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199,c1(C(N(C2CN(C(C3=C(C)OCC3)=O)CC23CC3)C)=O)ccc2nnc(C)n2c1 200,N1(C(CCC(N)=O)=O)CCCC2CN(C(c3ccc(CCF)cc3)=O)CC12 201,Cn1cc([N+](=O)[O-])cc1C(=O)NCC(C)(C1CC1)NC(C1C=CCC1)=O 202,CC1=C(C(=O)NCC2CC2NC(c2cccc(NCC(F)(F)F)c2)=O)CCC1 203,c1(OC)cc(CN2CC3CN(C(c4ccnc(OC)c4Br)=O)CC23)cc(C)c1 204,c1(C(=O)NC(C(C)C)(C)CNC(C2CCOC2)=O)cc2c(F)cc(F)cc2o1 205,c1(C(N2CCCCC(NC(C3(F)CCCC3)=O)C2)=O)cccn2nnnc12 206,CCCC(CC(=O)NC1CCN(OCC)CC1)NC(=O)C=C(C)C(C)(C)C 207,C(=O)(C(CO)NC(C1CCN(C(=O)C(c2ccco2)SC)C1)=O)OC 208,c1(C(=O)NC2CCCCN(C(C3C(C)CC(C)O3)=O)C2)nc2cc(F)ccc2s1 209,C1(C(=O)NCC(=C2CN(c3nnc(C(C)C)o3)C2)F)CCC(O)CN1C 210,CC1CC(C(=O)NCC(c2ccc(Cl)cc2)O)N(C(=O)CCc2ccco2)C1 211,N1(C(CC(=O)N(C)C)=O)CCC2CCC(NC(=O)CC3CN4CCN3CC4)C12 212,C12CCOC(C1)CCNC(=O)C2.C(CC(=O)NC1CC(CF)C1)OC(C)=O 213,c1(C(N(CCCNC(=O)C2CC2)CC)=O)nc(C(C)C)ncc1Cl 214,C(C(C(=O)N(C1CCC(NC(c2ccn(CC3CC3)n2)=O)C1)C)OC)OC 215,Cc1cc(CNC(C2(C(C)(F)F)CCO2)=O)ccc1F 216,CC1(C)CC(C)(NC(=O)C(CNC(=O)CCCC2CCCO2)CC2CC2)C1 217,N1(C(CC(C)O)=O)CC2(CNC(c3csc(-c4ncc[nH]4)n3)=O)CC1CO2 218,C1(CCC(=O)NCCc2cccs2)CCCCN1C(c1coc(C(F)F)n1)=O 219,C(=O)(C(CC(C)(C)C)NC(=O)CC(C)(F)F)NCC(CN(C)C)O 220,C(CC(C(=O)NC1CCOC1=O)NC(=O)C(C1CCC1)OCC)=CC 221,c1(COC)nc(NCc2c[nH]c(=N)s2)cc(N(CCCC2CCOC2)C)n1 222,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(C(C)OCCC#C)=O)C(OC)C1 223,C=CCCCC(C(=O)NCC1CC12CCOCC2)NC(=O)Cc1ncc(C)s1 224,c1(C(=O)NC2CC(NC(=O)CCSc3ccccc3)C2)csc2ccccc12 225,CCC(C)(F)C(=O)N1CC(NC(c2cc(-c3ccc(F)cc3)no2)=O)C(C)C1 226,C1(NC(C2C(C=C)OCC2)=O)CC12CCN(C(c1ncoc1CC)=O)CC2 227,C=CC(C)(C)C(=O)NC(CN(C)C(c1ccncc1CC)=O)CC 228,C(CCCCC(=O)NCc1nc(CC(=O)C(C)C)cs1)n1cc(C(C)C(=O)O)nn1 229,CC(C)C(CCN(C)C(C1(C(N)=O)CC1)=O)NC(C1(C)CCCCO1)=O 230,c1(NC(=O)CN2CCN(C(=O)CC3CCCCO3)CC2)ccc(I)nc1Cl 231,Cc1ccc2sc(NCC(CC(C)C)NC(c3ccc4oc(O)nc4n3)=O)nc2c1 232,c1(NCCc2nc[nH]n2)cc(OCC)ccc1OC.C1(C(=O)OC)CC1C(=O)CCN 233,C(C(C(=O)NCC1CCOCC1)N(C)Cc1ccsc1)(C1CC1)OCC 234,c1(NC(CSCC#C)=O)cccc(NC(C2CC2C(=O)NC)=O)c1 235,c1(COCC(C(=O)NCC(=O)NC(C(C)C)(C)C)(C)C)ccc(O)nc1 236,N#CC1CN(C(C2(Br)CCC2)=O)CC1NC(=O)Cc1ccc(OCC#N)cc1 237,c1(C(=O)NCC(CN(C)C(c2c[nH]nc2C2CCC2)=O)O)cnccc1N(C)C 238,C(C(N=c1[nH]c(NCC(C2CCCCC2)F)nc2c1SCC2)N1CCCC1)OC 239,Cc1nn(CC(F)(F)F)c(Cl)c1C(=O)NC1CCN(C(c2cnc[nH]2)=O)C(C)C1 240,C1(C(=O)NCC2N(C(C3C(C)CCS3)=O)CC2)CCN(S(C)(=O)=O)CC1 241,CC(C)CCC(C)NC(C1(c2nnnn2CCCNC2CC2)CCOC1)=O 242,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(NC(=O)CCC2OCCO2)C1 243,Cc1cc(NC(C2OCCN(C)C2=O)=O)ccc1NC(=O)CCC(C)(C)F 244,c1(NCC(C)(C2CC2)NC(c2cncc(OCC)c2)=O)nc2cc(Br)ccc2o1 245,c1(C(=O)NC2CCN(C(c3cc(C)nc(O)c3)=O)C2)cn2cc[nH]c(=O)c2n1 246,c1(OC)cc(C(N2CCCCC2c2nc[nH]n2)=O)nc2ccccc12 247,CC1(O)CC(NC(C2CSCN2C(=O)CCC2CCCC2)=O)C1 248,N1(C(c2c(CC)nc(=N)[nH]c2C)=O)CC2CCC1CN2C(C1CCCC1C)=O 249,Cc1cc(F)ccc1CC(=O)NC1CC(CNC(c2n[nH]c(C)c2F)=O)C1(C)C 250,c1(C(N2CCCC(CN(C(C3ON=C(C)C3C)=O)C)C2)=O)c[nH]c(=N)nc1O 251,C1(CNC(=O)C(O)CC2CCCC2)CC2(CC2)CO1.c12nc(n[nH]1)C1CN(C1)C2 252,CC(CN1CCOC1=O)N=c1[nH]c(=NCc2cnccc2Cl)[nH]c2c1COCC2 253,C(=O)(CCCCNC(=O)C(C)C)NC1C(NC(C2C(CCCCC)CCC2)=O)C1 254,Cc1ccc(Cl)c(CN)c1.c1(NC2(C=O)CCC2)ncnc(Cl)c1Br 255,CC(CC(F)(F)F)C(=O)NC1CCCC(N(C(=O)CSc2cccc(Cl)c2)C)C1 256,C1(NC(c2c(OCC)nccc2)=O)CCN(C(c2cnc(OC)nc2)=O)C1(C)C 257,CCC(CC)(C(=O)NC1CCC(CNC(c2cc(N)ccc2O)=O)CC1)OC 258,c1(N(C(c2ccc(NC(=O)NC3CC3)cc2)C(=O)NCCCO)C)ccc(Cl)cc1 259,C12C3CC4CN(C1C4C3)C(=O)CC1(CC1)OCC(=O)N2.c1(O)cccc(F)c1O 260,N1(C(C(C)(C)SC)=O)CCC(C2(NC(=O)CC(C)n3ccnc3)CC2)C1 261,c1(C(N2CCC(CCCO)C2)C(=O)NCC(C)C)nn(C)c(Cl)c1Br 262,N1(C(CCNC(=O)OC)=O)CC=CC1(C)C(=O)NCCc1ccc(O)cn1 263,C(CC(=O)N1CCN(C(C2(C(=O)OC)CC2)=O)CC1)(C(F)F)NC(=O)N.C(C)(C)(C)OC 264,N12CCC(CC1)C2.C1(C(CNC(C2(CCCC)CC2)=O)O)CCCO1 265,C(=O)(CCCCCF)NC(CN(CCOCCOC)C(C)C)C.C1C(=O)N1 266,C1(CC)C(=O)N(C)CCN1C(C1COCC1NC(c1cc2ccccc2[nH]1)=O)=O 267,CN1CCC(CCNC(C2(NC(=O)CNC(=O)CC(C)(C)C)CCCC2)=O)C1=O 268,C1(C)(C(=O)NCC(CC=C)N(C)C)CCCN(C(c2ccncc2)=O)C1 269,c1(C(C)=O)ccc(CC(=O)NC2C=CC(CCNC(=O)CCc3ccsc3)C2)cc1 270,c1(C(=O)NC(CNC(C(CCC)C)=O)C)cc([N+](=O)[O-])ccc1N(C)C 271,c1(C(N(C)CC2CCCN(C(C=CC(C)C)=O)C2)=O)ccc(F)c(F)c1 272,C=CC(CC)C(=O)N(CC(=O)N(CC(O)CNc1ccccc1F)C)CC(C)C 273,N1(C(C2(C(=O)OC)CC2)=O)CCCC2CCN(C(=O)C(Br)=C(C)C)CC12 274,c1(-n2c(CCn3cncn3)nc(C(CC)C)n2)cc(Br)ccc1OCC 275,S(=O)(=O)(c1ccc(Cl)c2ncccc12)NC1C(=O)N(c2cc(Br)c(O)cc2O)CCC1 276,C(CN=C(NCc1c(C)noc1C)NC1CCCCC1)N(C(C)=O)C 277,CCC(C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)(C)C)C(C)(C)CC 278,N1(C(Cc2cc(C)sc2)=O)CCCC(NC(=O)CCSc2ccccn2)CC1 279,C(CC(C)(C)C(=O)NCCC1CCCN(C(=O)C(C)CSC(F)(F)F)CC1)OC 280,C=C(Cl)C(C)(C)C(=O)NCCCN1CCC1(C)c1ccccc1 281,c1(C(=O)NCC(CNC(c2c(C)onc2C2CC2)=O)C)ccc([N+](=O)[O-])cc1F 282,CCCC(CCCNC(=O)CCC(=O)NCC)N=c1[nH]c(Cl)nc2c1CCOC2 283,CCCC(C)(CCC)C(=O)NC1CC2(C1)CC2C(=O)NCC(CO)N(C)C 284,CCC(CC(=O)NCCC1(C(N2CC(CC)C2)=O)CCC1)C(C)C 285,Cc1cc(CC(=O)NCC2CC3CC2N(C(=O)CN2CCCC2=O)C3)cc(F)c1 286,c1(C(=O)NC2(CC=C)CCN(C(C3CC=CCC3)=O)C2)ccc(C#N)n1C 287,C12(C(=O)NC3(C)CN(C(C4CN5CCC4CC5)=O)C3)CCCCC1NC(=O)CC2 288,C1(CC(=O)NC2CC(CCNC(C3CC34CCOC4)=O)C2)CC2(CCC2)C1 289,C1(C(=O)NC2(c3ccc(C)cc3)CCC2)CCCN(c2ccc(Cl)c(Cl)c2)C1=O 290,C(N=c1[nH]c2c(c(=NCc3n[nH]cc3C3CCC3)[nH]1)CCC2)c1cc(C)ncn1 291,Cc1ncsc1C(=O)NC(c1cn(CC(=O)N(CC)Cc2c[nH]ccc2=O)nn1)C 292,N1(C(c2n(CC)nnc2)=O)CCC2(CCC(NC(C3(OC)CC3)=O)C2)C1 293,C#CC1(NC(=O)CC2CN(C(=O)CC(C)(C)C3CC3)CC2C=CC)CC2CCCC12 294,Cc1ccc(C(=O)NC23CC(C2)N(C(=O)C=Cc2nccs2)C3)c(Cl)c1C 295,C#CCCC(O)C(=O)NCC1CCN1C(c1ccnc(C(C)(F)F)c1)=O 296,c1(C(C(=O)NC(C)CN(C)Cc2ccc(Cl)cc2)N2CCCC2)nc(Br)cn1C 297,C1(CCC(=O)N(CCN(C(=O)CN(C)C(N)=O)CC)CC)CCC(O)CC1 298,c1(NC(N(C)Cc2c(C)n[nH]c2)=O)ccc(C2CC2(F)F)cc1 299,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)COC2(C)CCOCC2)=O)c1F 300,CCCC(O)(CNC(c1ccc(NC(=O)CN(C)C)cn1)=O)CCC 301,c1(NC)ccc(C(=O)N(C)CC2CCCN(C(=O)Cn3ncccc3=O)C2)nc1 302,CC1(NC(C2CCC(CNC(=O)C(O)C3CC3)C2)=O)CC2CCC1C2 303,N(C)(C1CS(=O)(=O)c2ccccc21)CCNc1ccc2ccc(OC)cc2c1 304,c1(CC(=O)NC(C2CCCCN2C(c2cccn2C2CC2)=O)C)ccc(O)nc1 305,N1(CC(C)NC(=O)Cn2cc(C(C)O)nn2)CCN(C(=O)C(Cl)=CCl)CC1 306,S1(=O)(=O)c2ccc(cc2)OC2CCN1CC2.N1(CCCNC)CC=C(C)CC1 307,C=CCCCC(C1CC1)NC(=O)CCN(C(=O)CCC1CCCOC1)CCO 308,c1(C(=O)OC(C(=O)Nc2c(CC)cccc2)C)cnc(C)c(N)c1 309,C1(C)(NC(c2c(C(C)C)occ2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 310,CC1(CNC(=O)CC2CCOCC2)CC(F)(F)CN1C(c1cnsn1)=O 311,c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2nccnc12 312,C(=O)(C(=O)C(C)(C)C)N1CC(CNC(CN2CC(C)(C)C2)=O)(OC)C1 313,N1(C(C2C(C)(C)COC2)=O)CCc2[nH]nc(CNC(C3CCOC3=O)=O)c2C1 314,c1(C(N2CC(CC(=O)OC)OCC2)=O)ccc(F)c(-c2cc(F)ccc2F)n1 315,O(NC(=O)C(CCC1CC1)NC(=O)CSCCF)Cc1n(C)ncn1 316,c1(C(=O)NC2C(CNC(c3ccn4nncc4c3)=O)CC2)cc2cccnc2s1 317,N1(CC)CCN(C(C2(CO)C=CCN2C(=O)OC(C)(C)C)=O)C(C)C1 318,Cc1ncccc1CC(=O)NC1CC(CC(=O)Nc2cnccc2CO)C1 319,C1(C(=O)Nc2cscn2)CC(C(N2CC(=CCO)C2)=O)CCO1 320,C1(CN(C)C(=O)C2CC2)CN(C(C2(O)CC2(C)C)=O)CCO1 321,N1(C(C2N(C(c3c(C)nc(CC)o3)=O)CCC2)=O)CCCC(C)C1CO 322,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOCCC(C)O)C2 323,c1(C(=O)NCCC(C)N(C(C(C(C)C)SC)=O)C)c(C)nn(CCO)c1C 324,c1(CNC(C(COC)(C)C)c2nnnn2CCCSC)nn(C)c(Cl)c1Br 325,Fc1ccc(C2=CCN(c3nc(N4CCOCC4)nc4sccc34)CC2)cc1.CCO 326,c1(C(=O)NCCC(C)NC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 327,N1(C(C=CCCC=C(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccc1C 328,c1(C(N2CC(C)(NC(C3(C(F)(F)F)CC3)=O)C2)=O)ccc(=O)n(CCF)n1 329,CC(C(=O)N1CCC(CNC(=O)C(F)=C2CCCC2)C1(C)C)C(C)(C)C 330,c1(NC(c2cc(Cl)no2)C)[nH]c(=NCC2CCN(C)C(=O)C2)nc2c1cnn2C 331,C=CCCCC(C(=O)NCC1(C)CCC2CC12)NC(=O)CC(C)COC 332,CC1(C)CC(C(=O)NC(C2CCCC2)CNC(c2cc[nH]c2)=O)CC(C)(C)O1 333,c1(CNC(C2C3CCC23)=O)cnn2c1CN(C(C1CCCC13OCCO3)=O)CC2 334,c1(NCC2CCC(NC(C(CCC)OC)=O)C2)ccc([N+](=O)[O-])c(NC(C)=O)c1 