnn3)nnn2C)=O)C1 N1(CCCNC(C(C)NC(C2CCC2)=O)=O)CCN(C(C23CC(F)C2C3)=O)CC1 n1(CC)cnc(C(N2CC(C(C)NC(=O)CCn3ccc(C)n3)C2)=O)n1 C(c1cc(Cl)ccc1Cl)=CC(N1CCCC2(NC(c3c(C)onc3)=O)C1C2)=O C=CCCCCC(=O)NC1(C)CCN(C(C2CC23CCSCC3)=O)C1 C=CCC(C)(C)C(=O)NC(C)CN1CCN(C(c2n[nH]cc2OC)=O)CC1 CCC(C)C(C(=O)NC12COC(CNC(=O)CCc3csc(C)n3)(C1)C2)OC c1(C(N2C(C(C)C)C(NC(=O)C=CCO)CC2)=O)cc(=O)c2ccccc2o1 c1(NC(=O)NCC(=C)C)nc(C)c(CC2CCN(C)C2c2ccccc2)s1 Cc1c(C(N2CC(NC(=O)C(C)CF)C2)=O)cnn1C1CCCC1 c1(C(N(C2CCC(NC(=O)C(C)(O)C3CC3)CC2)C)=O)cccc(CF)c1 CC#CC1CCN(C(=O)C(CC2CC2)NC(=O)CN2CCCC2C)C1 C1(CC(=O)NC)CN(C(=O)CC2CCCCO2)CCN1C(c1cc(C)cnc1C)=O C1(NC(C2CN(C)C2)=O)CN(C(c2cncc(-n3cccn3)n2)=O)CC12CCC2 N1(C(C(CCCC)O)=O)CC2CCC(C1)N2c1cc(C)nc(Cl)n1 C1(c2cn(C)nc2)CCCCN1C(=O)NC(c1ccc(Br)cc1)C1CCC1 C1(NC(CC2CC(C(=O)OC)C2)=O)CCCCN(C(c2cc(C)c[nH]2)=O)C1 c1(C(=O)NC(C)CCCNC(C2CCCC(C)C2)=O)cn(C)c(=O)c2cncn12 C1(CNC(=O)CC2CCSCC2)CC2(CCN(C(C34CC(C3)C4)=O)C2)CO1 c1(CC(N2CCC(N(C)C(C3CCCC3)=O)C2)=O)ccc2c(c1)CCCO2 C(C(C(C)(C)C)NC(=O)C(C1CC1)C1CC1)NC(c1c(C)[nH]cc1)=O Cc1c(C(=O)NC(C)CCN(C)C(c2ncccc2O)=O)[nH]ccc1=O N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2C(=O)NCC1(O)CCC1 N1(C(C2N(C(c3c(C)noc3N)=O)C(C)C2)=O)CCN2CCCCC1C2 Cc1[nH]nc2c(C(N3CCC(NC(C4CCCOC4)=O)C(F)C3)=O)cccc12 C(CCCC(=O)NC1(CCNC(=O)CC2COC(C)(C)C2)CCOCC1)N(C)C N(C1CCCc2cccc(C)c21)C(c1c(CCC)n(C)nn1)=O C1(NC(C(CC)N(C)C)=O)CC(C)N(C(c2csc(Cl)c2OC)=O)C1 n1(CCC(=O)NC2CCN(C(C3(C(N)=O)CC3)=O)CC2)ccc2cccnc12 n1(CC)ccc2nc(N3CCC(NC(C4(C#N)CC4)=O)C(O)C3)ncc12 N1(C(C(CC)(CC)CO)=O)CC2(C1)CN(C(=O)CCC(C)OC)CC2CO N1(C(=O)NC(C)C=CCc2ccccc2)CCCN(CC(O)C(F)(F)F)CC1 C(C(=O)NCC1COCCN1C(=O)C(=O)C(C)(C)C)(C(C)(C)C)N(C)C C(=O)(CCCCC(N)=O)N(C1CC2CC1N(C(=O)CCOCC(F)F)C2)C N1(C(C2CC(C)CC(C)C2)=O)CCCC(O)(CNC(=O)CC2(O)CCC2)CC1 C1(CCNC(c2cc(C3CC3)[nH]n2)=O)CN(C(=O)C2=CCSC2)CCS1(=O)=O C1(N(C)C)CCN(C(c2cnc(C(C)(C)C#N)s2)C(=O)NC2CC2)CC1 c1(-c2cc(F)c(C(=O)OCC)c(F)c2)c[nH]c2ccc(Br)cc12 c1(C(N2CCC(NC(c3nc(CC)sc3)=O)C(F)C2)=O)c(C)ccc(C)c1C c1(CCN(C)CCC2CCCN(CCn3cc(I)cn3)C2)nc2ccccc2[nH]1 C(C(O)CN=c1[nH]cc(Br)cc1C#N)NC(c1c(C)sc(O)n1)=O c1(OC)cc(C(=O)NC(C2CCN(C(c3ccccc3F)=O)C2)C)ccc1Cl C(=O)(CCCCCN=[N+]=[N-])NC1CN(C2CN(C(C(CCO)OC)=O)C2)C(=O)C1 N1(C(CCCCC#C)=O)CCCC12CCN(C(=O)C(CO)c1ccccc1)C2 N1(C(CCN(C)CC)=O)CCN(C(=O)CN(C(=O)Cc2ccc(Cl)s2)C)CC1 c1(C(=O)NC2CCC(N(C)C(c3snc(O)c3Cl)=O)C2)ccc2ccnn2c1 c1(CC)ccc(C(=O)N(C)CCNC(=O)C(Cc2ccccc2)OC)c(C)n1 c1(OC)cc(Br)ccc1CN1CCC2(CC1)CC2.C12CC1C(=O)NC2 c1(C(=O)NCC2CN(C(C3C(C)=CCS3)=O)CC2O)cc(C)n(C2CC2)c1C c1(C(C(=O)NCc2scc(CNC(C(C)C3CCC3)=O)n2)(C)C)cccc(F)c1 C1(C)(CNC(C(C)N(C(CCC#C)=O)C2CC2)=O)CCC(=O)N1C C1(NC(C2CC(C)C2)=O)CN(C(c2cc(O)cs2)=O)C2(CCOCC2)C1 c1(NC(CCC)C2CCCC2)ncccc1S(=O)(=O)NCCc1cccc(Cl)c1 N1(C(c2ccc(Cl)cc2C(F)(F)F)=O)CCCN(C(=O)C2CC2)CCC1 c1(CCCC(=O)NCC2C(NC(C(C(C)C)(C)O)=O)C2)ccc2c(c1)CC(=O)N2 CC(C)CC(C)(CNC(=O)CC1CC2CCC1CC2)NC(C12CC(F)(C1)C2)=O Cc1cn2ccc(C(N3CC(NC(c4cc(Cl)cnc4C)=O)C(C)C3)=O)cc2n1 c1(C(=O)OC)ccc(C(N2CCCC(C(C)NC(=O)CSC(C)=O)C2)=O)c(F)c1 C(CCC(=O)NO)NC(C1(CC=C)CN(C(C2CCCCO2)=O)C1)=O c1(C(C)C(=O)NC2CC(c3ccccc3)CO2)ccc(F)c(F)c1 c1(NC(=O)NC(CC)COCc2ccccc2C(F)(F)F)c(C)noc1C(F)F n1(CCC)ncc(C(c2nnnn2C(C)CC)NCC(C)(CC)CC)c1C n1(C(C)C)ccc(=NC(=O)C2(C)CCCN(C(c3ccc4c(c3)CC4)=O)C2)[nH]1 Cc1noc2cc(C(N3CCN(C(=O)CC4CCOC4)CC4(CC4)C3)=O)ccc12 c1(C(N2CCC(NC(C(CCC#C)O)=O)C2)=O)cc(Br)cc(C)c1C c1(C(=O)OCC)ccc2c(n1)CN(C(=O)CCC1CCC(C(N)=O)O1)CC2 c1(C(N(CCNC(Cn2c(C)nnn2)=O)C)=O)ccc(O)c(CO)c1 C(=O)(C(O)C(C)(C)C)N(CC)CC1CCCN1C(c1cccc(CCC#N)c1)=O c1(C(C(F)(F)F)OC(C=CCOC)=O)ccccc1F C(CCCCC(=O)N1CC(COC)(NC(c2cn(C)c(C(F)F)n2)=O)C1)OCC C1(NC(CC(CCC)O)=O)CN(C(c2cc(C(N)=O)no2)=O)CCC1(C)C c1(CN2CCC(C(N(C3CC3)CC)=O)C2)c(C)cc(C)nc1O N1(C(COCC)=O)CCC(C2CC2)C1C(=O)Nc1ccc(C)cc1C C1(OC)COCCC1CC(=O)NCC(C(C)C)NC(C1CCC(=O)O1)=O c1(C(N(C2CCN(C(c3nc(C)n(C)n3)=O)C2)CCC)=O)cc(CO)c(C)o1 N1(C(c2cc(CC)no2)=O)CCN(C(=O)CN(C(=O)C(CC)CC)CC)CC1 N1(N2CCC(n3ncc(C)c3)C2)CCC(c2ccc(Br)cn2)CC1 CC1CN(C(C2CC=CC2)=O)CC1CNC(=O)CCOc1ccc(Cl)cc1 N1(C(C(CC#C)CC#C)=O)CCC2CN(C(=O)CCN(C)CC)CC2C1 CN=c1nc(N2CCCC(CC(=O)OC(C)(C)C)C2)cc(C)[nH]1 C1(CNC(c2c(CC(C)C)onc2)=O)COCCN(C(c2ccc(F)s2)=O)C1 Cc1ccc(C(=O)NCCCCC(C)NC(c2nncs2)=O)c(N=[N+]=[N-])c1 CC(CC(=O)NCC1CC1CNC(=O)C(C)(C)N1CCCC1)N(C)C CCCCCCC(F)C(=O)N1CCCC(CO)(NC(c2cc(Cl)c[nH]2)=O)C1 N1(C(C(C)C(C)O)=O)CC2(COC(CNC(C34C5C6C3C3C4C5C63C)=O)C2)C1 c1(CN2CC3C(NC(c4cnc(C)nc4)=O)C3C2)ccc(Br)cc1O c1(C(CC(=O)O)NC(CC)C(=O)NC(N)=O)cccc(Br)c1 CCC(F)(F)C(C)(C)C(=O)N1CC2CC2(CNC(c2cc(C)nc(C)n2)=O)C1 N1(C(C(CCOC)NC(C(CC#C)O)=O)=O)CC2(COC(C)C2)C1 CC(C(CO)NC(=O)CCC1CCCO1)NC(c1cc(-c2ccccn2)no1)=O N1(C(=O)C=Cc2ccc(F)cc2)CC2CCCCC2(NC(C2CCCS2)=O)C1 C1(CC)(NC(C2CCCC2)=O)CCCN(C(c2ccc(C(F)(F)F)nc2O)=O)C1 C(=O)(C(C(CC)CC)OC)NCC(CNC(c1cc(CC)nnc1C)=O)(C)F C1(N(CC#C)C(C2CC2(C)C)=O)CCN(C(c2ccc(O)nc2)=O)CC1 n1(C(C)(C)C)ncc(I)c1C(=O)NC(c1ccc(Br)cc1)CC(=O)O c1(C(=O)NC23CC(CNC(COC(CC)(C)C)=O)(C2)C3)cnc(O)c(F)c1 C(C(CNC(C1CCCS(=O)(=O)C1)=O)C(F)(F)F)NC(C=CC(=O)N(C)C)=O N1(C(C(C)n2ccnc2)=O)CC2CC(NC(=O)COCc3ccncc3)C(C2)C1 c1(CN2C(CNC(C)=O)CCC2)c(C)n[nH]c1C Cc1ncc(C(=O)N(CCC(C)NC(=O)C(C)C(C)O)C)cc1C#N C1(C(=O)NC2C(C(=O)NCC(N)=O)CCOC2)CCCC12CCC2 C(C)(C(=O)NCC1CCCN1C(c1cn(C2CC2)nn1)=O)(c1cccs1)OC C(=O)(C#CC1CCOC1)NC(C)(C)CCCCNC(=O)CC1(C)CCOC1 C1(c2cn(C(C)CNC(=O)C(C(C)C)n3cnnn3)nn2)(COC)CCOCC1 C1(CC)C(NC(=O)COC(F)(F)C(F)(F)F)CCN1C(C1CCC(OC)C1)=O CCC(C)(C)C(=O)NCCCOC1CCN(C(c2cn(CC3CC3)nn2)=O)CC1 CCC(CCCC(=O)N1CC(CS(C)=O)C1)NC(=O)CCOCCOCC c1(C(=O)NCC2CCN(C(COCc3ccc(C)cc3)=O)C2)cc(N)c(Cl)cn1 C(=O)(C(C)(C)C(=O)N1CCCC(CC(=O)Nc2cc(Cl)ccc2CO)C1)OC CC(CC(C)NC(=O)CC1(C)CC1(F)Cl)NC(=O)Cc1nncs1 C(=O)(C(=O)N=S(C)(C)=O)N(CCN(C(C1CC(C)(C)OCC1)=O)C(C)C)C c1(OC)ccc(C(C)C(=O)N2CCCn3cc(nn3)C2)cc1.C1(CO)CCCC1 Cc1cc(CCC(=O)NCCCCNC(=O)C(=C2CCCCC2)F)cc(C)c1 C(=O)(CCCn1cc(C2(NC(C3(C(F)F)CC(O)C3)=O)CCC2)nn1)OC C1(C(=O)NC2CN(C(C(C)N(C)C)=O)C2)CC2(C1)CC2F C1(NC(C(c2cccc(C)c2)C)=O)CC2CN(C(C3CCC(F)C3)=O)CC2C1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCCN(C(=O)CC(F)(F)F)C2)C1 C=CCC(CNC(C1(c2ccccc2)CC1)=O)C(=O)NCC(C)OC C1(C(=O)NC2CCCC2N(C)C)(CC)CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(F)F)CS(=O)(=O)NCc1cn(CC(F)(F)F)c(=O)nc1O CC(O)C(F)(F)C(=O)NCCCNC(C1(C#N)CCCO1)=O N1(C(C(=O)Nc2cc(C)c(C)nc2)=O)CC2CC(C1)C(N)C2CO N1(C(c2ccc(OC)cc2)=O)CCC2CC1CN2C(=O)CCCC(C)=O c1(C(=O)NC2CN(C(COCC)=O)CC2(C)C)cc2c(cc1N)CCCC2 C1(CC(=O)NCCCCSCC)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 C12(CNC(C(N(C)C(C3CCNC3=O)=O)C3CC3)=O)COC(C1)C(O)C2 CC1(NC(C2CCC=CCC2)=O)CCCCC1C(N1CCOC(C2CCC2)C1)=O C(C)(C)(CC(C)N=c1[nH]c(N2CC3CCC(C2)O3)nc2ccc(Cl)cc12)OC C(=O)(C1=CCCS1)N(C1CCCC1)CCCNC(C(C)Sc1ccccn1)=O CCCCC(CC(=O)NCC1(C(=O)OC)CC1)NC(=O)CN(C)C(N)=O C1(CN(C)C(C2CC2C2CC2)=O)CN(C(c2cccc(=O)o2)=O)CCO1 N1(C(C2(C)C(C(=O)OC)CC2)=O)CCCC(CNC(c2ccnc(S)c2)=O)CC1 c1(-c2nc(CCC)nn2CC2CCCCO2)ccnc(Br)c1F Cc1nc(C#N)ccc1C(N1CCC(NC(C2CC23CC3)=O)C(C)(C)C1)=O c1(CC)cccc(C(=O)NC2CC3C(NC(c4cscc4C(F)F)=O)C3C2)c1F Cc1cc(CC(=O)NCc2ncoc2CCNC(c2sccc2Cl)=O)no1 N1(C(C=CC(=O)NC2CC2)=O)CC2=C(C1)CN(C(=O)CNc1nccs1)C2 c1(C(=O)NCCCC(C)NC(C2OCCN(C)C2=O)=O)ncn2c1CCCC2 c1(C(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)C2)=O)cc(F)ccc1F N1(C(=O)CC2CCCSC2)CC(CO)C2(CCN(C(=O)CC3(O)CCC3)CC2)C1 CCCS(=O)(=O)C(C)C(=O)NCC1CCCN1C(c1cc2nc(C)ccc2o1)=O CS(=O)(=O)C1(C(=O)NC(CO)CCCNC(C2CCOCC2)=O)CC1 C(=O)(C(C)C(C)NC(=O)Cn1cc(-c2ncccc2F)nn1)OCC C(=O)(C(F)CC(C)(C)C)NCCCC1OCCN(C(c2n(C(C)C)ccc2)=O)C1 c1(C(=O)N(O)Cc2cn(-c3cccc(I)c3)nn2)ccc2c(c1)OCC2 N1(C(Cc2c(C)con2)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)C2CCC12 c1(NC(CC2CC(NC(c3nccc(C)c3)=O)C2)=O)cc(F)c(F)c(F)c1Br Cc1cc(=NC(=O)C(=O)NCC2(C)CCN(C(C3CCCC4CC34)=O)C2)[nH]o1 CN=c1nc(N2CC3CC3C2)[nH]c(=NCC(F)F)[nH]1.C1CC(=O)N1CCO CCCC(C(=O)N1CCC(N(CC(C)C)C(c2ocnc2CC)=O)CC1)C(C)C c1(OC)ncc(C(=O)OCCOc2ccccc2C)cc1C(F)(F)F C12(CNC(c3nc(C)sc3C)=O)CN(C(=O)Cn3cccn3)CC1(C(F)(F)F)C2 C1(N(C(C(CC)n2ccc(C3CC3)n2)=O)CC)CCN(C(c2ccc(C)s2)=O)CC1 C12(C(CNC(c3n[nH]cc3F)=O)NC(Cc3ccc(C)s3)=O)CCC(CC1)C2 N1(Cc2cccc(NC(=O)CCOC(F)(F)F)c2)CCS(=O)(=O)CC1 C(=O)(C#CC1CCC1)N1CC(CC(=O)NC(C(=O)NCC)C)(OC)C1 C1(NC(CCC(N)=O)=O)CN(Cc2ncccc2C(F)(F)F)CC(F)(F)C1 C1(CNC(C(C)O)=O)CCCCN(C(c2cc(-c3ccc(O)cc3)[nH]n2)=O)C1 C(CC(=O)NCc1cccc(CO)c1)(C(C)OC)NC(C(CC)SC)=O C1(CNC(c2c(COC)noc2)=O)CC(F)(F)CN1C(=O)CCn1cc(C)cn1 c12cccc(n1)C(=O)NCCn1cc(nn1)CNC2=O.N1(CC)CCCS1(=O)=O c1(C(=O)NC(C2CCCN2C(=O)C=Cc2cccc(Cl)c2)C)nnc(O)nc1O N1(C(c2cc(CC)ncc2)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 C1(NC(=O)Cc2ccon2)CC2CCC1CN(C(=O)Cc1ccccc1F)C2 N1(C(CCc2ccc(C)s2)=O)CC(C(=O)O)C2(CCC2)C1 C1(C(=O)NC2CC(F)(CNC(CC3C(COC)C3)=O)C2)CCS(=O)(=O)C1 c1(C(=O)NCC(C)N(C(=O)CC(C)SC)CC)cnc(O)c(C(C)=NO)c1 c1(CC)cc(-c2nc(C(C)C3CC3)nn2CCC(F)(F)F)ccc1Br c1(C(N(CCCN(C(CC(CC)C)=O)C)C)=O)nc(C)ccc1C c1(O)ccc(C(C)(C)CNCC(N)=O)cc1.C1(N(C)C)CCCCN1C c1(SCC(N2CCN(C(c3cc(OC)no3)=O)CC2)=O)cc(C)ccc1C C1(CC)CN(C(=O)CCC2CC2CC2CC2)CCN1C(=O)C(=O)NOC O=C(O)C#CC(=O)NC1CCN(C(=O)Cc2cc[nH]n2)CC1 Cc1cc(CNC2CCN(C(c3ccccc3F)=O)C2)c(O)c(Br)c1 N1(C(CC(C2CCN(C(=O)C3=COCC3)CC2)C)=O)CCS(=O)(=O)CC1 N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)Cc2ccc(C)s2)C(C)C1 n1(CCC(=O)NC(CNC(c2cc(C)oc2)=O)C(C)C)nc(O)c2c1CCCC2 N1(C2CN(C(Cc3c(C)n[nH]c3)=O)C2)CC(NC(C2CCC(=O)NC2)=O)CC1=O C#Cc1cccc(C(N2CC(NC(=O)Cc3ccsc3)C(CCC)C2)=O)c1F C=CC(C)(CC)C(=O)N1CCC(CN=c2[nH]nc(C)o2)(C)C1 c1(C(=O)NC(C)(CNC(=O)CCn2cnnn2)C2CC2)cc2cnc(Cl)cc2s1 c1(-c2ccc(N(C)C)o2)nc(Cc2cccc(Br)c2)nn1C1CSC1 c1(C(=O)NC(CC)CN(C(=O)CCc2c(C)noc2Cl)C)nccc(Cl)c1C c1(C(=O)NCC(C2CC2)NC(c2cccnn2)=O)nnc(O)nc1O N1(C(C(c2ccccc2F)OC)=O)CC=CC(NC(=O)C=C2CCN(C)CC2)C1 C(=O)(C1=C(F)CN(C(=O)C(C)(O)C(F)(F)F)CC1)NCCSCC(=O)OC(C)(C)C N1(C(C2(CC=C)CCOC2)=O)CC(O)CC1C(=O)NC1CC(C)(CC)C1 Cc1nc(CCC(=O)NCC2(O)CN(C(=O)Cc3c(C)cnn3C)C2)oc1C N1(C(CCC(C)=O)=O)CCCC(F)(CNC(=O)C(C)Sc2ccccn2)C1 N1(C(Cn2c(C)cnc2)=O)CCN(C(=O)Cc2nnc(O)s2)CC1C C1(N(C(=O)CC2CS(=O)(=O)C2)C)CCCC(NC(c2coc(C(C)(C)C)n2)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC(C)CCCCNC(c1scc2c1OCCO2)=O N1(C(c2nc(OC)oc2)=O)CCC2(C1)CN(C(c1c(C)n[nH]c1C)=O)CC(C)O2 C(c1cocn1)=CC(N1CC(CC(F)C(=O)C(N2CCC2C2CCCCC2)=O)C1)=O c1(CNC(C2C(C)C(=O)C2)=O)ccccc1CN(C(=O)COC1CCC1)C C1(N(C(C(c2cccs2)SC)=O)C)CCCN(C(=O)CC2CC2)C1 N1(C(C2CCN(C(CCNC(C)=O)=O)CC2O)=O)CC(C)N(C)C(C)C1 C(=O)(C1=CCCSC1)NC1C(NC(=O)CCOc2ccc(F)c(Cl)c2)C1 N1(CC(=O)NC)CCC(CNC(C2C3CCC(F)C23)=O)CC1 c1(CC)cccc2c(C(N3CCCC(N(CC(C)C)C(C)=O)C3)=O)c[nH]c12 N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC2(CC(NCc3cc(Cl)ccc3O)C2)C1 CCC(C#N)C(=O)NCc1cc(C(=O)NC2CCCCCC2)on1 c1(OC)ccc(F)c(C(C(=O)NC2CCCCC2)N(C2CCCC2)C)n1 Cc1ccc(C=CC(=O)NCc2c[nH]nc2C(=O)NCCc2nccn2C)o1 C1(C)(N(C)CC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CC3)C2)C1 C1(C(=O)NCCCN(C(Cc2c(C)nsc2)=O)C)CCCC(c2ccccc2)O1 c1(C(=O)NCC2CCC(NC(c3c(C#C)c[nH]n3)=O)C2)ccc2cncnc2c1 C=CC1CN(C(=O)COCC(F)(F)F)CC1NC(=O)C(c1ccc(F)cc1Cl)=O CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC1(C)CNC(=O)CN(C)C1CC1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 C1(CN(C(c2ncn(C(C)C)c2)=O)C)COCCN1C(c1cccc(Br)c1)=O Cc1cc(C(=O)NCC2(NC(C3C(C)(C)C3(C)C)=O)CCCCC2C)nc(O)n1 Nc1cc(C(=O)NCC2CCCC(NC(=O)CC3(O)CCC3)C2)ccc1Cl CC1CC1C1CC1NC(=O)C(F)CC1CN(C(=O)C=CC(F)F)C1 N1(C(C2C(C)C2)=O)CCOCC1CNC(C1(C(C)(C)O)CCC1)=O C1(N(C(CCCOC)=O)C)CCN(C(c2cnn(C)n2)=O)CC1C N1(C(C2(SC)CN(C(C3CC4CCC3CC4)=O)C2)=O)CCCC(C(N)=O)(CCC)C1 C1(NC(c2c[nH]nc2Cl)=O)CCCCC12CCN(C(=O)CC1CCSC1)C2 CC1CC=C(C(=O)NCCC2(CNC(C3CCSC(C)C3)=O)CC2)CC1 c1(C(=O)NCc2scc(CNC(CSCC=C)=O)n2)cccnc1C1CC1 CC1CCC(NC(c2coc(C3CC3)n2)=O)CN1C(=O)CC1OCCO1 N1(C(c2c(C)ncc(C)c2)=O)CCOC2(CCN(C(=O)CC3(O)CCC3)CC2)C1 Cc1cc(C(N2CCOCC2CNC(=O)CSCC(C)C)=O)c(N)c(Cl)n1 c1(OC)c(F)ccc(F)c1C(N1CCN(C(c2nc(=O)n(C)[nH]2)=O)C(C)C1)=O c1(OC)c(C)cc(C(N2CCC(NC(c3scnc3Cl)=O)C2)=O)cc1C c1(-n2c(CN(C)C)nc(CC(CC)C)n2)ccc2c(=O)[nH]ccc2c1 N1(C(c2cc(CC)sn2)=O)CCCOC(CNC(c2nccnc2C(N)=O)=O)C1 C(=O)(CCCCCCCC(=O)N1CC2C(NC(c3cscc3OC)=O)C2C1)OC N1(C(C(CC)OC)=O)CCCC(C)(C)C1CNC(C1CC2C=CC1CC2)=O CC(C)C(CCNC(=O)CC(O)c1cnc[nH]1)NC(=O)CCCC1CC1 c1(C(=O)NC(C(=O)NC(CCC)(C)CC)CC)cnn2c1CCC2 c1(CSCC)ccccc1C(=O)N(CC(O)CN(C(=O)C(C)n1cccn1)C)C C=CCC(CC)C(=O)NCC1(F)CCC(NC(c2nc(CC)sc2Br)=O)C1 C1(C(=O)NC2CC(CCn3cc(COCCO)nn3)C2)C2CCC(C2)S1(=O)=O N1(C(COC2CCN(C(=O)Cn3cccc3)C2)=O)CC(F)(F)C1C1CC1 Cc1c(C(=O)NC2CCCN(C(C3SCCCS3)=O)C2C)cccc1C1CC1 C1(CN(C(CCN(C)CC)=O)CC)CN(C(C2CSC2)=O)CCO1 c1(C(C(N2CCC(CNC(COC(CC)C)=O)C2)=O)C)ccc(F)cc1 c1(CCC(=O)NCC2CN(C(c3cccc(C#N)c3)=O)C2)ccc2ocnc2c1 C1(NC(c2ccc(Cl)cn2)=O)CC2CC1CN(C(C1CCOC1)=O)C2 N1(C(C(F)OC)=O)CC(NC(C2C=CC=CC=C2)=O)CC12CCCC2 c1(C(N2CCC3C(NC(C(C)OCCC(C)C)=O)C32)=O)cc(Cl)c(F)cc1N c1(C(=O)NC2CC(C)(NC(=O)CC(=O)NCC3CC3)C2)cnn2c1OCC(F)C2 C(CCCCCCO)NC(C1(CCNC(c2cc(OC)ns2)=O)CC1)=O [SH](=O)(=O)c1[nH]c(=NCCC(N)=O)ccc1Br.c1(C2CCN(CC)C2)cccc(F)c1 N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN(C(=O)CCc3cnccn3)C2)C1 c1(C(C(=O)NC2CN(C(C=CC(C)(C)SC)=O)CC2O)=O)ccc(F)c(F)c1F C(=O)(CCN(OC)C(=O)Cc1cccc(C#N)c1)NC1C(OCC)COC1 N1(CCC)CCCC(C(=O)NC2(CF)CCN(C(c3nncn3C)=O)C2)C1 CC(C(=O)NC(C)(C)CNC(c1cc2ccc(Cl)cc2o1)=O)C(C)C(C)(C)C c1(C(N2C(C3CCN(C(c4nc(O)n[nH]4)=O)C3)CCC2)=O)c(Cl)nsc1Cl C(=O)(C(C)(O)CC(C)C)NC1C(CO)CCN(C(C=C(CCC)C)=O)C1 c1(-c2cc(OC)ncc2OC)cccc2cc(C(=O)Nc3cccc(C)n3)sc12 Nc1cc(F)c(Cl)cc1C(N1CC2C(NC(C3CCCSC3)=O)C2C1)=O C1(C(=O)NC(c2ncc[nH]2)CO)CCC(C2CCCCC2)CN1 c1(C(=O)NC2CC3(CN(C(CC(C=C)(C)C)=O)C3)OC2)cc2cc(Cl)cnc2o1 c1(C(=O)NCC2(C)C(NC(C=CCC)=O)CCC2)cccc2nc(Cl)cn12 C1(NC(Cc2nc(C)sc2C)=O)CN(C(=O)C(C)n2ccnc2)CCC1O N1(c2nc(C)c(F)cn2)CCC2(CC1)CC(C(=O)N=c1cco[nH]1)CO2 Cc1cc(C(=O)NC(C2(CNC(C3(F)CCCOC3)=O)CC2)C)ccn1 C1(NC(Cc2cnc(OC)nc2)=O)CN(C(C2CC2(C)C)=O)CCC1C(F)(F)F N1(C(CCC=CC)=O)CC(NC(=O)Cc2ccc3c(c2)CC3)CC(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCCC(CN(C)C(c2c(Cl)cnn2C)=O)C1 c1(OC)cncc(C(=O)NCC=CCNC(=O)CCCc2csc(C)n2)c1C CCN=C(NCC(c1ccc(F)cc1)C)NC1CCN(C(=O)CC(F)(F)F)CC1 N1(C(Cc2nnc(C)s2)=O)CCCC2(CCCCC2NC(=O)C2=NOC(C)C2)C1 N1(C(c2cc(C)ncc2)=O)CCCCC1C1CCCN1c1ncc(C#N)cc1Cl C1(C(=O)NCCNC(c2cc(F)cnc2O)=O)CC2(CCCCO2)C1 C=CC(CC)CC(=O)N(c1ncc(F)cn1)Cc1ccc(F)cc1 NS(=O)(=O)c1cc(C(c2ccc3noc(-c4ccccc4)c3c2)=O)c(F)cc1Cl CCC(C)(C)C(O)C(=O)NC(c1ccccc1)CNC(c1ccc(N)cc1C)=O C1(C(=O)NCCN(C(=O)CC2CCC=CCC2)CCC)CCC(F)(F)C1 c1(C(=O)NC(CNC(CCC(=O)NCC)=O)C(C)C)cc(C)cc2cn[nH]c12 C1(NC(C2C(NC(C=C(C)C(F)F)=O)COC2)=O)CCN2CCC1C2 C(CC(CC)(CC)NC(C1CC2CC2C1)=O)NC(C(C=C)O)=O Cc1cn2c(n1)C(C(=O)NC(C)CNC(=O)C(C(C)C)C(C)C)CCC2 c1(CS(N)(=O)=O)ccc(C(N2CCN(C(C3C=CCC3)=O)CC2)=O)cc1 C1(C)(C(=O)NC2C(C)CN(C(c3ccnn3C3CC3)=O)CC2)CC2CCC(C1)S2 c1(C(N2CC3C(CNC(CCCC=C)=O)C3C2)=O)cn2c(n1)SCC2 N1(C(c2cnc(OC)s2)=O)CC2CCC2(CCNC(C2(C(N)=O)CC2)=O)C1 c1(C(N2C(C)CC(NC(c3cc(C)c(C)s3)=O)C2)=O)cccc(F)c1Br C1(C)(CCNC(CN(C2CCC2)C)=O)CCN(C(=O)COc2ccc(Cl)cc2)C1 C(=O)(CC(C)C1CCCO1)N(CCN(C(=O)Cc1csc(Br)c1)C(C)C)C C(CC)(C(=O)NCCCCCNC(c1sccc1F)=O)OCC CCCCC(O)C(=O)NC(CNC(=O)CCCc1ccc(F)c(F)c1)CCOC N(C=CC(=O)C(F)(F)F)C(C1N(C2CCN(C(C(C)C)=O)CC2)CC1)=O C=C1Cn2c(C(=O)NC(CN(C)C(C3CC4CCC3C4)=O)(CO)CO)nnc2S1 CC1CCCN(C(=O)C(=O)NC2CN(C(C3(C(C)(F)F)CC3)=O)CC2C)C1 c1(C(=O)NCCC(C)N(C(Cc2c(C)ccc(C)c2)=O)C)ccc(N)c(Cl)c1O C=C1CC2(C1)CC(C(=O)N(CCCOCCNC(c1cnc(O)cc1C)=O)C)C2 N1(C(C2C(C(C)C)OCC2)=O)CC(C(=O)NC(CCO)C(C)(C)C)C2(CCC2)C1 CC1CCN(C(=O)Cc2cc(Br)cs2)CC1CNC(C1OCCO1)=O Cc1cn2cccc(C(=O)N(C)CCN(C(=O)CCNC(=O)CO)C)c2n1 N1(C(C(CCCCC)O)=O)CC2CN(C(c3cc(OC)cc(I)c3)=O)CC2(C)C1 N1(C(CC(CCC)(C)C)=O)CCC2(CNC(c3ncc(C)cn3)=O)CCCCC12 C1(C(N2C(C(N3CC(O)(CCC)C3)=O)C=CC2)=O)CSCC(=O)N1 CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)NCC1CC(=O)N(C)C1=O)C(C)C CC1CC(NC(c2cnc3sccn23)=O)CCN1C(=O)CCc1cnn[nH]1 Cc1onc(Br)c1C(c1nnnn1CC(F)F)N(CCS(C)=O)CCO C1(NC(Cc2c(C)cco2)=O)CCN(C(=O)C(c2cccc(F)n2)(F)F)C1(C)C c1(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)cccnc1O c1(C(=O)NCCCOCCC(=O)N(CC#C)C(C)C)cc(F)c[nH]1 C1(C(N2CC(C)(NC(C3CC3C(F)F)=O)C2)=O)COc2c(F)cc(F)cc2C1 Cc1ccnc(C(N2CCC2(C)CC(=O)NCC(C)(O)CCO)=O)c1N N1(C(c2csc(Cl)c2)C(=O)NCCOCCO)CCC2NC(=O)NCC2C1 c1(C(CN(C(=O)C(CC2CC2)NC(=O)CC2(O)CCCC2)C)O)ccccc1 Cc1ncncc1C(N1CCC(NC(=O)COC2CCN(C)CC2)C1C)=O c1(C(N2CC(CNC(C3C(SC)CCC3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(SCC(=O)NC2(CCO)CN(C(C(C)OCCOC)=O)C2)ccc(F)c(F)c1 c1(C(=O)NCCCCC(C)NC(C(CC=C)CC=C)=O)cnc2c(c1)CCCC2 c1(OC)cc(C(N2CC(NC(=O)CCOC3CCC3)C(C)C2)=O)ncn1 c1(C(=O)NCC(CC)(CC)NC(c2cc(C)n(CCO)n2)=O)c(C)cccc1Cl N1(C(C(C2CCC(=O)N2)C)=O)CC(C(=O)NOC2CCOC2)C(C2CC2)C1 C1(NC(CC2CC(=C)C2)=O)CCC(O)CN(C(c2ccn3nnnc3c2)=O)C1 CC1(C(N2CC(NC(=O)CCCc3cccs3)C(O)C2)=O)CCC(=O)C1 N1(C(c2c(CC)cno2)=O)CCN(C(=O)CC2CCCOCC2)CC1CCOC N1(C(C2(C=C)CC2)=O)C2CCC1CN(C(c1nn(CC)cc1Br)=O)C2 c1(C(=O)NC2CC(CNC(C34OC(C)(C)C(C3)C4)=O)C2)ccc(Cl)c(N)c1Cl c1(OCC)cccc(CC(N2CCC(C)(NC(C3CCS3(=O)=O)=O)C2)=O)n1 C1(CC(=O)NCC(C)CNC(C2CNC(=O)O2)=O)CCC(=O)C1C Cc1nc2cc(C(=O)NCCC3CCN(C(C4CCCN4C(C)C)=O)C3)[nH]c2s1 CN1CCN(C(C2CCC(NC(=O)CC3CCOC3)CC2)=O)CC1(C)C N1(C(C(CNC(CCCC=C)=O)N(C)C)=O)CCC(C)(C#N)C1 c1(C(CC)C)cc(C(N2CCC2CNC(c2ccnn2C(F)F)=O)=O)on1 c1(C(C)(C(=O)N2CCC(NC(c3nc(CO)cs3)=O)C2)N(C)C)ccccc1Cl N1(C(C=CS(C)=O)=O)CCC2(CCC(CNC(c3coc(CO)c3)=O)CC2)CC1 c1(C(=O)NCC2CCCCN2Cc2cccc(Cl)c2F)nccc2[nH]ccc12 c1(C(c2n(CC=C)nnn2)NCCC2(COC)CC2)ccncc1C Cc1cccc(C)c1C1(C(=O)NC2CN(C(c3snc(O)c3Cl)=O)CC2C)CC1 c1(C(N2C(CNC(=O)NC)CCCC2)=O)ccc2occc2n1 N1(Cc2ccc(CN)cc2F)CCCCC2C1CCCN2C1CC1 C1(C(=O)NCCCC(=O)OCC)CCCCN1C(=O)C=Cc1ccc(C)o1 C(=O)(C1=CCCN(c2nc(C)cc(C#N)n2)C1)Nc1ccc(OC)c(C)c1C c1(N(CC)CC)ccc(C(=O)NC2CC2NC(=O)CC2C(=O)NN=C2C)cc1 c1(C(c2nnnn2C)Nc2cc(C)c(Cl)cc2)ncc2ccccn12 C1(CC(=O)NC(C(C)NC(C2(C=C)CCC2)=O)C)CC(C)(C)C(=O)N1 Cc1ccn2ncc(C(=O)NC3CCC(C)N(C(=O)CC4=CCCCC4)C3)c2n1 C#CCCC(C(=O)NCCCCOCC)NC(=O)C=Cc1ccco1 c1(NC(C2CC(OC)CN2C(c2cnc(O)[nH]2)=O)=O)cc(Cl)ccc1C(F)(F)F C(CCC(C)CC(=O)NCCC(C(C)C)NC(c1cn(C2CC2)cn1)=O)=C(C)C c1(C(N2CCN(C(CP(C)(C)=O)=O)C3(C2)CC3)=O)cnc2nc(Cl)ccc2c1 c1(OCC)cnc(C(=O)N(CC(C)(C)CNC(=O)C(C)OCC)CC)cn1 c1(NC(C2C3(CN(C(CC(C)C)=O)C3)C2)=O)cn2nc(Cl)ccc2n1 C(C(C)C)(C(O)C(=O)NC1C=CC(CC(N2CC(OC)CC23CCC3)=O)C1)OC CC1CCN(C(=O)C(C)Cn2ccnc2)CCN1C(=O)CC1(O)CCOC1 c1(OC)cc(Br)cc(F)c1C(=O)OC1(C(F)(F)F)CN(C(C2CCC(=O)N2)=O)C1 c1(NC(=O)CC2CCCN(Cc3cccnc3)C2)cc(Cl)ccc1Br n1(CCOC)nnnc1C(c1n[nH]cc1C)NCCCC1CCCC1 N1(S(CC)(=O)=O)CC2CCC(C1)C2NC(c1cc(C)cc(O)c1)=O c1(CC)cc(C(=O)NCc2nocc2C(=O)NC(C)CC2CCCO2)no1 c1(C(C)OC)noc(CCC(=O)NCCC2CC(NC(c3ccco3)=O)C2)n1 CC1CCCN(C(=O)C(=O)N(CCn2cc(C(C)(C)F)nn2)C2CC2)C1 c1(C(=O)NC2CN(C(C(CC(C)C)O)=O)CC(F)(F)C2)cc2n[nH]cc2cc1Cl CCCCC(C(=O)N1CCCC1CNC(c1cccc(C)n1)=O)ON=C(C)C C1(C)(CNC(C2N(C(CCC)=O)CCC2)=O)CCN(C(C23CC(C#N)(C2)C3)=O)C1 N1(C(c2c(C)csn2)=O)CC(C2CCN(C(=O)CC3CCCC34CC4)CC2)C1 CC(CCNC(=O)CCc1ccncn1)CCNC(c1cnc(C(N)=O)cn1)=O C(CC(C)(C)NC(=O)CCc1ccoc1)=CC(=O)NC1(CSC)CCC1 c1(NC(C23N(C(c4cccc(C)n4)=O)CCC2C3)=O)cccc(Cl)c1C c1(NC)ccc(Cl)c(C(=O)NC(C2CCOC2)CNC(=O)C#CC2CCC2)c1 C1(C(C)(C)CNC(=O)Cc2cccnc2)CCCCN1C(c1ccnc(O)c1)=O c1(C(=O)NC2C(C(N3CC(CC)OCC3)=O)CCC2)cc2[nH]ccc2cc1Cl CC1(C(=O)NCC(CO)NC(c2cnc(C3CC3)o2)=O)CCCCC1(F)F C1(C(=O)NCCCC2N(C(=O)NCc3c(CO)ccs3)CCC2)CCC(F)CC1 c1(CNCCOCCNC(C(C)C(=O)OC(C)(C)C)=O)ncnc2c1CCCC2 C1(C(=O)NC2C(NC(C(C#C)(C)C)=O)COCC2)CCC=CCCC1 c1(OC)cccc(NC(C2CC2NC(c2cc(Br)cc(F)c2O)=O)=O)c1C#N c1(CC(C2CCCN(C(c3ncccn3)=O)C2)N)ccc2ncnn2c1 N1(C(C(CC)C#N)=O)CC2OCCN(C(c3cccs3)=O)C2C1 C(=O)(CP(C)(C)=O)N1C(Cc2cn(CC(C)O)nn2)CCC1 O=C(CCCCNC(=O)COc1ccccc1)NCC1CCCCC1 N1(C(Cn2cc[n+](C)c2)=O)CC(OC)C(NC(c2csc(C(F)(F)F)c2)=O)C1 N1(C(c2cc(C)n(CC#C)c2C)=O)CC2CC1CN(C(c1ccn(CC)n1)=O)C2 C(CCCOC)(C(=O)NCc1cscc1C)NC(C(C(=O)OCC)F)=O C1(C(N(C)CCC2CCN(C(=O)Cc3ccoc3)CC2)=O)CC12CCOCC2 Cc1cc(=NC(C)c2nnc(CO)s2)[nH]c(=NCC2CC(F)(F)C(=O)N2)[nH]1 CCC(C)C(O)C(=O)NCC1=CCN(c2nnc(C)c(C)n2)CC1 c1(CC(N2CC(NC(C3C(CC)CCCC3)=O)C2)=O)ccc(Br)c(Cl)c1 N1(C(C(CCOC)OC)=O)CC2(CC(C(=O)NCCS(C)(=N)=O)CO2)C1 C1(C(N(CCC)C)=O)CC12CCN(CC(=O)N(c1ccc(Br)cc1)C)CC2 c1(C(C)C(=O)NC2CCCC2NC(C2CC(O)C2)=O)ccccc1[N+](=O)[O-] C1(NC(CC(=C=C)C)=O)CCN(C(=O)C(C)NC(C)=O)CC(C)(C)C1 N1(C(CSC)=O)CCC2(CCC(NC(=O)COC3CCN(C)CC3)C2)CC1 C1(CC(=O)N(CCCCC(c2scc(C(=O)OC)n2)C2CCC2)CC)CCN(C)CC1 C1(C(=O)Nc2c(C)cc(O)nc2)C2CCCC2CN1C(c1ccc(Cl)s1)=O CCCCS(=O)(=O)CC(=O)NC(CNC(=O)C(C)C(C)(C)C)CO C(=O)(C1=CCCC1(C)C)N(C1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1)C c12ccccc1N(C)C(=O)CCn1cc-2nn1.C1(CC(=O)OC)CC(OC)C1 C1(NC(c2cnc(O)o2)=O)CCN(Cc2cn(-c3cccnc3)nn2)CC1 N1(C(CN(CCOC)C)=O)C2CCC1CN(CCNC(=O)COC1(C)CCCC1)C2 Cc1ccc(F)c(-c2conc2C2CC2)c1O C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NCC1(CF)CC1)OC N1(C(C(C=C)OC)=O)CC(C2CCCN(C(c3[nH]nnc3CC)=O)C2)C1 C1(C)(C(=O)NCCN(C)C(c2ccc(CO)c(F)c2)=O)CCNC(=O)C1 c1(NC(C2(CNC(c3ccc(F)c(O)c3)=O)CC2)=O)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(C)CNC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)(F)C12CC2 N1(C(CCCCC)=O)CC(CN(C(=O)CSCc2cccs2)C)C2(CC2)C1 C1(C(=O)NC2CCN(C(C3CCN(c4ccccc4)C3)=O)C2)CC2(CCC2)C1 c1(C(N2CCC(CC=C)(NC(C3CCSC3)=O)C2)=O)c(C)nc(C2CC2)nc1O c1(C(N2CCC(C)(NC(CSC)=O)C2)=O)nc(-c2ccccc2)ncc1Cl N1(C(C(CCSC)O)=O)CCC2CN(C(c3nn(C)c(C)c3Cl)=O)C2C1 CC(C)CCC(=O)C(=O)NC1(C)CC(C(=O)N(C)Cc2cnn[nH]2)C1 C1(CNC(c2c(C)ccnn2)=O)CCCCN(C(c2ccccc2C(N)=O)=O)C1 CC1CN(C(=O)C(Cn2ccnn2)NC(=O)Cc2cnsc2)CCC1N(C)C c1(C(=O)NC23CC(NCc4ccc(OC)nc4)(C2)C3)ccc(C#N)cc1C C1(NC(CNC(CC(C)C)=O)=O)CCC(NC(=O)C(N2CCCC2)C2CC2)CC1 c1(C(N(CC(=O)NCC2OCC(C)C2)C)=O)cn(C)ccc1=O N1(C(C(C)N=[N+]=[N-])=O)CCCC12CCN(C(c1c[nH]nc1Cl)=O)CC2 N1(C(C(C(C)C)S)=O)CCc2nc(C(=O)N(CCO)C3CC3)ccc2C1 N1(C(C2(C(C)C)COC2)=O)C2CCC1CN(C(=O)CN1CCC(C)(C)C1)CC2 Cc1cc(C(N2CCC(NC(=O)CC3(N4CCCC4)CC3)C2(C)C)=O)cc(O)c1 C#Cc1cncc(C(=O)NC(C)(C(=O)NCCCOC(F)(F)F)C2CCC2)c1 c1(N(C)CCC2CCN(C(C3(C)CNC(=O)C3)=O)CC2)nc2ccc(O)cc2s1 C(CC(C)C)(C(=O)N1CC2CC2C1C(=O)NCC1CC(C#N)C1)OC c1(C(=O)NCC(CN(C(=O)CSC2CC2)CC)(C)C)cc(C)c(Cl)s1 n1(CC)ccc(C(=O)NCC2CCN(C(C3C(F)(F)C34CC4)=O)C2)cc1=O N=c1nc(C(F)F)[nH]c(=NC2CCCC(Nc3ncc(C(F)F)cn3)C2)[nH]1 Cc1noc(C)c1-c1cncc(F)c1.C12=CC=C(C=C1)C2NC(=O)C(C)(C)C CC(C(C)(C)C(=O)NCC1CCCO1)NC(=O)CNC(=O)NC1CC1 C1(NC(C(C)SC)=O)CC2CCC(C1)N2C(c1c(C(F)(F)F)coc1C)=O c1(CNC(c2cc(C)n(C)c2)=O)n[nH]c2c1CN(C(=O)COCC(F)(F)F)CC2 C1(NC(CCCNC(C(C)C2CC2)=O)=O)CC(C)(C)C12CC2 Cc1cc(C(=O)NCC(C)(C)CNC(=O)Cn2cccn2)c(F)c(Br)c1 C#Cc1ccccc1NC(C1CCCN1C(c1ccc(OC(F)(F)F)nc1)=O)=O C1(CNC(C2CC(O)CN2C(CC2(C(=O)OC)CCC2)=O)=O)Cc2nccn2C1 C1(C(=O)NC2CC(CCNC(c3cc(C(C)C)on3)=O)C2)CCC(=O)N1C(C)C Cc1cc2ncnc(N3C4CCC3C(C)C(NC(C3(C)CC(C)C3)=O)C4)c2[nH]1 C1(CNC(C(C)OC)=O)CCC(NC(=O)Cc2coc(C)n2)CC1 C1(C(=O)OCC)C2CC1CN(CC(C#N)C1CCOC1)C2 N1(C(c2cc(Cl)ccc2Sc2ccccc2)=O)CC2CCCN2c2ccccc21 C=CCC(C(=O)NC1(CCC(=O)N2CC(CC(N)=O)C2)CCC1)C(C)C C(=O)(C1=NN(C)C(=O)CC1)N1CC2CCC(NC(C(CCSC)(C)C)=O)(C1)C2 CC1(NC(c2cccnn2)=O)CCN(C(C2CCCN(C(=O)C3CC3)C2)=O)C1 c1(C(=O)NCCOCCCNC(C2(C(N)=O)CC2)=O)ccnc(CO)c1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CCNC(=O)Cc1csc(S)n1 C1(CCNC(C(C)CC2CCC2)=O)COCCN1C(=O)CC(C1CC1)C1CC1 C1(C(C)(C)C)CCCN(C(c2cc(Br)cs2)C(=O)NCc2ccccc2Cl)CC1 c1(C(N(C(C)CNC(c2ccco2)=O)C)=O)cccc(Cl)c1O C(=O)(NNC(=O)CN1CCCCC1c1ccccc1Br)c1ccc(C)cc1 C1(C(=O)NC(CCCC)CNC(=O)CN2CC3CC3C2)CC2CCCCCC12 c1(C(=O)NC2CC3(C(C(=O)NCc4cnn(CC)c4C)C3)C2)ccc(C#N)cc1 N1(C(C(C)OCCC2CC2)=O)CCCCC1C1CCN(CCO)C1 Cc1c(C(=O)O)cc(Cl)cc1S(=O)(=O)NC1CCCc2ccccc2C1 C#CC1(NC(C2(C)CCN(C(=O)C(C)n3ccnc3)C2)=O)CCC(C)CC1 C1(C(C(=O)NCCCC(=O)OCC)NC)CCC(C)(C)C1.c1(C)cccc(Cl)c1 C(=O)(CCC(=O)c1cccc(N)c1)NC1C(CNC(C(C)N(C)C)=O)CCC1 c1(C(N2CCC(N(c3ncncc3F)C)C2)=O)ccc(Cl)cc1 c1(C(N2CCC(O)(CCNC(COCC#C)=O)C2)=O)cc(O)ncc1Br c1(-c2cc(F)c(F)cc2)cnn2c1CN(Cc1c(Br)ccc(F)c1F)CC2 CCCCC(O)C(C)C(=O)NC(C)C(C(=O)N1CCC(=C(F)F)CC1)C(C)C c1(NC(COC(C(=C)C)=O)=O)nnccc1C C1(CNC(C2CC(CNC(COC(CC)C)=O)C2)=O)CC(C)(C)CO1 N1(CC(=O)NC(C2CCN(C(=O)COC(C)(C)CC)C2)C)CCCCCC1=O N1(C(C(CC=CCC)C)=O)CCCCCC(NC(=O)CCCC2CCCCC2)C1 C1(O)(C(C(=O)N(C2(CO)CC=CC2)C2CC2)O)CCOCC1 C1(C(=O)NCC2CCN2C(=O)Cn2cnnn2)CC2(COCCO2)C1 CC(CC(C)(C)C)C(=O)N1CCCC1CN(c1ncc(I)cn1)C CCCC(C)CCNC(=O)COC1CCN(C(=O)CC2CCCC2)C1 C1(C(F)(F)F)(C(N(CC(O)CNC(=O)C(C)(C)CN(C)C)C)=O)CC2(CCC2)C1 c1(C(C)C)nn(C)cc1C(=O)NCC1(NC(=O)C(C)C2CCOC2)CC1 C1(C(N2CC3C(C(=O)NCC(C)(C)F)C3C2)=O)CC(=O)CC(=O)N1 c1(C(N(CCC(=O)N(CCCCC)C)CCO)=O)csc(=N)[nH]1 c1(CNc2nnn(C)n2)ccc(CNC(=O)C(Cl)=CCl)cc1F CC(C(C)C(=O)NC1(C2CC2)CCC1)NC(=O)C=Cc1cn(C)nn1 CC(C)(C)CC(=O)N=c1ccn(-c2ccc(Br)cn2)[nH]1 N1(C(C2(CCOC)CC2)=O)CCOC(C(=O)N(C2CCCNC2=O)C)CC1 c1(N2CC(NC(CC3CCCC(OC)C3)=O)C2)nn2cc(C)nc2s1 C1(NC(CCOCC(C)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC(C)(C)C1 C1(NC(=O)Nc2c(C)c(N(C)C)ccc2)C2CCC1(C)C2(C)C CC1(C)CC(NC(c2ncccc2Cl)=O)CN(C(c2ccccc2[N+](=O)[O-])=O)C1 S(=O)(=O)(c1ccsc1C(=O)NC(C)C(C(C)C)NC(=O)C1=COCCC1)NC C1(NC(c2cccc(NC(CC)=O)c2)=O)CC2(C1)CN(C(C1CCC(=O)O1)=O)C2 C1(CNC(c2c(CC)occ2)=O)CC(OC)CN1C(=O)CN(C)S(N)(=O)=O c1(C(N2CC(NC(C(CCC)CC)=O)C(O)C2)=O)ccc2ncn(C3CC3)c2c1 c1(SC)cc(N2CC3CC2CN3C(C2CCCCS2(=O)=O)=O)nc(SC)n1 c1(-c2nc(NC(C(C3CCC3)OC)=O)sc2)ccc(C)cc1 Cc1cc(NC(C2CCC=CCCC2)=O)nc(Br)c1 C1(NC(C2(SCC)CC2)=O)CN(C(=O)C(C)(O)C(F)(F)F)Cc2ccnn2C1 C1(CC(=O)NC(C)(C)CF)CCCN1C(=O)CC1CC1 C(=O)(C1=CC2(CCOCC2)C1)NC(C)(CNC(C1(C2CC2)CCC1)=O)CO c1(N2CCCC(C)C2)cccc(S(=O)(=O)NC2CCC=C2Br)n1 N1(CC)CC(C)N(C(=O)CC2(NC(=O)CCN(C)C)CCC2)CC1C N1(C(CC2CCN(C(C)=O)CC2)=O)CCC2C(NC(C3CC34CCC4)=O)C2C1 c12cccc(F)c1O2.N1(c2ncc(C(=O)O)s2)CCOC(C2CC(F)(F)C2)C1 C1(NC(c2cc(COC)no2)=O)CC2CCC1CN2C(=O)CC(C)(C)C#N N1(C(CC(C)OC)=O)CC(OC)C(NC(=O)CSc2nncs2)C1 c1(C(=O)NCCNC(C(C)(C(C)C)NC(C)=O)=O)oc(S(N)(=O)=O)cc1C c1(C(=O)NC)cc(C)[nH]c(=NCCCC(C)(C)NC(C2CCC(F)CC2)=O)n1 C1(CNC(c2c(CC)ocn2)=O)C2CN(C(c3ccnc(OC)c3)=O)CC12 C(=O)(C(CCF)NC(=O)OC(C)(C)C)N(CC(c1ccc(F)cc1)(F)F)CC N1(CCONC(c2scc(CNC(C3C(C)(C(C)C)C3)=O)c2)=O)CCCOCC1 N1(C(C(C=C)C)=O)CC2CCCC(CNC(C34CCC(CC3)OC4)=O)C2C1 c1(NCCNC(C(C)c2ccco2)=O)cccc(NC(=O)Nc2ccncc2)c1 CCCC(C)CN(C)C(C1(N(C)C(c2cc(C(C)C)[nH]n2)=O)CC1)=O c1(OCC(N2CCC(C(C)NC(C(C(C)C)C)=O)CC2)=O)cc(F)ccc1F CCCCCCC(F)C(=O)NC(C)CNC(c1sc(CC)nc1C)=O n1(CC(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)ncc(C#N)c1N c1(COC(=O)NC2COCC2NC(C2C(NC(C)(C)C)C2)=O)cnc2sccn12 N#Cc1cccc(F)c1CC(N1CC(NC(C2CCCO2)=O)CC(F)C1)=O n1(CCSC)nnnc1C(c1cnc(Cl)s1)NC1CC(NC(N)=O)C1 S(=O)(=O)(c1ccc(N2CC3CC2CC3O)c(C#N)c1)NCC(CCC)O c1(OC)ccc(NC(C23CC(NC(=O)CCc4cnc[nH]4)(C2)C3)=O)c(C#N)c1 Cc1ccc(NC2CCOC(c3ccccc3)C2)nc1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NCC(C)NC(=O)C(C)(C)C1CCC1 C1(NC(C(C)O)=O)CCC2(CCN(C(=O)Cc3cnsc3)CC2)C1 C=C1Cn2c(C(=O)NC3CCCC(NC(=O)CCCn4ccnn4)C3)nnc2S1 C1(C(=O)NC2(CF)CCN(C(c3c(OC)ccs3)=O)C2)CC12CCC(C)(C)CC2 C1(C(=O)OCC)CCCO1.c1(C2CO2)ccsn1.C(=O)(COCC(=O)OC)NCOC CCC(CC(=O)N1CCCC1CC1CC1)NC(c1cc(O)nn1C)=O c1(C(N(CCCOCCNC(C(C)OCC#C)=O)C)=O)coc(Br)c1 C1(C(=O)NCC(CC)(CC)NC(c2nc(Cl)ccc2N)=O)CN2CCCN1CC2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(=O)CCn3cnnn3)CC1C2 N(C1c2ccccc2CC1C)C(c1ccc(OC)nc1Br)=O C(c1ccccc1F)=CC(=O)N(CC(CC)NC(=O)Cn1ncnn1)CC C1(N(C(CCN(CC)CC)=O)C)CCCN(C(c2cc(OC)ncc2F)=O)CC1 N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)COC2CCOC2)C(C2CC2)C1 C1(NC(=O)CSC2CCOC2=O)CCCCC1NC(c1cnccc1Cl)=O c1(C(=O)NC(C2CC2C(=O)NC2CCOCC2F)C)ccc(C#N)s1 Cc1cc(CN(C(C2(CNC(c3[nH]ccc3C)=O)CC2)=O)C)cc(F)c1 C12(C(N)=O)CCCC1(C(N1CC(NC(=O)CSCC3CCCO3)C1)=O)C2 C=C(C)CCCC(=O)NC1C2CN(C(C3CCOC(C(F)(F)F)C3)=O)CC12 Nc1cncnc1C(=O)NCC1(CO)CCN(C(=O)CN2CCNC(=O)C2)C1 c1(C(N2CC(CO)C3(CCC3)C2)C(=O)NCCC#N)ccc2ncccc2n1 N1(C(c2ccnn2CC(F)F)C(=O)NCCOC)CCC12CCN(C)C2 CC(C(=O)NC(N)=O)N(C)CCN(C)C(=O)NCc1ccsn1 CN1CCCC1(C)C(N1CC2C(CNC(c3cncc(-n4cccn4)n3)=O)C2C1)=O c1(OC)ncc(C(=O)NCCNC(=O)C(O)CCN(C)C)c(C(F)F)n1 C1(C=O)CC(C(=O)NCC(C)(C)OC(=O)C(F)(F)C2CC2)=NO1.C1CO1 N1(C(CC2(OC)CCOCC2)=O)CCC2CN(C(=O)CCc3cnc(C)o3)C2C1 C1(CC)CCCN(C(=O)CN2CCOCC2)C1C(=O)N(C)Cc1ccccc1C C1(N(C(C=C(C)C)=O)C)CCCCC1N(C(=O)CCCc1sccc1C)C Cc1nc([N+](=O)[O-])cn1CC(=O)NCC1CC1NC(=O)C(C)(C)n1cccn1 CC1CN(C(c2ncsc2C(F)(F)F)=O)CCC1NC(=O)CN1CC=CC1 c1(CN2CCCC(CC(=O)NCc3ccncc3)C2)cc([N+](=O)[O-])c(O)cc1O c1(CCC(=O)NC(C2CCOC2)CNC(C=C(CC)CC)=O)nc(C2CC2)no1 C(=O)(C(CCOC)NC(=O)CCC1CC1(C)C)NCC1CC(=C)C1 c1(C(N2CCC(COC)(NC(=O)Cc3n[nH]cc3Br)C2)=O)cc(C)n(C)c1C N1(C(C=COCC)=O)CC(NC(=O)C=Cc2ccncn2)CC(C)C1 CC(N=c1[nH]c(N2CCOC(C3CC3)C2)nc2cccc(F)c12)C1CC(F)(F)C1 C1(NC(c2ncc(C)cn2)=O)CCC2(CCCN(C(c3nnn(C)c3C)=O)C2)C1 c1(OCC=C)ccc([N+](=O)[O-])c(COC(=O)NC(CSC)CC)c1 C1(NC(c2c(C)c[nH]n2)=O)C2CC(NC(=O)CC3CCCC3C)CC12 c1(C(C)C)ccc(CC(=O)NC2CC(NC(C34CC(C)C3C4)=O)C(O)C2)cc1F C(=O)(C(CCC(C)C)NC(C1CC(=O)C1)=O)NC(CCOCC)C C1(NC(CCC(=O)OC)=O)CN(C(C2CC23CCCCC3)=O)CC(C)(C)C1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)Cc2cnsc2)CCO1 C1(C(=O)NCCOC)CCN(C(c2cc(OC)cs2)=O)C1C(C)C c1(C(=O)NCCN(C(C2C(CC)OCC2)=O)C2CC2)cccc(F)c1F N1(C(c2ncc(-c3n(C)ncc3)nc2)=O)CCc2ccc(F)cc2C1 Cc1cc(F)c(N)cc1C(=O)NC(CO)C(C)NC(c1ccc(Cl)c(F)c1)=O c1(C(C)C)nnc(N(CC(C)CNC(=O)C=CC2CCOC2)C)o1 C1(CNC(C)=O)CCCCN1C(=O)CC1CCCC(C2CC2)O1 C1(C)(C(N2CCCC(NC(C)=O)C2)=O)CCN(Cc2cnn(CCO)c2)CC1 c1(C(N2CC(C)(NC(=O)CCc3csc(=N)[nH]3)C2)=O)cccn2nnnc12 N1(C2CCN(CCC(C)C)CC2)C(=O)NC(C2CCc3ccccc32)C1=O c1(CC)ccc(C(=O)N(CCCNC(=O)CN(C)C)CC2CCC2)cn1 C(=O)(CC1OCc2ccccc21)NC1CC(CNC(c2n[nH]c(C)c2Cl)=O)C1 Cn1cc(C(=O)NCC2CCCCN2C(c2ccnn2CC#N)=O)c(O)nc1=O C(=O)(C(C)(C)C(=O)NC(CC(F)F)C(=O)NC1C2CCCC12)N(C)C C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(C(CSC)OC)=O)C2(C1)CC2 S(=O)(=O)(c1ccc(N2CC3CC3C2)nc1)NC1CC(C)N(c2ccccc2)C1 S(=O)(=O)(c1ccc(F)c(F)c1)N(C1C2CCC1CNC2)Cc1ccc(C)cn1 C12(NC(c3ccoc3C(F)(F)F)=O)CCC(C1)N(C(C1CC=CCC1)=O)C2 CCC(C(=O)NCCN(C1CCCC1)C(=O)COc1cc(F)ccc1F)C(C)O c1(C(=O)NCC(C)SC)cc(=NC(=O)CNC(=O)C(C)(C)C)[nH]n1C N1(C(C(C(CC)O)(F)F)=O)Cc2ccccc2C(NC(=O)COC2CCCC2)C1 c1(C(N(CCC)CCNC(=O)C(F)(F)C2CCOCC2)=O)ccc(C(F)F)nc1 c1(OC)ccc2cc(C(=O)NC3CC(C)CN(C(C4CCCS4)=O)C3)ccc2c1 c1(C(=O)OC)ccc(CN2CC3CCC2C3C(=O)O)c(OC)c1 c1(C(N2C(CNC(=O)CCCN=[N+]=[N-])CC(OC)C2)=O)cnc2n(c1=O)CCS2 N1(C(C2C3(CC(NC(c4c(C)oc(CO)c4)=O)C3)C2)=O)CCC(C#N)CC1 CC(C)C(C(=O)NC12CC(NC(=O)C(Cc3ccsc3)NC=O)(C1)C2)NC=O c1(C(=O)NC(CC#C)C(=O)N(C(C)CSC)C)cc(C)ccc1F c1(CC(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)C)cccc(Cl)c1 C1(C(=O)NCC2N(C(C3C(C)CC3)=O)CCC2)CC(C)(C)CO1 C1(CNC(C(CC)(C)ON=C(C)C)=O)CCCC2CN(C(=O)C3=CC(C)(C)C3)CC12 N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1[nH]ccc1C)=O)C2 CCC(C)CC(C)CC(C)C(=O)N1CCCS(=N)(=O)CC1.c12ccc(cc1)o2 CCCC(C(=O)N1CCN(C(=O)C(C)Cc2ccccn2)CC1)N(C)C CC1=C(C(=O)N2CCC(NC(C3CCS(=O)CC3)=O)C(C(C)C)C2)CCC1 C=CCCC(C(=O)NCCC(C)F)NC(=O)CCC(CC)OC c1(N2CCC(NC(C(CC3CC3)NC(C)=O)=O)CC2C)nc(C)nc2c1cnn2C Cn1cc(C(F)=CC(=O)NCCC2CCN(C(C3CC4(CC4)C3)=O)C2)cn1 CC1(C)CN(C(=O)Nc2ccc(C(F)(F)F)c(Cl)c2)CC1Nc1ncncc1I N1(C(C2(CC)CCC2)=O)CCC(C)C(NC(=O)CSCc2c(C)noc2C)C1 c1(CC(=O)NC2CN(C(CCCOCCC)=O)CC2C)ccc(CC)c(F)c1 N1(C(C(C(C)O)N)=O)CC2CCCC2C1C CC1(C)CC1(C)CNC(c1csc(O)n1)c1nnnn1CCCC1CC1 C1(NC(COCC#C)=O)CN(C(=O)CCCSC(C)(C)C)C2(CCC2)C1 c1(-c2cn(C(COCC)C(N3CCC(C)C3COC)=O)nn2)ncc(F)cn1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)CCOCC(O)C1 c1(C(N2CCCC23CCN(c2nnc(C4CC4)s2)C3)=O)c[nH]c2cccc(F)c12 C1(NC(CCCOC(C)=O)=O)CC2CCC1(NC(c1cc(C)n(CCO)n1)=O)C2 N1(c2n(CC(=C)C)c(-c3ccoc3C)nn2)CC(C)OC2(CCCOC2)C1 CS(C)(=O)=Nc1ccc(C(N2CCCC(NC(=O)CCOCC3CC3)C2)=O)cc1 c1(C(=O)NC2(CNC(C3(C)CCC(C)C3)=O)CCCC2)ccc(P(C)(C)=O)cc1 c1(C(N(CC(C)NC(=O)C(O)C(C)c2ccccc2F)C)=O)ccc(F)cc1N N1(C(c2cccc(Cl)c2C)CC)CC2CCC(C1)N2CC(c1ccccc1F)O C(=O)(C(C)(C)CCCNC(=O)C(C1CC1)OCC)NC(CC#C)CO c1(C(=O)NC(CNC(C(C(C)(C)C)OC)=O)(C)CO)cnc2sc(C)cn12 Cn1cc([N+](=O)[O-])cc1C(N1CC2CCC(C1)C2NC(c1cscn1)=O)=O c1(C(=O)NCCC(C)NC(CC2(NC(C)=O)CC2)=O)ccc(C2(C)CC2)cc1 C(CC(C)CC)(C(=O)N(C)CC1(O)CCCCC1)NC(C=CC)=O c1(C(N2C(C(=O)NCC(=O)OC)CCC2)C(=O)OC)c(Cl)c(C)nn1C Cc1ccc(NC(C2CCOC2CNC(c2nonc2N)=O)=O)c(C)c1O CCCC(C)NC(=O)CSC.CCC(C)(c1nccs1)NC(=O)O N1(C(C(C)SCCCC)=O)CCCC(NC)C1.c1(C(=O)NCCN)coc(C(F)F)c1 Cc1ccc2c(CNC3CCCN(Cc4ccccc4)C3C)cc(=O)oc2c1 C(=O)(CC(C)CC(F)(F)F)NC(CCNC(C1CC(C)(C(=O)OC)C1)=O)C C1(N(C(c2sccc2Cl)=O)CC)CCCN(C(=O)CCCc2cc[nH]n2)CC1 