335,c1(C(=O)NC(C(=O)NC(CCCCC)C)CC)cc2cccnc2[nH]1 336,c1(C(=O)NC2C(NC(C(CC=C)c3ccccc3)=O)C2)csc([N+](=O)[O-])c1 337,c1(-c2n(N(C)CC3(C(F)(F)F)CC3)ncc2)cn(C)nc1-c1ccc(Cl)s1 338,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C(=O)NCC2CC2)C(CF)C1 339,N1(C(c2nnc(CC)s2)=O)CCCC(C2CC2NC(C2CCCS2)=O)C1 340,C1(CC)CCCN(C(c2csc(CNC(=O)CCc3cnc(C)s3)c2)=O)CC1 341,c1(C(N(C2CC3CCC(C2)N3)C(CC)CO)=O)csc2ccc(Br)cc12 342,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 343,C#Cc1ccc(C(=O)NCC(c2scnc2C)(C)C)o1 344,c1(NC(C2(COC)CN(C(=O)CCC3(C)CC3(F)F)C2)=O)cccc(CO)n1 345,C12(CC(=O)N(C(CCNC(c3cnc(C)n3C)=O)C)C)CC3CC(CC(C3)C1)C2 346,C1(CN(C(C(C)=CC2CC2)=O)C)CCCN1C(=O)CSc1ccccc1 347,N1(C(C(C)O)=O)CCc2nc(CNC(c3ccc4ccccc4n3)=O)sc2C1 348,C1(C(CNc2n(CCC3(C)CC3(F)F)nnn2)(C)C)CCS(=O)(=O)C1 349,C(=O)(CCCc1nccs1)N1C(C)(C)C1.c1(S)ccccc1.C(C(=O)N)=C(C)Cl 350,CCCC(C(=O)N1CC(NC(c2ccc(C(C)C)cc2)=O)C1)S(N)(=O)=O 351,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 352,CC1CC(NC(=O)C=Cc2cncs2)CCN1C(C1CCC(C(N)=O)C1)=O 353,CC1(CN)CN(C(c2cc(-c3ccco3)nn2C2CC2)=O)CCO1 354,c1(OC)ccc(F)cc1C(=O)C(=O)NC(CNC(=O)C1=C(C)OCC1)C1CCC1 355,c1(OC(C)C)cncc(C(=O)NC(C2CCCN2C(=O)Cn2ccnc2)C)c1C 356,C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CC(N(C)C(c2cc3ccsc3s2)=O)C1 357,C(=O)(CC(C)CC(=O)OC)NC1(CC(=O)NC2(CC(=O)OC)CC2)CC1 358,C(CN=c1[nH]c(=NCC2CCCO2)[nH]c2cccc(F)c12)c1cnc(C)s1 359,c1(CC(N2CCC(NC(CCC3C(C)C3)=O)C2C)=O)c[nH]c2cnccc12 360,C(=O)(C(O)C(F)(F)F)N(C(CC(=O)NCC(C)(C)OCC)(C)C)C 361,C1(C(N(CC(C)CO)C)=O)C2CC(O)C(C2)N1C(C1CN(C)CCO1)=O 362,CCCCCCCCCC(C)CC(=O)NCCN(C)C(c1ccnc(Cl)c1Cl)=O 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452,Cc1ccc([N+](=O)[O-])c(NNC(=O)c2c[nH]c3cc(Cl)ccc23)n1 453,C1(CNc2nc(COC)nc(N3CCC(CF)C3)c2)CC2(CCC2)CCO1 454,c1(C(=O)NC2C(NC(C(C)OCC#C)=O)C2)cnc(Nc2cccnc2)cn1 455,N1(C(c2cccc(OC)c2)=O)CC(C2CN(C(C3CC4CCC4C3)=O)C2)C1 456,c1(OCN(C(=O)Nc2ccc(-n3cnnc3)cc2)C2CC2)cccc(F)c1 457,c1(C(=O)NCCC(C)CCNC(=O)C(F)CC2CCCC2)cccc2ccnn12 458,C(N=c1[nH]c(=NC2CC=CCC2)c2[nH]ccc2[nH]1)c1ccc(C(F)(F)F)nc1 459,Cc1c(C(=O)NCCCn2ccnn2)ccc2nn[nH]c12 460,N1(C(C(CC)=CC)=O)CC(C)CN(C(c2ccc(SC)cc2)=O)CC1C 461,C1(C(=O)NC(c2ccccc2F)C)CC(F)CN1C(=O)C(c1ccccc1)O 462,N1(C(C(C2CCOC2)NC(CCn2ncc(C)c2)=O)=O)CCC(CCO)CC1 463,N1(C(=O)C(F)(F)F)CCc2nc(C)sc2C1.C#Cc1ccncn1 464,C=C(Cl)CCC(=O)NCC(C)(CNC(c1csc(C(C)=O)n1)=O)OC 465,c1(-c2c(CNC3C(c4cccc(F)c4)CC3)cno2)cccc2ccccc12 466,C1(NC(C(C=C)(F)F)=O)CCC2CN(C(c3csc(S)n3)=O)CC2C1 467,c1(C(CN(C)C)NC(C)CN2CCSCC2)c2c(nn1C)CCCC2 468,C=CC1CN(C(c2ccc(F)c(C)c2)=O)CC1NC(C1CCCS1)=O 469,N1(C(CCCCC#N)=O)CCC(CNC(c2cccc3nccn23)=O)C(F)(F)C1 470,c1(C(=O)NCCCC(C)NC(c2cnc(SC)s2)=O)c(F)cncc1Cl 471,c1(CC)cc(F)c(NC(c2ccc(OC)c(Br)c2Cl)=O)c(F)c1 472,C1(N(C(c2c(C)oc(CO)n2)=O)C)CCCCN(C(=O)C2=CCSC2)C1 473,c1(OC)ccc(CNC2CCCN2C(c2cnc(I)cn2)=O)cn1 474,C1(C(=O)NCC(C(C)C)O)CCN(C(C2CC3CCC2C3)=O)C1(C)C 475,C1(C(N(CCC)Cc2cn(C)cn2)=O)COCCN(C(=O)CCOCC2CC2)C1 476,C1(CNC(C(C)N(C)C)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 477,c1(NC(N2CCN(c3ccccc3Br)CC2)=O)ccc(Cl)cc1C1CCCN1 478,Cc1c(NC(c2ccc(C(C)C)cc2)C)ncnc1NCC1COC(C)(C)C1 479,C(C)(CCCC(C)C)NC(CC1(C=C)CN(C(=O)C=Cc2ccc[nH]2)C1)=O 480,Cn1ccc2cccc(C(N3CC(F)CC3CNC(c3cc(N)ccn3)=O)=O)c12 481,C(=O)(CCCCC(=O)N1CC2(CC2C(=O)NC2CC(CO)C(O)C2O)C1)OC 482,C(=O)(C(O)C(C)CC)NC(c1ccc(OC)cc1)(C(=O)OC)C 483,c1(N2CCCC(C(C)NC(CSCC(N)=O)=O)C2)nc2ncc(Cl)cc2s1 484,C12CCS(=O)(=O)CN1C(=O)NCCO2.C=CCCCOC(C)(C)C 485,C(=O)(C1CCSc2ccccc21)NC(C(=O)OC)Cc1cc2c[nH]nc2cc1F 486,C1(NC(c2sccc2F)=O)CC2CCC1CN2C(=O)Cn1cc(CO)nn1 487,C#Cc1cc(NC(=O)C(CNC(=O)C(C)(CO)OC)OC)cc(F)c1 488,N1(C(C2C=CC(NC(C#CC(C)(C)O)=O)C2)=O)CCOC2(CCCC2)C1 489,N#CC1CCCCN1C(c1cccc(CNC(=O)Cc2ccc(F)cc2)n1)=O 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690,CCCC(CC(=O)NCC1(O)CCCC1(C)C)NC(c1c[nH]nc1Cl)=O 691,c1(NCC2C(NC(c3cc(C(C)=O)on3)=O)CCC2)nn(C)cc1[N+](=O)[O-] 692,c1(CC(=O)NC2(CO)CN(C(CS(CC)=O)=O)C2)cc(F)ccc1F 693,CCC1=NOC(CC(N2CC3CC3(NC(C3CC(=O)N(CC)C3)=O)C2)=O)C1 694,C1(C(=O)NCC2C(C(=O)NCC3(CC(=O)OC)CC3)C2)CCCCN1C 695,C1(CNC(=O)CONC(=O)C2CCOC2)(COC2CC2)CCOC1 696,Cc1nc(NC2CN(C(C3C=CC=CC=C3)=O)CCC2C(F)(F)F)c(C)c(O)n1 697,C1(NC(C(C)NC(N)=O)=O)CN(C(=O)CSc2cccs2)CC1C 698,c1ccccc1F.C1(C)(NC(C(C)OCC)=O)CC(NC(=O)CC)C1 699,c1(CC)cc(C(=O)NC2C3CN(C(c4cc(C)c(Cl)cn4)=O)CC23)ccc1F 700,CC1CC(NC(c2ccc(C(F)F)cc2)=O)CN1C(=O)C(F)=CC1CC1 701,c1(C(=O)N(C(N2CC(C3CCCO3)C2)=O)C2CC2)c(O)ccc(F)c1Br 702,N1(C(c2c(C)noc2C)C(=O)NCCC#N)CCC2(CCC2)C1 703,c1(N(C2CC=CCC2)C(c2n(CC)nnn2)C2CC2)ccc(-c2ccnn2C)cc1 704,c1(NC(C(C)NC(c2ccc(CO)nc2)=O)=O)cccc2ccoc12 705,C(=O)(C(O)C1=CCCCC1)NCCCCCCC(=O)NCC1(C)CC1 706,N1(C(C=CC(C)(C)SC)=O)CCN(C2CCN(C(C3CC(C)C3)=O)CC2)CC1 707,c1(C(=O)NC(C)C(C)(C)NC(C2CCC2C(C)(C)C)=O)ccc2cn(C)nc2c1 708,c12ncc(Cl)cc1C(=O)N2.c1(-c2cncc(C(=O)OC)c2)cccc(CO)c1C 709,N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1[nH]cnc1CC)=O 710,C1(C)COCCO1.C(=O)(C1C2C(C2)C(=O)N1)OC.C(F)(F)F 711,C1(C(N2CCC(CCOC)(NC(=O)CCOCC(F)F)C2)=O)CCCC(C)(C)O1 712,C12CC(CCN1C(=O)CC1COCCO1)NC2=O.C12(SC)CC(C1)C2 713,N1(C(C(c2ccc(C)o2)C)=O)CCC(C(=O)NCCCN2CCC2)C(C)(C)C1 714,N1(C(C23N(C(CC4=NNC(=O)C4)=O)CCC2C3)=O)CCc2nocc2C1 715,O=C(C(F)CC1CCOC1)NCCCc1cnn[nH]1 716,N1(C(N2CCOCC2Cc2cnc(C)s2)=O)CCC2CCCCCC2C1 717,c1(COC)ncc(I)c(C(=O)NCc2cn(C(C)(C)C(=O)O)nn2)n1 718,CCCC(C)CC(=O)NCC(C(F)(F)F)N1CCN(C(c2ccco2)=O)CC1 719,C1(CCNC(c2ccc(C(F)F)o2)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 720,c1(C(=O)NC2C3(CC(NC(C(C)CN4CCCCC4)=O)C3)C2)cccc(N)c1F 721,C1(CC(=O)NC2C(C)C2(C)C)C2CCCC2N1C(=O)C(C1CCOCC1)=O 722,C1(C(=O)OCC)COCCN(C(c2cc(C)cc(Cl)c2)C(=O)NC2COC2)C1 723,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1CC(N(C(C=C(CC)C)=O)C)C(C)CC1 724,C1(CC)CN(C(=O)C=CCOCCOCc2coc(SC)n2)CCS1 725,N1(C(C(=O)N(CC=C)C)=O)CCn2cc(C)nc2C1.c12ccc(cc1)SCC2 726,C1(c2nnnn2CCSC)(NC(CC)C2CC2)CC2(C1)OCCO2 727,CC(C)C(C(=O)NC1CC(NC(=O)CCCc2cccs2)C1)c1ccncc1 728,C1(C(N2CCC(NC(c3ccncc3)=O)C2)=O)C2CC2CN1C(=O)C1CC1 729,N1(C(c2cn(CC)nc2)=O)CCN(C(=O)COc2ccc(F)cc2)C(C)C1C 730,C1(CNC(c2c(CC)nc[nH]2)=O)CN(C)CCN1C(=O)COc1ccsn1 731,C(=O)(C#CC1CCCO1)NC1C(CNC(C(=O)Nc2ccc(C)cc2C)=O)CCC1 732,S(=O)(=O)(c1cc(C(=O)O)ccc1Cl)N1CC2C(NC(C(C)OC)=O)C2C1 733,CCC(C(=O)NCCCC(CO)NC(c1ccc(C)nc1N)=O)C(C)C 734,C1(CNC(C2(COC)CCCO2)=O)CCCCN(C(c2ncn(C)n2)=O)C1 735,N1(C(C2CC(C)CN2Cc2c(Cl)cnn2C)=O)CCC(=O)N(C)CC1 736,C1(C(=O)NC2(CC(=O)NC(CN(C(C)C)C)C)CC2)CN(c2nncs2)C1 737,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C(C)C2CCCC2)CC1C)=O 738,C1(C(C)NC(C(F)OC)=O)CCN(C(c2ccccc2OC)=O)CC1 739,C1(C)(C(N2CCCCC(CNC(CC(C=C)C)=O)C2)=O)CCC2(CC1)OCCO2 740,N1(C(c2cc(CC)oc2C)=O)C2CCC(C2)C1C(=O)N(C1CCN(C)CC1)C 741,c1(SC)ccc(C(=O)NC2CCCCC2NC(=O)C(O)C(F)F)c(Cl)c1 742,c1(OCC)nc(NCCC(C)NC(=O)C(CO)c2ccccc2)ncc1Cl 743,C1(C(=O)NC2CCC(NC(=O)C(C)SC)CC2)(OC)CCCCC1 744,N1(C(c2c(C)nncc2)=O)CCC(n2cccn2)(CNC(C2CCSCC2)=O)CC1 745,N1(C(CN(CC)CC)=O)CC(CSC)C2(C1)CN(C(=O)CS(C)(=O)=O)C2 746,Cc1cccc(CNC(C23CC2CN(C(C2CCC(=O)N2C)=O)C3)=O)c1O 747,c1(NC(CNC(C2(C)CCC(C)C2)=O)C2CC2)cc(=O)n2cc(Cl)ccc2n1 748,n1(CC)ccnc1C=CC(N1CCC1CNC(=O)C(c1ccc(Cl)cc1)O)=O 749,C1(CCC(=O)NCC(C)CN(C(=O)CN(c2cnccn2)C)C)CCCCN1C 750,C1(C(=O)NC(CCCNC(C(C)NC(=O)OC)=O)(C)C)CCc2nnc(O)cc2C1 751,C#CCC(C)(C(=O)NC(c1cnc[nH]1)C)NC(C1CCCC(=O)CC1)=O 752,c1(N2CC(C)C(CNC(c3ccco3)=O)CC2)ncnc2c(Br)cccc12 753,C1(C(N2CC3(CN(C(C(C4CCCC4)OCC)=O)C3)C2)=O)CCc2ccnn2C1 754,C1(C(=O)NCCCCNC(Cc2nc(-c3ccc(C)o3)sc2)=O)COCC(C)O1 755,C(=O)(CCCCCC(C)(C)C)NC1(CF)CCN(C(CCc2n(C)cnc2)=O)C1 756,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)cccc3Cl)=O)CC2)C1 757,C1(NC(C(C)(C)N2CCCCC2)=O)CC2(C1)CC(NC(C1CCC1C#N)=O)C2 758,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(F)(F)F)nn2)=O)n[nH]1 759,c1(CC(=O)NCC(CN(C(C(C2CCCC2)OC)=O)C)O)cccc2occc12 