c1(C(=O)NC2CN(C(C3CC(CC)C3)=O)CC(O)C2)nn2cccnc2c1Cl C=C(Cl)C(C)(C)C(=O)NCC1(COC)CCN(C(c2ccncc2O)=O)CC1 c1(CNC(CCC)(C)C)nc(O)c2c(C)c(C(C)C)sc2n1 N1(C(c2ccc(CSC)cc2)C(=O)NCc2ccco2)CCOCCC1C1CC1 C1(C(=O)NC(C=C)C)CCC(c2ccccc2)CC1 C1(CCCCNC(C(C)n2cncn2)=O)CCN(C(=O)C=Cc2cn[nH]c2)CC1 C(c1ccc2c(c1)OCO2)=CC(=O)NCC1CCN(C(C2(F)CCOC2)=O)C1 c1(OCC)nccc(C(=O)NCC2CN(C(=O)CCS(=O)(=O)NC(C)C)C2)c1F c1(OC)cccc(C(N2CCN(C(=O)C(CO)C(C)C)CC2C(C)C)=O)c1F CCC(COC)C(=O)N(CC(O)CNC(=O)C=CSC)C C(=O)(C1=C(C)CCCC1)NCc1cn(CC(C)NC(C(CCC)C)=O)nn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C2CCC12 O=S(=O)(c1cccs1)NCC1(O)CCCN(Cc2cc(Cl)ccc2Cl)C1 N1(C(C2(CC)CCOC2)=O)CCN(C(=O)CCCOC)C(c2ccc(Cl)cc2)C1 c1(C(N(CCNC(C(n2ccc(C(F)(F)F)n2)C)=O)C)=O)ccc(S(C)(=O)=O)o1 C1(C)(C(=O)OCCN(C(=O)OC)C)CN(C(=O)OC(C)(C)C)CC1(F)F Cc1cc(Br)cc(C)c1CNCC12CC1CN(C(=O)Nc1cccc(Cl)c1Cl)C2 Cc1nc(NC2CC23CC(NC(=O)C(N2CCSCC2)C)C3)ccc1[N+](=O)[O-] Cc1nnc2n1CCCC2C(=O)Nc1cnc2n1CC(C(F)(F)F)CC2 N1(C(COCCCC#C)=O)CCN(C(=O)NC2CN(C3CCC3)C2)CC(O)C1 N1(C(C2C=CC(NC(c3ccc(COC)o3)=O)C2)=O)CCC(C)C1CO CC1C(NC(c2ccc(-c3ccccn3)nc2)=O)CCN1c1nnco1 c1(SCC(=O)NCCC(C)N(C(=O)CCNC(c2nc[nH]n2)=O)C)ccccn1 C(=O)(C1CCc2c[nH]nc21)NC(CC(C(=O)N(CCN=[N+]=[N-])CC)F)(C)C C(=O)(C(C)(C)CN(C(=O)Cc1ccnn1C)C)NCCC1CC(C)C1 c1(C(=O)NC2CC2CNC(C2(O)CCOC2)=O)cc(Cl)c(Cl)s1 c1(C(N2CC(NC(C(C)SC(C)C)=O)C3(C2)CC3)=O)cccc2c1COC2 c1(C(N(CCC)CCNC(=O)CCCc2ncc(C)o2)=O)ccc(C)c(F)c1F c1(C(N2CC(C=C)C(NC(=O)CCc3cnco3)C2)=O)cncc2[nH]ccc12 Cc1cccc(C)c1NC(C1CCCN(S(=O)(=O)CC23CCCC2OCC3)C1)=O CN1CC2(CCN(C(C3C4CC3N(Cc3ccc(Br)cn3)C4)=O)CC2)C1 C(=O)(CC(C)(C)CC(F)F)N1C2CC(CNC(C(C)OCCCC)=O)C1CC2 C1(NC(c2cnc3ncccn23)=O)CCC2CN(c3nnco3)CC2C1 Cc1cc(C(=O)NCC2(C)CCCN2C(c2cocc2C)=O)ncc1CO CC1CCN(C(c2cnn(CCF)c2)=O)CCN1C(=O)C(F)CC(C)(C)C c1(COC)cc(C(=O)N(C2CCN(C(=O)C(C)NS(C)(=O)=O)C2)C)c(C)o1 Nc1c(F)ccc(Cl)c1C(N1CCOCC(CNC(=O)C=CC(N)=O)C1)=O C1(CC(=O)N(C2CCN(C(=O)CCn3cccc3)C2)CCC)CCCCCO1 C1(C(N(CC#C)CC=C)=O)C2CC2CN1C(=O)CCOC1CCCC1 C1(C2(C)CC2)(C(N(CCCCNC(C(CC2CCC2)OC)=O)C)=O)CC1 c1(C(=O)NC(CNC(C(CC)O)=O)CC)c(C)cc(=O)n(C)c1C c1(C(=O)NCCN(CCOC)C(c2cc(F)cs2)=O)cnc(C)[nH]1 C12(NC(=O)C=CC3CCCCC3)CCN(C(=O)Cc3c[nH]ccc3=O)CCC1C2 C=C=C(C)CC(=O)NC1C2CCN(C(=O)C(C)Sc3ccccc3Cl)C12 CN=c1[nH]c(=NCC2(c3ccccc3)CCCO2)[nH]c(=NCC2CC23CCC3)[nH]1 CCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(OC)n(C)n1)=O C1(N(C(CCOC2CN(C(C(C(=O)OC)C)=O)C2)=O)C)CCC(=O)N(C)C1 c1(C(=O)OC)c(NC(=O)C(C)(O)Cn2cc([N+](=O)[O-])cn2)sc(C)c1C C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCF)C(CO)C1 C(Cn1cncn1)(C(=O)Nn1cnnc1C)NC(c1ccc(C)[nH]1)=O N1(C(C2CC(C#N)(OC)C2)=O)CCC(C)C(NC(=O)CC2CCS(=O)(=O)C2)C1C Cc1ccc2occ(C(N3CCC4CN(C(C5CNC(=O)O5)=O)CC4C3)=O)c2c1 N1(C2CN(C(CNC34CC(CC(=O)Nc5cccnc5)(C3)C4)=O)C2)CCCC1=O N1(C(c2cc(F)c(F)cc2Br)=O)CCOCC(N=c2[nH]cnc3cc(I)sc23)C1 CC12COC(C(=O)NCCC3(O)CN(C(=O)CCCn4cncn4)C3)(C1)C2 c1(NC(C2CC23CCN(C(c2cccnn2)=O)C3)=O)cccc2c1OCO2 C(=O)(CCS(=O)(=O)N(C)C)NCCC1CC(NC(C=NOC)=O)C1 c1(OC)cc(CNc2nc(C(N3CCCC3(C)C(N)=O)=O)sc2)cc(Br)c1 c1(C(N2C(CN(C(C(C3CCOCC3)C)=O)C)CCC2)=O)cn(C)c(=O)nc1O c1(CC)nccn1C(C)CC(=O)NCCC1CCN(C(c2ncc[nH]2)=O)C1 c1(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)ccc2cnccc2n1 CCC(CCCC(=O)NC1C(OC)CC1O)NC(=O)Cc1cc(C)on1 c1(C(=O)NC23C(CN(C(c4cncc(CC)c4)=O)C2)C3)cc(F)c(N)cc1OC Cc1nn2cccnc2c1C(=O)NC(CNC(=O)CN1CCCOC1=O)CO C1(CNC(c2c(N(C)C)cccc2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC1(C)C(CC(N2CCC(CCF)CC2)=O)CCN1C(C1CC2CCC(C1)O2)=O N1(C(C(CC)C)=O)CCN(C(c2ccc(C)c(C)n2)=O)C2(CCC2)C1 Cc1cc(OCCCn2nnnc2N(c2c(C)cccc2C)C)cc(C)c1 C1(C(=O)OC)(N(C)C)CC(NC(c2nc(C(C)(C)C)cs2)C)C1 C1(C(=O)NC2CC(N(C(C(c3ccc(C)cc3)F)=O)C)C2)CCOC(=O)CC1 Cc1c(C(N2CC3CC(NC(=O)C(F)C4CCC4)C2C3)=O)[nH]c2cc(F)ccc12 N1(C(c2nc(C)nn2C)=O)CCC2(NC(=O)CNC(N)=O)CCCC12 C(=O)(C1=C(C)OCCC1)N1C(CN(C(CC2CCC(C(C)=O)CC2)=O)C)CCC1 N1(C(CCc2n(C)ccc2)=O)CCC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O c1(C(=O)OCCC(C(=O)NC(CC#C)C(=O)OC)(C)C)cc2cc(F)cc(C)c2[nH]1 C1(NC(C(COC)NC(C)=O)=O)CC(CO)N(C(=O)CSc2ccccn2)C1 c1(NC(C2CC2C(N2CCCCC(O)C2)=O)=O)cc(F)ccc1Br N1(C(C2CC(CN(C)C)C2)=O)CCC(NC(=O)Cn2nnc(-c3ccco3)n2)C1 C12(CC=CCC1)C(=O)N1CC(C1)C2.N1(OC)CCN(c2ncco2)CC1 N1(C(c2csc(C)c2C)=O)CCN(C(=O)COC2CCCOC2)C(C(F)F)C1 N1(C(c2c(CC)cc(F)cc2)=O)CCC2(CC1)OCCC2NC(=O)C(O)CSC C(=O)(C(O)CC(C)(C)C)NCCCCCNC(C(C(C)C)SCC)=O C(C)(CCC(C)(C)O)(c1n(C(CC)(C)C)nnn1)NC1(CCO)CCOC1 C(=O)(CC(C)(C)n1ccnn1)NC(CCN(C(=O)CC1CSC1)CC)C c1(OC(C)C)cccnc1C(=O)NC1CC(CCNC(=O)CC(=O)OC)C1 c1(NC(CNC(CC(C)=O)=O)=O)cccc(Br)c1OC(F)F Cc1cccc(C(=O)NC2CCCC2NC(c2sccc2F)=O)c1 C(=O)(C(C#N)(CC)CC)NCCC1CN(C(C(c2ccc(OC)cc2)CC)=O)C1 Cc1onc(C2CC2)c1C(=O)NCCC1CN(C(C2(F)CCOCC2)=O)CC1C N1(C(C2(C)COC(=O)C2)=O)CCCC(CO)(NC(c2cc(O)nc(O)c2)=O)C1 c1(C(C)(C)C(=O)N2CC(NC(C3CC(=C4CCC4)C3)=O)C2)cccnc1F S(=O)(=O)(c1c[nH]ccc1=NC1CCCOC1)NCc1cc(OCCC)nn1C N1(C(C2(C)N(C(c3cccc(C)c3N)=O)CCC2)=O)CCC(=C(F)F)CC1 Cc1ccc(CCNC(=O)C(C)(C)NC(=O)CCCN(C)C)cc1 N1(C(CC2(C=C)CN(C(C3(C(N)=O)CC3)=O)C2)=O)CC2CCCCC12C N1(CC(=O)NC(CNC(c2c(C)oc(C)c2C)=O)C)C(=O)NC(C)(C2CC2)C1=O C1(NC(C(N2CC(C)OC(C(F)(F)F)C2)=O)=O)CC2(C1)CC1CCC(C2)N1 C1(C(C(=O)NCCCC(=O)OCC)N(C(c2ncc[nH]2)CC)C)CCC(C)CC1 c1(CC(N2CC(CNC(C(C(C)C)OC)=O)C2)=O)nn(C)c(=O)c2ccccc12 N1(C(C2(C(C)C)CC2)=O)CCC2(CCCN(C(c3nc(Cl)sc3Cl)=O)C2)CC1 C1(NC(CCC=C)=O)CCCN(C(c2cc(-c3cccnc3)n(C)n2)=O)CCC1 c1(CN2CC(CC)N(C(=O)CCc3ccc(C)cc3)CC2)c(F)ccc(C)c1F C(=O)(C(O)C(F)(F)F)N1C(CNC(c2ccc(CCC)[nH]2)=O)(COC)CCC1 c1(C(N2CC(C(C)NC(CCCOC)=O)OCC2)=O)ccc(=O)n(C(C)C)c1 N1(C(c2c(C)coc2C2CC2)=O)CC(NC(C2C(F)(F)C23CCC3)=O)C2(CC2)C1 Cn1cc(C(=O)NC2(C)CC(NC(C3CC4CCC4C3)=O)C2)ncc1=O c1(-c2n(C(n3ccnc3C(C)C)OCC)ccn2)ccc(OC)cc1 C1(C(F)(F)F)(Cc2cn(CCOC)nn2)CCCCC1 Cc1c(-c2noc(C(c3cn(CCCN(C)C)nn3)C)n2)cc(C#N)n1C C=CCCCCCCC(=O)NCC1CCCC1C(=O)NC(Cc1ccco1)CO CC(C)C(F)C(=O)N1CCC(C(O)CNC(c2ccc(OCCF)cc2)=O)CC1 N1(C(=O)CSC2CC2)CCCC2(CCN(C(c3csnn3)=O)C2)C1 c1(NC(C2(SC)CC(O)C2)=O)ccc2nc(C)[nH]c2n1 N1(C(C(CCC2OCCO2)CNC(=O)OC(C)(C)C)=O)CCc2cc(C#N)ccc2C1 C1(CC(=O)N(C)CC#N)CCC(C(=O)Nc2ccncn2)CC1 c1(CC)ccc(C(N2CC(NC(C34COCC(C3)C4)=O)C(C)C2)=O)cc1 N1(C(CC(=O)OCC)=O)CCOC(C(C)NC(c2cn(C(C)C)nc2C)=O)C1 CCC(CC(F)(F)F)C(=O)NCC1CN(C(=O)CCNC(=O)CC(C)C)CC1O c1(C(N2C(C)CC(NC(C3C(C)(CC)C3)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(O)(C(C)NC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CC1 N1(C(C2C(C)N(C(=O)CCc3cncnc3)CC2)=O)C2CCCC1CN(C)C2 c1(CC)cc(CC(=O)NCCCn2cc(-c3ccc(C(=O)O)nc3)nn2)ccc1C C(=O)(C(C)C(C)c1ccco1)NC(CN(C(COCc1onc(C)n1)=O)C)(C)C Cc1ccnc(N2CC(CO)(NC(C34CC3COC4(C)C)=O)C2)c1[N+](=O)[O-] Cc1cc(C(=O)NC2COCCC2NC(=O)C=Cc2cn[nH]c2)cc(F)c1 CS(=O)(=O)C(CNC(C1(O)CC1)=O)CNC(c1n[nH]c2c1CCC2)=O c1(C(=O)NC2C(CNC(=O)C(=CC3CCCCC3)F)C2)ccc(=O)n2c1CCC2 c1(CC(C(=O)N(CC(CNC(CN2CC(CC)C2)=O)C)C)C)c(C)n[nH]c1C Cn1cc([N+](=O)[O-])c(=NC2CCN(C(C3CCC=CCC3)=O)CC2)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2CC2)(CNC(C2(C)CC=CCO2)=O)C1 C(=O)(C(CC)CCOC)N(C(CCNC(C1C(CC)CCCC1)=O)C)C N1(C(C(=O)NC(c2ccncc2)=O)=O)CCC(F)(C(=O)NCC2(NC3CC3)CC2)C1 c1(N(C)C)nccc2c1CN(C(=O)C(=O)Nc1ccc(S(C)=O)cc1)CC2 n1(CCOC)cc(C(=O)NC(CNC(=O)CCc2nncs2)C(C)C)cn1 C1(C(N(C(CC)CC(=O)NC2CCCCC2C)C)=O)CC2(C1)CC(C)C2 N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CCCCN(C(C3CCC4CC4C3)=O)C2)C1 c1(C(=O)NCC(C(C)(C)C)NC(C(C(C)C)n2cnnc2)=O)ncc(Cl)nc1Cl N1(C(C(C2CCN(C(C(C)(C)SC)=O)C2)C)=O)CCC(O)(CCO)CC1 N1(C(c2c(CC)nc[nH]2)=O)CC2(C1)CN(C(=O)C(F)(F)Cl)C2 O=C(CC=C(Cl)Cl)NCCCN(C(c1ccnc(SCCO)c1)=O)C1CC1 c1(CC(N2CC(NC(C=C(COC)C)=O)C(F)CC2)=O)coc2cc(Cl)ccc12 C1(C(=O)NC2CC(NC(C3(CC=C)CCC3)=O)C2)CC=CC(O)C1 CC1CN(C(c2ccoc2C(F)(F)F)=O)CC1NC(C1(C)CC2(CC2)C1)=O C1(C(C(=O)NCC(CNC(c2cc(C)n(C)c2)=O)OC)C)CCCCCC1 c1(NCC(C)NC(c2c(C)nccc2)=O)nc2c(cc1C#N)CCC(C)(C)C2 C1(NC(CCN(CCCCC)C)=O)CCCN(C(C2CC3CCC3C2)=O)C1 N1(C(C(c2ccc(C)o2)C)=O)CCC(C(=O)NC2CCC(O)C2)C12CC2 CC1CCC(NC(C2(C3CCC3)CC2)=O)CN1C(c1cc(F)ccc1Br)=O c1(C(=O)OC)c(C)[nH]c(C(=O)NCCCc2cn(CC3(CO)CCC3)nn2)c1C C(C(=O)N1CCC(CO)(NC(=O)CN2CCNC(=O)C2)CC1)(C(C)(C)C)SC C1(C(=O)OCc2cc(C)sn2)CCC(=O)C(C)C1(C)C c1(C(N2CCC(C)C2CNC(=O)C=CC2CCC2)=O)cc2ccc(Br)cn2c1 C=CCC(CNC(c1ncccc1CC)=O)C(=O)NCC(CO)C1CC1 C1(CNC(C2(CCNC(C3(C)CCCC3)=O)CC2)=O)CCCC2(CC2)C1 c1(C(=O)NCCC(C)N(C(=O)Cc2cccc(Cl)c2Cl)C)cnc2[nH]cncc1-2 CN=S(C)(=O)c1ccc(C(=O)NCC2CN(C(=O)CC3CC3)CC23CCC3)cc1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC(F)(CNC(=O)C(F)C2CCOC2)C1 c1(C(N2CCC(CCNC(CCCC#C)=O)CC2C)=O)cccc2c1NCC2 S(=O)(=O)(CC(=O)NCC1CCCCC1NC(=O)CC(C)(F)F)NC(C)(C)C N1(C(C2C(OC)CN(C(C3CN4CCN3CC4)=O)C2)=O)CCC2(COC(=O)N2)C1 CC(CN(C(=O)Cc1nccn1C)C)C(=O)NC1(C2CCCO2)CCC1 N1(C(C(C)NCCC#N)=O)CC(C)(C)C(NC(=O)C=CC(=O)N(C)C)C(C)(C)C1 Cc1nc(C(N2CC(OCCNC(c3ccc(=O)oc3)=O)C2)=O)c(C)o1 N1(C(CSC)=O)CC(OC(C2CSC2)=O)CC1CC(N1CCN(C(C)=O)CC1)=O Cc1c(C(N2CCC(C)(C(=O)NCc3ccc[n+]([O-])c3)CC2)=O)cncc1F c1(OC)cc(C(=O)NCCC2CCN(C(=O)C#CC(C)(C)C)C(C)C2)ccc1F Cc1cc(N)cnc1C(=O)NCC(C)N(C)C(c1ccc(C(C)(C)C)s1)=O C12(NC(c3c(Cl)c(C)n(C)n3)=O)COCCC1CN(C(=O)C1=CCCCC1)C2 C1(NC(=O)Cn2nnc(=O)[nH]2)CCCCN(C(=O)CSc2ccccn2)C1 Cc1ccc(Cl)c(OC(C)C(=O)NCC(C(C)(C)C)NC(=O)C=CC(F)(F)F)c1 c1(OCOC)ccc(-c2cnc(CNC(c3cc(I)c[nH]3)=O)nc2)c(C)c1 c1(CN2C(C(=O)OC)CC(C(C)(C)C)CC2)cn2c(n1)CCCC2 N1(C(CCC(=O)NC)=O)CCC2(NC(=O)CP(C)(C)=O)CCCC12 C(=O)(C(C)C(C)(C)c1ccccc1)N1C(CNC(Cc2c(C)nc[nH]2)=O)C=CC1 c1(C(CNC(c2cccc(Oc3ccccn3)c2)=O)F)ccc(F)cc1F N1(C(c2n[nH]c(C)c2Cl)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC(C)(C)C1 c1(C(=O)NCCC2CN(C(C(C)OCCN(C)C)=O)C2)cc2occc2s1 c1(OCCC(=O)NCCC(C)NC(=O)CC2CC3(CC3)CO2)ccc(F)c(Cl)c1 C(=O)(C(F)(F)CCn1cc(C(N2CCOCC2)(C)C)nn1)NCCC(=O)OCC c1(C(=O)NCC(c2ccc(C(C)(C)C)cc2)O)cc(N=[PH](C)(C)=O)ccn1 N1(C(c2cc(C)ns2)=O)CCCC(NC(C2CCC(C)(C)OC2)=O)C1C C1(CC)CN(C(=O)COc2ccc(F)cc2)CCC1NC(C1C2CCC(=O)C12)=O c1(C(C(=O)NCC2CCN(C(C(C(C)SC)O)=O)CC2)=O)ccc(F)c(F)c1F N1(C(=O)CSCc2ncc[nH]2)CCCC2C1CCCN2C(c1c[nH]ccc1=O)=O N1(C(c2ccc(Cl)cc2)=O)CCn2ncc(-c3cnn4c3CCC4)c2C1 CC1(CC(=O)NCC(O)CCNC(=O)Cc2ccccc2Cl)CCCCCC1 CCCCC(C(=O)NC1CN(C(=O)C(C)CC2CCCCC2)CCC1C)C(C)C c1(C(N(C2CCN(C(=O)CCc3cccn3C)C2)CC#C)=O)cnn(CCO)c1 N1(C(C(CC)F)=O)CC(NC(=O)CCc2ccc(OC)cc2F)CC(C)(C)C1 c1(C(C)C(=O)NCC=CCNC(C23CCCC2C3)=O)cccc(C(F)(F)F)c1 N1(C(C2C=CC(NC(=O)CCC(F)(F)F)C2)=O)CC2CCC(O)C(O)C12 N1(CC(N2CCCC(C(C)NC(C(OC)OC)=O)C2)=O)Cc2ccccc2C1=O Nc1cncc(C(=O)NCC2C3CN(C(C4CCCC(O)C4)=O)CC23)c1 C(C(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O)NC(CCCOCCOCC)=O CCN=c1[nH]c(C(=O)NCC2CC(F)(CNC(C3CCN(CC)C3)=O)C2)cs1 c1(CC(=O)NC2(CNC(c3c(CC)c[nH]n3)=O)CCOC2)c[nH]c2ncccc12 N1(C(c2c(NC)cccc2)=O)CC2N(C(c3ccc(Cl)o3)=O)CCC2(C)C1 c1(CC(=O)NCC(CC)NC(=O)CC2CCCOC2)cnnn1C C1(NC(CCC#CC)=O)CCN(C(=O)C#CC(C)C)C12CC2 c1(CNC(C(c2nscc2Br)N(C)CCn2ccnc2)=O)cc(Cl)nc(Cl)c1 C#CC1(O)CC(C(N2CCCCC2CNC(c2oc(SC)cc2C)=O)=O)C1 c1(NC(C(C)CF)=O)cccc(F)c1C#N C(=O)(C(CC(C)C)C(C)C)NCCC1CCN(C(C(C(=C)C)(C)C)=O)CC1(F)F CN1CC(N(C(=O)CCCCC(=O)OC(C)(C)C)C2COC2)CCC1C(F)(F)F CC1(C)CCCCC1=CC(N1CCOC(C)(CNC(=O)CN2CC3CC3C2)C1)=O C1(C(N(CC(O)CNC(=O)CCOC2CC2)C)=O)CSC2(C)CCC(=O)N12 C(=O)(CCCCC(N)=O)NC(C)C(C)NC(C1(S(N)(=O)=O)CCCC1)=O Cc1nocc1CC(=O)NC(C)CN(C(=O)C(NC(C)=O)=Cc1cccs1)C c1(C(=O)NC(CC=C)CNC(C2CC2CC)=O)cc([N+](=O)[O-])ncc1Br c1(C(N2CCC(CNC(CC(CC)O)=O)C2(C)C)=O)cc2c(nc1O)CCCC2 O=C(CO)N=c1ccn(CC(=O)Nc2cc(Br)c(F)cc2Cl)c(O)n1 n1(CC)ncn(NC(=O)C2CCC=CC2NC(=O)C(C)CN(C)C)c1=O N1(C(C(CC)SC)=O)CC2(C(=O)NCC3(C)CCCO3)CCC1CC2 C1(CC)(CO)CCN(C(C2C3COCC23)C(=O)NC2CC(F)(F)C2)CC1 Cc1nocc1C(=O)NC(C1(O)CN(C(=O)CC(=O)OCCC(C)C)C1)C C(=O)(C#CC1CCCOC1)NCC1CC(OC)CN1C(C1CCC(=O)N1)=O c1(NC(CCC)CCCNC(=O)CCOCCOCC)ncc2ncnc-2[nH]1 O=S(=O)(c1c[nH]ccc1=NC1COC2(CCC2)C1)NCC1(Br)CC1 C(=O)(C(C)C(O)C(C)C)N1CCN(C(Cc2cc(C)nn2C)=O)C(C(C)C)C1 N1(C(C(C2(O)CCN(Cc3ccc(N(C)C)nc3)C2)C)=O)CCc2sccc2C1 c1(OC)ncc(CN2CCOC(CNC(c3conc3C)=O)C2)cc1Br C(=O)(N1CCCc2nncn21)C1(C(=O)NOCc2cccn(C)c2=O)CCCO1 N1(C(CSCCN(C)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)C12CCC2 Cc1ccc2nc(C)c(C(=O)OCC(=O)NCCCc3cccc(Br)c3)n2c1 n1(CCC(=O)NCC2CN(C(C(COCC)C)=O)C2)cnc2ccccc12 CCCC(CCC)C(=O)N1CCC(O)(Cn2cc(CCN(C)S(N)(=O)=O)nn2)C1 Cn1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)cs2)=O)C2CCC2)ccc1=O c1(C(N(C2(C3CN(C(=O)CC4CCC5CC45)C3)CC2)C)=O)cc(Br)ccc1N c1(OC)cc(N)cc(OCCc2ccc3cc[nH]c3c2)c1[N+](=O)[O-] C1(NC(c2cccc(OC)n2)=O)CCOC12CCN(C(=O)C(O)P(C)(C)=O)CC2 c1(C(C)=O)cnn(C)c1C(=O)NC(CNC(=O)CC(O)Cc1ccccc1)CO Cc1cc(O)ncc1NC(=O)C(C)N(C(c1cc[nH]c(=N)n1)=O)C1CC1 CC(C)CC(C(=O)N1CCC(CCNC(=O)Cc2ccc(Cl)c(F)c2)C1)C(N)=O c1(C(N2CC(N(C(=O)COC(C)C)CC)C2)=O)cnc2c(C)cccc2c1 c1(C(COC(C2C(C)(C)CCO2)=O)=O)cnc2n1CCC2 Cc1ccc(C(=O)NC(CNC(C23CSC(C2)C3)=O)C(C)(C)C)n1C CC(C)C(C(=O)N1CCC(C(=O)NC(c2ncccc2F)C)O1)C1CCC1 c1(N2C(C(=O)NCCC(F)(F)F)CCC2)nccc(Br)n1 C1(C2CC2)(N(C(=O)C(O)C2CN(C(=O)CC3CC(=O)C3)C2)C)CC1 c1(C(N2CC=C(CNC(C(C)CC3CCC3)=O)CC2)=O)n[nH]c2c1CC(C)(C)C2 Cc1cn(C)cc1C(=O)NCC(C)(C)CNC(C1CC(C)(c2ccccc2)C1)=O CCCCC(=O)N1CSCC1C(=O)N(C)CCc1cccs1 C1(C(=O)OC)CCC(C(=O)NC(C)CN(C(=O)CCCOC2CCOCC2)C)C1 C(=O)(N=c1[nH]cc(C(=O)O)nc1Cl)C1N(Cc2nc(C)sc2)CC(C)C1 C(=O)(CC1=CCOCC1)NCC1C(C(N(C(CF)CF)C)=O)C1 c1(C(N2CC(C(C)NC(c3cscc3F)=O)OCC2)=O)cc2c(ncn2C)s1 C(=O)(C1=C(C)OCCS1)NCC(CC=C)C(=O)NC1COC(C)(C)C1 c1(NC(C2C(C(=O)NCC(C)(C)N(C(=O)C=C(Cl)Cl)C)C2(F)F)=O)ccc(F)cc1 C=CC1COCC1NC(=O)CC1CC1CNC(c1cccc(CO)c1)=O.C(N)=O Cc1cccc(C(=O)NCC(C2CCN(C(c3cc(C)n(C)n3)=O)CC2)F)c1C C1(CNC(c2nncs2)=O)CCN(C(C23CC2C3)=O)CC1 C(=O)(C(C)(C(C)C)OC)NCC(=O)NCC1(OCC)CN(C(c2ccoc2)=O)C1 C(C(C)CC(=O)NCC1CCN(C(=O)CNC(c2ccco2)=O)CC1)OC C1(C(N2CC3C(CNC(C4(COC)CCOCC4)=O)(C3)C2)=O)CC(=O)OC1(C)C CC(F)(C(=O)N1CC(NC(=O)CNC(N)=O)C1)C1CC1 C1(C(=O)NC2(CC)CCOC2)C2CC2CN1C(=O)CC1C(C)(C)C1(C)C C1(F)(CNC(=O)CC2CC(n3cnnc3)C2)CC(NC(c2cncnc2)=O)C1 c1(CC)nn(C)c(NC(C)=O)c1NC(c1ccncc1C)=O C1(CC(=O)N(CC)CC2CC2)CN(C(C2CCC(C3CC3)C2)=O)C(C)(C)C1 c1(C(=O)NC(CC)CN(C)C(C2CCC2C(F)F)=O)cscc1SC N1(C(COCCCOC)=O)CC(C)CN(C(=O)CCCc2ccccn2)CC1C O=C(C1Cc2ccccc21)NC1CCN(C(=O)C(c2ccccc2Cl)O)CC1O c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cnc(N(C)C)c(Br)c1 c1(N)sc(C2CCCOC2)nc1C.CCCCSCC(=O)N(CCN)CC1CC1N CCCCC(C(=O)NC1(C)CC(NC(=O)Cc2cc3ccccc3o2)C1)C(C)C C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(c2n(COC)ncc2)=O)CC(O)C1 c1(C(N2CC(C)(NC(c3cn(C(C)C)nn3)=O)C2)=O)ccc2c(c1)C(C)C(C)O2 C1(CP(C)(C)=O)C(=O)N1.C(c1ccc(OC)cc1)=CCNC1CC(C(=O)OC)C1 c1(C(=O)NCC2C3CN(C(C(C)(C)F)=O)C2C3)ccc2n[nH]cc2n1 C=CCCCC(C1CC1)NC(C1CC1C(C)NC(c1ccc(F)cn1)=O)=O N1(CC)CCOCC1C(=O)NC(COC)CC(=O)NCCN1CCOC1=O c1(NC(=O)CCC2CCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)cccc2c1CCO2 N1(C(C=CC(=O)OCCCC)=O)CCC(O)(CNC(c2cnccc2OC)=O)CC1 c1(N2CC(C(=O)NC(C3CCN(C(c4cscc4F)=O)C3)C)C2)ncccn1 c1(OC)ncc(C)cc1NC(C1(NC(C2(C)CC3C=CC2C3)=O)CC(F)C1)=O N1(C(c2cccc(CC)c2O)=O)CC2(CC(NC(=O)C(C)=CC3CC3)CO2)C1 Cc1cc(C)c(C(=O)NC2CCCC2n2cc(CCS(N)(=O)=O)nn2)cn1 n1(CC(=O)NCC2C(NC(CCCc3ncc(C)o3)=O)C2)nc([N+](=O)[O-])cc1C N1(C(C2C(CCC)CCC2)=O)CCC2CCC(NC(=O)CCCCN(C)C)C12 CC12C3C4C1C1C2C3C41C(=O)NCC1CCN(c2ccccc2)C1 C1(C(=O)NC(CNC(CCC(C)C)=O)CO)CCCc2ccccc2C1 n1(C(C)(C)C)ncc2c1CCCC2NCc1cccc2nncn12 C1(CNC(C2CC(CNC(=O)COC(=O)CO)C2)=O)Cc2nccn2C1 c1(CC)cnccc1C(N1CCC(CC)C1CNC(C1CC(C)=NO1)=O)=O C(CC(F)F)(C(=O)NC1CC1)NC(CN(C(=O)COC1CCC1)C)=O Cc1ncn(C)c1C(=O)N(C)Cc1cn(C2CCN(C(C)(C)C)CC2)nn1 c1(C(=O)OC)oc(CN2CCSCC2)cc1C.n12cc(nn1)C(C)NC(=O)CC2 C1(C(=O)NC2CCC(NC(Cc3c(C)n[nH]c3)=O)C2)CC1C1(C)COC1 N1(C(C(C(C)C)O)=O)CC2COCCC2(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 C(CC1=CCCCC1)N(C(C1(CC=C)CN(C(C2CC(C3CC3)C2)=O)C1)=O)C c1(OC)ccc(F)cc1CCC(=O)NCC(O)CNC(C12CC(C1)C(C)(C)O2)=O Cc1nc(C(=O)N(CCCOCCN(C)C(c2sccc2Cl)=O)C)sc1C c1(C(C)CC(=O)N(C2CCCC2)CCNC(C2CCCSS2)=O)ccc(F)cc1 C1(N(C)C)CN(C(=O)C(O)CCNC(c2cccc(O)c2)=O)CC1F C#Cc1ccc(C(=O)NC2CC3(CCOCC3)C2)cc1Cl C1(OCC)CCCCC1n1cc(C(N2CC(COCP(C)(C)=O)C(O)C2)=O)nn1 C1(CCC)(NC(=O)CC(C)n2cccn2)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C(C(C)(C)CC(=O)NCCSCc1ccccc1)OC.C12CC1CC(=O)N2 N1(C(CC2N(C(c3cc(C)ncn3)=O)CCCC2)=O)CCCC2(C1)N=N2 c1(C(=O)OC)ccc(CN2CCCC2CNC(C2(c3ccccc3)COC2)=O)s1 c1(CN(C(=O)OC(C)(C)C)CC2CCCC(CC)C2)c(C)[nH]c2cccc(Br)c12 N1(C(CCC#C)=O)CC2(CNC(=O)C=CCCC(C)C)CC1CCO2 S(=O)(=O)(c1ccc(F)c(F)c1F)N1CC(C(=O)NCc2c(O)cccc2F)C1 c1(CN2CCC(C(=O)Nc3onc(C)c3Br)C2)cc(Cl)cc(Cl)c1Cl C(=O)(C1=C(C)OCCS1)N(C1(C2CCCN2C(=O)C(C)C#N)CC1)CC C12(CNC(c3c(CC)c[nH]n3)=O)CC1CN(C(C1CC=CCC1C(F)(F)F)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cnc(CC)cn1 C=C(C)CC(C)C(=O)NCCCCN(C(=O)C(C)(C)C1CCCCO1)C CS(=O)(=O)c1cscc1C(N1CCC(F)(F)C(CNC(=O)Cc2cc[nH]c2)C1)=O C(=O)(C(C)C1CC1)NCCN(CCOCC)Cc1nncs1 c1(NC(=O)NCCc2nnc(C)o2)cnc2n1CCOCC2 c1(C(=O)NC(C(=O)OC)Cc2cc(Cl)sc2Cl)ccc(OC(F)(F)F)cc1F C1(C(=O)NCCN(C(=O)Cc2csc(C)n2)CC)CCCCC(C)(C)C1 C12(CNC(c3cc(F)ccc3F)=O)CCC(CC1)N(C(=O)C(F)=CCCF)C2 N1(Cc2cn(CC)nn2)CCC2(CCN(C(=O)Cn3ccc(C)cc3=O)CC2)C1 C(=O)(CCCC(C)(F)F)NC1C(N(C(C(=O)N2CCCC2)C2CC2)C)CCCCC1 c1(NC(C2OCCN(C(C(C)=CCC)=O)C2)=O)c(CO)cccc1C N1(C(C2(CCCC)CCCCC2)=O)CC(NC(=O)CSCC(C)C)CC(F)C1 N1(C(CC)=O)CCC(C)(CNC(=O)CCc2scnc2C)C1 c1(C(=O)NCC2CC(CNC(=O)C(F)OC(F)(F)F)CO2)cccc(CO)n1 N(C(=NCCCCl)NC1CCC(=O)NC1)CC1(NC(=O)OC(C)(C)C)CC1 N1(c2c(OC)cncn2)CC2(CCC(NC(c3cc4cccnc4s3)=O)C2)C1 CCCC(CC)C(=O)NC(c1ccccc1F)CNC(c1cnc(S)[nH]1)=O C(=O)(C#CC1CCOC1)NCC1C(NC(C=CC(=O)OC(C)(C)C)=O)C1 C1(C(=O)NCC(NOC)=O)CN(C(=O)C=Cc2nccs2)CC12CCC2 N1(CC(=O)NCCC)CC2CCC(NC(c3ccc4c(c3)OCCO4)=O)CC2C1 c1(C(N2CC(OCC(=O)N(CC(CC)C)CC)C2)=O)sccc1CO C1(C(=O)NCC2CC(NC(CN3C(C)CCC3)=O)C2)CCOCC1(C)C C(=O)(C(CO)C(F)(F)F)N(CCCC(=O)Nc1c(COC)csc1)C c1(CN2CCN(C(C)CC3(C(F)(F)F)CC3)C3C2C3)c2cc(Br)ccc2nn1C N1(C(C(C)(O)C2CCOCC2)=O)CCC2(CCC2)C(NC(=O)C=C2CCC2)C1 c1(C(N2CC(NC(c3c(OC)c(F)ncc3)=O)C(O)C2)=O)cc(F)c(F)cc1N C1(NC(COC2CN(C(C(C)(F)F)=O)C2)=O)CC2OCCCC12 CC(C)CC(O)C(C)C(=O)N1CC(O)(CCNC(=O)Cc2ccc(O)c(Cl)c2)C1 c1(OC)ccc(C(N2CC(C)(C)C2CO)=O)c(C(F)(F)F)c1 CC(C)(C)C(O)C(=O)NC1CC(CCNC(=O)CCCc2ncco2)C1 C(CCCCNC(c1[nH]nnc1C1CC1)=O)NC(=O)COC1CCCOC1 C(=O)(C(CO)C(F)(F)F)NC1(CC=C)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 C1(CC)CCCCC1C(=O)N(CC(C)NC(=O)C(C)(C)C1CCCCC1)C C1(C(=O)NC(C)C(CO)NC(c2ccc(O)nn2)=O)CCN(C2CC2)S1(=O)=O C(=O)(C(C)CCCc1ccccc1)N1CCC(C)(CNC(C=CCCC)=O)C1 C(C(CCN=c1[nH]c(=NC(C)CCN(C)C)[nH]c2ccccc12)C(C)C)OC C(c1cc(Br)ccc1Sc1ccccc1)=CC(=O)N1CCC1 CCCCS(=O)(=O)CC(=O)NC1C2CC1N(C(=O)Cn1cc(C(F)(F)F)nn1)C2 c1(NC(C2N(Cc3cccc(OC)c3F)C3C(C2)C3)=O)ccc2nc(O)[nH]c2c1 c1(C(N2CCC(CCOC)(NC(=O)CN(C)C)C2)=O)coc2ccc(Br)cc12 N1(C(COCC#C)=O)CCCC(C)(CNC(c2ncccc2C)=O)C1 C(=O)(CCCN(C)C)NCCC(C)NC(c1cccnn1)=O N1(C(c2n(C)nnc2)=O)CC2CCCCC2(CNC(c2c[nH]c(C#N)c2)=O)C1 Cn1cc(C(C(=O)Nc2cccnc2)NC(c2ccc(I)s2)=O)cn1 N1(C(c2scc(C)c2)=O)CC(CCNC(=O)C=CC(=O)NC2CC2)C(C)C1 c1(NC(C2C(C3CCN(C(C4(C)CC(=C)C4)=O)CC3)C2)=O)nc2cccnc2s1 C1(NC(C(N2CC(C(C)C)SCC2)=O)=O)CCc2c(cnn2CCO)C1 c1(CC)ccc(C)c(NC(=O)C(Cn2cncn2)NC(C2CC(=O)C2(C)C)=O)c1 C1(C#N)(C(N(C(CCNC(c2cccc(OCCC)c2)=O)C)C)=O)CC2(CC2)C1 C1(F)(C(N(C)CC2N(C(c3c(C)cns3)=O)CCC2)=O)CCS(=O)(=O)C1 C1(NC(C23CC(C)(C2)C3)=O)CCC(NC(=O)C(O)(C2CC2)C2CC2)CC1 N1(C(c2cc(Br)cs2)C(=O)NCC(=C)C)CCC(CN(C)C)CC1C CC1CN(C(C2CC(C)(C)C2)=O)CC2(CCN(C(=O)C(F)(F)c3nccs3)C2)O1 CC1(C)CC(NC(C2(C)CCCNC2=O)=O)CCN(C(=O)COC2CCCC2)C1 CC(=O)CCN=C(NCCC1SCCS1)N1CCN(c2nnc(C)c(C)n2)CC1 CC(=O)CCCC(=O)NCCC1CC(NC(c2cn3c(n2)SCC3)=O)C1 C1(NC(c2cc(CCCC)oc2C)=O)CN(C(C2CC(F)C(=O)N2)=O)CC12CC2 N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1CC(F)F N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2cncnc2O)C2CCCCC2C1 N1(C(C(C)C)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC12CCCCC2 N1(C(C(CC(C)C)CNC(C2CC3CCC3C2)=O)=O)CC2(CCC2)C12CCC2 C(=O)(C(C)(CNC(=O)COc1ccsc1)CC)NCC1N(CC)CC1 N1(C(c2ccc(C#C)c(F)c2)=O)CCCC2CN(C(c3scnc3C)=O)CCC12 N1(c2ncnc(C)c2Br)CCc2sc(C(=O)NCCC3CCOCC3)cc2C1 N1(C(CC(CC=C)(C)C)=O)CC2CC3CC2C1C3NC(c1scc(C)c1C)=O c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)C(C)C)cnn2c1NCCC2 c1(N(CCC)CCNC(=O)CN2CC3CCC2C3)nc2c(cc1C#N)CCOC2 CC1OC2(C(N3CC4CC4(NC(c4ccc5c[nH]nc5n4)=O)C3)=O)CCC1CC2 N1(C(C2CC(NC(C=CCCC(C)C)=O)C2)=O)CC(C)OC(C)(C)C1C Cc1ccc2nc(CSCc3coc(C(=O)O)n3)cc(=O)n2c1 C1(OC)CCC(C(=O)NCCCCCCNC(c2coc(N(C)C)n2)=O)CC1 c1(C(=O)NCC(CCCC)NC(C2(S(C)(=O)=O)CCC2)=O)cc(C)c(O)c(N)c1 C1(N(C(c2ccccc2C)C(=O)OC)CC2CCOCC2)CCC2COC1O2 c1(C(C)C)ncc(Cl)c(C(=O)NCCCCN(C)C(c2ncncc2F)=O)n1 c1(C(=O)NCC2CCN2C(=O)CC2C=CCC2)cccc(N2CCNC2=O)c1 CC1CCCCCCN1C(C1CC2CCC1N2C(C1(CCF)CCC1)=O)=O C1(C)(NCC(C)=CC(N2CCC2CC(=O)Nc2ccsn2)=O)CC=CCC1 C1(C(N2CCC(=C)C2)=O)CCN(C(=O)CCc2cnco2)CC1C c1(C(N2CCC(CN(C(=O)CC3C=CCCC3)CC)CC2)=O)cnc(O)c(F)c1 Cc1cc(C#N)nc(Nc2cnc(Cl)cc2C(=O)Nc2cncc(C#N)c2)n1 N1(C(c2sc(C(=O)OC)c(C)c2)=O)CCCC2CN(C(C3CC(O)C3)=O)CCC12 C1(C#CC(=O)NCCOC2CN(C(c3cc(C(F)F)[nH]n3)=O)C2)(CC)CC1 C1(CNC(C(C2CC2)OCC)=O)CN(C(c2cn(C)nc2COC)=O)CCCO1 c1(N(CCCC)C(=O)NC(CCCC)CC)cccc2scnc12 N1(C(C(c2ccc(Br)cc2F)C)=O)CC2(CCCC2NC(=O)CNC(=N)N)C1 c1(C(N2CC(C(C)NC(c3cccc(SCCC)c3)=O)C2)=O)cc(F)cc(F)c1 N1(C(c2c(OC)nsc2OC)=O)CCC(CCNC(C2CC2F)=O)C(F)(F)C1 C#CC1CN(C(c2cc(C)nn2CC)C(=O)NCC(=C)C)CCO1 c1(CC(=O)NCC2CN(C(=O)C(F)=CC3CC3)C2)cc(Cl)ccc1O c1(C(=O)NC(CN(C(=O)C(N2CCNC2=O)C)CC)C)ccc(O)c(C(C)C)c1 C1(CNC(C=CC=CC)=O)CN(C(c2cc(F)c(F)cc2F)=O)CCC1(F)F CC1CC(C(N2CC=CC(C(=O)NCCC3C=CCC3)C2)=O)CN1C CC1(C)OCCC1NC(C1CC(CCNC(=O)CCN2CCCC2)C1)=O C1(C(=O)OC)CCCN(CC(=O)Nc2ccccc2Oc2ccccc2)C1 O=C1NCC(C(=O)N(C2(C(=O)NC3(CCF)CCC3)CCC2)C2CC2)N1 C=C(C)CCCC(=O)N1CC(CC(N2CCC(OC)C2(C)C)=O)C2(CC2)C1 N1(c2ccnc(C(C)C)n2)CCC(NC(=O)C(C)NC(c2ccco2)=O)C(C)C1 C1(CNCc2cn(C(C)(C)C)nc2)COCC(C)(C)O1.N12CC(C)(C1)CC2=O C(=O)(C(F)(CNC(=O)C(c1cnn(C)c1)=O)C(C)C)NCC(=C)C C(=O)(CCN(OC)C(=O)C1(F)CN(C(=O)C(C)OCCN(C)C)C1)OC Cc1cccc(CN(C)Cc2nc(C(=O)NC(C)CNC(=O)CC(C)C)sc2)c1 CC1(C)CN(C(=O)CC2(OCc3cccc(F)c3)CC2)CC(C)O1.C1(C(=O)N)CC1F c1(CC(=O)NCCCNC(C2N(CCC)CCCC2)=O)cc(F)ccc1Cl CSC1=C(C(=O)N(C)CCN2CCN(C(C3CCSC(C)C3)=O)CC2)CCCC1 C1(C(=O)NC2CCC(NC(CC3C(C)=NNC3=O)=O)C2)CCCCC1(C)C CC1CN(C(C2CCC=CCC2)=O)CCN1C(C12CCC(F)(CC1)C2)=O N(C(=NCC1CCC2(CC2)C1)NC1CCOCC1)CC(C=C)(F)F Cc1ccc(C=CC(N2CCN(C(=O)CC(C)(C)F)C(C3CC3)C2)=O)cc1 NS(=O)(=O)c1ccc(C(=O)NC2CCC23CN(C(=O)CCc2cnc(O)[nH]2)C3)s1 C(=O)(C(C(C)(C)C)OC)NCC(C(=O)NCc1c(OC)cccc1)O C1(CNC(c2cc(C)[nH]n2)=O)CCCC2(CN(C(=O)CC3(N4CCCC4)CC3)C2)O1 c1(CNC(C2CC(F)CN(C(c3sccc3Cl)=O)C2)=O)ccc(CO)cc1F N1(C(C2CC3C=CC2C3)=O)CCCC(O)(c2cn(-c3ccc(Cl)cc3Cl)nn2)CC1 c1(NC(C2CN(C(=O)NC(C(=O)OC(C)C)C)C2)C)ccc(Cl)c(O)c1 CC1(C)CCCN(C(C2CCC2C(C)(C)C)=O)C1C(=O)NC1(C)CCCC1(F)F C1(C(=O)NCCCCSC)CCC(C2CC2)N1C(=O)Cc1cccnc1O CC(C)C(CNC(C1CCCCCC1)=O)C(=O)NCCN1CCCC1 CCC(C)(CNC(c1cc(OC)ns1)=O)C(=O)NCCN(C)C1CC1 N1(C(CC2CCCN(C(C3(C#C)CC3)=O)CC2)=O)CCCCC(C)(C)C1 CC1CC2CN(C(=O)CCc3nccn3C)CC2N1C(C1CC2C=CC1CC2)=O N1(C(C(=O)NCC(CC)NC(=O)OC(C)(C)C)=O)CC(C)(C)OC2CCCC12 C(=O)(C(C)CS(C)(=O)=O)NCC12N(C(C3CCC(CC)O3)=O)C(CC1)CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCC(CCC(=O)N(CC(C)C)CC(C)C)C1 C1(NC(C2CC3(C2)CC3(F)F)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(C(CC=C)(C)O)=O)CC2(C=C(C(=O)NCC(C)CC(F)(F)F)CO2)C1 C1(C)(CC(=O)N(C)CC2CCN(C(C)=O)C2)CCN(C(=O)Cc2cnc(C)s2)C1 O=C1NCCN(C(C2C(O)CCN2C(=O)Cn2cccc2)=O)C1CCO Cc1snc2sc(C(N3CC(C)(NC(=O)CC4COCCO4)C3)=O)cc12 C1(CNCC2(C)OCCO2)CN(Cc2cc(C(F)(F)F)cc(Cl)c2)CCC1O c1(CNC(C2C(CC)OCC2)=O)cccc(C(=O)NCC2=NOC(C)C2)n1 N1(C(CC(C(=O)OC)C)=O)CC(NC(=O)CSC2CC2)C(S(C)(=O)=O)C1 c1(C(=O)NCCC2CCC(NC(=O)C=CBr)C2)cc2n(n1)CCO2 c1(C(N2C(CNC(C(CC)=CCCC)=O)CC2)=O)ccc(F)c(C(C)(C)C#N)c1 C12CCC3(CC1)CN(C3)C(=O)CN2Cc1ncc[nH]1.c1(NC(C)=O)cncn1C C=CC1(NC(=O)CC2C3CN(C(C45CCC(C4)C5)=O)CC23)CCCCC1 c1(C(=O)NC2CC(NC(C3(C)CC3(F)F)=O)C2)ccc(-c2cncnc2)cc1F C1(CNC(C(C(C)c2ccccc2)N)=O)CC(=O)N(C)C1c1ccc(Cl)c(Cl)c1 C=CC(CCC)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(C1)C(C)O2 O=C(C1=CCCCCC1)NCC(C1CCOC1)NC(=O)CC1(CO)CC1 C(C(C)(C)CCO)NC(C(C1CN(C(C2OCCC2C)=O)C1)OC)=O CN1CC(NC(C2CN(C(C3CCC(C)(C)CC3)=O)CC2(F)F)=O)C2(CC2)C1=O C1(NC(C2C(C=C)C2)=O)CN(C(=O)CCCc2nc(C3CC3)no2)CC1OC c1(C(N2CC3(CN(C(c4c(CC)c[nH]c4)=O)C3)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NCC(CC2CC2)CO)(CC)CCN(C(c2cscc2C)=O)CC1 c1(C(N2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)=O)ccc(C)c(F)c1 N1(C(C(CCN(C)C)O)=O)CC(NC(=O)CCc2cnc[nH]2)CC(O)C1 C1(C(N2CC(OC)C(C(=O)NC34CCCC3C4)C2)=O)CC(C2CC2)=NO1 C=C(Cl)CC(C(=O)NCCc1cnn(C)c1)NC(=O)CC=CC(C)(C)C c12cc(ccc1[N+](=O)[O-])SC2.N1(C(=O)OCC)CCOCC1C(C)(C)C C1(C(N2CC(N(C)C(C3CC(F)C3)=O)C2)=O)CC(N(C)C)CCO1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(CCN(C(c3cc(O)cnc3N)=O)C2)C1 C(=O)(C1COc2ccccc21)N(C1CN(C(=O)C(c2ccccc2)C2CC2)C1)C c1(N(C(=O)NCC(C)Oc2ccccc2Br)C)cccc(Br)c1Cl CCC(C)CCCCC(=O)N1CCC(NC(C2CCS2(=O)=O)=O)C(C(N)=O)C1 c1(C(=O)NCC2C(NC(C=CSC)=O)C2)ccc(C(F)(F)F)nc1N Cn1nccc1C=CC(N1CCCC1C1CCN(C(C2(C)CNC(=O)N2)=O)CC1)=O Cc1[nH]c2ccc(C(=O)NCc3nc(CNC(=O)CC4CC4)cs3)cc2c1C c1(C(N2CC(SC)C(NC(C3CC3[N+](=O)[O-])=O)C2)=O)cnc2cc(O)ccc2c1 C12(C(=O)NCC3CC(NC(c4cocn4)=O)C3)CCC(CO)(CC1)C2 c1(OC)ccc2cc(C(=O)NCCCC(C)NC(=O)C(C)SC(F)(F)F)[nH]c2n1 N1(C(c2nncn2C)C(=O)NCCOC)CCC2(CC1)OCC(O)C2O c1(N(C)C)ccc(C(=O)NCC2(NC(=O)CN3CC4CC4C3)CCOC2)cc1 C=C(C)CC(C(=O)N1CCN(C(=O)C(c2cnn(C)c2)C)C(CC2CC2)C1)OC C1(CCNC(C(C)=CC)=O)(OC)CN(C(c2cnc(-c3ccncc3)s2)=O)C1 C1(C(N(CCCO)CCC)=O)CCCN(Cc2cc[nH]n2)CC1 Cc1c(C(=O)NC2CC(NC(=O)CC3(O)CC3)C2)oc2cc(Cl)ccc12 c1(C(=O)NCC(CN(C)C(C2CCCN2C)=O)O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCCC2CCN(C(c3c(C)cncc3)=O)CC2)ccnc2[nH]cnc12 N1(CC(c2ccccc2)OC)CC2CCCN(C(c3csc4nccn34)=O)C2C1 N1(C(C(CCC#C)NC(c2coc(CO)c2)=O)=O)CCCC2(CCCO2)C1 N1(C(C(N2CCC(O)CC2)C)=O)CCC(NC(=O)CC(O)C2CC2)CC1C C1(NC(N2C(CC)C(=O)NCC2)=O)COc2cc(C)c(C)cc2C1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC(C)C2)cnn2ccn(C)c12 C1(COC)CCC(C(=O)NCCN(C)C(=O)C2CC2)C1 c1(-n2cc(CCC(C)C)nn2)cnc2c(c1)CNCC2 c1(SC)cccc(N2CC3CC(NC(C4(S(N)(=O)=O)CC4)=O)CC3C2)c1[N+](=O)[O-] C1(CNC(C(C)OCC)=O)CCCC2CN(C(=O)Cc3nc(C)no3)CC12 Cn1cncc(C(=O)NCC2CN(C(=O)C(O)C(F)F)CCO2)c1=O CC(C)(CC(=O)NCCN1CCCN(C(C2CCC23CCCO3)=O)CC1)C(F)F C=CCC(C)C(=O)N(CCCN(C)C(c1cccc(OC(C)C)n1)=O)C c1(C(N2CCC(O)(CNC(C(C)C)=O)C2)=O)cc(C2CC2)nc2c1cnn2C C1(OCC(=O)OCCOC)CN(C(=NCCSC)NC(c2ccccc2)C)C1 CCCCC(F)C(=O)N1CCN(C(=O)CNC(c2cc(SC)c(C)o2)=O)CC1 C(=O)(CC(C)C(=O)NC(C1CC1C(N1CC(C)(C)C1)=O)C)OC c1(C(C)CC(=O)NCC2(NC(=O)CN3CCC(F)C3)CCCC2)ccc(F)cc1 O=C(CCCC(F)(F)CO)NC1CCCN(C(c2cc3c(nn2)CCCO3)=O)C1 c1(CNC(CCN(C(=O)CCC(=O)N(C)C)C)=O)cccc(F)c1 c1(C(=O)NC(C(=O)NC2CCNC2=O)C2(C)CC2)cnn2cccc2c1 N1(C(COCCCCC)=O)CCN(C(C2(SC)CCC2)=O)CC1CC1CC1 Cc1cc(=NC(=O)C2CC(F)CN(C(c3ccc4cnc(C)n4c3)=O)C2)[nH]n1C C(=O)(C(C)(C)F)N(CCN(C(C(C)OCCC=C)=O)C)C Cc1cc(=NC2CCN(C(c3cn(C)nc3C(C)(C)C)=O)CC2C)[nH]c(CO)n1 C1(F)(C(=O)NCC2C(CNC(=O)C(O)C3CC3)C2)CC=CCC1 Cc1cc(C(C)Nc2cc(NCC(c3ccccc3F)(F)F)ncn2)cc(C)c1 N1(C(CN(C2CC2)CC)=O)CC2CC(NC(=O)COC3CCCOC3)CC1C2 C1(C(=O)OC)CN(C(=O)C(C)(C)C)CC1c1cccc(Br)c1 CC1CCc2c(C(=O)NC3(C)CN(C(C4CC4c4ccsc4)=O)C3)csc2C1 C=CC(C)(CC)C(=O)NCCCC(C)NC(c1ccccc1SCC(F)(F)F)=O C1(NC(=O)CCC2CC2)CCOC12CCN(C(=O)C(=Cc1cccnc1)F)CC2 C(=O)(CC(=O)N(C1CCN(C(c2snnc2C(C)C)=O)C1)CCO)OC C1(C(=O)NCCC2(O)CN(C(C34CC(CO3)C4)=O)C2)(OCC)CCOCC1 C(=O)(NNC(=O)C(=O)OCC)c1nc(-c2cncc(C(=O)OCC)c2)sc1 CCCCC(C)(F)C(=O)NC1CCCCC1NC(=O)CN=S(C)(C)=O C1(C(C)C)CCC(C(=O)NCC(C2(O)CN(C(C3CC(C)CO3)=O)C2)(C)C)CC1 c1(C(=O)NC(C(=O)NCCS(=O)(=O)NC)C2(C)CC2)cccc(C)c1C C(=O)(CCS(N)(=O)=O)NCC1(O)CCN(C(c2c(OC)c(C)sc2)=O)C1 C1(C(=O)OC)CCCC(C(=O)N(C)CC2CCCN2C(=O)C(C2CCC2)OC)C1 CC(C)(C#N)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccncc1)O c1(C(=O)NC2(CO)CCCN(C(C=C3CCN(C)C3)=O)C2)ccc(C#N)cc1O C(=O)(C#CC1(C)CCCO1)NCCC(C(C)C)NC(c1ccc(CC)c(Cl)c1)=O c1(CN2CC(CC#N)N(C(=O)Cn3nccn3)CC2)cc(Br)cc(F)c1F C1(CCNC(c2n(CC)cnc2)=O)CCCN(C(c2c(C)ncn2O)=O)CC1 C1(NC(C(CC2CCCCC2)OC)=O)CN(C(=O)C(N)=O)CC1C c1(OCCN2C(=O)C(C)(C)C2)cccc(C#N)c1.CCC(C(=O)OC)N c1(C(N(C2C3CN(C(C(C)NC=O)=O)CC32)C)=O)cc2nc[nH]c2cn1 C1(C(CNC(C(CC)O)=O)C)CCN(C(=O)CCCCNC(=O)CC(C)C)CC1 N1(C(c2n(CCOC)cnn2)C(=O)NC2CCCCC2)CCC(C#N)CC1 CC1(C)C(C)(C(N2C3CC2CN(C(c2cc([N+](=O)[O-])sn2)=O)C3)=O)C1(C)C c1(OC)ccc(N)c(C(=O)NCC2CN(C(C3CC4CC4C3)=O)CC2C)c1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCCN(C(c2c(CC)nc(C)s2)=O)C1)C c1(C(=O)NCCNC(C2C3CCC2(c2ccncc2)C3)=O)ccc2sncc2c1 Cn1cnc(C(N2CCC(CNC(c3c(C(F)F)cnn3C)=O)C2)=O)cc1=O C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(C2CC2)C1 Cc1nn2c(c1CNC(=O)C(O)CC(F)(F)F)CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(SC)nc(Cl)c(COCC2(C(=O)Nc3cc(Cl)c(OC)cc3Cl)CC2)c(Cl)n1 C1(C(NOCC(=O)NC2CC(=C)C2)=O)CCOCC1(C)C C(C)(C)(CCC(=O)NCc1ccccc1O)NC(c1ccc(CC)cc1)=O c1(NC(C(C(C)SC)N)=O)c(C)cccc1F c1(NC(C(CO)NC(Cc2c(C)n(C)cn2)=O)=O)ccc(O)cc1F c1(OC)cnc(C(=O)N(CCNC(C2CC2(C)C)=O)C2CC2)c(F)c1 N1(C(C2CCN(CC)C2)=O)CCC2(CC2C(=O)NC2(C)CC3CCC2C3)C1 C1(CNC(CN(CCOC)C(C2OCCC2C)=O)=O)CCCC1CF C1(C(=O)NCC2(C#N)CCC2)CN(C(C2CC3CCC2CC3)=O)CC12CC2 c1(C(=O)NCCCCCNC(Cc2n(C)cnc2)=O)cc(C#N)n(C)n1 N1(C(c2ncc[nH]c2=O)=O)CCN(C(=O)COc2ccc(Cl)cc2Cl)CC(O)C1 C(C1c2ccccc2CCN1C(c1cccn1C)=O)NC(CSCCOC)=O C12(NC(CCCC)=O)CCN(C(C3CCN(c4ccncn4)CC3)=O)CC1C2 N1(C(Cc2ccn(CC)n2)=O)CC(OC)C(OC)C1CNC(=O)CC1CC12CC2 Cc1cc2ccc(C(=O)NC3CCCCC3N(C(=O)C(=O)NC(C)C)C)cn2c1 CC1Oc2c(C(N3CC(CNC(c4ccnc(CO)n4)=O)C3)=O)cccc2C1C C1(NC(C(CCCC)O)=O)CC2CN(C(=O)CC(O)c3cc(C)cs3)CC2C1 C1(C(=O)NC2CCN(C(c3ccc(C(C)C)o3)=O)C2)C2CCN1CC2 c1(C(N2C(C)(CNC(C(CC#C)C)=O)CCC2)=O)cc(OC)ccc1[N+](=O)[O-] C(C)(C)(CCC(=O)NC1CC2(C1)CN(C(C1CN(C(C)=O)C1)=O)C2)OC c1(C(=O)NC2CCCCN(C(CC(C=C)CC)=O)C2)ccsc1S(N)(=O)=O c1(C(=O)OC)cncc(C(N2CC(F)(CNC(=O)C(C)Cc3ccco3)C2)=O)c1 C(=O)(CC(C)C(C)C)NCC1(O)CCN(C(c2n(CCOC)ncc2)=O)C1 N1(C(c2cccc(C(C)C)c2)=O)CCN(Cc2cc(F)c(I)c(F)c2)CC1C#N C1(C(=O)NC(CC=C)CNC(=O)CN(C)C)CCN(C)C1c1cccs1 C1(NC(c2cc(C)nc(C)c2)=O)C(C)CN(C(c2cnc[nH]2)=O)CC1C c1(C(=O)NC2CCCN(C(C=NOC)=O)C2)ccc2nc(CO)[nH]c2c1 C(=O)(CCCC(F)(F)Br)N1CCC(n2cc(C(N3CCCCC3=O)C)nn2)C1 c1(C(=O)NC(CC)(C)CCNC(=O)C(CN(C)C)C(C)C)cn2ccnc2cn1 CC#CCCCC(=O)N(CCCCCC)CCNC(C1CCC=CCCC1)=O C1(CNC(c2onc(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)C1(C)C C1(OC)(CNC(=O)CC2CC(N(C)C)C2)CCN(C(C2(C(N)=O)CCC2)=O)C1 C1(C(=O)OC)CC(=O)N(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)C1 C(=O)(C(C)(CC)C(N)=O)N1CCN(C(c2nc(COCC)sc2)=O)C(CF)C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)CCc2ccn(C)n2)CCC1C c1(C(N(CC)CC)=O)ccccc1C(=O)NCC1CCCN1C(c1ccon1)=O C1(CNC(C2(OC)CCSC2)=O)COCCN(C(c2c(Cl)csc2Cl)=O)C1 C12(CNC(=O)CCCCO)CC(CO1)N(C(C1CC1C1CC1C)=O)C2 C1(C)(C(N2C(CC)(CC)CCC2)=O)CC=C(C)CC1 Cc1cc(C(=O)NC2(C(=O)NCCC3OCCC3(C)C)CC2)cc(O)n1 N1(C(c2cccc(CC)c2)=O)CCC2(NC(=O)Cc3ncoc3C)CC2C1 C1(CC(=O)N(CCC(=O)N2CC(O)C2)CC#C)CC(CC)=NO1 C=CC(C(=O)N(CCC(C)NC(c1cn(CCCF)nn1)=O)C)OC C(=O)(C(O)CC(F)(F)F)NCCOC1CCN(C(C(C(C)C)NC(N)=O)=O)CC1 c1(NC(C(C)NN(CCN2CCOCC2)C(C2CCCCC2)=O)=O)cccnc1 C(=O)(C1=CCCCCC1)N1CCC(NC(=O)Cc2n[nH]cc2Br)C(O)C1 C(=O)(C(O)C(C)(C)C)N(C(C)CNC(C1CC(=O)N(C2CCCC2)C1)=O)C C=CCC(C)(C)CC(c1nnnn1C)NCC1CC1c1c(F)cccc1Cl c1(SC2C3CN(C3)C(=O)N2)nc2c(s1)CC(C)(C)CC2.C(=O)(CC)OC N(C1c2ccccc2CC1NC(=O)CCCC1CC1)C(C(C(C)O)N(C)C)=O Cc1cc(C(=O)NCC2C3CC2N(C(=O)Cc2cnn(C(C)C)c2)C3)nc(C)c1 C1(C(=O)NC(CCC)C2CCCC2)CN(C(c2sc(C)nc2C)=O)CCO1 C(C(CC(C)C)C(=O)NC1CCCC1N=[N+]=[N-])NC(CCSC)=O Cc1nc(C(F)(F)F)oc1C(N1CCOC(CNC(c2cc(Cl)c[nH]2)=O)C1)=O N(C1c2ccccc2CC1NC(C1CCCC12CC2)=O)C(C(CCC)N(C)C)=O c1(NCC(CCC)OC)nc(C)cn2nc(C(F)(F)F)cc12 c1(SCC)cc(C(=O)NCC2CC2CNC(C2CCCC3(CC3)C2)=O)ccc1C N1(N2C(CC)CCCC2)CCN(C(=O)Cn2cnc(C=O)c2)CC(C)(F)C1.C(C)=O Cc1oc(SC(F)(F)F)cc1C(=O)NC1CN(C23CC(C(=O)OC)(C2)C3)CC1C c1(C(=O)NCC2CC2CNC(c2cscc2C2CC2)=O)cc(C(F)F)cc(F)c1 c1(C(N2CCSCC2)=O)ccc(C(N2CCCC2c2ccc(F)cc2)=O)nc1 CC1CC(C(F)(F)F)(NCc2ccccn2)CC(C)O1 C1(C)(C(=O)NCC(C)C)CC12CCN(C(C)CC1CCCCCN1)CC2 c1(CCC(=O)NCCN(C2CCCCC2)C(C2C(C#N)C2)=O)ccccc1F Cc1cccc(C(=O)NCC(=O)N(C)CC2CCN(C(=O)C(C)C3CC3)C2)c1 N1(C(c2c(CC)n(C)nc2)=O)CCC2CN(C(=O)C(O)CCSC)CC2C1 Cc1ccc(C(N2CCCCC2C(C)NC(=O)Cc2ccccc2C)=O)cc1C C(=O)(C1=CC2CCCC12)NCCC1CCCN(C(C2(CC)COC2)=O)C1 N1(C(CCSCC)=O)CCN(C(=O)CN(c2ccccc2)C)C(CCOC)C1 C1(NC(CC(C)(C)Cn2cc(CC3(O)CC(C(=O)O)C3)nn2)=O)CCC(C)CC1 C1(NC(C(C)(C)C)=O)CC2(CCCN(C(c3ccnc(OCC4CC4)c3)=O)C2)C1 c1(CCC)cc(C(N2CCOC(CNC(C3CC(OC)C3)=O)C2)=O)nn1C c1(CC)cc(F)c(C(=O)NCCOCCCNC(=O)CC(CC)SC)cc1F CC1(C)CN(C(=O)C(O)C(F)F)CCC1NC(c1ncn(-c2ccccc2)n1)=O CCC(F)(F)C(C)(C)C(=O)NCC(C)CNC(c1cnn2cc(C)cnc12)=O N1(C(CCCC=C)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)C2C1 c1(C(=O)NC(CCOC)CNC(C2C(Cl)(Cl)C23CC3)=O)c(F)ccc(C)c1Cl N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2CCCCS2(=O)=O)=O)C(C)C1 N1(C(CCOCC#C)=O)CCC2(CCCN2C(c2ccnn2CCCC)=O)C1 C=CCCN=C(NCc1coc(C)c1)NCC1CCC(C)O1 CN1C2CCCC1C(NCC(=O)NC1(C)CCOCC1)C2 c1(C(N2CC(NC(C(CC)SC)=O)C(C)C2)=O)csc(=NC2CC2)[nH]1 N1(C(c2sccc2CO)=O)CC2CCC(C1)N2C(c1c(O)cccc1F)=O C1(C2CCN(c3nnc(C(N)=O)s3)CC2)(NC(C2CCN(OC)CC2)=O)CC1 C1(NC(c2cc(C)c(C)nn2)=O)CCC2CC1CN2C(C1(C2CCC2)CC1)=O CCC(C)(CO)NC(=O)CC1C(NC(c2cocn2)=O)CC1O N#Cc1cc(C(=O)NC2(CO)CCCN(C(C3CC=CCC3)=O)C2)cc(F)c1F c1(OCC(=O)NCC(CNC(c2nn[nH]c2Cl)=O)CO)ccccc1O N1(c2c(F)cnc(C)n2)CCC2(CCCCC2NC(c2cnc(C3CC3)s2)=O)C1 N1(C(C2C(C)(C)C2(F)F)=O)CC(NC(=O)CCn2cc(Br)cn2)CC1(C)C c1(CC)nnc2n1CCN(N(C)Cc1nnc3ccccn13)C2 C#Cc1c[nH]nc1C(=O)NCC1CCCC1NC(=O)Cc1csc(C(=O)OC)c1 CC(C(C)(C)C)=CC(=O)N(C(C)CCNC(C1CC(CN(C)C)C1)=O)C C(CC(=O)N1CC(CO)(OC)C1)(C1CC1)NC(CC1CC(=C)C1)=O CC(C)C(C(=O)NCc1csc(=N)[nH]1)NC(=O)CC1(c2ccccc2)CC1 N1(C(c2ccc(CC)o2)=O)CC(NC(=O)CC2CCCN2C(C)=O)CCC1C Cc1cc(NC(=O)C(F)C(C)CNC(=O)Cc2cc[nH]n2)cnc1O C1(CCNC(c2cccc(OC)n2)=O)CC(F)(F)CN1C(C1C=CC=CC=C1)=O CC(C)CC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCCCC1O)=O N1(C(C(C)OCCOC)=O)CCC(F)(C(=O)NCCCCCCN(C)C)CC1 N1(C(C23C(C)OC(CC2)C3)=O)CC(O)(C2(CNC(C3CCSCC3)=O)CC2)C1 C(CC(O)CC(=O)N1CCOC(CCNC(=O)C=Cc2cc[nH]n2)C1)SC C(c1ccc2c(c1)OCO2)=CC(=O)NCC1CC(NC(=O)C2=CCCO2)C1 c1(OC)ccc(C(N2CCCC(N(C)C(C3CC3CF)=O)CC2)=O)cc1Cl C(=O)(C(C)(C)CC(F)F)NCC(CC(=O)NCc1c(CC)nn(C)c1)C1CCC1 C1(C(N(C(CN(C(c2ncn(C(C)C)n2)=O)C)C)C)=O)CCC2(CCC2)C1 C1(CNC(CCOC)=O)CCCN1C(=O)CN(c1ccccc1)C Cc1nc2c(o1)CCCC2CC(=O)N1CC(Nc2ncnn3c(Br)ccc23)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CC2(C1)CN(C(C1COC(=O)C1)=O)C2 c1(C(=O)OC)ccccc1-n1cc(CN(O)C(C2CCCC(=O)N2)=O)nn1 C(C(=O)N(C)CCNC(C1CCCN1C(=O)C(C)(C)C)=O)(C(C)C)NC(=O)OC C(=O)(C(F)C(C)(C)O)NCCC1(NC(C2CC(C(=O)OC(C)(C)C)C2)=O)CC1 N1(C(CCSCCC)=O)CC=C(CCNC(C2(CCF)CC2)=O)CC1 C1(C(=O)NCC(C)(COC)CC)(CC)CCCN(C(C2CCC2)=O)C1 C(=O)(C#CC1CCCO1)N1CC(CNC(c2ccc(CSC)cc2)=O)C(C)C1 N1(c2ccc(C#N)cn2)CC(NC(C2(C3CCC3)CCC2)=O)C2CCCCC12 N1(CC(=O)N(c2ccc(OC)c(C(F)(F)F)c2)C)C(=O)c2ccc(Br)cc2C1=O C(=O)(N=c1cc2ccccn2[nH]1)C1CN(C(CC(C)OC)=O)CC(C)(C)C1 c1(C(N)=O)cc(C(=O)NC2CCN(C(C3CN(C4COC4)C3)=O)C2)n[nH]1 C(C(C)(C(N)=O)NC(=O)CC1CCN(C(=O)Cc2ccccc2Br)C1)OC c1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(O)C2)cccc2nccn12 C(=O)(C(C)CC(F)F)N1CC(C)C(NC(=O)COC(C)(C)C)C1 C(=O)(C1CCc2c[nH]nc21)NC(CCC(N1CCN(C(=O)NC)CC1)=O)C c1(OC)oc(C)nc1C(=O)NC(C)CCNC(=O)CCc1ccncn1 N1(C(c2scc(C)c2)=O)CCCC(NC(=O)CC2CCCO2)C1C c1(NC2(C)CC(NC(c3cc(CC)oc3C)=O)C2)ccc(C#N)nc1 C#CCC(C(=O)NC)NC(c1cnc(CNC(C2(C#N)CC=CC2)=O)nc1)=O c1(CCC)cc(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)ccn1 c1(OC)ccc(C)c(NC(c2c(CNC(=O)C(C(C)C)OC)nnn2C)=O)c1 c1(CCCCC)nc(-c2sc(Br)nc2C)n(C(C)CCC)n1 C1(C(C)C)CN(C(c2ccncc2F)=O)CCC1NC(c1cnn(CCF)c1)=O N=c1nc(O)c(CC(N2CCCC(CCNC(=O)CC3=CCCC3)CC2)=O)c[nH]1 N1(C(C(C)(O)c2ccccc2)=O)CC2CC2(NC(=O)Cc2cccs2)C1 N1(C(CC(C)n2cccn2)=O)CC2(CCNC(C3CCCN3C)=O)CCC1CC2 C(=O)(CCCCC(=O)NCC1(C)CCC(NC(=O)CCCC(F)(F)F)C1)OC N1(C(C2CC(CC)C2)=O)CCCCCC(NC(=O)Cn2nc(C)oc2=O)C1 C(=O)(C#CC1CCOCC1)N1CCCC(NC(C(C(C)O)C)=O)CC1 C(=O)(CC(C(F)F)NC(=O)CCCF)NCc1cc(CC)[nH]n1 C(=O)(CC(F)(F)C(C)C)NC1CCCN(C(c2c(C)nc(=N)[nH]c2)=O)C1 c1(OC)ccc2nc(N3CC(CN(C)C(c4coc(Cl)n4)=O)C3)c(C#N)cc2c1 c1(OC)cccc(C(=O)NC2COCC2NC(=O)CNc2ccc(C)cc2)c1F CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(C3CC3)no2)=O)C(C(F)(F)F)C1 c1(OC)cccc(C(C(=O)NCC(=C2CN(C(=O)C(C)CF)C2)F)OC)c1 Cc1cc(C(=O)NCC23CC(CN2C(=O)COC(F)(F)F)C3)nnc1C Cc1nn(C)c2sc(C(N3CCCC4CN(C(C5CC5(F)F)=O)CC34)=O)cc12 C1(CNC(=O)NCc2cccc(OC(CC)C)c2)OCCC12CCC2 c1(OCCC(N2CCC(N(C(CCC#C)=O)C)CC2)=O)cc(F)ccc1F Cc1c(Cl)ccc2[nH]c(C(=O)NC3CC34CCN(C(=O)C(N)=O)CC4)cc12 c1(C(N2C3C(C(N4CC(C)OCC4C)=O)C(C3)C2)=O)c[nH]c2cccc(Cl)c12 Cc1cc(O)ncc1C(c1nnnn1Cc1ccccc1)NC1(C)CC1(C)C CC1(C)CC(C#N)(CNC(=O)C(O)C2CN(C(c3nnsc3N)=O)C2)C1 C1(CC)(NC(c2cn(C3CCC3)nn2)=O)CCN(C(=O)COCC(C)C)CC1 N1(C(CC2CCN(C)C2=O)=O)CC(NC(c2cnccc2C(F)F)=O)C2(CC2)C1 C(C)(CN=[N+]=[N-])NC(C1C(NC(C(C)OC)=O)CC1)=O C1(CNC(c2nc(OCC)sn2)=O)CN(C(=O)CCC(C)CN(C)C)CC12CC2 C(C(CCCC)NC(C1(OCC)CCSCC1)=O)NC(c1cn(CC=C)nn1)=O C(CCN=C(NCCOCCS)NCC1CCCCO1)CS(C)(=O)=O c1(C(=O)NCCOC2CN(C(CC#N)=O)C2)c(O)nnc2c1COCC2 c1(C(N2C(CNC(C(c3ccccc3)C)=O)CC2)=O)cnn(C(C)(C)C)c1 C(CN=C(NCC1(C2CC2)CC1)NC1CCS(=O)(=O)C1)N(C1CCCCC1)C CCC(C(=O)NCC(O)CNC(c1ocnc1C)=O)OC1CCCCC1 C12(C(=O)NC(CCOC)CNC(=O)C(O)CSC)C3CCC(CC13)C2(F)F Cc1cc(N)c(C(=O)NCCC2CCC(NC(=O)C3=C(Cl)CC3)C2)cc1C C#CCC(C(=O)N1CCC(C(=O)NCCCc2ccsc2)(CC)C1)C1CC1 Cn1cc2ccc(NC(C3CC(O)CCN3Cc3ccnc(O)c3)=O)cc2n1 N1(C(C(=O)NCCC)C(C2CCCC2)OC)CCC(S(=O)(=O)C(C)C)CC1 C(=O)(CC(C)(C)C(=O)NCC1CCN(C(=O)CNC(N)=O)CC1C)OCC C(=O)(CS(=O)CC)N(CCC(=O)NC(c1ncnn1C)C)CC=C N1(C(Cc2c(C)ncs2)=O)CCC2(CO)CN(C(=O)CCc3cn[nH]c3)CC2C1 c1(NCc2nnc(C(F)F)o2)nccc(=NCc2cnc(C(F)(F)F)s2)[nH]1 c1(OC)ccc(C2CC2)c(C(N2CCN(C(=O)C3CC3)C(CC3CC3)C2)=O)c1 c1(C(=O)NCC(CC=C)NC(c2cc(C(F)F)cc(F)c2)=O)ccc(N)c(F)n1 C(CC(CC)C(=O)NCC(C)N(C)C(c1nnsc1C)=O)=CC c1(C(=O)NCC2C(NC(COCC)=O)C2)cc(-n2cccc2)cc(Cl)c1 c1(N(CC(N2CC=CC2)C)CC)ccc(C(=O)OC(=O)CSCC(C)(C)C)cc1 Cc1nnc(CC(=O)NCCC2CCC(NC(=O)Cc3nncn3C)C2)o1 c1(C(N2CCC(OC(C)C)C2)C(=O)NCCCSCC)csc(C#N)c1 C1(OC)CCCCN(CC(=O)NCC(C)(Cc2ccccc2)C(C)O)C1=O C1(NC(C2C3CCC(F)(F)C23)=O)CN(C(C2SCCS2)=O)CC12CC2 c1(OC)cccc2cc(C(N3CCCC3CCCNC(C3CC3(F)F)=O)=O)[nH]c12 C1(CNC(CC(C)C2CC2)=O)CN(C(=O)CNS(N)(=O)=O)CCCO1 CC1CCCN(C(C2CCCN(C(C(=O)O)c3ccsc3)C2)=O)C1 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC1CN2C(=O)C(O)Cc1cnc[nH]1 Cc1ccc(C)c(C(=O)NC2(CNC(=O)CC(C)c3ccco3)CCCCC2)n1 C12(NC(C(CC)C)=O)COC(C1)C(NC(c1ccc(F)cc1OC(F)F)=O)C2 N1(C(C2C(NC(=O)C(C3CCCCC3)O)CC2)=O)CCC(CC2CC2)CC1 c1(C(=O)NC2CC(C)(CNC(c3c(CC)nn[nH]3)=O)C2)cccc(N)c1C CCC(C)CCCCC(=O)N1CCC(Nc2ccc(C(=O)OC)c(C)n2)C1C c1(C(=O)NCC#CCNC(c2ncccc2C(F)(F)F)=O)cnc2n1CCC2 N1(C(C2=NOC(CNC(C(SC)SC)=O)C2)=O)CC(CO)C2(CCC2)C1 C(=O)(C(C)S(N)(=O)=O)NCC(CC(=O)NC1CC(CC(=O)OC)C1)C c1(C(=O)NC2CC(NC(C=CCC)=O)C2)cccnc1-c1nncn1C c1(OC)cc(=NC(=O)C=CCC(C)(C)NC(=O)C(C)Cn2cccn2)[nH]n1C c1(C(=O)NC2CC(CC(=O)NCC3C(OCC)C3)C2)cnc(-c2cccnc2)s1 C(C(CC)(CC)C(N)=O)NC(C1CC(CC)N(C(c2cc(OC)n[nH]2)=O)CC1)=O CCC(C(=O)N(C(C)(C(=O)NCCC1CCC(=O)N1)C1CC1)C)C(C)(C)CC C1(NC(C(CSC)O)=O)CC2(CCN(C(c3cccc(SC)c3)=O)CC2)C1 C1(C(=O)NCc2cnc(C(C)OC)s2)COCCN1CC(F)(F)F C1(NC(c2ccc(C)cc2)=O)CCCC12CCN(C(c1sc(=N)[nH]c1C)=O)CC2 C1(C(N2CC(NC(c3ccc(CO)nc3)=O)C2)=O)C2CCCCC12 c1(OC)cc(N)cc(C(=O)NCC(C)(C)CNC(C2CC2CC(C)C)=O)c1OC c1(C(=O)OC)ccc(C(=O)NC(C)CCNC(=O)C#CC2CCC2)c(OC)c1 c1(C(=O)NCC(CCCC)NC(=O)CC2(OCC)CC2)cc(N)ccc1CC Cc1csc(=NCC(=O)NCC2(C)CCCN2C(=O)CNC(=O)CCCCO)[nH]1 C1(NC(c2ccc(OC(C)=O)cc2)=O)CCCCN(Cc2cccc(Br)n2)C1 CS(=O)(=O)C1CCC(C(N2CCC(NC(=O)CC(F)(F)C(F)F)C(O)C2)=O)CC1 C1(CNC(c2c(COC)ccs2)=O)CCCN(C(C2(c3ccno3)CC2)=O)C1 c1(C(N2CCC(=CCNC(c3nncc(OC)c3)=O)CC2)=O)nnc(O)nc1O C1(N(C)C(c2ccn(C3CC3)n2)=O)CCCC(N(C(=O)CC2CC2)C)C1 c1(C(N2CCC3C(NC(c4cc(CC)c(C)s4)=O)C32)=O)cc(N)cnc1Cl c1(C(N2CCC(OCCNC(C(C)OC)=O)C2)=O)ccc(CO)nc1 c1(OC)ccc(CC(c2ccc(OC(F)F)cc2)NCc2nnnn2C)cc1 Cn1cc(C(=O)CN(C(=O)Cn2nnc(C(C)(C)C)n2)CCO)nn1 c1(C(=O)NC2C(C(N3CCN(C=O)CC3)=O)C2)cc2ccccc2oc1=O c1(C(C(=O)NCC2N(C(c3n(CC)ccc3)=O)CC2)O)ccccc1F c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(c3[nH]ccc3C)=O)C2)c1F Cc1cc(C(=O)NCc2ccc(C(=O)N(C)CC3CCCC3O)cc2)c(C)s1 c1(C(=O)NCC23CC(NC(C4CCC5CCC4O5)=O)(C2)C3)cccc2c1OCO2 C1(CNC(CCCCC#C)=O)CN(C(=O)CCCCOCC)CC(C)(C)O1 N1(C(c2ccc(CCC)c(N)c2)=O)CCCC2(NC(=O)CC3CCCC3)CC2C1 N1(C(C(C)CC2CCOCC2)C(=O)NC2(C)CC2)CCC(S(=O)(=O)C(C)C)CC1 c1(OC)cnc(F)c(C(=O)NC2CC(F)CN(C(c3ccc(CSC)o3)=O)C2)c1 CN1CCN(C(=O)Cn2nc(O)ccc2=O)C(CNC(=O)Cc2cccn2C)C1 N1(C(=O)Nc2ccc(NC(C)=O)cc2O)CCC(C2CC2)C1c1nnc(O)n1C N1(C(C2(C)SCCCS2)=O)CC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 C1(NC(CCCOCCC)=O)CN(C(=O)Cn2cnc(C#N)n2)CCC1C CCCCC(CC)C(=O)NC1CCC(C)(CNC(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(=O)NCC(CC)NC(c2c(Cl)nn(C)c2Cl)=O)CCCNS1(=O)=O c1(OC)ccc2c(C(=O)NCC3CCN3C(=O)C3=CCSC3)ccnc2c1 Nc1ccc(Cl)cc1C(=O)NCC12CC(NC(c3c[nH]nc3C3CC3)=O)(C1)C2 C1(NC(CCC(CC)OC)=O)CCN(C(c2ccc3sccc3c2)=O)CC1(C)C N1(C(C2(Cc3ccc(O)cc3)CC2)=O)CC2CC2(C(=O)OC)C1 c1(C(=O)NC(C2(CNC(c3ccc(CC)o3)=O)CC2)C)cc2c(Cl)cccn2n1 c1(C(c2n(CCC)nnn2)NC2CCCS(=O)(=O)C2)cc2cccnc2o1 c1(SC)ccc2sc(CN(C)CCCCCN)nc2c1 C1(CC(=O)N(CCN(c2c(C(=O)OCC)cccn2)C)CC)CCCCCCC1 Cc1cc(C#N)cnc1C(=O)NC1(C(=O)Nc2cn(C)nc2C)CCC(C)(C)C1 CC#CCC1C(=O)N1CC1CC1.c1(OCCCNC(=O)OC(C)(C)C)cccnc1 c1(C(=O)Nc2nc(C)cc(C)n2)ncn2cc(-c3cncn3C)sc12 C1(F)(C(N2CC(NCc3cn(C)nc3)OCC2)=O)CCCCC1(F)F CC1(CNC(=O)Nc2ccnc(OC(F)F)c2)CCCCCC1 Cc1c(C(=O)NC(C)CNC(=O)COCc2cccnc2)cccc1O c1(C(N2CC(COC)(NC(=O)C(F)CC3CCC3)C2)=O)nc(C(C)C)ncc1Cl c1(C(=O)NC2CC2NC(c2cnn[nH]2)=O)ccc2nc(O)cc(O)c2c1 C1(OC)CC(CNC(=O)CN(C2CCCC2)C)N(C(C2C=C(C)CS2)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CCC(C)(CNC(c2cnn(C(F)F)c2)=O)C1 C1(F)(C(N2CC(F)(CNC(c3cc(SC)ncc3)=O)C2)=O)C(C)(C)C1(C)C c1(N(CCCC(F)(F)F)CC(F)(F)C2CC2)cc(Cl)ccc1Cl C1(C(=O)NC(CC=C)(C)C)CCC(C)(C)N(C(=O)CC2C=CCC2)C1 N1(C(C)=O)CCC(CC(=O)N(CC(C)CNC(=O)CCC2CCC2)C)CC1 c1(CN2C(C(=O)NC(C(C)(C)C)CO)CNCC2)ccc2cncn2c1 c1(C(N(C)CCOCCCNC(=O)CC2(C(F)F)CC2)=O)cn(C(C)(C)C)nn1 C1(C(=O)NCCN(CCCC)CCCC)CCCN(C(=O)COCC(F)F)C1 C12(NC(C3N(CC)CCC3)=O)CCN(C1)C2=O.c1(NC)cnc(Cl)nc1 c1(C(N2CCC(=CCNC(C3C(C)(C)CO3)=O)CC2)=O)cc(O)nc(C2CC2)n1 c1(OCC(=O)NC(C2CCCC2O)CNC(CC)=O)ccsc1Cl C1(NC(c2c(SC)scc2)=O)CC2CCC1N2C(=O)C(C)OC1CCCC1 C1(C(=O)NC(C=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1c[nH]c(C)c1)=O N1(C(CCOCCOC)=O)CCC2(CC2)CC1C(N1CC(C)N(C)C(C)C1)=O CC(CC(=O)N1CCCC1(C)CNC(c1ccc(O)nc1Cl)=O)C(F)F C1(CC)CCC(C)N(C(C2CC(O)(CNC(=O)CNC(C)=O)C2)=O)C1 C1(C)(SC)CCC(=O)NC1.c12nc(no1)C2NC n1(CCNC(C2C=CC(NCc3ccc(O)cc3Br)C2)=O)nnc2ccccc12 Cc1ccc(C(C)C(=O)N2CC(CC(C)NC(c3ccsc3C(F)F)=O)C2)cc1 C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)(NC(CNS(CC)(=O)=O)=O)C1 CCC(CC)(CCNC(C1CCCC(=O)N1)=O)NC(C1OCCCC1(C)C)=O C(C)(N=c1[nH]c(N2CCC(C3CCC3)C2)nc2cc[nH]c12)c1c(C)nc(C)[nH]1 C1(C(=O)NC(C(=O)NCC(=O)NCCC)CC)OCCC1NC Cc1oc(C(=O)NC2CC(CCNC(=O)CCC3CCCO3)C2)cc1CO Cc1cncnc1N1CCCC(CCNC(C2(C(C)C)CC2)=O)C1 CN1CC(C(=O)N(C)CCN(C)C(c2ccc[n+]([O-])c2)=O)C(C(F)(F)F)C1 N1(C(C2(C(=O)NC)CC2)=O)CC(NC(=O)CCC2CCC(=O)N2)C(O)C1 CC#CCCCC(=O)NCCOCCN(C(=O)C(c1ccc(F)cc1)C1CC1)C c1(N2CCC(=CNC(c3cnn[nH]3)=O)CC2)ccncc1[N+](=O)[O-] c1(C(=O)NC2CC(C)N(C(=O)C=CI)CC2)cc2n(n1)CCCO2 CC(C)(C)C(O)C(=O)N1CC2(CC(NC(=O)CN3CCCCCC3)C2)C1 CC1CCC(=CC(=O)NC(C)(CNC(C2(c3ccccn3)CC2)=O)C(C)C)CC1 N1(C(c2cc(Cl)c(Cl)c(Cl)c2)=O)CCC2C1CCCN2C(C12CC(C1)C2)=O Cc1cc(O)ncc1C(=O)NCCN(C(=O)CC1COC2CC1C2)CC1CC1 n1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2F)cnc([N+](=O)[O-])n1 C1(CNC(CN(C)C)Cc2ccccc2)COC2(CCOCC2)O1 CC1(C)CC2(CC(C(=O)NC3CC(CNC(c4cccn4C4CC4)=O)C3)C2)C1 N1(C(Cc2ccc(C)o2)=O)CCCCC1CC(=O)NC(CN(C)C)CCO Cc1cccc(C)c1C(O)C(N1CCC(C2CCCN2C(=O)CC2CC2)CC1)=O C1(NC(c2c(C)cncc2C)=O)CN(C(=O)Cn2ccccc2=O)C2(CCC2)C1 c1(C(=O)NC(CCNC(C(CCC)C(C)C)=O)(C)C)ccc2c(c1)CCC2(C)C N1(C(C=CC(=O)OC(C)(C)C)=O)CC2CC2(NC(=O)CC(O)c2ccccc2)C1 c1(NCc2c(C)ccs2)[nH]c(=NC2COCC2C2CC2)nc2c1ncn2C(C)C C1(CNC(C=NOC)=O)CC2(CCOCC2)CN1C(=O)C(C)OC1CCCC1 N1(C(c2cnc(CC)s2)=O)CC(CNC(c2cnc(=N)[nH]c2)=O)C(C)C1 N1(C(C2CCCN(c3cc(C)nn3C)C2)=O)CC2(CC(S(C)(=O)=O)C2)C1 C1(NC(COCCOCC)=O)CCCC12CCN(C(c1nnn(C)c1N)=O)CC2 Cc1ccc(CNC(=O)NC(C)C(C)NC(c2ccnn2CC(F)(F)F)=O)cc1 C(=O)(NNCC(F)F)NCC1(COC)CCCO1 C1(NC(C2(CCOC)CC2)=O)CCC2CC1CN2C(=O)C=Cc1nc(C)cs1 C1(NC(C(C(C)C)C)=O)CC(F)CN(C(c2ccc(CC(N)=O)cc2)=O)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NCc1cn(C)nc1 c1(NC2CN(C(=O)CC3CCS(=O)(=O)C3)C2)ncnc2c1CCC2 S(=O)(=O)(c1ccc(Br)cc1NCc1nc2ccccc2n1C)NC(CC)CO N1(C(c2ccc(C)c(F)c2F)=O)CCC2CCC(C1)N2C(=O)C(C)CC(C)(F)F c1(C(=O)NCC=C2CCN(C(CC(C=C)(C)O)=O)CC2)cn2nccc2nc1C c1(NC2(CNC(C(CSC)C)=O)CC2)ncnc2c1cnn2C C=CC1(CC(=O)NC2(CC3CCC3)CC2)CN(C(=O)CC2CC2)C1 N1(C(C=NOC)=O)CCCCC1C1CCN(C(=O)C(C)Cc2c(C)noc2C)C1 N1(C(C(C)NC(N)=O)=O)CCOCC1CNC(c1ccc(C(F)(F)F)s1)=O Cc1[nH][nH]c(=NC(=O)C23CC2CN(Cc2ccc(CBr)cc2)C3)c1C C1(OC)(OC)CC2(CN(C(=O)N(CCS(N)(=O)=O)C3CC3)C2C(C)C)C1 c1(C(N2CCCC(N(C(=O)Cc3occc3C)CC)C2)=O)cc(C)cc(F)c1N N1(CC(=O)N(CCCN(C(=O)Cc2cccc(Br)n2)C)C)CCC(C)(O)C1 c1(CC(=O)NCC(CNC(C(COCC)C)=O)C)ccc(O)c([N+](=O)[O-])c1 CC1(C(=O)NC2CCC(NC(=O)CCSC(F)(F)F)CC2)CCC12CCC2 C1(C(N2CCC(C(=O)NC(CC#CC)CO)(OC)C2)=O)CC2CC(=O)C1C2 Cc1nc(C(=O)NC(CNC(=O)C(C)Oc2ccccn2)C2CCC2)cs1 C(C(=O)N1CCCC(F)(CCSc2cncc(C)n2)C1)(c1ccccc1)=C(C)C N1(C(C=CC=CCC)=O)CC(O)(C2CCCN2C(=O)CCc2ccsc2)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCN(C(=O)CC(C)(C)SC)CC1c1cn[nH]c1 CC(F)CCN=c1nc2c(ncn2C)c(NCc2nc(C(C)(C)C)ns2)[nH]1 Cc1c(NC(=O)CC2(C)CN(C(=O)COC3(C)CCC3)C2)ccc(Br)c1Cl N1(C(CC(C=C)CC)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 c1(C(=O)OC)cc(CC(=O)N(CCCNC(=O)C(C)n2ccnc2)C2CC2)[nH]n1 Cc1c(CC(=O)N(CC(C)CNC(c2ncncc2Cl)=O)C)cccc1[N+](=O)[O-] Cn1cnc2cccc(C(N3CC(NC(c4cccnc4S)=O)C4CC34)=O)c12 C12(C(N(CC(C)(C)NC(c3cn(CC)nc3C)=O)C)=O)CCC(F)(CC1)C2 N1(C(C(C)O)=O)CCCC2(CCN(C(c3cnc(F)c(F)c3)=O)C2)C1 C1(C(=O)O)CN(C(=O)CCBr)CC12CN(C(C1CCCO1)=O)C2 CC(C)C(F)(CNC(C1C2CCCCC12)=O)C(=O)NC1(C2CCCC2)CC1 C(CC(F)F)(C(=O)NCc1nn[nH]c1C1CC1)NC(CCC(C)OCC)=O N1(C(C2CC(NC(C)=O)C2)=O)CCC(NC(=O)CC2CC2(Cl)Cl)CC1 Cn1cc(CN=C(NCC(F)F)NC2CCC2)c(C(F)F)n1 C1(NC(C(C=C)OC)=O)CCCCC12CCN(C(c1[nH]ccc(=O)c1C)=O)CC2 N1(C(c2cccc(N(C)C)c2)=O)CCCC(F)(CNC(C2CCCN2C=O)=O)C1 C12(CNC(=O)Cc3ccoc3)CCCC1N(c1ccn3c(Br)cnc3n1)CCC2 C#Cc1ccc(C(=O)Nc2c(C)cnn2CC2CCC(C)CC2)cc1C c1(N(C2CCCC2)CCCC)ccc(C)c(OC(c2cccc(SC)c2)=O)c1 c1(CNC(=O)NC2(C3CCCC3)CC2)cncc2n[nH]cc12 c1(CN(CC)Cc2ccnn2CC2CCCO2)ocnc1C1CCC1 c1(CC)cc(C(C(=O)NCC(C)C)N(C2CCC(=O)NC2)CC)n(C)n1 C=CCCC(C(=O)O)Nc1ccc(C(=O)OCC)c(C(=O)OC)c1 C1(NC(C=Cc2nnn(C)n2)=O)CCCCN(C(=O)C(c2ccccc2)F)C1 c1(C(N2CC(C)C(CNC(=O)C(C)(C)C(F)(F)F)CC2)=O)c(O)cc(F)cc1F Cc1ncnc(C)c1C(=O)NCCC(C)NC(C1(CC(C)C)CCCC1)=O C1(NC(c2c(CC)cno2)=O)CC2CC1N(C(=O)CC1CN3CCC1CC3)C2 c1(N2CC3N(C(c4ccccc4F)=O)C(C3)C2)ncc2cn[nH]c2n1 N1(CC(=O)NCCN(C(CC2C(C)=NNC2=O)=O)C(C)C)CCc2sccc2C1 c1(N(C)C(=O)NC(CC)=O)ccc(S(=O)(=O)N2CCCC(C)(COC)C2)cc1F CC1(C)CC(=O)NCC1C(N1CC(O)(CCNC(=O)CC2(O)CCCCC2)C1)=O c1(CN2CCC(C#N)(NC(CCN(C)C)=O)C2)ccc2cc(O)ccc2c1 c1(CCC(=O)NC(C(C)NC(c2c(C)ccnn2)=O)CO)cc2ccccc2o1 c1(C(=O)NCC2N(C(C(=O)Nc3c(OC)cccc3)=O)CC2)sc(C)c(C)c1C N1(C(C2C(CC)CCN2C(=O)C=CCN2CCC2)=O)CCc2nc[nH]c2C1 CC1CN(C(=O)Cc2cc(F)cc(F)c2)CCCN1C(C1OCCN(C)C1=O)=O N1(C(c2ccc(C)cc2C)C(=O)NC(C(=O)OC)C)C2CCCC1CC(F)(F)C2 C=CCC(CC(F)F)C(=O)NCC1CCC(C)(C)CN1C(=O)CC1CCCN1C C1(C(N2CC=CC(NC(C=Cc3ncn(C)c3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(CC)CCC)N1CCC(N(C(CC(=C)Br)=O)CCO)CC1 c1(C(=O)NCC(c2ccccc2)CNC(C=C=C(C)C)=O)cn2cccnc2n1 c1(NC(C(C)NC(C2(C(=O)O)CCCSC2)=O)=O)ccc(CC#N)cc1 C#CCCCCC(C(=O)NC(C)CC)N1CCNC(=O)C1C CCCCCCC(O)CCC(=O)NCC1(C)CCCN1C(=O)CCCCCF N1(C(c2nc(C)sc2C)=O)CCOCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1 n1(NC(C2C3CN(c4nc(CC)nc(Cl)c4F)CC32)=O)c(C)nc2ccccc12 N#CCCCCC(=O)NCC1CCN1C(=O)C(c1ccc(Cl)c(Cl)c1)O C1(CNC(CSCC(=O)OC(C)(C)C)=O)CN(C(c2ccsc2)=O)CC1C(F)F c1(OC)ncc(C)cc1CNC(=O)NC(C(F)(F)F)C1CCOCC1 C1(C(=O)NCC(C(C)C)=O)CCCN(C(c2cccc(CN)c2)=O)C1 N1(C(C=COCC)=O)CCCC2CCN(C(=O)CCc3ccc(Cl)s3)CC12 N1(C(C2CC(CCC)C2)=O)CCC1(C)CC(=O)N(C1CCOC1)CCF C1(CC(=O)NCCSCC(=O)NCCN(C)C)CCC2CC12 c1(SC)cc(C(N2CCC(C(F)C(=O)NCCc3csnn3)C2)=O)co1 O=C(C(O)C(F)(F)F)NCC1CC2CCC1N2C(c1ccnc(CO)c1)=O N1(C(COC(C)C)=O)CCC(CNC(c2cnc(C(N)=O)s2)=O)CC1C c1(C(=O)OC)cc2ccc(-c3cccc(N4CC(F)(F)CC4C#N)c3)nc2[nH]1 C1(O)(CNC(C(C)CC2CC2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC1 c1(C(N(C2CCN(C(C3(C)CCCOC3)=O)C2)C)=O)cc(OC(F)F)nc(Cl)c1 n1(CC(=O)OC)cc2c(n1)C(NC(N1CCSCC1c1ccc(C)o1)=O)CCC2 C1(NC(CC(CCC)O)=O)CN(C(=O)Cc2ncc(Cl)s2)CC12CCOCC2 N1(CCC(N2CC(O)CC(NC(COC)=O)C2)=O)CCCc2ccccc21 c1(C(=O)NC(c2cc(Br)ccc2Br)C)c(F)cc(Br)cc1Br C12(CNC(CCC#C)=O)CCCCC1CN(C(=O)C(C)(C)C1CCC1)C2 Cc1nc2sccn2c1C(=O)NC1CC(CNC(c2ccc3cncn3c2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(C1CCC1)C1CCC1)NC(C(C)O)=O C1(NC(c2cncc(C)c2C)=O)CC2(CCN(C(c3cnc(S)[nH]3)=O)C2)C1 N1(CC(=O)NC(C=C)C)CCN(C=O)CC1=O.c1(C)cc(Br)c(C)cn1 c1(CC)ccccc1CN1CCCC(N(C(=O)Cc2ccc(C3CC3)o2)CC)C1 N1(C(c2c(NC)scn2)=O)CCC2(CCCN(C(c3c(C)noc3C)=O)C2)C1 CC1=NOC(C)(C(=O)NC2CN(C(=O)C(C)(C)COCC(F)F)CC2CO)C1 CCC(O)C(C)C(=O)NCCC1(NC(=O)CNC(c2ccc(Cl)cc2)=O)CC1 C(=O)(C(F)(F)CCCC1CC1)N(C)CC1(CC(C)C)CC1 N#Cc1cncc(C(=O)NCCC(O)CNC(=O)CC23CCC(CC2)C3)c1 c1(C(=O)NCC2OCC(CNC(C(=O)N(C)C)=O)C2)cccc(N)c1 C(=O)(C(Cc1ccoc1)NC(C1SCCS1)=O)NCC(C1CCCC1)OC c1(NC(NC(C2CN3CCN2CC3)C)=S)nc(Cl)ccc1F c1(SC)cccnc1C(=O)NCC1(CNC(C2CCCC(CC3CC3)C2)=O)CC1 C=C(C)CCC(C)NC(=O)CCCCNC(=O)CC(=O)OC C(=O)(CCC(C)(C)F)NCCC(C)CCNC(=O)CCNC(c1ccccc1)=O Cc1c(Br)noc1C(=O)NC1CCCC1NC(=O)C(N1CCNC1=O)C C12(C(N3CC(CC(=O)Nc4ccc(N(C)C)cc4)OCC3)=O)CCC(CC1F)C2 c1(C(=O)Nc2ccc(OC)nc2)ccc2c(C(=O)Nc3cnc(O)[nH]3)n[nH]c2c1 CCC1=NOC(C(=O)NCC2CCN(C(=O)NCc3ccco3)CC2)C1 C(C1=NOC2CN(C(c3cc(CO)[nH]n3)=O)CC12)NC(C(C)=C1CC1)=O C#CCCCCC(=O)N(C)CC1CC(F)CN1C(C1(CCOC)CCCC1)=O N1(C(C2CCCS2)=O)CCC(N(C(=O)CC2CC=CCC2)CCO)CC1 c1(N(C)CCO)ccc(S(=O)(=O)N(CC2CCOC2)CC)cc1Cl.CCC(C)O c1(C(=O)NC(C(C)NC(C(CC)(C)CC)=O)C)oc2c(Cl)cccc2c1C C1(NC(c2n(CC=C)ccn2)=O)CCN(C(c2ccsc2Cl)=O)C1C C1(O)(CN(C(CN(C(C)=O)C)=O)C)CN(C(=O)C(C)CC2CC2)C1 C1(CC)CN(C(C2OCC3CCCC23)=O)CCN1C(=O)C(O)C(C)C N1(C(C(C(C)C)OC(C)=O)=O)CCC(N2CC(NC(c3ccco3)=O)C2)C(C)CC1 C1(CNC(C(CCC)CC)=O)CCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 CC1CN(C(=O)C(C)(C)C2(O)CCOC2)CCC(C(F)(F)F)O1 c1(CCN(CCCOC)C(C)C)nc(-c2ccc(C)s2)no1 N1(C(COCCCOC)=O)CC(C(C(=O)N(C2(CSC)CCC2)C)OC)C1 CCC(O)C(C)(C)C(=O)NCC1(OC)CN(C(c2cc(Cl)ccc2F)=O)C1 N1(C(=O)OCCC)CCC2(CCC(C(=O)NS(=O)(=O)CC)C2)CC1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CN(C(=O)CN(C)CCO)C)C2C1 c1(C(N(CCCN(C(C2C(C)CC(=O)NC2)=O)C)C)=O)cnc2c(c1)ncn2C Cc1cc(N)c(C)nc1C(N1CCC(O)(C(C)NC(c2ccn(C)n2)=O)C1)=O N1(C(CCC)=O)CCN(C2CCN(c3cccc(Cl)c3)C2=O)CC1C c1(C(N(C2CCN(c3ncnc(C(F)(F)F)c3Br)C2)C)=O)cnc2[nH]ncc2c1 N1(C(COCCCC)=O)CCCC1(C)C(=O)NCC1OCCC1C c1(OC)ncnc(OC)c1C(=O)N(CCCCNC(=O)CN(C)C)C C1(NC(CC(C)SC)=O)COCCN(C(c2ccc(OC(C)(C)C)cn2)=O)C1 CCCCCC(C)CC(=O)NCC(C)CNC(c1cc(-c2ccccn2)no1)=O CN=c1cc(C(=O)NCC2(CNC(C3CCSC3)=O)CC23CCC3)cc[nH]1 Cc1c[nH]c(C(N2CCCC2(C)C(=O)NCCN2CCOCC2)=O)c1C Cc1ncc2n1CC(C(N1CCC(CF)(NC(C3CC3C)=O)C1)=O)CC2 Cc1ncc(C(N2CC=CC2CNC(c2cn(C(C)(C)C)nn2)=O)=O)cn1 c1(N2CC(NC(C3CCOCC3)COC)C2)cnoc1-c1ccoc1 N1(C(CCC#C)=O)CC2CCC1CN2C(C1CCCN1c1ccccc1)=O C(=O)(C1CN(C2CC2)c2ccccc21)NCCCNC(C1CN(S(C)(=O)=O)C1)=O N1(C(CCC(C)OCC)=O)CC=C(C(=O)Nc2ccc(C)c(O)c2)CC1 CC(C(=O)NC1CN(C(c2cc3ccsc3s2)=O)CC12CC2)S(N)(=O)=O CC(CC(=O)NC1CC(C(N2CC3CC4CC3C2C4)=O)C1)CC(C)(C)C N1(C(=O)NCC(C)OCC=C)CCC(c2nccn2C)C1 Cc1c[nH][nH]c1=NC(=O)C1CCCCN1Cc1ccc(Cl)nc1Cl C(CN=C(NCC(C)C)NCc1ccccc1)C1CC(COC)C1.c1cc(C)on1 c1(OC)ccc(C(N2CCN(Cc3cc(Br)ccn3)CC2CC#N)=O)cc1Br C(=O)(C(C)CNC(C1CCCC1OC)=O)N(CC)Cc1ccoc1 CCCC(CC)C(=O)NC1CC2CC1N(C(=O)C1=COCCC1)C2 C(=O)(CCCC(F)(F)F)NC(c1ccc(C(C)C)cc1)CNC(C(CC)O)=O N1(C(C2C(C)C2)=O)CCC(NC(=O)CCCCCc2ccccc2)CC(C)(C)C1 CCCCC(CNC(=O)Cc1sc(C)nc1C)NC(C1CC1CF)=O N1(C(c2c(C)cno2)=O)C2CCC(C2)C1CNC(c1ncsc1C(F)(F)F)=O C(=O)(C(F)C(C)(C)O)NC(c1ccc(F)cc1)CNC(C=C(CC)C)=O c1(C(=O)NC2CCCN(C(CC3CN(C)C3)=O)C2)ccc2nn[nH]c2n1 c1(C(=O)NC2CCN(C(C(C)=CC)=O)C2C)c(C)nn(C(C)(C)C)c1C N1(C(c2nc(CC)oc2)=O)CCCCC1C1(NC(=O)CCc2cc(Cl)no2)CC1 c1(C(=O)NCC(C)(C)NC(Cc2ccc(C)c(O)c2)=O)cn2cccc(Cl)c2n1 Cc1ccc(CCC(N2CCC(CN(C(=O)CCC(C)(C)F)C)C2)=O)cc1C C1(NC(C2CC3(C2)CC3F)=O)CC2CN(C(C34CCC(O)(CC3)CC4)=O)CC2C1 CC(C)CCCC(=O)NC1(C)CCN(C(c2cnn(C(C)(C)C)c2Br)=O)C1 c1(C(N2C(CNC(=O)C3=CCSC3)CC(C)(C)C2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] C1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)CC)CCCC(C)(C)C1 C1(CC=C)(NC(c2csc(C(F)F)n2)=O)CCN(C(c2nn(C)cc2C)=O)CC1 C(CC(C)(C)C(=O)NC1CCC1CNC(c1sccc1NS(C)(=O)=O)=O)SC c1(C2C(CC)CCC2)nc(-c2cccc(Cl)c2)nn1CCN(C)C N1(C(c2c(C)nc(C3CC3)o2)=O)CCN(C(=O)CCCCC2CC2)C2CCC12 c1(C(N2CC3(CN(C(C)(C)C)C3)C2)=O)cccc2nc(C3CC3)sc12 N1(C(CCSCC)=O)CCc2ccccc2C1CCNC(=O)CCS(N)(=O)=O c1(C(N2CCCC(N(C(CNC(CC)=O)=O)CC)CC2)=O)nccc2nn[nH]c12 C(CCSC)(C(=O)NC1(C)CC(NC(=O)CNc2ccccc2C)C1)OC C(=O)(C(C)(C)C(=O)N1CC=CC(NC(=O)Cn2cc(Cl)cn2)C1)NC N1(C(C(c2n(C)ncc2)NC(=O)CCN2CCCC2=O)=O)CC(O)C(O)C1 C1(CNC(CCN(CC)CC)=O)CCCN(C(=O)C(C)(C#N)CC)CC1 C(=O)(C(CCC(C)(C)C)N(C)Cc1ccc(C(C)C)cc1)NCC c1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CCCC2)cc(Cl)ccc1N C(=O)(C1=CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NCC1(CN(C)C)CC1 CC(C(=O)N1C(C(=O)NCC(O)CC2CCCC2)CCC12CC2)S(C)(=O)=O N1(C(c2cc(C)ns2)C(=O)NCCC2CC2)CC(F)(F)CCC1C c1(OC)cc(C(N2CCC(NC(c3cc(F)ccc3O)=O)C2)=O)cc(F)c1F CP(C)(=O)C1CCC(C(=O)NCC(N)CC2CCCC2)C1 c1(C(N2CCC(CNC(C3(CC#C)CC=CCC3)=O)CC2)=O)n[nH]cc1[N+](=O)[O-] C#CCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1cc(C)n(C(F)F)n1)=O C1(c2nnnn2C)(C(c2ccc(Cl)cc2)C)CNC(=O)Cc2ccccc2CC1 C1(CC)CCCCN1C(C1CC(NC(C2(CC)CC2)=O)C(O)C1)=O c1(NC(c2nc(C)oc2)=O)ccc(NCc2ccc(CO)cc2)nc1 C1(C(N2CCCCC(NC(CN(C)S(N)(=O)=O)=O)C2)=O)CCn2nncc2C1 C12(C(N(CCCNC(c3ccc(CO)cn3)=O)CC)=O)CCC(CC1=O)C2(C)C c1(C(=O)OC)ncccc1NC(=O)N(C1CCCC1)Cc1ccc(COC)o1 C(=O)(C(CNC(=O)CCC(C)CN(C)C)CC(C)C)NCC(CCC)OC C(c1ccccn1)=CC(=O)NC1(C)CC(NC(=O)Cc2cc[nH]n2)C1 C=C(F)C1(CC(=O)NC2CC(C(=O)NCC(=O)N(C)OC)C2(C)C)CCC1 c1(NC(C(=O)NC(CCC)C(=O)NC2CCC(C3CC3)C2)C)cccc(F)c1C O=C(CCCn1cccc1)NCC(C1CC1)NC(=O)CCN1CCC(F)C1 C(=O)(C(C(=O)NC1CC(N(N2CCN(CC(C)O)CC2)C)C1)OC)OC c1(C(=O)NC2CCN(C(C(C)N(C)C)=O)C(C)C2)cn2c(n1)COCC2 O=C(C#CC1CCCCO1)NCC1CCCCN1C(c1ccc2c(c1)OCO2)=O N1(C(c2ccc(COC)s2)=O)CC(O)CC1CNC(C1(C)CCCCC1)=O C1(C(=O)NCC2=CCN(C(c3ccoc3)=O)CC2)CCc2nccn2C1 C(=O)(C#CC1CCC1)NC(C1CC=CCC1)C(=O)NCCCNC(=O)OC c1(C(=O)NCCCCNC(C=CC=CCC)=O)ccnn1C(C)C N1(C(CN2C(C)CCC2)=O)CCC(C(=O)NCCCC2CC2C)C12CCC2 C1(CC=C)(NC(C2CC2C2CC2)=O)CCN(C(c2cc(OC)ncn2)=O)CC1 N1(C(c2cn(CCC)nc2C)C(=O)NCC2CC2)Cc2ccc(C#N)cc2C1 Cc1cc(Br)ccc1C(N1CCCC(N(C)C(c2cn(C)cn2)=O)C1)=O C1(NC(C(CC=C)C)=O)CS(=O)(=O)C2CN(C(=O)C#CC3CC(F)(F)C3)CC12 c1(C(=O)NC(CC)CN(C(=O)CC2C=CCC2)C)cnc(S)nc1 C(CCC(=O)N(C(c1ccccc1)CNC(=O)C(c1cccnc1)C)C)=C(C)C c1(C(N2CCCC(CC=C)(NC(c3cc[nH]c3)=O)C2)=O)ccc2cccnc2c1 Cc1ccc(C(=O)NCCOCCOCCNC(=O)C(O)CSC)cc1SC.C(C)C CCC(CC(F)(F)F)C(=O)NCCN(C)C(c1cccn2nncc12)=O C1(CNC(C(CCCC)C)=O)CC2(CCC2)CN1C(c1ccc(N)cc1Cl)=O c1(-c2nnc(-c3c(OC(F)F)ccc(C)c3)o2)cc2n(c1)CCS(=O)(=O)C2 c1(C(=O)NCC(C)(C(C)C)NC(C=C(COC)C)=O)cn(C)c(=O)c(C)n1 Cc1ccc(C2(CN(S(=O)(=O)CC(F)F)C(=O)OC(C)(C)C)CCC2)cc1 c1(CNC(C(C)N(C(=O)CC2CCCO2)CC)=O)csc(C)c1 c1(C(=O)NC2CCN(C(C3CNC(=O)N3)=O)CC2O)n[nH]c2c1CCOC2 N1(C(c2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(C)CCCC2O)C1 CC(C)C(C)CC(=O)N1CCN(C(c2cc(O)nc(O)n2)=O)C(CF)C1 N1(C(C(CC=C)C)=O)CCC(COC)(NC(=O)CC2CN(C(C)=O)C2)CC1 N1(C(C)=O)CCCCC1COC(=O)C(C1CN(C(=O)NC23COCC2C3)C1)OC CC(=O)CCCC(=O)N1CCCC(NC(c2ccc(Cl)nc2N)=O)C1 C1(NC(Cc2onc(C)n2)=O)CCSC12CN(c1nc(C(C)C)ccc1C#N)C2 c1(NC(C(=O)OC(c2cccc(OC(F)(F)F)c2)C)=O)c[nH]c2ccc(Cl)cc12 c1(C(C(F)F)NC(C2C(C)(C)NC2)=O)ccccc1F N1(C(CC(=O)NC)=O)CCCC(C)C1CNC(C1CCC(CC2CC2)CC1)=O CCCC(C(=O)N1CCCC1C(C)NC(C1(C(F)(F)F)CC1)=O)S(N)(=O)=O N1(C(C(C)(C)C#N)=O)CCCC2(C1)CN(C(=O)CCCCCCCCO)CCO2 C1(C(=O)NC2C(CNC(C3(C)C(C)C3)=O)COC2)CC(C)(C)OC1(C)C C1(NC(c2c(CC)nco2)=O)CC2CCC1C(NC(=O)CCOC)C2 C(=O)(C1=CCCC1C)NC(c1cccnc1)C(=O)NC(CCCC=C)C1CC1 C1(NC(C(=C)Cc2ccccc2)=O)CN(C(c2ccc(CC)cn2)=O)CC1F Fc1ccc2sc(CN3CCN(c4ccc(Br)cn4)CC3)nc2c1 Cc1ccc(CC(=O)NCC(O)CCNC(c2ccc3c(c2)CC3)=O)c(F)c1F C(CN=c1[nH]c(=NCC2CN(CC(F)(F)F)C2)c2[nH]ccc2[nH]1)c1occc1 CC1(C)CN(C(=O)CCc2cnccn2)CC1CNC(C1(C(F)F)CC1(F)F)=O c1(C(N(C2CCCN(C(c3cc(N)ccc3Cl)=O)C2)C)=O)scc2c1CCCC2 c1(C(=O)NCC2CN(C(C(N3CCC(C)CC3)=O)=O)CC2C)n[nH]c2c1COC2 Cc1cc(C)n(Cc2ccc(C(=O)NCCCNC(C3CC3(F)Cl)=O)o2)n1 CC1OCCC1C(=O)NCC1CC(C(=O)NC(C(N)=O)C2CC2)C1 N1(C(c2cc(CNC(C(C)(CO)OC)=O)no2)=O)CC2(CCCO2)C1 C#CCC(CC#C)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(C2OCCN(C)C2=O)=O)CC12CCN(C(c1ccc(CO)o1)=O)CC2 O=C1CC(NCCN2CCN(Cc3ccccn3)CC2)CC1(F)F Cc1cc(C(N2CCC2C(=O)NC(C)C)=O)c[nH]c1=N C12(CCNC(C3CC(O)(CC#C)C3)=O)CCC1CN(C(=O)C=CCOC)C2 C1(C)(CNC(C2ON=C(CC)C2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 c1(OC)ccc(C(=O)NCC(C2CC2)NC(=O)CCN2CCCCC2)s1 Cc1cccc(N)c1C(=O)N(C)CCC1CCCCN1C(c1ccoc1)=O CC1(COC(c2cnc(-c3ccsc3)s2)=O)CCCCC1 C12(C(N3CC(n4cc(C(=O)NCCOC)nn4)C(O)C3)=O)CC1COC2(C)C N1(CCC2N(C)CCC2)CCOCc2ccc(Br)cc21 Cc1cc(C(=O)NCC2(F)CN(C(c3ncccc3F)=O)C2)c(Cl)cc1F C1(CNC(CC(CC)C)=O)CN(C(C2CCCN2C)=O)CCC1(C)C C1(C(=O)NC(CN(C)C(c2sccc2Br)=O)(C)C)C(C)(C)C1(F)F c1(C(C(=O)N(CCCCNC(C(CN(C)C)(C)C)=O)C)(F)F)cc(Cl)ccc1Cl c1(C(=O)NCCN(C(=O)CN(C)C(N)=O)C(C)C)cn2c(n1)CCC(C)C2 C1(C(=O)NCC(CC)(C)NC(C2CC23CCCC3)=O)CCCCCN1C Cc1nn(C)c(N2CC(n3cc(NC(=O)C(O)CC(C)C)cn3)C2)c1Cl Cc1ccc(C(=O)OCC=CCO)c(N(C(=O)CCC(C)C)C(C)(C)C)c1 c1(C(=O)NCCC2CCC(NC(CN(CCC#C)C)=O)C2)ccc2sncc2c1 c1(C(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CC2)cc(Cl)ccc1N C1(NC(C(c2ccccc2)N)=O)CCN(c2ccccn2)CC1 c1(N2CCC(OCC=C)C2)nc2c(c(=NCc3nc(O)n[nH]3)[nH]1)COC2 N1(C(C2C(C)CC2C)=O)CCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 c1(C(=O)NCCCNC(c2c(CC)ncnc2)=O)cccc(C(F)(F)F)c1C N1(C(Cc2cccc(C)c2)=O)CC(C(=O)NC2CCCCC2)CC(C)C1 c1(CN(CC)CC)ccc(C(=O)NC(C)(C)CCNC(C2(N=[N+]=[N-])CC2)=O)cc1 C1(NC(c2cccc(C)n2)=O)C2CCC(C2)C1C(N1CCCC(CN=[N+]=[N-])C1)=O Cc1cc(C(=O)OCC(c2sc(Cl)cc2Cl)=O)c(O)nn1 N1(C(COCCCC)=O)CC(C)N(C(=O)CCCn2cccn2)CC1C N1(C(C(c2n(C)ncc2)(F)F)=O)CC2CCN(C(=O)C(O)P(C)(C)=O)CC12 N1(C(C(C)(C)CCl)=O)CC2CCC(C1)N2C(c1cc(F)c(Cl)nc1Cl)=O N1(C(C=CCCC)=O)CC2(CCNC(C3(C(N)=O)CCC3)=O)CCC1CC2 c1(C(=O)NC(C)CCCNC(=O)Cc2cccc(O)c2)ncnc2c1OCCO2 C1(CCC)CCCC1C(=O)NCC1CC(NC(=O)COc2cn[nH]c2)C1 c1(OC)ccc(Br)cc1CC(N1CCC2(CC2C(N2CC3CC3C2C#N)=O)C1)=O C1(c2cn(C3CCCC(C)C3)nn2)C2CCCC1N(C(c1cc(I)c[nH]1)=O)C2 C#CC1N(C(c2cccc(N(C(c3c(F)cccc3F)=O)CC)c2)=O)CC1(C)C C1(C(N(C)C)=O)CN(C(c2cccc(C(=O)NC3CCCC(N)C3)c2)=O)CC12CC2 c1(OC)ccc(C2(C(=O)NCCNC(=O)CC3COCCO3)CC2)c(SCC)c1 C1(N(C)C)CN(C(C2CCN(c3ccc(Cl)cn3)CC2)=O)CC1C(=O)O c1(CC(=O)NC2COCCC2NC(C2(n3cnnn3)CC2)=O)ccc(Cl)cc1F N1(C(C(C)OCCCC)=O)CC2CCCC2(NC(=O)Cc2ccc(Br)cc2)C1 c1(CC(N2CCC(NC(C=C(CC)C)=O)C2CC)=O)cnc(Cl)cc1C C(c1cc(Br)ccc1F)=CC(=O)NCc1nc(C(CC)C)on1 C1(C)(CNC(CC(CN(C)C)O)=O)CC(F)(F)CN1C(c1ccncc1O)=O C1(F)(CNC(CN(C(C)=O)C)=O)CCN(C(=O)COC2(C)CCC2)C1 c1(CC)nc(C)oc1C(=O)NC1CCOCC1C(=O)NCCC1(C)CC1 N1(C(C(C)=CC)=O)Cc2ccccc2C(NC(C2(COC)COC2)=O)C1 c1(C(=O)NC(CCNC(c2c(CC)non2)=O)C)cc([N+](=O)[O-])cc(C)c1Cl c1(OC)cccc(C)c1NC(N1CCN(C(CN(C(=O)C(C)CO)C)=O)CC1)=O Cc1snnc1C(=O)N(C1CC1)CC1CCCN1C(c1ccsn1)=O C1(C(N2CCCC(CO)C2)=O)CC(O)CN1C(=O)CCc1ccccc1F C1(NC(C=C(C)Cl)=O)C2CC3CN(C(=O)CCc4n[nH]c(=N)s4)C1C3C2 C(C(C)CC(=O)N1CCCC1C(C)(C)NC(C1CCS(=O)(=O)C1)=O)OC CC(CC(=O)NCC1(O)CC(C(=O)NCCCCCN(C)C)C1)C(F)(F)F N1(C(C(C(C)C)SCC)=O)CCN(C(C2(C)CC2)=O)CC12CC2 N1(C(CCCC2(C)N=N2)=O)CCOCC(NC(C2(CO)CCOCC2)=O)C1 c1(CC(N2CC3(CN(C(C45CC(C)C4C5)=O)C3)C2)=O)cccc([N+](=O)[O-])c1 C#CCC(CC(F)F)C(=O)NC(C(N1CC(F)CC1C)=O)C1CC1 c1(N2CCC(C(C)NC(C(C(C)C)C)=O)CC2)nc(Cl)nc2[nH]cnc12 c1(C(C(=O)NCC(C)NC(=O)CCn2cc(Cl)cn2)O)cc(F)c(F)cc1F Cc1c(C(=O)NCC2(NC(C3COC4(CCC4)C3)=O)CC(F)(F)C2)cccc1F C1(C(=O)NCCC(C)N(C(=O)C=CC(N)=O)C)Cc2nccnc2C1 CS(=O)c1cccc(C(=O)NCc2cc(O)nc(CNC(=O)C#CC3CC3)n2)c1 c1(OCC)c(F)cc(C(N2CC3=C(C2)CN(C(c2cnco2)=O)C3)=O)cc1Cl c1(C(=O)NC2CCN(C(c3ccc(COC)s3)=O)C2)n[nH]c2nccc(Cl)c12 c1(C(=O)NC(C2N(C(C=C(COC)C)=O)CCCC2)C)cccc2ncccc12 N1(C(C2(C#N)CC2)=O)CC(C2CCCN(C(C3CC4(CCC4O)C3)=O)C2)C1 C(=O)(C(C)C(O)C(C)CC)N1CC(C(=O)Nn2cncn2)(CCC=C)C1 c1(C(=O)NC(CCOC)CNC(=O)COCC2CC2)cccc2c(C)ccnc12 c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCC3)C2)cc2ccncc2s1 CCS(=O)(=O)c1ccccc1C(=O)N(CC(C)(C)NC(C1COC(=O)N1)=O)C C1(CNC(CCSC)=O)CC(C)N(C(=O)C(C)=C2CC2)C1 CC#CCCCC(=O)N1CCC(C(C)C(=O)NCC(CC)C(C)(F)F)C1 N1(C(C2CCN(C(CC)=O)C2)=O)CCOCC1CO.C1(C(=O)N)CC(=O)N(C(C)C)C1 c1(C(=O)NCC(C)NC(c2ccc(OCC)nc2)=O)ccc(CC)c(OC)c1 CCCC(C(=O)N1CCCC1CCCNC(=O)C=C1CCCC1)N(C)C c1(CC)nc(C(=O)NCC2(C(=O)NCCC#CCO)CCCCC2)c(C)o1 N1(C(C2(C)C(C)(C)C2)=O)CCC(C2CN(C(C3CC4(CCC4)CO3)=O)C2)CC1 c1(CNC(C(CC2CCCOC2)N(C)C)=O)ccc2ccccc2c1Br C1(C(=O)NC(c2ccc(N(C)C)cc2)C)CN(C(=O)C=C2CC2)CC1CC(C)(C)C c1(NC(C)=O)cccc(CC(=O)NCCCC(C)NC(=O)C(O)C(C)C)c1 c1(-c2c(S(C)=O)cccc2)ccc2c(C(=O)Nc3cc(O)ccn3)nsc2c1 c1(NC(N2CCC2CF)=O)cc(O)c2ccccc2n1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(CCNC(c1c(CC)cncc1)=O)C c1(C(=O)NC2C3CN(c4cc(C(C)C)nc(Cl)n4)CC32)c[nH]nc1S(N)(=O)=O c1(OC)cc(OC)c(C(N2CCN(C(=O)C(C)=C(C)C)CC(O)C2)=O)cc1OC c1(C(C(=O)NC2(c3nnc(C(=O)OCC)s3)CC2)(F)F)ccc(F)cc1C C12(CNC(CC3CCCN(C(C(C)(C)OC)=O)C3)=O)CCC(C1)C(=O)N2 c1(C(=O)O)ccc2nc(C3CC3)oc2c1.C12CCN(CC1)CC(C1CC1)N2 O=C(C1=NOC2(CCCN(C(c3ccc(Cl)cc3F)=O)C2)C1)N(CCO)C1CC1 Cc1cc(C(C)C)ccc1C(N1CCC(NC(c2cc(O)ncn2)=O)C(F)C1)=O CCN=c1ccc(C(=O)Nc2cccc(NC(C3CC4CCC3C4)=O)c2)c[nH]1 Cn1ccc2c(C(=O)NCC3(F)CCCN(C(=O)CCC(C)(F)F)C3)ncnc12 CC1CCCCC1(CNC(c1nc[nH]c1C(F)(F)F)=O)NC(=O)C=CCO C(=O)(C1=C(C)OCCS1(=O)=O)NC1CCC(CCNC(c2cc(OC)no2)=O)C1 C(=O)(C(C)(C)C(=O)N(C)C)NC1C(N(C)C(C2CCC2c2nc[nH]n2)=O)CCCC1 C1(C(N2CC(O)(CN(C(C(C)OCC3CC3)=O)C)C2)=O)CC2(C1)CC(CO)C2 C(=O)(C1=CC2(CCN(C(=O)C=Cc3nccs3)C2)C1)NCC(CC(=O)NC)C Cn1cc(S(C)(=N)=O)c(CNC(c2cc(Br)ccc2-n2cnnn2)=O)n1 N(C1CCOc2ncccc21)S(c1ccc(C(N(CCC#N)CC)=O)cc1)(=O)=O c1(OC)ccc(C(=O)NC2CN(C(c3cc(C(N)=O)cc(F)c3)=O)C2)c(F)c1F CC(CC(=O)NC1CN(C(c2occ3c2CCC3)=O)CCC1F)CC(F)(F)F C(=O)(CC(C)(C)CC(=O)N1CCCC2CN(c3ncnc(Cl)c3C)CC12)OC c1(C(N2C(C)(C)C(C(=O)NCC(O)CO)CC2)=O)cnn2ccccc12 Cc1cccnc1C(=O)NC1CC(NC(C2CCC(NC(N)=O)C2)=O)C1 C1(C(N2CCCC(CC3CC3)C2)C(=O)NCCCF)CCCN(CCO)C1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(OC)CC(NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 Cc1ccc(C(=O)NC2(CO)CCN(C(C3(C)CCOC3)=O)C2)cc1C#N N1(C(C(C(C)C)=O)=O)CCC(C)(C(=O)NC2CCC(F)(F)CC2)CC1 C1(NC(CNC(=O)NC)=O)(CO)CCN(C(=O)Cc2cc(Cl)ccc2OC)CC1 C(CC(N)=O)(C(=O)Nc1ccc(C)c(C(N)=O)c1)NC(C1CCC(C)(CC)O1)=O N1(C(C(CC=C)CC)=O)CC2(C1)CN(C(c1cc3c(cc1Cl)NCC3)=O)CCO2 Cc1ccccc1CN(C(=O)C(F)C(C1CC1)C1CC1)c1ccccc1 N1(C(C(C)c2ncco2)=O)C2CCC1CN(C(=O)COc1ccc(F)cn1)C2 CC1CN(C(C2CCC(O)CC2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)O1 Cc1nnc2n1CC(NC(=O)NCC1COCCOC1)CC2 C12(CNC(c3n(CC)cc(Cl)c3)=O)CCC(CNC(C3CC3Cl)=O)(CC1)CO2 C1(CC(=O)NC(CCCC=C)C2CC2)CCC2(CCN(NC(=O)OC(C)(C)C)C2)C1 N1(C(CCC(C)(C)F)=O)CCC2CN(C(c3cnn4c3OCCC4)=O)CC12 c1(C(=O)OC)cccc(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c1 C(=O)(C1CCCc2scnc21)NC(CCCCNC(CSC)=O)C C1(CCC)CN(C(=O)CNc2cccc(Cl)c2)CC1NC(=O)COC1CC1 Cc1c(C(N2CC(C)(CNC(c3ccc(Cl)c(Br)c3)=O)C2)=O)cccc1O C1(NC(C2CC(OC)C2)=O)CCSC12CN(C(=O)CC(=O)OC(C)(C)C)C2 N1(C(C2(CC)COC2)=O)CC2(CO)CC1(C(N1CCC(SC)CC1)=O)C2 c1(OCCCCOC(COC(CC)=O)=O)ccc(S(C)(=O)=O)cc1 C1(CC)CC(C(=O)N(C2CC2C2CC2)C)CCN1C(c1ccsc1C#N)=O C1(C(=O)NCC(=C)C)CCCN(Cc2ncccc2Br)C1 C1(C(N2CCC(C(=O)NC)C2)=O)CN(C(=O)Cn2ncnn2)CCN1C Cc1nc[nH]c1C(=O)NC1COCC1NC(=O)COCC(F)(F)F C1(NC(C(CC)OC)=O)CCN(C)C12CCCN(C(C1(CC)COC1)=O)C2 CC1(C)CN(N2CCN(c3ncnc4[nH]ccc34)CC2)CCC1CO N1(C(CCSCCC)=O)CC(NC(c2ncsc2Br)=O)C(C2CC2)C1 C1(C(=O)NC(c2ccc(F)c(F)c2)(C(=O)OC)C)CSC(c2cccs2)=N1 c1(COC)ccnc(C(=O)NC(C)CN(C(=O)COCC2CCCOC2)C)c1 c1(CC)nc2ccccn2c1C(=O)NNC(=O)C1CNC(CN)C1 C(c1ccc(F)c(C)c1)=CC(=O)NC1CC(C)(NC(C(CC)SC)=O)C1 c1(NC(C2(SC)CN(C(c3sc(O)nc3C)=O)C2)=O)ccc2ccncc2c1 C12(C(N3CC(NC(C4C(C)(C)CO4)=O)(CO)C3)=O)CCCN(CC1)C2 Cc1c(C(N2CC(NC(=O)C(CO)N(C)C)C(F)C2)=O)nnn1C(C)C