760,C(=O)(C1=CCCCCC1)NC1CC(N(C)C(C2CC23CCOC3)=O)C1 761,C1(C)(C(N2CCC(N(C(=O)CNC(N)=O)CC#C)C2)=O)CCOC(C)C1 762,C1(C2CCCN(C(=O)C=C(C)C(F)F)C2)(NC(CN(CCOC)C)=O)CC1 763,c1(NCC(=O)NC(=O)OC)c(NC(C2(C)CC(C)=NO2)=O)cccc1[N+](=O)[O-] 764,Cc1cnn(C(C)C(=O)NCC2CCOC2C(=O)NCC=Cc2ccco2)c1 765,C(=O)(CCS(=O)(=O)CC(C)C)NC(C)CC1CN(C(C2CCOC2COC)=O)C1 766,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 767,C1(CC)CCN(C(C2CCCC(OC)C2)=O)C(C(=O)NCCn2nncc2C)C1 768,c1(C(N2CCCC(CN(C(C3CC(C(=O)OC)C3)=O)C)C2)=O)cnc(O)c(C)c1 769,C1(C)(C(=O)Nc2cc(NC(c3c(C)nn(C)c3C)C)ncn2)CC2(C1)CC(F)(F)C2 770,N1(C(C2C(=C)C2)=O)CC2(CCN(C(c3sc(Cl)c(Cl)c3OC)=O)CC2)CC1C 771,C1(C(=O)NC2(CO)CN(C(CC3C(C)C3)=O)C2)CCC(Cc2ccccc2)CC1 772,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(C1CCN(C)CC1)=O 773,Cc1cnc(CC(=O)N(CCCNC(=O)C(=O)NC2CC2)C(C)C)o1 774,C1(CC(=O)NC2CC2O)CCN(C(C2CC2(Cl)Cl)=O)C1 775,C#CCCN=C(NCC(C)Cc1cc(C)oc1C)NC1CCCC1 776,Cc1cccc(C(C(=O)NC2CC(CNC(C3(Cl)CC3)=O)CC2O)N(C)C)c1 777,C1(NC(C2CCS(=O)(=O)C2)=O)CC2CN(C(C3(n4ccnn4)CC3)=O)CC12 778,C=CCCCCC(=O)N1C2CCC1C(C(=O)N(C)CC1CCCOC1)C2 779,Cc1cc(Br)oc1C(N1CCC(Cn2cc(CC(O)C3CC3)nn2)CC1)=O 780,S(=O)(=O)(c1ccc(=NCCCCCCO)[nH]c1)NCCCc1ccc(C)c(F)c1 781,C1(C(=O)NCC(C)(CC(C)C)NC(CCOCCC)=O)COc2ccccc2C1 782,c1(CCNC(=O)CCC2(NC(C3CCCCO3)=O)CCC2)ncccc1F 783,C1(C(N2CCC(CN(C(=O)C)C)C2)=O)CCC(C(=O)NCCN(C)C)S1.CO 784,N1(C(CCCOC(C)C)=O)CC(O)CC1C(=O)Nc1cnccc1C(N)=O 785,N1(C(C=C(CCC)C)=O)CCN(C(c2ccc(CC)cc2C)=O)C(CCO)C1 786,CCCCC(C)CCC(=O)NCCOCCNC(c1cc2nn[nH]c2cc1F)=O 787,C1(C(=O)NCC(C2(O)CN(C(c3cc(C)[nH]n3)=O)C2)(C)C)CCC(=C(F)F)CC1 788,N1(C(C(CC)(C)CC)=O)CCCC2(C1)C(NC(=O)C(C)SC)CCN2C 789,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 790,c1(C(N2CCCN(C(C(C(CC)C)C)=O)CC2C)=O)nc(C)n2ccccc12 791,c1(CN2CC3C(C(N4CCC(CO)C4)=O)(C3)C2)ccc2occc2c1 792,CCN=C(NCCNC(C1CCC(NC(=O)OC(C)C)C1)=O)NC(C)(C)C 793,c1(OC(C(=O)N(CC(C)(C)NC(C(=Cc2ccco2)C)=O)C)C)cccc(C)c1 794,c1(NCC)ccccc1C(N1CCCC(COCC(=O)NCCN(C)C)C1)=O 795,N1(C(c2ccc(C(=O)OC)cc2)=O)CCC2CN(C(=O)CSCC(N)=O)CC2C1 796,c1(C(=O)NCC(CN(C(c2c(C)nn(C)n2)=O)C)(C)C)nc2ncccn2n1 797,C1(F)(CNC(C2(OCC)CCOC2)=O)CCCN(C(=O)C=Cc2ccsc2)CC1 798,C(CCCCC(=O)NCCCCNC(=O)CC1(C(F)(F)F)CCCC1)NC(C)=O 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1245,C1(CC2CN(C(CC3C=CC(C(=O)O)C3)=O)C2)CC2(CCO1)CC2 1246,Cc1cc(Br)cc(C)c1C(=O)N(CC(N1CCCC(C(F)F)C1)=O)C 1247,CCC(CC(=O)N1CCN(C(C2CCCN2C(=O)OC)=O)C(CO)C1)C(F)F 1248,N1(C(COCCC=C)=O)CC2CCC1C(OC(C1CCC1)=O)C2 1249,c1(OCCCC)ccc(NC(c2nocc2-c2cccc(Cl)c2)=O)c(C)c1 1250,c1(N2CC(C)(CCN(C)C)OCC2)nc(N2CCOC(C)(C)C2)nc2c1COCC2 1251,Cc1cc(NC(=O)CC2(C)CNCC2)c(C)nn1 1252,C1(CCC(=O)NCCN(C(C)C)C(C)C)CCCN(C(c2[nH]cnc2CO)=O)C1 1253,C(=O)(C1=C(C)CCN(C(c2noc(Cc3ccc4nccn4c3)n2)C)C1)OC 1254,c1(C(N2CCC(C(C)NC(C34COCC3C4)=O)C2)=O)cc(F)c(F)cc1N 1255,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1256,c12ccc(cc1)C(=O)NC2.N1(C(Cc2ncn(C)c2)=O)CC(O)CC1CCCO 1257,N1(C(c2nn(CC)nc2C)=O)CCC(C)C(CNC(C2CNC(=O)N2)=O)C1 1258,S(=O)(=O)(c1ccc(-c2cn(CC(=O)N(C(CCC3CC3)C(=O)O)C)nn2)o1)NC 1259,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1260,c1(CCC)cc(C(N2CC(F)(C(=O)NCC3CC(O)C3)C2)=O)n[nH]1 1261,C(=O)(CC1OCCc2ccsc21)NCCN(C(=O)C=CCOC(C)(C)C)C 1262,c1(NC(C2CCCC(NC(CCC#C)=O)C2)=O)cnc(Cl)c(F)c1 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1281,c1(OC)ncc(C)cc1C(=O)NC(CNC(=O)CC1COC(=O)C1)C1CC1 1282,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C(C)C(C)C)CC3C2)c1C#N 1283,C1(C(N2CC3CCN(C(=O)C4=COCCC4)C3C2)=O)CCCCC(F)(F)C1 1284,N1(C(C2CC(=O)N(CC3CC3)C2)=O)CCOCC1CC(N1CCCCCCC1)=O 1285,c1(OC)cc(C(N2CC(NC(=O)C(C)CN(C)C)CCC2C)=O)cc(Cl)c1O 1286,c1(CN2C(C(=O)NC3CC(C(C)O)C3)CCC2)ccccc1O 1287,C(=O)(CCC(F)(F)C(F)F)NC(C)CNC(=O)COCc1nc[nH]n1 1288,C1(C)(C(N(CCCNC(=O)CC(=O)Nc2nccs2)C)=O)CS(=O)(=O)C1 1289,Cc1ccc(C)c(-c2nnc(CN3CCNC(=O)C3c3ccccc3)o2)c1 1290,C1(CNC(=O)C2CC2)CN(C(=O)C(C2CCCCCC2)O)C2(CCC2)C1 1291,N1(Cc2n(C)c(O)nn2)C2CCC1CN(C(c1cnc(C3CC3)nc1)=O)C2 1292,C1(C(=O)OCC)CN2CCN1CC2.C1(N)CC(C)CN(C(=O)C(F)(F)C=CC=O)C1 1293,C(CCSC)(C(=O)NC(C)(CNC(C12CCC(CC1)C2)=O)CO)OC 1294,N1(C(C2N(C(CC)=O)CCCC2)=O)CCC(CNC(=O)CCN(C)C)C(O)C1 1295,c1(C(N(C2CCN(C(=O)CCCN(C)C(=O)CC)C2)CCC)=O)cnc(O)n1C 1296,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CCC2 1297,c1(C(=O)NC2C3(CNC(C(C)(C)N(C)C)=O)CCC(C2)C3)cccc2ccsc12 1298,N1(C(CC2(C)CCCO2)=O)CCN(C(C2CC3CCC(C2)O3)=O)C2(CCC2)C1 1299,C1(CC)CN(C(c2cc(N)cc(O)n2)=O)CCC1NC(=O)C(C)(C)CN(C)C 1300,N1(C(=O)NCc2cc(C(=O)OC)sc2)CC2CC(C)C2C1 1301,N1(CC(=O)NCCN(CCC)C(c2ccnc(OC)c2)=O)CCOCC1C 1302,CC(C)C(C)C(=O)N1CCN(CC(C)NC(=O)CCc2cn(C)cn2)CC1 1303,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1304,N1(C(c2cc(C(C)C)on2)=O)CC(NC(=O)Cc2cnco2)C2(CCOCC2)C1 1305,N1(C(CCCc2cc(C)sc2C)=O)CC2CC(NC(=O)C=CCF)C(C2)C1 1306,CCC(CC)C(C(=O)N1CCN(CCNC(C23CC(C)(CCO2)C3)=O)CC1)OC 1307,c1(CC)ccnc(C(=O)NC2CC23CC(NC(=O)C(F)(F)CN(C)C)C3)c1 1308,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1Br)=O)CC2 1309,N1(C(CC(=O)NCCSCC(C)C)=O)CC(NC(C23CC(C)(CO2)C3)=O)CC1C 1310,C1(CNC(=O)C=CC2CCCC2)CN(C(c2cn3c(n2)CCC3)=O)CCC1(F)F 1311,N1(C(C2C(CCOC)C2)=O)CCC(C)(N(C(C2(C(F)(F)F)CC2)=O)C2CC2)C1 1312,C=CCCC(C(=O)OC)NC(C1CN(C(c2cscn2)=O)C1)=O 1313,C1(CC(=O)NCC2C(CNC(C(CC)N(C)C)=O)C2)CCC2(CC1)CC2 1314,c1(-n2c(C3N(CC)CC3)nc(-c3cccs3)n2)ccc(OC)cc1F 1315,C(CCCCCN(C(=O)CCn1cccn1)C)NC(C(C)c1ccco1)=O 1316,N1(C(c2nccc(C)c2N)=O)CCC2(CCCC(CNC(=O)C=CCO)O2)CC1 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1335,C(C(=O)N1CC(C(=O)N(CCN=[N+]=[N-])C)C(F)(F)C1)(C(C)(C)C)SC 1336,C1(C(=O)NCC(C)NCCO)CCN(C(N2CCCC2)=O)C1 1337,c1(C(N2CCC(NC(CCCN(C)C)=O)C23CC3)=O)cc2n(n1)CCOC2 1338,c1(C(=O)NCC2(NC(c3cn(C)c(=O)n3C)=O)CC2)coc2ccc(F)cc12 1339,c1(C(=O)NCC(CC)(C)NC(=O)COCCO)cc(Cl)ccc1N.c1(S)nccn1C 1340,C(=O)(C(CC1CCC1)C1CCC1)NCCCCN(C(=O)C(c1cccnc1)O)C 1341,c1(C(C)C)ccc(CNC(Cc2ncco2)C(=O)O)o1 1342,C1(C(N2CC3CC(NC(c4csc5nccn45)=O)C3C2)=O)CCc2ccnn2C1 1343,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1344,C1(C(=O)OC)CN(C(C2(F)CN(C(C3CCCOC3)=O)C2)=O)CCC1O 1345,O=C(CCC(=O)NC1CCC(F)(CNC(=O)CSC2CC2)C1)c1cccs1 1346,CCCC(CNC(C1C=CCN1CC)=O)C(=O)N(CCN(C)C)CC 1347,CC#CCCCC(=O)NC(c1ccc(NC)cc1)C(=O)NC(C)COC(F)(F)F 1348,C1(Nc2c(C(=O)OC)scc2)CCCN(c2nccc(Br)n2)CC1 1349,c1(CN(CC(CO)NC(C(C)NSC(F)(F)F)=O)C(c2cnc[nH]2)=O)ccccc1 1350,C1(O)(CN(C(=O)CSC(C)(C)C)C)CCCN(C(=O)CC(O)C(C)C)C1 1351,c1(C(N2C(CNC(COCCCC(C)C)=O)C=CC2)=O)cc2nnn(C)c2s1 1352,c1(N(CCNC(C(c2ccccc2F)C)=O)C(c2ccsc2)=O)cncc(F)c1 1353,C1(C(=O)OC)C2C=CC(CC2)C1C(N1CCC(NC(C2CC2c2cnc[nH]2)=O)C1)=O 1354,C1(N(C(CCC(=C)C)=O)C)CN(C(c2ncccc2O)=O)CC12CC2 1355,C1(C(=O)OC)CCC(O)CN(C(=O)NC(c2cnn(Cc3ccccc3)c2)C)C1 1356,c1(CC(=O)Nc2sccc2NCC(=O)NCC(=O)OC)cccc(N(C)C)c1 1357,C1(C(=O)NC(COC)(C)COC)CN(C(=O)CC2(O)CCCCC2)CCC1(C)C 1358,N1(C(C(CC)(F)F)=O)CC2C3CCC(C2C1)N(C(=O)C(c1cscn1)C1CC1)C3 1359,CCC(C(=O)NCCCN(C(=O)C(=O)NC1CCCC1)CC)C(C)O 1360,C1(C(C2CCCN(C(=O)CC3CCC(C)(C)O3)C2)SCC)CCC(C(=O)NC)CC1 1361,N1(CC(N2CC(CN(C)C(C3COCCO3)=O)C2)=O)CCCCC1=O 1362,c1(NC(C(CC2CCCC2)NC(C2CC(O)C(F)C2)=O)=O)cc(OC)cc(F)c1 1363,CO[Si](CCC(C)(C)C)C(=O)N1CCSCC1C 1364,C12(NC(CC(=O)N(C)C)=O)CCC(CNC(c3cn(C)cn3)=O)(C1)OC2 1365,N1(C(c2cc(C)cc(O)n2)=O)CCC(C2CC2)C1CNC(=O)C1=CCCOC1 1366,N1(C(C2(CNC(C(COC)C)=O)CC2)=O)CC(C)(C)C1C(=O)N(C)C 1367,N1(C(CSCC)=O)CCC(F)C(NC(c2ccc(Oc3ccccc3)nc2)=O)C1 1368,N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC(CCNC(C2CCCC(=O)N2)=O)CC1 1369,c1(C(=O)NC2CC3(C2)CN(C(C2CCS(=O)(=O)N2)=O)C3)cc2cccnn2n1 1370,CCC#CCN=c1nc(N2CCC(c3ccccn3)CC2)c2c([nH]1)CCC2 1371,c1(C(=O)NCCC(C)NC(=O)COCCCF)coc2c1C(=O)NCC(C)(C)C2 1372,c1(C(CNC(c2nc(C3CC3)cs2)=O)NC(C(C)C)=O)ccccc1[N+](=O)[O-] 1373,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCN(C(C)C)CC1)CC(C)C 1374,CN1CC=C(CC(=O)NC2CCN(C(C3CC3C(=O)NCCO)=O)C23CCC3)CC1 