c1(C(N(CC(CC)NC(=O)C(C(C)C)N(C)C)C)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCCN(C(=O)C(O)c2ccco2)C)csc2cncn12 S(=O)(=O)(c1ccc(O)c(C(=O)O)c1)N1C(C)(CC(C)C)CCC1 c1(SC)ncc(C(=O)N(C)CCN(C(=O)CSc2nncn2C)C)s1 C12(C(=O)NCC3CN(C(C4C(C)CC4)=O)C(C)(C)C3)CC3CC1C2C3(F)F C1(CC(=O)NCCOC2CCC2)(OC(=O)CCC2CCC2)COC1 C1(NC(C2CC3(CC(F)C3)C2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1F CON(Cc1ccc(Cl)cc1)C(=O)CC1(C)CCC(=O)NC1 N1(C(C2(CCC)CCC2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 c1(C(N(CC(CN(C(C=CC=CC)=O)C)O)C)=O)c(C)noc1N C1(C(=O)NCCN(C(C2CCC(N(C)C)CC2)=O)CC)CCC2CCCCN12 C1(OC)CCC2(C(N3CSCC3C(=O)NCCC(C(C)C)OC)=O)CC12 C(=O)(C#CC1CCOC1)NC1C(NC(c2cc(C)c(C)s2)=O)CCOC1 c1(C(=O)O)cc(CN2CCC(F)(C(=O)Nc3c(Br)ccnc3Br)C2)ccc1O C1(NC(CCC2C(C)=NNC2=O)=O)CN(C(c2cnc[nH]2)=O)CC2(CC2)C1 c1(NC(c2cc3sccn3c2)=O)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(CNC(c2ncc(OCC)nc2)=O)O)CC(=O)CC12CCC2 N1(C(=O)COC2CN(C(C3CCCCO3)=O)C2)CCc2cccnc2C1 c1(CC(=O)N(C2CCN(C(COCC#C)=O)C2)CC#C)cc(Cl)cc(Cl)c1 N1(C(CCSC)=O)CC(NC(=O)C(c2cncn2C)O)C(C2CC2)C1 S(=O)(=O)(c1ccc(F)cc1)NCCNC(c1scc(C)n1)C c1(C(=O)NC2CCC(NC(c3cccc(CO)c3)=O)C2)cnnc(C2CC2)c1 c1(C(N(C2CCN(C(C3CCC(=O)N3)=O)C2)CC)=O)n[nH]c2c1CCC2 C1(CNC(C2CC(C(=O)OC)C2)=O)(CNC(=O)CC2COC(=O)C2)CCCCC1 Cn1nc(-n2cc(CNC3CCC3c3ccccc3)nn2)nc1Br c1(COCC)nc(C)cc(=NC2CC3CN(C(c4csnn4)=O)CC23)[nH]1 C1(NC(C2(COC)CCC2)=O)CCC(C)N(C(=O)C2=COCCO2)C1 n1(C2CN(C(C3(F)C(C)C3)=O)C2)cc(CNC(=O)C=CC2CCCC2)nn1 C(=O)(C1CCc2snnc21)N1C(CNC(C2(C(=O)NC)CC2)=O)CC(O)C1 N12CCc3cccc(c3C1)C2=O.CC1=CCCC(C)C1C(=O)NC(C)(C)C C(CC(C(C)C)NC(c1ccc(SC(F)(F)F)cc1)=O)NC(C(COC)O)=O C(C(N=[N+]=[N-])C(=O)N1CCC(CCC(=O)N(C)CCO)CC1)OCC CC1(NC(=O)C=C2CC2)CCC(NC(c2cccc(CF)c2)=O)CC1 C(c1cnc(C)nc1O)=CC(=O)NCCC1(NC(c2c(CC)nco2)=O)CCC1 CCCC(O)CC(=O)N1CC(O)(CN(C)C(c2cnn(C(C)CC)c2C)=O)C1 C1(NCCC)CCCN(C(c2ccc(-c3cccnc3)s2)C(=O)NC(C)C)CC1 N1(C(C(Cc2cn[nH]c2)NC(C(c2ccccc2)OC)=O)=O)CCN(CCF)CC1 C1(C(N2C(CC(=O)NCc3c(CC)n[nH]c3)CC2)=O)CCCC1C1CC1 c1(N2CCC(NC(CN(C(=O)NC)C)C)C2)ncc(S(=O)(=O)NC)cc1Cl N1(C(c2c(C)ncnc2)=O)CC2CCC(N(C(=O)C(O)C(F)(F)F)C)C2C1 c1(C(=O)NC2(CNC(=O)Cc3ccc(Br)s3)CCC2)ccc(OC(F)F)cc1 N1(C(CCCC)=O)CC(C)N(C(=O)C=Cc2ccc(C)s2)CC1C C(=O)(C(C(C)(C)C)C1CCC1)NC(CNC(c1cc(C)on1)=O)(C)C c1(SCCC(=O)N(c2cccc(Cl)c2)CCC)nnc(-c2cccs2)n1CCC c1(C(=O)NC2(CO)CCCN(C(CCC(CC)OC)=O)C2)n[nH]c2c1COCC2 CC(C)(C)CCCCC(=O)N1CC(=O)NCC1C(N1CC(CCO)C1)=O c1(C(CC(C2CCOC2)NC(=O)CCC2CCC2)=O)cn(-c2cccnc2)nn1 Cc1cccn2ncc(CNCC(c3cc4ccc(Br)cc4s3)=O)c12 CC1(NC(C23CSCC2C3)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(CNC(=O)NCc2cc(C3CCOCC3)no2)ccc(C(F)(F)F)cn1 N1(C(C(C)=C(CC)C)=O)CC2(CNC(C3CC3(C)COC)=O)CC1CO2 Cc1cc(F)c(CC(N2CCC(C(C)NC(=O)CC3CC3(Cl)Cl)CC2)=O)cc1F c1(N(CC(CN(C)C(c2cc(CC3CC3)on2)=O)O)C)cc(CO)nc(Cl)n1 c1(OC(C(=O)N(C2CCN(C(C(CC)(C)O)=O)C2)CCO)C)ccc(O)c(F)c1 N1(C(C(C)OCC=C)=O)CCC2CN(C(C3CC(n4ccnn4)C3)=O)CC12 C1(C(=O)NCC)CCCCC1SN1CCC1C(N)=O.c12cccc(n1)C2 C1(CNC(C(C)(CSC)NC(CC(C)SC)=O)=O)Cc2nccn2C1 CC1CC(c2ccc(F)cc2)CN1C(=O)CS(=O)(=O)N1CCN(C)CC1 Cc1csc(CNC2CC2C(=O)NCc2ccc(O)cc2)c1C CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(COCC)N=[N+]=[N-])CC1CO C1(CC)CN(C(=O)C(O)C(C)C)CCN1C(=O)CCCN(C)C(C)=O c1(NC(=O)COCCC(C)C)cccc(C)c1.C(C)(C(=O)N1CC2CC2C1)OC CC1=NNC(=O)C1CC(=O)N(C)CC1CCCN1C(=O)CCC1CC1(F)F c1(C2(C)CC2)nc(N2CCN(C(C3CCCC(C)C3)=O)CC2)cc(Cl)n1 C(=O)(C(C)(C)CNC(=O)C(C1CCN(C(c2c[nH][nH]c2=N)=O)C1)F)NC c1(C(N2CCCN(C(c3ccc(C)nn3)=O)CC2C)=O)sc2nnc(S)n2c1C C(=O)(C1CSc2ccccc21)NC1CC(CNC(C(=Cc2cccs2)C)=O)C1 C1(CC(N2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C(O)C2)=O)CCC2(CCC2)CO1 C12(CCNC(=O)C(C3CCCCC3)O)CCC(CC1)N(C(=O)CN1CCCC1)C2 c1(C(=O)NCC2OCCCN(C(C3C(C#N)C3)=O)C2)cccc2ccoc12 C1(C(N2CC(O)(CNC(c3c(C)sc(Cl)n3)=O)C2)=O)OCC2CCCC12 C1(C(N2C(CNC(C(CCCOC)C)=O)CC(F)C2)=O)CN=C2N=CNN2C1 C(=O)(C(C(C)F)NC(C)=O)NCC1CC(CCNC(CC2CC(OC)C2)=O)C1 C=Cc1ccc(C(=O)NC2CCCC2NC(=O)C(F)C2CCCC2)cc1 C1(CNC(CCC(=O)OC)=O)(CNC(=O)CCC(C)(C)C)CC2CCCC2C1 C(CCS(N)(=O)=O)C1CC(n2cc(-c3c(C)n[nH]c3)nn2)C1 CCCCCCCCCCCCCC(O)COC(=O)C(F)CC(C)C c1(C(=O)NCC2(O)CCN(C(c3cncc(O)c3)=O)C2)cc2c(Cl)cccc2[nH]1 C1(O)(CNC(CC)=O)CCN(C(c2ccnnc2NC2CC2)=O)C1 N1(C(c2c(C)n(C(C)C)nc2)=O)CCC(C)C(N(C(=O)C(C)O)C)C1 C#CC1(O)CCCN(C(c2cnn(Cc3cc(C)ccc3F)c2)=O)C1 C#CC1CCCN1C(=O)C(C)CNC(=O)CCC(=O)C1CC1 Cc1nc2c(s1)CCCC2C(=O)N1CCC(CNC(c2cnsc2)=O)C(F)(F)C1 c1(N(CCOC)C)cc(N2CCC(CC(N)=O)C2)nc(NCC2CCCO2)n1 C1(CC(=O)NCCOC(C)=O)CCCCC1NC(=O)Cc1ccc(C)s1 c1(C(=O)NC2CCN(C(Cc3nc(C)sc3C)=O)C2)cc2nc(Cl)ccc2s1 N1(C(C(C)C(F)F)=O)CC(NC(c2cc(F)ccc2Br)=O)C(C2CC2)C1 C1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)CC2CCC(C1)C2 C(c1c(C)coc1C)=CC(=O)NC1C(C)(CNC(C(COC)O)=O)CCC1 C1(C(=O)NC2CC(NC(COc3cn(C)nc3)=O)C2)CN2CC3CC2(CO1)C3 CCCCC(C(=O)N1CCCC1C1CCN(C(c2nocc2Br)=O)CC1)N(C)C Cc1cnc(F)cc1C(=O)NC1CCCCN(C(C23CC2C3)=O)C1 c1(N(C)Cc2ccoc2)nc(N2CCCC(F)CC2)c2c(n1)CCOC2 c1(OC)ccc(NC(=O)C(=O)NC(c2cnsc2)C)c(C#N)c1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)NCCCS(N)(=O)=O)C(F)C1 C12(C(=O)NCC(C)N(C(=O)Cc3ccccn3)C)CCC(C1)C2(C)C c1(CC)nncn1NC(=O)C(CCC(C)C)NC(c1cccc(C)c1F)=O C(=O)(CCCC(=O)NCC1C2CN(C(C3COCCO3)=O)CC12)NC(C)C CC1=C(C)CC(C(=O)NC2CC(C(=O)NC3CCCC3CN)C23CCC3)CC1 CC(C(=O)NCC(C1CC1)N(C)C(c1cnnc(O)c1)=O)C(F)F N1(C(CNC(CC)=O)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 Cc1nn(C)cc1C(C)C(=O)NC(C)CNC(C1(S(N)(=O)=O)CC1)=O C(CC[Si](C)(C)C)NC(C(N1CCC(CCC(=O)NC(C)C)C1)=O)=O C1(CCOC)(NC(c2cc(C)n(C)n2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1 CC(C)(C)C(CNC(C1(C#N)CC1)=O)NC(c1cnncc1O)=O C1(C(=O)NCCOCCOC)(OCCSCCON(C)C)CC1 C(CC(O)C(F)(F)F)CONC(CCC1N(C(CCc2onc(C)n2)=O)CC1)=O CC1CN(C(C2CCCCCN2C)=O)CCC1CN=c1ccnc[nH]1 N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CC1(C#N)CCCCC1 C1(COCC)CCN(C(=O)CCCNC(C2COCCN2C2CCCC2)=O)CC1 c1(-c2cn(C3(NC(COCP(C)(C)=O)=O)CC3)nn2)cccc(O)c1 N1(CC(=O)N(CC(C)NC(=O)CC2CC(F)C2)C)CC(=O)NC1=O N1(C(C2(OC)CCC2)=O)CCN(CC2CN(C(c3cnc(O)o3)=O)C2)CC1 C12(C(N(CC(COC)O)C)=O)CC(CN(C(=O)CCS(N)(=O)=O)C1)C2 c1(C(=O)NC23CC(C(=O)NCC4(C#N)CC4)(C2)C3)ccc(OC(F)F)c(F)c1 c1(C(N2CCCC(C(C)NC(=O)C3=CCSC3)C2)=O)c(F)cc(F)cc1F c1(C(N(C2CN(C(COCCC#C)=O)CC2F)C)=O)cc(C)n(CC)c1C N1(C(C(CCC)C)=O)CC2(C1)CN(C(=O)C(C)S)CC2C(=O)O c1(C(=O)NCCCCCCC=C)ccccc1S(=O)(=O)N1CCCCC1C C1(CNC(C(COC)C)=O)CCCCN(C(=O)C(C)N(C)C)C1 N1(C(CCC)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)o2)CC12CCCC2 C(=O)(C1CCc2nnc(C)n21)C1(C2N(CCc3c(C)cc(O)cc3)CCC2)CC1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)c(S)n1 C1(C(=O)NCC2CC(C(N3C(C(C)C)CCC3)=O)C2)CCN(C)C(=O)C1 Cc1ccc(C(N2CC3C(CNC(=O)CCCCC(N)=O)C3C2)=O)c(O)c1C Cc1cn2c(CC(=O)NC3CC(NC(c4ccc(F)cc4F)=O)C3)csc2n1 CN(C)S(=O)(=O)N(C)CC(=O)NCCCC1CCN(C(C2CCS2(=O)=O)=O)CC1 c1(CC)cccc(NCC2CCC(C(=O)OC)O2)c1 c1(CN2CC3C(C(=O)NCCCOC)C3C2)cccc(OC)c1OC c1(COC(CC2C(OC)COCC2)=O)nc2cc(Cl)ccc2s1 Cc1cc(C#N)cnc1N(C1CCCN(C(C2(F)CCOC2C)=O)C1)C c1(C(N(C2CCCN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)C)=O)cc2c(s1)CCC2 c1(N(C(C(C)Cc2ccnn2C)=O)C(C)C)cnnc(Br)c1 c1(C(=O)NC2C(CNC(C(N3C(CC)CCC3)=O)=O)CC2)cccc(CO)n1 c1(C(=O)NC(C(C)C)CNC(c2cn(C)ccc2=O)=O)cc(N)c(N)cc1F c1(C2(NC(=O)C(F)=CC3CC3)CN(C(c3cccc(Cl)c3)=O)C2)ccc(F)cc1 C(=O)(C(C#N)C(C)C)NCC#CC(=O)N(CC(COC)C)C c1(CC)ccc(C=CC(N2CCCC2CCNC(=O)C(F)n2ccnc2)=O)cc1 CC#CCCCC(C)(c1nnnn1C(C)C)NC(C)Cc1ccc(OCC)cc1 c1(C(=O)Nc2c(OC)nc(F)cc2)cc(-c2cccc(F)c2)cc2c[nH]nc12 C1(NC(Cc2cc(C)sc2)=O)CC(=O)N(C2CN(C(=O)C(C)C(C)C)C2)C1 C1(CNC(c2ccnc(C)n2)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)F Cc1nn(CCO)cc1C(=O)NC1CC(C)N(C(=O)COc2ccc(F)cn2)C1 N1(C(CCCCOC)=O)CCC2(CC2NC(c2ccncc2F)=O)C1 CN1CCOCC1C(=O)NCCn1cc(C(=O)NCC2CC(F)C2)nn1 c1(C(=O)NC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-n2cnnn2)cc1Cl C(=O)(C(C)(C)C1=CCSCC1)NCCC(C)NC(C1CC1C(F)(F)F)=O C1(NC(c2cnccc2Cl)=O)CCC12CCN(C(=O)CC1CCCCO1)CC2 C1(C(=O)NC2(C)CC(NC(C3C(C)(C)OC(=O)C3)=O)C2)CCCCN1S(N)(=O)=O C1(NC(=O)CC2CN(C(c3cnc(Cl)cc3I)=O)CCO2)CCC(F)(F)CC1 c1(C(N2CCC(NC(C3(CF)CCOCC3)=O)C(F)C2)=O)cc(Cl)cc(Cl)c1Cl c1(OC)cc(CN2CC(O)CC2C(=O)Nc2ccnc(O)c2)ccc1Br CC1(C(=O)NCCCCNC(c2ccc(F)cn2)=O)C2Cc3ccccc3C12 c1(C(=O)NCCn2c(C)ncc2)ccc2c(n1)CN(C(C1CC(C)(O)C1)=O)CC2 CC1(C)CC(C(N2CCC(C(F)F)C2)=O)CN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)NCc2n(C)nnn2)CCCCC1(C)NC(=O)CC1CNC(=O)O1 C1(CC(N2CCN(C(CC)=O)CC2)=O)CC(C)(C)CN1C(=O)CN1CCCCC1 C=C(C)C(C)(C)C(=O)N1CCN(C2CCCN(C(=O)COC(C)(C)CC)C2)CC1 N1(C(C2(c3ccccc3F)CC2)=O)CCN(C(C2CC3CC3C2)=O)CC12CC2 C(C(CC(C)C)NC(c1ccc(C(=O)NC)cc1)=O)NC(C(C)N(CC)CC)=O Cc1[nH]nc(C(=O)NC(C(=O)NCCCC(C)O)C2(O)CCC2)c1C C=C=CC(C)C(=O)N(CCC(=O)NCCN(CCC)CCC)CC C1(C(=O)NCC23OCC(CNC(=O)C4=CCCCO4)(C2)C3)CC2CCC(C1)C2O c1(OC)nccc(CNC(C2CC(NC(C3COC(=O)N3)=O)C(O)C2)=O)n1 c1(COC)ccc(NC(=O)CCN(C)C(c2cn(C(C)C)nn2)=O)cc1 c1(OCOC)ccc(C(=O)NC(C)Cn2cc(C(C3CC3)N(C)C)nn2)cc1 C(CS(=O)(=O)CC(=O)NCC(C)CN(C)C(C1CCCN1C)=O)OC C1(NC(c2cnc(Cl)s2)=O)CCCCC12CCN(C(=O)C1=CC(O)CCC1)CC2 c1(NC(CC)CNC(C2CCCC2(C)C)=O)ccc(C#N)cc1[N+](=O)[O-] C(CC(=O)NCC1(O)CCCCCC1)(C(F)(F)F)NC(c1nn(C)c(=O)cc1)=O C=C(C)CC(C(=O)N(CC(C)(C)C(=O)NC1CCOCC1C)C)OC c1(-c2cc(C(=O)NCC)ncc2)n[nH]c2c1CN(C(c1cccc(Br)c1F)=O)C2 c1(CCC(=O)NC2C(CNC(CN(C(C)C)C)=O)C2)cnn(-c2ccccc2)c1 C1(CNC(C(C)CO)=O)CC2CCC(C1)N2C(c1cnn(C)c1N)=O c1(C(N2CC(NC(CC(CC)OC)=O)CC3(C2)CC3)=O)cc2c(C)n[nH]c2cn1 C1(CC(N2CC(CCNC(C3CCC(C)(C)O3)=O)C2)=O)CCc2sccc2C1=O c1(C(C)=O)cc(C(=O)NC(C2CCOC2)CNC(c2ncoc2C)=O)no1 c1(OC)ccc2[nH]cc(CN3CC4CC3CN4C(C3CCCCC3(F)F)=O)c2c1 O=C(CCC(=O)N1CCOCC1)NCC(CO)NC(c1cn(C2CC2)nn1)=O c1(NC(COC)=O)ccc(Cl)cc1C(=O)NCC(c1ncc(Cl)n1C)=O c1(-n2c(N3C(COC)CCC34CC4)nnc2C2CCCCC2)cc(F)cc(Br)c1 S(=O)(=O)(c1cnn(CCO)c1)N1CC(Nc2cc(OC)cc(OC)c2)N(C)CC1 c1(CNC(C(=O)NC(c2c(C)cnnc2)C)=O)ccc(S(=O)(=O)N(C)C(C)C)cc1 Cc1cn2c(n1)C(C(=O)N1CC(CCNC(c3ccc(C4CC4)s3)=O)C1)CCC2 C(CC(F)F)(C(=O)NC1CCCC1(C)C)N(C(c1nnn(CC)c1C)=O)C N1(C(C(C)OCCOC)=O)CC2CCC(NC(=O)COC(C)C)CC2C1 c1(C(=O)NCCCC(C)NC(c2nccnc2C(F)(F)F)=O)ccc(F)c(Cl)c1 S(=O)(=O)(c1ccc(NC2CCOC2)cc1Br)NC(C)C(c1c(Cl)cccc1Cl)O C1(NC(COCCSC)=O)CCC(CNC(c2ccccc2COC)=O)CC1 Cc1ccc(-n2nc(CC(F)(F)F)nc2C2CC2(c2ccccc2)C)c(C)c1 c1(C(=O)NC2CC(C)(NC(C=NOC)=O)C2)ccc(C2CC2(Cl)Cl)cc1 N1(C(C=C=C(C)C)=O)CCC(C)(CNC(C2CCN2C)=O)CC1 c1(C(N2CCC(NC(C3(C)CCC3)=O)C(F)C2)=O)cc(O)c(O)c(O)c1 c1(NCCn2cc(-c3cnn(C)c3C(N)=O)nn2)ccc2cccnc2n1 N1(C(C2C(CC)C2)=O)CCC2(CCN(C(=O)C(F)CCC(C)C)CC2)C1 N1(C(C2N(C(C3CCC(C)(C)OC3)=O)CCCCC2)=O)C2CCC1CC1(C2)N=N1 c1(CN(C2CCN(C)C2)Cc2csc(Cl)c2)cccc(C(=O)O)c1 c1(CC)c(C(=O)NCCCCNC(c2csc(C)n2)=O)[nH]c(C)c1C(N)=O c1(NC(=O)NCCN(CC)CC)ccc(NCC(c2ccccc2C)(C)C)cc1 N1(C(C2(C#N)CCCO2)=O)CCC(F)(CNC(c2ccc(F)c(Cl)c2)=O)CC1 C(N=c1nc(N2CCCCC(SC)C2)c2c([nH]1)CSC2)c1cc(OCC)ncc1 C12(C(=O)NCC(CC)NC(=O)C(F)CC3CCCC3)CCC(O)(CC1)CC2 C1(C(N2CCC(N(C(C3C4COCC34)=O)CC)CC2)=O)OC(C)(C)OC1(C)C c1(C(=O)NCC2(F)CC(NC(CCS(=O)(=O)N(C)C)=O)C2)nccc2[nH]ccc12 N1(C(N=c2ccn(C(CC)C)[nH]2)=O)CC2(CO)CC(C)(C1)C2 C1(C2CN(C(=O)C(C)S(C)(=O)=O)C2)(NC(c2c(SC)cccn2)=O)CC1 Cn1[nH]c(=NC(=O)C2CCN(Cc3c(Br)cc(F)cc3Br)C2)cc1Cl N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(c2ccnc(C(F)F)c2)=O)C(C)C1 N1(C(C(N)=O)=O)CCOC(CCNC(=O)CCC(=O)c2cccc(F)c2)C1 N1(C(CCOCCC)=O)CCOC(CNC(=O)C#CC2CC2)C1 c1(SC)ccc(C)c(C(=O)NC2CCCC2NC(C2CC23CC(F)(F)C3)=O)c1 N1(C(=O)C(C2CCCC2)C2CCCC2)CCC2(C1)CN(C(C1(F)CCCC1)=O)C2 c1(C(N(CC(CN(C(c2c(C)scc2)=O)C)O)C)=O)nccc(Cl)c1F C(CC(=O)N1CCC(O)(CO)C1)(C(F)F)NC(=O)Cn1cc(CO)nn1 c1(C(=O)NCC2CCCCN2C(=O)CCn2ccnc2)ccc2c(c1)CCC=C2 c1(NC)cc2c(cc1Cl)NC(=O)CO2.C12CC3CC1CN3C(=O)C1CN2C1 C1(c2ccc(F)cc2)(C(=O)NCC2C=CCN2C(c2ccon2)=O)CCCCC1 C1(CCOCCOCCNC(C(C)(C)OCC)=O)CCC(C(C)C)CC1 c1(CN(C2CCC2)C(C2(c3ccncc3F)CC2)=O)ccc(Cl)cc1F C(CC(C(=O)N1CCC(NC(C2CC2[N+](=O)[O-])=O)C1C)OC)OC c1(OCCC(N2CCC(C)(CNC(=O)CCC#N)C2)=O)cccc([N+](=O)[O-])c1 C(C)(C)(C(F)(F)F)NC(CN(C(=O)Cc1ccccn1)CC1C(C)CCC1)=O C1(c2nn[nH]n2)C2CC3CN(C(=O)CCCNC(CCC(=C)C)=O)C1C3C2 c1(C(N(C2CCN(C(c3ncc[nH]c3=O)=O)CC2)CC)=O)cnc2ccoc2c1 c1(CCC)cc(C(N2CCOCC(NC(C3CSCC(=O)N3)=O)C2)=O)ccc1Cl c1(NC2(CNC(C3CCC(C)CC3)=O)CCOCC2)cc2nncn2cn1 c1(C(=O)NCCC2CCC(NC(CC=C)=O)C2)nccc2c1[nH]c1ccccc21 C(=O)(C1Cc2ccccc21)NC(CC=CC(=O)NC(CC=CC)CO)(C)C C(CN=c1ccnc(SC#N)[nH]1)c1ccc(C(=O)O)cc1Cl C1(CCOC)CCN(C(=O)C=C(Br)Br)CC1 c1(CC(=O)NC(CNC(C2C(c3ccc(C)s3)C2)=O)(C)C)cccc(Cl)c1F c1(N2CCCC(NC(=O)CCc3ccc(Cl)s3)CC2)nc2cccc(Br)c2o1 N1(C(=O)C=CBr)CCC2CCC(NC(C3(C4CC4)CC3)=O)C1C2 C(CS(=O)(=O)C(F)(F)F)OCC.c12cc3c(cccc3o1)NCCn1nnnc1-2 C(=O)(CC(O)C(C)C)NCC(CCOC)NC(=O)CN(C)C(=O)OC n1(CC)c(C)nn(CC(=O)N(C(C)CNC(=O)C(CCSC)N(C)C)C)c1=O C1(C(N2CCC(C)(CCNC(CNC(=O)OCC=C)=O)C2)=O)C(F)(F)C12CCC2 C1(C(N(C)CCNC(=O)CCc2nncn2C)=O)CCC(C)(F)CC1 c1(OC)c(Cl)cc(C(N2CCOCC2CNC(C2CC(F)C2)=O)=O)cc1Cl N1(C(Cn2nnc(C)n2)=O)CC(C)CC1C(=O)NC1(CC(C)C)CC1 C1(NC(c2c(C)nc(Br)o2)=O)CC2CCC1CN(C(=O)C(C)C(C)O)C2 c1(CC(=O)NCc2ccccc2CNC(C2(F)CCCC2)=O)ccc(Cl)cc1Cl Cc1nc2ccc(C(=O)NCCN(C(=O)Cn3cccn3)C)cc2s1 C(=O)(CC1OCCc2ccccc21)N1CCC(CN(C(c2cc(C)sn2)=O)C)C1 C1(OC)CN(C(c2cc(C)n(C)c2C)=O)CCC1NC(c1cc(Cl)ncc1Cl)=O c1(C(N2CCC(CCOC)CC2)=O)n[nH]c2ccc(-c3nncs3)cc12 c1(C(=O)NC2(CO)CN(C(C(C)CN(C)C)=O)C2)ccc(CC(C)(C)C)cc1 c1(C(=O)NC2CCN(C(CS(CCCC)(=O)=O)=O)C2)ccccc1C#CC1CC1 c1(C(=O)NCC2C(NC(C(C)OCc3ccncc3)=O)C2)nccc2n[nH]cc12 C1(C(N2CC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)(OC)CCOC1 c1(Cc2nc(CC3CN(c4n(C)nnn4)C3)on2)ccc2cccnc2n1 C1(CN(C)C(C2CC2c2ccsc2)=O)CCCN1C(=O)CCc1cncs1 C1(NC(C(CC)F)=O)CCCC1(C)CNC(=O)CCC1CCC1 C12(CNC(C(CCCC)O)=O)CCC(CN(C(C3(C)CCCN3C(C)=O)=O)C1)C2 c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC(C1(O)CCN(C(C2CCCC2)=O)C1)C N1(C(c2ccc(N(C)C)nc2)=O)CC(NC(c2snc(Cl)c2Cl)=O)CC2(CC2)C1 c1(NC(C(=O)N(C2CCC2)C)=O)ccc2c(c1)COC2(C)C C(=O)(C(O)CC(F)F)N1CCC(CCNC(c2c(C(=O)OC)c[nH]n2)=O)CC1 N1(C(c2nc(SC)sc2)=O)CCC2(CC1)CC(NC(=O)Cc1conc1C)CO2 C#CC1(C(=O)N(C)CCN2CCCC2=O)CCN(C(=O)CC2CC(C)=NO2)C1 c1(OC)cc(C(F)F)ccc1CNC1CN(C)CC1(C)C C1(CNC(C=CSC)=O)CC2(CC2)CN1C(=O)C(c1cccc(C#N)c1)C(C)C c1(C(=O)NCCN(C(=O)C(=O)NCC(F)(F)F)C)ccc2ncn(C)c2n1 C1(CNC(C(C)CN(C)C)=O)CCN(C(c2cnn(C)c2F)=O)C12CC2 Cc1nn2cc(C(=O)NCC3C(C)CCN3c3ncns3)nc2s1 CC(C)C1CNC(=O)c2cc(OCCOCc3cnc4ccc(Br)cc4c3)ccc21 C1(CS(N2CC3C(N(C)C)C3C2)(=O)=O)CC2(CCNCC2)CO1 Cc1c(C(=O)NC(C2(O)CN(C(c3ccc(C#N)s3)=O)C2)C)cnn1C1CCC1 c1(C(=O)NC2CCN(C(C3CSCCS3)=O)C23CC3)c[nH]c2cc(Cl)ccc12 C1(NC(c2cncc(OC)n2)=O)CCC2CC1CN2C(=O)Cc1ccc(Cl)cn1 CCC(C)(CO)C(=O)NCCCCCN(C)C(C1(F)C(C)(C)C1(C)C)=O N1(C(C2(C(=O)OC)CC2)=O)CCC(CCNC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 N#Cc1ccccc1OCC(=O)NC1CC(O)(CNC(=O)CC2CCCCO2)C1 c1(C(=O)NCC2C3CN(C(c4cc(OC)n[nH]4)=O)CC32)nc(Cl)ccc1Cl c1(C(=O)NCC(C)N(C(=O)CN2CCOCC2)CC)cccnc1C c1(NC(N2C(C(N(OC)CCSC)=O)CC(O)C2)=O)cccc2[nH]ccc12 N1(C(CCC(C)c2ccccc2)=O)CC(=O)NCC1C(N1CC2CC1CN2C)=O C1(C(N(CC(CC)C)C)=O)CCN(C(=O)C(C2CCC2)OC)C1 N1(C(C(C)Nc2ccccn2)=O)CCCC(C(C)NC(=O)CNC(=O)C2CC2)C1 C(=O)(CC1COc2ccccc21)OC(CN(CCC)CCOCC)C N1(C(C(C=C)O)=O)CCC2(C1)CN(C(C1(OC)CS(=O)(=O)C1)=O)CCO2 C1(NC(CCC(=C)C)=O)CN(C(c2cc(F)c(N)c(F)c2)=O)CC(C)(C)C1 c1(SCC#C)cccc(C(=O)NCC2(NC(=O)C(C)C(C)C)CCOCC2)c1 C1(NC(C2(CC=C)CCC2)=O)CCC(NC(C2CCOCC2C)=O)CC1 c1(OCC)cnncc1C(=O)N(C)CCOCCNC(=O)CNC(N)=O C1(C)(C(=O)NC(CC)CNC(c2csc(-c3ccsc3)n2)=O)CCCOC1 c1(C(=O)NC(C(C)(C)NC(CC2(OC)CC2)=O)C)ccc(N2CCOCC2)cn1 N1(C(c2cc(C)[nH]n2)=O)CC(F)CC1CN(C)C(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC1COCc2ccccc21)NC1(C)CN(C(c2cc(Cl)c(Cl)s2)=O)C1 c1(C(N2CC(NC(c3n(CC)nc(C)c3)=O)C(C)C2)=O)ccc(F)c(F)c1N N1(C(C(C2CC=CCC2)NC(=O)CSC2CC2)=O)CCCC2(CC2)C1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CCn2ccnc2C(C)C)C1 N1(C(c2c(C(C)C)ncs2)=O)CCOCC(NC(C2(n3cnnn3)CC2)=O)C1 c1(C(=O)NCC2C(NC(CN(CC)CC)=O)CCC2)ccc2cccnc2c1O Cc1cc(C(=O)NC2COCCN(Cc3ccc(Cl)nc3Cl)C2)ccc1O CCC(CC)C(C(=O)N1CCCC1C(C)(C)NC(=O)C=Cc1cnccn1)OC Cc1ccc(C)c(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)n1 C1(C2CN(C(C3CC3C(F)(F)F)=O)C2)(NC(C(c2cn(C)nc2)=O)=O)CC1 C(=O)(C1COc2ccc(F)cc21)NC1CN(C(C2(C#N)CCOCC2)=O)C1 O=C(CC1OCc2cc(Cl)ccc21)NCCNC(=O)C(c1cccc(Cl)c1)(F)F C(C(C(=O)NC(CC)C1CC1)NC(=O)C(C1(C)CCOC1)C)OCC c1(OC)ccc(C(C)=CC(=O)N(C2CCN(C(=O)C3CC3)CC23CC3)C)cc1 c1(C(=O)NCC2C(NC(=O)CC3CC3(Cl)Cl)C2)cc(C(F)F)cc(F)c1 c1(C(N)=O)ccc(C(N2CCC(N(CCO)C(C3CCCCC3O)=O)C2)=O)c(F)c1 C=CC(C)CC(=O)NCC(C1CCN(C(=O)C(C)OCCOC)CC1)O CS(=O)CCC(=O)N1CCC(CCCCCNC(=O)CCC2CCOCC2)CC1 c1(CC(=O)N(C2CCN(C(C3CC(OCC)C3)=O)C2)C)ccc(Br)c(O)c1 c1(C(=O)NC2CN(C(C(c3ccc(F)cc3)OC)=O)CC2C)ccnc(F)c1N c1(C(=O)NC(C)CNC(=O)C(C)(C)Oc2ccccc2)cccc2nc(O)oc12 C(=O)(CCC(C)(C)C)N1CCC(CN(C(=O)Cc2cnns2)C)C1 c1(CNC(c2nnnn2C2CC2)C2C(c3ccccc3)C2)cc2ncccc2o1 C1(C(=O)NCCC2ON=C(C)C2)CCCC(NC(c2ccc(CO)cn2)=O)CC1 CCC(CC(=O)N1CCC(C)(CC(=O)Nc2cncc(SC)c2)C1)OC c1(CC)nc(C)[nH]c1C(=O)NCC(F)CNC(=O)C(CCSC)OC c1(C(=O)NCc2c(C(=O)NC3CC(C)SCC3)n[nH]c2)c(C#N)ncn1C c1(C(=O)NC(C)CCNC(=O)CC2CCC(=O)N2C)cnc2c(c1)CCOC2 N1(C(CSCCC#N)=O)CCC2(CC1)CCN(C(=O)CCc1cc[nH]n1)CC2 c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)NCC2COCC2O)o1 C(=O)(C(O)CC[S+](C)C)N1C2(CN(C(C3C(C)OCCC3)=O)C2)CC1 c1(C(=O)NCC(CCNC(C(C)OC(C)(C)C)=O)O)c[nH]c2ccccc2c1=O Nc1cc(F)c(CC(N2CC3CCC(C2)N3C(C2CCCC(O)C2)=O)=O)cc1F N1(C(C23CCCN(CC2)S3(=O)=O)=O)CC(c2nn[nH]n2)Oc2ccccc21 C1(NC(C2(C(C)NC(CCCC#C)=O)CC2)=O)CC2(CNC(=O)O2)C1 c1(CC(N2CC(C3(NC(CC(C=C)(C)O)=O)CC3)C2)=O)ccc([N+](=O)[O-])cc1 C(CN(C)C(C1CN(C)CC1C)=O)(CO)(CO)NC(C(C)=C(CC)C)=O c1(C(=O)NCCCNC(CN(C(COC)=O)C)=O)oc(C)cc1C C1(NC(c2ccn(CC)n2)=O)CCCCC1NC(=O)C=CC(C)(C)C N1(C(C(C)OCCC=C)=O)CC(N(C)C(c2ccc(OC)o2)=O)C2(CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CCCCN(C(C(C(CC)C)OC)=O)C1 Cc1ccc(-n2nc(-c3ccc(C)o3)nc2C(=O)NC2CC2)cc1 c1(NC(c2ccc(-c3ccco3)o2)=O)cncc(-c2ccccc2)c1 CS(=O)(=O)c1ccc(C(O)CNCC2CC3CNCC23)cc1 C1(OC)CC(NC(c2cnn(C(F)F)c2)=O)CN(C(c2cccc[n+]2[O-])=O)C1 C1(C(=O)NCc2c(C(=O)NCCS(CC)=O)[nH]cc2)CC1C1(C)COC1 c1(NC(C2(C)CCN(Cc3cccc(Br)c3F)C2)=O)ccc(C#N)c(O)c1 CC(CCC(=O)N1CC(CC(N)=O)C1)NC(c1c[nH]cc1C1CC1)=O n1(CC(=O)N(C(C)C)CCN(C(=O)CC#N)C)cc(CN2CCC2)nn1 c1(C(=O)NC(C(C)NC(C(CSC)O)=O)CO)c(C2CC2)nn2ccccc12 C(=O)(C1=CCC(C)CC1)NCCC1CCC(NC(c2cc(CC)c(CC)o2)=O)C1 C(=O)(C(C(C)CC)NC(=O)C1=C(C)CC1)NC(CCC=C)CO c12cc(cc(Br)c1)NC2=O.CC1CCCC1COC1CC1 CS(=O)(=O)c1cncc(C(N2CC3C(C(=O)Nc4ncc(F)s4)C3C2)=O)c1 c1(OCCC(=O)NC2C(NC(CCNC(C)=O)=O)COC2)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(C)N(C(C34CCCC3C4(F)F)=O)CC2)cc2nccn2c(O)n1 C(=O)(C1=NOC(C)C1C)NCC1(CNC(C(C)c2ccsc2)=O)CC1 CC1c2ccccc2N(C(=O)CN2CCCC3(CCCNC3)C2)C1C C1(CC(=O)NCCCN(C(C=C(CCC)C)=O)CC)CC2CC2C1 N1(C(Cc2cccc(OC)n2)=O)CCN(Cc2cc(F)ccc2OC)CC1C#N C1(C(=O)NC2CN(C(COC)=O)C(C)(C)C2)CC(c2ccccc2)=NO1 CC1CC(O)CCN(C(C2CCCCN2C(c2cccc(=O)n2C)=O)=O)C1 C(C(C)(C)C(=O)NCCCC(C)NC(=O)C=CC(=O)OCCCC)OCC=C C1(F)(NC(C(C)CCN(C)C)=O)CCN(C(=O)C(=O)NCC2CC2)CC1 c1(C(C)OC)nc(C)c(C(=O)Nc2ccc(N3CCCCCC3)nc2)s1 C1(C(=O)NCC(C)(CO)NC(CC=CC)=O)CCCCC12CCC2 C1(CC=C)(NC(c2coc(Br)c2)=O)CN(C(c2cnn(Cc3cnn(C)c3)c2)=O)C1 c1(C(=O)NCC(CC)n2cccn2)c[nH]c2ccc([N+](=O)[O-])cc12 S(=O)(=O)(C1CCCC1OCC)NCCC1CC(OCC)C1 CC1(C)CC(CNC(=O)CC2CC(F)(F)C2)N(C(c2csnc2Br)=O)C1 C(c1cncn1C)=CC(N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCC1)=O N1(C(COCCCC(C)C)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CCOC)CCCCN(C(c2nonc2N)=O)C1 N1(C(C(C(C)C)c2cccnc2)=O)CC(C2(NC(=O)CC(C)C3CC3)CC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccnn3C(CC)CC)=O)CC2C1 c1(CC(=O)N(CC(C)NC(=O)CCc2cncs2)C)ccc(C#N)c(F)c1 N1(CC#C)CCC(C(N2CCC(C)C2CNC(=O)C(F)=C2CCCC2)=O)CC1 N1(C(CONC(=O)OC(C)(C)C)=O)CCC(NC(C2CCC(=O)N2)=O)C(C)(C)C1 c1(NC(C2N(C(c3ncc(C#C)cc3C)=O)CC(O)C2)=O)ccc2nccn2c1 C1(CC=C)(NC(=O)CSc2cccs2)CCCN(C(C2CC2C(N)=O)=O)C1 C(=O)(C(C)C(=O)NCc1occc1C(=O)NC1CCN(C(N)=O)C1)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)Cc2cncs2)CC1CCO Cc1cnc(NC(C)Cn2cncn2)c(S(=O)(=O)NC2CC=CCC2C)c1 C1(NNC(C2C=CC(NC(C3(CC=C)CCOC3)=O)C2)=O)CCCN(C)C1=O.C=O C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)Cn2nc(C)oc2=O)CC(C)(C)O1 n1(CCC)cc(CNC(=O)C=CCNC(c2cn(C3CC3)cn2)=O)nn1 c1(C(N(C2CN(C(C3CC(O)C3)=O)CC23CC3)C)=O)cc2ccccc2s1 Cc1ccnc2ccc(C(N3CCN(C(c4cccnc4S)=O)C4CC34)=O)cc12 C1(CNC(C=CC(C)(C)SC)=O)CCC(C(=O)NC2CCOC2C)CC1 c1(OC)ccc(C(=O)OC)cc1NC(C1CCN(Cc2c(Br)cncc2Br)C1)=O c1(C(N2C(CNC(c3cc(C)nc(O)c3)=O)COCC2)=O)cc(F)cc(C)c1C C(=O)(C=C1SCC(=O)N1C)NC1C(NC(CSC)=O)COC1 C1(C)(CC)CC(NC(c2cnoc2C2CCC2)=O)CN1C(=O)CCC(C)(C)OC C1(CCNC(c2cc(C(=O)OC)on2)=O)CN(C(C23CC2C3)=O)CCS1(=O)=O N1(C(CC)=O)CCC(NC(C2CCC3(CC2)CC3)=O)C(CO)C1 C1(C(=O)NCC2(COC)CN(C(C3(O)CCSC3)=O)C2)CSc2ccccc2O1 c1(NC(C2CC23CN(C(c2cncs2)=O)C3)=O)cc(F)c(O)cc1Cl C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)N(CCC)CCNC(c1cnc[nH]1)=O N1(C(C2C(COC)C2)=O)CCC(CNC(c2ccc(C)cn2)=O)C(C)C1 N1(C(C(CCC)(C)CC)=O)CCCC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(CC2(C)CC2F)=O)CCC(C2CN(C(=O)C3=CCCC3)C2)CC1 C(=O)(C(C)(C)C(C)O)N1CCC(N(C(Cn2c(C)cnc2)=O)C)C1 c1(CNC(=O)C(N2CCC(OC(F)F)C2)=O)ccnc(OC(F)F)c1 C1(C)(CC)CC(NC(C2(C)CC2)=O)CN1C(=O)CCc1cc(Br)cs1 CC1(CNC(C2CCS2(=O)=O)=O)CCCN(C(c2ccc3c(c2)CC3)=O)C1 c1(C(N2CC(C)C(NC(=O)CC3CCN(C)CC3)C2)=O)nnc(Cl)cc1N C=CCCCCCNC(=O)C(CO)NC(c1ccoc1CC)=O Cc1cc(C(N2CC(NC(=O)CN(C)C)C3(CC3)C2)=O)nnc1C Cc1c(N2CC(C)OC(C)C2)nc2c(F)c(Br)ccc2c1Cl Cc1cc2nc(C(N3CC(=O)NC4(CCCC4)C3)=O)cc(=O)n2o1 C(=O)(C(O)CC(N)=O)NC(C(=O)N(C(C(=O)OCC)C)C)CCF N1(C(CC(C2CC2)NC(CCC(C)SC)=O)=O)CC(CO)CC12CCC2 Cc1cc(C(N2CCC23CN(Cc2cc(O)ccc2Cl)C3)=O)cc(O)c1 N1(C(CNC(N)=O)=O)CCC(F)(F)C(CNC(=O)C=Cc2ccccc2)C1 C12(CCNC(C=CSC)=O)CCC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 N1(C(C2(COC)C=CCC2)=O)CC2(C1)CN(C(=O)C(C)Cc1ccc(C)cc1)C2 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(C)(NC(C=C(COC)C)=O)C1 C(C(C)(C)CC(=O)NC1CC(C)(NC(c2cnc(-c3ccccn3)s2)=O)C1)OC CS(=O)c1ccc(C(=O)NCC2CC2NC(=O)CN(C2CCC2)C)cc1 C1(CNC(C2C(C)C2C)=O)CC(F)CN1C(c1cnn(CCN(C)C)c1)=O c1(CC(=O)NC(CC)(C)CNC(=O)C#CC2CCC2)cc(F)c(F)cc1F N1(C(CCN(C(C)=O)C)=O)CCC(NC(=O)CC2(C)CC2)CC1C1CC1 C1(CNC(C2CN(CC)C(=O)C2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 C1(CCNC(C=C(CCC)C)=O)CN(C(=O)CCCCC)CC1C c1(CCC)n[nH]cc1C(N1CC(N(C(=O)C(C)CC2CCC2)C)C1)=O N1(C(CC2(C=C)CN(C(=O)C(CO)C(C)(C)C)C2)=O)CC(C)OCC(C)(C)C1 C(=O)(CCNC(=O)C=CC(C)(C)C)N(C1CCOC1)CC#CC CCC(C)(CC(=O)O)NCc1cc(Oc2ccccc2)cc(Cl)c1 N1(C(C2(CC)CCCC2)=O)CCN(C(C23CC(OC)C2C3)=O)C(CC(C)(C)C)C1 Cc1cc(C(N2CC(NC(c3cccc(Br)c3)=O)C(C)C2)=O)c2c(C)noc2n1 Cc1nc2cc(Cl)cc(C(N3CC(NC(C4CCOC4)=O)CC34CCC4)=O)c2[nH]1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(=O)CCS(C)=O)C2(CC2)C1 c1(C(=O)NC2CCN(C(c3c(C)cnnc3)=O)CC2)c(Cl)cccc1Br Cc1cccc2nc(C(N3CCCC3C(C)NC(=O)C(CO)C(C)(C)C)=O)cn12 CC1CCN(C(=O)CCC(=O)NCCC(N)=O)CC1NC(C12CC(CCO1)C2)=O c1(CN2C(C(N3CCCC(c4ccccc4)C3)=O)CCC2)cncc(Cl)n1 Cc1cncnc1C(=O)NC1(C)CN(C(=O)Cc2ccoc2)C1 C#CC1CCN(C(=NCCSCC)NCc2ccc(Cl)nc2C)C1 c1(C(=O)Nc2cccc(CCC)n2)[nH]c(C)c(C(=O)NC2CSC2)c1C CC(N=c1[nH]c2ccc(C#N)cc2s1)C(C1CCCCC1)NC(C1CC1(Cl)Cl)=O C1(C(N2CC(C)C2)=O)(CO)CCCN(C(C2(c3ccccc3)CCC2)=O)C1 C(=O)(C1=CCCC1)N1CCC(CNC(C2C(C)C2)=O)C1 c1(C(N2CCC(CCNC(c3c(CC)cno3)=O)C2)=O)nn(C)c(N)c1C c1(CN(C(=O)CC2CCCO2)C)cnn2c1CN(C(C1(F)CCCCC1)=O)CC2 c1(OC)ncc(C(=O)N(C2CCCN(C(=O)C(=O)NC3CC3)C2)C)nc1C c1(C(=O)NC2C(NC(c3cc(OC)ns3)=O)COCC2)noc2ncccc12 C(CN=c1[nH]c2ccccc2s1)NC(C1CC2CC2C1)=O.C1COCC1 Cc1c(NCC(C2CCC2)NC2CC2)ncnc1SC1CC1 C1(C(N(CCCN(c2ccc3nnnn3n2)C)C)=O)CCc2nnc(O)cc2C1 N1(C(C(c2ccccc2)C)=O)CCCCC1C1CCCN(C(C2(CO)CCC2)=O)C1 N1(C(CC2(C(=O)OC)CC2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccccc1)C2 CC1=CCC(C)(C(=O)NCC2CC(NC(c3cnc(C4CC4)s3)=O)CC2O)CC1 Cc1nn(CC(=O)NC2CCN(CCc3cn(CCCF)nn3)CC2)c(C)c1C CC(COc1cccc(Br)c1)N=c1[nH]c(=N)[nH]c(=NC2CC2C2(C)CCOCC2)[nH]1 C(C1CCCc2cccnc21)NC(C1CCNC12CCSCC2)=O C1(CNC(C2CN(CC)C(=O)C2)=O)CC2C=CC1CC2.C12(CCCCC1)C(=O)N2 CC(C)(C)C(CNC(=O)C1=NOCC1)C(=O)NCC1CC2C=CC1O2 C(CN=c1[nH]cncc1Cl)C1(O)CCN(C(c2cccc(C3CC3)n2)=O)CC1 C1(NC(c2n(C(C)C)cc(Br)c2)=O)CC2CC(NC(c3cn[nH]c3)=O)C2C1 c1(OC)cc(=NC(=O)C2=NN(c3ccc(N(C)CC)cc3)C(=O)C2)[nH]n1C.C(C)(C)O N1(C(C(n2ncc(C)c2)C)=O)CCC2CCN(C(=O)C(F)OC(F)(F)F)CC12 c1(C(=O)NC2CCN(C(CC3NC(=O)OC3)=O)C23CC3)cncc2cnccc12 C1(CC(=O)NCC(CC)CO)CCC(NC(=O)CNc2cccnc2)CC1 C(=O)(C1CCc2c[nH]nc21)NCC(CCOC)NC(c1cnc(O)n1C)=O C1(C(N(CCN(C(c2c[nH]c(=NCC)s2)=O)C)C)=O)CC(C)(C)OC1(C)C c1(OC)cccc(OC(C)C(=O)NCCNC(c2c(SCC)cc(OC)[nH]2)=O)c1 N1(C(c2nn(CC)c(O)c2)=O)CCCCC(CNC(=O)C(C)NC(=O)COC)C1 C12(C(=O)OC)CC1CN(C(=O)C(F)CC1CN(C(c3ccc(C(C)=O)o3)=O)C1)C2 c1(C(=O)OC)ccc(C(=O)NC2C3CN(C4CC4)CC23)cc1F N1(CCC(=O)NC2C=CCN(C(CC(CCC)O)=O)C2)CCCc2ccccc21 C1(N(C(CC(CNC(C2C=C(CO)CCC2)=O)OC)=O)C)CC(C)CC(C)C1 c1(C(=O)NC2CCC(NC(C3(CCOC)CC3)=O)C2)cc(C)ccc1OC(F)F N1(C(C2(C)CCCCC2O)=O)CCc2sc(CNC(=O)Cn3cnnn3)nc2C1 CCC(CC(=O)N1CCCC(NC(C)=O)C1)N(C(=O)Cn1cc(C)cn1)C c1(OC)cc(F)c2c(c1)CN(S(=O)(=O)C1CC=CCC1)CC2 C1(C(C)NCc2cccc(C(=O)OCC)c2)CC2(CCOCC2)CO1 c1(NC(CC(=O)NCc2cccc(Br)c2Br)c2ccccc2)cc(Br)nc(Br)c1 C1(NC(=O)COc2ccccc2)C2CC3C(C2)C13C(=O)NCc1cncnc1 CN1CCC(O)(C2(C(N3CCC(CF)(NC(=O)C4=CCCCO4)C3)=O)CC2)CC1 Cc1nn(C)cc1C(N1CCC(C(N2CCC(O)(CN(C)C)C2)=O)C1)=O c1(C(=O)NC2C(NC(CSCC=C)=O)CCCC2)cnc(C)nc1OC c1(CNC(C2N(C(C(CN(C)C)(C)C)=O)CCC2)=O)cc(F)cc([N+](=O)[O-])c1 CC1CN(C(=O)Cn2ncccc2=O)CC(CNC(=O)CNC23CC4CC2C3C4)O1 Cc1cccc([N+](=O)[O-])c1NCC1(F)CC(NC(=O)C=Cc2ccccc2F)C1 C=C(Br)CC(C)(C)C(=O)N(C)CC1CCCCN1C(=O)CSC1CC1 c1(C(=O)NCc2ccc(CCNC(C(C)C#N)=O)cc2)ccc2c(n1)CCCC2 c1(C(C2COC2)N(C(C2(c3ccnn3C)CC2)=O)CC)c(F)cncc1Br Cc1cnc(C(=O)N(C)CCOCCN(C)CCC2CCCC2(F)F)c(C)c1 c1(C(N(CCCOCCNC(CCc2cnc(C)o2)=O)C)=O)cc(CO)n(C)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cnn(C)n2)=O)CC1C Cc1ncc(CC(N2CC=CC2C(=O)NOCCF)=O)s1 C1(C(N(CCN(C(=O)CC2COCC(C)(C)O2)C)C)=O)CC(F)(F)C1(C)C C1(CC(=O)NC(CNC(C=CCC)=O)(C)CO)CSc2ccccc2NC1=O c1(C(N2CCC(F)(CNC(CCC(C)N(C)C)=O)C2)=O)ccn2ncccc12 CC1CN(C(=O)Cc2ccoc2)CCCN1C(=O)CCc1ccc(C#N)cc1 N#CCCCCCC(=O)NCC1CCN(C(C2CCCS2)=O)C1 C1(NC(c2n(CC)ccc2)=O)CCCCN(C(=O)C(C)OCCC(C)C)C1 N1(C(C2(C=C)CCCC2)=O)CCC(c2cn(C3CCCC(OC)C3)nn2)CC1C N1(C(c2c(CC)n(C)nc2)=O)CCC(C)C(CC(=O)NCCCCC(C)C)C1 C1(c2nc(SC)nn2-c2nccn2C)CCC2(CCN(C(=O)OC(C)(C)C)C2)O1 c1(C(=O)Nc2cccc(CNC(=O)NCC)c2)ncn2c1COCC2 C1(C(N(CC(C)(CO)CO)C)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 C(c1c(Cl)cccc1Cl)=C(C(=O)NC1(COC)CN(C(=O)C(O)CCSC)C1)C c1(C(C)=O)[nH]c(C)c(C(N2C3CCC2(CNC(=O)COCC(F)F)CC3)=O)c1C S(=O)(=O)(c1ccc(C#N)c(N2CC=CCC2)c1)NC1(C=C)CCC1 C1(C(N(C2C(C)CCC2)C)=O)CC2(CC2)CN1C(=O)CCc1cnc[nH]1 C1(CC)CC(CC(=O)N(C)CC2(CNC(c3ccccc3O)=O)CC2)CCO1 C1(N(C(C2CCC(CN(C)C)O2)=O)C)CCCN(C(c2ncncc2Cl)=O)C1 c1(C(=O)NCCCCC(CO)NC(=O)Cc2nc[nH]n2)cc2ccc(O)cc2[nH]1 C1(N(C(C2C(CNC(CNC(=O)OCC)=O)CC2)=O)C)CCCC1(F)F C1(NC(CC2C(CC)C2(F)F)=O)CN(C(c2c[nH]nc2OC)=O)CC12CCC2 c1(-c2cn(CC(CNC(C(C)NC=O)=O)(F)F)nn2)cccc(Cl)c1 C1(NC(Cc2cccc(C)c2)=O)CC2(C1)CC(C(=O)NC(C)(C)CN(C)C)C2 N1(C(c2ccncn2)=O)CCOCC2(C1)CN(C(C1CCOCC1)=O)CCCO2 c1(CC(N2CCN(C(CC(CC)C)=O)CC2CC)=O)ccc2c(c1)OC(F)(F)O2 C1(NC(c2ccc(F)c(Cl)c2)=O)CCc2nnc(O)n2C1.C12(CC1)C(C)N(C1CC1)C2 C1(CN(C(=O)Cc2ncc(Br)cn2)C)CCN(C(C2CC2F)=O)CC1 c1(OCC(N2CCCN(C(C(CC#C)O)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(C)(C)NS(C)(=O)=O)occc1CN(C(=O)OC)Cc1cocn1 N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)C(c2ccccc2)F)CC1CC(F)F N1(C(CCCc2cn(Cc3c(C(C)=O)cccc3)nn2)=O)CCS(=O)CC(C)C1 C(=O)(C(F)C1CCCC1)NCCN(C(=O)C(C)C1CCCC1)CC(C)O C1(OC)COc2cc(C(=O)NC3CCC(C)(C)CC3C)nn2C1 n1(CC(=O)OCC(=O)OC)[nH]cnc1=NCc1ccccc1CN=[N+]=[N-] C1(NC(CCCNC(=O)OC)=O)CS(=O)(=O)CC1NC(=O)Cc1ccon1 CC(C)C#CC(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)CC1 N1(C(c2n(C)cnc2)=O)CC(NC(=O)CC23CCCC2C3)C(C)(C)C1 CCCCCCC(=O)N(C1CCC(NC(=O)COC(C)CC)CC1)C C1(CC(=O)N(CCC#C)CCOC)(CO)CCC1 N1(CC(=O)Nc2ccc(CCC)cc2)CC2CCC(F)(C2)C1 CC1=C(C(=O)NC2C=CCN(C(=O)COc3cc(F)cc(F)c3)C2)CCCC1 C1(O)(CC(=O)NCC(CN(C(CCn2c(C)csc2=O)=O)C)O)CCCCCC1 CCC(C#N)C(=O)N(CCCN(C(=O)CCc1ccc(Cl)s1)C)C N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)Cc2csc(N(C)C)n2)C(C)C1 N1(Cc2cc(OC)c(O)cc2)CCCC2(CCN(C(C3CCC(O)CC3)=O)C2)C1 N1(C(C(C(=C)C)(C)C)=O)CCC2(CCC(CNC(=O)C(C)(C)C(N)=O)CC2)CC1 C(=O)(C(C)(C)C(C)NC(=O)CC1(O)CCC1)NCCC1C(C)C1 N1(C(c2c(C)onc2C(F)(F)F)=O)CCCCC(CNC(C2CCNC2=O)=O)C1 c1(OCC)cc(F)ccc1NC(C1OCCC1NC(=O)Cn1ncn(C)c1=O)=O C1(NC(c2c(C)nc(C(C)OC)s2)=O)CN(C(=O)C=CSC)C(C)(C)C1 c1(CN2CCCC(C(=O)NCCNCCO)C2)cc2ccoc2cn1 C1(C(C)O)CN(C(=O)CN(C)C(C2CC23CC3)=O)CCO1 Cc1ccc(SCC(N2CCC(NC(c3[nH]ccc3C)=O)C2)=O)cc1 C1(NC(C(CC=C)C)=O)C2COCC1CN(C(c1cc(C)[nH]n1)=O)C2 C12(CC(=O)NCC(C)CNC(=O)C(C)n3ccnn3)CCCN1CCC2 c1(CNCCOCCC(C)CO)ncccc1O C#CCC(C(=O)NOCc1ccccc1)NC(=O)COCC=C c1(C(=O)NC2C(CNC(c3c(CC)onc3)=O)C2)cc(Cl)cc(C)c1C CC(CCNC(=O)CCOC1CN(C(C2CCCCO2)=O)C1)C(C)(C)C N(C(=NCC=CC1CC1)NCc1ccco1)CC1(C)CCCO1 c1(OC)ccc(CC(=O)NC2CCN(C(c3cccnc3N)=O)CC2F)c(F)c1 C(=O)(C1CNC(=O)NC1)OC(C)(C)C.c1(C2CC(F)(SC)C2)ccccc1 Cc1ncc(C(=O)N(C2CN(C(=O)CCNC(=O)CO)CC2(C)C)C)cc1C#N CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1COC2)C1CCOCC1 Cc1[nH]nc2c1CC(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC2 Cn1ccc(C(=O)NCC2CCC(N(C(=O)C=C3CCSCC3)C)CC2)cc1=O N1(C(CSCC#C)=O)CCN(CC(=O)NCC2CC(CCC)C2)CC1 c1(OC)cccc(C(c2nnnn2C(C)(C)C)NC2(C)CCOC2)c1 N1(c2cc(NC)[nH]c(=N)n2)CCC2CC(C(=O)NCCCCCCO)C2C1 c1(CNC(C(C2CC2)OCC)=O)cncc(C(=O)NC2CC(=O)N(C)C2)c1 C(C)(C)(C(N)=O)NC(C=CC(C)NC(=O)CC1CC1(C)C)=O c1(C(N2CCN(CC(O)C3CC3)CC2)C(=O)NCC(C)C)ccnc(Cl)c1Br [N-]=[N+]=NCCCC(=O)NC1CCCCCC1NC(=O)Cn1cc(Cl)cn1 C1(NC(CC(CC)SC)=O)CCC2(CCN(C(c3ccnc(Cl)c3N)=O)CC2)C1 C(=O)(C1=NOC(C)C1C)NC(CCC(=O)NCC(CCOC)O)(C)C c1(C(=O)NC2(CCO)CN(C(=O)CC3CCOC3)C2)cccc2sncc12 Cc1scc(C(=O)NC2C3CC2N(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1C Cc1cc(C(N2CCC(N(CCO)C(c3occc3C)=O)C2)=O)ccc1C1CC1 C(=O)(C(C)COCCOC)NCCC(=O)OC.C12CCC1NC(=O)CSC2 c1(C(C2CC2)NC(CC=CCC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)F)NC1(CC(=O)NC(CCC)CO)CCCCC1 N12CC(F)(F)CC1C2=O.c1(NC(c2ccc(COC)cc2)=O)nnc(Cl)cc1Br c1(C(N(C2CCN(C(C(CSC)O)=O)CC2)CCO)=O)cnc2cccnc2c1 C1(COCC)CC2(CC2)CN1C(c1cc(I)ccc1Cl)=O.C12N(CC1(C)C)C2=O N1(C(c2c(C)scc2)=O)CC2(CCN(C(c3ccc(O)cc3Cl)=O)C2)C1 N1(C(c2c(C)onc2C2CC2)=O)C2CCC1CN(C(c1ccncc1F)=O)CC2 N1(C(C(=O)NCCC2CC2)C2CCCC2)CCCCC(C2CCOCC2)C1 C1(COC)(NC(=O)NCCCN(C(=O)CC2CC2C)C)CCCCC1 c1(CC=O)cccc2c1OCCO2.N12CCCN1C(CO)C2.C=CCCC=O N1(C(C(C2CCCC2)NC(CNC(C)=O)=O)=O)CC2(CCNC(=O)O2)C1 S(=O)(=O)(c1cncc(Br)c1)NCC(=O)OCC(c1ccc(C(F)(F)F)cc1)=O C1(C(=O)OC)CCN(C(=O)Nc2cccc(C3SCCS3)c2)C2(CC2)C1 C1(CC(=O)N(CC(=O)NCCCc2cnccn2)CCC)C(=O)NN=C1C C=CCC(F)(F)C(=O)N1CC(NC(=O)Cn2ccccc2=O)CC(C)C1 N1(C(Cc2c(C)con2)=O)CC2CCN(C(C3CC(C)(C)OC3(C)C)=O)CC2C1 Cc1nc2ccc(C(=O)NC(C)CC3CCN(C(C4CC4CF)=O)CC3)cc2[nH]1 C1(C(N2CCC(CN(C(=O)C=C3CCC3)C)CC2)=O)CC2(C1)CC(F)C2 N1(C(c2cc(C)c(-n3cncn3)cc2)=O)CCC(CNC(=O)CNC=O)C(F)(F)C1 c1(C(N(CC(C)NC(C2CC(n3cnnc3)C2)=O)C)=O)cc(C#N)on1 CCCCC(CNC(=O)CCC1CCC(=O)N1)NC(=O)CSCCOC C1(CNC(CCN(C)CC)=O)CC2CN(C(C3C=CC=CC=C3)=O)CC12 c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)ccnc(C(C)(F)F)c1 c1(CC(=O)NC2C(C)(CN(C(C(C)=C(C)C)=O)C)CCC2)cnn2c1CCCC2 Clc1cc(-n2nc(C3CCC3)nc2-c2cn[nH]c2)cc(Cl)c1Cl O(NC(=O)C(C)C(C)NC(=O)C(C)(C)O)C(COC)COC CC1CCN(C(c2ncoc2C(F)(F)F)=O)C(C)C1NC(=O)C=Cc1nccs1 CCC(O)(C(=O)N(C(CNC(c1ccc(C)nc1)=O)C1CC1)C)c1ccccc1 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CN(C(C(c1ccccc1F)(C)OC)=O)C)O CCCCCCC(=O)NCCC1COCCN1C(=O)C=CI c1(CC(N2CC(CCNC(c3nc(OCC)oc3)=O)C2)=O)ccc(C(N)=O)nc1 C1(C(N2CC(OCC)(CNC(c3coc(O)n3)=O)C2)=O)C2CCC(C2)C1(C)C C1(NC(c2ccc(C)cn2)=O)CC(CNC(=O)Cc2cc(C)[nH]n2)C12CCC2 C1(CC(=O)Nc2cnc(C)s2)CCCCN1C(c1ccccc1-c1nn[nH]n1)=O C(=O)(C(C)(F)C(=O)NC1CC1NC(=O)CS(=O)(=O)Cc1cccs1)OCC C1(C(C2(C(C)(C)O)CC2)C)CCCCC1NC(=O)CC1(CNCC2CC2)CC1 C(c1cnccn1)=CC(=O)N(C1CCC(NC(C2(SC)CCC2)=O)C1)C C1(C(=O)OC)CCCN(C(=O)NCC2(Nc3ccccc3)CCN(C)C2)CC1 c1(C(N2CCC(C)C(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2)=O)c(N)cc(F)cc1F C(=O)(C1(C)CCCc2ccccc21)NC1C(NC(c2c(C)ccc(F)c2N)=O)C1 N(C1CCc2sc(Cl)cc21)C(c1c(C)n(-c2cnn(C)c2)nn1)=O C1(C(=O)NC(C(O)CO)C2CC2)CN(C(C2(O)CCCCC2)=O)CC12CCC2 C=CCCN=C(NCCC1CN(C(C)C)C1)N1CCC(CC)C1 S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCC3)C2)cn1)NC C1(N(C)C(c2cc(C(F)F)no2)=O)CN(C(c2cc(O)nn2C)=O)CC1(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)NC1C(CC(=O)OC)CC1 Cc1c(C(=O)NCC2CCC2NC(C2CCNC2=O)=O)sc2[nH]cnc(=S)c12 C1(NC(CCCCCCSC)=O)CC2CCCC(C1)N2C(c1ncncc1F)=O c1(C(N(C(C)CNC(c2ccc(CC(N)=O)cc2)=O)CC)=O)cnc(=N)[nH]c1 CCCC(C)CCN=c1cc[nH]cc1S(=O)Cc1ccc(C(C)(C)C)cc1 n1(CCC(=O)NCC2(COC)CCCNC2)cc[nH]c(=O)c1=O C1(C(=O)NCC=CCOCC)(NC(=O)C=CC(C)C)CC(F)C1 c1(NC(C(CC2CCC2)NC(C(CCCOC)C)=O)=O)cccc([N+](=O)[O-])c1 n1(C(CC)C)ccc(=NC2(CF)CCCOCC2)[nH]1.c1(CSC)nnnn1CCC CC(C)C(C(=O)NCCNC(C1CSCCS1)=O)S(=O)(=O)C1CCCCC1 O=C(CC1OCCc2ccsc21)NCC1(CNC(c2ncc(C(F)F)s2)=O)CC1 C(c1ccncc1C)=CC(=O)N(C)CC1(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CC=C)cccc2)=O)CC2CCCC(C1)N2C(C1CC(C)(C)CO1)=O CCCCCCC(C)C(=O)NC1(C)CCN(C(c2cnc(O)cc2OC)=O)CC1 C1(C(=O)NC2CC(CCNC(CCc3n(C)ncc3)=O)C2)CCc2nnnn2C1 C(CN=c1[nH]cnc2c1COC2)N(C(C1C(CC)OCC1)=O)CC S(=O)(=O)(CC(=O)NCC1(F)CC(CNC(=O)C(c2cccc(F)c2)C)C1)NC C1(CNC(CC2CC(C)C2)=O)CCC(N(C)C(c2sccc2C(C)(C)C)=O)CC1 C1(=CC(=O)N(CCC(C)(C)NC(Cc2cc(C)on2)=O)C)CCN(C)CC1 N1(C(CCNC(c2cn(CC=C)nn2)=O)=O)CCCC(CO)C1 c1(C(N2CC(C)(NC(C(CSC)C)=O)C2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)NCC(C(=O)NC(CN(CCC)CC)C)N(C)C)cc[nH]c(=NC)c1 c1(NC(C2N(C(Cc3n(C)ccc3)=O)C3C(C2)C3)=O)cc2c(cc1Br)OCCO2 Cc1cnc(Cl)[nH]c1=NC1CC2CN(C(=O)C(C)C(C)C)CC12 CN=S(C)(=O)c1ccc(C(N2CC(CNC(=O)COC(C)=O)C(O)C2)=O)cc1 N1(C(C2CC(CC)C2)C(=O)NCCC#N)CCC(C)(O)C(C)(O)C1 Cc1cc(C)c(C(N2CC(O)CC2C(=O)NCC2CCOC2C)=O)s1 C(C(CC(=O)NCCC1CC=CCC1)NC(c1cn(C)cc1C)=O)OC C(=O)(C=C1SCC(=O)N1C)N(C1CCN(C(=O)C2=NNC(=O)CC2)CC1)CC#C c1(C(N2CC3(CC(NC(C(C(C)C)(C)C)=O)C3)C2)=O)sc([N+](=O)[O-])cc1Cl C=CCC(C(=O)N1CCC(C)(NC(c2cc(C(=O)C(C)C)c[nH]2)=O)C1)NC(C)=O Cc1nc2ncnn2cc1C(N1CC2CC(NC(=O)Cc3cccnc3)C1C2)=O c1(N2CCC(COC)C2)nc(N2CCN(C)C(=O)C2)c2ccccc2n1 c1(C(=O)NCC(C)CNC(=O)CN2CCOCC2=O)sccc1S(N)(=O)=O n1(CC)ncc(C(N2CC(NC(=O)COC3CCCCC3)C(CO)C2)=O)c1C N1(C(c2n(C)c(-c3ccc(F)cc3)cc2)=O)CCc2ccc(F)c(Br)c2C1 Cc1cc(Br)c2c(c1)CN(C(C1C3CCOCC13)=O)CC2 c1(C(=O)NC2CCN(C(C(CO)N(C)C)=O)C2)cc(C(F)(F)F)ncn1 C#CCCCCCC(=O)NCC(=O)N.C(C(C)C(C)(C)C)CNC(COC)=O n1(CC#C)c(C)cc(C(=O)NC2CCC(NC(c3ccc(F)c(O)c3)=O)C2)c1C Cc1c(Br)ccc(S(=O)(=O)N2CCCN(CCS(C)(=O)=O)CC2)c1F c1(C(=O)NCCN(C(C=C(C)C)=O)CC(C)O)cn2c(Br)c(C)nc2s1 Cc1ccc(I)c(NC(C2CN(C(=O)Cc3cccc(C(F)(F)F)n3)CCN2)=O)c1 c1(C(N(C)C[Si](C)(C)C)C(=O)NC(C)C)cc2cc(F)ccc2o1 Cc1nc(N2CCC(C)C(NC(=O)CCOc3ccccc3C)C2)c(C)c(Cl)n1 C1(CNC(C(C)NC=O)=O)N(C(=O)C(=O)C(C)(C)C)CCC1(C)C Cc1cccc(CC(=O)NCC2CC(F)CN2C(=O)CC2(C)CCCCC2)c1F c1(C(=O)NCC(n2cc(C3(O)CCOC3)nn2)C)cnnc(Cl)c1 C1(CC(=O)NCc2n(C)ncc2)CCCCN1C(=O)CCn1cccn1 C(=O)(C(CC)(CC)OC)N1C(CN(C(C=CCN(C)CC)=O)C)CCC1 C1(NC(C2(COC)CC(=O)C2)=O)CCN(C(=O)C(Cl)=CCl)CC1C c1(C(C(=O)NCC2C(NC(C(C)(C)OC)=O)CCC2)OC)ccc(OC)cc1 c1(C(=O)NCC(CN(C(CCOCC)=O)C)(C)C)cnc2ccoc2c1 C1(NC(c2c(C)ccn2C)=O)CC2(CCC(NC(C3CC4CCC3C4)=O)CC2)C1 c1(NC(C2CC(NC(CC=C)=O)C(O)C2)=O)cccc2c1CCC2 C1(NC(CCC=C)=O)CC(OC)CN(C(c2c(C(F)(F)Cl)n[nH]c2C)=O)C1 C1(NC(C2CN(C(C(=O)Nc3cccc(C)c3)=O)C2)=O)CC2(C1)CC2(F)F C1(NC(CC(CC)O)=O)CN(C(=O)COC(C)CC)CCC1C(F)(F)F CCCC(C(=O)NOCC(=O)OC)NC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CC2)cc(Cl)sc1Cl c1(OCC(=O)N(C2CC(NC(c3cc(O)ncn3)=O)C2)C)ccc(Br)cn1 c1(C(N2CCOCC(NC(CC=C)=O)C2)=O)c(C)nc(C(C)C)nc1O N1(C(CC2(C#N)CC2)=O)CCN(CCNC(C2CC(n3ccnn3)C2)=O)CC1 Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]n3)=O)C2)=O)cc([N+](=O)[O-])c1Cl Cc1ccnc(C(=O)NC(CNC(=O)COC2CCCCC2)CC(C)C)n1 C(CNC(c1cc(Br)sc1C)=O)(C(C)(C)C)NC(CNC(=O)OC)=O c1(C(N(C2CCCN(C(C3C(=C)C3)=O)C2)C)=O)cc2c(F)cc(F)cc2o1 C1(NC(C=CCNC(C(C)(C)OC)=O)=O)CCCSCC1 c1(C(=O)NCC(CC(C)C)NC(C2(CC)CCNC2=O)=O)c[nH]cc(F)c1=O N1(C(CCCCCC#C)=O)CC(CNC(=O)C(=O)NCC)CC12CCOCC2 C(=O)(C(O)CCC(F)(F)F)N1CCC(CN(C)C(C2CC3(CCO2)CC3)=O)C1 C(CCCC(C)NC(=O)Cn1nnnc1C(C)C)NC(C1(SC)CC1)=O C(=O)(C(C(=O)NCc1ccc(C(=O)NCC(C)(C)N(C)C)s1)OC)OCC Cc1cn2c(C(=O)NC(C3CCN(C(C4CCC(=O)C(C)C4)=O)C3)C)cnc2s1 N=c1nc2c(c[nH]1)CC(C(N1CCCN(C(c3ccsc3)=O)CC1CO)=O)CC2 N1(C(C)C)C(=O)CCC1C(=O)NCC(C)(C)NC(C1CC1c1ccc(Cl)nc1)=O c1(CC(=O)NCCN(CCCN(C)C)C(C2C(C=C)C2)=O)ccccc1O C(=O)(C#CC(C)(C)CNC(=O)CC1CCCSC1)NCc1c(C)nccn1 c1(C(=O)NCC(CCCC(=O)OC(C)(C)C)=O)cc2n(n1)CCCNC2=O c1(OC)ccc(O)c(C(=O)N(C)CCNC(C2(CF)CC2(F)F)=O)c1 C1(C#N)(C(=O)NC(C2CCN(C(C3CC(=O)NC(=O)C3)=O)C2)C)CC2C=CC1C2 N1(C(C2(C)CC2F)=O)CCN(Cc2nc[nH]n2)CC1 c1(C(N2CC(NC(c3cnnc(C4CC4)c3)=O)C(O)C2)=O)ncc(Cl)cc1F N1(CC(=O)NC2C(NC(C3C(C=C)CC3)=O)CCC2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(F)c(F)c1F)N1CC(NC(C2CCC(OC)CC2)=O)C1 C1(C(C)NC(N2CCC(COC(C)(C)C)CC2)=O)CCCC(CN)O1 CC1CCCC(NC(=O)COCC2CCCN(C(c3cnoc3C3CC3)=O)C2)C1 C1(C)(CC(=O)OC)CCCN1C(=O)NCc1ccccc1-c1cn[nH]c1 S(=O)(=O)(c1ccc(Cl)cc1C(F)F)NC(c1ccc(Cl)c(F)c1)C c1(C(c2n(C(CC)C)nnn2)NCCOC(=N)O)cc(F)c(Cl)cc1F N1(C(C(C(C)C)c2cccs2)=O)CC2(CCN2C(N)=O)C1 CC1(C)C=CC(NC(c2cc(CNC(=O)CCN3CCCCC3)cs2)=O)CC1 N1(C(C2(OC)CCOC2)=O)CC2CC(C1)N2C(=O)C(O)CSC C(=O)(C1CCCn2cnnc21)NC(CNC(Cn1ncc(C#C)c1)=O)C1CC1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2(CCCC2C(=O)NCCNC(C)=O)C1 CCC(CC(F)(F)F)C(=O)NCCC1CN(C(=O)CC2CC3(CC3)C2)CC(C)O1 C1(N(C(=O)CCC2CCCN(C)C2)C)CC2CCC(C1)N2CC1CCOC1 CC1OC(C)CC1C(N1CCN(CCc2cn(CC3CCCOC3)nn2)CC1)=O CCS(=O)(=O)CC(=O)N1CCCCC(N(C(=O)C(C)NC(c2ccco2)=O)C)C1 C1(CNC(CC(CCC)O)=O)CN(C(=O)C=CC=C(Cl)Cl)CC2(CCC2)O1 N#CC1(CC2CCN(c3cccc(OCc4ccccc4)c3)C2)CCOCC1 c1(C(N(CC(CC)NC(c2ccncc2)=O)CC)=O)ccnn1C1CCCCC1 C=CC(CCC)CC(=O)N1CCN(C(=O)CC(O)CC(C)C)C(C)C1 N1(C(CNC(CC)=O)=O)CCC(CNC(c2ccc(Br)cc2O)=O)C1(C)C CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)COCCSC)CC1 N1(C(C(C2CCCO2)NC(CC(=O)NCC#C)=O)=O)CCC(C)(C(=O)OC)C1 N1(c2n(CCOCC=C)c(C(C3CCCO3)C)nn2)CCC2(CC1)CC2(F)F c1(CCNC(C2C(C)CCCC2)=O)cn2c(n1)CCCC2 N1(C(C2(CC=C)CCCNC2)=O)CCN(Cc2ccc(Cl)cc2)CC(O)C1 C(=O)(CCC(C)(C)F)NC1CCCC(N(C(CNC(c2c(C)occ2)=O)=O)C)C1 C1(CNC(=O)NCC(CC(=O)OC)c2ccc(Br)cc2)CC(F)(F)CCN1 CC1CCCC(C(N2CCC(C3CCCN3C(=O)CC3CCCC3)C2)=O)CC1 c1(C(N2C(C(C)NC(CN3C(C)CCC3)=O)CCC2)=O)cccc(O)c1Cl c1(CNC(CCNC(=O)OC)=O)n[nH]cc1C(C)C c1(C(N2C3CC(NC(C(C)Cc4ccco4)=O)C2CC3)=O)sccc1S(N)(=O)=O C=CC1(CC(=O)NC2CCN(C(C)=O)C2C)CN(C(=O)COC)C1 c1(-c2c(SC)cc(F)cc2)ccc2c(O)c(C(=O)NC(CO)CC(C)C)sc2c1 C#Cc1cc(C(=O)NC(CNC(=O)C(CC(C)C)OC)C2CCC2)cc(N)c1 c1(C2(C(=O)NCC34N(C(C(C)O)=O)CC(C3)C4)CCC2)ccc(S(N)(=O)=O)cc1 c1(CC(=O)N(C2CCCCC2)CCCNC(CCOC)=O)sc(C)cc1C C1(CC(=O)NCCN(C(=O)CCCc2cnccn2)CC2CC2)COC(=O)N1 C1(C(=O)NC2CC2N(C)C)(CC)CCCN(C(=O)C=CSC)C1 C1(C(=O)OCC)CC2(C1)CN(CCCC1CC(C(C)(C)C)C1)C2 C#CC1CCN(C(C2CC(NC(c3ccc(CO)s3)=O)CCO2)=O)C1 C=CCCC(O)CNC(C1(CO)CCN(C(=O)CC2CCC(C)CC2)C1)=O c1(CC(C)C(=O)NCC2(NC(C3CC3F)=O)CCC2)ccc(F)cc1 c1(OC)ccc(OC(=O)NC(C)(C)C)c(NS(=O)(=O)C2CN(C(C)=O)C2)c1 N1(C(C(CCC)NC(=O)Cn2ccc(C)n2)=O)CC2(CC(N(C)C)C2)C1 C1(NC(C=CC(C)(C)C)=O)CN(C(c2ccc(C(O)CF)cc2)=O)CC1(C)C c1(NCC2CC(NC(C3(C(C)C)C(C(=O)OC)C3)=O)C2)ncc(OC)nc1OC N1(C(C(=O)NCCOC)=O)CCC(CO)C(NC(c2oc(Br)nc2C)=O)C1 CC(CC(C)(C)C)C(F)C(=O)N1CC(CCNC(=O)C=Cc2cocn2)C1 Cc1ccc(Cl)c(N=c2scc(-c3cc(C)n(C)n3)n2CCSCC(C)C)c1Cl c1(CC(=O)NCC2CCN(C(CC3CCC(=O)NC3)=O)C2)ccc(O)c(F)c1 c1(C(N2CCC(OCCCF)CC2)C(=O)NCC(F)F)ccc(C2CC2)cc1 C(=O)(C1=Cc2ccccc2C1)N1CC2C(C(N3CCC(CCC)C3)=O)C2C1 C(CC(C(N)=O)OC)OC(C(NOCC(=O)NC)=O)C1CCC1.C c1(C(=O)NC2C(NC(c3nc(C)[nH]n3)=O)CCOC2)ccc(Br)c(C)c1 C(=O)(CCC(C(C)C)NC(=O)C(C)(Cl)Cl)NCC(C(=O)NC)(C)C O=C1NC(=O)C(CNC(=O)CC2(NC(C3CC(=C4CCC4)C3)=O)CC2)N1 N1(C(COC(C)C)=O)CCC2CN(C(c3ccc(N)c(Cl)c3)=O)C2C1 C(=O)(C(F)C(=O)N1CCSCC1C(=O)Nn1cncn1)OCC C(=O)(C(CC)CCCCC)N1CCN(C(CC(=C)Br)=O)CC1CO CN1CCCC(C(=O)NC2CCC(Cn3cc(CCCO)nn3)CC2)C1.C1CO1 N1(C(CCc2c(C)noc2Cl)=O)CCCC2(NC(c3cc(C)n(C)c3)=O)CC2C1 Cc1cc(C(=O)NCc2cc(C(=O)NCCCC(=O)NO)no2)ccc1C#N C12(NC(=O)C=CC(F)(F)F)CCCC1CN(C(c1cccc3[nH]ccc13)=O)C2 N1(C(CNC=O)=O)CCC2CN(C(c3ccoc3C3CC3)=O)CC12 c1(OC)ccnc(C(N2CC(NC(C3CCCCO3)=O)CCC2C)=O)c1N CC1=C(C)CC(C)(C(=O)NCCC2CSCCN2C(=O)COC2CCCC2)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CCN(C(=O)Cc3ncccn3)CC12 C1(NC(=O)CCC2CCCOC2)CN(C(c2ccco2)=O)CC1(F)F N1(C(CC(COC)C)=O)CCC(NC(c2ccc(C)cn2)=O)CC1C C1(NC(CC=CC)=O)CCC(C(=O)NCCN2CCC(O)CC2)CC1 CC(C)(F)CC(=O)N1CCC(CCNC(=O)Cn2ccccc2=O)C1 C(=O)(C1CCCn2cnnc21)N1CCC2CN(C(=O)Cc3sc(O)nc3O)CC21 C1(C(N2CCC3CN(C(c4c(C#N)csc4)=O)CC32)=O)CS(=O)(=O)CC12CCC2 N1(C(c2ccc(N(C)C)cc2)=O)CC2(CC(NC(=O)CCOC3COC3)CO2)C1 c1(C(C(=O)NCCCNC(c2c(COC)onc2)=O)C)ccc(Cl)c(Cl)c1 O=C(CC(C(F)F)NC(C1CC12CCCC2)=O)NC12CCN(CC1)CC2 Cc1c(C(=O)NCC2(NC(c3ccsn3)=O)CC2)cnc2c(Cl)cccc12 CC1(C)CN(C(=O)C=CC2CCC2)C(CNC(C2CC2(F)F)=O)CO1 c1(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)nnc(O)cc1O Cc1[nH]nc(C(=O)N(C)CCC2CCN(C(C3CC(F)C3)=O)CC2)c1C Nc1c(C(N2CCC(NC(C3CCc4nccn4C3)=O)C2)=O)nc(O)nc1O N1(C(c2cc(CC)nn2C)=O)CC2CC(C1)N(C(C1CC(C)CC(=O)N1)=O)C2 C(=O)(C(C)C(C)NC(=O)CCOC1CCC1)NC(CC#C)C N1(C(C(=O)Nc2cccc(C)c2NS(C)(=O)=O)=O)CCc2ccncc2C1C C1(CCNC(c2n[nH]c(C)c2O)=O)CN(CCOCC(C)C)CCS1(=O)=O c1(N(C(=O)NC(C(C)C)C)CC2CC(=O)N(C)C2=O)c(Br)c2ccccc2n1C C1(CC=C)(C(N2C(C)(C(=O)OC)C=CC2)=O)CCN(C(=O)COCCCOC)C1 c1(CCC(=O)NC2CN(C(c3nc(C)sc3)=O)C3C2C3)c[nH]c2cccc(C)c12 N1(C(CC2N(C(C)=O)CCC2)=O)CCC(C2(NC(c3sncc3C)=O)CC2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(CNC(c2ccc(C)o2)=O)CC(C)(C)C1 C1(CC(=O)N(C(C#C)C)CC)(NC(=O)CCNC(N)=O)CCC1 N1(C(C(C)(C)OC)=O)CCCC(O)(CCNC(=O)C(C2CCOCC2)O)C1 CCS(=O)(=O)C=CC(=O)N1CC(CC(C)NC(c2csc3ccccc23)=O)C1 c1(Cn2cc(N(CCO)CC3CCCSC3)nn2)ccc2c(c1)OCO2 C(=O)(C(O)Cn1cncn1)NC1CC(OCC(=O)N(C)Cc2ccoc2)C1 C(CC(C(C)C)NC(=O)C(C)NC(=O)C1CC1)N(C(c1c(OC)ccs1)=O)C C1(C(N2CC(CCNC(=O)CN(C)S(N)(=O)=O)(OC)C2)=O)CCN(C)C1=O N1(C(C2C(C)(C)CC2)=O)CCOCC2(COCCN2C(c2snc(Cl)c2Cl)=O)C1 c1(OCC)c(NC(=O)CCCCN2CCOCC2)cccc1Cl C1(C(N(C2CC(O)C2)C)=O)CCC(O)CN1C(C12CSCC1C2)=O c1(C(=O)OC)scc(-c2ccc(C)cc2)c1NC(=O)Cc1cc(C)no1 c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cnc(C(F)(F)F)cn1 c1(C(N2CC(NC(C3N(CCC(C)C)CCC3)=O)C2)=O)cnccc1C(C)(C)C c1(C(C)C(=O)NC2CC(NC(c3c[nH]cc3Br)=O)C2)ccc([N+](=O)[O-])cc1F Cc1nc(=NNC(=O)c2c[nH]c(C(F)(F)F)c2)s[nH]1 Nc1cc(C(N2CCCC(NC(C34CCCN(CC3)C4)=O)CC2)=O)ncc1F c1(C(=O)NC2(CCNC(C(C3CCCC3)OCC)=O)CC2)ccc(O)c(C)c1C C(CCCC(=O)NCC1CN(C(=O)C(=O)NCC(F)(F)F)C2CC12)SC N1(C(CCCN(C(C)C)C)=O)CCCC2(C1)CN(C(=O)CCS(C)=O)CCO2 N=c1[nH]cncc1C(=O)NCC12CC1CN(C(c1cnccn1)=O)C2 C1(O)(CNC(CCN(C(C)=O)C)=O)CCCN(C(C2CC2(C)C(F)(F)F)=O)CC1 N1(C(c2n(C=C)nnc2)=O)CCC2(C=C(C(=O)N3CC(=O)NCC3C(N)=O)C2)C1 N1(C(C(C#C)(C)C)=O)CC2CCC1C1CN(C(c3cccc(N)c3F)=O)CC21 c1(NC2C=CCCCC2)nc2c(c(=NCc3nc4cccnc4[nH]3)[nH]1)CSC2 C1(C)(C(=O)NC23CN(C(C(C)C4CC4)=O)C(C2)C3)Oc2ccccc2NC1=O c1(OCCC(C)(c2nnnn2C2CCOC2)NCCC(N)=O)ccc(F)cc1 C12(NC(CNC(CCC)=O)=O)CCC(CNC(c3cnsc3)=O)(C1)OC2 c1(OC)c(F)ccc(F)c1C(N1C2CN(c3nccc(Br)n3)CC12)=O c1(CC(C(=O)N(CCC(C)NC(c2c(CC)cno2)=O)C)C)ccccc1C C(C(C(C)C(C)C)NC(=O)CCc1nc[nH]n1)NC(C(c1ccc(CC)s1)=O)=O Cc1[nH]nc2ncc(C(=O)N(C3CCCC3)CCCNC(=O)C(C)(C)F)cc12 c1(C(N2C(CNC(C3C(C)OCCO3)=O)CC(F)C2)=O)ccc(N)c(N)n1 CCC(C)C(=O)C(=O)NC(C1CCOC1)CNC(C1CC=CC1)=O c1(-c2ccc(CC)nc2)cccc2ccc(C(=O)Nc3cnc(Cl)cc3Cl)nc12 C1(CNC(=O)C=CC2CCC2)CC(N=c2nc(C3CCOCC3)[nH]s2)CCO1 C1(CCC(=O)NCC(C)(CO)NC(=O)Cc2csc(Cl)c2)NC(=O)NC1=O C1(C(=O)NC(c2ccccc2)CC=C)CN(C(C)=O)CCO1 C1(NC(c2c(C)n(CC(F)F)nc2)=O)CCN(C(C2OC(C)CC2C)=O)CC1C CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(=O)CC1C(C)(C)C1(C)C C1(COC)(CNC(C2CSCCS2)=O)CCN(C(=O)C(C)(O)COC)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CC(NC(c2csc([N+](=O)[O-])c2)=O)C(O)C1 N1(C(C(CCC)C)=O)CC2CCC1CN2C(c1nc(-c2ccc(Cl)cc2)no1)C C1(C(=O)NC2(CCCNC(c3ccc(C(F)F)o3)=O)CC2)CCCCS1 C#C[Si](C)(C)CCCNC(=O)NCC1CC1C1CCCC1 N1(CC)CCOC(C(=O)N(CC)CC2CCS2(=O)=O)C1 C1(C(=O)NC(C2CN(Cc3csc(-c4ccccc4)n3)C2)C)CN2CCN1CC2 C1(C(=O)NC2(C)CC(C(=O)NC(c3cncnc3)C)C2)CN(C)CCN1C CC1CC(CC(=O)NCc2nc[nH]n2)CN1C(c1csc(C#N)c1)=O c1(C(C(=O)NCCCN(C(CC(C)F)=O)C)O)ccc(F)cc1Br Cc1c(Br)ccc(C(=O)NCC(C)(CO)NC(C2CCCOC2C)=O)c1F c1(NC(C2CCCCN2C(c2cncc(Cl)c2)=O)=O)cccc(F)c1F N1(C(c2cc(C)c(C)nn2)=O)CCN(C(=O)CCc2nccs2)CC(C)(C)C1 CC(CS(N)(=O)=O)NC(=O)C(C1CC1)NC(=O)C=Cc1cc[nH]c1 N(C(=NCC(C)SC)N1CCC(CF)C1)CC(=O)NC(C)C C1(NC(C(CC)OCC)=O)CC2CC(C1)N(C(=O)C(C#N)=CC1CC1)C2 N1(c2nnc(C)s2)CC2CCC1C(NC(=O)CC1CCCS1(=O)=O)C2 CCCCC(C)C(=O)N1CC2C(N(C)C(C3CC4CCC(C3)S4)=O)C2C1 c1(C(N2C(C)CCC(NC(C3CCSC3)=O)C2)=O)nnc2c(F)cccc2c1O C1(N(C(C2(COC(C)C)CC2)=O)C)CCC(NC(C2CN3CCC2C3)=O)CC1 C(CCCCNC(=O)C(n1ccc(C(F)(F)F)n1)C)NC(C(C)OCC(C)C)=O O(NC(=O)CC(C)CNC(=O)C=Cc1cnn(C)c1)C(C1CCCCC1)C c1(C(N2CCCC(c3ccn(C)n3)C2)C(=O)NCC)cc(F)nc(F)c1F c1(C(=O)NC(CCN(C(C(C(C)C)N(C)C)=O)C)C)cccc2nncn12 c1(C(=O)NCC2CC(NC(C(C)c3ccsn3)=O)C2)ccccc1-n1cccn1 C(C(C)(O)C(C)(C)C)NC(c1c(CNC(C2C(C(=O)OC)C2)=O)noc1)=O c1(C(N2C(CNC(c3ccnnc3S)=O)CC(OC)C2)=O)cc2oc(C)cc2[nH]1 N1(CC(COC)O)CCC(NC(=O)C(C)(C)c2cccs2)CC(C)(C)C1.C1=CC1 N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC1CC12CC(O)C2 CS(=O)(=O)c1ccc(F)c(-c2noc(CN3CCC(C4CCC4)C3)n2)c1 S(=O)(=O)(c1ccc(N(C)Cc2cnnn2C)c(F)c1)NCC(C)O c1(C(N2C(CNC(COC)=O)CC(O)C2)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 c1(OC)ccc(C(=O)NCCN(C(=O)C(O)P(C)(C)=O)CC(C)O)c(Cl)n1 O=[N+]([O-])c1ccc(F)c(CS(N2CCC3C(F)CC23)(=O)=O)c1 C1(C(=O)NCc2occ(C)c2)CCC=CC1NC(c1ccon1)=O C1(NC(C2(SC)CCC2)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1C C1(C(N(C2CCN(C(c3csnc3Br)=O)C2)CCC)=O)OCCC1C C1(C(=O)NC2CN(C(c3c(C)noc3C)=O)C(C)C2)Cc2ccccc2C(=O)O1 C(=O)(CN=c1cc[nH]cc1)NCC1(NC(C(CC)=CCCC)=O)CCCC1 c1(NCC(CCCCC)O)ccc(S(=O)(=O)NC2(CCOC)CCCC2)cn1 C=CCC(C(=O)N1CC(NC(C)=O)(CNC(c2cc(C3CCC3)no2)=O)C1)OC c1(C(N(CCCNC(C2CCOC2)=O)CC)=O)ccc(OCC)cc1.C1(=O)CN1 CC(C)C(C(=O)N1CCCCC1C(=O)NOC1CC2CCC1C2)C1CCC1 C(=O)(C1=CC(O)CCC1)NC1(NC(=O)CCCSc2ccccc2)CCCCC1 c1(C(N2CC3CN(C(COCC)=O)CC32)=O)c(F)ccc(Br)c1F c1(C(=O)NCCC2C(C)CCCN2C(c2ccsc2Cl)=O)ccc2c(n1)CCC2 C1(C(=O)NC(c2nnc(O)o2)C)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O c1(CN2CC(C(=O)OC)[SH](C(=O)OC(C)(C)C)CC2)ccc2c(Cl)ncnc2c1 N1(C(CC)CNC(=O)C(C)C(=O)OC)CCN(C(=O)C(c2cccnc2)OC)CC1 C1(CC(=O)NCCC2CCCN(C(C3C(C#N)C3)=O)C2)CCc2ccccc2C1 c1(CC(=O)NCC2(F)CCN(C(c3nc(C(C)C)oc3)=O)C2)c(O)ncnc1O CCC(C)CCC(=O)NC1CCC12CN(C(=O)COCc1ccc(OC)nc1)C2 c1(CNC(CCNC(=O)COCC2CC2)=O)ccc2c(c1)OCCCO2 C(=O)(C(N=[N+]=[N-])C(C)C)NCC(C(=O)N(CC(C)OC)C)C N1(C(C(C(=O)OCC)F)=O)CCC2CCN(C(=O)C(C)O)CC12 C12(CC)CCCN(C1)C(=O)C1(CC1)N(C)C2=O.CCC(CC(=O)OC)SC C1(C)(C(=O)NC2CC(CNC(c3c(SC)cccn3)=O)C2)CCN(C)CC1 c1(OCC)cc(C(N2CCCC2CNC(C2CCC2c2nc(S)n[nH]2)=O)=O)on1 C1(C#N)(C(N2C(CNC(CCOCCC)=O)(COC)CCC2)=O)CC2CC2C1 N1(CCCNC(C2C(C(C)C)OCC2)=O)CCN(C(c2cccnc2)=O)CC1 CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)C(=O)NCC1(C2CC2)CC1 c1(C(N2C(CCOC)CN(C(=O)C(C)CSC)CC2)=O)cc2ccccc2nn1 N1(C(C2C(CNC(CN3CCC(C)C3)=O)OCC2)=O)CCC(CN=[N+]=[N-])CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC(C)(O)CNC(C1Cc2nncn2C1)=O N1(C(C=CCOC)=O)CC(C2CCN(C(c3cccc(C(C)(C)C)c3)=O)C2)C1 C1(NC(Cn2c(C)nnn2)=O)CC2(C1)CC(C(=O)NOCC1CC=CCC1)C2 N1(C2CN(C(C3N=C(C)SC3)=O)C2)CCN(C(=O)Cn2cccn2)CC1 c1(C(=O)NC(C)C)ccc(NC2CC(C(=O)OCCO)C2)cc1 c1(C(=O)NCCCN(CC(=O)NCCC)CC)ccc2oc(S)nc2c1 C(=O)(CC(C)C(C)C)NCC(Cc1ccccc1)NC(c1oc(CC)c(C)c1)=O C=C(Br)CC(=O)NC1CCC(NC(=O)C(F)C2CC2)C1 Cn1nc(C(=O)NC2CCC2NC(C2(CC3CCC3)CC2)=O)ccc1=O Cc1ccc(N(C)C)c(C(=O)NC2CC(CNC(C3CC34CC4)=O)CC2O)c1 CC1CN(C(=O)CC(C)n2cc(Br)cn2)CCCN1C(=O)Cn1cccc1 N1(CCC)CCCC(C(N2CC3CC3(CNC(=O)C3=CCSC3)C2)=O)C1 C(=O)(C(CCC(=O)NCc1ncc(F)cc1Cl)N(C)C)OC C(c1ccncc1)=CC(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C Cc1ccc2oc(C(=O)N(C3(C)CC(C)(C)C3)C)c(C)c2c1 C1(NC(C2C3COCC23)=O)CN(C(C2CCCOC2)=O)CC12CCC2 CC1(C(=O)NCC(CO)NC(c2cc[nH]c2C2CCCC2)=O)CCCNC1=O C1(NC(c2ccn(CC)n2)=O)CCC12CN(C(=O)Cc1ccc(COC)cc1)C2 C1(C(N2C(C(C)NC(=O)COCC(F)(F)F)CCC2)=O)CC(=O)NC1(C)C c1(C(N2CC(C(C)(C)O)(CNC(c3cnc(C)[nH]3)=O)C2)=O)c([N+](=O)[O-])cnn1C Cc1cc(CO)ccc1N.c12cnc(s1)C1(CC1)N(N1CC(C3CCCO3)C1)C2=O Cc1ccccc1CCC(=O)NC(c1cccc(Cl)c1)CNC(=O)C(O)C(F)F N1(CC)CCN(CN2CCC(N3CCCC3)C2)C(=O)C1=O N1(C(C(C(CC)C)N(C)C)=O)CCC(C2CC2)(CNC(=O)C(C)(C)CO)C1 c1(C(=O)NCc2ocnc2C(=O)NCCN2CC=CCC2)cc(Cl)cnc1O c1(CNC2CC(NC(c3ncn(-c4ccccc4)n3)=O)C2)ccc(I)c(F)c1F c1(C(N(C)Cc2scc(C)n2)=O)ccc(CNC(=O)C(C)CC2CC2)cc1 C1(C(N(C2CCN(C(=O)C3=C(C)CCOC3)CC2)CC)=O)CC12CCC(=O)CC2 c1(C(=O)Nc2c(OCC)cc(C#N)cc2)cncc2cnccc12 N1(C(CCCCCSC)=O)CCN(C(=O)CC2CC(OC(F)F)C2)CC(CO)C1 C1(C(N2CCC(C(C)NC(CN(CC)CC)=O)CC2)=O)COC(C)(C)CO1 c1(C(C(=O)NCCC(C)NC(C2COCC2C(F)(F)F)=O)O)ccccc1Cl CCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(C)Oc2cccnc2)C1 c1(CN=c2[nH]cc(-c3cccc(OCC#N)c3)s2)cc(O)c(O)c(Cl)c1 C1(CNC(C2(C(C)(C)OC)CC2)=O)C2CN(C(c3cc(Cl)cn3C)=O)CC12 N1(C(CCOC)=O)CCCC(N(CCO)C(c2sccc2CN(C)C)=O)C1 N1(C(CCCN(C)C(c2ccccc2CC#N)=O)=O)CCC(C)(O)C1 Cc1cccc2[nH]c(C(=O)NC3CCCN(Cc4c[nH]c5ncccc45)C3)cc12 CC(CC(=O)NC1(CNC(=O)C=Cc2ccoc2)CC1)c1cccnc1 n1(CC(C)NC(c2cnn(C3CC3)c2)=O)cc(CNC(C2CC(F)(F)C2)=O)nn1 C(c1ccc(C(F)F)o1)=CC(=O)NC1(C)CN(C(C2C(C(C)(F)F)C2)=O)C1 C(=O)(CCC(N)=O)N(CC(=O)NCCN(C)C)C(C)C Cc1cc([N+](=O)[O-])c(NC(=O)C(=O)NCC2(c3ccccc3)COC2)cc1Br N(C1CCCc2c1cnn2C)CNC(CCN1CCCC(N(C)C)C1)=O C1(CNC(C(CCF)NC(=O)CCCC2CCCO2)=O)CC2OC1C1CC21 N1(C(C2CCCN(C(CCOCCC)=O)CC2)=O)CCc2ccc(C)cc21 c1(NC(c2cn(C(C)(C)C)nc2)=O)ccc2c(c1)CCN(C(=O)C#CC(=O)O)C2 CCC(CCC(=O)NCc1cc(C)ncn1)NC(=O)C(C)NC(=O)NC N1(C(C2N(C(C(SC)SC)=O)C3C(C2)C3)=O)CCCC(O)(C2CC2)C1 c1(N)ccc(S(=O)(=O)Nc2cccc(C)c2C)c(Cl)c1.C1(CC)CCCCN1 C(=O)(C(CO)C(C)(C)C)N1CCC(COC)(NC(=O)CCOC2CCCC2)C1 C(c1ccc2ncccc2c1)=CC(=O)NC1CCCC1NC(=O)CC1CCOC1 c1(C(=O)NC(CC)CNC(=O)CCCc2ccsc2)cccc(S(C)(=O)=O)c1 C=C(C)CC(C(=O)N1CCC(CC2CCC2)C1)NC(=O)CC1CCC(=O)NC1 N12CCC(F)(C1)C2=O.N1(C(=O)CCOC2CCC2)CCN(CCF)CC1 c1(C2CCCN(Cc3n(C(C)C)ncc3)C2)cc(F)ccc1F C1(NC(C2CC(NC(C3CCN(CC)C3)=O)C2)=O)C=CCCC1CO C(=O)(CC(C)n1cc(Br)cn1)NCC(CC)NC(=O)CCCc1cnn[nH]1 c1(C(=O)NC2COCC2NC(C2(C3CCCO3)CCC2)=O)cc2cccnc2[nH]1 c1(CC)ccc(C=CC(=O)NC(C)CN(C)C(c2ccnn2CC)=O)o1 n1(CC)nc(C)cc1C(N1CCC1CNC(C1(n2ccnn2)CC1)=O)=O c1(C(=O)NC2C(C)(C)N(C(=O)C(Cl)=CCl)CC2)ccc2nn[nH]c2n1 CCC(CNC(=O)COC)(CC)C(=O)NC(c1cc(C)on1)C C#CCCN=C(NCc1ccc(C2CC2)cn1)NC(C)CCS(C)(=O)=O N1(c2n(CC(OCC)OCC)c(C3C=CCC3)nn2)CC2CS(=O)(=O)CC2(C)C1 CC1CN(S(=O)(=O)CCNC(=O)N(C)CCc2ccccc2)CC(C)O1 O=C(CS(=O)(=O)C1CC1)N1CCN(C(C2C=CCS2)=O)CC1 CC1CCN(c2nnc(Cc3cscn3)n2CCC(=O)N(C)C)CC1C c1(C(C(=O)NCC(C)C)N(C(C)CC2CC2)C)ccc(C2CCC2)cn1 C1(CNC(c2occ(C)c2)=O)CCN(C(=O)C(O)CC(C)C)C12CC2 N1(C(C=C(C)c2ccccc2)=O)CC2CC(C)N(C(C3CC3F)=O)C2C1 Cc1ccc2c(N(C)Cc3cn(C)cn3)nc(=NC3CCCC(C)C3)[nH]c2c1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2(NC(C3CC(C)(C)CO3)=O)COC1C2 S(=O)(=O)(c1ccccc1C#N)N1CC2CCN(C(C#CC)=O)C2CC1 c1(CC)cc(C(N2CCCC(N(C(=O)C=CSC)CCO)C2)=O)ccc1F N1(C(CSC)=O)CC2CC(C1)C2NC(=O)C(CC(C)C)n1ccnc1 C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1CC(N(C)C(c2cc(Cl)ccc2O)=O)C1 C1(C(=O)NC(CNC(C(CC#C)O)=O)CO)CCCC2(CC2)C1 c1(C(=O)NC2C3CC(NC(c4cnc(C)[nH]4)=O)CC32)c(C)ccc(F)c1O c1(C(N2CCCCC(CNC(c3ccsn3)=O)C2)=O)cc2cccnc2o1 C1(C(N(C2CCOCC2)CC)=O)CCC2(CC1)CCN(Cc1ccc(I)o1)CC2 O=C(Cc1cc(Cl)cs1)NN=c1ccn(C2CC2)[nH]1 C12(NC(CCC(C)OC)=O)CCC(C1)N(C(=O)CNC(C1CCCC1)=O)C2 CC1CN(C(=O)C(C2CC2)N(C)C(C2CCCC(=O)C2)=O)CCS1=O N1(Cc2ccc(OCCCCCCCN=[N+]=[N-])cc2)CCC(C2CCOC2)C1 c1(C2CC(C(=O)NC3CC(NC(C4(C(=O)OCC)CCC4)=O)C3)C2)ccc(F)cc1 C12(NC(CCCOC)=O)CCC(F)(F)CC1CN(C(=O)C(C(C)(C)C)OC)C2 N1(C(C(n2ccc(C)n2)C)=O)CCC(C(N2CCC(C#N)C2)=O)C1C(C)C N1(CCNC(C(CSCC)NC(=O)CC(C)C2CC2)=O)CCCCC1=O N1(C(C(CC(N)=O)O)=O)CCC(CNC(c2nc3cnccc3s2)=O)C(F)(F)C1 c1(C(=O)Nc2c(O)ccc(C)c2)n[nH]c2c1CN(C(=O)CC1CCN(C)CC1)C2 N1(CC2CCC2)CCC(NCc2c(COC)onc2)CC1 C1(NC(C(n2cc(-c3ccc(Cl)cn3)nn2)C)=O)CCCN(O)C1=O c1(COC)ccc(C(=O)NCC2CCCC2NC(C23CC(C)C2C3)=O)o1 CC(C)(C)C(C#N)C(=O)NCCC(O)CNC(=O)Cn1cc([N+](=O)[O-])cn1 c1(C(=O)NCC(C)NC(c2cncc(F)n2)=O)cc(C2CC2)cnc1Cl O=C1CCCC(C(N2CC=CC2C(=O)NCC2(CO)CC=CC2)=O)C1 C1(NC(CC(C)(C)C)=O)CC(F)CN(C(c2ccc(O)c(F)c2)=O)C1 C12(CNC(CN(C3CCC3)C)=O)CCC(Nc3ncc(I)cn3)(CO1)C2 N1(C(c2cscc2Br)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N#Cc1ccc(SCC(=O)NCCOCCNC(=O)CNC2CCOCC2)cc1 CCS(=O)(=O)CC(=O)NC1COCC1NC(C1CC2CCC2C1)=O c1(C(=O)OCC)oc2ccccc2c1NC(=O)NCC1(n2cccn2)CC1 N1(C(C=CCCC(C)C)=O)CCC(C)C(N(C(=O)Cc2ccon2)C)C1 C1(Nn2cc(-c3c(C)con3)nn2)CC(C)OC(C)C1 N1(C(c2c[nH]c(=N)o2)=O)CCCCC(NC(=O)Cn2ccc(C3CC3)n2)C1 N1CCN(c2ccncc2)CC1.c1(CCC(C)=O)ccccc1OC(F)(F)F.OCl c1(C(=O)NCCOCCOCCNC(c2ccns2)=O)cnc2ncccn12 N1(C(c2ncc(C)cc2C)=O)CCCCC12CN(C(c1cc(C#N)oc1C)=O)C2 c1(OC)ccc(Cl)cc1CC(=O)N(C(C)CNC(=O)Cc1cccs1)C CC1=C(C)CC(C(N2CC3(C2)CN(C(=O)Cn2cnnc2)C3)=O)CC1 Cc1ccccc1COCC(=O)NC(C1CCCN1C(c1cccnn1)=O)C C(=O)(CCCCCC#N)N1C(CC(N2C(CC)CN(CC)CC2)=O)C2CCCC21 CCC(CC(=O)NC1CC(O)CN(C(=O)CC2=CCCC2)C1)CC(F)(F)F Cc1ncc(C(=O)NCC(C)(C)CNC(C2CC(CF)C2)=O)cn1 c1(C(N2CCN(C(C(C=C)C)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1 C1(NC(C(C)(F)F)=O)CN(C(=O)C=CC2CCCCCC2)C2(CCCOC2)C1 C1(NC(CNC(C)=O)=O)CCCC1C(=O)NCC1(N2CCOCC2)CC1 C1(NC(C(C)O)=O)CCN(C(=O)CC(c2ccccc2)C2CC2)CC1 C1(CC=C)(NC(=O)CCCC2CCC2)CN(C(=O)CC2CCNC2=O)C1 c1(C(N2CC(CNC(C(N3CCOCC3=O)C)=O)C2)=O)ccc2[nH]ccc2c1F N1(C(CNC(=O)OC)=O)CCC(NC(=O)CC(C)C(F)F)C(CO)C1 C1(C(=O)NCC2N(C(c3nnn(C)c3N)=O)CC(F)C2)CCCC(C)(C)O1 c1(C(C)C)ccc(C(=O)NCCC(C)(C)NC(=O)CC(=O)OC(C)(C)C)s1 C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)(CNC(C1CC2CCCC2C1)=O)CC c1(OC)cc(C(=O)NC2CCCC2NC(=O)C(COC(C)(C)C)N(C)C)n(C)c1 c1(CCC)ccccc1C(=O)NC1CCN(C(c2cc(CC)oc2C)=O)C1C C(CCC(C)(C)C(=O)Nc1ccc(NC(c2n[nH]cc2Cl)=O)cc1C)OC N1(CC(=O)NCCC2CCCN(C(c3cc(C4CC4)no3)=O)C2)C(=O)CNC1=O C(=O)(C1CCCc2ccnn21)NC1(CF)CCN(C(C(C)C2CCCC2)=O)C1 C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2snc(O)c2Cl)=O)C1 CCCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)C(C(C)CC)OC)C1 C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)Cc1csc(C(C)OCC)n1)CC c1(NC(C(CC2CCC2)NC(C2CC3(CCC3)C2)=O)=O)ccc(CCO)cc1 c1(C(N2CC3CCC(CNC(COC)=O)(C2)C3)=O)cnc([N+](=O)[O-])cc1C C1(C(N2C(CCC(=O)N3CC(c4ccon4)C3)CCC2)=O)CC2(C1)CC(O)C2 CC(C)CC(CNC(c1cc(=N)[nH][nH]1)=O)C(=O)N1CCCC1(C)C(C)(C)C C(c1cc(Cl)c2c(c1)OCCO2)=CCNC(C1ON=C(CC)C1)=O c1(C(C(N2CCCC(N(CC(=O)OC)C)C2)=O)CN)ccc(OC)c(OC)c1 c1(OC)cccc(C(C)NC(=O)CN2CCC(NC(C3CCNC3=O)=O)CC2)c1 N1(C(C2(C(=O)NC)CC2)=O)CCC2(NC(C34CC3COC4(C)C)=O)CCCC12 N1(C(C(C)N(CC=C)CC=C)=O)CCN(C(c2cccnc2)=O)CC1 Cc1cc(C(=O)N(c2cccc(Cl)c2)CCCO)c([N+](=O)[O-])c(O)n1 N1(C(C2N=C(C)SC2)=O)CC(F)(F)CC1(C)CNC(c1cn(CCO)nn1)=O C(=O)(CCC(C)(C)O)N(C1CCN(C(=O)C(CC=C)c2ccccc2)C1)CCOC N1(C(c2c(CC)oc(C)c2)=O)CC(NC(c2cnc(C(C)OC)s2)=O)CC(O)C1 C1(CC(=O)NCC(CNC(C2(CC)CCCCC2)=O)O)COCC(C)(C)O1 CCCCC(CC)C(=O)N(CC(O)CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)C C1(NC(c2ncn(C)n2)=O)CCSC12CN(C(=O)CC1CCC(C)(C)C1)C2 C(=O)(C(F)(F)CC1CCCO1)NCC1(C(C)NC(Cc2nc(CC)sc2)=O)CC1 CC(c1ccccc1C)=CC(N1CC(CO)(NC(c2cccnn2)=O)C1)=O N1(CC(C)NC(=O)C(O)Cc2ccccn2)CCN(C(C2(O)CCC2)=O)CC1 Cc1cncc(NC(c2nnnn2CC2CC2)CC2CCCCO2)c1 C1(NC(c2n(C(C)C)ncc2)=O)CCC(N(C(=O)CC2CCN(C)C2)C)CC1 c1(C(C(=O)Nc2c(CN(CC)CC)noc2)C2CC2)ccccc1F N1(C(C2(OCC)CCOC2)=O)CC(CC(=O)Nc2cncc(C#N)c2)C2(CC2)C1 C=CCCC(C(=O)N(C)CCSC)NC(c1cocn1)=O C1(C(=O)Nc2c(O)cccc2Cl)COC2(CCN(C(c3ccnnc3)=O)CC2)C1 CC1CN(C(C2(NC(C3CC(N(C)C)C3)=O)CCC2)=O)CCC1(O)C(F)(F)F C1(NC(C(C)(C)O)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CCC3)=O)C2 c1(C(c2nnnn2CC2CCOC2)Nc2cn(CC)nc2)cn(C)nc1C C(C(=O)NC1CCCC1CC(N1CCC2CCC12)=O)(C(C)C)OC c1(OC)nccc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)C2)c1F N1(C(CCCCC#C)=O)CC2OCC(NC(C3C(C(F)F)C3(C)C)=O)C2C1 N1(C(C(CCCC)=O)=O)CCC(C)(C)C(C(=O)NCCC(O)C(F)(F)F)C1 CCC(C)(CNC(c1ccc(O)cc1)=O)C(=O)NCC(O)C(C)(C)C C1(CC)(CC)CC(NC(c2ccc(Cl)c(O)c2)=O)CN1C(=O)C(F)OC(F)(F)F c1(NC(CN(CC)CC)C)ccc(S(=O)(=O)NCc2nccs2)c(Br)c1 n1(CC(=O)NCCNC(=O)C=Cc2ccc(F)nc2)ccc2cc(F)ccc12 Cc1nc(C2CC2)sc1C(N1CC=CC(NC(=O)Cn2ccnn2)C1)=O c1(C(=O)NCC2(CCNC(CN(CCOC)C)=O)CC2)nccc2c1NCCC2 C1(NC(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(c1nnco1)C2 N1(C(CC(=C)C)=O)CCC2(NC(c3cnn4ccsc34)=O)CC2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CN(C(=O)CC4CCC4)CC3C(F)F)c2[nH]1 c1(C(=O)NCC(=O)NCC(N2CC(OC(=N)O)C2)=O)cc(O)ccc1C Cc1ccn2ncc(C(=O)NC34CCCN(C(c5n[nH]cc5Br)=O)CC3C4)c2c1 C1(C(N(c2ccccc2)C)=O)CCCN(Cc2cccc(I)c2)CC1 c1(C(N2CCCC(N(C(C3CCNC3=O)=O)CC)C2)=O)c(OC)ccnc1O C(=O)(C1=NOCC1)NCC(CNC(c1c(CC)nc[nH]1)=O)O Cc1ccc(Cn2ccnn2)cc1.N12CC(C1)NC(=O)C1(CC1)CC1CC1C2=O C1(CC(=O)NCCOCCC(=O)NC(C)Cc2nc[nH]n2)CC=CCC1 C(C(=O)NNC(=O)c1cc(C)n(-c2cccnc2)c1C)C1CC1.Cc1cc(C)[nH]n1 Cc1cc[nH]c(=N)c1C(=O)NC1CCC(NC(=O)COc2ccc(F)cc2Cl)C1 CCC(C)(O)C(=O)NCC12CC1CN(C(c1ccc(OCOC)cc1)=O)C2 c1(NC(C2(C#C)CN(C(=O)CCSCCCC)C2)=O)cnc(F)c(C)c1 N1(C(Cc2ncc(CC)[nH]2)=O)CCCC2(CNC(=O)C(Br)=C(C)C)CCCC12 Cc1c(Br)cnn1CC(=O)N(C(C)CCNC(c1ccc(N)cn1)=O)C c1(C(C)NC(Cn2cc(-c3scc(C)n3)nn2)=O)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)SC)c1[N+](=O)[O-] n1(CC)nc(C(N2CCC(NC(c3ncccc3OC)=O)CC2)=O)cc1C1CC1 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)CC2)cc(S(N)(=O)=O)co1 C(=O)(C(C)CS(C)(=O)=O)N1C2C(NC(c3c(C)n(CCN(C)C)nc3)=O)CC(C2)C1 c1(C(N2CCC(C(CNC(C(CC)F)=O)C)CC2)=O)nnc2ccccc2c1O Cc1coc(C=CC(=O)NCCN(CC(C)O)C(c2ccc(Cl)o2)=O)n1 N1(C(C2COC3(CO)CC2C3)=O)CCCC(O)(CNC(=O)C(F)(F)C(F)F)CC1 N1(C(C2(COC)CC2)=O)CCCCC(NC(=O)CC(C(F)F)c2ccccc2)C1 CCCS(=O)(=O)CC(=O)OCC(=O)Nc1ccc(Br)cc1F C1(N(CC(C)OC(F)F)C(=O)CC2CCC(C)C2)CC2C=CC1C2 c1(C(=O)NCC(CO)NC(Cc2ccn(CC)n2)=O)cccc(S(C)=O)c1 C1(C)(CNC(CCC=CCC=C)=O)CCC(NC(C2COCCO2)=O)CC1 C1(NC(C2(OC)CCSC2)=O)CCN(C(c2snnc2C2CCC2)=O)CC1F N1(C(C(=O)OC)C(C)C2CCCC2)CC2CC1CCC2NC(=O)OC(C)(C)C C1(CC)(CO)CCCN(c2cc(Cl)nnc2O)C1 C1(CC(N2CC(C(C)NC(=O)CC3CC3)OCC2)=O)CCC2(CCC2)CO1 C(=O)(C(CC)OC1CC1)N1CC(OCCNC(C2C=CCC2)=O)C1 N1(C(C(C)C2CCC2)=O)CCC(NC(C2(S(C)(=O)=O)CC2)=O)C(CO)CC1 CC(C(C)(C)C(=O)NC1CC2C(C1)C2(F)F)NC(c1n[nH]c(=N)[nH]1)=O Cc1ncc(Br)cc1NC(C1CC1C(=O)Nc1cnc(C#N)nc1)=O N1(C(C=CC(C)C)=O)C2CCC1CC(NC(=O)C(c1ccc(F)c(F)c1)O)C2 C(C(O)C(=O)NC1(C(F)F)CC(NC(=O)C=Cc2nccs2)C1)OC c1(C(=O)NC(C(C)NC(C2CCC(N(C)C)C2)=O)C)ccnc2[nH]cnc12 c1(C(=O)NC(CC)CN(C(=O)COC2CC2(F)F)CC)cc2c(s1)CCOC2 C1(O)(CNC(C2CCCN2CC(F)(F)F)=O)CN(c2nnc(O)s2)C1 N1(C(c2c(C)c(I)nn2C)C(=O)NCCSC)CCC(O)CC1(C)C C1(CNC(C(C)n2cccn2)=O)CN(C(=O)CC(C)(C)CN(C)C)CC1(C)C CC1=C(C(=O)NCC(C)(C)CN(C)C(c2coc3c2CCCC3)=O)SCCO1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCC(NC(C2CC(F)C(=O)N2)=O)CC1 c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)oc2)=O)oc(C)nc1C(F)F N1(C(C2N(CC)CCC2)=O)CCC2CN(C(c3ccc(N(C)C)cn3)=O)CC2C1 C1(C(N(CCC#C)CCO)=O)CCN(C(C2CC=CCC2C)=O)C1CC CC1OCCC1CC(=O)N(CCNC(=O)C(C)(C)n1ccc(C2CC2)n1)C1CC1 c1(N(C)C)nc2ccc(C(=O)NC34COCCC3CN(C(=O)C3CC3)C4)cc2s1 c1(C(=O)NC2C=CC(C(=O)NCC3CC3[N+](=O)[O-])C2)cnc(Cl)s1 N1(C(C(CC=CC)CC)=O)CC2CC(NC(c3n[nH]c(CC)c3Cl)=O)C(C2)C1 c1(NCC2CCN(C(C3(C)CCCCO3)=O)CC2)cccc(F)c1[N+](=O)[O-] c1(CN2CC(c3cn(CCCC(=O)C(c4ccc(I)s4)=O)nn3)C2)ncc(Cl)cn1 CCC(C)CC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(c1cc(C)[nH]n1)=O c1(C(=O)NC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)ccc(N)c(F)n1 c1(OC)cc(OC)c(-c2ncsc2C(=O)NCC2CCC(=O)N2)c(OC)c1 c1(CC)ncc(C(=O)NC2CCN(C(c3csc(C)c3N)=O)C2C)c(C)n1 C1(C(=O)NCC(C)(C)NC(C2CC(C)OC(C)C2)=O)Cc2cc(F)ccc2O1 Cc1cccn2cc(C(N3CC4CCCC(C3)N4C(=O)C3=CCCC3C)=O)cc12 Cc1cc(C(=O)NCC2CCC(NC(C3Cc4nccn4C3)=O)C2)cc(N)c1O c1(C(=O)NC2C(C)(C)CN(C(=O)CN3CC(=O)NC3=O)C2)cnc2sccc2c1 C1(C(=O)NCC(C)NC(c2ccc(F)c(N)c2)=O)C(C)OC(C)C1C c1(C(N(CCCNC(=O)C=Cc2ccoc2)CC)=O)ncc(C(F)(F)F)cc1Cl CCCC(C)(C)CN=c1[nH]c(=NC2CCCCC2CC)[nH]c2c1SCC2 O=C1CC(CC(=O)N(C2CCCN(C(C3(F)CCCCC3)=O)C2)CCF)CCCN1 c1(C(=O)NCC(C)(C)NC(C=C(C)Cl)=O)cn(C)nc1C1CCCCC1 c1(C(=O)OCC)nc(CN(C(CN(C(=O)OC(C)(C)C)C)=O)C)cs1 N#Cc1cnn2cc(C(=O)NC3CN(C(C4CSC4)=O)C4CCCCC34)cnc12 C1(=CC(=O)N(CCCNC(C2CCCCS2)=O)C)CCCCCC1(F)F c1(NCC(C2CCC2)OC)nccc(=NCC2CCC=CCC2)[nH]1 CC(CSC(F)(F)F)C(=O)NCC1CCCC1NC(=O)C(C)N(C)C c1(C(N2CC(C)CC(NC(C(C(CC)C)O)=O)C2)=O)ccc2ccoc2c1 c1(C(=O)NC(CCNC(C2(C(=O)NC)CCC2)=O)C)cc(-c2ccco2)on1 N(C(=NCc1ccc(Cl)nc1)NCC(=O)N(C)OC)C(CCC=C(C)C)C C1(CNC(CC(C)O)=O)CCCCC1C(=O)NCCNC(C1CCC1)=O n1(CC)cc(C(N2CC(C)(NC(=O)C(O)CC3CC3)C2)=O)c(C(F)(F)F)n1 N1(C(C2CCN(C(CC(CC)O)=O)CC2O)=O)CCN(CC)C(C)(C)C1 C=C(C)CC(C(=O)N1CC(CC(C)NC(=O)C2=CCCSC2)C1)OC N1(C(c2c(F)ccc(F)c2O)=O)CCC2C(CCN2C(c2cccc(Cl)c2)=O)C1 C(CCC(=O)NCC1CC1CNC(C1CN(C2CCC2)C1)=O)OC C1(NC(C(C2CCN(C(c3csnn3)=O)CC2)C)=O)CC2CC1CC21CC1 c1(CC(=O)N(CCOCCN(C(=O)Cn2nnc(=N)[nH]2)C)C)ccsc1Br c1(C(=O)NC23CCC(CNC(C=CCOC)=O)(OC2)C3)c(C2CC2)nc2sccn12 C(=O)(C(C)(C)C(C)(C)O)N1CC(NC(c2cn(CC)nc2C)=O)(COC)C1 CC(C)C(C(C)NC(=O)C=Cc1ccccn1)NC(c1ncncc1Cl)=O N(C1CCc2c1ccc(Br)c2F)C(=O)NCC(C)Oc1cccc(C)c1 CC1(C)CC(CC(=O)NC2(C)CCN(C(c3cn(CC(F)(F)F)nn3)=O)C2)CO1 Cc1cncc(C(=O)NC(Cc2cn[nH]c2)C(=O)N(CCCO)CCO)c1 N1(C(CCC=CC)=O)CC(CC(=O)N(C)Cc2ncn(C)n2)CC1(C)C CCC(CC)C(C)C(=O)N(C)CC1COCCN1C(c1ccc(S(C)(=O)=O)o1)=O C(=O)(CCCCCF)NCCCn1cc(-c2scc(C(=O)OC)c2)nn1 CC1(C)COC(CCC(=O)NCCN(C(=O)C(F)=CC2CC2)C2CCCC2)C1 c1(-c2cc(OC)c(Br)cc2)n[nH]c2c1CN(C(=O)C(C)N(C)C)CC2 N(C(=NCCC=C(C)C)NCC(C)(C)C)CC1(OCC)CCCOC1 C(=O)(CCCCCn1cc(C2CCN(C)C2)nn1)N(CC(=O)OC)C(C)C c1(C(=O)NC2C3CN(C(c4c(C)cc(O)nc4)=O)C2C3)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCS(C)(=O)=O)N1CC(N(C(c2c(C)nc(CC(F)(F)F)s2)=O)C)C(O)C1 N1(C(CCOCCOC)=O)CC2CC1C2CNC(=O)C(C)C(F)F n1(CC)nc(C(=O)NC(C)CCNC(=O)C(O)C(C)(C)C)c(Cl)c1Br CC1(C)CCCC(NC(N2CCOCC2c2ncno2)=O)C1 C1(CNC(C(C)SC)=O)CN(C(=O)COCC(C)(C)C)CC(C)(C)O1 N1(C(C2N(C(C3CCCO3)=O)CCC(CC)C2)=O)CCc2nc(C)[nH]c2C1 C1(NC(CC2CC(COC)C2)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1)=O C12(NC(CCCC#C)=O)CCOCC1CN(C(c1noc3ccc(Cl)cc13)=O)C2 CCC(C)CC(=O)N(C1CC(NC(=O)C(c2ccc(C(F)(F)F)cc2)(C)C)C1)C N1(C(C=C(CC)C)=O)CCC(COC)(NC(=O)C(C)C)C1 Cc1cc(C)n(CC(=O)NC2CC(C)(CNC(C3(F)CCOC3)=O)C2)n1 C1(C(C)NC(CNC(C2C(OCC)CC2)=O)=O)CCN(C(=O)Cc2cc[nH]c2)C1 C12CN(CCC1CO)C2=O.n1(CC)nnc(C)c1C=O.n1(C2CC2)ccc(CO)n1 C1(C(=O)NCC(C)CN(C)C(c2ccc3ccoc3c2)=O)CCc2cncn2C1 C1(NC(=O)NC(COCC)C)N(C(c2cccc(C)c2)=O)CCC1(C)C N1(C(C=CC)=O)CCC2CCC(NC(c3ccc(F)cc3[N+](=O)[O-])=O)C1C2 n1(CC(N2CC(NC(C(C(C)OC)O)=O)(CO)C2)=O)cc([N+](=O)[O-])ccc1=O C=CC(CC)CC(=O)NC(c1ccccc1)CNC(=O)CC1(OC)CCCC1 c1(C(C)C)ccnc2c(C(=O)NCC(C)NC(=O)CCF)cnn12 N1(C(C(C)O)=O)CCC(C2(O)CCN(C(c3cc(Br)ccc3N)=O)C2)CC1 O=C(N1CC2COCC2O1)C1CCN(c2ccc(Br)cc2)CC1 c1(CC)nncn1CCNC(=O)CCOCCN(C(=O)C(c1ccn(C)n1)C)C C1(NC(c2nc(C(C)OC)oc2)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)CC1 c1(C(=O)NC2CN(Cc3cn(C(CC)C)nn3)C2)cccc(C)c1 C1(C(=O)NCCNC(C)=O)CCCCN(C(C2CCC(C)(C)OC2)=O)C1 C1(C(=O)NCC2(C(=O)NC3CN(C(CC)=O)C3)CCCO2)CCN(C)C1=O C(=O)(NNc1cc(C#N)ccc1F)NCCN(CC(F)F)C CON1CC(C(=O)NC(C)(CNC(c2cn(C)nn2)=O)C2CC2)CC1=O c1(C(=O)NCCCCN(C(C(C)CC2CC2)=O)C)ccc(S(C)=O)cc1 C(C)(N=c1[nH]c2c(c(=NCC3(C)CCC3)[nH]1)CCCCC2)c1scc(C(C)C)n1 C1(C(=O)Nc2ccc(CC)nc2C)C(C2CC2)CCN1C(=O)CC(Cl)Cl c1(CC(=O)NCCN2CCN(C(c3c(C)ccs3)=O)CC2)ccccc1S(C)=O Cn1ccc2[nH]c(C(=O)NC3CN(C(C4CC45CC5)=O)C4(CCC4)C3)cc12 c1cccnc1S.C(C(F)(F)F)=CC(=O)NCC1CC1C(=O)NCCNC(=O)C=C C1(n2cc(C(O)C(C)C)nn2)(NC(C(CC2CCC2)OC)=O)CCSCC1 c1(CNC(c2cc(C)nn2C)c2n(CCOC)nnn2)cnc2ncccn12 c1(C(CCC(=O)N(C(CCNC(COC(C)C)=O)C)C)=O)csc2ccccc12 C1(C(N2CC3(CN(C(C=CCC)=O)C3)C2)=O)CCc2ccc(F)cc2O1 c1(C(N2CC(O)(C(C)NC(=O)CSCCN(C)C)C2)=O)sc2cccnc2c1Cl CC1CCN(C(=O)COc2ccc(Br)cc2)CC1NC(=O)C=C1CCCCC1 n1(CC)cc(Br)cc1C(N1CCN(CC2CCN(C(=O)C(C)C)CC2)CC1)=O c1(CNC(CC2(C)CC2F)=O)ncoc1C1CN(C(=O)CNC=O)C1 C(C(=O)N1CCC(F)(c2cn(CCN(C)CCO)nn2)C1)(C(C)C)NC(C)=O Cc1cccc(C)c1S(=O)(=O)Oc1ccc2ccc(Br)cc2c1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(=O)Cc1nccn1C n1(CC)nccc1C=CC(=O)NCCC(C)CCNC(c1ccc(C(N)=O)o1)=O CC1CN(C(C2CCCCS2)=O)CCN1C(=O)COC1CCCOC1 C1(O)(C(=O)NCCN(C(=O)CSc2nccn2C)C)CCOC1 N1(C(C(CC)(C)CC)=O)CC2CCC1C(NC(=O)C=C1CCC(C)C1)C2 CC1CC(C)(C(=O)NCC(=O)NCC(=O)NCC2CC23CCC3)C1 Cc1ncc2c(n1)CCCC2N=c1[nH]c(=NCc2ncc(Br)s2)[nH]c2ccsc12 N1(C(c2cncc(C)n2)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O c1(C(=O)NC23CC(C(N4CC(CO)CC(CO)C4)=O)(C2)C3)coc2ccccc12 c1(C(N(CC(CNC(c2nc(CC)oc2)=O)C)C)=O)cc(Cl)c(F)c(Cl)c1 N1(C(C)=O)CC2CCCC(C1)N2C(C1CN(C(C(C)(C)C)=O)CCS1(=O)=O)=O