1375,Cc1ccc2cc(C(=O)N(C3CN(C(=O)CC4CCOC4)CCC3O)C)cn2c1 1376,C1(CC(=O)NCCCC(C)NC(=O)CCc2cnn[nH]2)COC2(CCC2)CO1 1377,c1(C(N(CC(CO)(CO)NC(C(COC)OC)=O)C)=O)c[nH]c2c(F)cccc12 1378,C(C(O)CCNC(C1CN(C2CCOC2)C1)=O)NC(c1cccs1)=O 1379,C(=O)(C(CNC(c1ccc(C)nc1)=O)C(C)(C)C)NCCC(COC)O 1380,c1(CC(=O)N(C(CNC(C2(N(C)C)CCC2)=O)C2CC2)C)cnoc1 1381,C(=O)(N=c1c(Br)c[nH]cc1Br)C1C2(CCN(c3cc(OC)nc(C)n3)C2)C1 1382,N1(C(C2CCC(NC(C(NOC)=O)=O)CC2)=O)CCCC(C2(C)CC2)C1 1383,N1(C(c2ccc(C(C)(C)C)o2)C(=O)OCC)CCCC(C(=O)NCC)C1.CCCC 1384,C(=O)(N=c1ccn(CC)[nH]1)OCc1c(SC)cc(Br)cc1 1385,c1(OC)ccccc1CCn1cc(CNC(c2cc(O)cs2)=O)nn1 1386,C(C1=NOC2CCCCC12)C(=O)NCCc1cn(C2CCCC2)nn1 1387,Cc1ccc(N)cc1C(N1CCCC(OC(=O)C(=O)N(C)C)C1)=O 1388,C1(NC(C(C2CCCN(C(=O)CC3CCCCC3)C2)C)=O)CCC([N+](=O)[O-])CC1 1389,C1(C(=O)NCc2n(C(C)C)ncn2)CCN(C(=O)Cc2cccc(F)c2)C1CO 1390,c1(C(=O)NC(CN(C(=O)CCOc2ccccc2F)CC)C)cccc(F)c1N 1391,N1(C(CC2CCC(C)CC2)=O)CCOC2(CCN(Cc3nc(O)n[nH]3)C2)C1 1392,N1(C(C(C)=C(CC)C)=O)CCC(C2CC2)C1CNC(c1ccc2n[nH]cc2c1)=O 1393,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1394,C(=O)(C(C)(c1ccccc1)OC)N(CC(C)NC(C1SCCCS1)=O)CC 1395,C12(C(=O)NCCOCCCCOCC)COCC1CN(CC1CCCOCC1)C2 1396,C(CC(C)(C)C)(C(=O)NC(C)CC1(O)CCC1)NC(C(CCC)C)=O 1397,c1(CC)ccc(C(N2CC3CC3(CNC(=O)C3=C(Cl)CC3)C2)=O)cc1Br 1398,c1(C(=O)NC2(CC(=O)NC3CC(CC)(CC)C3)CC2)cccc(OC)c1O 1399,N1(C(=O)NC2C(CS(C)(=O)=O)C2)CCCC(CSc2ccc(Cl)cc2)C1 1400,c1(C(=O)NCC2C(NC(c3cnn(C(C)C)c3C3CC3)=O)C2)c(F)cccc1F 1401,C(c1cc(F)c(F)c(F)c1)=CC(N1CCC(N(C(C(C)OC)=O)C)C1)=O 1402,N1(C(CCC(C)C)=O)CCCCC(C(=O)NC2CCS(=O)(=O)C(C)C2)CC1 1403,C1(NC(c2c(C)cn(C)n2)=O)CC2(C1)CC(NC(c1csc(C)c1N)=O)C2 1404,N1(C(C2(O)CC2)=O)CCC(C(N2CCOC(c3ccco3)C2)=O)C2OCCC12 1405,c1(CC(CN2CCN(C(CC(C)NC3CC3)=O)CC2)=O)ccc(C#N)cc1F 1406,C(=O)(C1CCCc2n[nH]cc21)N(CC(C)NC(c1ccc(CC)cc1N)=O)C 1407,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)(C)O)ccc2ncncc2c1 1408,CON=C(C(=O)NCC1(C)CCN(C(=O)CCC(C)N(C)C)CC1)c1ccco1 1409,n1(CC(N2CC(CNC(C3(C)CC3)=O)C2)=O)nc2n(c1=O)CCCC2 1410,C1(CC=C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1411,c1(C(=O)NC2CC(NC(C(C)(C)c3cnsc3)=O)C2)ccn2c1CCC2 1412,Cc1nc(C(=O)NCC(O)CNC(c2ccc(Br)s2)=O)cn1C(F)F 1413,c1(OCC)ccc(Br)cc1CC(=O)NC1COCCC1O 1414,C1(CNC(C2C(C(C)NC(CN(C)CC)=O)C2)=O)CC(C)CO1 1415,CC(C)(C)CC(=O)NC1CC2C(NC(=O)CCOC3CCCOC3)C2C1 1416,Cc1ccc(CC(=O)NC2(CO)CN(C(=O)CN(C)CC3C(C)CC3C)C2)cc1 1417,c1(C(=O)NC(C(N2CC(OC(C)=O)C2)=O)c2ccoc2)coc(CSC)c1 1418,c1(C(=O)NC(CCOC)CNC(c2ccccc2F)=O)nsc2c(Cl)cccc12 1419,n1(CC=C)nnnc1C(C1CC=CCC1)NCCC(=O)NC 1420,CC1CCN(C(C2(c3cccc(Cl)c3F)CC2)=O)CC1NC(=O)CC1(C)CCC1 1421,C(C)(CCC(=O)NCC(C1CCN(C(=O)C(C)(C)c2ccsc2)CC1)C)OC 1422,C1(C(=O)Nc2cn(CC#C)nc2)CC2C=CC1N(C(=O)Cc1cnn(CC)c1)C2 1423,c1(CNC(C2(O)CCN(C(C3CC3c3ccoc3)=O)C2)=O)cccc(C(=O)O)c1 1424,C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(C2(CC#C)CCCCO2)=O)CC1 1425,C=CC(CC)C(=O)NCCOC1CCN(C(C2C=CCC2)=O)CC1 1426,C1(C(N2CCC(C(C)NC(C3(CN(C)C)CC3)=O)C2)=O)CCCCC(C)(C)C1 1427,CC1CCC(C(N2CC(CC(F)C(=O)N3CCC3(C)C)C2)=O)C1 1428,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1429,CCC(CC)C(C(=O)NC(C)(C)C(=O)NC(CO)CCCO)OC 1430,C=CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1CNC(C1(C(C)C)COC1)=O 1431,CCC(c1cccc(Cl)c1)=CC(=O)NCC(C1CC1)NC(=O)Cc1ccccc1O 1432,CC1CCCC1(C)NC(C1(CNC(c2cnn(C)n2)=O)CCCCC1)=O 1433,CC1CCCC(O)(C(=O)NC2CCN(C(=O)COc3ccc(F)cn3)C2)CC1 1434,c1(CCCC(=O)NCC2CC(NC(C3CCC(C)O3)=O)C2)ccc(Cl)cn1 1435,c1(N(CC(=O)Nc2nc3ccccc3o2)C)ncc(Br)c2cccnc12 1436,N1(C(C23CCC(C)(CC2)OC3)=O)CCCC2CN(C(C3CC3C3CC3)=O)CCC12 1437,C(C)(C(c1nnnn1C)Nc1cnn(-c2ccccn2)c1)(C1CC1)OC 1438,c1(NC(CC2N(C(c3cc(CC)oc3C)=O)CCC2)=O)c(Cl)ccnc1Br 1439,c1(C(N2C(C(N3C(COC)C(O)CC3)=O)CC2)=O)ccc(C)c(C#N)c1 1440,C1(C#CC(=O)N2CCC(NC(=O)COc3cccc(C)c3F)C(O)C2)(CC)CC1 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1511,C1(CC(C)C)CC(N=c2[nH]c(N3CCOC(c4ccco4)C3)nc(=N)[nH]2)CCO1 1512,C(=O)(C(C(C)NC(C1CCN1CC)=O)C(C)C)NCCC(=O)NCC#C 1513,N1(C(CC2CC(C)(C)C2)=O)CCN(C(C2CCO2)=O)CC1c1cccc(Cl)c1 1514,CN1C(=O)NCC1C(=O)NCCN(C1CCCC1)C(c1ccc(F)cc1)=O 1515,C1(C)(Cn2cc(CC=C)nn2)CCCN1C(=O)C(C(C)C)N(C)C 1516,C(C)(C)(CCN=c1cc(Cl)nc(C)[nH]1)NC(CC(CC)c1ccccc1)=O 1517,C(=O)(C#CC1CCOCC1)NC1CCC(N(C(Cc2n[nH]c(=NC)s2)=O)C)CC1 1518,N1(C(=O)C(O)Cn2cncn2)CCc2ccccc2C1C(F)(F)F 1519,C1(CN(C)C(C2CC23CC(NC(C24CCC(C2)C4)=O)C3)=O)CCCCC1(C)C 1520,C#CCC(C)(CC)C(=O)N1CCC1CNC(C1(O)CCSCC1)=O 1521,Cc1ccc2c(NC3CCC(c4ccccc4)N3)nc(N(CCCO)C)nc2c1 1522,C(C)(C(CC(=O)N(C)CCN1CCCCC1)NC(=O)Cc1ccc(F)nc1)OC 1523,C1(NC(c2n(CCC)nc(C)c2)=O)CCN(C(C23CC(C)C2C3)=O)C(C)C1 1524,CC(C(C(=O)OC(C)(C)C)N(C)C(=O)Cc1cnn(C2CCOCC2)c1)C(C)(C)C 1525,C1(CNC(c2cn(C(C)C)cc2C(F)(F)F)=O)CCCCN(C(=O)C=CC(N)=O)C1 1526,c1(CCC(=O)NC(CCNC(C2C(C(=O)OC)CCC2)=O)C)ccccc1OC 1527,CCCCCC(=O)NCC(C)N(C(=O)Cc1cccnc1)C 1528,Cc1cc(F)ccc1CN(C(c1cc2occc2[nH]1)C(=O)NCC1CC1)C 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1565,N1(C(C(=O)NCCC)CCC2CCCCC2)CCCC(C2CCN(C)C2)C1 1566,CN=c1[nH]c(C(N2CCN(CC(C)NC(C3CC34CC(O)C4)=O)CC2)=O)cs1 1567,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)CCN2CCCC2)CCC1(C)C 1568,c1(C(C)C)nccc(C(N2CC(n3cc(CCNS(N)(=O)=O)nn3)C(O)C2)=O)n1 1569,N1(C(c2c(CC)oc(C)c2)=O)CC(CNC(C2(CCF)CCC2)=O)CC12CCC2 1570,c1(CNC(C(CC)(O)c2ccccc2)=O)cccc(S(=O)(=O)Nc2ccc(F)cc2)c1 1571,Cn1ccn2ncc(C(c3ncc(C(F)F)o3)NCc3ccc(F)cc3)c12 1572,c1(N2CCN(C(c3ccc(C)[nH]3)=O)CC2C)cc2nncn2cn1 1573,C1(CC)CN(C(=O)C(C)(O)COC)CCC1NC(=O)CCCOC 1574,C(=O)(C(C)CCCC(C)C)N(CCC(=O)OC)CCC(c1cnn(C2CC2)c1)=O 1575,c1(N(CCSC)CC)nc(N2CCc3c(N)cccc3C2)c2c(n1)c(C)nn2C 1576,N1(C(C2N(C(c3ccn(C)c3)=O)CCC(CC)C2)=O)CCCC(C2CCC2)C1 1577,CCC(CC(=O)N1CC(CC(F)C(=O)N2CC(CN3CCCC3)C2)C1)C(C)C 1578,C(CC(C(=O)NCC1CC2CC2C1)NC(c1cnc(C2CC2)o1)=O)OC 1579,C1(CC)CCN(C(C2COCCO2)=O)C1CNC(c1cccnn1)=O 1580,Cc1ccccc1CCC(C)NC(C1(CO)CCC1)=O.C(C)(C)(C)O.C1(=O)NC1.O 1581,N1(CC(C)(C)NS(=O)(=O)c2cnc(=N)[nH]c2)CCCN(N2CCS(=O)(=O)C2)CC1 1582,C=C=C(C)CC(=O)NCCOCCC(=O)NCc1cccnc1CCCC 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1601,C1(O)(CNC(c2cn(CC)nn2)=O)CCCN(C(c2cnc(NC)cn2)=O)C1 1602,c1(C(N2CC(F)(C(=O)NCc3ncon3)C2)=O)ccc(Cl)nc1 1603,C1(O)CCC2(CCCC2)O1.CC1CCCC1(OC)CNC(=O)NCCOC(C)(C)C 1604,c1(C(N(CCCNC(c2cccs2)=O)CCC)=O)ccc(F)c(O)c1 1605,c1(C(=O)NCCCC(C)NC(CC(CC)(C)C)=O)cc2ncccc2o1 1606,CCC(C)CCCCC(=O)N(C(C)=O)CC1CCCN1c1ncnc2[nH]cnc12 1607,C(=O)(CCS(N)(=O)=O)N1CC(C(C)NC(=O)CCC2CC2(C)C)C1 1608,C1(NC(CCC(CC)NC(c2c(C)coc2C)=O)=O)CC(C2CCCC2)C1 1609,C12(C(=O)NCC(CCCC)NC(C3CCC3(C)C)=O)CC3CC(CC(C3)C1)C2 1610,Nc1ccc(C(N2CC(NC(C3CC3C3CCC3)=O)C(F)C2)=O)cc1[N+](=O)[O-] 1611,c1(C(N2C(C3CCN(C(CC=C)=O)C3)CCC2)=O)ccc(=O)n(-c2ccccc2)c1 1612,c1(C(=O)NC(COC)CC(=O)NCC=CCSC)cc(C)cc(O)n1 1613,c1(CN(CCSC)C)cn(C2CCc3cccnc32)nn1 1614,C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(C(N2C(CC)CCC2)=O)=O)C2CCC1C2 1615,C1(CC)CN(C(=O)CCc2ccc[nH]2)CCC1CNC(c1cnc(C)cc1Cl)=O 1616,C(=O)(CCC(F)(F)F)NC(C(C)C)CNC(c1cccnc1N(C)C)=O 1617,C#CC1(NC(=O)CN(C(=O)C(CC)n2ccnc2)CCC)CCCCC1 1618,c1(C(c2n(CCC)nnn2)NC2CC2F)cc(F)cc(C#N)c1 1619,c1(C(N(Cc2cn(C(C)(C)C)nn2)O)=O)ccc2c(c1)CC(C)(C)O2 1620,C1(C(=O)NCC(C)NC(=O)C(C)C2=CCCC2)CCc2[nH]nc(C(F)(F)F)c2C1 1621,c1(C(N2CC(CC(C)NC(C(C3CCC3)OCC)=O)C2)=O)cc(C)c(F)cc1N 1622,CC1c2ccccc2CN1C(=O)NCCNS(C)(=O)=O.N12CCCCC(C1)C2=O 1623,Cc1nc2[nH]cc(C(N3CC4CC4(NC(c4cnn5c4OCC5)=O)C3)=O)c2cc1F 1624,Cc1c[nH]cc([N+](=O)[O-])c1=NCC1CC(C)N(C(=O)C(F)=CC2CC2)C1 1625,c1(C(=O)NC23CCN(C(c4n(C)ccc4)=O)CC2C3)cc2ccsc2c(O)n1 1626,c1(-c2nc(OC)c(C(N3CCN4CCOCC4C3)=O)cc2)cc2nc(C)ccc2o1 1627,C1(CNC(Cn2c(C)cnc2)=O)CCCN(C(=O)Cc2cscn2)CC1 1628,N1(C(c2nc(C)oc2)=O)CCOC2CCN(C(=O)C(C)CSC(F)(F)F)CC12 1629,C1(C(=O)NCCOCCC(=O)N(C2CCCC2)C(C)C)CCCCC1C.C(C)S 1630,c1(C(CNC(CN(C)C2CC2)=O)CNC(=O)Cn2cnc(Br)c2)ccccc1 1631,Cc1cc(F)ccc1C1(C(=O)NCC(CNC(C2(N(C)C)CC=CC2)=O)CO)CC1 1632,C1(NC(C(C2CN(C(=O)Cc3ccncc3Cl)C2)OC)=O)CC=CCC1C 1633,Cc1cc(CNC(c2ccc(C(F)(F)F)cc2)C)cc(C)n1 1634,c1(C(N(CC(C)(C)NC(=O)CNS(C)(=O)=O)C)=O)ccncc1F 1635,c1(CCC(=O)N(CCCNC(C23CC(F)(C2)C3)=O)CC)cnn(CC(F)(F)F)c1 1636,C1(F)(C(=O)Nc2ccc(N(C)C)nc2)CCCN(C(C2CCC3(CCC3)C2)=O)C1 1637,CC1CCCn2ncc(C(=O)NC3(C(F)F)CCCC3)c21 1638,C1(OC)CN(C(=O)C(CCSC)NC(C)=O)CC1NC(c1c[nH]c(=O)cn1)=O 1639,C#CCCCCC(=O)NC(CO)CCCNC(C1(C#N)CC1(C)C)=O 1640,c1(C(N(C)CCNC(=O)CC(F)(F)c2ccccc2)=O)cccc2oncc12 1641,c1(OCC(=O)NC(CNC(C(C)OCCOC)=O)CC)ccc(C)nc1 1642,c1(OC)cc(CC(N2CCN(C(=O)C(=O)NCCN(C)C)CC2C)=O)ccc1Br 1643,C1(NC(c2cc(C)n(C)n2)=O)CC(F)CN(Cc2cc(F)cnc2Cl)C1 1644,C12(C(=O)NCC3C(CNC(c4ncc(C)cc4F)=O)C3)C3CCC(CC13)C2(F)F 1645,c1(C(N(C2CCCN(C(C(COC)C)=O)C2)CC2CC2)=O)cccc(C)c1Cl 1646,C12(CNC(COCC)=O)CC(CO1)N(C(=O)CCCSc1nccn1C)C2 1647,c1(N(CCOC)CCNC2CC(C)(C)C2C(F)(F)F)nc(CO)c(C)cc1C#N 1648,O(N1CCC(CC(N2CC3CCC3(NC(=O)CC34CC(C3)C4)C2)=O)CC1)CC 1649,C1(N(C(c2cnc(C)[nH]2)=O)C)CCCN(C(C2CCCN(CC(C)C)C2)=O)C1 1650,Cn1cnc2ccc(C(=O)NCC3CCC(F)(CNC(C4CC4Cl)=O)CC3)nc12 1651,N1(C(c2c(CC)n[nH]c2)=O)CC2CC2C1C(N1CCC(n2cncn2)C1)=O 1652,C(=O)(C(=O)N=S(C)(C)=O)Nc1ccc(OC2CN(C(C3(C)CCCS3)=O)C2)c(Cl)c1 1653,c1(OC)cc(Cl)ccc1C(N1CC(CNC(=O)CC2(C)CCC2)CC(C)C1)=O 1654,C1(C(N2CCC(=CCC)C2)=O)CCN(C(c2cocc2C)=O)C12CC2 1655,c1(C(N(CCCCNC(CS(CC)(=O)=O)=O)C)=O)cc(S(=O)(=O)NC)c[nH]1 1656,C1(O)(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2CC2F)=O)CC1 1657,C1(CC(=O)N(CC(O)CNC(c2conc2C(F)(F)F)=O)C)CCN(C)C1=O 1658,c1(SC)cc(=NC(=O)C2CC2NC(C2CNC(=O)N2)=O)[nH]n1C 1659,C(CCC(=O)NC(C)(C)C=CC(=O)N(C)C)N(C(=O)Cc1ccsc1C)C 1660,C1(C(=O)NCCC(=O)N(CCCNCC2CCC2)C)(C2CC2)CCCO1 1661,N1(C(c2c(OC)ccs2)=O)CCOC(C)(CNC(=O)C(C)n2cnnn2)C1 1662,N1(CCNC(C(C)(C)N(C)C)=O)CCN(C2CCCC2O)CC1 1663,CC1(C)C2CN(C(C3COC4(C3)CN(C(c3cnsn3)=O)C4)=O)CC12 1664,C(=O)(CC(C)C(=O)OCCCNC(c1cc(N2CCCC2)ccn1)=O)NC 1665,C(=O)(CC(CN(C)C)C(F)(F)F)NCCCN(C(CC1(CC=C)CCCC1)=O)C 1666,C1(C(=O)NC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)CCc2nnnn2CC1 1667,C#CCCCCCC(=O)NCC1CCN(C(=O)C(C)CSc2ccccc2)C1 1668,c1(C(=O)NCc2ccc(C(N3CCC(COCC)C3)=O)s2)n[nH]c(C)c1Cl 1669,c1(C(=O)NC2C(CNC(=O)CN3C(=O)CNC3=O)C2)cc(F)cc2nn[nH]c12 1670,c1(OC)cncc(C(=O)NC2(Cc3nnc(-c4ccc(OC)cc4)s3)CCC2)c1 1671,N1(C(C(CCC2CC2)NC(C2N(C=O)CC2)=O)=O)CC2(CCC(O)CC2)C1 1672,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(c1c(N)sc(C)c1C)=O)(C)O 1673,c1(CN2CCC(C(=O)Nc3c(OC)cc(O)cc3)C2)c(F)cc(Cl)cc1F 1674,c1(C(=O)NCC2(C(C)NC(CC=C(C)C)=O)CC2)cc(N)c(C)c([N+](=O)[O-])c1 1675,N1(C(C(CCC=C)NC(c2ccc(N)c(F)n2)=O)=O)CC2CCC(O)C2C1 1676,C(CNC(=O)Cn1cc(C2CC2)nn1)(CC(F)(F)F)NC(c1nc(CC)sc1)=O 1677,N1(C(c2cc(CC)no2)=O)CCC(O)(CCNC(=O)C(C)CSC)C1 1678,N1(C(c2[nH]cc(C(C(C)C)=O)c2)=O)CCCN(C(=O)CN2CCCC2=O)CC1 1679,C1(C(=O)NC2CC(C#N)(OC)C2)(OC)CCN(C(c2cnc(C)nc2O)=O)CC1 1680,C1(NC(c2cnc(C(N)=O)s2)=O)COCCN(C(c2n[nH]c3c2CCC3)=O)C1 1681,CP(C)(=O)C(O)C(=O)N1CCC(O)(CNC(c2ccc(=O)oc2)=O)CC1 1682,c1(C(N2CC(CNC(C(CC(C)C)O)=O)C2)=O)cc(N)c(=O)n(C)c1 1683,c12ccc(cn1)S(=O)(=O)N2.CC1(C)CC(NCCC(F)(F)F)CC(O)C1 1684,c1(CC(=O)NCC(CC)NC(c2cn(CC(F)F)cn2)=O)ccc(F)cc1OC 1685,C1(CNC(C2N(C(C(C(C)C)SCC)=O)CC2)=O)CCCCCCC1 1686,S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1CC(NC(c2c(C)cc(C)nc2)=O)C1 1687,CC1(C(=O)NC2CCC(CCC(=O)NCCc3noc(=O)n3C)C2)CC=CCC1 1688,N1(C(C2C(C)CCN2C(=O)CC2CCC=CCC2)=O)CCNC(=O)CC1 1689,N1(c2nc(COC)nc(Cl)c2)CCS(=O)(=O)C(CCNC(=O)CCS(C)(=O)=O)C1 1690,N1(C(C(C)NC=O)=O)CC2(CC2)CC1C(=O)N1CC=CCO1 1691,N1(C(c2cc(C)ns2)=O)CCC(NC(=O)Cc2ccsn2)C1C 1692,Cc1nc(O)ccc1C(N1CSCC1C(=O)NCC(C)(C)C#N)=O 1693,c1(C(=O)NCCNC(c2ccccc2C(N2CCOCC2)=O)=O)ccc(Br)cc1 1694,c1(C(=O)Nc2c(-c3cc(C)oc3)nccc2)ccc2[nH]cc(C#N)c2c1 1695,c1(C(=O)NC2(C)CCCC2NC(=O)Cc2ccsc2)ccnc(O)c1F 1696,CN1CC=C(CC(=O)NCC2COCCN2C(=O)Cc2c(O)ncnc2O)CC1 1697,C1(C(N2CC(C3N(C(C=C(C)Cl)=O)CCC3)(O)C2)=O)CCC2CC2C1 1698,c1(C(=O)NC2(CCNC(=O)COC3CCOC3)CCC2)ccn2nncc2c1 1699,C1(CC(N)=O)(NC(C(NOC)=O)=O)CCCN(C(c2ccccc2O)=O)C1 1700,CC1(C)CCC(O)(C(N2CC(CNC(c3csc(C(F)F)n3)=O)C(O)C2)=O)CC1 1701,CC1CN(C)CC1NC(c1cccnc1CNC(C1CCC1C#N)=O)=O 1702,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(=O)Cc2cncnc2O)CC1 1703,CC(C)(C)C(O)C(=O)NC1CCCN(C(c2cc(F)ccc2O)=O)CC1 1704,c1(C(c2n(CCOC)nnn2)NCC2COC(=O)N2)ncc(C)cc1C 1705,N1(C(c2cncc(Cl)c2)=O)CC2CCCN(C(=O)C(=Cc3cccnc3)F)C2C1 1706,c1(NC(c2n(C)ncn2)=O)sc2c(c1C(N1CCOCC(O)C1)=O)CCCC2 1707,c1(C(=O)NC2(CO)CCN(C(C3CC(C)(O)C3)=O)C2)cncc2ccsc12 1708,n1(C(C(=O)NCC2(C)CCN(C(COC)=O)C2)C)cc2ccccc2n1 1709,S(=O)(=O)(c1ccc2oc(C(=O)OC)cc2c1)NC1CC(N(CCC)C)C1 1710,Cc1cc(C(N2CCC2C(N2CCC(O)C(C)C2)=O)=O)ccc1F 1711,N1(C(c2ccc(C=C)cc2)=O)CCN(C(=O)C(C)(C)C)CC2CCCCC12 1712,N1(C(c2c(OC)nn(C)c2)=O)CCCC(N=c2[nH]c3cc(C)nn3o2)CC1 1713,c1(C(=O)NCC(CN(C(C(c2cccc(C)c2)=O)=O)C)(C)C)cc2n(n1)CCC2 1714,c1(CC)cc(C(=O)N(C(C)CNC(=O)C=CCOCCSC)C)sc1C 1715,CCC(O)C(C)C(=O)N(CC(C)CNC(C1(OC)CCSC1)=O)C 1716,C(CN=c1ccc(S(=O)(=O)NC(C)Cc2cccc(Cl)c2)c[nH]1)NS(CC)(=O)=O 1717,CC(C(=O)NC1C=CCN(C(C2CN(C3CCOC3)C2)=O)C1)C(F)(F)F 1718,n1(CCNC(=O)NC(CN(C)C)CCO)cnc([N+](=O)[O-])c1 1719,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1720,c1(-n2cc(CC(C)N(C)C)nn2)nc(-c2ccncc2)nc2sccc12 1721,CCCC(CNC(=O)CCNC(=O)CO)C(=O)NCC1COC(=O)N1 1722,N1(C(c2cnc(CNC(CC(CC)(C)C)=O)nc2)=O)CCC2C(CCN2C)C1 1723,c1(C(N(CC(C)NC(=O)CNc2ccccn2)CC)=O)cccc(F)c1F 1724,N1(CC(=O)NC2CC(F)(CNC(CN(C)C(N)=O)=O)C2)CCCCS1(=O)=O 1725,C1(c2n(C)nnn2)(Nc2ccc3c(c2)CCO3)CC2(CCCCC2)C1 1726,C1(N(C)C)CC(N=c2[nH]c(=NC3CCC(C4CC4)CC3)[nH]c3c2COC3)C1 1727,C(CC(=O)OCc1ccc(SC)cc1O)(C1=CCCC1)OCC 1728,C1(CCNC(C(CC#C)O)=O)CCN(C(c2cc(C(F)F)no2)=O)CC1(F)F 1729,c1(C(=O)NCC(C2CCC2)NC(C(C)SC)=O)cc(C)ccc1Cl 1730,CC(C)CC(CC(=O)NC(=O)C=C(Cl)Cl)NC(C1CCCN1C(=O)C1CC1)=O 1731,c1(C(C(=O)NCCC)N(CCC#C)C)cc(C(F)(F)F)cc(C)c1 1732,CN1CC(C(=O)NCCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)CCC1=O 1733,c1(CC(=O)N(C2CCN(C(CCC(C)OC)=O)C2)CCO)ccc(Cl)cc1O 1734,C1(NC(CC(=O)OC)=O)CCN(CC)CC1n1cc(C2CCC(C)=C(C)C2)nn1 1735,c1(C(=O)NCC(C(C)C)NC(C(F)(F)C2(OC)CC2)=O)ccc2c(c1)COCCN2 1736,C1(CC(=O)NCC2CCN(C(c3c(N)nc(Cl)cc3)=O)C2)Cc2ccccc2O1 1737,n1(C2CCN(C(c3ccc(C)o3)C(=O)NC3CCOC3)C2)ccc2ccccc12 1738,c1(C(=O)NCC2N(C)CCN(C(c3coc(Br)c3)=O)C2)cccn2cncc12 1739,c1(C(N2C(CNC(C(CC(=C)C)C)=O)CCC2)=O)ccc2nsnc2c1 1740,C1(C)(NC(c2c(C)csc2)=O)CCN(C(=O)CCSC2CCCC2)C1 1741,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)o2)=O)C1 1742,c1(C(N(C2CN(C(C=CCOC)=O)C2)C)=O)cc(=O)cc[nH]1 1743,C(=O)(C1=CC2(CCOC2)C1)N1CCC(N(C(C2SC3C=CC2CC3)=O)CC)C1 1744,c1(C(N(CCN(c2c(OCC)ccnc2)C)CCOC)=O)ccc2occ(C)c2c1 1745,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(CCC)=O)CC1 1746,c1(OC)ncnc(C(=O)NCC2(C)CC(NC(=O)Cn3cncn3)C2)c1F 1747,c1(C(N(CC(C(=O)NC(CC#C)C(=O)NC)(C)C)C)=O)cccc(C#N)c1C 1748,c1(CC(=O)NCC(CNC(=O)C=C2CCC2)F)ccccc1 1749,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1750,c1(OC)cc(C)cnc1NC(=O)CC1CC(O)CN1C(=O)C(C)n1ccnc1 1751,C1(O)(CC)CCCN(C(=O)C=CCN(C(=O)CCn2nc(C)nc2C)C)C1 1752,Cc1nc2cc(C(=O)N(CC(C)NC(=O)CCC3(C)CC3)C)cc(O)c2o1 1753,CC(C(=O)N1CCC1CNC(=O)Cc1cscn1)n1ccnc1 1754,C1(OC)CCC12CC(C(=O)NCC1CCN(C(=O)CN3CCCCC3)C13CC3)C2 1755,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1c(CCC)nns1)=O 1756,C#CCCCC(C)C(=O)NCC(CO)NC(c1cc(C(N)=O)[nH]n1)=O 1757,C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(=O)CC1(O)CCOC1)OC 1758,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1759,N1(C(c2cccc(C)n2)=O)CCCCC(NC(C2(C3CCCO3)CCC2)=O)C1 1760,Cc1[nH]c(C#N)cc1C(=O)NCC(C)(C)NC(C1CC(C)(C)CN1C)=O 1761,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1762,Cn1ccc2c(C(=O)NCC3CN(C(c4cnccc4Cl)=O)CCO3)ccnc12 1763,c1(CC(N2CC(CNC(C(C)OCC)=O)(COC)C2)=O)ccccc1Br 1764,c1(C(=O)NC(C(C)C)(C)CNC(=O)CSCC(N)=O)cnc(Cl)c(C2CC2)c1 1765,S(=O)(=O)(c1cccc(C(=O)N(C)Cc2nc(=O)o[nH]2)c1)N(CC(=O)NC(C)C)C 