c1(C(N2CC(F)(CNC(c3cc(F)ccc3Cl)=O)C2)=O)cc(F)cc2nn[nH]c12 N1(C(C(CSC)OC)=O)CCC2(CCCN2C(c2cccc(C(N)=O)c2)=O)C1 n1(CF)cnc2c(NCCN3CC4CCC3C4)nc(N3CC4C(C3)C4(F)F)nc12 C1(C)(NC(C)=O)CCN(C(=O)CC2C=CC(NC(c3cccc(CO)c3)=O)C2)C1 C1(OC)CC(CNC(=O)Cc2cncn2C)N(C(c2ccncc2Br)=O)C1 N1(C(C2CC(CNC(c3n(C)cnc3)=O)C2)=O)CC2CC3CC2C1C3O C1(C(N2CCC(N(C(c3onc(CC)n3)C)C)C2)=O)CCN(C)CC1 Cc1cc(N)cnc1C(=O)NCC(C)(C(C)C)NC(=O)CC1OCCC1(C)C C(CCCCNC(=O)NCC12CC(F)(C1)C2)N(C)C c1(C(N2CCCC(NC(C(C)(C)CC3CC3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C=CC(F)F)CC1O c1(C(N2CCC(COC)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(N2CCC(N3CC(C)(C)C3)C2)nccc(N2CCOC(CC(=O)N)C2)n1.CCl c1(C(=O)NC2CCN(C(COCCOC)=O)CC2C(C)C)ccc2ccoc2c1 C1(COC)CN(C(c2cc(C)on2)=O)CCN1C(c1cc(C)ccc1I)=O N1(CCn2cncn2)CCCC(C(N2CCCNC2)C)C1 c1(C(=O)NCC2(O)CC(NC(C(COCC)C)=O)C2)ccc(C(C)(C)C)cn1 N1(C(C(C)Oc2ccccc2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C2CC12 N1(C(c2ccn(C)c2)=O)CCCC(CNC(c2c[nH]c(=O)cn2)=O)CC1 CCCCC(C)(F)C(=O)N(CCCNC(=O)CC(=O)Nc1cccc(C)c1)CC N1(C(C2C(C)(C)C2(C)C)=O)C(CNC(C23CCC(CC2)OC3)=O)CC2CCCC12 C1(CNC(Cc2nnc(C)o2)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C Fc1cc(NC(c2cnccn2)c2nnnn2C2CCOC2)c2c(c1)CCO2 c1(C(=O)NCC2CCCCN(C(=O)C(F)CC3CCC3)C2)cccc([N+](=O)[O-])c1 Cc1cc(C(N2CC=CC2C(=O)NCCCc2ncn(C)n2)=O)cs1 c1(CC(=O)NC2CN(C(c3cc(C)n(C)c3C)=O)CC2O)cccc([N+](=O)[O-])c1 C(CNC(=O)C(C)(C)Cl)(C(C)(C)C)NC(CCC(=O)NC)=O C(=O)(CC(CC)C(C)C)NCC(CC)NC(=O)Cc1c(C)nn(C)c1C C=CCCCC(C)N=c1[nH]c(=NCCCn2cccn2)[nH]c2cccc(F)c12 C(C(COC)CC(=O)NCCC1CCN(C(=O)Cc2ccsc2C)CC1)OC C(=O)(C(CC(C)C)C(C)C)N(C(CNC(C(CCC(N)=O)OC)=O)C)C c1(-c2c(C(=O)NC3CC3C(=O)OC(C)(C)C)c(C)n(C)n2)cccc2c1COC2 CC1CC(=O)CCC1C(=O)NCC1(NC(=O)C=Cc2cccnc2)CCOCC1 C1(C(=O)NC)CCCCCN1C(C(=O)NCC(C)C)C1CC=CC1 C1(C2(O)CN(C(C3CC(F)(CO)C3)=O)C2)(CNC(=O)Cc2ccc(Cl)cn2)CC1 C(=O)(C(C)C(C)C)NC(CN(C(CCNS(CC)(=O)=O)=O)C)(C)C c1(C(=O)NCCNC(C)=O)ccc(-c2ccc(F)c3ccoc23)c2cc[nH]c12 N1(C(C)=O)CCC2(CC1)OC1(C)CC2(NC(=O)CCCc2ccc(C)c(C)c2)C1 C1(C(N2CCCC(CNC(c3c(COC)nn[nH]3)=O)C2)=O)CC2C(C1)C2(C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(O)(CNC(c2ccnnc2S)=O)CC1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCCC(C(C)NC(=O)C2=CCC2)C1)=O c1(CCNC(C2C(=C)C2)=O)ccc(CNC(c2sccc2OC)=O)cc1 N1(C(CCC2CCC(C)O2)=O)CCCC(C2CCCCN2C(c2coc(Cl)c2)=O)C1 N1(C(=O)CC2OCCCO2)CCC2C(C(N3CCOC(C4CC4)C3)=O)C2C1 C1(C(N2CC(F)(CNC(Cn3c(C)cnc3)=O)C2)=O)CCn2ccnc2C1 N1(C(C2=C(C)CCCC2)=O)CCC(NC(=O)Cc2c[nH]ccc2=O)C2(CCC2)C1 C12(CNC(C(C(C)C)NC(C)=O)=O)CCC(CC1)CN2C(=O)CC1CCCC1 C1(NC(c2nnc(C(C)C)s2)=O)C(C)CCN(C(C2CCC(=O)NC2)=O)C1C c1(CC)nc(C)cc(=NC(C)C2CN(C(=O)CSCc3csc(C)n3)CCO2)[nH]1 C1(N(C(Cc2scc(C)c2)=O)C)CN(C(C2CC2C(C)(F)F)=O)CC12CC2 c1(C(N(CCOCCOC)C)=O)n[nH]c2ccc(C(F)(F)F)cc12 c1(NC(C2C(NC(c3ccc(F)nc3)=O)C2)=O)ccnc(Cl)c1 c1(C(c2nnnn2C2CCOC2)NC(CCCSC)(C)C)cccc2c[nH]nc12 CCC(CCO)N=c1nc2c(ncn2CC)c(NC(CC)CCO)[nH]1 c1(CNC(CN(CCCN(C)C)CC)=O)[nH]c(=N)ccc1C c1(C(=O)NCC2N(C(CC(CC)C)=O)CC(O)C2O)cnc2c(ccn2C)c1 O=C(C1=CS(=O)CCC1)NC1(CO)CCCN(C(c2cccn3ncnc23)=O)C1 c1(C(=O)NC2C(NC(C(C(C)C)OC)=O)CCOC2)cc2c(F)cc(F)cc2[nH]1 Cc1oc(CO)cc1C(N1CCCCC1C(=O)N(CC(C)CO)C)=O N1(C(c2cccc(C#C)c2)=O)C2CCC1CC(N(C(=O)C(F)CCCC)C)C2 C(CC(O)C(=O)NCc1ncccc1CNC(=O)CCn1cccn1)SC N1(C(CNC(C)=O)=O)CCC(CNC(c2c(C)noc2-c2ccccc2)=O)C12CC2 C1(O)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 C(=O)(CCC1=CCc2ccccc21)NC1CC(NC(C(CCC)C#N)=O)C1 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)CSCC(N)=O)CC1c1cccnc1 C(=O)(C(C)C(F)(F)F)NC1C=CC(CC(=O)NC2(c3nc(C)on3)CC2)C1 C1(CCNC(C(=O)NCC)=O)CCN(C(C2CC2C(C)(C)C)=O)CCC1(F)F C(=O)(CCN(OC)C(=O)C(C)C1CCOC1)N(C(c1nn[nH]n1)C)C1CC1 c1(C(C)C)cnc(O)c(C(=O)NCCCN(C(=O)C(C)(C)COCC(F)F)C)c1 N1(C(C(CC)SC)=O)CC2=C(C1)CN(C(C1CCCCN1N=O)=O)C2 N1(C(C=CCOC)=O)CC(CNC(c2cccc(C)c2C)=O)CCC1C N1(C(C(c2cccc(F)c2)OC)=O)CC(n2cc(C3CCCO3)nn2)C(C)C1 C1(C(=O)NCc2cnc[nH]2)COCCC12CCN(C(C1CCCS1)=O)CC2 N1(C(C2CC(OC)C2)=O)CCCC(C)C1CCNC(c1ccn(C2CC2)c1C)=O Cc1ccc(C(=O)NC(CNC(=O)C2=C(Cl)CC2)C(C)C(C)C)c(=O)n1C Cc1ccc(Cl)c(OCC(=O)NC2CC3C2CCN3C(c2ccnc(C)c2)=O)c1 C1(CCOC)CN(C(=O)CC2CN(C)C2)CCN1C(=O)C=CC(=O)NC1CC1 C1(C(N2C(CNC(CC3(C(=O)OC)CCCC3)=O)CC2)=O)CCS(=O)(=O)C1(C)C Cc1cc(OC(c2ccccc2)C)ncc1-c1ccc(Nc2c(I)cnn2C)s1 N1(C(C=CC)=O)CCN(C2CCN(C(c3cncc(N)c3)=O)C2)CC1 Cc1nc(N2CCCC(CNC(=O)C(C)(C)CN(C)C)CC2)[nH]c(=N)n1 C(=O)(CCC(N)=O)N(C1CCN(C(=O)C=Cc2ncc[nH]2)CC1)CC#C c1(C(N2CCC(C3N(C(CC4C(=O)OCC4)=O)CCC3)C2)=O)c[nH]c(=O)cn1 N1(C(CCOC)=O)CCN(C(=O)CC2CCC(OC)CC2)CC1c1nccn1C c1(CNC(C2CC(O)CN2C(C2CN(C(CC)=O)C2)=O)=O)cc(=O)n(C)cn1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(NC(CC(CCCC)O)=O)CC1 N1(C(C)C)CC(C(=O)NCCC(C)NC(=O)Cc2cccn2C)CC1=O C1(C(N(CC)CC2CCN(C(=O)C(C)CO)CC2)=O)CC2CC1CC2O C1(NC(C(N2CCOC2=O)C)=O)CC=C(C(=O)N(C2(CC3CC3)CC2)C)C1 c1(CC)cc(C(N2CC3CC3(CNC(c3ncccc3C(F)F)=O)C2)=O)ccn1 CC1OCCC1(C)NC(C1(CCNC(=O)C(c2ccccc2)N(C)C)CCC1)=O CC1CC(NC(C2(C)CC2)=O)CCN1C(c1csc(C(C)(F)F)n1)=O N1(C(c2nnn(COCC)c2N)=O)CCCN(C(C2CC2(C)CC)=O)CCC1 N1(C(CCNC(=O)OC)=O)CCC(CNC(C2CCS(=O)CC2)=O)C1(C)C c1(C(=O)NCC2CCN(C(C=CCC)=O)CC2C)cc(Cl)cc(Cl)c1OC(F)F C1(C(N(CCNC(CCc2ccc(C)cc2)=O)C)=O)CC(c2ccncc2)=NO1 CCC(CC(=O)NCC(CC(C)C)NC(=O)CCN(c1ccncc1)C)C1CC1 Cc1cc(=NC(=O)COCCNC(=O)Cn2cc(C#N)cn2)[nH]n1C C(C(=O)NC1CCC(NC(c2cnoc2-c2ccc(Cl)s2)=O)C1)(C(C)C)SC C(=O)(C1=C(Cl)CCC1)N1CC(F)(C(NOCC(C(C)(C)C)O)=O)C1 N1(C(C=CC)=O)CCN(C(=O)CC(F)(F)F)CC1CS(C)(=O)=O c1(C(C)(C)C)cc2n(n1)CCN(CC1CCc3ccccc3C1)C2 N1(C(CCC#C)=O)CC(C)OC2(CCN(C(c3cc(O)cc(Cl)c3)=O)CC2)C1 C(CCCC(=O)NCCc1ocnc1CNC(=O)C(C1CC1)C1CC1)OC N1(C(C)=O)CCCC(C2CCCCN2C(c2cn(-c3cccnc3)nn2)=O)C1 C1(NC(CC2C(C)=NNC2=O)=O)CCC2(CC1)CC2NC(c1nn(C)c(Cl)c1Cl)=O c1(CC)[nH]nc(C(=O)NC2CC(O)C2CC(=O)NCC2(C)CCN(C)C2)c1C CCC1(CNC(=O)OC(C)(C)C)C(=O)N1.N1(C(C)=O)CCCCC1 C1(NC(c2cc(C)no2)=O)CCCN(C(=O)C(C)n2cccn2)CCC1 S(=O)(=O)(c1cc(F)c(F)cc1F)N1C2CN(C(c3cc(C)cc(C)c3)=O)CC21 c1(C(N(CCNC(C(C)(C)CF)=O)C2CC2)=O)ncc(Cl)cc1Cl C=C(C)CC(C(=O)N1CC2CC2(NC(=O)Cn2cnc(C(N)=O)n2)C1)OC C(=O)(C(O)CCCCC)NCC(CC=C)NC(=O)CCOc1ccc(C)cc1 C1(NC(CNC(CNC(c2cc(CC)ncn2)=O)=O)=O)CC12CCCCCC2 CCCCCCC(=O)N1CCC(COC)(NC(c2cnc(C(N)=O)cn2)=O)C1 C1(C(=O)NCC(C2CCC2)NC(CC=CCC)=O)COC2(CCC2)CO1 Cc1cnn(CC(N2CC(c3ccccc3)(NC(=O)Cc3n[nH]c(C)n3)C2)=O)c1 O=C(CC1OCCc2ccccc21)N1CCN(C(=O)COC2CCC2)C(CF)C1 C1(C(=O)NCC2(OC)CN(C(=O)C(C)Cc3c(C)noc3C)C2)CCC(C)(C)O1 c1(SCCNC(CNC(CCC)=O)(C)Cn2cccn2)ccc(S(N)(=O)=O)cc1 C1(NC(C2CC3CC3C2)=O)CCCC12CN(C(c1csc(Cl)c1Cl)=O)C2 C1(NC(COCC(=C)C)=O)CCCC(NC(c2cnc(C)nc2C(C)C)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)N1CCCC(CN(C(C(CCCCC)F)=O)C)C1 C1(c2onc(C)n2)CCCN(C(=O)Nc2ccccc2C(C)C)C1 N1(C(=O)CN(C(C2(C(=O)NC3CC3)CC2)=O)C2CC2)CCN2C(=O)NCC2C1 CCC(CCCC(=O)NC(CO)CCC(C)C)NC(C1(C(=O)NC)CCC1)=O C1(N(C)C(C2C=CCC2)=O)CCCCC1N(C)C(c1cc(Br)ccn1)=O c1(C(C)=O)cccc2c(CC(=O)NCc3cnc(C(C)O)s3)c[nH]c12 c1(C(=O)NCC2COC(CNC(C3CN(C4COC4)C3)=O)C2)n[nH]cc1[N+](=O)[O-] CCC(C)(C)C(=O)C(=O)N1CC2CC1CN(C(=O)COC1CCOC1)C2 c1(C(=O)NCCNCCCN2CCC(C(=O)OC)C2CC)cc2cccnc2[nH]1 C1(C(N2CC(CC=C)(NC(=O)CCOC3CC3)C2)=O)CCC(N(C)C)CC1 C1(C(=O)NC2CC(NC(=O)C=Cc3cnc[nH]3)C(O)C2)CCCC2(CC2)C1 N1(C(CCCc2onc(CCC)n2)=O)CC2CCC1CN2C(C1CC(SC)C1)=O c1(C(=O)NCC(c2ncc[nH]2)C)ccc(CNC(C2CCSC2)=O)nc1 C1(C(c2ccc(F)cc2)NC(c2ccc(-n3ccnc3)cn2)=O)CCCCCC1 N1(C(C=CCC)=O)CCCC(C(C)(O)CNC(c2ccsc2Cl)=O)C1 c1(OC)ccc(CNCC(N2CCCC2C(C)NC(C2(C)CCCS2)=O)=O)cc1 N1(C(c2cc(C)nn2C)=O)CC(C(=O)NCC2(n3ccnn3)CC2)CC1(C)C C1(C(N(CCCNC(=O)C(O)C2CCCC2)CC)=O)CC12CCSCC2 C1(C(C)(C)C)CCCC(C(=O)NC(C)(CNC(=O)CCc2ccco2)C2CC2)C1 CC1CCC(CC(=O)N(CCCN(C)C(c2cnn(C)n2)=O)C)O1 N1(C2CCN(C(C=C(CC)C)=O)C2)CCN(C(=O)C(CC)n2ccnc2)CC1 C1(O)(C(N2CCC(C(C)O)C2)=O)CCN(CC=Cc2ccco2)CC1 N1(C(C(C)n2cncn2)=O)CCC(CO)C(NC(=O)CCN2CCN(C)CC2)C1 c1(CN(C2COC2)CC#C)ccc(NC(C2CCN(C(=O)NC)C2)=O)cc1 C=CC(C)CC(=O)N1CCOC(CCCNC(c2ccc(CC)[nH]2)=O)C1 c1(N2CCC(=CCNC(c3c(Cl)nc(N(C)C)s3)=O)CC2)ccc2nnnn2n1 c1(C(=O)NC(CC)CN(C(=O)C=C2CCOCC2)CC)cn(C)c(C)n1 C=C(C)CC(C)C(=O)NCCCCNC(=O)CC1C=CCC1 c1(C(=O)NCC2N(C(c3nc(C(C)=O)sc3)=O)CC2)ccsc1S(N)(=O)=O c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)CC)cnc(C)nc1C1CC1 C(CC)(C(=O)N(CC(C)(Cn1cccn1)NC(=O)COCCC(C)C)C(C)C)OC n1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2ccc(C(C)=O)o2)=O)c1C c1(C(=O)NCC2(O)CN(C(C3(OC)CCS(=O)(=O)C3)=O)C2)cc(C)c(O)c(C)c1 N1(C(c2n(C)nnc2)=O)CCC2(CCC2CNC(C2(C)CCNC(=O)C2)=O)CC1 c1(OC)ccccc1C(C)CC(=O)NC1CCCC1(C)N1CCOCC1 CC1CN(C(c2nnn(C)n2)=O)CCC1N(C)C(c1ccc(C(F)(F)F)nn1)=O c1(N2CCC(NC(CCn3c(C)csc3=O)=O)C(O)C2)nn(C)cc1[N+](=O)[O-] c1(CC(=O)NCC(CNC(C(C2CC2)SC)=O)C)ccc(C(N)=O)nc1 c1(NC(=O)C(c2cccs2)NC(C2CC(CF)C2)=O)cncc(C(N)=O)c1 N1(C(c2cnc(C)[nH]2)=O)CCC(F)(F)C(CNC(=O)CN2CCCNC2=O)C1 C1(NC(C(C)=CC)=O)CCC(C)(CNC(=O)C(C)NC(=O)COC)CC1 n1(CC)ncc(Cl)c1C(=O)N(C)CC1CCN(C(c2cnc(C(N)=O)cn2)=O)C1 CCCC(C)CCCC(=O)N1CCCC1C(C)(C)NC(C1CCS(=O)(=O)CC1)=O c1(C(=O)OCC)nc(C(=O)N(C(C)CCNC(C2(CC)CCC2)=O)C)cs1 N=c1[nH]c(=NCC2(Br)CC2)[nH]c(=NC2CCN(C3CC3)C(=O)C2)[nH]1 N1(C(c2cc(OC)ns2)=O)C2CCC1CC(NC(C1(N(C)C)CCCOC1)=O)C2 c1(C(=O)NCC(C)(CO)NC(C(CC)n2cncn2)=O)ccc2n[nH]cc2n1 N(C(=NCCN1CCC(C)(C)CC1)NC1CSCC1C)CCOCC N1(C(CC(C(C)C)O)=O)CCCN(C(c2cc(N)cnc2Cl)=O)C(C)C1 C(=O)(C1NCCc2ccccc21)Nc1c(NC(C)=O)ccc([N+](=O)[O-])c1 C1(C(=O)NCC(C)N(C(C2C(C)C2)=O)C)C2CCC1(c1ccn(C)n1)C2 Cc1cc2c(cc1C)C(C(=O)N(C)CC1C3CN(C(c4cccs4)=O)CC13)CO2 N1(C(C2CC2CF)=O)C(Cn2cc(-c3ncoc3C3CC3)nn2)CC2CCCCC12 CC1CN(C(=O)C(F)=C2CCC2)CC1NC(c1csc(-c2ccoc2)n1)=O N1(C(C2(CSC)CC2)=O)CC(CCNC(=O)CSc2nccn2C)(OC)C1 C1(C(=O)NC2CC(CNC(=O)Cc3cccc(Cl)c3)CC2O)OC2CCC1CC2 N1(C(C(C)O)=O)CC(C)(NC(c2ccoc2I)=O)C1 C(C)(N=c1[nH]c(N2CCCN(CC)CC2)nc2ccsc12)c1c(CC)cncc1 Cc1ncccc1NC(c1nnnn1CC(F)F)C1CCSC1 N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)CC2CNC(=O)CCCSC c1(C(N(C(CC)CNC(c2cn(CCOC)nn2)=O)C)=O)cnc2ccccn12 C1(CNC(CC(c2ccccc2Cl)C)=O)CCN(C(=O)COC2CC2)CC1C C1(C(=O)NCC(C)(C)C2(O)CCC2)CC12CCC(F)(F)CC2 N1(C(C(CCC)OC)=O)CCCN(C(=O)COc2cccnc2)CC1C(C)C C(N=c1[nH]c(C)cc(=NC2CCC3CC2CO3)[nH]1)C1CCN(CC)C1 C(CCF)(C(=O)NC(C)C)NC(C(C)NC(C1(OCC)CCOC1)=O)=O C1(CC)CCCC1(C)C(N1CCN(CCCNC(=O)C2CC2)CC1)=O N1(C(c2c(C)cc(C)s2)=O)CCC(C)C(CC(=O)NC2CCCC(O)C2O)C1 CP(C)(=O)CC(=O)N1CCCC1C1(NC(=O)COc2ccc(Cl)cn2)CC1 C(=O)(CCCC(=O)C1CC1)N1CCC(N(C(=O)CCC2CC2(Cl)Cl)C2CC2)CC1 O=C(CC(C1CC1)NC(c1c[nH]cc1C1CC1)=O)NCC(O)CO C(C(C)(O)CC(=O)N1CCC(C(=O)NCCC(F)(F)CO)(C(C)C)C1)OC C#Cc1cccc(C(=O)NCC2(CCNC(C3(COC)CCOC3)=O)CC2)c1F c1(OC)c(Br)ccc(CN(CC(F)C(F)(F)F)C)c1O C1(NC(c2nc(CC)sc2)=O)CN(C(=O)COCC2CCCC2)C2CC12 Cc1nc2c(CCC(N3CCC(CNC(=O)CCOC(C)C)C3)=O)cccc2o1 C12(C(=O)NCC(C#C)OC)C(NC(=O)CC3CCOC3)C3CC1C2C3 C(CCCCCC(=O)NCC1CCSC(C)C1)NC(COCCCCC)=O C(Cn1cccn1)(C(=O)Nc1conc1CC)NC(C=C(CC)C)=O c1(C(=O)NC(CN(C(CC(CC)C2CC2)=O)C)C)cc(S(C)(=O)=O)ccc1OC N1(C(c2c(CC)cno2)=O)CCCC(F)(CNC(C2CC(F)(CO)C2)=O)C1 c1(C(N2C(C(C)(C)NC(C(C)C(F)F)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NC2(CC=C)CCN(C(C3CCN(C)C(=O)C3)=O)C2)cnc(Cl)cc1N CC1=C(C(=O)NC(C(=O)NC(C)CC2CCCCC2)c2cccs2)SCCO1 N1(CC(=O)NC2CN(C(=O)CN3CCCC3)CCC2F)CCCCS1(=O)=O C1(NC(C2CC(NC(=O)NCc3cc(C)cc(F)c3)C2)=O)CCc2nn[nH]c2C1 c1(C(=O)NC2(CC(=O)N(CCOC)C)CCC2)ccc(C)cc1O C=CC(CC)CC(=O)N1CCCC(NC(=O)C(=O)Nc2ccc(C)cc2)C1CC C1(CCC(=O)NC(C(c2ccccc2)NC(C2CC(OC)C2)=O)C)CCOCC1 CCCN=C(NCc1ccc(Cn2ccnc2C)cc1)NC1CC12CCCC2 C1(NC(C(C=C)CC)=O)CN(C(=O)C(c2ccccc2F)O)CC1C=C N#Cc1cc(NCC2CCCC23CCC3)c(N)cc1F CC(C)(C)C(CC(=O)N1CC(F)(CO)C1)NC(=O)CC1CC1C1CC1 Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)CC(C)c2cnn(C)c2)nc1C Cc1cccc(C)c1OCCC(N1CC(NC(=O)CC2CCCOC2)C(F)C1)=O c1(C(=O)NC2CN(C(C(N)=O)=O)CC2c2ccccc2)ccnc2ccncc12 C1(C(=O)NC2(CC#C)CCOCC2)CC2CN(C(=O)CSCc3cscn3)CC12 c1(C(=O)NCC2CCC(NC(c3c(CC)nns3)=O)C2)cnc(C2CC2)nc1O c1(C(N2CCN(C(C=CCOC)=O)C(C(C)C)C2)=O)ccn2c(C)ncc2c1 Cc1cc(C)c(C(=O)NC(Cc2cn[nH]c2)C(=O)NC(C2CCCC2O)C)cn1 O=C(CC1OCc2ncccc21)NCCSCC(O)CO c1(C(=O)NCC2(CNC(Cc3c(C)nc[nH]3)=O)CCC2)csc([N+](=O)[O-])c1 CCC(C#N)C(=O)N1CCC1C(=O)N(CCCOC)C C1(NC(C2CCCC2CF)=O)CCN(CCC(=O)Nc2ccc(F)cc2)CC1O c1(C(=O)NC(C2(O)CCN(C(CSCCC)=O)C2)C)cccc2nncn12 C(C(O)(C(=O)NCC(C)(CNC(=O)CCCCC(F)(F)F)OC)C(F)(F)F)OC Cc1cc(C(C)C)nc(N(C)CC2CCN(C(=O)CC3CC(C)(C)CO3)CC2)n1 N1(C(CC(C(=C)C)O)=O)CC(C)(C)OCC1CNC(c1cc(C2CC2)on1)=O c1(C(N2CCCC(C(=O)NC(C(=O)OC)C(=O)O)CC2)=O)ccc2cncnc2c1 c1(CN2CC(C(=O)N(C3CC3)Cc3ccccc3)OCC2)c(F)ccc(F)c1F N1(C(C2CCC2(F)F)=O)CCC(F)(C(N2CCN(CCO)CC2)=O)C1 c1(C(=O)OC)[nH]c(=NC2CC23CC(NC(=O)C(C)SC(F)(F)F)C3)sc1C c1(C(=O)NCC2CCCCN(C(c3cnncc3O)=O)C2)cccn2cncc12 C1(C2CCN(C(c3cnc(S)n3C)=O)C2)(NC(CC=CCC)=O)CC1 c1(C(=O)O)ccc(C2CCCN(C(=O)CCOC3CCCCC3)C2)cc1 N1(c2nc(N3CCN(C)CC3)c(Cl)cn2)CCC2(CC1)CC(N(C)C)CO2 C(=O)(C1=CC2CCCCCC12)NC(C(c1ccc(OC)cc1)OC)C C1(C(N2CC(N(C)C(C3CCC3)=O)C3(C2)CC3)=O)Cc2cc(Cl)ccc2O1 C1(OC)CCC(C(=O)NC2CCN(C(c3ccc(C(F)F)nc3)=O)CC2)CC1 Cc1csc2c(C(=O)NCC3CCN3C(=O)CC3(O)CCCCCC3)cccc12 C1(NC(COCCCC(C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCC1C C1(C(N(C(CC)CNC(=O)CNC(C2CC2C)=O)C)=O)CCCCC1 C1(OC)CCC(CNC2CCCN2C(=O)COc2ccccc2)CC1 CC(C)(C(=O)NC1CC(CNC(c2cc[nH]c2)=O)C1)C1CCCCO1 N1(C(Cc2ccc(C(=O)NCC=C)cc2)=O)CCC(N)CC1c1ccccc1 N#Cc1c[nH]cnc1=NC1CCC(NC(=O)CN2CCCCCCC2=O)C1 c1(CC(=O)NC(C)(CNC(=O)CSC2CC2)CO)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NC2C(CN)CN(Cc3ccccc3)C2)CC2CCC(C1)S2(=O)=O c1(-c2nc(CC(CC)C)nn2CCC(C)C)cc(C)ccc1Br C(C(C)(C)C(C)(C)C)NC(CNC(CNC(c1cc(OC)no1)=O)=O)=O c1(C(COC(=O)Cc2cccc(OC(F)F)c2)=O)cc2ccccc2s1 O=C(C1CCc2cc(O)cc(=O)n21)NC1CC1C(F)F c1(NC(CC2(O)CN(CC=C)C2)=O)nc(Br)ccc1OC C=C(Cl)C(C)(C)C(=O)NCCC1CCN(C(c2cccc(C(N)=O)n2)=O)C(C)C1 C1(OC)CC2(C1)CN(C(=O)C(C)CNC(C1(C)CCNC1=O)=O)C2 C(C(COC)C(=O)NCCN(C(=O)CC1CCCOCC1)C)OC c1(CC)ccc(C(=O)N(C)Cc2cccc(Br)c2)c(OC)c1 C1(CN(CC)CC)CCCCN1C(=O)Cc1cnn(C)c1C N1(C(C2CN(C(C3(SC)CC(=O)C3)=O)CC2F)=O)CC(C)=CC(C)C1 c1(C2C(NC(=O)CCCC3N=N3)C2)cccc2ccccc12 N1(C(c2c(C)nccc2)=O)CCC2(CC1)CC2C(=O)NC1CCC1(C)C C1(N(C(c2nc(OCC)oc2)=O)C)CCC(NC(=O)CCC(=O)N(C)C)CC1 CCC(CC)CC(F)C(=O)NC1CC(CN2CCNC2=O)C1 c1(C(=O)NCC(CO)NC(c2ccc(OC(F)(F)F)nc2)=O)c[nH]cc(F)c1=O C1(C(=O)NCC(C)OCC=C)CC=CCC1NC(=O)COc1ccn(C)n1 C(C)(C(=O)NCCN1CCC(NC(C2CCS2(=O)=O)=O)CC1)(C(C)C)OC c1(C(N2CCCC2CO)=O)ccc2c(c1)CCN(Cc1cccc3ccoc13)C2 C(=O)(C(C)CC)N(CCC)Cc1sccc1C CCCC(CNC(C1CCN(C(=O)C=Cc2cc[nH]c2)C1)=O)OC C(=O)(C(O)(C(F)(F)F)C1CC1)NC(CN(C(c1nc(CC)oc1)=O)C)CC c1(OCC)cc(Cl)ccc1C(N1C2CCC1(CNC(C1CCC1(C)C)=O)CC2)=O c1(OC)nscc1C(N1CCCC1CC(=O)NC1CC1C(F)(F)F)=O N1(C(CC(C)OC)=O)CC(CO)C2(CCN(C(c3csc(C(F)F)n3)=O)CC2)C1 N1(C(C(C)(c2cccs2)N(C)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)O)CC1 C1(C(=O)NCc2nnn(CC)n2)(NC(CCC)=O)CCCC1C c1(C(c2n(CC=C)nnn2)NCC2(C)COC2)cnn(CC(F)(F)F)c1C1CC1 C(=O)(C(C)(F)C(F)(F)F)N(CC)CC1CCN(C(C2CC2c2ncc[nH]2)=O)CC1 Cc1csc(=O)n1CCCC(N1CCCCC1C1CCCN(CC(C)O)C1)=O C(=O)(C1=NOC2COCC12)N(CCC(=O)NC1C(COC)CCC1)C N1(C(C2C(C)CC2)=O)CCc2[nH]nc(CNC(=O)Cc3cc(Cl)cc(Cl)c3)c2C1 C1(C)(C(=O)NC2CCC(CNC(C(C)(C)c3ccno3)=O)C2)CCCNC1=O CCS(=O)(=O)CC(=O)N1CCC(C)(N(C(=O)C(c2ccccn2)C)CC(F)F)C1 CCC(CC(=O)NCC1COCCN(c2ccncc2C#N)C1)C(C)(C)C N1(C(C(C)OCCCC)=O)CCC(CNC(c2cn(CCC3CC3)nn2)=O)CC1 c1(CNC(CC2(OC)CCC2)=O)n[nH]cc1C(=O)NC(CO)C(C)C N1(C(C(CC(C)C)NC(C(COC)(C)OC)=O)=O)CCc2ncsc2C1 c1(C(N2CCCC(NC(=O)Cc3ccns3)C(F)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(NC(C2(F)CCC2)=O)ccc(C2CCN(Cc3ccnnc3)CC2)cc1 N1(C(C2C(C=C)OCC2)=O)CC(CNC(C2CSC2)=O)C(C)(C)C1 CC1CC(C(=O)N(CC(=O)NCC(O)Cn2cccn2)CC2CC2)CN1C c1(OC)cc(=NC(=O)C(F)(F)C2CCCN(Cc3ccccc3)C2)[nH]n1C c1(NC2CC(C)C(C)(C)CC2)ccc(S(=O)(=O)NC2CCCCC2)cn1 CC1(NC(=O)NCc2cnoc2SC2(n3cccn3)CC2)CCNC1=O CCCC(C)(C)CC(=O)NCC1CN(C)CCN1C(C1CCC2(CCC2)OC1)=O c1(C(=O)OCC)cccc(N(C(=O)NCc2ccc(C)cn2)CC)c1 N1(C(C2CCCN2C(=O)CCn2cccc2)=O)CCCC(OC(F)F)C1 c1(C(=O)NCC2CCCC(NC(=O)CSC(F)F)C2)ccc2nc[nH]c2c1 C1(C(N(C)CCC2CC2)=O)CSCCN1C(C1CC1C(C)(F)F)=O C1(C2CN(C(C(CC#C)C3CCCCC3)=O)C2)CC(C)(C)CN1C S(=O)(=O)(c1ccc(-c2cccc(C)c2F)s1)CCSC(C)=O c1(CSCC(=O)NCCC2CCN(C(=O)C(=O)NC(=O)CO)C2)cccnc1 c1(CNC(=O)CC2CCCCCN2)ccc(S(=O)(=O)N2CCOCC2)cc1 C(=O)(C1CCc2cccc(O)c21)N1CC(CNC(C=CCOC)=O)C(F)(F)CC1 CCCC(C)C(c1nnnn1CC)NCCCc1noc(C(C)(C)C)n1 C(=O)(C(F)(F)C(F)F)N1C(CCNC(C(c2scc(C)n2)C)=O)CCC1 N1(C(c2ccc(=N)[nH]c2)=O)CCC2(CCC(NC(c3cn(C4CC4)cn3)=O)C2)C1 CCC1=C(C(=O)N2CCN(C(=O)C(F)C3CCOC3)CC2CCO)CCCO1 C(CN=c1[nH]nc(C2CC2)s1)=CCNC(c1cnc(Cl)c(C2CC2)c1)=O c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C(C)C)NC(N)=O)C(C)C)c(C)n1 CCC(C)(C)CCCC(=O)NCC1CCN(C(c2cnc(SC)n2C)=O)CC1C CC(C)CC(O)C(=O)N1CC(c2cccc(C(F)(F)F)c2)C(C)C1.C1CN1C(C)=O c1(C(N(CCCCN(C(C=CCC)=O)C)C)=O)ccc(C(C)(C)C)cc1N Cc1cccc(Br)c1C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)C(C)C C1(CNC(c2ccn(C(C)(C)C)c2)=O)CC2(CC2)CN1C(=O)CCC(=O)C1CC1 C1(OCC(=O)NC(c2cccs2)C)CN(C(C2C=CCS2)=O)C1 Cc1c(-c2csc(C(=O)Nc3cccc(F)c3OC(F)(F)F)n2)ccnc1Cl c1(CCOCC(=O)NC2(CNC(C=CC=CC)=O)CCOC2)ccc(Cl)cc1 C1(CC)CN(C(=O)CC=CCNC(=O)C(C2CCOCC2)F)CCS1 C12(NC(C(CNC(C=C(CCC)CCC)=O)C)=O)CC3CC(CC1C3)C2 C1(NC(C=CCC(C)(C)NC(=O)CP(C)(C)=O)=O)CCC(O)CC1 C(CCN=C(NCc1ccc(F)c(F)c1)N1CCC(C)(F)C1)SC c1(OC(C(=O)Nc2nccc(CC)n2)C)ccc(Cl)cc1C C1(CC(=O)NC2(C(=O)NCC3(C4CC4)CC3)CCC2)CC2(CC2)C1 C1(C(=O)NC2(CO)CN(c3ncnc(Cl)c3F)C2)C2Cc3ccccc3C12 c1(C(=O)NCC2CCCN(C(C(CC)OC)=O)C2)cn(CCO)c(=O)nc1O C(C(C)(CO)CO)N(C)C(C1OCCC1NC(C1COCCN1C)=O)=O C(CC(C(=O)N1CC(CO)CC1CO)NC(=O)CC1(O)CCC1)N(C)C CC(C)CC(C)(CNc1ncc(C(F)F)cn1)NC(C1C=CC=CC=C1)=O Cc1cc(N)c(C(=O)NC(C)CCNC(C2CC2[N+](=O)[O-])=O)c(F)c1 C1(NCc2ccc(CC(=O)O)s2)CC2CCCC(C1)C2(F)F C(=O)(C1=NN(CCO)C(=O)CC1)NC(C1CCCCN1C(=O)CCCN=[N+]=[N-])C C1(NC(=O)CC2CC2)CC2CC(C1)N(C(C1CCCN1C(N)=O)=O)C2 N1(C(C2(CC)CCN(C(=O)C=CC3CCOC3)C2)=O)CCOCC(C)(O)C1 c1(C(=O)NCC2(CC(=O)N(CC(CC)O)C)CC2)cncc(NC)c1 C1(C)(CNC(CCC=CCC=C)=O)CCN(C(C2(C)CCCCO2)=O)CC1 Cc1cccc(C(C)NC(=O)C(O)CNC(C2(Cl)CC2)=O)n1 C1(c2n(CCCOC)nnn2)(NCc2ccoc2)CCC(C(C)C)C1 CON1CC(C(N2CC(C)(C(=O)NC3(CCO)CCCC3)C2)=O)CC1=O N(C(=NCCC1CCCC1)NCc1ccco1)CC1C(N(C)C)CCCC1 c1(CNC(c2cccnc2N(C)C)=O)ccc(C(C)NC(CCC)=O)cc1 c1(OCCC)ccc(C)cc1-c1ccc(C(=O)Nc2c(O)cccc2Br)c(C)n1 C(C)(C(C)CCC)NC(CCN(C(CCC)=O)CC1CC1)=O c1(CC)cnc(C(=O)N(C(C)CCNC(=O)C(c2cccnc2)O)C)s1 c1(OC(C)C(=O)NCC=C2CCN(C(C3(C)COC3)=O)CC2)cccc(F)c1 N1(C(C2N(C(C3OCCC(C)C3)=O)C(C3CC3)CC2)=O)CCC2(CCC2)CC1 C1(C(N2C(CNC(CCCCOCC)=O)CC3CC32)=O)CCc2c(n[nH]c2C)C1 c1(SC)ccc(C(=O)NCc2ccsc2C(N2CC(c3nncn3C)C2)=O)o1 C1(C(N2CCCC(CNC(=O)COC(F)(F)F)C2)=O)(OCC)CCOCC1 C(=O)(C1(C)CCc2ccccc21)N1C(CNC(CNC(C)=O)=O)C(C)(C)CCC1 N1(C(C2CC(CC)OCC2)=O)CCCC(O)(CNC(c2nc(C)oc2C)=O)CC1 N1(C(CC)=O)CCCc2cc(N(C3CC4CCC(C3)N4)C(C)=O)ccc21 c1(-c2ccc(OC)nc2F)c[nH]c2ccc(C(=O)NC(c3ccccn3)C)cc12 C1(CC(=O)NCCCN(CCC)C(c2cnc[nH]2)=O)CCCC1C c1(C(=O)NCC=CCNC(C(C)OCOC)=O)cnc(C)nc1C Cn1cc2c(n1)CC(C(=O)NC1COCCN(C(c3coc(O)n3)=O)C1)CC2 CCCCCC(F)C(=O)NCCC(C)NC(=O)CC(C)(C)SC c1(OC)ccc(C(C(=O)NCC2CC2)N2CCC2C2CCC2)c(Br)c1O C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCC(CNC(c1c(C)n(C)nn1)=O)O N1(C(Cc2c(C)con2)=O)CC2(NC(c3ccc(=O)n(CCF)n3)=O)CCC1C2 C(=O)(C1CCCn2ncnc21)NC(C)CC1CN(C(C2CC3(C2)CC(O)C3)=O)C1 C1(CNC(=O)Cc2cncnc2)CC2(CCN(C(c3cnccc3Cl)=O)C2)CO1 c1(C(=O)NCCCN(C(c2ncoc2C2CC2)=O)CC)cnn2c1OCC(O)C2 c1(C(=O)NC(C(C)(C)C)CNC(C2OCCO2)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(CNC(CC2C(C)CCC2)=O)COCCN(C(c2ncc(C(F)F)s2)=O)C1 N1(C(C=C2CCC(C)CC2)=O)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1C1CC1 N(C1CCOc2c(Br)cccc21)C(=O)Nc1cc(NC(=O)OCC)c(C)cc1 N1(C(=O)NCC2(O)CN(C)C2)CCc2nc(O)ccc2C1 O(P(=O)(COC(c1cnc(-c2cccs2)nc1)=O)OC(C)C)C(C)C c1(CC)oc(C(=O)N(C)CC2C3CCCC23)cc1C C1(NC(c2ccc(-c3nc[nH]n3)nc2)=O)(CO)CCN(C(c2ccc[nH]2)=O)C1 c1(C(N(CC(CC)NC(=O)C(C)(C)O)C)=O)ccc2c(c1)S(=O)(=O)NC=N2 CC(C)(C)C(O)C(=O)NCC1(NC(=O)CSCCN(C)C)CCCCC1 N1(C(C(C)(C)SC)=O)CCCC(N(C)C(c2cc(C)nn2C(C)(C)C)=O)C1 C=C1CC(NC(=O)C(C2CC(OC)C2)NC(C2(SC)CC2)=O)C1 c1(C(=O)NCC(C)CNC(C2(F)CC2)=O)cc(N)ccc1C(F)(F)F CS(=O)(=O)C1(c2cn(C3CCN(C(c4cnc(C(F)F)s4)=O)C3)nn2)CC1 c1(CCC(=O)NC2COCC2F)ccc(Cl)nc1 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(=O)COC1CCCOC1 c1(SC)cc(C(=O)NC2(CO)CN(C(=O)C(C)NC(C3CCC3)=O)C2)oc1C N1(C(Cc2c(C)con2)=O)CCC(CNC(=O)C(C)C(C)C)C12CCC2 C=CC(COCC)N=c1[nH]c(=NCCCCCCCCOCC)[nH]c2ccc(Cl)cc12 c1(CC)conc1C(=O)NC(CC1CCCC1)C(=O)NC(CC1CC1)CO C=CCCC(C)(C)CNC(=O)C=CC1CCCN1C(=O)C=C1CCC1 c1(C(=O)NCCC(C)NC(C2ON=C(C)C2)=O)ccc2c(c1)nc(C)n2C1CC1 C1(N2CCN(c3c(C)nccc3)CC2)CCCCN(C(c2ccn(C)c2)=O)C1 C12(C)CCN1C2=O.c1(OC)conc1CNC(=O)C(C)(C)OC(C)=O C1(NC(CCS(C)=O)=O)CN(C(c2cc(C(F)F)cs2)=O)CCC1(C)C N1(C(C(C)OCCC=C)=O)CC2CCOC2(CNC(c2cn(C)nc2CC)=O)C1 C(=O)(C(C)(C)CC1CC1)NC(CCN(C(CSc1n(C(C)C)cnn1)=O)C)C C1(CNC(c2c(C)csc2)=O)CC12CCN(C(c1scnc1C)=O)CC2 Cc1ccoc1C(=O)NC(C)C(=O)NCCS(C)(=N)=O C1(OC)CCC(c2nnnn2CC2CC2)(NCCCSC)CC1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCCN2C(C2(O)CCCC2)=O)cn1 C(=O)(C(O)C(F)(F)F)N(CC(CNC(c1n[nH]c(C)c1Br)=O)C)C C(CN(C(=O)C(C1CCN(C(=O)CCN2CCCC2=O)C1)C)C)(C(C)C)OC N1(C(=O)Cc2ccc(Cl)nc2)CCN(C(C23CCCC2CC3)=O)CC12CC2 c1ccc2c(c1)CC(NC1=NCCN1C1CCOCC1)C2 CC(CC(=O)NC1CC(CO)C1)C(C)(C)NC(C1CC1(F)Cl)=O N1(C(CC(=C=C)C)=O)CCCCCC(NC(c2nnc3ccccn23)=O)C1 c1(-c2cn(CC3CCC(NC(CC4(C#N)CC4)=O)C3)nn2)ccnc(Cl)c1.C1CCC1 C(=O)(C#CC1CCOC1)N(CCCC(=O)NC1CC2(CCCC2)C1)C C(CCCCCNC(=O)C(C)n1cccn1)NC(=O)COC(c1c(C)nco1)=O C1(CC)CN(C(=O)C=CC(C)C)CCC1NC(c1ccc(=O)n(C2CC2)c1)=O c1(CN2C(C)CCC2C(=O)Nc2ncc(C#N)cc2I)cc2cccc(F)c2s1 N1(C(CCC(C)OC)=O)CCN(c2ncc(C(=O)OC)cn2)CC(C)(F)C1 c1(C(N2CC=CC(NC(c3ccc(C(F)F)cc3)=O)C2)=O)nc(Cl)ccc1F CC1(C)CC(NC(c2ncccc2F)=O)CN1C(C12CCC(F)C1CC2)=O N1(C(C(C2(O)CCC2)NC(c2cn(CCC)nc2)=O)=O)CCN(CC)C(C)C1 N1(C(C(COC)N(C)C)=O)CCOCC(CNC(=O)CCc2cc(C)on2)C1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2ccc(N)cc2C)=O)C(C)C1 N1(C(C=CC(C)(C)NC(=O)Nc2cc(-c3cnn(C)c3)[nH]n2)=O)CCC(CO)C1 C1(CC)CCC(NC(=O)C(CCNC(=O)CCCN(C)C(C)=O)OC)CC1 C12(C(=O)NCCOCCCNC(c3c(C)[nH]cc3)=O)CC1COC2(C)C C(C)(C)(C(=O)N1CC(CCO)(NC(=O)C(C)CN(C)C)C1)OC N1(C(COC(C)(C)C)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(CCO)C1 c1(C(=O)NC(c2cn(CCCNC(=O)C(O)c3cnc[nH]3)nn2)C)c(Cl)cnn1C CN(CC1CCN(S(C)(=O)=O)CC1)N1CCOC(c2ccc(C#N)cc2)C1 c1(C(C)(C)C#N)ccc(C(=O)NCC(C)(O)CNC(=O)CNC=O)cc1 N1(C(C2(SC)CCC2)=O)CCC(CCNC(=O)Cc2csc(Br)n2)C1 C1(OC)CC(O)C12CCN(Cc1cc(Br)cc(N)c1N)CC2 N1(C(C(C)OCCOCC)=O)CCOCCC1C(N1CCC(CC)C1)=O C1(NC(C(C2CCC2)NC(C(C)NC(CC)=O)=O)=O)CNC(=O)C1(C)C C1(C(=O)NC(CC)COC)(CNC(=O)CSC(C)(C)C)CC2(CC2)C1 C(=O)(CC1=CCN(C(c2cnc(C3CC3)o2)=O)CC1)N(C)Cc1nc(C)[nH]n1 c1(OC)cc(NCc2cc(Br)c(C)cc2OC)ccc1S(C)(=O)=O CC(C)(C(=O)NCC(C)(C)C#CC(=O)NC1(C(C)(F)F)CC1)C(F)(F)F c1(C(N2CC(C(C)(C)O)(CNC(CCc3nc(C)sc3)=O)C2)=O)nc(=O)n(C)[nH]1 C1(OC)CNCCC1CNCc1cnc(N2CCOCC2)n1C C(=O)(C1=CC2CCC1C2)N1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 c1(C(=O)NCC2N(CC(=O)NC3CCC4CC34)CCCC2)cccn2cncc12 CN1CCN(c2ncc(Cl)c(O)n2)C(CNC(c2ccc(F)nc2F)=O)C1 c1(C(=O)NCCN(C(CN2C(C)CCC2C)=O)C)cc(Cl)c(F)cc1F C1(N(C(=O)CCc2cc(Cl)cs2)C)CN(C(=O)CC2COCCN2C)CCC1O c1(CN2CC(C(N)=O)CC(C)C2)n[nH]c2ccc(-c3ccc(C(F)(F)F)s3)cc12 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC(CNC(c2ncc(F)cc2F)=O)C1 c1(SCC(N2CCC(CNC(c3cscn3)=O)CC2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCC#N)NC(CNC(COc1c(C)ccc(Cl)c1)=O)C C12(C)CCCN1C2.Cn1ccc(N(CC(C)(C)n2ccnc2)C(c2coc(Br)n2)=O)n1 N1(C(CCCCC)=O)CCOC(C)(CNC(C23CSC(C2)C3)=O)C1 Cc1cc(C(=O)N(CC(C)NC(C2(Nc3ccccc3)CC2)=O)C)c(Cl)cc1N c1(C(=O)NC(C)CC(C)NC(C23CC(F)(C2)C3)=O)cc(=O)c(Br)c[nH]1 C=C(C)CC(C)C(=O)NCCC1CCCCN1C(=O)CCCn1nc(C)nc1C C1(C(=O)NCC(CC(N2CCN(C(C)C)C(=O)C2)=O)OC)CC2CCC(C1)C2 c1(C(=O)NCCCOCCNC(CCCC=C)=O)ccc2c(n1)OCC(=O)N2 c1(OC)ccc(C=CC(=O)N(CC(C)(C)CNC(=O)C(C)CS(C)=O)C)nc1 c1(C(=O)NCC(CC=C)NC(c2cnc(N(C)C)cn2)=O)cc2cccn2cn1 C1(NC(c2cc(-c3cccc(OC)c3)[nH]n2)=O)COc2ncccc2C1 C(=O)(CC(C)C(F)(F)F)NC(C(=O)NCC1CCCN(CC)C1)C(C)O C(=O)(CCCCC(=O)c1ccccc1)NCC1(C)CCOC1 C1(C)(CC(=O)NCC(C=C)(C)C)CCN(C(c2cc(O)cs2)=O)C1 CC1OCCN(C(=O)CC2(C#N)CC2)C1C(N1CCCN(C(N)=O)CC1)=O N1(c2cc(CC)nc(Cl)n2)CCCC12CCN(C(=O)COCCN1CCCC1)C2 C1(C(N(C2CCN(C(CC(=C)Br)=O)CC2)CCC)=O)CCn2c(O)nnc2C1 N1(Cc2cc(C)n(C)n2)CCOC(C)(CNC(=O)CCC2CCOC2)C1 c1(C(N(C2CCCN(C(=O)CCS(=O)(=O)NC)C2)CC)=O)csc2nccn12 C=CC1(CC(=O)NCc2cc(Cl)cs2)CN(C(c2cccnc2OC)=O)C1 c1(C(N2CCN(CCCNC(=O)CC3CNC(=O)C3)CC2)=O)cc2c[nH]nc2s1 C(C(C(=O)N1CC=CCO1)NC(=O)C#CC1CC1)OC c12nn(C)cc1CNC(=O)COC(C)(C)CNC2=O.C1(CC)CCCSC1C N1(C(c2c(CC)nccn2)=O)CCC(C(=O)NC(C)CN2CCOCC2)=C(F)C1 c1(C(=O)OC(C)CF)ccccc1N1CCCS1(=O)=O N1(C(C2(OC)CC2)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(CF)C1 c1(NC2(C)CCN(CCCCCC)C2)ccc(OC(F)(F)F)cc1C c1(C(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)(C)C)ccc2oc(=N)[nH]c2c1 C1(NC(c2nocc2Cl)=O)CC(CO)N(C(=O)C=Cc2ccc(Br)o2)C1 CC(C)CC(C(=O)NCCC(N1CCCC1C1(C)CC1)=O)C(C)C c1(OC)c(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)oc2ccccc12 N1(C(CCCOCCOC)=O)CC2CCCC2C1C(=O)NCC(C)O c1(C(N2CCC(C(=O)OCC)C2)C(=O)NCCCF)cc(Cl)c(F)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CCC(C(C)(C)NC(C2CCCCN2N=O)=O)C1)OC N1(C(c2cc(OCC)no2)=O)CCCC2(NC(=O)C(C)(C)CC)CCCC12 c1(C(=O)NC2CN(C(C3C(C)(C)C3)=O)CC2N=[N+]=[N-])cc2c(s1)CCCCCC2 C(C)(CCC(=O)NC(C)Cn1cc(-c2ccc(-n3cccn3)cc2)nn1)SC c1(C(=O)NCC2N(C(C3CC(C)C(C)CC3)=O)CCC2)ccc2c(c1)CCN2C c1(C(N(CCC(C)NC(c2c(C)nc(C)n2O)=O)C)=O)cccc(C=C(F)F)c1 C(C)(C)(S(C)(=O)=O)c1cn(CC2CCN(C(C(C)NC(CC)=O)=O)C2)nn1 N1(C(c2c(CC)nn[nH]2)=O)CC(C)(C)CCC1CNC(=O)CNS(=O)(=O)N(C)C C1(C(=O)NO)CCN(CCCC=C)C1CC.c12ccsc1NC2=O Cn1cc(C(N2CC(CCNC(=O)C(C)(C)C(N)=O)C2)=O)c(=O)c(Br)c1 Cc1c(C(=O)NC(CNC(=O)C2CC2)C(C)(C)C)c(=O)oc2ccc(O)cc12 C1(CC=C)(OC)CC2CCC(C1)N2C(C1CC1C1CC1)=O.C12(COC1)CC(=O)N2 CC(C)CS(=O)(=O)CC(=O)NC1CCN(C(C2CCCS2(=O)=O)=O)C1 N1(C(c2c(C)oc(CO)c2)=O)CC2CC(C1)N(C(=O)Nc1cnc3[nH]ccc3n1)C2 C1(C(=O)OC)CCN(CCO)C(=O)C1.N12CC(C1)N(C)CC=CC2=O c1(OCCCC)ccc(C(=O)NCC(F)CNC(C2(C)CCNC2=O)=O)cc1 c1(CC(=O)NCC2OCCC(NC(CC3C(C)(C)C3)=O)C2)ccc2occc2c1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(F)(F)C(=O)NCC2CCCN2C2CC2)C1 c1(C2CC(C(=O)Nc3cccc(N4CCCOC4=O)c3)C(O)C2)cccc2nncn12 CCC(C(=O)N(CCCCC(=O)N1CCCC(CCCO)C1)C)C(C)C c1(-c2ccc(CN3CCC(OC)C3C)cc2)ccccc1[N+](=O)[O-] N1(CCOC(C(C)CC2CCCC2)=O)C(=O)CNC1=O c1(C(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)CC2)noc(C)c1C(=O)OC CC1=C(C(=O)NC2CCC(CC(=O)NCC3C=CCC3)CC2)CCCO1 C(=O)(C(F)CC(CC)CC)N(CCN(C(C(C1CCCC1)OCC)=O)C)C C=CCCCCC(=O)NC1COCC1C(=O)NC1CCC=CCCC1 c1(C(=O)NC(CC)(C)CNC(c2cc(Br)n[nH]2)=O)cnc2n1CCCC2 C1(NC(CC=C)=O)CC(OC)CN(C(C2(COC)CCOCC2)=O)C1 C1(CC)CC(CC(=O)NC2CCCC2NC(=O)C=CCO)CCO1 C1(C(=O)NCC#CCNC(CNC(=O)OC)=O)CC(CO)C1(C)C C(=O)(C1CCc2cc(Cl)ccc21)NCCC1N(C(C(CCCCC)O)=O)CCC1 C(C1CCc2cccnc21)NC1CCC(C#N)(c2ccccn2)CC1 C1(F)(CNC(C(C)SCC)=O)CC(CNC(c2c[nH]c(Br)c2)=O)C1 c1(OCC)ccc(-c2nc(Cc3sc(CC)nc3C)n(CCC(F)(F)F)n2)cc1 c1(C(N2CCN(C(c3cccc(C)c3C)=O)C(CF)C2)=O)cnn2ccccc12 CC1=C(C(=O)N2CCC(NC(=O)CC(F)(F)Cl)C(CO)CC2)C(C)(C)CCC1 CC(N=c1[nH]c(N(C)CCSc2ccccc2)nc(=N)[nH]1)c1ncccn1 N1(C(c2ccn(C)c2CC(=O)O)=O)CC2(C1)CN(C(c1ccc(Br)cc1)=O)C2 C12CCCN(C1)C2=O.C12CCN(CC1)C2=O.C1(NC(N)=O)CCOC1 c1(C(=O)NC2CC(C)N(C(c3ccnnc3Cl)=O)CC2)ccc2cc[nH]c2c1 c1(OC)ccc(-c2noc(C3CC4(OC)CC3C4)n2)cc1Br C(C(C)C(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)CC1)OC N1(C(CCSCC)=O)CCC2(CCCC2CNC(=O)C(O)CC2CC2)CC1 c1(C(C(=O)NCC2CCN(C(C=CC(C)C)=O)C2)O)ccc(O)c([N+](=O)[O-])c1 c1(CC)nc(C)cc(=NC2C3CN(C(=O)C(C)Cc4cccc(Br)c4)CC23)[nH]1 Cc1cnc(O)c(NC(c2n[nH]cc2CNC(C2CCC3(CC3)C2)=O)=O)c1 Cc1cc(F)cnc1C(N1CCC(C)C(NC(c2cc[nH]c2C)=O)C1)=O C=CC(C)(C)C(=O)NCCC1(O)CCN(C(C2CCC2(F)F)=O)C1 N1(C(C(CCCC)O)=O)C2CCC1C(F)C(NC(=O)Cc1ccc(C)cc1C)C2 N1(C(CC)=O)CCCC(C(=O)N(C)CCC(=O)C(C)OCCC(C)C)C1.C1CO1 C1(Cl)(C(=O)NCC(C)(C)CNC(C2CCCN2S(C)(=O)=O)=O)CC12CCOCC2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)C2CCC1CC(NC(c1n[nH]cc1Cl)=O)C2 C#CCC(C)C(=O)NCCc1ccc(NC(c2cscc2C)=O)cc1 Cc1ccc(-n2ncc(-c3nc(CP(C)(C)=O)no3)c2C)cc1 N1(C(C2(C)C(C)C2)=O)CCN(C(=O)C(c2cc(F)ccc2F)(F)F)CC(C)(F)C1 c1(C(N2CC(NC(CC(C)F)=O)C3(C2)CC3)=O)cc(F)cc(N)c1F C1(NC(c2n(C=C)nnc2)=O)CN(C(c2cnoc2CC)=O)C2CCCC12 C1(NC(c2c(CC)csc2)=O)C(C)CCN(C(=O)Cc2ccc(C)nc2Cl)C1C C1(C(N(C2(C(=O)NC3CCC(C)C3)CCC2)C2CC2)=O)CCN(C)C1=O C1(NC(C(=Cc2cccnc2)C)=O)CC(O)CN(C(c2c[nH]nc2C2CC2)=O)C1 c1(C(=O)NC2C(NC(C(C)OC)=O)CCCC2)cc(F)c(Cl)cc1Cl c1(C(N2CCN(C(c3cnc(C)s3)=O)C(CO)C2)=O)cccc([N+](=O)[O-])c1Br c1(OC)cc(CC(=O)NCC2(C)CN(C(c3ccccc3)C)CCO2)cc(Cl)c1 C1C(C)(CO)NC(=O)C(=O)N1C.C(C(F)F)NC=O.C(C)(C)(C)O C(=O)(C(O)C(F)F)NC(C1CCN(C(c2cccc(N)n2)=O)C1)(C)C Cc1ccnc2c(C(=O)NC(C)CN3CCN(C(=O)CCC(N)=O)CC3)cnn12 C12(C(=O)NC3(CC)CC(C)(C)C3)C(NC(c3ccc(C)cc3C)=O)C3CC1C2C3 C1(C(=O)NC2(C(=O)OC)CCCC2)CCC2(CN(CCCC(=O)O)C2)O1 c1(CN(CC)CC)nnc2n1CCN(CCCNC1c3ccccc3CC1C)C2 c1(COC)cc(=NCc2cccc(Br)c2Br)[nH]c(Cl)n1 c1(C(N2CCC(NC(c3c(CC)n(C)nc3)=O)CC2)=O)c(F)ccc(Br)c1C c1(NC(C(CCC=C)NC(C2CC(=O)N(OC)C2)=O)=O)cc(C#N)ccc1C C1(CCC)CN(C(C2(COC)CNC(=O)C2)=O)CCN1C(=O)CCS(N)(=O)=O c1(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)coc2c1COC2 C1(F)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)CCC(=O)Nc2nccs2)C1 CC1(C2CCCN(C(C3CC(F)CCN3C(c3nonc3N)=O)=O)C2)CC1 Cc1cn2c(n1)C(C(=O)N1CCCC(O)(CNC(=O)CSC3CC3)C1)CCC2 C1(C(=O)NCC2C(C)C2C)CC2CC1CN(C(=O)C#CC1CCC1)C2 C1(C(=O)Nc2c(C)noc2)CCC(C2CC2)N1C(=O)CC1CSCCO1 N1(C(c2c(CC)oc(C)c2)=O)CCCC(C)C1CNC(c1cccc(=O)o1)=O Cc1noc(C2C(C(=O)NC3CCC3CNC(c3ccsc3)=O)C2(C)C)n1 C(=O)(C1COc2ccc(F)cc21)NCC1(O)CN(C(Cc2nc(=N)[nH][nH]2)=O)C1 c1(C(C)(C)C)n[nH]c(=NCCCC(C)NC(=O)Cc2cccc3[nH]ccc23)s1 c1(CC(=O)NC(C(=O)NCCC=CC)CC2CCCC2)ccc(F)nc1 N1(C(CNC(=O)COC2CCOCC2)=O)CC(C)(COCCSC)CC1(C)C CC1CN(C(C2(C)SCCCS2)=O)CC1NC(=O)CNC(C1CCC1)=O C12(NC(c3c(C)con3)=O)CCCC1N(C(c1cc(Cl)sc1Cl)=O)CC2 CC(C)CC(C(=O)NCCc1cnnn1C)ONC(C1(C)CC=CCC1)=O N1(C(CCOCC#C)=O)CC(NC(c2ccc(N3CCCC3=O)cc2)=O)CC1C C(=O)(C(C(=O)N1CCC(C(=O)N(C)CC2CCCC2(C)C)(CF)C1)OC)OCC N1(C(c2c(CC)cn(C)n2)=O)CCOC(C)(C(C)C)C1 c1(C(=O)NCc2n[nH]cc2Cl)ccc(CCN(CCC2C=CCC2)C2CC2)cc1 C1(OC)CN(C(c2c(CO)n[nH]c2C)=O)CC1NC(c1cn[nH]c1)=O Cc1cccc(C(=O)NCCC(=O)NCCC(O)C2CC2)c1 N1(C(COc2cn(C)nc2)=O)CC=C(C(=O)NC2CCCC(O)C2O)C1 C(=O)(CCS(N)(=O)=O)NCC(CC)N(C(=O)C=CSC)C N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)C2 C#Cc1cn(C)nc1C(=O)NC1CCN(C(C2(OC)CCOCC2)=O)CC1 C1(CNC(C=C2CCC(C)C2)=O)CCCCN1C(=O)CCCNC(N)=O C(=O)(C(F)(F)C(C)(C)O)NC1CC(C)CN(C(c2ccnn2C2CC2)=O)C1 Cc1cc(C(=O)NC2CC3CC(C2)N(C(C24CC(C)(CO2)C4)=O)C3)ccc1C#N C1(CNC(C2(c3c(C)ccc(C)c3)CC2)=O)CC2COCC2N1C(=O)CCF c1(NC(=O)Nc2cc(CN(C)C)ccc2F)nc(Cl)cn2ccnc12 C1(C(=O)NCC(CC(=O)NCC(COC)(F)F)OC)CC2(CCCO2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC(C1)N2C(c1ccnc(F)c1)=O Cc1cc(C#N)ccc1C(N1CC(C)(CNC(=O)CCCCN(C)C)C1)=O CC(C)(F)C(C)(F)C(=O)N1CC(NC(C23CC(CC(F)F)(C2)C3)=O)CC(O)C1 c1(OC)ccccc1CCC(=O)NC1CN(C(=O)CCc2cnoc2)CC1C N1(C(C2N(C(C)C)CCC2)=O)C(CC(=O)NCCCC(F)F)C2CCCC12 c1(CC(C(=O)NC(CCC=C)C(=O)O)(C)C)cc(OC)c(OC)cc1OC c1(C(N2CCN(C3CN(C(CS(CC)=O)=O)C3)CC2)=O)cc2c(s1)CN(C)CC2 N1(C(C(=O)NC(C)C)=O)CC2(CCC2NC(=O)C(O)Cc2ccc(F)cc2)C1 C[Si](C)(C)c1cccc(-c2ccc(CNCc3cc(Br)c[nH]3)cc2)c1 c1(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)cncc(Cl)c1 c1(C(=O)NCC(CO)NC(CCC(CC)C)=O)sc2ncccc2c1N N1(C(c2ccc(CCC)s2)C(=O)NCCOC)CCC(P(C)(C)=O)C1 C(N=c1[nH]c2c(c(=NCC3(P(C)(C)=O)CC3)[nH]1)CCCC2)C1(CC)CC1 C1(CNC(c2cc(OCC)n[nH]2)=O)CCCN(C(=O)C(=Cc2c[nH]cn2)F)CC1 c1(CC(N2CC(NC(=O)Cn3cc(CO)nn3)C(F)C2)=O)ccc2c(c1)CCO2 C(=O)(CC(C)(C)CC(F)F)NC(C1(O)CCN(C(C2CC2C(C)(F)F)=O)CC1)C c1(C(=O)NCC#CCNC(C(C)c2ccco2)=O)sccc1Cl C(=O)(C(CCOCCO)NC(=O)CCn1ccnc1)N1CC(C#C)C1 C1(C(=O)NCC2CCCS2)CCN(C(=O)CCOCC2CC2)C1 C1(C(N2CCCC(C(C)NC(c3cc(F)c[nH]3)=O)C2)=O)CCCC1(C)F Cc1ccc(CCC(=O)N(CCCN(C(=O)CC2CCCC2)C)C)s1 N1(C(C(C)C)=O)CCC2(CC1)CC(NC(C1CC1(C)C(C)C)=O)CCO2 C1(O)(C(=O)NCC(CC)NC(c2c[nH]c(C(F)(F)F)c2)=O)CCCC(C)CC1 c1(C(=O)NCCC2N(C(C=CSC)=O)CCC2)ccc(Br)c(C)n1 C(CC(C(=O)NC(C)(C)C)OC(C1(c2cccc(Cl)c2)CCC1)=O)SC C(=O)(C(F)CC(C)C)NCCN(C(c1ccc(C)nc1O)=O)CC N1(c2c(C)cccc2)C(=S)NC(c2csc(C#N)c2)C2=C1CCNC2=O C1(C(N2C(C(=O)NCc3ncc(Cl)cc3Cl)CC(O)C2)=O)CCc2nc[nH]c2C1 CN1CCC(N(C)C(C2CC2(c2ccccc2Br)F)=O)C1=O