1766,Cc1cnn(CCCNC(=O)CCN(C)CCO)c1.C1(=O)CC2(CC2)N1 1767,C(CCC(=O)NC(C)CNC(=O)CCc1nc(C)no1)=C(C)C 1768,C12(NC(C3CC(C)OCC3)=O)CC(CNC(c3cncn3C)=O)(C1)OC2C 1769,C1(C(=O)Nc2c(CC)ncs2)CC12CCN(C(c1ccc(C3CC3)cc1)=O)C2 1770,CS(=O)CCC(=O)N1CCCC(N(c2nccc(C(F)(F)F)n2)CCO)C1 1771,C1(CC(=O)NC2CCOC2=O)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1772,N1(C(C(N2CCCC3C(C)(C)C2C3)=O)=O)CC2CS(=O)(=O)CC2C1 1773,N1(C(C(C)N)=O)CCCC(NCCO)C1.CCCCCCC(=O)C(c1ccc(Cl)s1)=O 1774,c1(C(N(C2CCN(C(c3onc(C)c3C)=O)C2)CC)=O)c(Cl)cnn1C 1775,Cc1noc(C)c1C=CC(=O)NC1CC2CCC1(NC(C1(O)CCCC1)=O)C2 1776,c1(CC(=O)NC2C(CO)CCN(C(C=CC(CC)C)=O)C2)cn2ccccc2n1 1777,c1(OCC)ccc(Cl)cc1NC(=O)C(c1cccc(Br)c1)N1CCCC(NC)C1 1778,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CCC2)C1 1779,c1(OC)c(C(=O)NCCC2CSCCS2)ccc(Cl)c1Cl 1780,C1(C(=O)NCCCOCCSC)(COC)CCCN1C(=O)C(C)(F)F 1781,c1(C(C(=O)NC2(CNC(COCC(=C)C)=O)CC2)C)cccc(C(N)=O)c1 1782,C1(C(=O)NCCC(CNC(=O)CC(=O)Nc2nccs2)O)CC2C=CC1CC2 1783,c1(C(C2CC2)NC(C2CN(CC3CC3)C2)=O)ccc(I)nc1 1784,N1(C(CCC=C=C)=O)CC2CCN(C(C3CCN(C(=O)NC)CC3)=O)CC2C1 1785,N1(C(Cc2cn(CC)nc2)=O)CCN(CCOCCNC(=O)C(C)N2CCC2)CC1 1786,c1(NC(C23CC(NC(c4ccncc4Cl)=O)(C2)C3)=O)ccc2c(Cl)n[nH]c2c1 1787,C(=O)(C(=O)NNC(=O)C1CC(N)C1)NC(C)Cc1ccccc1 1788,C(=O)(C1SCCc2sccc21)NCC1N(C(c2cc(C)n(C(F)F)n2)=O)CCC1 1789,c1(C(=O)NCC2(CNC(c3c(CC)onc3C)=O)CC2)cc(OCC)nc(C)c1 1790,N1(C(c2c(OC)nsc2)=O)CCCCC1C(C)NC(c1cnoc1C)=O 1791,N1(C(COCC(C)C)=O)CC(CNC(c2csc(Cl)n2)=O)OC(C(F)(F)F)C1 1792,C(C1CCOC1)=CC(N1CC(C)(CCC(=O)NC(CCNC(C)=O)=O)C1)=O 1793,c1(C(N2CCN(C(C(C)C(F)(F)F)=O)CC2CO)=O)cnc2cccc(F)n12 1794,CC(O)C(C)(C)C(=O)N1CC(NC(c2ncc(Cl)cc2Cl)=O)C(CC2CC2)C1 1795,C=CCCC(c1nnnn1C1CCOCC1)(c1cccs1)NC(C)CCC(C)C 1796,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1797,c1(C(=O)NC2CC3(CN(Cc4cn(C)nc4)C3)C2)n[nH]c2cc(Br)ccc12 1798,N1(C(COCCCCC)=O)CCC(NC(=O)C(C)SC(F)(F)F)C(C)C1 1799,C1(NC(c2cc(Cl)sc2Cl)=O)CC2CC(NC(C3SCCS3)=O)CC2C1 1800,C1(C(=O)NC(C(=O)N(C(C)C(=O)N(C)C)C)Cc2cn[nH]c2)CC2CC(=O)C1O2 1801,c1(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)ncnc2c1nnn2CC 1802,C1(NC(COCCCC#C)=O)CC2(C1)CC2NC(=O)CCCOC1CCCCC1 1803,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1804,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1805,N#CCCCCC(=O)N1CCN(C(=O)C=CCN2CCCC2)C(CCO)C1 1806,C1(OC)CC(C(=O)NC(CNC(c2cn(C(C)C)cn2)=O)C2CC2)CC1OC 1807,Cc1cc(N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2C)n2nc(C)nc2n1 1808,C(=O)(CN=c1[nH]c(C)cs1)NCCN(C(CC1(CC)CCOCC1)=O)C 1809,C(=O)(C1=CC2CCC=CCCC12)NCC1CC(O)(CNC(C(=O)N(C)C)=O)C1 1810,C1(CN(C(=O)COCCOc2ccccc2)C)COCCN1C(=O)CS(=O)CC 1811,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1812,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1813,C12(OC)CCC(C(=O)N(CC(C)NC(c3cc(F)ccc3C(N)=O)=O)C)(CC1)C2 1814,c12c(cccc1F)C(=O)NC2.c1(OC)cc(C(=O)NC2(CO)CCC2)[nH]n1 1815,CC1CCCCN1C(=O)CCN(c1nc(-c2ccc(F)cc2)cs1)C(=O)C1CC1 1816,c1(C(=O)NCC2CC2CNC(C2CC(O)(c3ccccc3)C2)=O)ccc(O)cn1 1817,C(C(C)CC(=O)NC(C(=O)N(C)CCOC(C)(C)C(F)(F)F)C1CC1)SC 1818,C1(NC(c2c(CC(C)C)nc(C)s2)=O)CC2CC(NC(=O)Cc3cn[nH]c3)CC12 1819,C=CC(CCC)CC(=O)NC(COC)C(=O)N(CCCCC)C(C)C 1820,C(CC(O)CNC(=O)C(Cn1ccnn1)NC(=O)CC1(O)CCOC1)OC 1821,Cc1ccc(CC(=O)NC2CCC(N(C)C(c3nocc3Cl)=O)CC2)c(F)c1 1822,CC(CC(=O)NC1CCCN(C(=O)CNC(c2cnc(O)nc2O)=O)C1)C(F)F 1823,c1(C(=O)NC2CC3CC2CC3c2ccccc2)cc2c[nH]nc2c(C(F)(F)F)n1 1824,c1(C(C)=O)cn(CC(N2CC(C)(N(C(C3CCCCS3)=O)C3CC3)C2)=O)nn1 1825,c1(OCC(=O)NC(CNC(C2(CC)CCCC2)=O)(C)C2CCC2)ccc(F)cn1 1826,c1(C(=O)NCC2(O)CCN(C(C(C=C)(C)CC)=O)C2)cccc([N+](=O)[O-])c1O 1827,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1828,c1(CC(N2C(CNC(C(C)C3(O)CCC3)=O)CCC2)=O)cc(O)ccc1Br 1829,C1(OC)CN(C(C2(CF)CC2)=O)CCC1NC(=O)C(O)CCSCOC 1830,c1(C(=O)NC(C(=O)NC2CC(CC(C)(C)C)C2)C2(O)CCC2)ccccc1 1831,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1832,CC1CCCCCN1CC=CCS(=O)(=O)Cc1ccccc1-c1ccc(Cl)c(F)c1 1833,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1834,Cc1cc(C(N2CCC(CO)(CNC(=O)CC3CCCC3(F)F)C2)=O)ncc1N 1835,C1(NC(C(CNC(CSC)=O)NC(=O)CSC2CC2)=O)CCC2CC1CO2 1836,Cc1cc(C)c(C(=O)Nn2cncn2)cc1C.C12CN(C1)CNC2Cc1ccoc1 1837,c1(C(=O)OC)cc(SCCn2cc(-c3ccn(C)n3)nn2)cs1 1838,Cc1cc(S(=O)(=O)NC2CC(C)(C)OC2(C)C)c(C)cc1Br 1839,CC1(CNC(c2cnco2)=O)CCN(C(=O)Cc2nnc(-c3ccccc3)o2)C1 1840,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1841,C(=O)(CC(F)(F)C(F)F)N(C)CC1CC(NC(=O)CSC(C)(C)C)CCO1 1842,N1(C(C)=O)CCC(C2OCCC2NC(=O)C=C(C)C(C)C)CC1 1843,C12(C(=O)NCC3CCC(NC(c4ccc(Cl)nn4)=O)C3)C=CC(CC1)C2 1844,C(C)(CC(=O)NCC(C1CC1)NC(=O)CC#N)(C(F)(F)F)N(C)C 1845,n1(C(C2CCCCC2)C)nc(-c2cnn(C)c2)nc1-c1ccc(N)n1C 1846,c1(CC)cc(C(N2CCCC2CN2CC(CC(=O)OC)C2)=O)ccn1 1847,c1(C(N(C2C(C)CN(C(C34CC(F)(C3)C4)=O)CC2)C)=O)ccnc2cc[nH]c12 1848,Cn1cc(C(=O)NC2CC(O)CN(C(c3scnc3C3CC3)=O)C2)ccc1=O 1849,N1(C(C2(C(C)C)COC2)=O)CCCC(C2CCN(C(=O)CSS(C)(=O)=O)CC2)C1 1850,CCCCC(CNC(=O)CN1CC2C=CC1C2)NC(c1cncc(C)n1)=O 1851,c1(CC)nnc(CNC(=O)CCN(C(=O)Cc2cccnc2)C(C)C)o1 1852,CCCC(C)CC(=O)NC1CCCC(CNC(c2c(C)nc(C)n2O)=O)C1 1853,CC1CC(N(C)C)(CO)CN1C(=O)CCCC(c1ccccc1F)O 1854,c1(C(N2CC(NC(C(C)(C(C)C)OC)=O)CC2(C)C)=O)c(C)nc(O)nc1C 1855,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1856,c1(C(=O)NC23C(CN(C(C4CC(=O)N(O)C4)=O)C2)CC3)sc2sccc2c1Cl 1857,C1(N(C(c2ccc(CN(CCC)C)o2)=O)C)CCCN(C(=O)CCNC(N)=O)C1 1858,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1859,c1(C(N2CCCC(N3CCCC3)C2)=O)ccc2ncsc2c1 1860,Cc1ccc(=O)n(CC(=O)NCC2CC2NC(=O)COC2(C)CCCC2)n1 1861,C1(NC(C=C(C)Cl)=O)CCCCCN(C(c2cc(C3CCCC3)on2)=O)C1 1862,O=C(C1=CCCN(C(C2(C(F)(F)F)CC2)=O)C1)NC(CO)C1CC1 1863,C12(NC(c3ccc(COC)o3)=O)CC1CN(C(C1CCC=CCC1)=O)C2 1864,C1(C(N2CCCC(C)(NC(c3cccc(F)c3F)=O)C2)=O)Cc2cccnc2C1 1865,c1(OC)ccc(O)cc1C(N1CC=C(CNC(C2(OC)CC2)=O)CC1)=O 1866,CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CCN1C(C1CC1C(C)O)=O 1867,CN1CCN(C(c2ccc(Br)o2)=O)C(CNC(c2csc(CO)n2)=O)C1 1868,c1(C(=O)NC(C(=O)OCC)Cc2cocn2)noc2c1CCCCC2 1869,N1(C(C2CCOCC2)=O)CCCN(C(C2C(F)(F)C23CC3)=O)C(CO)C1 1870,C1(NC(c2c(C)n(C(C)C)cc2)=O)CCN(Cc2ncnn2C)CC1O 1871,N1(C(c2c(CC)nc[nH]2)=O)CCCC(C(C)NC(=O)CN2CC3CC3C2)C1 1872,c1(CC(=O)NCC2COCCN2C(C2CC2c2ccncc2)=O)ccc(Cl)cc1 1873,N1(C(C2CCN(CCC#C)CC2)=O)CCC(CO)C(NC(=O)CP(C)(C)=O)C1 1874,C(=O)(C(C)(C)C(C)C)N(CC(N1CCC(C(=O)NC(C)C)C1)=O)CCOC 1875,C(=O)(CCCCCN=[N+]=[N-])N1C(C)C(C(=O)NCC2CCC=CCC2)CC1 1876,CC1CCN(C(c2cnn(C(F)F)c2)=O)C1CNC(=O)COC1CCOCC1 1877,CCCC(CNC(c1ccsc1C)=O)C(=O)NCC(F)(F)C(C)(C)O 1878,c1(C(=O)NCC2COC(CNC(c3cc(Cl)no3)=O)C2)cccc(CO)n1 1879,CC(C)(C)C(=O)NC1CCC(CC(=O)NCCCCO)C1 1880,Cc1sc(N2CCCC2C2(C(=O)O)CC2)nc1-c1ccccc1 1881,C1(C(N2CCC(CNC(c3c(CC)occ3)=O)CC2)=O)CC1C1CCCC1 1882,CC1CCC(NC(c2cc(C#N)c[nH]2)=O)CN1C(=O)CCN1CCOCC1 1883,c1(N2CCN(C(CSc3ccc(C)cc3)=O)C3C2C3)ccnc2ccnn12 1884,c1(C(C)(C)C)ccc(CC(=O)NC2(CCCNC(C3CC=CC3)=O)CC2)cc1 1885,c1(OC)ccc(C(=O)NCCN(C(C2(C)CCC(C)C2)=O)C(C)C)c(N)c1Br 1886,C1(C(N(C2(C)CC2)C)=O)CCN(C(=O)C2CC(CSC3CC3)C2)O1 1887,CCCC(O)CC(=O)N1CCC(C(C)(C)NC(=O)CCS(C)(=O)=O)CC1 1888,CC(C)S(=O)(=O)CC(=O)NCC1(CCNC(C2CC3(C2)CC32CC2)=O)CC1 1889,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1890,N1(C(C2N(C(C=Cc3ccc(C)o3)=O)CCC2)=O)CCCC(CO)C1C 1891,N1(C(COCC(=C)C)=O)CCC(NCc2cncs2)CC1 1892,N1(C(c2cc(Cl)cc(Cl)c2O)=O)CCC2CCN(C(C3C4COCC34)=O)CC12 1893,C1(C)(C(N(CCCNC(c2c(OC)cccc2)=O)C)=O)COC(C)COC1 1894,CC1(C)CC(NCCCC2CCC2=O)c2ccccc2O1 1895,C(C)(C(=O)NCC(C)(C)CNC(=O)CC(C)C1CC1)(C(C)C)NC(C)=O 1896,C(=O)(CC(C)(O)COC(C)C)NC1CCN(C(c2c(NCC)nccc2)=O)C1C 1897,C1(CN=C(NCC(C)(C)C#N)N(C)Cc2ccco2)CCCCC1(C)C 1898,Cc1ccc(CC(=O)NC2CCC2NC(c2ccc[nH]2)=O)s1 1899,N1(C(C2CCC(C)CC2)C)CCC(C)C(NC(=O)OC(C)(C)C)C1 1900,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(=O)Cc2cccnc2F)c1O 1901,C1(NC(N)=O)CCC2(CCN(C(=O)CCSc3c(C(=O)OC)ccs3)CC2)C1 1902,c1(NC(C2C(O)CCN(C(C3C(C)(C)C3)=O)C2)=O)c(Cl)cc(Br)cc1Cl 