c1(OC)cnc(F)c(C(N2CCCC2C2CCN(C(C3(O)CCC3)=O)CC2)=O)c1 Cc1cc(NC(=S)NCc2cc(C)on2)c(C)c(C)c1 c1(C(N2C(CC(=O)N(C)CC3N(CC)CCC3)CCC2)=O)ccnc2cc[nH]c12 NS(=O)(=O)c1cc(C(=O)NCC2C=CCN2C(=O)Cc2cc[nH]c(=N)c2)co1 N1(C(C(C)C2(O)CCC2)=O)CCCC(CCNC(c2cnn(CCO)c2)=O)CC1 c1(C(N(C2CCC(NC(C3(C)CC4CC4C3)=O)CC2)C)=O)cccc(=S)n1O c1(C(=O)NC2(C)CCN(C(=O)CC3(N4CCCC4)CC3)C2)cc(O)ccc1Cl C1(NC(CSCC=C)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC1CO Cc1nccnc1C(=O)NCC1CCN1C(=O)C(N1CCCCC1)C C(=O)(C1CCCn2nccc21)N1CCN(C(COc2ccc(C)cc2F)=O)CC1 N1(C(CS(C)(=O)=O)=O)CC2(CCCC2NC(=O)CCOC2CCOC2)C1 C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(c2cccc(F)c2Cl)=O)C1 CC1CCCCC1(CNC(=O)CC1CC2(CC2)CO1)NC(C12CC(F)(C1)C2)=O N1(C(c2cc(OC)nc(Cl)c2)=O)CC2CCN(C(C3C(C)(C)OC3(C)C)=O)C2C1 C[Si](C)(C)C1(CNC(C2(CCNC(=O)CC3CCCO3)CC2)=O)CC1 C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(c2cc(C)cs2)=O)C12CCC2 c1(C(=O)NC23CC(CNC(c4nc(CCC)sc4)=O)(C2)C3)ccc2sncc2c1 c1(C(=O)NCC2C(NC(C=COCC)=O)CCCC2)cc2ccccc2o1 c1(CCC(N2CC(OCCNC(CN(C3CC3)CC)=O)C2)=O)ncc(C)[nH]1 c1(N(CCC)CC)ncnc2cccc(OC(=O)CCc3nccs3)c12 c1(C(N2C(CNC(=O)C3CC3)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(=O)NC2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)cn(C)c2ccccc12 Cc1noc(C)c1C(C)CC(=O)N(C)CCN(C(=O)CCNc1ccccn1)C C1(C(=O)NCC2N(C(c3cc(C)sc3)=O)CCC2)CCCCCS1(=O)=O N1(C(c2c(C)cco2)=O)CCC2(NC(c3cccc(N(C)C)n3)=O)CCCC12 N1(C(c2cc(=N)[nH]cc2)=O)CCC(CNC(c2scnc2Cl)=O)C12CC2 N1(C(=O)Nc2c(C)c(C)cc(C)c2C)CCCC2(CC1)CNC(=O)O2 N1(C(CCn2c(=O)cc(C)nc2)=O)CC(C)CN(C(C2CN(C)C2)=O)C(C)C1 C1(CCNC(CCC(=O)OC(C)(C)C)=O)CC2CCC1CC2 C(CCS(C)(=O)=O)NC(C1(NC(Cc2cc(C)no2)=O)CCSC1)=O Cc1oc(CNC(C2CCC2(F)F)=O)nc1C(=O)NCC1CCCC(=O)N1 C1(CNC(CCCOCC=C)=O)C(CC)CCN1C(c1ncncc1N)=O C(CCC)(C(=O)N1CCC(N(C(=O)CN2CC3CC3C2)C)C1)=CCC C=CC(CCC)CC(=O)N(CCCOCCN(C(=O)CC1CCCOC1)C)C C(CO)(C(F)(F)F)NC(C(CC1CCOCC1)NC(c1cc(=N)[nH][nH]1)=O)=O C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(=O)Cc2ccccc2O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(C=CCC)=O)C C1(NC(C(C)C2CCCO2)=O)CCC(N(C)C(C2C=CCCC2)=O)CC1 N(C1CCCn2ncnc21)C(c1cc(CNC(C2SCCS2)=O)cs1)=O c1(-c2c(C(=O)Nc3nccc(Br)c3Cl)cc(Cl)cn2)ccc2[nH]nc(O)c2c1 CC(CC(F)(F)F)NC(=O)CCC1CC(NC(C2CCCS2)=O)C1 Cc1[nH]c(=N)nc(N2CCCC(C)(C(=O)NCC3CCCC3)C2)c1C Cc1ncncc1C(N1CCN(CCN(C)C(C2(Cl)CC23CCC3)=O)CC1)=O c1(C(=O)NC2CN(C(CN3CC(C)C3)=O)C(C)C2)cc(S(=O)(=O)N(C)C)c[nH]1 C1(=CC(=O)NC2CCC2NC(c2ccc3c(c2)OCC3)=O)CCCCCC1(F)F c1(CC(=O)NCCC(C)NC(CCSCC)=O)ccc(C(=O)OC)cc1Cl c1(CC(=O)N(C)CC2CCN(C(c3n(CCC)ccc3)=O)C2)ccc(Cl)nc1 C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(C=C)(F)F)=O)C2C(C1)C2 c1(COC)nc(C(=O)OC(c2cnn(Cc3ccccc3)c2)=O)n[nH]1 N1(C(C2(C#C)CCCC2)=O)CC2(C1)CN(C(=O)Cn1ncc(O)nc1=O)CCO2 N1(C(c2cn(CCC)nn2)=O)CC(CNC(c2cncn2C)=O)CCC1C N1(C(CN(C2CC2)CC)=O)CCc2ccc(-c3ccc(Cl)cc3)cc21 C(=O)(C1=CCCOCC1)N1C(C(C)NC(c2ccn(C(C)C)n2)=O)CCC1 C(C)(C(C)C(=O)N1CCN(C(C)C)CC1)NC(c1cnc(CC)s1)=O S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCC(C)F)[nH]1)COCC2)NC C1(C(=O)NC2CC(NC(c3[nH]cc(C)c3)=O)C2)CC(S(N)(=O)=O)C1 c1(C(=O)NCCC(C(C)C)NC(=O)CCCC(N)=O)cc(F)cc2ccncc12 N1(C(c2ccc(OC)nc2C)=O)CCC2CN(C(=O)C(C)O)CCC12 c1(C(N2C(C)CC(NC(c3c[nH]c(Br)c3)=O)CC2)=O)cnn2cccc(Cl)c12 c1(CN(C(CCN(C(c2nc(C)sc2)=O)C)=O)C)cccc(O)n1 C1(C(N(C)CC2CCN(C(=O)COc3ccon3)C2)=O)CN(C)C(=O)N1 N1(C(=O)Cc2ccc(Cl)s2)C2CC3C4CC(C3C2O)C1C4O N1(c2snc(SC)n2)C2CCC1CC(NC(=O)COC1CCCC(C)C1)C2 C12=CC(=NCCC(=O)N1)NC=N2.C(CN(C)C)(C1CC1)OC C(=O)(C1=CCCN(Cc2cc(F)c(O)c(F)c2)C1)NCc1c(Br)ccc(OC)c1 C1(C)(C(N(CC=C)C)=O)C=CCN1C(c1cnc(C2CC2)o1)=O c1(OC)ccc(C)cc1NCCC(=O)NC1CC1NC(=O)Cc1nccn1C CC1CCCN(C(=O)C(=O)NCC2(C)CCN(Cc3cc[nH]n3)C2)C1 CC(C#N)CN=c1nc2sccc2c(NCC2(C)CC2(F)F)[nH]1 C(=O)(C(COC)CC(C)C)N1C(CC(=O)NC(CCCC)C)C2CCCC21 c1(OC)cccc(-c2ccnc(N3CCN(C(=O)C=CCBr)CC3)c2)c1 C1(C(N2CCC(CNC(CCCc3c(C)ccs3)=O)C2)=O)(CF)CCOCC1 C1(CNC(CCC2(COC)CC2(F)F)=O)(CO)CCC(=O)N1 N1(C(C(CC)O)=O)CCc2sccc2C1CNC(c1ccc[n+]([O-])c1)=O c1(C(N2C(CNC(C(C(CC)O)C)=O)C3CCC2C3)=O)ccnc2[nH]cnc12 CCCC(O)CC(=O)N(C1CCN(C(=O)C(C)(C)COC)CC1)CCC c1(SC)cccc(C(=O)NC(CNC(=O)C2=CCC2C)CO)c1[N+](=O)[O-] Cc1cccc2c(C(=O)NCC3C(C)(C)C3(F)F)c[nH]c12 N1(C(C)=O)CC(O)CC1C(=O)NC1CCC1NC(c1nc(O)c(C)s1)=O c1(C(=O)NCC2(O)CN(C(=O)C=C(Cl)Cl)C2)coc2c1CS(=O)(=O)C2 c1(OCC(=O)NCCN(C(=O)CCc2ccccc2Cl)CCOC)ccccc1C c1(C(N2C(CNC(c3csnc3C3CC3)=O)CC(OC)C2)=O)ccc(C)cc1C C1(C2CC2)(CNC(CC(CC)O)=O)CCN(C(c2cnc(O)nc2O)=O)C1 N1(C(Cn2c(C)ncc2)=O)CCN2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CC(C)(C)C2CC2)CCC1C C12(C(=O)NCC3CCN(C(CC(C)P(C)(C)=O)=O)C3)CC3CC(C1)CC(C)(C3)C2 Cc1ccc(CNC(C2CC2C(=O)Nc2nc(C#N)cs2)=O)cc1[N+](=O)[O-] c1(C(=O)NC2C(C)N(C(c3cnc(O)n3C)=O)CC2)cnc2nc(O)ccc2c1 c1(C(=O)NC2CCC(NC(C3(CO)COC3)=O)CC2)cnc(O)c2cccnc12 CCCC(CC(C)C)C(=O)N(C1CCC(CNC(=O)C(C)OC)CC1)C C(=O)(C(C(F)(F)F)OC(C)=O)NCCN(C(=O)CC1CC1C1CC1)CC N1(C(CCN(C)C(C2CCC(N=[N+]=[N-])C2)=O)=O)CCC2(CCOC2)CC1 C1(CNC(c2cn(CCC)nc2C)=O)CC(N=c2[nH]c3c(C)c(C)ccc3s2)C1 C1(O)(CCNC(COCCCCC)=O)CCN(C(=O)C(C)(F)CC)C1 C1(C(N)=O)CC2(C1)CN(C(c1csc(C(C3CCC(O)C3O)=O)c1)=O)C2 C(CS(=O)(=O)CC(=O)NC1(C(=O)NCc2ccc(CO)cc2)CC1)OC C(=O)(CCCCCCC(=O)O)NC1CC(N(C)C(C)=O)C12CCCC2 C(=O)(C(C)(C=C)CCOC)NCC(C(=O)NCCCC(C=C)(C)C)OC Cn1cc(C(=O)NCC2CC(F)CN2C(c2csnn2)=O)c2cc(F)ccc12 N1(C(CC2CCN(CC)C2)=O)CC(N(C(c2nc(Cl)c(CC)[nH]2)=O)CC)C(O)C1 C(=O)(CC(C(C)(C)C)NC(=O)CC1CCCO1)NC(C(=O)OC)C N1(C(CN(CCC)C)=O)C(CNC(=O)CN(C)S(=O)(=O)N(C)C)CC2COCC12 c1(OC)cc(C(N2CCC3CCN(C(C4CC4F)=O)CC23)=O)c(C)cc1[N+](=O)[O-] C1(C(=O)NC(CNC(CCOC(C)=O)=O)(C)CC(C)C)CCc2nc(O)[nH]c2C1 CC1(CNC(=O)CCCc2cnccn2)CCCC1NC(c1ccc(Cl)s1)=O C1(CC(N2CC(C)C(NC(C3CC(C4CC4)C3)=O)C2)=O)CCCCC1(F)F N1(C(c2cccc(CC)n2)=O)CC2CCC(N(C)C(c3cc(O)ncn3)=O)C2C1 c1(C(N(CCN(CC(=O)NC(F)(F)C(F)(F)F)CC)CC)=O)cccc(C)c1 N1(C(C=Cc2c(C)ccnc2)=O)CC2(CC2)n2nccc21 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N1CC(C)CC(NC(C(COCC)C)=O)C1 CCC(O)C(C)(C)C(=O)N1CCC(CO)(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 c1(CC)cccc(C(=O)NC2CC(NC(=O)C(F)CC3CC3)C2)n1 c1(C(n2cc(C3CCCCN3C(=O)C(N)=O)nn2)C)ccc(F)cc1 CCC(C)(F)C(=O)N1CC(OCCNC(=O)COc2cc(C)sc2C)C1 N1(C(C(NOC)=O)=O)CC(CNC(=O)CN2CCC(O)CC2)CCC1C c1(C(CCC)C)n[nH]c(=NC(=O)N(C2CCCCC2)c2ccccc2)s1 CN1CC2C(CCCN2C(=O)CCCn2cc(-c3c(F)cccc3Cl)nn2)C1=O C1(C(C(=O)NCC(=C)C)N(C(C)C)CC)CCCC1(C)C Cc1n[nH]c(=NCCC(C)(C)NC(=O)C(C2CCOCC2)C)s1 CC(C(C)(C)C(=O)NCCN1CCNC1=O)NC(=O)Cc1ccccn1 N1(C(C=CCCC)=O)CCC(CC(=O)N(C)C(C2(C)CC2)C)CC1 CC#CCCCC(=O)NCC(CNC(c1ccccc1SCC(N)=O)=O)OC CP1(=O)CCN(CC(N2CC3(C2)CN(C(c2ncccc2Cl)=O)C3)=O)CC1 c1(C(=O)NCC(CC)(C)NC(=O)CCC2CCCN2C)cnn2c1CCC2 c1(C(=O)NC2CC3CN(C(C(C)(C)OCC)=O)C2C3)cc(S(C)(=O)=O)oc1C CC1=C(C(=O)NC2CCCCC2NC(C2CC(C(C)C)=NO2)=O)CCCO1 C1(NC(C(CCOC)C)=O)CCCC2CN(c3cc(C#N)nc(C)n3)CC12 C(c1cccc(OC)c1)=CC(=O)NCC1CC(F)(CNC(C(CC)C)=O)C1 N1(C(CCC)C)Cc2ccc(NC(=O)N(C)CC3CCC(=O)N3)cc2C1 c1(C(=O)Nc2c(-c3ccc(N(CC)CC)cc3)csc2)c(F)c(F)cc(F)c1F C1(N(C(C2(C)CC2(C)C)=O)CC)CCCN(C(c2cncc(N(C)C)n2)=O)CC1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(CCN2C(=O)C(C)=C(C)C)C1 c1(N(C(C)(C)C)C(c2sccc2C)C)ccc(OCC(=O)N(C)C)cc1[N+](=O)[O-] C1(NC(C2=CCN(C(C(CC=C)(C)O)=O)C2)=O)C2CCC(C2)C1(C)C c1(N2CC3(CC(CC(=O)N(C(C)(C)C)CCO)OC3)C2)c(N=[N+]=[N-])cnnc1O c1(CC(=O)NCCN(C(C=Cc2occ(C)n2)=O)C2CC2)ccc2ncsc2c1 CS(=O)(=O)c1ccc(O)c(C(N2CC3CC3(C(=O)O)C2)=O)c1 CC(C)(C#N)CCC(=O)NCC1CC(NC(C2CCCCN2C(N)=O)=O)C1 Cn1cnc2nc(N3C4CCC3C(CNC(C3(C)CCCCNC3=O)=O)C4)ncc12 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC12CC(C1)N(C(=O)CC(F)(F)C(F)F)C2 c1(C(C(F)(F)F)NC(C(C)=CC2CC2)=O)ccccc1C#N c1(C(=O)NCCC2(NC(C3=C(C)OCC3)=O)CCC2)ccc(S(N)(=O)=O)cc1 C1(NC(c2c(C)nncc2)=O)(CO)CCCN(C(C2(C#N)CCOC2)=O)C1 C=CCC(CC(=O)NCC(C)CC(=O)OC)NC(C1(C)CCN(C)C1)=O c1(C(C(=O)NC(C2(O)CN(C(C(C(C)C)CO)=O)C2)C)C)cc2ccccc2o1 c1(N(CC(CC)(C)OC)C)nc(=NCC(C(C)C)OCC)[nH]c2cc[nH]c12 c1(OCC(=O)NC2C(NC(C(C)c3cccs3)=O)C2)ccccc1C(F)F c1(C(=O)OC)c(C)noc1CC.C1(C(=O)O)CCC1(C)C(=O)NC1CN(C(CC)=O)C1 C12(C(=O)NC)COCC1CN(C(=O)CN(C)C(=O)C1CC1)C2.C1CCN1 c1(C(=O)NC(C)CN(C)C(c2ccn(C3CC3)n2)=O)ccc(N)cc1F c1(C(C(=O)Nc2ccc(Cl)cc2)N(C)C)n[nH]c2c(F)cccc12 S(=O)(=O)(c1ccccc1OC(F)F)N1CC(NS(CC)(=O)=O)C1 c1(-c2cn(C(C)C(=O)NCC3CN(C)C(=O)O3)nn2)ccc2cc(Br)ccc2c1 CC(C)C(C)(O)C(=O)NC(CNC(c1cc(-c2cccs2)on1)=O)CO c1(CC(=O)NC2CC3CN(C(C(C)OC)=O)CC2C3)coc2cc(CC)ccc12 C1(C(N2CC(C)C(CNC(=O)CCn3cccc3)C2)=O)CC2CCC1CC2 N1(CC)CCOCC1CC(=O)NCCC(C)N(C(=O)Cc1cnns1)C CC1CC2(CC(NC(=O)CC3CC4(CC4)CN3C(=O)C=CCF)C2)C1 Cc1ncc(C(=O)NC(C(=O)N(C)CC2CCCCC2O)C(C)(C)C)cc1C#N c1(C(=O)NC(C2CCN(C(=O)CCC3CCC(C(N)=O)O3)C2)C)ccc(F)cc1Cl CC1CC2CN(C(C3CCC(C)(C)OC3)=O)CC2N1C(=O)C(F)CC1CCOC1 c1(NC(c2ccco2)=O)ccc(N2CCOC2=O)cc1 N1(C(CCCC2CC2)=O)CCC2(C=C(C(=O)NC(CC3ON=C(CC)C3)=O)C2)C1 C1(OC)CC(CF)N(C(=O)CC(CNC(=O)CC2CCSC2)C2CCC2)C1 C(CCC(=O)NC(C)CN(C)C(C1CC1(C)C(F)(F)F)=O)OCCC CC1CN(C(=O)Cc2c[nH]nc2O)CCCN1C(C1OC2CCC1CC2)=O c1(NC(CCC=C)C)ncccc1S(=O)(=O)NC(c1cccc(F)c1C)C C1(C(=O)NC2(C(=O)NCCOCCOCF)CC(C)(C)C2)CC2CC1CC2=O N=c1[nH]c(=NCCOc2ccc(Cl)c(F)c2)[nH]c(=NC2CC3CCCCC23)[nH]1 C1(C(=O)NCC(CC)NC(=O)Cc2nc[nH]n2)CCCCC1C(C)(C)C c1(C(=O)NCCCOCCNC(C2(C(=O)OC)CCCC2)=O)c(C)ccc(F)c1N c1(C(N2CCC(C(N3CCC(Br)C3)=O)CC2)=O)ccccc1F c1(CNc2c(C(=O)OCC)cnn2C(C)C)cc(Cl)c(N)c(Cl)c1 C1(NC(=O)CCc2cnco2)CC2CC(NC(c3ncnc(O)c3Cl)=O)CC12 N1(C(C(CCCC)O)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(CO)C1 C1(NC(C2CCCCCC2)=O)CC2CC1CN(C(c1nc(Cl)sc1Cl)=O)C2 N1(C(C2(F)CN(C(C(C3CCCC3)OC)=O)C2)=O)CC2CCC(C1)C(=O)N2 N#CC1(C(N2CC3CC(CNC(=O)Cc4cc[nH]n4)C3C2)=O)CC12CCOCC2 c1(C(C)NCC(N2CCC(C(OCC)OCC)C2)=O)nc2ccccc2[nH]1 C(=O)(C(O)CC(C)C)NCC(C(=O)NC(COC)C)(C)C Cc1ncc(C(N2CC=CC2(C)C(N2CCC(OCCF)C2)=O)=O)n1C Cc1csc(C=CC(=O)NCCC(O)CNC(=O)C(Cc2ccsc2)NC=O)n1 c1(C(=O)NC2C(NC(CC3N(C)CCC3)=O)COC2)ccn2nccc2n1 N1(C(c2cccc(CC)c2N)=O)CC(C)(C)OCC1CNC(=O)Cn1cnnn1 CCC(O)C(C)C(=O)N1CC(F)CC1CNC(c1cnn(C2CC2)c1Cl)=O c1(CC(=O)NCC2C(NC(c3c(CC)cco3)=O)COC2)cccc(O)c1 CC1=NOC2(C1)CC(C(=O)NC1C=CCN(C(=O)CN(c3ccncc3)C)C1)C2 c1(C(=O)OC)nc(NC(C2CC2CF)=O)cnc1OC(C)(C)C c1(C(=O)NCC(C2CCOC2)NC(C(CC)(C)CC)=O)cc(S(N)(=O)=O)cs1 C1(CCCC)(COCC(C)(C)NC(C2CC2CNC)=O)CCCC1 c1(NC2(C(F)F)CC(NC(c3ccc(OC)nn3)=O)C2)nc(OC)cc(C)n1 c1(C(=O)NC2C(CC)CN(C(c3ccoc3C)=O)CC2)ccc(C)c(F)c1N N1(C(CN(CCOC)C)=O)CC(CNC(C2CCCN2C(=O)CC)=O)C(O)C1 N1(C(c2ncc(C)nc2)=O)CC2(CNC(c3c[nH]nc3C)=O)CC1CCO2 C(=O)(C(CO)C(C)C)N1C(CN(C(c2ccc(OC)cc2)=O)C)CCC1 N1(C(C(Cc2cn[nH]c2)NC(C2C=CC=CC=C2)=O)=O)CCC(C2CCCC2)C1 c1(NC=O)ccc(CCC(=O)NCC2C=CCN2C(=O)CC2CC2(Cl)Cl)cc1F C(=O)(CC1=CCN(C(C2(Cl)CC2C(C)=O)=O)CC1)NCC(CC(=O)OC)O Cc1nccc(C(=O)NC2CN(C(c3n[nH]c4c3CCC4)=O)C2)c1C c1(C(=O)NC(C(C)NC(C=CCCC=C(C)C)=O)C)ccc(Br)cc1N(C)C N12CCc3ccccc3C1CN1C(=CC=C([N+](=O)[O-])C=NC(CCC)C1=O)C2=O c1(C(=O)NCCC2N(C(C3CC(=O)NC3)=O)CCC2)cc2c(cn1)COCC2 C1(C(=O)NCC2CCCN(C(COCCCCC)=O)C2)CC2(C1)CC1(CC1)C2 Cc1c(CC(=O)NC2CCCC(NC(=O)CCn3ccccc3=O)C2)ncn1C C1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(F)(F)C2)CCCCC12CC2(F)F C1(CNC(c2c(COC)cc[nH]2)=O)COCCN1C(=O)CCC1C(=O)NN=C1C C1(C(C(N2C(CC(=O)N(CC(C)(C)C)C)CCC2)=O)=O)CCCCCC1 C12(NC(c3c(C)ncnc3)=O)CC(CNC(=O)C(c3ccccc3)C)(C1)OC2C C1(CC(=O)N(CCCC)C)C2CCC(C2)N1C(=O)CSCCOC C1(CCOC)(NC(=O)C(F)n2cccn2)CCN(C(=O)CCC2CC(C)C2)C1 c1(C(N2CC(CNC(CCSC)=O)C3C2C3)=O)cc(Cl)c2c(c1)OCO2 C1(C2(C(N(CC(CNC(COCC(C)C)=O)O)C)=O)CC2)CCCCO1 CCC(CC(C)C)C(=O)NC(CNC(c1cnn(CC)c1C)=O)C(C)C C(=O)(CC(C)C(=O)c1ccccc1)N(C1CCC1C(c1ccc(C)s1)O)C(C)=O C1(CNC(c2[nH]cc(CC)c2)=O)CCC12CCN(C(=O)C(F)(F)COC)CC2 C(=O)(C1=C(C2CC2C)N(C)C(=O)N(C)C1c1cc(C)cc(O)c1)OCC CCC(C(=O)NCC1C2CCC(C2)N1C(c1cc(C)cc(N)c1)=O)C(F)(F)F c1(C(N(C(C)CN(C(=O)Cc2ccc(CO)cc2)C)C)=O)cn(C)c(=O)nc1O C1(CNC(=O)C=CC2CCOC2)(CO)CCN(C(c2ccc(O)nc2)=O)C1 N1(C(CC#C)CC)CCC(C)(C2CC2)CC1 C1(CC(=O)N(C)CC2CCN(C(C3(C(F)F)CC(O)C3)=O)C2)CN2CCN1CC2 c1(N2CCC(CN(C(c3c(CC)nn[nH]3)=O)C)C2)ccc([N+](=O)[O-])c(OC)c1 C#Cc1cnc(C(=O)NCC2N(C(=O)OC(C)(C)C)CC2(C)C)c(C)c1.OCC Cc1cnc(-c2nc(CCCO)nn2C2(C)CCCCC2)c(C)c1 CC1CN(C(=O)C(Cc2cc[nH]n2)NC(c2ccoc2Cl)=O)CCC1CO CCN=C(NCC1(N2CCSCC2)CCCC1)NCc1cnc(N(C)C)s1 CC1(CNC(=O)C2=CCCO2)CCN(C(c2ccnc(C3CC3)n2)=O)C1 S(=O)(=O)(c1ccccc1S(=O)(=O)N1CC(c2ccc(C#N)nc2)C1)NC N1(C(COC(C)=O)=O)CCCC(C)(C(=O)NCC23CCCC2CCC3)C1 CCC(CCCO)NC(=O)C(N1CCCCC1CC(=O)NCCOC)=O N1(C(CCC(=O)NCCC)=O)C2CCC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 Cc1nc2ncccc2cc1CCC(=O)NNC(=O)c1cocn1 c1(C(=O)OC)ccc(C(=O)NCC2(O)CC(NC(C3(C#N)CCCO3)=O)C2)cc1 C12(CC(=O)NC(C(C(C)C)NC(=O)CNC(=O)C(F)(F)F)C)CCC(CC1)CC2 c1(C(=O)NC2CCC(NC(c3snc(C)c3N)=O)C2)c(C)cncc1C N1(C(C(Cc2ccco2)NC(C)=O)=O)CCCCCCC1C.C12CC(C1)CC(=O)N2 CCCCC(C(=O)N(CC(C)C(=O)NCCc1ccc(C)cc1)C)NC(N)=O c1(C(N2CC(NC(CCCC#C)=O)C2)=O)c[nH]c2cc(OC)c(OC)cc2c1=O CC(CCCc1ccccc1)C(=O)N1CCCC(C)(NC(c2ncn(C)n2)=O)C1 C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(C(C)C)N(Cc2cncnc2)CC1)=O c1(NC(CC2(O)CCN(C(c3nc(C)oc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCCN(C(CSCC=C)=O)CC)cnn2cnnc2c1 N1(C(c2cc(CNC(C3C(=O)NCC3)=O)sc2)=O)CC2C=CC1CC2 C1(NC(c2ccc(C(C)=O)o2)=O)CCN(C(c2ccncc2O)=O)CC1.C1(S)CC1 Cc1ccn2ncc(C(=O)NCC3CC(C)(C)CN3C(c3ccnn3C)=O)c2c1 CC(C)(O)C(F)CNC(=O)CC1(C)CCN1C(C1CC=CCO1)=O N1(C(CCC2CC(NC(c3ccc(=N)[nH]c3)=O)C2)=O)CCC2CCC(C1)S2 C1(CNC(c2c(C)ccs2)=O)CN(C(=O)CNC(C2CCC2)=O)C2CC12 c1(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(CO)CC2)=O)cc(F)c(F)cc1F N1(C(CC2(CC)CCC2)=O)CCSCC1CCNC(=O)Cc1csnc1C N1(C(C2(C)CC(=C)C2)=O)CC2(CCC2NC(=O)C(C2CCCCC2)O)C1 C=C(C)CC(C)C(=O)NCC1CCCN(C(c2c(CC)nc(C)n2C)=O)C1 c1(NC(c2ccc(O)cc2)=O)ccc(NC(c2cc(Br)c[nH]2)=O)nc1 C1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NCC)s2)=O)CCc2cncn2C1 CC1=CC(C)CN(C(=O)CC(CC2CC2)NC(=O)Cn2c(O)nnc2O)C1 c1(C(=O)NC(C)(CNC(=O)Cc2ccnc(Br)c2)CO)cc2n(n1)CCC2 c1(CC)nc2sc(C)cn2c1C(=O)NC1CC1CNC(C1CC1C#N)=O C1(OC)CN(C(=O)CCC(N)=O)CCC1NC(=O)CC1(CO)CC1 N1(C(C=C(C)c2ccco2)=O)CC2(CCC2)CC1C(=O)NC1CNC(=O)C12CC2 C1(C(N(CCC)CCC)=O)(CNC(=O)CC2C=NN(C)C2=O)CC(F)(F)C1 N1(C(C2(CCC)CC2)=O)CCC(C2CCCN(C(c3c(Cl)cccc3Cl)=O)C2)C1 Cn1ncc(C(=O)NCC2(C)CCN(C(=O)CNC(c3cccs3)=O)C2)c1N C12(C(N3CC(C)(NC(C4COC5(CCC5)C4)=O)C3)=O)CCC(CO)(CC1)CC2 C1(C(=O)NCC2(F)CC(CNC(=O)CCF)C2)CN2CCN1CC2 N1(CCC)CCC(CNC(=NCc2cc(C)on2)NCC(=O)NC)CC1 C1(NC(c2ccc(C)s2)=O)CC2CCC1(NC(=O)CCc1ccc(C)c(Cl)c1)C2 C=CC(CC)CC(=O)N1CCC(C)C(CNC(C23CC4CC2C3C4)=O)C1 Cc1nc(CC(N2C(C(=O)Nc3ccccc3Br)CC3CC23)=O)c(C)s1 c1(C(=O)NC(CNC(c2cccc(SCC#C)c2)=O)C)cccc(=O)n1C CCC(C(=O)N1CCC(NC(c2cnc(S)n2C2CC2)=O)C(F)C1)C(C)C c1(C(CC)C)nc(N2CC3(CN(C(c4cc5sccc5[nH]4)=O)C3)C2)cc(C)n1 N1(C(CC2(C)CCN(C(c3c(C)cnn3C)=O)C2)=O)CCCC(C)C1CO CC(CS(C)=O)C(=O)N1CC2CC1(CNC(=O)CCSCc1ccccc1)C2 c1(C(=O)NC2C(NC(C3(C)CNC(=O)C3)=O)C2)cc([N+](=O)[O-])c(Cl)cc1Cl Cc1c(C)c(C)c(S(=O)(=O)NC2c3ccccc3OCC2C)c(C)c1C N1(C(C2(CC=C)CC2)=O)CCC(N(C(=O)C=CCn2cncn2)CCO)CC1 C1(CNC(C=CSC)=O)CCCC(CNC(=O)C(C)n2ccnn2)C1 c1(CCOC)ncc(C(=O)N(C2(CNC(=O)CNC(C)=O)CC2)C)[nH]1 C(CC(F)(F)F)NC(=O)CN1CC(N(C)C(C2CC(F)(CO)C2)=O)C1 CC1CN(C(C2CN(C)CCN(C)C2)=O)CCCN1C(C1OCCN(C)C1=O)=O c1(OCC=C)ccccc1C(=O)NCC1(CNC(C2CCCC2(F)F)=O)CCC1 CC(CC(=O)N(C1CCN(C(=O)CC=CC(C)(C)C)C1)C)c1ccncc1 N1(C(C2CC(SC)C2)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)nc1C)=O)C2 C1(OC)(OC)CCC1C(=O)N(CCC(=O)N(CC(c1nn[nH]n1)C)C)CCO C1(NC(c2ccc(Cl)c(-n3nnnc3C3CC3)c2)=O)CCCNC12CCC2 C1(C2CCN(C(C=NOC)=O)C2)CCCN(C(=O)CC2(C)CC2)C1 C1(C)(C(N2CCC(C(=O)OC)C2C)=O)CCCN(CC2CCOCC2)C1 CC(C)C(C)C(=O)NCCC1(CNC(=O)C(C)Oc2cccc(F)c2)CC1 c1(SCC(N2CCC(NC(c3c(C)nns3)=O)C23CC3)=O)nnc2ccccn12 N1(C(=O)OC(C)(C)C)CCCC2(C1)CN(Cc1cccc(C#N)c1)CCO2 Cc1ccc(C(F)F)c(C(=O)NCC(C)N(C)C(C2CCN(C3CC3)C2=O)=O)c1 c1(C(N2CC(NC(CC3CC(=O)NC3)=O)C2)=O)cnc(C2CCCC2)nc1O C1(NC(C(CNC(C=Cc2c(C)cccc2)=O)O)=O)CC2(CCCCC2)C1 CC1CCCCC1C(=O)N(C)CC1(O)CN(C(=O)CS(=O)(=O)N(C)C)C1 Cc1nc(C(=O)NCC(C(C)C)NC(C2(O)CC2(C)C)=O)nn1C C(CC(=O)NC(C)C(=O)NCCF)N(C(=O)C(C)C1(O)CCC1)CC C=CCCCC(=O)N1CCC(N(CCC)C(c2cnccc2Br)=O)C1 c1(OC)ccc2c(C(=O)NC3(C)CN(C(c4cc(=O)cc[nH]4)=O)C3)ccnc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCSC1)NCCN(C)CCO C1(C(N2CC(O)(C(C)NC(c3cc(CC)on3)=O)C2)=O)CC(OC)C(OC)C1 c12cc([nH]n1)C(=O)N2.c1(CC(=O)NCCNC(C2CN(CC)C2)=O)cn(C)cn1 N1(CCCC=C)CC2CCN(C(=O)CCc3ccc(CCCC)cc3)CCC2C1 C(CC(C)(C)C(=O)NC1(CC(=O)NCC2(C)CCCOC2)CC1)OC N1(C(C(CN)OC2COC2)=O)CCC(OCCC(F)(F)F)CC1 C(=O)(CCC(CC)CC)NCCCC(CCC)NC(c1nc(C)ccc1O)=O C1(C(=O)NCCCN(C(=O)CCc2nnc(C)n2C)CC)OCCOC1C CCC(O)C(C)(C)C(=O)NCC1(F)CC(NC(c2cccc(SC)c2)=O)C1 c1(C(N(CCNC(CCn2ncn(C)c2=O)=O)C2CC2)=O)cnc2nccn2c1 N1(C(C=Cc2cnc(C)s2)=O)CCC(NC(C2CCCC(=O)N2C)=O)C(C)C1 N1(C(CCCC)=O)CCC(C(F)CNC(C2(C)CC=CCC2)=O)CC1 c1(C(=O)NCCN(C(=O)C(C)C(C)C)CC)cncc2n[nH]cc12 C(=O)(CN1C(=O)Cc2ccccc21)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O CN1CC2(CC2)CC1C(=O)NC(CC1CCCC1)C(N1CCC(O)(CO)C1)=O c1(N(C)C)ccc(F)c(CNC2CCC23CCCC3)c1F c1(NC(C2CCN(Cc3ccc(CO)o3)CC2O)=O)cccc2c(I)n[nH]c12 N1(C(C2(C(C)(C)NCCC#N)CC2)=O)CC(C)C1.CO CC1OCCC1CC(N1CC(C)(NC(CNC(C2CCC2)=O)=O)C1)=O c1(C(c2nnnn2C2CCCCC2)NCCOCCOCC)cnc(C)[nH]1 C#CC1(NC(=O)C(CCC)NC(c2cc(C)cc(F)c2)=O)CCC(C)CC1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C1(NC(c2c(C)cnc(F)c2)=O)CN(C(=O)CS(N)(=O)=O)C2CCCCC12 Cc1nccnc1C(=O)NCCC1CCC(NC(=O)C=Cc2cnc[nH]2)C1 Cc1c(C(=O)NC2CN(C(=O)C(=O)NCC3CC3)CC2C(F)(F)F)nnn1C C(CCCCC(=O)N(C(C)CNC(=O)Cc1sccc1Br)C)SC CC(C)(CF)C(=O)NCCC1CCN(C(c2ncc(C(F)(F)F)s2)=O)C1 C1(NC(=O)N(C(CCN(C)C)c2cccs2)Cc2ccncc2F)CC2C(C1)C2(F)F c1(-n2c(C(COC)NC3(CC)CC3)nnn2)ccc(Cl)cc1F c1(CNC(C2OCC(C)(C)OC2)=O)ccc2c(c1)CN(C(=O)C(O)C(F)(F)F)C2 C1(N(CC(=O)O)C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC2(CCNC2=O)CC1 c1(C(N2CCC(NC(=O)CC3CCCCC3(F)F)C2)=O)cnc2scnc2c1 C(=O)(CCC(=O)c1cccnc1)NC12CC(NC(CNC(CN(C)C)=O)=O)(C1)C2 C=C(C)C(CC(=O)NC1CN(C(c2cnc(C)s2)=O)CCC1C)OCC Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCC(NC(=O)C(=O)NCC(F)F)CC1 N1(C(C2N(C(C(CC#C)C3CC3)=O)CC2)=O)CCC2CCCC2C1 C1(NC(C(N2CCCCC2)C)=O)(CO)CCN(C(c2cccc(CO)n2)=O)C1 N1(C(C(CCC)OC)=O)CCC2(CC1)CN(C(C1CC(F)C(=O)N1)=O)C2 C1(NC(C2C(OC)CCC2)=O)(CNC(C2CC=C(C)CC2)=O)CC2CCC1CC2 n1(CCCC(=O)NCC(C)(C)NC(c2cnc(C3CC3)s2)=O)c(O)nnc1O N1(C(C2(C)C(CC)CCC2)=O)CCc2cc(O)c(S(=O)(=O)N(C)C(C)=O)cc2C1 CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)Cn2ncnn2)C1)OC C(c1ccc(F)c(F)c1)=CC(=O)NC(CCC)CCCNC(=O)C(C)(C)CSC C1(C(=O)NCCOC)CC12CC(NC(=O)COC1(C)CC1)C2 CC1CC(C(=O)N2CCC23CN(C(C2COCCN2C)=O)C3)=NO1 CCC(C(=O)N1CCC(C2CCCCN2C(=O)COCC(C)(C)C)CC1)C(C)C C(=O)(C(CCF)NC(=O)C(C)C1CCC1)NCC(=O)OC.CCCCO C1(CC(=O)N(C2C(OC)COC2)C)N(C(=O)CNc2ccccn2)CCC1(C)C CON1CCC(C(N2CC3CC(N(C)C(c4cnn(C5CC5)c4)=O)C2C3)=O)CC1 C(=O)(C(C)CC(C)CC)N1CCC(CNC(C2C(=C)C2)=O)C12CC2 c1(C(N(C)CC2CCN(C(CC(C=C)CC)=O)CC2)=O)cc2occc2n1C N1(C(c2c(C)noc2)=O)CCN(C(=O)CCc2cccnc2Cl)CC1C(C)C C#Cc1ccc(C(N2CCC(CC(N)=O)(NC(=O)C(CC=C)OC)CC2)=O)cc1 c1(CC(=O)NCC(O)C(=O)NC(CCO)C2CCC2)cccnc1O C(=O)(NNc1c(F)cccc1F)OC.C12CCC1(C)NC2 c1(C(=O)NCCC2CCN(C(C3C(C)OCC3)=O)CC2)cccc(C(F)F)c1Cl c1(C(N2CCC(C(C)(C)NC(C3C(CC)CCC3)=O)CC2)=O)ccc(C)cc1F N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(C3CCN(C)C3=O)=O)C1C2 C(=O)(C(O)C(C)(C)C)NC1CCN(C(CC(C)SC)=O)C1 CC1C(=O)CC1C(=O)NCC1CC(NC(=O)CCn2cnnn2)C1 C1(NC(C(CCF)NC(CCCCN(C)C)=O)=O)C(O)C2CCCC12 C(N=c1nc2c(ncn2C)c(NCCc2ncco2)[nH]1)c1cc(C)nc(C)c1 N#Cc1cnn2ccc(N(C(=O)CCCC(F)(F)F)C3CC34CCNCC4)nc12 Cc1cc(C(N2CC(CNC(=O)C(c3cscn3)N(C)C)C3(CC3)C2)=O)ccc1F N1(C(C(C)N(CCC)C(c2ccn(C)c2CC)=O)=O)CCCC2CC1C2(C)C N1(C(CCc2onc(C)n2)=O)CCC2CCC12CNC(c1cccnc1N)=O c1(C(C(=O)N(CCC(=O)NCCOCCC=C)C)C)ccnn1C C1(O)(C(=O)NCCCC(C)NC(c2ccc(OC)c(Cl)n2)=O)CCCC(C)CC1 C1(CNC(c2cc(OC)nn2C)=O)CC2COCC2N1C(=O)C(C)OC(C)=O CC1CCc2ncc(C(=O)NC3CN(C(C4C(C)(C)C4(C)C)=O)CC34CC4)n2C1 N1(C(CC2(N(C(c3cc(C)c(F)cc3)=O)C)CC2)=O)CCC2CN(C)CC2C1 c1(OC(C)C)cccc(C(=O)NCC(O)CNC(=O)C2=CCCOC2)c1F C(=O)(C1=Cc2cc(OC)ccc2OC1)NC1C(CNC(C(CC)CC)=O)CCC1 Fc1ccc2c(Nc3cc(-c4cnn(C5CCCCO5)c4)ccn3)ncnc2c1 CC(O)C(C(=O)NCCCN(CCCNC(=O)Cn1cccc1)C)NC(N)=O N1(C(c2cc(C)c(C(N)=O)cn2)=O)CC2CN(C(=O)Cc3ccsc3)CC2(C)C1 C1(C(N2CCC(C(C)NC(C)=O)C2)=O)(NC(C(F)=CCC)=O)CCOCC1 CC(C(=O)NC(C(=O)NCCNC(=O)C1CC1)C1CC1)S(N)(=O)=O c1(C(C)(C)C(=O)NCC2CC(NC(c3cncn3C3CC3)=O)C2)ccc(Cl)nc1 c1(CC)nc(C)c(C(=O)NC(C2(O)CN(C(c3ccc(CN(C)C)o3)=O)C2)C)s1 C1(=O)C(O)CN1C(=O)OC(C)(C)C.C=C(C)C(=O)NCC(C)NC(=O)OC C(CC(C(=O)N(CC(CO)(CO)NC(C12CCCCC1C2)=O)C)NC=O)SC N1(C(c2nc(C3CC3)cs2)=O)CCN(C(C2C=CCC2)=O)C(C2CC2)C1 C1(C(=O)NC2CCN(S(CC3(C(=O)O)CCC3)(=O)=O)C2)C2CC3C(C2)C13 N1(C(C=CCCC)=O)CC(CNC(=O)CC2CC2)C(O)C1 CC1(C)C2CN(C(=NCCCSC(F)F)NC3CC(c4ccccc4)C3)CC12 c1(OC)cc(Br)c(CN2CC3CC2CN3C(=O)CNC(=O)C2CC2)cc1O N1(c2onc(C3CCC(N)C3)n2)CCCC(c2nc(O)n[nH]2)C1 C#Cc1c[nH]nc1C(N1CCC(OCC(=O)NCCN(C)C2CC2)C1)=O c1(CC)n[nH]c(=NC2CC(CNC(=O)CC3(O)CCCOC3)C2)s1 c1(N(C(Cc2nc(CC)sc2)=O)CCNC(C2CCN2)=O)cnc(C)nc1 C1(C)(OC)CC(NC(=NCC2CC2)NC(C)(C)Cc2ccccc2)C1(C)C N1(C(c2cc(C)c(C)s2)=O)CC(C)CN(C(=O)CN2CCC(C)C2)CC1C N1(C(C(C)Oc2ccccn2)=O)CCC(NC(=O)C=CC2CCCC2)CC1 C1(C(=O)NC2CCN(CC)C2=O)CCN(C(=O)C=Cc2cc[nH]c2)C(C)C1 C1(C(=O)NC(C2(C)CCC2)CC)CN(C(c2cccnc2)=O)CC1C(C)C N1(C(c2nccc(OC)c2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1C(C)C C1(C(N2CCN(CC)CC2)=O)C2CC3C(C2NC(c2ccc(C#N)n2C)=O)C13 N12CCC(C3CCN(C3)C1=O)C2.CN1CCS(=O)(=O)CC1CSCCOC(C)(C)C N1(C(c2c(OCC=C)cccn2)=O)CCN(C(=O)COC2CCCC2)C(CO)C1 c1(C(C)C)ccc(SCC(=O)NC2CN(C(=O)COC3CC=CC3)CC2C)cc1 O=S(=O)(c1ccncc1Cl)NCc1ccc(-c2cccnc2)cc1 c1(CNC(C(C)N(C)C(c2cccn2C2CC2)=O)=O)ncn(C2CC2)n1 CC(C(=O)NCCCN(C)C(c1cn(C)nc1-c1ccccc1)=O)P(C)(C)=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCN(C(=O)CCCF)C(C)C1 N1(C(c2cc(Cl)no2)=O)CCC2C(CCCN2c2ncncc2Cl)C1 C1(O)(C(C)NC(c2cc(C)nn2C)=O)CCN(C(C2CC(F)C2)=O)CC1 N1(C(Cc2n(C)ccc2)=O)CCC2C(CCCN2C(c2ccc(C#N)cc2)=O)C1 C1(n2cc(CCCC(N3CC(C#C)C3)=O)nn2)CC2CC1CC2OC S(=O)(=O)(c1cnc(Cl)nc1)N1CC(C)(C(=O)Nc2c(C(=O)OC)cc(I)cn2)C1 c1(C(=O)NCC2CCN(C(CC(CCCC)O)=O)CC2)c(N)nn2ccccc12 c1(C(=O)NCCN(C(=O)CC2OCCC2C)CCOC)nnn2c1CCCC2 C1(NC(N(C2CCS(=O)(=O)C2)CC=C)=O)CCCCC1C(C)(C)C N1(C(C(F)=CC)=O)CC2(CCN(C(=O)CC(C)C(=O)c3ccc(Cl)cc3)C2)C1 c1(N(C)C)ccc(C(N2CC(C(=O)NCC3(C)CC3)C3CC23)=O)c(F)c1 Cc1cccc(-n2cc(CN3CCN(C(C4CCC(=O)NC4)=O)CC3)nn2)c1O N1(C(Cn2ccc(C)cc2=O)=O)CCN(C(c2cnc(O)cc2C)=O)CCC1C C1(C(N2CC(C=C)C(NC(=O)C(CCC)N(C)C)C2)=O)CCc2ccccc2C1 CC1(C)COC(C(=O)NCC(=O)NC2C=CCCC2)C1 C1(CCCNC(C2(CC=C)CC2)=O)CCCN1Cc1nc(CC(C)C)no1 c1(CC(=O)OC)ccc(NCc2ccnc(Br)c2)cn1 N1(C(CC2(NC(C(C)CC3CC3)=O)CC2)=O)CC2CCOC2C1 c1(C(=O)NC2(CC=C)CN(C(CSCC#C)=O)C2)c(OC)cccc1C c1(C(=O)NC2CC(NC(c3cc(C)cc(CO)c3)=O)C2)c(Br)cc(F)c(Cl)c1F Cn1nc(C(=O)NCC2CCCCCN2C(C2C3CCCOC23)=O)c(Cl)c1Cl C=CCCC(CC(C)C)C(=O)N(C)CCN(C)C(c1cn(C)nc1Br)=O C#Cc1cccc(C(=O)NCC2CC2NC(=O)C=Cc2ccc(Cl)cc2)c1C N1(C(c2ccc(S)cc2)=O)CC2CC1CN2C(c1c(Cl)cccc1Cl)=O C1(C(N2CCC(N(C(=O)CCc3ccc(Cl)s3)C)C2)=O)CCCC12CCC2 CC1=C(C(=O)N2CC(CNC(c3cnn(C)c3C#N)=O)C(C)C2)SCCO1 C(=O)(C1=CCCCC1)N(C)CCOCCCCN(C(=O)C(C1CCOCC1)F)C C1(NC(C)=O)CN(C(=O)CN(c2cncn2C)Cc2ccccc2)CC1O c1(C(=O)NCCCOCCC(=O)N(C(CC#C)C)C)ccnc(O)c1 C1(NC(c2cc(CNC(c3ccc(C(C)=O)[nH]3)=O)sc2)=O)CCC(C)CC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C3CC3)NC(C)=O)=O)C2)cccc(F)c1C N#CC1(C(N2CC(n3cc(CNCc4cc(=O)cc[nH]4)nn3)C2)=O)CCOC1 c1(N(C)CC)nc(=NCC2CSC2)[nH]c2cccnc12.c1(C)cccc2c1O2.OC C1(CNC(N2CCC(C)(CS(C)(=O)=O)C2)=O)CC2OC1C1CC21 C1(c2nnnn2C2CC2)(NCc2c(C)cccc2)CCC(C)(C)CC1C N1(C(CC=C(C)C)=O)CCCC2(NC(=O)CN(C)S(N)(=O)=O)CCCC12 C12(C(=O)NCC(=C)C)CCN(C(c3cc(Cl)n(C)n3)=O)CCC1C2 C=CCC(Cc1ccccc1)C(=O)NCCCNC(=O)C=C(Cl)Cl N1(C(C2CCN(CCC)CC2)=O)CCN(C(=O)C2=CCCC2)C(CO)C1 C1(NC(c2c(CC)ccc(F)c2)=O)CCC2(CCCN2C(c2cocn2)=O)CC1 N1(C(CC(C)CF)=O)CCN(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC2(CC2)C1 Cc1cc(C(F)(F)F)c(C#N)c(N2CCC3C(CCN3C(C3CCC3)=O)C2)n1 CC1(C)CCC(C(N2CCC(NC(c3csc(CO)n3)=O)C2(C)C)=O)OC1 N1(C(=O)Cc2ccc(Cl)cn2)CCCN(C(C2(CF)CC2)=O)CC1CO N1(C(c2cc(C)sn2)=O)CCCC(NC(=O)C(C)CC2CCC2)C1C C1(C(=O)NCCOCCNC(=O)CCC2CC(F)(F)C2)CCCC2CCCN12 c1(C(=O)NC23CCC(CNC(C4CNC(=O)O4)=O)(OC2)C3)cccc2ccnn12 C1(NC(COCCC)=O)CCC(N(C)C(c2cc(C3CCCC3)no2)=O)C1 Cn1c(C(=O)NC(CO)C(=O)NCc2cn[nH]c2)cnc1Cl c1(C(=O)NC2CC3CN(C(C(C)(C)C(F)F)=O)C2C3)csc2ncnc(O)c12 [N-]=[N+]=Nc1ccc(Cl)cc1NC(c1ccc(OCCF)cc1)=O Cc1nn2cc(CC(N3CCCC(CNC(c4oncc4C)=O)CC3)=O)nc2s1 Cc1ccc(F)c(CN2CCC(Nc3ccccc3)CC2)c1Cl C1(C(C)NC(CSCC(C)=O)=O)CCN(C(=O)Cc2nc(O)n[nH]2)C1 N1(C(C(=O)NCC(F)(F)F)=O)CCCC2(CCN(C(=O)Cc3cscc3F)C2)C1 CCC(CC)CC(=O)NCC1CCC(C)N(C(=O)C(c2ccccc2C)C)C1 CCCC(CCC)CC(=O)NC1CC2CN(C(c3cc(C4CC4)nn3C)=O)CC12 C1(OC)CN(C(c2cnoc2C2CCC2)=O)CC1NC(C1CCCC1)=O c1(NC(CCNC(C=Cc2cccc(C)c2)=O)C)ncnc2cc(F)c(F)cc12 c1(CCC(N2CCC(Cc3cn(C4CCC4)nn3)C2)=O)cnc2ccccc2c1 N1(C(=O)OC(C(C)(C)C)=O)CCN(C(N2CC(c3cnc(C)[nH]3)C2)=O)CC1 c1(C(=O)NCC(=O)NC2CC2CNC(=O)CC2CCC2)cccc(Br)n1 C1(CCC(C)C)CCN(C(C2CCCN2C(=O)CCOC2CC2)=O)CC1 CCC(CCC(=O)NC1(C2CN(C(C3CCCCC(=O)N3)=O)C2)CC1)OC CC1(NC(=O)CC2CSCCS2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(C(N2CCC(F)(CNC(c3coc(Cl)c3)=O)C2)=O)coc2ccc(Cl)cc12 C1(C)(OC)CC(NC(=O)C(F)CC2CN(C(=O)CC3(O)CCOCC3)C2)C1(C)C C(C(=O)NCCN(C(=O)C(O)Cc1ccccc1)C1CC1)(C(C)C)SC c1(CC(C(=O)NC2CN(C(c3nc(Cl)cs3)=O)C2)O)ccc(F)cc1 c1(C(=O)NCCC(CCc2ccccc2)NC(C)=O)ccc(C(C)C)cc1N N1(C(N2CCCC(N(C)C(=O)OC(C)(C)C)C2)=O)CCC2(CCC(C)(O)CC2)C1 C(=O)(CCC(F)(F)F)N1C(C(=O)Nc2n(CC)ncc2)CC(C)C1 N1(C(C(COC)C)=O)CCC(C2CCC2)(CNC(=O)Cc2nnc(S)n2C)CC1 N1(C(C(CCC)O)=O)CCN(C(C2(F)CCOCC2)=O)CC1CC C(c1nc(CC2CCCOC2)no1)=C(COCC)C(F)F N1(C(c2c(C)snc2)=O)CCOC2(CCCN(C(=O)C(F)C(C)C(F)(F)F)C2)C1 Cc1cc(S(=O)(=O)N2CCCC(C)(C(N3CCOC(C)C3)=O)C2)ccc1Br CP(C)(=O)CCC(=O)NCCn1cc(CNC(C2CC3CCC2O3)=O)nn1 C1(CC(=O)N(CCn2cc(CCS(=O)(=O)NC(C)=O)nn2)C)CC(O)C1(C)C N1(C(C2C(CC)C2)=O)CCC(CN2CCN(C(=O)C(C)(C3CC3)OC)CC2)CC1 N1(C(c2c(N)n(CCO)nc2)=O)CCN(C(=O)CC=C(Cl)Cl)C2CCCCC2C1 C1(C(C)NC(=O)CCOCC2CC2)CCCCN1C(=O)CC1CCOCC1 C1(OCC)CC2CN(C(=O)C(CC(C)C)N(C(=O)CC3CCC(C)(C)O3)C)CC12 C1(N(C(C2(CCOC)CC2)=O)C)CCN(C(=O)C=C2CCC(C)C2)CC1 C(C(=O)NCC1=CCCOC1)(C(C)C)NC(C(COC)C)=O c1(C(=O)NCC(C)NC(C2(COC)CCCCO2)=O)cc(C)ccc1O N1(C(c2c(NC)ccc(F)c2)=O)CCC2CC1CN(C(=O)CCC=C(C)C)C2 C1(NC(=O)CC2C=CCCC2)CCC2(CC1)CN(C(=O)C(=O)NCC(F)F)C2 c1(CC(=O)NCCCCCCn2cc(C(C)NC)nn2)nnc2n1CCOC2 C1(NC(C2N(C(Cn3ncc(C)c3)=O)CC=CC2)=O)CN(C)CCC1O N1(C(C)=O)CCCOC(COC(c2nc(CS(C)(=O)=O)cs2)=O)C1 S(=O)(=O)(CCCCCS(N)(=O)=O)NCCC1C(C)(C)NCC1 C1(C(N2C3C(NC(=O)CC4CCS(=O)(=O)C4)C(C3)C2)=O)CC12CCOCC2 C=CC1CCCCN1C(=O)COC1CC(NC(c2ccccc2CCOC)=O)C1 C=CC(C)C(C)C(=O)N1CC2(NC(=O)Cn3ccccc3=O)CC1(COC)C2 c1(C(N2CC(COC)N(C(c3nccn3C)=O)CC2)=O)ccc2c(c1)COCO2 C(=O)(CC(O)C(C)(C)C)OC(C(=O)N(S(=O)(=O)c1cccs1)C(C)C)C c1(C(=O)NCC(C)(C)CNC(=O)C(CC(F)F)C2CCC2)ccc(N)cc1F CC(F)(F)CCCC(=O)NCC1CC(NC(c2cccnc2O)=O)CC1O C1(CNC(c2cc(CC(C)C)on2)=O)CN(C(=O)CN(C)C(=O)C2CC2)CCO1 O=C(N=c1ccn(C2CN(Cc3ccc(I)c(F)c3)C2)[nH]1)c1c(F)ccnc1Cl c1(CC(=O)N(C)CC2(NC(c3ccnnc3)=O)CC2)nc(F)c(F)cc1F C1(C(=O)NCC23CC(NC(C4SCCCS4)=O)(C2)C3)C2Cc3ccc(Cl)cc3C12 C1(CNC(C(c2ccccc2)OC)=O)CCN(c2ncc(F)cn2)C12CCC2 N1(CCCC)CC2CCC1C(NC(=O)C(C)Oc1ccc(OC)cc1)C2 CS(=O)(=O)c1cccc(C(N2CC(NC(c3ccnc(Br)c3)=O)CC(F)C2)=O)c1 N1(C(Cc2cc(C)on2)=O)CC(C2CN(C(=O)CC3SC4=NCCN4C3=O)C2)C1 CC(C(=O)N1CCC(O)(CNC(C2CCC3(CCC3)C2)=O)CC1)C1=CCCC1 Cc1nn(C(F)F)c(C)c1S(=O)(=O)N(C)CC1CCCCO1 C1(CCS(C)(=O)=O)COCCN1C(=O)Nc1ccc(Br)cc1 C1(C(=O)NC2C(NC(c3ccc(F)c(Cl)c3F)=O)C2)CCc2cc(F)ccc2O1 C1(NC(CCCC#C)=O)CCc2nc(NC(c3cc(F)cc(Cl)c3)=O)sc2C1 CCC(C)(COC)CNC(C12CC1CCN2C(=O)CNC(C1CC1C)=O)=O C1(NC(C2CCC(F)(F)CO2)=O)CC2(C1)CN(C(=O)C=Cc1cncs1)C2 C1(C(N2CC(SC)C(N(C)C)C2)=O)N(C(=O)CN2CCCCC2)CC12CCCC2 c1(CC(=O)N(CCC(C)NC(=O)Cn2ncnn2)C)csc2ccccc12 C1(C(N(CC(=O)N(C)C)CC)=O)CN(C(=O)Cc2cnoc2)CC1(F)F Cn1ncc(C(N2CC(F)(CNC(=O)CCCOC(C)(C)C)C2)=O)c1F N1(C(c2c(C)scc2)=O)CCC2CN(C(c3cnc4n3CCS4)=O)C2C1 c1(C(C)C)nc2c([nH]1)CC(C(=O)N(C(C)CNC(=O)CN1CCSCC1)C)CC2 c1(C(N(C(CNC(c2cnc(C)nc2C)=O)C)C)=O)scc2c1OCCO2 c1(C(N2CCCC(C(C)Nc3cn(C)nn3)C2)=O)cccc2ncnc(O)c12.C CC1(C)CC(NC(C2CC3CC2C2CC32)=O)CN(C(c2ccnc(Cl)c2)=O)C1 c1(C(N2CCC(NC(=O)NC(C(=O)OC)C)C(O)C2)=O)ccc2ccccc2n1 O=C(C1=CCCS1)NC1CCN(C(C2CCNCC2)=O)CC1 C(=O)(C1Cc2ccccc21)NCC(C)NC(c1cc(C(=O)OC)no1)=O c1(C(N2C3(COC)CC(NC(C4CC4C)=O)(C2)C3)=O)cc(S(C)(=O)=O)ccc1O c1(C(N2CC(CCNC(=O)CC3CCCC3)(OC)C2)=O)cn(C)c(=O)n1C c1(C(c2cccc(Oc3cnccn3)c2)OCCCC(C)C)cccc(Cl)c1Cl C1(CC(=O)NCCCSC)C2CCC(C2)N1C(c1ncccc1CO)=O c1(C(=O)NCCCNC(=O)COC(F)F)cc2c(nc1O)CCCCC2 c1(OCC(=O)NCC2C=CCN2C(=O)CSCC(F)(F)F)ccc(F)cc1O C1(CNC(c2snc(O)c2Cl)=O)CCCC(CNC(=O)C(F)(F)C2CC2)C1 CC1CC(C(=O)N2CCC(CC(N3CC(n4ccnc4)C3)=O)C2(C)C)=NO1 c1(C(N2CCC(CNC(C(C)(C)CO)=O)C2)=O)cnn2cc[nH]c12 c1(C(N(C(C)CNC(C2(C(F)(F)F)CC=CCO2)=O)C)=O)cc(F)c(F)cc1N C1(C(=O)NC(COC(C)=O)CO)CC(C)CN1C(c1cc(C(C)C)[nH]n1)=O CC1CCN(C(c2c[nH]ccc2=N)=O)CCN1C(c1cc(F)n(C)n1)=O N1(C(C=C(C)C)=O)CC(C)CCC1CNC(c1cc(C)nn1C)=O c1(NC(C2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)cccc(Cl)c1C c1(C(=O)NC(c2ccco2)CO)ccc(-c2ccccc2F)cc1 C1(C(N2CCN(C(CC)=O)CC2)=O)(NC(=O)CC)CC2(CC2)C1 Cc1cc(C(F)F)nn1CC(=O)NC(CNC(c1ccc(C(N)=O)[nH]1)=O)CC(C)C C1(OC)CCCN(C(C2CC3CCC2O3)C(=O)NCC(C)C)CC1 CCC(C(=O)NCC=CC(=O)N(C)CC1(CO)CC1)C(C)C n1(C2CCN(C(C3C(c4onc(C)n4)C3(C)C)=O)C2)cnc2ccccc12 c1(C(=O)NCC(C2CC2)NC(C2CN(C(C)C)C2)=O)cnn(C2CC2)c1 C(c1cncn1C)=CC(=O)N(C1CN(C(C2(Oc3cnn(C)c3)CC2)=O)C1)C C1(CCC(=O)NC2CC(CNC(C3(CS(N)(=O)=O)COC3)=O)C2)CC2CCC1C2 C1(CNC(Cn2c(C)cc(C)n2)=O)CCCCCN1C(=O)C(F)CC1CCC1 N1(C(C2(OC)CCCC2)=O)CC2C(NC(=O)C=C3CCCCC3)C2C1 c1(C(=O)NC(C2CN(C(C=C(C)C)=O)C2)C)nn(C)c(C(F)(F)F)c1Cl c1(NC=O)nc(CC(=O)N(C2CCN(C(C3CC3C(F)F)=O)C2)CCO)cs1 C#CC1(C(=O)NCCCCC(=O)OC)CCN(OC(C2CC2C2CC2)=O)C1 C1(N(C(=O)CCOC2CCCOC2)C)CCCC(NC(=O)CSc2cccnc2)C1 C=CCC(CNC(c1ccn(CCC)n1)=O)C(=O)NC1CC(CC)C1 N1(C(C(C)(C)C#N)=O)Cc2ccc(CNC(=O)C=CSc3ccccc3)cc2C1 CCCCC(C(=O)N1CCCC(CO)CC1)NC(c1cc(=N)[nH][nH]1)=O CN=c1nc(C(N2CCC(O)C(NC(=O)CC3CCC4CC34)C2)=O)cc(C)[nH]1 c1(C(=O)NCc2cn(CC(=O)N(C(C)COC)CC)nn2)cnn2cccnc12 c1(C(=O)NCCC(C)N(C(C2=CC(C)(CC)C2)=O)C)cn2cnnc2cn1 c1(C(=O)NCC2C(NC(=O)C=Cc3cn[nH]c3)C2)ncc2n1CCCC2 C(=O)(CCCCCC#N)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO Cc1nc(CO)sc1C(=O)NCCCCCC1CCN(C(=O)CC#N)CC1 C1(CC2CC2)CC12CCN(C(=O)CC13CCCC1C3)C2.Cc1cc(C)n(CC(=O)N)n1 N1(C(C)=O)CCCC(C(N2CCN(C(=O)CNC(=O)CC3(CO)CC3)CC2)=O)C1 N1(C(C2N(C(N)=O)CCC2)=O)CCN(C(=O)CNC(C2CCC23CCC3)=O)CC1 S(=O)(=O)(c1ccc(-c2ccc(O)c(C3C(CC)CN(CC)CC3)c2)o1)NC(F)(F)F C12(C(=O)NCC(CC=C)NC(=O)C(C)Oc3cccc(Cl)c3)CCN(CC1)CC2 c1(N2C(C)CC(CNC(CCCC(=O)NCCC)=O)C2)ncnc2cc(Br)sc12 N1(C(C(CCC)CCC)=O)CCC2(CO)CN(C(=O)C(=O)NC(C)C)CC2C1 C=C(Cl)CCC(=O)NC1(C(=O)N(CCN2CC=CC2)CC)CC(CO)C1 c1(OC)ccc(C)c(C(=O)N(C(CNC(=O)C(C2CC2)C2CC2)C2CC2)C)c1 c1(C(N2C(CCNC(C(=O)NC3CC3)=O)CSCC2)=O)cccc2occc12 CCCCC(CC)CC(=O)NC1CCCN(C(=O)CSCc2ccccn2)CC1 C1(CN(C(C2(C(C)C)CCOC2)=O)C)CN(C(=O)C(F)(F)CN(C)C)CCO1 c1(C(N(CCCN(C(c2nc(CC)sc2)=O)C)C)=O)cc(SC(F)(F)F)oc1C C12(C(=O)NC3(CN(C)C)CC3)C(NC(=O)CC3CCOC3)C3CC1C2C3 C(N=c1nc(N2CCCC(C)C2)c2sccc2[nH]1)c1cccc(OC)c1C c1(N(C)C(=O)Oc2ccccc2)ccccc1CN1CC2CC1CO2 CCCC(C)(O)C(=O)NCCCOCCOCCNC(=O)CSc1cnn(C)c1 C(C(F)(C(=O)N1CCC1(C)C(=O)N(C)C)C(C)C)NC(C(C(=O)OC)C)=O C1(NC(c2c(C(C)C)cccc2)=O)CCCC2CN(C(C3CC4(CC4)C3)=O)CC12 Cc1c(Br)cc(C(=O)NCCCCNC(C2(C)CC(C)C2)=O)c(=O)n1C CCCCCCN1CCC(CC(=O)ON2CCCC2CC(=O)NCC(=O)NC)C1 C(=O)(CC(C)C(C)(C)NC(N1CC(C)C(F)(F)C1)=O)OC N1(C(CCC(C)=O)=O)CCC2(CC1)CN(C(c1cnn(C)n1)=O)CCO2 C(=O)(CS(=O)C(F)(F)F)NCCC1CCN(C(C2C(CC)N(C)CC2)=O)CC1 c1(CNC(CC2C(C)(C)C2)=O)ccc(CNC(C2CCCOCC2)=O)cc1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(O)(CNC(=O)C(O)CSC)C1 N1(C(c2c(C)scc2)=O)CCC12CN(C(C1CNC(=O)CC1C)=O)C2 N1(C(C2(CC)CN(C(=O)CN(C)C(C)C)C2)=O)CC2(CCOC(=O)N2)C1 C(CCC(=O)NC1(C(=O)NOCCF)CCSC1)OCCOC C1(C(N(CCCCNC(Cc2cc(C)no2)=O)C)=O)CCCC(CF)C1 N1(C(CC2(OC)CC2)=O)CCC(O)(C(C)NC(=O)Cc2cc(C3CC3)no2)CC1 c1(C(N2CCC23CN(C(c2cscn2)=O)C3)=O)cnc(Cl)cc1Cl c1(C(N2CC(NC(Cc3cc(C)n(C)n3)=O)C(O)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1ccc2ncc(C(N3CCC4CN(C(c5cnn(C)n5)=O)CCC34)=O)n2c1 N1(C(=O)C(F)OC(F)(F)F)CC2(C(=O)NCC3CCCSC3)CC1CO2 c1(C(=O)NC2CCC(NC(=O)CSc3ccccc3Cl)C2)cccc2nncn12 CCC(CC)CCC(=O)NC1CCC1NC(C1(Br)CC1)=O Cc1ccc(C(=O)NCC2CCCCC2NC(C2OCCCO2)=O)c(Br)c1 c1(C(=O)NCC2CC(NC(C3CCC=CCCC3)=O)C2)ccc2cnccc2c1 C(=O)(CCC(=O)N(C)CCN(C)C(c1c[nH]nc1Cc1ccccc1)=O)N(C)C c1(CC(=O)NC(C)CN(C(=O)C=CBr)C)cc(C(F)(F)F)n(C)n1 N1(C(c2nc(OC)oc2)=O)CCC(NC(=O)Cc2cccc(Cl)c2OC)C(C)C1 N1(C(CN2CC(C)(C)C2)=O)CCCC(NC(c2coc(O)n2)=O)CC1 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)NC(CC(C)(C)C)c1cccnc1 C1(C(N2CC(OC)(CNC(=O)C(C)CC(F)F)C2)=O)CC2CCC(C1)C2O c1(C(N2CCC(C)(CCNC(c3c(SC)n(C)nc3)=O)C2)=O)cc2n(n1)CCO2 c1(C(=O)NC(CC)CNC(C2(C)CCOC2)=O)nc(Br)c2n1CCCC2 C=CCCCCCCCCC(=O)NC(CNC(C1CCCN1N=O)=O)CCCC c1(C(N(CCC)Cc2cccc(C3CC3)c2)=O)cc(C2CC2)ncc1Br N1(C(C(C)Cc2ccco2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(NC(C2(F)CCN(C(=O)C=Cc3cnccn3)C2)=O)cnc2ccc(Br)cn12 N1(C(c2c(C#C)c[nH]n2)=O)CCN(CCNC(=O)C(O)CCSC)C2(CCC2)C1 c1(C(C)=O)cc(C(=O)NCC(C)(C)NC(=O)CC2CC2(Cl)Cl)co1 N1(C(C2CCC(C(C)C)CC2)=O)C2CCC1CN(C(C1(C)CC3CC3C1)=O)CC2 C1(C(=O)NCC2CC(F)(CNC(CCC=CCC=C)=O)C2)COCCN1C C(=O)(C(CCC(C)C)NC(c1ncccc1F)=O)NCc1nc(C)sc1C CC(CC(C)(C)C#N)Nc1c(C(N)=O)c(C(F)(F)F)nn1C C1(CC)CCCC1(C)C(=O)N(C)CC1COCCN1C(=O)CSc1n[nH]c(O)n1 N1(S(C(C)C)(=O)=O)CCC(F)(C(N2CCN(c3cc(Cl)ccn3)CC2)=O)C1 c1(C(=O)NCC2CCN(C(c3ncncc3F)=O)C2)c(F)cccc1Br c1(C(=O)NCCN(C(Cc2cc(COC)on2)=O)C)cccc2nnn(C)c12 c1(-c2onc(C(=O)NC3C(CNC(C4CC(SC)C4)=O)C3)n2)cccc(F)c1 C1(O)(CN(C)C(C2CC2Cc2ccccc2)=O)CN(C(C2CC(C)(C)C2)=O)C1 N1(CC)CCOC(C(=O)N(CC(CO)(CO)NC(C2CC(F)C(=O)N2)=O)C)C1 C1(NC(c2c(C)oc(CNC(=O)C(C)CC3CCC3)n2)=O)CCCCC1(C)C C1(CCNC(=O)Nc2cnc(-n3cccn3)o2)CCCC12CC2 N1(C(C2(NC(CCCN(C(C)C)C)=O)CCOCC2)=O)CCOC2CCOCC12 FCCN=C(NCc1cc(Cl)ns1)NCc1nc(C2CCCCC2)no1 c1(OC)cccc(C(Cc2ccc(F)cc2)NC2CCOC2)c1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)CC4)C2)nc(C)c1 c1(CNC(c2ccc(-c3ccc(CN)cc3)o2)=O)ccc2ncccc2c1 c1(NC(C(CC(C)C)ONC(C2COCC(C)O2)=O)=O)cccc2ccncc12 C12(C(N3CCC(COC)(CNC(c4ccoc4)=O)C3)=O)CCC(C)(CC1)OC2 C1(CC(N2C(c3ccc(C)o3)COCC2)=O)CCC2CNCCC2C1 c1(C(=O)NCC2CCC2NC(c2cnc(C3CC3)[nH]2)=O)ccc(OC(F)F)nc1 CCCC(C(=O)NC12CC(NC(=O)C(C(=O)OCC)N(C)C)(C1)C2)N(C)C c1(C(=O)NCC(C2CCCC2)NC(CC(=C)C)=O)c(S(C)(=O)=O)cnn1C C1(CN(C(=O)CC2CCC2)C)CN(C(=O)CC2(c3ccccc3)CC2)CCO1 CCC(F)(F)CC(=O)N(C1CCCCC1NC(C1C(Cl)(Cl)C12CC2)=O)C c1(CCC)cc(C(=O)NCC2(CNC(=O)CCC(C)N(C)C)CC2)cc(O)n1 N1(C(CN(C(CSCC=C)=O)C)=O)CC(F)(F)C(F)(F)C1 c1(C(N2CCCC(NC(c3cncnc3)=O)C(F)C2)=O)cc2c(s1)CCCCC2 C(C(C)CC(=O)NCc1cc(NC(=O)OC(C)(C)C)cn1C)OC C#Cc1ccc(NC(=O)C=C(C)CNC(c2ccc(C)nc2O)=O)c(C)c1 N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1C(=O)NOCCC1CC1 N1(CC(N2CC(C(C)NC(=O)C(c3ccc(Cl)nc3)(C)C)C2)=O)CC(=O)NC1=O N1(C(C2(CC)CCOCC2)=O)CCC2(CC(NC(c3sc(C)c(C)c3C)=O)C2)C1 CCCCC(C)CCC(=O)N1CC2CC1CN(C(c1cnn(C(C)C)c1N)=O)C2 C1(NC(C(C)N(C)C)=O)C(C)CCN(C(c2cc3ncccc3[nH]2)=O)C1C c1(OC)cc(OC)cc(CC(N2CC(NC(c3ccc(F)cc3)=O)C(C)C2)=O)c1 c1(NC(C2CN(C(c3c[nH]nc3C(F)F)=O)CC2F)=O)cc(Cl)cnc1O N1(C(c2c(C)cc(F)s2)=O)CCC(CO)(NC(c2ccc(O)nc2)=O)CC1 N1(C(C2(CC)CC2)=O)CC2CCCC(CNC(C3CC(F)C3)=O)C2C1 c1(N2CC(NC(c3nc(CC)oc3)=O)C(C)CC2)nc(C)nc2n[nH]cc12 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2(CC)CC2)=O)o1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 C(=O)(CCCCCCCC(=O)N(CCCNC(=O)CC1(C)CCCCC1)C)OC C(=O)(C#CC1(C)CCCO1)NC(C)(C)C.CC12CN(CCO1)Cc1nc[nH]c12 C(=O)(C(=O)C=Cc1cccs1)NCC(C)N(C)C(c1ccnn1C)=O C1(C(N(CC=C)CC=C)=O)CCC(n2cc(C3CCN(C)C3)nn2)C1 c1(CN(CC(=O)O)C(C)=O)ccccc1Br.c12cn(cn1)C1CN(C1)C2=O C1(CCCC)CN(C(C2CC(C(F)F)(OC)C2)=O)CCN1C(=O)C(C)N(C)C CC1CC(C(N2CCOCC(C(=O)NC3(C4CC4)CC3)C2)=O)CC(C)C1 C#CCCCCC(=O)NC1CCC(CNC(=O)C(C=C)c2ccccc2)C1 c1(CC(N2CCC(N(C(=O)C(F)n3cccn3)C)CC2)=O)cnn2c1CCCC2 N#Cc1cc(C(=O)NCC2(F)CCN(S(=O)(=O)C(Cl)(Cl)Cl)CC2)ccc1O c1(C(=O)NCC(CO)NC(C(CCC)CCC)=O)c(C)ccc2nonc12 C1(C(=O)Nc2cccc(NC(CCCCOCC)=O)c2)Cc2cc(C)ccc2O1 c1(C(N2CC(CC(=O)NCCC(C)CO)OCC2)=O)ccc(C#N)cn1 CCC(CC(=O)NCC(C)(C)CNC(C1(N(C)C)CC1)=O)C1CC1 O=C(CCC1CCCC(=O)N1)NNc1ccc(C2CC2)nn1 C1(C(=O)NCCCN(C)C(=O)OC(C)(C)C)CNC(=O)C1.c12c[nH]nc1CNC2=O c1(NCC2CC(NC(C)=O)C2)ccc(S(=O)(=O)N2CCOCC2)cc1 C(=O)(CC(C)(C)C(=O)N1CC(C)C1C(N1CC2COC(=O)C2C1)=O)OC c1(C(=O)NCCCNC(C2CCC2)=O)cccnc1-c1ccccc1 N=c1[nH]c2ncc(C(=O)NCC#CCNC(c3ccc4sccc4c3)=O)cc2s1 Cc1ccc(OCC(=O)NCC2(O)CCN(C(C3(C)CC=CC3)=O)C2)c(F)c1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(NC(=O)C(C)(C)CCF)C(O)C1 C1(CNC(c2c(C)n(C(C)C)cc2)=O)CC2(C1)CN(C(=O)C=CC(F)(F)F)C2 CC1(C)CC2(CN(C(C3CN(C(C4CCC4(F)F)=O)C(C)(C)C3)=O)C2)C1 S(=O)(=O)(c1ccc(NC2C=CCCC2)cc1Br)N1CCCC(C)(CCC)C1 Cc1c(CC(=O)NCC(C2CC2)NC(C2CC3CC3C2)=O)nc(Br)n1C Cc1nc2cccc(C(N3CCCCC(N(C(=O)C(C)CF)C)C3)=O)n2n1 c1(CNCCC(C)N(C)C)cc(Br)ccc1Br C1(NC(C=CC)=O)CCC12CCN(C(c1c(F)ccc(Br)c1F)=O)CC2 c1(C(=O)NC23CC(C(=O)Nc4c(C(=O)NC)cccc4)(C2)C3)cc(Cl)ccc1I N#CCCCC(C(=O)Nc1cccc(-c2ccco2)c1)N1CC2CCCC(C1)N2 c1(C(=O)NCCN(C(=O)Cc2cccnc2Br)CC)c[nH]c2cc(C)ccc12 N1(C(CCC=CC(C)C)=O)CCC2(CC1)C(N(C(=O)CC(C)(C)O)C)CS2(=O)=O CC1CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C(=O)NCCCc1cnn(C)c1 Cc1cnc(CNC2CCCCC2C(=O)Nc2ncc(Br)cc2C(F)F)cc1Br N1(C(C(CC)(F)F)=O)CCC(CNC(=O)Cc2ccc(C)o2)C(C)C1 N(C(=NCCCCc1ccccc1)NC(c1ccccc1)C)C1CN(CC)C1 c1(C(=O)NC2(C)CCN(C(C(CCSC)O)=O)CC2)cnnc2ccccc12 Nc1cccn(CC(=O)N(c2cccc(F)c2)C2CCC2)c1=O Cc1[nH]cc(C(=O)NC2CCCCC2NC(=O)CCC(N)=O)c(=O)c1Cl c1(C2(C(=O)OCCCSC)CC2)ccc(Br)cc1 N1(C(C2(CSC)CC2)=O)CC(C2CCCCN(C(=O)CC3CCCO3)C2)C1 c1(CC)cc(C)ccc1C(=O)NCC(CNC(c1ccccc1CC#N)=O)OC c1(C(N(CCNC(=O)C(C)(O)C2CC2)CC)=O)snnc1C1CC1 c1(N2CCC(CC(C)=O)CC2)cc(C)nc(NC(c2nc[nH]n2)C)n1 c1(C(c2n(CCC)nnn2)NC(c2ccc(Cl)s2)CC)ccc(OCC)nc1 C#CCCN=C(NCCCN=c1cc[nH]cc1)N1CCC2(CCCN(CC)C2)C1 CCC(C)C(CNC(=O)C(F)CC1CN(C(=O)Cn2ncn(C)c2=O)C1)CO c1(OCC)cc(C(N2CSCC2C(=O)NCc2cc(Cl)no2)=O)on1 c1(C(N(C2CCC(NC(CCc3c(C)ncs3)=O)C2)C)=O)cnc(C(F)F)nc1 N1(C(C=CC(=O)OCC)=O)CCN(C(c2ccc(SC(C)C)cc2)=O)C(C)C1C c1(CN(C(c2ccc(C(=O)OC)s2)C(=O)NCCC2CC2)C)cn(C)nc1C C1(O)(CNC(c2csnn2)=O)CCN(C(=O)C(F)(F)Sc2ccc(F)cc2)C1 c1(CCC(=O)NC(C)CC2CN(C(=O)CCC3CC3(Cl)Cl)C2)cn(C)cn1 c1(CC(=O)NC(CNC(CC2(COC)CCCC2)=O)C)nncnc1O c1(OC)cccc(NC(=O)NCC(C(C)(C)C)NC(=O)OC(C)(C)C)c1[N+](=O)[O-] C=CCC(C(=O)N1CCC1CNC(c1cnc(CC)[nH]1)=O)NC(C)=O C1(CN(C)C(C2(n3cc(CN)nn3)CC2)=O)COCCN1CCF Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC(C)CCC2CC2)ncc1N CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)CCc1ccc(Cl)s1)C2C c1(C(N2CCC(NC(C=NOC)=O)C2)=O)ccc(C)c(F)c1 C1(NC(CN(CCOC)C)=O)COCC1NC(=O)COCC1CCCOC1 N12CCOCC1CC(=O)NCCn1cc(cn1)C2=O.C(C(C(=O)OC)OC)SC.CC Cc1cccc(O)c1C(N1CC2(CCC2NC(c2cnn(C)c2)=O)C1)=O CC(CCCNC(=O)CCc1ccoc1)NC(=O)COc1ccccc1 c1(C(=O)NCC(C)Oc2ccccc2Cl)cncc2n[nH]cc12 c1(NC(C)C)ccc(C(=O)NCCCCCNC(=O)CC2(O)CCC2)cn1 n1(CC(N2CC(C)N(C(=O)C3=C(Cl)CCC3)CC2)=O)ccc(=O)c2ccccc12 c1(OC)ccc(NC(c2cccc3ncn(C)c23)=O)cc1S(N)(=O)=O N1(C(C(CC)OC)=O)CC(N(C(=O)CCn2nc(C)c(C)c2C)C)C(C)(C)C1 C1(N(C(c2cc(SC)oc2)=O)C)CCN(C(=O)C(=Cc2cccnc2)F)CC1C c1(C(=O)NC(CC)CN(C(=O)C(C)=C(C)C)C)sc(N2CCOCC2)nc1Cl C=CC(C)(O)C(=O)NC(C)CNC(=O)CSc1ccncc1 C(=O)(CC(CN(C)C)CC)NC(CC=C)CNC(=O)CSCCC#N C1(F)(C(N2CC(CC)C(NC(=O)CCC3CCOC3)C2)=O)C(C)(C)C1(C)C N1(N(CC(O)CC)CC(=O)N(CC(O)CNC)C)CCOCC1.CC N1(C(C(C)NC(=O)NC)=O)CC2CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 N1(C(CC2C(C)CCC2)=O)CC(C2CCN(C(C3(O)CCCCC3)=O)CC2)C1 C1(CC)CN(c2nnc(C)n2Cc2ncc(C(F)(F)F)n2C)CCS1 N1(C(c2n(CCOC)ncc2)=O)C(CNC(=O)CSC)CC2COCC12 Cc1nn(C)cc1CC(=O)N(C1CCCC1)CC(=O)NC(C)C C1(NC(c2csc(O)n2)=O)CN(C(c2cccc(Cl)c2)=O)CC12CC2 C1(CC)(NC(c2ncn(C)c2C)=O)CCCN(C(=O)CC2(O)CCCOC2)C1 CC(CC(=O)NC(C1CC(F)(F)C1)C)C(C)(C)NC(C1CC(=C2CC2)C1)=O c1(OC)ccc(Cl)c(CC(=O)N(C2CCCN(C(=O)CC(C)OC)C2)C)c1F Cc1cnn2cc(C(N3CC(NC(C4(O)CCSC4)=O)C(C4CC4)C3)=O)cnc12 C(=O)(N1CCC(C(=O)NC(c2ccncc2F)C)O1)c1c(CC)nn[nH]1 C(CCS(C)(=O)=O)(C(=O)OC(C)(C)C)NC(=O)OCC(CCO)C(F)(F)F c1(OCC(=O)N(C(C)C)CCN(C(=O)CCC#N)C)ccc2c(c1)CCC(=O)N2 C(=O)(CCCC(=O)OC)N1CCC(N(C(=O)C(C)CC2CCCO2)CCC)CC1 c1(CC(=O)N(C2CCN(C(=O)C=Cc3ccc[nH]3)C2)C)nccc2ccccc12 C1(OC)CC(CNC(=O)CNC(=O)CCC(C)C)N(C(c2nc(C)oc2C)=O)C1 N1(C(C2CC(N(C)CC)C2)=O)CCC2(CC1)CCN(C(=O)C(C)CO)CC2C C1(NC(C2(C=C)CC2)=O)CC2CCC1C(NC(=O)C(C)Cc1cccc(Cl)c1)C2 c1(C(=O)NCCN(C(COC(CC)CC)=O)C(C)C)cc(C(C)(C)O)on1 C1(C(=O)NCC=CC(=O)OCCC2CCOC2)CCC2CC12 N1(C(c2c(C)cn(C)c2)=O)CCC(C)C(NC(c2ccncc2Cl)=O)C1C c1(OC)nc(C(F)(F)F)c(C(=O)N(C2CCN(C(=O)C(=O)C3CC3)C2)C)s1 C(CCCCC(=O)N(C1CCCN(C(C2(C)CC=CC2)=O)CC1)CC)OC N1(C(c2ccc(CN(C)C)nc2)=O)CCC(C2CCN(C(=O)C(N)=O)C2)CC1 Cc1cc2occ(CC(N3CC(O)(C(C)NC(C4CC4(Cl)Cl)=O)C3)=O)c2cc1C Cc1cc2ccccc2cc1C(=O)NC1CN(C(=O)C(C)c2ccsc2)CC1C C(C)(CNC(=O)C(=Cc1ccccc1)C)(C(C)C)NC(CCCNC(C)=O)=O N1(C(C(CC)NC(C)=O)=O)CCN(C(c2ccc(CO)cc2)=O)C(C)C1 N1(C(C(CNC(C(CC)C(=O)OC)=O)C)=O)CCc2cncnc2C1 Cc1cc(C(F)(F)F)sc1C(=O)NCC1C2CC2C2CC12 N1(C(c2cc(C)ns2)=O)CC(NC(=O)C=C2CCCCC2)C(F)C1 c1(CCNC(C)(CCI)c2nnnn2C2CCOCC2)nnc2n1CCC2 C1(C(=O)NCCOC2CN(C(CN(CCC)C)=O)C2)CC2(C1)CC(F)C2 C1(CC(=O)N(CCC)C2CC2)CN(C(c2[nH]ccc2COC)=O)CCC1C C1(C)CCC(=O)NC(C)(C(C)C)CNC(=O)CN1.c1(OCC)cnn(C(C)C)c1 C1(CN(C)C(c2cccc(Br)n2)=O)CN(C(c2ccc(Br)nc2)=O)CCO1 C1(CC)(NC(C2OCC2(C)C)=O)CCN(C(C2CCCC(C(=O)OC)C2)=O)CC1 C1(C(N2CCC(CCNC(C(C)=O)=O)C2)=O)CCC(F)CC1 N1(C(=O)Cc2ccon2)CCCN(C(c2cn(CC(F)(F)F)nn2)=O)C(CO)C1 S(=O)(=O)(c1cc(F)cc(F)c1)N(C)C(C1CC2CCC1N2C(=O)OC(C)(C)C)=O C(=O)(CC(O)CCC)N(C1CCN(C(c2cc(C(N)=O)cn2C)=O)CC1)CC#C N1(C(CN2CCN(CC)CC2)=O)CCC(C)N(C(c2ccc(C(N)=O)o2)=O)CC1 O(NC(=O)C(C(C)O)N(C)C)C(C(=O)NC(C1CCCCC1)CC)CC(C)C C(N=c1nc(NCC2CCC(O)C2)c2c([nH]1)c(C)nn2C)c1c(O)ncc(C)c1 c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)CC23CC3)cccc2c1CNC2=O C(=O)(CC(C(F)F)NC(C1CSC(C)=N1)=O)NCCOCC C1(CC=C)(NC(C2CCCC2O)=O)CCCN(C(C2CCC3(C2)N=N3)=O)C1 C(=O)(CCCCCNC(C12CCC(C1)C2)=O)NCCC1C(C)(C)CCO1 c1(C(=O)NC(CCCCNC(CCC=C=C)=O)C)ccn(CC)c(=O)c1 C1(CCNCc2c(C)cc(O)nc2)CCc2ccccc2N1 c1(C(=O)OC)cc(N(C)CC2CCCCN2C(=O)C2=CCCC2)cc(C#N)c1 C1(CNC(c2c(CC)[nH]nc2Cl)=O)CN(C(c2cccnc2)=O)C2CCCC2O1 c1(C(=O)NC2CCC(NC(CC3CC(OC)C3)=O)C2)cnc2c(F)cccn12 c1(CN(C(C2(CC#C)CCC2)=O)C)ccc(CNC(C2(C)CS(=O)(=O)C2)=O)cc1 c1(C(C)N(C)C(c2cnc(-c3ccnn3C)cn2)=O)ccccc1F CCCC(C#N)C(=O)NC1CC(CCC(=O)NC2CCCCCC2F)C1 C(CC(=O)NC1(CCF)CC1)N(C(=O)CCC1CCCC1)CC C1(C(N(C)CC2CCCCCC2)=O)C2CC2CN1C(=O)C=CC(C)(C)C c1(CC)oc2ccccc2c1CC(=O)NCC(C)(C)NC(=O)CC(C)CC c1(C(=O)NC2C(OC)CN(C(C3CCOC(=O)N3)=O)C2)cc(C)cc(F)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(=O)NCC(F)(F)F)CC1C c1(C(=O)OC)cnc(N2CCN(C(=O)C(c3cnn(C)c3)O)CC2C)nc1C c1(C(N(CCC2N(C(C(COCC)C)=O)CCCC2)C)=O)n[nH]c2ccccc12 c1(CC)ccc2c(c1)OCO2.S1(=O)(=O)CCN1.C1(Br)(C(=O)OC)CCC1 C1(C(N2CCC(CNC(c3ccc(C4CC4)o3)=O)C2)=O)(SC)CC(F)(F)C1 N1(C(C(C)Sc2ccccn2)=O)C2CCC1C(NC(=O)CCc1ccc(Cl)s1)C2 N1(C(CCOC)=O)CCN(C(C2CCC(F)(F)C2)=O)C(C2CCC2)C1 Cc1cnc(C)c(C(=O)NCCC2CN(C(c3cc(C#N)c[nH]3)=O)CC2C)c1 C1(C(N2C(CNC(C(C)n3cncn3)=O)CC(O)C2)=O)CC12CCSCC2 Cc1n[nH]c(C)c1CC(=O)NC1(CCNC(C2CC23CCOC3)=O)CCOCC1 C1(CNC(c2c(C)n[nH]c2)=O)CCCN(C(C2CCN(C)C2)=O)C1 c1(C(=O)NC(CCOC)CNC(c2oc(C)cc2C)=O)cnc2cc[nH]c2c1 Cc1ccc(F)cc1C(C(=O)O)N(c1cccc(F)c1)CC1CC1 C(CC(=O)N(C)C)(C(N)=O)OC(C)=O.C1(C(=O)OC)CCC(C)(C)CO1 c1(C(N2CCCC(CNC(C3C4CC(=O)CC43)=O)C2)=O)occ2c1CCCC2 CN1C(=O)NCC12CN(C(C1CN(C(C3(C)COCCO3)=O)CC13CCC3)=O)C2 C(=O)(CCCC(=O)NCC(C)(C)CN(C(=O)Cc1cc(Cl)ccc1OC)C)NC C1(NC(C(C)O)=O)CCOC12CCN(C(c1cncn1C1CC1)=O)CC2 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(c1cn(CC)nn1)=O c1(C(=O)NCCNC(C2CCOCC2)C2CC2)ccc(C2CCCN2)o1 C1(CC)CN(C(=O)C=CCN(C)CC)CCC1CNC(C1CC(=O)CCO1)=O C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(=O)CC2CCCC2(F)F)CCC1CO C(=O)(C(C(C)(C)C)NC(=O)C=CC1CCN(C(c2cccc(=O)o2)=O)CC1)NC C#Cc1cnc(C(=O)NC(C)(CNC(=O)Cc2nnc(C)o2)CC)c(C)c1 N1(C(C(CCSC)NC(c2cocc2C)=O)=O)CCCC2(C1)N=N2 Cc1noc(C)c1C(C)(C)C(=O)OCCn1ccnc1C CC1(C)NC(=O)CC1C(=O)NC1COCC1NC(C1(CC2CC2)CCC1)=O c1(NC(C2CN(C(C(F)=CCC)=O)CC2F)=O)ccc2ccncc2c1 c1(C(C)OC)nc(C)c(C(=O)NCC(C)(O)CNC(c2ncccc2N)=O)s1 N1(C(CC2CCC(C)C2)=O)CCCC(N(C(=O)Cc2cnoc2)CC2CC2)C1 N1(C(C2(F)CN(C(CC(C)F)=O)C2)=O)CCC2(CCOCC2)C1 n1(CC)ccc(C(=O)NC2CCC(C)(CNC(=O)Cc3csnc3C)C2)c1C c1(NC(C2(CO)CN(C(C(C)C(C)n3cccn3)=O)C2)=O)cc(S(N)(=O)=O)cs1 c1(N2CCC(C)(CC)CC2)nc2ccc(Cl)cc2c(=NCCCN(C)C(C)C)[nH]1 Cc1ccn(CC(N2CC(NC(C3CCCN3C(N)=O)=O)CC2(C)C)=O)c(=O)c1 C1(C(=O)NCC(c2ccccc2)O)CC(F)CN1C(c1cccc(O)c1)=O N1(c2nc(SC)nc(C)c2)CC2CC(NC(c3ncc(Cl)s3)=O)CC2C1 C12(NC(CNS(NC)(=O)=O)=O)CCOCC1CN(C(c1sccc1C(F)F)=O)C2 N1(C(C(n2cc(CC(O)C(C)(C)C)nn2)C)=O)CCC(C=CC(=O)O)CC1 O(NC(=O)CC(C(C)CC)NC(c1ncn2c1CCC2)=O)CCCC#C Cc1nc2ncnn2cc1C(=O)NCCC(C)NC(c1ncc2ccccn12)=O c1(C(N(C2CCN(c3nnc(C(F)F)s3)C2)CC)=O)ccc(C)nc1Cl c1(-c2cc(NC(CSc3ccc(C)cc3)=O)sc2)ccc2ncnn2c1 N(C(=NCCCc1nccs1)NCC(F)F)C1CCCN(S(C)(=O)=O)C1 C(C)(C(=O)NC1CCCN(C(=O)CCn2nc(C)cc2C)C1)(C(C)C)NC(C)=O CCCS(=O)(=O)CC(=O)NC1CCN(C(=O)Cc2occc2C(=O)OC)C12CCC2 c1(C(C)NC(CC(C)NC(C2N(CC)CCC2)=O)=O)ccc(F)cc1 n1(C(CC)C)nnnc1C(c1nc(COC)cs1)NCCC1(COC)CC1 C(=O)(C(O)CC(F)(F)F)NC1C(SC)CN(C(c2ccnnc2)=O)C1 C1(N(C(C(CC)F)=O)CC(C)C)CCN(C(c2cc(-c3cccs3)on2)=O)CC1 C1(C(=O)NCC2CC2NC(=O)CC2(C#N)CC2)(CC)CCCCO1 c1(CC)ccnc(NC(c2noc(=O)n2C)c2nnnn2CC2CCCO2)c1 C=CCC(C)(O)C(=O)NC1CCC(NC(C2CCC3CC23)=O)C1 Cc1cc(F)sc1C(=O)Nc1cccc(CNC(C2CC3C=CC2C3)=O)c1 N1(C(C23OCC(C(C)C)(C2)C3)=O)CC(NC(C2CC(S(C)(=O)=O)C2)=O)C2(CC2)C1 C1(CCC)CCC(CN(C(c2cc(O)ncn2)=O)CC)CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CC(C)(C)NC(C(S(CCC)(=O)=O)C)=O)C N1(Cc2ccc(NCC)[nH]2)CCOCC(C(N(CC)CC2CCCCN2C)=O)C1 c1(N(C(CC)CCSC)C)[nH]c(=NC2CC2CC(C)(C)C)nc2c1ncn2CC C(=O)(C1=COCC1)NCC(CCOC)NC(=O)CSCc1ccccc1F C1(CNC(CCP(C)(C)=O)=O)CCN(C(c2ccc(CO)nc2)=O)CCC1(F)F c1(C(N2C3(CN(C(=O)CSCC(F)(F)F)C3)CC2)=O)ccc(S(=O)(=O)CF)cc1 O=C(C(O)C1CCc2ccccc21)N1CCOC(C(F)F)CC1 CCC(C)(C)C(O)C(=O)NCC(C1CCCCC1)NC(C1CC2(CCC2)CO1)=O N1(C(c2ncn(CC)n2)=O)CC(NC(C2CCCC(OC)C2)=O)C2(CC2)C1 C(C(O)CC(C)(C)CO)N1CCC(Oc2c(OC)cccc2)C1 c1(C(=O)NCC2(O)CC(NC(CC(CC)C3CC3)=O)C2)cnc2cnccc2c1 c1(CNC2C(C(=O)Nc3ncc(C#N)nc3)CCC2)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1C(=O)NC1(CC(N2CCCC(C#N)C2)=O)CCC1 O(NC(=O)C(C(C)CC)NC(=O)C(CC(C)C)OC)CC=C N1(C(C=C(CCC)C)=O)CCC(NC(c2ccccc2OCCOC)=O)C(F)C1 CC1C(NC(C2(CF)CCC2)=O)CCN1C(C1CCN1Cc1ccccc1)=O C(=O)(C1=CC(C)(COC)C1)N1CCC(CC=C)(NC(=O)C=CC(CC)=CC)C1 CCCCC(CO)NC(=O)CCN(C(=O)CC1CCC(=O)C1)C1CC1 c1(C(=O)NC(CC)(CNC(=O)C(C)C(C)COC)CC)ccc2c(c1)NC(=O)C2 N1(C(C(C)(C)OC)=O)C2CCC1(CNC(=O)C(C)(C)c1ccno1)CC2 c1(C(N(C(CC)CO)C2CC2)=O)coc(CNC(=O)C(O)CN(C)C)c1 C1(CNC(Cn2ncc(C)c2)=O)(NC(c2c(C)cncc2C)=O)CC2CCC1C2 N1(C(CCSCC(C)C)=O)CCC(C)(NC(C2CCC2(F)F)=O)C1 c1(C2(C(=O)Nc3ccc(CC)cn3)CC2)ccccc1C#N N1(C(CCCC#CC)=O)CCC2C(CCN2C(c2cccc(SC(F)F)c2)=O)C1 Cc1cc2c(CC(=O)NC3CC(n4cc(-c5cn(C)cn5)nn4)C3)csc2s1 C1(CNC(c2c(C)onc2C(F)(F)F)=O)CCN(C(=O)CC(C)O)C1(C)C C(=O)(C1=NNC(=O)CC1)N1C(C)CC(NC(CCCCNC(C)=O)=O)C1 C(c1cccc(O)c1)=CC(N1CCC(CC(=O)NCC(O)CF)CC1)=O C1(NC(C2(NC(CCN(C)CC)=O)CCC(C)(C)C2)=O)CCOCC12CCC2 C(CCCC(C)(C)NC(=O)C=Cc1cncs1)NC(C(C)Cc1ccncc1)=O c1(C(=O)NCc2cccc3[nH]ccc23)cnc2nc(O)nc(O)c2c1 C(=O)(C(C(C)C)NC(=O)OC(C)(C)C)NCCCNC(c1c(CSC)cco1)=O c1(NCCC2(CSC)CC2)ncccc1S(=O)(=O)N1CC(C)C(C)C1 C1(C(N(CC(COC)C)C)=O)CN(C(C2CN(C)CCN2C)=O)CC12CCC2 c1(NC(N2C(C(=O)OC)C3CC3C2)=O)ccc(OC(F)(F)F)cc1Br c1(C(N(CCOC)CCNC(c2csc(Cl)c2)=O)=O)nccc2nn[nH]c12 C1(NC(=O)CCc2ncc[nH]2)CC2CCCC(C1)N2C(c1ncncc1Cl)=O C(=O)(CC(F)(F)Br)NCCOCCN(C(=O)C=CC=C(Cl)Cl)C c1(CCC(=O)NC2C(NC(C(C)(C)NS(C)(=O)=O)=O)CC2)ccc(F)cc1 C1(NC(C2(C)COCCO2)=O)CCC2(CC1)CC2NC(=O)Cc1ccccc1O N1(C(C=NOC)=O)CC=C(CNC(=O)CCc2csc(C)n2)CC1 c1(C(N(CC(C)N(C)C(c2cnc(O)o2)=O)C)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(C)(NC(c2c(COC)noc2)=O)CCN(C(=O)C(c2ccc(C)cc2)(F)F)C1 c1(C(=O)NC(C(C)C)C(C2CCCCC2)NC(C2CCC2)=O)ncc(F)cc1F C1(C(=O)NC2CCN(C(C(c3ccc(F)cc3)=O)=O)C2)CCC12CCOCC2 c1(C(=O)NC2CC(F)(CNC(CCOCCN(C)C)=O)C2)c(F)cccc1F Cc1cc(C(N2CCC(N(C(=O)CCCC(F)F)C)C2)=O)cnc1O c1(NC(C2CCN(Cc3c(C)[nH]c(C)c3C)CC2)=O)ccc2c(c1)CCC2 c1(C(N(CC(=O)N(CCCC#C)C)CC#C)=O)cc(C)nc(O)n1 c1(C(=O)NC2C(C)N(C(=O)CC3(C)CC3)CCC2)ccn2c1CCCC2 C1(C(N(C)CCNC(c2cnsn2)=O)=O)CCC(c2nc[nH]n2)CC1 O=C(C1=NOCC1)NC1CN(C(=O)Cc2cc(Cl)cs2)CC1O CC1CN(C(C23CCC(C(=O)O)(CC2)C3)=O)Cc2cccc(Br)c21 CC1CCCn2c(CC(=O)NCCNC(=O)Cc3ccccc3)cnc21 C12(CC(=O)NC3CC(CNC(CCC(C)N(C)C)=O)C3)CCCCC1C2(F)F c1(NC(=O)Nc2cccc(CS(C(C)C)(=O)=O)c2)cc(F)c(F)cc1I C1(CNC(C(=O)NCC)=O)CCC(C(=O)N(C)CCC)CC1 C1(C(=O)NCCC(CC)(O)CC)CC(N=[N+]=[N-])CN1C(C1CC(C)=NO1)=O C#Cc1ccc(C(N2CCC=CC2C(=O)NOCCCCCC2CC2)=O)cc1 C1(C(=O)NCC(CNC(COc2cn(C)nc2)=O)O)C(F)(F)C12CCC2 C=CC1(C(=O)NCc2c[nH]nc2C2CC2)CCN(C(c2cnc(N)cn2)=O)C1 C1(NCc2ccc(CC(C)C)cc2)CCS(=O)(=O)CC1 Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccco2)s1 C(CO)(CCCCNC(=O)C(C)(C)F)CNC(c1cccc(SCC)c1)=O N1(C(C(C)=C(CC)C)=O)CCC(C)(C)C1CNC(=O)Cc1nn(C)cc1Cl C12(C(=O)NCC(CNC(CCn3c(C)ncc3)=O)O)CCOC(C)(C1)C2 c1(C(=O)NCC(CC)NC(c2nccn2CC)=O)oc(C(F)F)cc1C C(CC(C)C(=O)N(CC(=O)OCc1ccccc1)CC1C(O)C(O)CO1)=CCC c1(C(N2CC(OC)C(NC(=O)CC#N)C2)=O)c2c(nn1C)CCOC2 c1(C(=O)NCC(N(C(C(CC)CC)=O)C)C2CC2)ccc2c(c1)NC(=O)CN2C N1(C(CC(CC2CC2)NC(CCSCCCC)=O)=O)CCCC(C)CC1 N1(C(C=C(C)C(F)F)=O)CC(NC(=O)C(c2cccc(C)c2)C)CC(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3cocn3)=O)CC2)=O)cc(Br)c1C C1(CNC(c2cccc(C)n2)=O)CC(C)(C)CN1c1cc(-c2cccs2)ncn1 C1(NC(c2cc(C)[nH]n2)=O)CC(C(=O)NC2CN(c3ncco3)C2)C12CCC2 CC(=O)CC(C)(C)CC(=O)N1CCC2(CCC(OC(C)(C)C)C2)C1 C#CC1(C)CCCN(C(C2CCCN(C(c3ccc(C)nc3)=O)C2)=O)C1 c1(C(=O)NC2C(NC(COCP(C)(C)=O)=O)COCC2)cnc(O)c2ccccc12 Cc1cnn(C)c1S(=O)(=O)N1CCN(CC(=O)Nc2ncc(Cl)cc2Cl)CC1 c1(C(=O)NC2CC(Cn3cc(-c4c(C)csc4)nn3)C2)cc(Br)c(O)cc1Br c1(C(N2CCC3(NC(C4(O)CCC4)=O)C(C2)C3)=O)cccc2nn[nH]c12 CC(C)C(CC(=O)NCC12CCC(CC1)N(C(c1cnc(S)[nH]1)=O)C2)C(C)C CCCC(CC)CCC(=O)N1CCCN(C(=O)Cc2ccc(O)cc2Cl)C(C)C1 C1(OC(C2CCN(C)C2)=O)COC2(C1)CN(C(=O)OC(C)(C)C)C2 c1(CC(=O)NC2(C)CC(NC(C3CC(F)(CO)C3)=O)C2)ccc(F)c(Br)c1 c1(NC2CCN(C(C(CC)F)=O)C(C)C2)nc(Cl)nc2sccc12 C1(NC(CCCCC)=O)CC2(C1)CC(CNC(C1(C(=O)N(C)C(C)C)CC1)=O)C2 Cc1cccc(C(N2CCC(C)(CC(=O)NC(C)C(C)(C)CO)C2)=O)c1C C(=O)(C(CC)C(=O)NCC1CCC(NC(=O)CCc2cccc(O)n2)C1)OCC Cc1cc(C(=O)NC(CNC(c2cc(CF)on2)=O)C(C)(C)C)[nH]c1C n1(C(=O)N(CCO)CCO)ncn2nccc2c1=O CC1CCN(c2ncc(C(N3CC(NC(c4csc(Cl)c4Cl)=O)C3)=O)s2)CC1 N1(C(CC=C=C)=O)CCCC(C(C)(O)CNC(=O)Cc2cn(CC)nc2C)C1 c1(OC)ccc2c(c1)CC(C)N(C(c1csc(Cl)n1)=O)C2 c1(OC(C)C)cc(-c2csc(NC(c3ccc(C(C)(C)C)cc3)=O)n2)c(F)cn1 C(C(C(=O)NCC1CCN(C(=O)CCc2ccncn2)C1)N(C)C)OC Cc1ccc(C(c2ccccc2)NC(=O)NCC(N)C(F)(F)F)cc1 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(Cc2ncc(C)o2)=O)C1(C)C C=CCC(C(=O)N1CC(C)C1C(=O)NC(C)C(C)C)OC C(=O)(C(C(C)(C)C)c1ccccc1)N(Cc1nn(C)c(F)c1)C1CC1 CC1=C(C(=O)NCC2CC2CNC(c2ccc(C)c(C)c2)=O)CCCO1 C(=O)(C(CO)C(C)(C)C)NC1(C(=O)NCC(CCC)CCC)CSC1 Cc1nc(N(C)C)sc1C(=O)NCC1(NC(C2CC2F)=O)CCC1 c1(NC2(C3CN(C(C(Cc4ccc(C)cc4)C)=O)C3)CC2)nc(C)nc(O)c1C c1(C(=O)NCCCC(CCC)NC(=O)C(C)N(C)C)ccc2c(c1)C=CCC2 C(=O)(C1=C(Cl)CCCC1)NC(C)CCN(C)C(c1ccccc1C(C)(C)C)=O CC(C)C(CCN(C)C(C1CC1(F)F)=O)NC(c1c(Cl)cnn1C1CCCC1)=O C1(NC(C2CC(C)(CC)C2)=O)CCCC1(C)CN(C(=O)C=Cc1sccc1C)C N1(C(C(CC)n2nccc2C)=O)CCCC(C)(NC(c2cc(C(C)C)[nH]n2)=O)C1 NS(=O)(=O)CCC(=O)NC1CN(C(=O)Cn2nnc(-c3ccco3)n2)CC1O C1(C(=O)NCC(CC)n2cccn2)CN(C(=O)Cc2csnc2C)CC12CC2 c1(C(C)=O)ccsc1C(=O)N(CCC(C)NC(=O)CC1CCCCO1)C c1(C(=O)NC(CC(C)NC(C2CCC(C)(C)O2)=O)C)cc2ccccc2c(=O)o1 C1(NC(C(COC)C)=O)CCSC12CN(C(=O)C=Cc1ccccc1OC)C2 c1(NC(C2(O)CCN(Cc3c(C)cccc3)C2)=O)nc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)CO)=O)CC(F)CC1CNC(=O)Cn1nnc(-c2ccccc2)n1 CC1(NC(c2ccnc(O)c2)=O)CCC(NC(C23CCCC2C3Br)=O)CC1 C1(C(N2CCC(CN(C(C(CC#C)C)=O)C)C2)=O)CCC2(CC1)CC(O)C2 c1(C(=O)NCCCN(C2CC2)Cc2ccncc2C(F)F)nc[nH]c2ncnc1-2 n1(CC(=O)N(CCOCCCNC(COC)=O)CC2CC2)cc(C(C)O)nn1 C1(NC(CCC(CC)NC(C2CC=C(C)CC2)=O)=O)CCCCC1N=[N+]=[N-] C1(NC(C(CNC(COC2(C)CCC2)=O)CC2CC2)=O)CC2(C1)CC(C)(C)C2 C(=O)(CC(C)CC(=O)N(C1(CC(=O)NCc2nccn2C2CC2)CC1)C)OC C(N=c1[nH]c(SC)ncc1C)C1OCCN(C(c2c(OC)cc(O)cc2)=O)C1 C(CCCC(C)NC(=O)C(C)CCO)NC(C1(C)CC(=C)C1)=O c1(CN2CCC(CN(C(C(COC)O)=O)Cc3cccnc3)C2)ccccc1F C12(C(=O)NC3C(C)CN(C(=O)Cc4ccsn4)C3)CCCCN1CCC2 c1(C(N(C(C)C(=O)NCc2ccc(O)nn2)C)=O)ccnc2cc[nH]c12 N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)C=CC2CCCO2)CC(C)(C)C1 C1(C(=O)NCC2N(C(CC3(OCC)CCCC3)=O)CC2)Cc2cc(C)ccc2O1 N#Cc1ccc(CNC(c2scnc2-c2cc(C(=O)O)ccn2)=O)cn1 C(=O)(CS(=O)(=O)C1CC1)N1C(CCCNC(c2c(C(N)=O)nccn2)=O)CCC1 c1(C(N(C(C(=O)NCCN(C(C)C)C)C)C2CCC2)=O)cnc(N)cn1 c1(C(C(=O)NCC(CO)NC(=O)Cc2ccoc2)NC(N)=O)cc(F)cc(F)c1 c1(C(=O)NCCCOCCN(C(CC2CC(=C)C2)=O)C)cccc(C=C(F)F)c1 N1(C(C(C)c2ccsc2)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)CCC1C C1(C(N2CC(N(C(CC3(OCC)CC3)=O)C)C2)=O)(COC)CCOC1 C(=O)(C#CC1CCCOC1)N1CCCC(NC(c2cc(N)c(Cl)cn2)=O)(CO)C1 N1(C(CCC(CC)OC)=O)CCCC12CCN(C(c1cnn(C)n1)=O)C2 C1(CS(N)(=O)=O)CCC(N=c2[nH]c(=NCC3CC3C3CC3)[nH]c3c2CCCCC3)C1 N1(c2cc(C)nc(N(CC(C)(F)F)C)n2)C(C)C2CCCCC2C1C N1(C(=O)CN2CCCS2(=O)=O)CC2C3CCC(C2C1)N(CCn1cc(Cl)cn1)C3 C(C(=O)N1CC2C(CN(C(=O)CN3CCOCC3)C)C2C1)(C(C)(C)C)SC C1(C)(C(N2CCC(NC(C)=O)CC2)=O)CN(C(C2C3CCCC23)=O)C(C)(C)C1 c1(N2CCC(C)(NC(C3C4CCCC34)=O)C2)ncc(Cl)c(O)n1 N1(C(C2CC23CC3(F)F)=O)CCn2c(CNC(C3(O)CCCCC3)=O)nnc2C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC1(C2CN(C(C3N(C)CCOC3)=O)C2)CC1 C1(CC)(Nc2ccnc(OCCO)c2)CC(F)(F)C1 C1(C(N(C(C)CCNC(C2CC(C)(C)CN2C)=O)C)=O)Cc2ccccc2N1C C1(c2nnnn2Cc2nnn(C)n2)(NC(COC)CN2CCOCC2)CC2CC2C1 C(C)(C)(CCCC(=O)NC1CC(CO)C1)NC(CC1N(C)CCC1)=O CN(CCCC(=O)NCCC1(O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C1)N=O N1(C(C(CC)C)=O)CC2(CCN(C(C3(c4cccc(C)c4)CC3(F)F)=O)CC2)C1 C1(CC=C)(C(=O)N(CC(O)CC)C)CCCN1C(c1cn[nH]c1)=O c1(C(N2CC(OC)C(NC(c3cnco3)=O)C2)=O)cc(N)ccc1C(F)(F)F C1(CC(=O)NC2C(NC(C3(C#N)CCOC3)=O)C2)CCCCCCC1 C(=O)(C(CC(C)C)C(N)=O)N1CCC(CC=C)(NC(c2ncc(F)cn2)=O)CC1 c1(C(N2CCCCCC(NC(CC=C(C)C)=O)C2)=O)[nH]nc2c1CCCC2(C)C c1(C(N2CC(NC(c3ccc(OC)cc3)=O)C(F)C2)=O)cccc(Cl)c1Br c1(C(=O)NCC2CN(C(C(COCC)(C)C)=O)CC2C)cc(C)cc(Cl)c1N N1(C(C=NOC)=O)CC2(C1)C(NC(C1CC(OC)CN1C(C)=O)=O)CCS2(=O)=O Cc1cc(F)ccc1C(O)C(=O)NC1CC(C)N(C(C2CCC=CO2)=O)C1 CC1(CNC(C23CSCC2C3)=O)CCCN(C(c2ccc(O)nc2)=O)C1 N1(CCNC(C2CCC3CCC23)=O)CCCN(C(c2cccnc2)=O)CC1 N1(C(Cc2nc(-c3ccc(OC)cc3)sc2)=O)CC2(CCC2NC(=O)CCF)C1 Cc1ccc(C=CC(N2CCN(C(=O)CC(C)C3CC3)CC2C2CC2)=O)cc1Cl C(=O)(C1=C(C)OCCC1)NC(C(N1C(C#C)COCC1)=O)C c1(C(=O)NCC(CC(C)C)NC(C2CC(O)C2)=O)ccc2occc2n1 CCCC(C)(O)CC(=O)NC1CCCN(C(=O)C(F)=C(C)C)C1CC C(=O)(C(F)C(F)(F)F)N(CCC(c1cccs1)NC(COC(CC)CC)=O)C C1(C)(NC(C(CCNC(c2cncc(O)c2)=O)OC)=O)CCCC1(C)C c1(C(N2CCC(C(=O)NOC)CC2)C(=O)NC(CC)C)nc(C)c(C)n1C N1(C(COCCN(C(=O)CCOC2CCC2)C)=O)CCN(C2(C)CC2)CC1 C1(C(=O)NCC(C)(C)NC(CCc2nc(C)sc2)=O)OCC2COCCC12 C1(CNC(C2CC(C)C2)=O)CN(C)CCN1C(c1ccon1)=O CCCCCCCCCC(=O)N1CCN(C(=O)CCCC(=O)OC)CCC1C C1(CC)CCC(C)CN1C(=O)CCCN(C(=O)Cc1cccn1C)C c1(C(=O)NC2CC(C)N(C(c3cnc(O)s3)=O)CC2)cccc(S(C)(=O)=O)c1 c1(CC)nnc2n1CCCC2C(=O)N1CC(NC(C2CN(S(N)(=O)=O)C2)=O)C1 c1(C(N2CC(C(N3CCC(OC(C)C)C3)=O)C2)=O)c(Cl)cc(F)cc1Br C(=O)(CCC(=C)Cl)NCCCC(C)NC(C1(CC#C)CCOC1)=O C1(C)(NC(=O)Nc2n(C)ccn2)CCCN(C(=O)C(CO)Nc2ccccc2)C1 CCCCCCC(C)C(=O)N1CCCC1CN(C(=O)CCN(S(C)(=O)=O)C)CC N1(C(C(CC)N(C)C(c2cnc(S)nc2)=O)=O)CCC(C)OC(C)C1 N1(C(c2cnc(C)s2)=O)CC2(CNC(=O)C(F)n3cccn3)CCC1CC2 c1(C2(n3c(-c4cnn(C)c4)nc(CC(C)(C)C)n3)CC2)ccc2ccccc2c1 c1(NC(CS(Cc2c(C#N)cccc2)(=O)=O)=O)ccc2c(c1)OCCO2 Cc1cc(C)c(C(=O)NCC(C)(O)CNC(=O)C(O)CCN(C)C)c(N)c1 C1(CC(=O)NCC(CC)(CC)OC)CC2(C1)CN(C(=O)CCc1ccn(C)c1)C2 n1(-c2ccc(C)cc2)cc(C#CCNC(c2cc(Cl)cc(Br)c2F)=O)nn1 Cc1ccc(C(=O)NCCc2ccc(C(=O)NCc3ccncc3)cc2)c(O)n1 c1(CC)ccc2occ(C(=O)NC3CCC(NC(=O)CCn4ccnn4)C3)c2c1 N1(C(CCCOC)=O)CC2CCC(C1CO)N2C(=O)C(C)Oc1ccccc1 c1(C(N(CC(OC)OC)CC(C2CC2)OC)=O)cc(Cl)ccc1C c1(CC(=O)N(CCCCN(C)C(c2cc(Cl)cs2)=O)C)nc(C2CC2)cs1 c1(OCCNC(c2cccc(C3CC3)c2)C)cc(F)cc(Cl)c1 c1(C(N2C3CN(Cc4cc(Br)cc(Br)c4F)CC23)=O)cc2n[nH]cc2cc1Cl C1(NC(Cn2c(C)ccn2)=O)CN(C(=O)C=CCn2cncn2)CCC1F C1(N(C)C(c2cnc(C(C)(F)F)s2)=O)CCC(NC(C2CCC2(F)F)=O)CC1 C1(OCC)C2CC3CN(C(C4CC(C)CCC4CC)C(=O)NC(C)(C)C)C1C3C2 N1(C(C2CC3CC2C2CC32)C(=O)NCCC2(C)CC2)CC(C)(C)OC2(CCOC2)C1 C(=O)(CC(C)(C)O)NCC1C(CNC(C=C(CCC)C)=O)C1 O=C1CN(C(=O)CC2CCC(NCCNS(=O)(=O)CCl)C2)CCCN1 CC(C(C)(C)C(=O)NCC1CCCOC1)NC(C1COCCC1C)=O N1(C(CN(CCC)C)=O)C2CCC(C2)C1CC(=O)NCC(C)CC(=O)OCC C(c1ccc(OC)cc1)=CC(=O)NC(CCCC)CNC(=O)CC(C)OC C1(NC(c2c(CC)non2)=O)(CNC(=O)Cc2sc(S)nc2C)CC2CCC1C2 C1(n2cc(CN3CCC(N(CCC)CCC)CC(N)C3)nn2)C2CS(=O)(=O)CC12 N1(CC)CC2(CN(C(=O)CC=CCNC(=O)CC3CCCOC3)C2)C1 N1(C(=O)CC2C3CCCC3N2C(=O)CC2CC=CCC2)CCc2n[nH]cc2C1 CC(CC(F)F)C(=O)NCC(c1ccccc1F)NC(c1n[nH]cc1F)=O c1(OC)c(C(=O)NC(CO)C(C)NC(=O)Cn2ncn(C)c2=O)cc(Cl)cc1Cl CN1CCC(C)(C(=O)NCC2(C(C)(C)C)CCN(C(=O)OC(C)(C)C)C2)C1=O c1(N(C(CSC)C(=O)O)C(=O)CC2CC2C)ccnc(-c2ccoc2)c1 C1(CNC(c2c(Cl)cn(C)n2)=O)CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2 c1(C(N(CC(C)N(C)C(C23CC(C(F)F)(C2)C3)=O)C)=O)cnccn1 C(=O)(C1=NOC(C)C1)N1C(C(=O)NCC2(C#C)CCC2)CC(O)C1 C1(OC)CN(C(=O)C(C)SC(C)C)CCC1NC(c1ccc(C(N)=O)[nH]1)=O C1(NC(c2cnc(OC)s2)=O)CN(C(=O)C(C)(C)C2CC2)CC(C)(C)C1 c1(C(N2CCN(C(CN(C)CC)=O)CC2C2CCC2)=O)cccc2[nH]c(=N)oc12 C(C(C)CC(=O)NCCOCC1CCCC1)NC(Cc1onc(C)n1)=O CCC1=NOC(CC(=O)NCC2CCCCN2C(c2cc(C(=O)OC)sn2)=O)C1 C(=O)(CC(O)c1ccccc1)N(CC(CN(C(=O)COCCCF)C)O)C c1(C(N(CC(C)NC(=O)C(C)CCCOC)CC)=O)ccc2nc(C)sc2c1 C1(NC(c2ccc(C)nn2)=O)CCCC12CN(C(=O)CCOC1CC1)C2 N1(C(=O)OC(C)(C)C)CCC2(COC(COC(c3n[nH]c4c3CCCC4)=O)C2)C1 c1(OC)cc(OC)c(C(=O)NC2CCN(C(=O)CN3CCNC(=O)C3)C2C)cn1 C1(NC(c2cc(C)c(C)nn2)=O)COC2(C1)CN(C(c1ccc(Br)o1)=O)C2 C1(C(=O)NCC(=C)CCN)CC(N=[N+]=[N-])C1 C1(CNC(C(C)SC)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 Cn1ccc(CCC(=O)NC2CC(NC(=O)C=CC(F)(F)F)C2)c1 N1(C(C2C(OCC)C2)=O)CCCC2CN(C(=O)CSc3nccn3C)CC12 N1(C(C=CC)=O)CCc2ccccc2C1CNC(c1sc(Br)cc1F)=O C(=O)(C1=CCC(C)CC1)N1CC(NC(c2c(C)nc(C(C)(C)C)s2)=O)(CO)C1 N1(C(c2cc(C)cc(F)c2N)=O)CC2CCCC(NC(C3CC34CCC4)=O)C2C1 C1(CNC(Cc2c(C)cc(C)s2)=O)N(C(=O)CC2CC2C2CC2)CCCC1(C)C N(C1c2ccccc2CC12CCC2)C(c1cc(=O)n2ccsc2n1)=O N1(C(C(C)NC(CC)=O)=O)CCC2CCC(C1)N2C(=O)CCc1nc(C)cs1 C1(CN(C(=O)C(c2ccc(F)cc2)F)C)CCC(NC(=O)C=C(Cl)Cl)CC1 CC(C(=O)N1CCCC(CNC(=O)C(C)(C)n2cc(Br)cn2)C1)C(F)F C1(C(N2C(CNC(C(CC)OC)=O)CC(F)C2)=O)CCCC2C1C2(F)F N1(C(c2c(C)con2)=O)CC2CS(=O)(=O)CC2(CNC(=O)C2=CCS(=O)(=O)C2)C1 c1(C(=O)NC2C(C(=O)OC)CCC2)sccc1S(=O)(=O)N1CCSCC1 N1(C(c2cc(F)c(O)c(F)c2)=O)CCC2(CCCN(C(c3coc(O)n3)=O)C2)C1 C1(NC(C2(C(C)NC(C=CCOC)=O)CC2)=O)C=CCCCC1 C1(C(=O)NC2C(CNC(COCCC=C)=O)C2)CCCN(c2ncccn2)C1 N1(C(C2C(C)OCC2)=O)CCCN(C(=O)CCN2CCN(C)CC2)CCC1 c1(NC2CN(C(C(CC)CC3CCCC3)=O)CC2C)[nH]c(=O)n(C)c(=O)c1C#N CCC(C(=O)NCCCN(C(C1(CCO)CC1)=O)C1CC1)C(C)(C)CC c1(OCC)ccc(C(=O)NCCCC(CO)NC(=O)C(O)C2CCCC2)cc1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(c2csc(S)n2)=O)C1 N1(C(=O)OC(C)(C)C)CCC(C)(CNC(=O)NCC(c2ccccc2)OC)C1 N(C(=NCCC1COC1)NC1CC12CC2)Cc1cn(C)nc1 N1(C(C2(CC)CCCC2)=O)CCC2(CCC2)C(CNC(C2C=CC=CC=C2)=O)C1 c1(NC(C)=O)cccc(CC(=O)NC2CCC2NC(c2cc(C)c(C)[nH]2)=O)c1 n1(CC(C)NC(c2cc(Cl)no2)=O)cc(-c2ccncc2)nn1 N1(C(=O)OC(C)(C)C)CCC(O)C(C(=O)NCCNCc2ccc(=O)oc2)C1 Cc1c(C(N2CCN(CCCNC(C3CC3C#N)=O)CC2)=O)cccc1Cl c1(CS(=O)(=O)N(C(C)C(C)(C)C)C)cccc(Br)n1.C123CC(C1)(C2)NC3=O CC1c2cccc(F)c2CCN1Cc1sc(Cl)cc1Br C1(CC(=O)NCC(C)OC(F)F)CN(C(=O)COC2CCCCCC2)CC12CC2 c1(CC(=O)NC2CC(CO)N(C(c3ccc(Cl)[nH]3)=O)C2)ccc(F)cc1F C1(NC(C(C(C)C)SC)=O)CC=C(C(=O)NCc2ccc(C#N)cc2)C1 C(=O)(C(F)CC(C)(C)C)NCC1C(C)CCN(C(C2(CC=C)CCCC2)=O)C1 c1(C(=O)NC(CC)C(C)O)cnn2cccc(-c3cc(OC)ccc3O)c12 C(=O)(CC(O)C(C)C)NCC1CCN(C(C(C)NS(CCCC)(=O)=O)=O)CC1 Cc1cc(CN2CC(C)(CNC(=O)C(CO)c3ccccc3)C2)nc(C)c1 C(=O)(C(CC1CCCC1)NCC(=O)OC)N(CCOCCOC=C)C c1(OC)ccc(CC(=O)NCCC2(O)CN(C(=O)Cn3cc(Br)cn3)C2)cn1 C(=O)(C(C(=O)NCCCN(C(=O)CCSc1n[nH]c(C)n1)C)C(C)C)OCC c1(CNC(C(C)(C)CCl)c2nnnn2C2CCCCC2)nc2ccc(Cl)cc2[nH]1 Cn1ncc(C(F)(F)F)c1C(N1CCN(C(=O)Cc2csc(NC=O)n2)CC1)=O N1(C(C(C)C)=O)CCC2CCN(C(c3cnn(C4CC4)c3)=O)CC2C1 c1(OCC)c(-c2cnc(C(N3CCCCC3CO)=O)cc2OC)ccc(F)c1F C1(CC(=O)NCc2ncco2)CCCC1NC(=O)CC1CSC1 c1(C(N2CCC(C)C2)C(=O)NCCCSC)ccc(C(F)(F)F)o1 c1(CC(=O)N(C2CN(C(c3cc(F)cnc3O)=O)CC2(C)C)C)cc(F)ccc1Cl N1(C(c2c(SC)ccs2)=O)CCC(F)(CNC(=O)C(F)C2CC2)CC1 c1(C(=O)NCc2ccc[n+]([O-])c2)cnn2c1NCC2 c1(COCC(=O)NC2(CCC(=O)NC3CCCO3)CCC2)c[nH]ccc1=O CC1CCC(NC(=O)C(C2CCCCC2)N(C)C)CN1CC1C2CC3C(C2=O)C13 c1(C(N2CCC(C)C2CNC(=O)CNC(=O)CC(C)(C)C)=O)coc2c1COC2 c1(OCC)cccc(C)c1C(=O)NCc1csc(CNC(C2(F)CC2)=O)n1 C1(C(N2CC(O)(CCNC(C3CN4CCN3CC4)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C(N2CC3CC2(CNC(C24CCCN2CCC4)=O)C3)=O)ccc1C#N CCC(C)(CC(=O)N1C2CCCC1CN(C(=O)C=CCCC(C)C)C2)C(=O)OC c1(C(N2CCC(C)(NC(C=CSC)=O)C2)=O)c(Br)cncc1[N+](=O)[O-] N1(Cc2cccc(C(=O)OC)c2F)CCC2(CC1)OCc1ccccc12 c1(N2CCC(C(F)(F)F)(CC)C2)nc(=NCCC2(C)CC2)[nH]c2c1CCCCC2 c1(OC)cccc(N(c2nnc(C)n2Cc2cccnc2OC(C)C)C)c1 N1(C(C2(N(C)C)CCCC2)=O)CC(C(=O)O)CC(c2ccccc2)C1 C1(NC(CCCCOC)=O)CC12CCN(C(c1cc([N+](=O)[O-])n(C)n1)=O)CC2 C1(C(N(CC(C)NC(CN(C(C)=O)C)=O)C)=O)CC(O)CN1C(=O)OC(C)(C)C c1(C(N2CCN(C(c3n[nH]cc3Br)=O)CC2)=O)cccn(CC(F)(F)F)c1=O C1(CNC(c2cccnn2)=O)C(F)(F)C12CCC2.N12CCN(CC1)C1CCN2C1 CCC(CC(C)C)C(=O)N1CCCC(C(=O)NCCOC2CCC2)CC1 c1(C(N(C2CCN(C(c3c(OC)nc(C)nc3)=O)C2)C)=O)ccn2c1CCCC2 C=C1CCCN(C(=O)CCN(C(C2CC=CCO2)=O)CC2CC2)C1 C1(C(=O)NCc2occ(C(=O)NCc3nc(C)oc3)c2)CN(C)CCO1 c1(C(=O)NC(C)CC(C)NC(c2ccco2)=O)cc(Cl)ccc1OC(F)F Cc1cnc(C(=O)NCC2C3CC2N(C(=O)CSc2n[nH]c(=N)s2)C3)nc1 c1(SC)nc2ncnc(NC(CCNC(C3NC(=O)CC3(C)C)=O)C(C)C)c2s1 c1(C(=O)Nc2cccc(NC(C(C(C)OC)O)=O)c2)c(C)nc(C)nc1C N1(C(Cc2ccc(C(N)=O)nc2)=O)CCCOC(CCNC(=O)C(F)(F)CO)C1 N1(C(C2C(NC(C(C)(C)OCC)=O)CC2)=O)CCCC(CC(N)=O)C1 N1(C(CCCCC(=O)NC)=O)CC(C2CCN(C(c3ccc(C)s3)=O)CC2)C1 C1(NC(C=CCN(CC)CC)=O)CN(C(=O)CC2CC(N(C)C)C2)C(C)(C)C1 C1(NC(C(C)(C)C#N)=O)CC(NC(=O)Cn2nnnc2-c2ccsc2)C12CCC2 C12(C(N)=O)CC(CNC(C3CCOC4(CCCC4)C3)=O)(C1)OC21COC1 CC1CC=C(C(=O)NCC2=CCN(C(c3ccoc3Br)=O)CC2)CC1 S(=O)(=O)(c1cc(C(N2CC(CO)(NC(=O)C(F)C(C)C)C2)=O)ccc1F)NC c1(N2CCC(N(C(C)=O)C)CC2)nc(NCCCCCF)c2ccsc2n1 N1(C(C(Cn2cccn2)NC(CCC(C)OC)=O)=O)CCOC(C#N)C1 C(=O)(C(F)CC(C)(C)C)NC(C1(O)CN(C(=O)CCCC2CCCCC2)C1)C N1(C(c2cc(OC)no2)=O)CCCN(C(=O)CC(c2ccccc2)N(C)C)CC1 S(=O)(=O)(c1cccc(N2CCC(CCO)C2)n1)NCCCCN(C)C c1(CC)cc2c(c(=O)o1)C(c1c(Cl)scc1Cl)NC(=O)N2C(=O)OC C(=O)(C(C(=O)OC(C)(C)C)C(C)C)N1C(CNC(Cc2c(C)ocn2)=O)CC1 N1(C(C(n2ccc(C)n2)C)=O)CCC(C(=O)NCC(C)S(N)(=O)=O)CC1 C(N=c1[nH]c2c(c(=NCC(C)OC(F)F)[nH]1)CCCC2)C1N(CCC)CCC1 C1(N(C(CNC(CCCC)=O)=O)C)CN(C(=O)Cc2ncsc2Cl)CC1(C)C C(CCCCCCO)CNC(=O)CCc1ccoc1.C12(CC1)N(C)C2=O n1(CC)nc(C(=O)NCC2(C)CCC(NC(=O)CSc3nncs3)C2)cc1C C(=O)(C1=CCCCC1)N1CC(N(C)C(C2CCCCN2C2CCCC2)=O)C(O)C1 N1(C(C(c2ccccc2)OC)=O)CCC(C(C)NC(c2cc(Cl)nn2C)=O)CC1 c1(C(N2CCC(CN(C(CNC(C(CC)C)=O)=O)C)C2)=O)ncc(C)cc1F C(=O)(CC(CC(C)C)NC(=O)CCCCOC)NC1CCCC(C=C)C1 CC1CCC(O)(C(=O)NCC2CC(O)(CNC(C3SCCCS3)=O)C2)CC1 N1(C(c2nc(Cl)cs2)C(=O)NCCC)C2C=C(c3ccccc3)CC1CC2 C(C)(C)(CCC(F)F)NC(c1cccc(Br)c1)C N1(CC=C)C(=S)NC(c2sc(Cl)nc2Cl)C2=C1CCN(c1ccc(F)cc1)C2=O C(=O)(C(C)CC(C)C)N(CCC(=O)NC(c1ccnn1C)CC)CC#C CCCC(C(=O)N1CCN(C(c2cc(N)cnc2C)=O)C(C)C1C)C(C)C c1(NC(C(CC)NC(=O)C=Cc2cscn2)=O)ccc2c(c1)OCO2 CC(C)(CC(=O)N1CCC(C)(CCNC(C23CCN(CC2)C3)=O)C1)CC(F)F C(CNC(c1sccc1C#N)=O)(CC(F)(F)F)NC(CN1CCC(C)CC1)=O c1(CC)onc(C(N2CCCC2C2CCN(C(c3c[nH]c(Br)c3)=O)C2)=O)c1C c1(C(=O)NCC2N(C(CC3N(C)CC=CC3)=O)CC2)c(F)cc(CO)cc1F c1(C(N2CC(O)CC(NC(C(CCC)OCC)=O)C2)=O)nc(C)c(C)nc1C c1(C(=O)NCC(CC)(CC)NC(=O)C(F)=C(C)C)cncc2ncccc12 Cc1cccc(C(C)C(=O)NC2CC(CNC(=O)CCc3cncc(O)c3)C2)c1 Cc1nc2cc(C(=O)NC3CCC3NC(c3n[nH]c4c3CCC4)=O)ccc2s1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(C(C)NC(=O)NC)=O C1(CCNC(C2(OC)CC2)=O)CCN(C(=O)Cc2cncnc2O)C(C)C1 CC(C)(C)C(O)CNC(C1CC(=O)CN1C(C1COCC1C(N)=O)=O)=O Cc1cc(C(=O)NC(C2CCCN2C(c2ncoc2C)=O)C)ccc1Br C1(N(C(c2cnccn2)=O)CC)CCCN(C(=O)C(C)n2cnnn2)C1 c1(C(=O)NCCN(c2ccc(C(F)(F)F)cc2)C(CCC)=O)cccnc1NC Cc1ccn(CC(=O)NC2(CC(=O)NC3CSC3)CCC2)n1 C1(NC(c2cnc(CCCC)s2)=O)CC2CC(C1)N(C(C1(C3CC3)CCC1)=O)C2 N1(C(c2c(C)c[nH]n2)=O)CC(NC(c2cc3occc3[nH]2)=O)CC(F)C1 Cn1nccc1C=CCNC(C1(C(=O)N(C)C)CC1)=O C(=O)(CC(C)CC(C)C)N(C1CN(C(c2ccc(C)c(C)n2)=O)CC12CC2)C C(C(=O)N(C)Cc1ccncc1)(C(C)(C)O)NC(C(C)=C1CC1)=O c1(C(=O)NC2CC(OC)CN(C(COCCSC)=O)C2)cnc2ncc(Cl)cn12 C1(NC(=O)NCC(=O)OCC)CCC(CC(C)C)CC1.N12CCCC(C1)C2=O N1(C(=O)C=Cc2nccs2)CCCCC1CCNC(C1(c2nccs2)CC1)=O