1903,C(CN=c1nc(Cl)[nH]c(C)c1C#N)C1CCN(C(c2cc(SC)oc2C)=O)C1 1904,C1(CNC(C(C)Cc2cnc[nH]2)=O)(NC(=O)COCCCF)CCCCC1 1905,C1(NC(C)=O)CCC(C(=O)NCC(c2cccc(C)c2)N(C2CCCC2)C)CC1 1906,c1(C(=O)OC)cc(S(=O)(=O)N2CCOCC(CNC(C3CCCO3)=O)C2)c[nH]1 1907,C1(NC(c2cscc2C(F)F)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1908,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1909,CC1CC(CNC(=O)CN(CC(C)(C)C)C)CN1C(C1C2COCC12)=O 1910,CC(C)(C(=O)N1CCCCC1)C1=CCN(C(=O)C=CCN(CCCOC)C)C1 1911,N1(C(CC2CC(NC(=O)COC3CCCOC3)C2)=O)CC(CO)C2(CC2)C1 1912,C(CCC(C)(C)NC(=O)CC1CC1COC)NC(COCCOCC)=O 1913,CC1OCCCC1C(=O)NC(C1CN(C(C2CCCN2C=O)=O)CCO1)C 1914,CCC(CC)(CO)C(=O)NC(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1)C 1915,Cc1cnc2c(C(N3CC4(CCC4NC(=O)CC4CCC4)C3)=O)cccn12 1916,C1(C)(C(c2n(CCCOC)nnn2)NCc2cscc2F)CC2(C1)CC2(F)F 1917,N1(C(C2C3(CN(Cc4ccc(C(=O)OC)c(F)c4)C3)C2)=O)CCC(O)C(F)(F)C1 1918,C1(C)(CC(=O)N(C)CCNC(c2ccnc(OC(C)(C)C)c2)=O)CCS(=O)(=O)N1 1919,c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)=O)ccc(N)c(Cl)c1 1920,c1(N2c3ccc(cc3)CNC2=O)cc(Cl)nnc1O.N1(CC(C)OC)CCCCC1 1921,c1(OC(C(=O)NCCN(C(=O)C(CC#N)N(C)C)CCC)C)ccccc1F 1922,c1(CC(=O)N(C)CC2(NC(C3CCC3CO)=O)CC2)ccc2c(c1)CCC2 1923,c1(CN(C(CC)C)C(C2CCCC23CC3)=O)ccc(F)cc1 1924,c1(N(C2CCN(C(CN(C)CCSC(F)F)=O)C2)C)ccc(O)cn1 1925,c1(OC)nc(C)cc2ccc(-c3ccc(CNC(C4CCNC4)=O)cc3)cc12 1926,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1927,C1(CC(C)NC(=O)CNC(N)=O)CCN(C(=O)C(F)(F)CO)CC1 1928,C1(CNC(c2n(CCC)ncc2)=O)CN(C)CCN1C(c1cc(C)n(CC)n1)=O 1929,Cc1scc(C(=O)NCC(c2ccc(F)cc2)NC(c2nnsc2C)=O)c1C 1930,CC1CCC=C1C(=O)N1CCC(C(N2CCC(F)CC2)=O)C12CC2 1931,Cc1cc(F)c(C(=O)NC2CC(O)CN(C(c3ccn(C)n3)=O)C2)c(Br)c1 1932,c1(C(=O)NC2CCN(C(C(CC=C)C)=O)CC2OC)c(F)ccc2occc12 1933,N1(C(c2cc(SC)n(C)c2)=O)CCC2C(CCN2C(c2occ3c2CCC3)=O)C1 1934,C1(C(N(CCCCC(C)C)C)=O)C2Cc3cc(Br)ccc3C12 1935,c1(OC)ccnc(O)c1C(=O)N(CC(C)N(C)C(c1cc(CO)[nH]n1)=O)C 1936,CC(C)(CCCCNC(=O)C(O)C1CC1)NC(c1cc(Cl)n[nH]1)=O 1937,C(=O)(C1CCCn2ccnc21)NC.C1(=O)C(C)(C)OCCCN1C(C)C 1938,c1(NCC(CNC)(C)O)ccc(S(=O)(=O)NCc2ccnc(SC)c2)c(Cl)c1 1939,C1(C(N2CC(C(C)OC)C2)=O)N(C(C2COC(=O)N2)=O)CCCC1(C)C 1940,c1(N(C(CC2(C)CCC2)=O)Cc2ccco2)cccc2c1NCCC2 1941,N#Cc1sc(=NC2(C3CN(C(=O)CNCS(=O)(=O)C(F)(F)F)CC3)CCC2)[nH]c1Cl 1942,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1943,C1(NC(C(C)n2cncn2)=O)CCN(C(C23CCN(CC2)C3)=O)C12CCC2 1944,C1(CCCNC(=O)CC2CC2C(F)(F)F)CCCCN1C(C1CCC(O)CC1)=O 1945,c1(C(N(C)Cc2cc(OC)no2)=O)cc2ccncc2c(O)n1 1946,S(=O)(=O)(c1ccc(NCc2ccco2)cc1Cl)N(CCCNc1ccncn1)C 1947,C1(c2ccc(C)cc2)CCN(C(=O)C(CN=[N+]=[N-])C2CCC2)CC1(C)C 1948,c1(C(=O)NCC2C(NC(=O)CC3CS(=O)(=O)C3)COC2)ccc(C2CCC2)cc1 1949,N1(C(COCC)=O)CCC(C2(NC(c3nc(O)nc(O)n3)=O)CC2)C1 1950,C1(C(N2CCC(Cc3cn(CC(=C)CC)nn3)CC2)=O)CCc2ccccc2C1 1951,C1(C(=O)NCC2CN(C(=O)CCc3ccsc3)CCO2)CCc2nncn2CC1 1952,C(=O)(C(C)(CC)CO)NC1CCN(C(C=CC=CCC)=O)C1C 1953,C(CCN=C(NCC(=O)N(C)C)NC1CCC2CC12F)N1CCN(C)CC1 1954,N1(C(C2(OC)CCCC(C)C2)=O)CC2CCCC1C2CNC(c1cc(C)co1)=O 1955,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1956,Cc1cnc(NCCCCCF)c(S(=O)(=O)NCCCC2CCS(=O)(=O)C2)c1 1957,C1(C(C(=O)N(CC(CC)O)C)(C)C)CCCN(C(C23CC(F)(C2)C3)=O)C1 1958,N1(C(C(C)N(CC)CC)=O)CCN(C(c2sccc2SC)=O)CC1.C(CC)N 1959,c1(C(=O)NCCCC(C)NC(c2cnc(C)nc2)=O)cc(C#N)[nH]c1C 1960,C(CCN(C(=O)Cc1cn[nH]c1)C)(C(C)(C)C)NC(CCC1CC(C)C1)=O 1961,c1(C(N2C(C)CN(Cc3ccc(Cl)c(Cl)c3)CC2)=O)cn2cccnc2n1 1962,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(CC)CC)nn1 1963,N1(C(C=C2CCN(C)CC2)=O)CC2CN(C(=O)CC3CCCO3)CC2C1 1964,C1(NC(C2CCN2C(=O)C(O)C2CCC2)=O)CC2CCN(CC1)C2 1965,CN(CCC1(O)CN(Cc2ccccc2)C1)N1CCCC2C(O)C(C)(C)C12 1966,C12(C(N(C3CCCN(C(c4[nH]cc(C)c4)=O)CC3)C)=O)CCCC(CCC1)C2 1967,CCCCC(C)(C)C(=O)NC1CCC1NC(c1cnccc1C(=O)OC1CC1)=O 1968,C12(NC(Cc3cccc(OC)c3)=O)CCC(CC1)N(C(c1cccc(F)c1)=O)C2 1969,N12CC3CCC1CN3C(=O)C1(CCCOC1)C2=O.c1(OC)cc(O)nc(O)n1 1970,N1(C(c2nnn(C)c2N)=O)CCC(C)(C)CC1C(=O)NC(C)(CO)CO 1971,C1(C(N(C2CN(C(c3sc(CC)c(C)c3)=O)C2)CCOC)=O)C(C2CC2)C1(F)F 1972,N1(C(C=C(C)C(C)C)=O)CC(C(=O)NC(c2cn(C)nc2C)C)C(F)(F)C1 1973,C=CCCCCCCC(=O)NC1CCCC1NC(C1C=C(C)CS1)=O 1974,N1(C(=O)Cc2ccccc2)CCCCC(Nc2ccnc(I)n2)C1 1975,C1(C(N2CCC(COC)(NC(=O)CC3CC(F)C3)CC2)=O)C2(CCC2)C12CCC2 1976,n1(CC(C)NC(N)=O)cc(CC2CC2)nn1.C12CCCC1CNC2=O 1977,c1(C(C(=O)OCC(c2cn(CCCC#N)nn2)=O)=O)ccc(O)c(Br)c1 1978,C1(NC(CCCC#C)=O)CC2CCC1CN(C(C1CCC(=O)NC1)=O)C2 1979,c1(C(=O)NCCC2(O)CCN(C(C34OC(C)C(C3)C4)=O)C2)cccc2occc12 1980,C1(N(C2CSC2)C(C2CCN2C(C)(C)C)=O)(C(=O)NCC)CSC1 1981,n1(CCC)ncc(C(N2CC(NC(=O)CC(C)(C)C)C3CC23)=O)c1C 1982,c1(C(=O)NCC(C2CCC2)NC(c2csc(Cl)n2)=O)ccc([N+](=O)[O-])cn1 1983,C12(NC(=O)COc3ccc(CO)cn3)CCC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 1984,C12(CNC(CC(=O)OC)=O)CN(C(=O)Cn3ccnc3C(C)C)CC1CCO2 1985,N1(C(=O)NC2CN(C(C)C(=O)Nc3ccco3)C2)CCC2(CCC(O)C2)C1 1986,C1(NC(C2CCC(CC)O2)=O)(CO)CCN(C(=O)CCN2CCC2)C1 1987,Cc1ncnc(C)c1CC(=O)NC1(F)CCCN(C(=O)C(C)C(C)O)C1 1988,c1(C(=O)NC(CC=C)CNC(=O)C(F)n2cccn2)ccc(Cl)nc1F 1989,Nc1c(C(N2CCC(NC(=O)C=Cc3cc[nH]n3)C23CCC3)=O)ccc(Cl)c1Cl 1990,C1(CCCC)CCN(C(=O)CCN(C(=O)CN2CC3CC3C2)CCO)C1 1991,C1(CC(=O)NCCn2cc(-c3ccnn3CCO)nn2)CC2COCC12.C1CC1 1992,N1(C(C2C3(CCN(C(CC4(N(C)C)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 1993,c1(C(N2CCOCC(NC(c3c(C)onc3)=O)C2)=O)cc2c(Cl)cccc2[nH]1 1994,N1(C(C2CC(C)C2)=O)CCc2onc(C(=O)NCC3CCN(C)C3)c2C1 1995,C1(CC)CN(C(C2(C3CC3)CC2)=O)CCC1NC(=O)C(C)=CC(C)(C)C 1996,c1(OC)ccccc1C(=O)NC(CNC(=O)C(c1cccc(Cl)c1)OC)CC(C)C 1997,CCC(C)(CCCNCC1c2cccc(c2)O1)C1CC1.OC 1998,C1(NC(=O)CCF)CCOCC1NC(=O)Cc1ccn(-c2ccc(Cl)cc2)n1 1999,C(=O)(CCC(C)(C)NC(c1ccc(F)cc1)=O)NC(C#C)CC 2000,C(=O)(C(O)C1=CCCCC1)NC(C)CCC(=O)NC(CCO)C1CC1 2001,N1(C(c2cn(-c3c(COC)c(O)ncc3)nn2)=O)CCC(C(=O)O)=C(F)C1 2002,c1(CC)cccc2c1CN(C(=O)C(=O)Nc1ccc(Cl)cc1)CC2 2003,c1(NC2C(NC(c3cccc4nc(O)oc34)=O)CC2)ncc(Cl)cc1[N+](=O)[O-] 2004,CCCC(O)CC(=O)N(CC(O)CNC(=O)Cc1cc(N2CCCC2)ncn1)CC 2005,Cc1cccnc1CCNC1CCN(CCS)C1.c1(O)ccccc1C 2006,C(=O)(C(C)C(CC)CC)N1CC(CC(=O)N(CC(NOCC)=O)CC)C2(C1)CC2 2007,c1(C(=O)NCC(C)CN(C(=O)CC2COCCO2)C)ccc(-c2ccccc2)o1 2008,c1(OC(CC2(C(CCCOC)=O)CCSC2)=O)cccc(F)c1 2009,C=C=C(C)CC(=O)NCC1(F)CCC(NC(=O)Cn2ncc(Br)c2C)C1 2010,CC(N=c1ncc(Cl)c[nH]1)C1CCCN(C(=O)C(CO)c2ccccc2)C1 2011,C1(C(=O)NC2CC3(C(NC(=O)Cn4cncn4)C3)C2)CCc2ccc(F)cc2O1 2012,c1(COCC(N2CCC(CCNC(C(CC)O)=O)C2)=O)ccccc1Cl 2013,Cn1cc(C(N)=O)c(=NC(=O)C2CCC(NS(=O)(=O)c3ccccc3Br)CC2)[nH]1 2014,C1(OC)(CNC(=O)Cn2cc(Br)cn2)CCN(C(C2C3COCC23)=O)C1 2015,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2016,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2017,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2018,C(C(C)C(=O)NCCCNC(C1CCC(=O)C1)=O)OC(C)=O 2019,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2020,N1(C(=O)C=CC=C(Cl)Cl)CCc2ccccc2C1CNC(C1(CCF)CCC1)=O 2021,C1(N(C(=O)C(C)NC=O)CCOC)CCN(C(=O)CCC2CCC2)CC1 2022,c1(C(N(C(C)C(=O)NCC(C)S(C)(=O)=O)CCC)=O)cnn(C)c1Cl 2023,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=O)[nH]1)CC2 2024,C1(C(N2C(C(N(C)CC3COCCO3)=O)CC2)=O)CCC2(CCC2)O1 2025,c1(CCCC)ccc(C(=O)NCC2CC2CNC(C2CCCO2)=O)cc1N 2026,C1(NC(COC(CC)(C)C)=O)CCN(C(C2CSCC(=O)N2)=O)CC1OC 2027,C1(C(N2CC(NC(c3c(OC)ccs3)=O)C(C)C2)=O)CN2CCCC2CO1 2028,c1(N(C(c2cc(-c3ccccc3)nc(O)c2)=O)C2CC2)cnnc2ccccc12 2029,C1(C(N(CCC(=O)NCC2CCCS2)CCO)=O)C=CCCC1 2030,c1(CNC(C(C)=O)=O)cnn2c1CN(C(C1(F)CCC1)=O)CC2 2031,c1(OCC)c(Cl)cc(NC(c2ccc([N+](=O)[O-])o2)=O)cc1Cl 2032,O=C1COC(C(=O)NCC2CN(C(c3ncn(-c4ccccc4)n3)=O)C2)C1 2033,N1(C(C2N(C)CC(C)(C)C2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C(F)(F)CC1 2034,N1(C(C(N2CCOCC2=O)C)=O)CC2CCC2(NC(=O)CC2CCCOCC2)C1 2035,c1(CN(C(C(C)c2ccsc2)C2CC2)C2CC2)ccc(Cl)c2cccnc12 2036,N1(C(C(C)(C)CF)=O)CCN(C(c2cccc(F)c2)=O)CC1CC1CC1 2037,C1(CNC(=O)COc2ccccc2)CCC(NC(C2CC2C2CC2)=O)CC1 2038,CCCC(C)CC(=O)NC1CCC(NC(C2CCCOC2)=O)C1 2039,C1(CNC(C(=O)NC(C)C)=O)CCCCN(C(c2cc3[nH]ccc3s2)=O)C1 2040,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2041,c1(C(=O)NCCSCCC(F)(F)F)cnc2c(Br)cc(Br)cc2c1 2042,C1(CN(CCCC#C)C)CCCN(C(=O)C(c2cccc(C)c2)O)C1 2043,C(CC1=CCCCC1)NC(N(CCCS(C)(=O)=O)c1ccccc1)=O 2044,N1(C(c2ccc(COC)[nH]2)=O)CCCC2CN(C(C3(F)CCC(C)CC3)=O)CC12 2045,c1(C(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)C2)=O)cccc2cnccc12 2046,C=CCC(CN(C(c1ccn(CCF)n1)C(=O)NC(C)CC)C)CC(C)C 2047,C(CCCCCNC(=O)Cc1ccc(F)cn1)NC(c1c(SC)csc1)=O 2048,C1(CC)CCCN(C(c2ccc(OC)s2)=O)C1C(=O)NC(C12CCC(CO1)C2)C 2049,c1(CCC)c(C(N2CC(O)(C(C)NC(=O)OCC)C2)=O)nnn1CCC 2050,c1(C(C)C)nnsc1C(N1CC(CCNC(=O)CCc2ncccn2)C1)=O 2051,c1(C(=O)NC2C3CC(NC(c4cncs4)=O)CC32)ccc2[nH]ccc2c1 2052,C12(NC(c3cnns3)=O)CCN(C(=O)CCc3cncc(Br)c3)CC1C2 2053,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)C=CCO)CC1CC(F)(F)F 2054,c12c(Cl)ccc-1c2Cl.N1(CC)CCN(C(c2cnccc2C)CN(C)C)CC1 2055,c1(C(N(CCC(C)NC(CCC)=O)C)=O)cnc(OCC(=O)NC)cc1OC 2056,N1(C(C(CC)n2cncn2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1CC1CC1 2057,C=CCC(CC)C(=O)NCCC1CN(C(=O)CCC(=O)NC2CC2)CCS1(=O)=O 2058,c1(C(N2CCC(CNC(C3CN4CCC3C4)=O)C2)=O)cn2ccccc2n1 2059,C1(C(=O)NC(CNC(C2(C)ON=C(C)C2)=O)(C)C2CCC2)CC2CC1CC2O 2060,CS(=O)(=O)c1ccccc1C1=CCN(C=O)C1.C(C)(C)(C)OC=O 2061,C(C(=O)NCc1ccco1)(c1ccns1)N(CCOC)CC1CC1 2062,C1(CCC(=O)NCC(C)CN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)CCCOC1 2063,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC(C)C)CCC2CO)c1 2064,Cn1ncnc1CNC(=O)C(O)C1CN(C(=O)CC2OCCO2)C1 2065,O(C=C(C#N)C(=O)N1CCC(CCNC(=O)COCC2CCCO2)C1)CC 2066,c1(C(=O)NC2CCCC(NC(Cc3c(C)n[nH]c3)=O)C2)ccc(S(=O)(=O)CF)cc1 2067,C=Cc1cnn(C)c1NC(=O)C(=O)NCc1cc(OCCOC)ccc1F 2068,c1(C(C)C)ccc(C(=O)NCC2C=CCN2C(=O)CSC(=O)OC2CCCCO2)s1 2069,N1(C(c2nc(C)oc2)=O)CCC(O)C(NC(=O)CCCOc2ccc(Cl)cc2)C1 2070,C1(N(C)C)CCCCC1C(=O)NC(CNC(=O)C(O)CC1CCOCC1)C1CC1 2071,N(C1CCCOc2c(Br)cccc21)C(=O)NCCn1cc(CCS(=O)(=O)NC)nn1 2072,C12(CC(=O)NCC3(F)CN(C(C4C(C)C4)=O)C3)CCCN1CCC2 2073,C(C(C)(C)CNC(=O)Cn1nnnc1C)N(C(C(C)OCCC#C)=O)C 2074,c1(C(C(=O)N(C2CCN(C(C3CN(C4CC4)C3)=O)C2)CC)C)c(C)noc1C 2075,CCCCCCC(C)NC(=O)CC1C2CCC(C2)N1C(c1ccc(C(F)F)o1)=O 2076,c1(C(=O)NCC(CN(C(=O)CO)CC)O)cc(C)n(C)c1C.c1(OC)ccsc1 2077,c1(C(C)C)nccc(C(N2CC3C(NC(=O)CCCC4CCOCC4)C3C2)=O)n1 2078,c1(OCC=C)cccc(C(C)NC(C23CC(C)(CN2)C3)=O)c1 2079,c1(Cc2nc(C)nn2C2C(C)CCCC2C)cnc2sc(C)nc2c1 2080,CCCC(CC(=O)N1CC(NC(C2CCCN2)=O)C1)c1ccccc1 2081,Cc1cc(C(N2CC3CC(C(N4CCOC(CN=[N+]=[N-])C4)=O)(C3)C2)=O)cc(O)c1 2082,Cc1nccnc1C(=O)NC1CN(C(c2ccc(OCC3CC3)nc2)=O)CC1C 2083,c1(CN2CC(C#N)C(NC(c3nccnc3Cl)=O)C2)cc(O)c(O)c(O)c1 2084,CC1CC(C(=O)NCc2ccc(-c3cccs3)cc2)N(C(C2(Br)CCC2)=O)C1 2085,C1(NC(c2c(C)cn(C)c2)=O)CN(C(=O)CC(F)(F)Cl)C2(CCOCC2)C1 2086,C1(NC(=O)NC2CN(CCCC(=O)OC)C(C)CC2)CCN(C)C(=O)C1 2087,CCCCC(O)C(C)C(=O)NC(C)C(=O)NCCOC1(C)CCC1 2088,c1(NC(C23CC(C)(C2)C3)=O)cccc(OC(F)(F)F)c1 2089,c1(CC(=O)NC23CCN(C(=O)CCc4ccsc4)CC2C3)ccc2sccc2c1 2090,CCCCC(C)C(=O)NC(c1nc(C(=O)NC(c2cccc(O)c2)C)co1)C 2091,c1(C(N2C(SCC(C)(C)OCCF)CC2)=O)ccc(NC(C(C)(C)C)=O)cn1 2092,Cc1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)c[nH]c2nccc1-2 2093,Cc1ccc(OC(C)C(=O)NCC2CC(F)CN2C(=O)CC=C(Cl)Cl)cc1 2094,c1(C(N(CC(CNC(c2[nH]cc(C)c2)=O)C)C)=O)cn(C2CCC2)nc1C 2095,c1(CC)ccc(C(=O)NC2(C)CCCN(C(c3cc(N)cc(O)c3)=O)C2)c(F)c1 2096,C(=O)(CC(C)CC(F)(F)F)NC(CC1CN(C(CC2(COC)CC2)=O)C1)C 2097,c1(CN=C(NCC(=O)NCCOC)NC2CCOC2)nccc2ccn(C)c12 2098,C(=O)(C(F)C1=CCCCC1)NC1C2CN(c3nnc(CC)s3)CC21 2099,C123CCC(CO1)(C2)C(=O)NC3.C(=O)(CC(C)(F)F)NC1(C(CC)(F)F)CC1 2100,N1(C(CNCc2n(C)c(S)nn2)=O)CCCC(S(N)(=O)=O)C1 2101,C1(NC(c2ccsn2)=O)CCC2CCN(C(c3conc3C3CCCO3)=O)C12 2102,c1(C(=O)NC(C)(C)CNC(C2(C)CCC(=O)NC2)=O)ccc([N+](=O)[O-])cc1F 2103,C#Cc1ccc(NC(=O)C(C)(C)C2CCCN2C(=O)COC2(C)CCCC2)cn1 2104,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cc(N)c(O)c(F)c2)=O)CC(C)(F)C1 2105,N1(C(c2c(COC)nn[nH]2)=O)CC(NC(c2cnn(C)c2C)=O)CC1C 2106,C12(CNC(C(C)C3CCC3)=O)CCCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 2107,c1(C(=O)NCCC2CN(C(C3(CN(C)C)CC3)=O)C2)ccc(O)nc1 2108,Cc1cc(NC(c2cc(Cl)ncc2NC(c2ccno2)=O)=O)ncc1F 2109,C(=O)(C1c2c[nH]nc2CCC1C)N1CC(CNC(Cc2ccc(C)s2)=O)OCC1 2110,Cc1ccccc1NC(CCSC1CC(F)CN1C(=O)CC(C)(F)F)=O 2111,N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(c2ccncc2Cl)=O)C2COCC12 2112,C(CC(F)F)(C(=O)NCC1(O)CCCC(C)C1)N(C(c1n(CCC)ccc1)=O)C 2113,C1(CC(=O)N(C)CC2CN(C)C2)CN(C(c2cncnc2)=O)CC12CC2 2114,C(CC(C(=O)NC(CN(C)C)C(C)C)CCOC(C)(C)C)=CC=CC.C(=O)(CCO)N 2115,C1(NC(C2CCN2C(C23COCC2C3)=O)=O)CCC=CCCC1 2116,c1(C(=O)NC(C)CCC(=O)NC2CC2OC(C)(C)C)c[nH]c2ncccc12 2117,c1(CC)ccc(C#N)nc1.n12cc(C(=O)N(CCC(C)NC(=O)NC)C)c-1n2 2118,c1(C(=O)NC(C)CC2CN(C(c3cccc(C(F)F)c3)=O)C2)ccn(C)c(=O)c1 2119,N1(C(Cc2n(C)ncc2)=O)CCC2CCN(C(c3n[nH]c(C4CC4)c3Cl)=O)CC12 2120,C12(CCC)CC(C(=O)NCCOC3CN(C(=O)CCC4CCCO4)C3)(C1)C2 2121,c1(C(=O)NCC(CNC(C2CC23CCCC3)=O)OC)ccc(C#N)cn1 2122,N1(C(C(C=CCCC)O)=O)CCCCC(NC(c2ccc(SCCF)cc2)=O)C1 2123,CCC(C)(COC)C(=O)NC1CCC1CNC(c1cccc(OC(F)F)c1Cl)=O 2124,C(=O)(C1=CSCS1)N(CCCN(C(=O)C=Cc1cc[nH]c1)C)C 2125,C1(NC(C2CCO2)=O)(CO)CCN(C(c2ccc(SC(F)(F)F)cc2)=O)C1 2126,c1(C(N2CCN(C(C#CC3(CC)CC3)=O)CC2C)=O)cccc2cc(F)ccc12 2127,N1(C(c2cn(CCC)nn2)=O)CCCC(N(C(=O)Cn2cc(COC)nn2)C)C1 2128,Cc1nn(CC(=O)NC(C)CNC(=O)Cc2ncc(Cl)s2)c2ncccc12 2129,CC(F)CC(=O)NC1CCC(NC(=O)Cc2cc[nH]n2)C1 2130,c1(OC(C)C(N2CCCCC2CCNC(C2(C)CC2(Cl)Cl)=O)=O)ccccc1F 2131,N1(C(C2CCCC(NC(C3=NOC(C)C3)=O)C2)=O)CC2(CCN(C)CC2)C1 2132,c1(C(=O)NCCOCCN(C)C(c2cccnc2Cl)=O)nn(C)c2ccccc12 2133,N1(C(CCc2n(C)cnn2)=O)CCC2(COCC(CNC(C3(CO)CC3)=O)O2)C1 2134,c1(OC)ncc(C(=O)NCC2CCN(C(C3CC(F)C3)=O)C2)cn1 2135,c1(C(=O)NCC2C(CNC(c3c(C(C)C)cco3)=O)C2)ccc(N)c(N)n1 2136,c1(C(=O)NC2C(CC)C2)c(-c2ncon2)ncn1C 2137,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2cnc(C3CC3)o2)=O)cc(F)c1 2138,CC(O)CCC(=O)NCC(C)N(C(=O)CCc1ccc[nH]1)C 2139,Cc1ncc(Cl)cc1C(N1CCNCC1c1ccc(F)cc1)=O 2140,CS(=O)(=O)c1cnn(CC(=O)NCCCNC(=O)CC2OCCC2(C)C)c1 2141,C(=O)(CN1C(=O)C(NC(CC)=O)CCc2ccccc21)NCCC1CCCN1C 2142,N1(C(c2n(C)nc(Cl)c2)=O)CCOC2(CCN(C(=O)C(=O)NCC(F)(F)F)C2)C1 2143,c1(NC(C)C2CC2)ccc(S(=O)(=O)NCc2ncn(C)n2)c2ccncc12 2144,C1(CCNC(C2C(CC)CCC2)=O)CCN(C(=O)C=CC(CC)=CC)CC1 2145,c1(CC(N2CCC(C(C(N3CC4C(CC)C4C3)=O)F)C2)=O)cccc(C)c1O 2146,C(=O)(CC(F)(F)F)NC(CNC(=O)NC(CCNS(C)(=O)=O)=O)C(C)C 2147,N1(CC)CCC(C(C)C)CC1.N12CCCC1C2=O.C12CCC1C(=O)NC2 2148,C1(OC)(OC)CCC1C(=O)NCc1nc(CNC(c2cnn(C(C)C)c2)=O)cs1 2149,N1(C(C(C)(C)CO)=O)CCC(NC(=O)CC2CC3CC3C2)CC(O)C1 2150,c1(N2CCCC(C(=O)NC3(c4cc(C)no4)CC3)C2)ncc(Br)cc1C#N 2151,N12CCCC(C)(C)C1C(=O)N(C)CCC2=O.c1(CNC(=O)OC)ncco1 2152,c1(C(N(C(CC)C(=O)N(C2(C)CC2)C)C)=O)ccc2n[nH]cc2c1 2153,N1(C(CCc2cc(C)no2)=O)CC2C(NC(c3c[nH]nc3F)=O)C2C1 2154,c1(NC2CN(C(C)=O)C2)ncccc1S(=O)(=O)N1CCC(=C(F)F)CC1 2155,C1(CNC(CCCCN(C)C)=O)CC1C1CCCCC1.C12CC1CNC2=O 2156,C1(C(=O)NCCC(CNC(c2c(C)ccs2)=O)O)Cc2c(F)cccc2O1 2157,N1(C(=O)CC2(C(F)F)CCOCC2)CCS(=O)(=O)CC1c1ccccc1 2158,N1(C(CC(n2c(CC)ncc2)C)=O)CCOCC1CNC(c1csnc1Cl)=O 2159,c1(C(=O)NC(CCC)CNC(=O)CCc2nc(SC)no2)ccc(C(F)F)cc1 2160,c1(C(=O)OC)c(C)[nH]c(C(=O)NCC(C)C)c1C.c12c[nH]c(c1)NC2=O 2161,N1(C(=O)Nc2ccc(C(=O)OC)c(C)n2)Cc2cccc(Cl)c2C1 2162,c1(C(N2CC(CO)CC(C)C2)C(=O)NCCCSC)cc(Br)ccc1C(F)(F)F 2163,C1(NC(C(C)N(C(c2cccc(=O)n2C)=O)CC)=O)CN2CCC1(F)CC2 2164,c1(C(C)OCC)cccc(C(=O)N(CCN(C(=O)C(C)=C2CC2)C)C(C)C)c1 2165,C1(C(=O)NCC(=O)N(C2CCCC(CO)C2)C)CC(=O)NC(=O)C1 2166,C1(NC(=O)NC(C(C)C)CN2CCCC2)C=CC(C)(C)CC1 2167,c1(-n2c(CCCCCOC)nc(CCOC)n2)cc(C)ccc1C 2168,C1(CNC(CCC(C)C)=O)(NC(=O)CN2CCN(C3CC3)C2=O)CCCCCC1 2169,C(=O)(C(C)(C)C(C)NC(=O)C=CC1(C)COC1)NCC1CCN(CCC)C1 2170,C1(C(=O)NCC(CN(C(=O)CNS(N)(=O)=O)C)O)CC12CCOCC2 2171,N1(C(c2n(C)nc(CNC(c3ccc(O)nn3)=O)c2)=O)CC2(CCC(=O)O2)C1 2172,CCC(Cc1ccccc1)C(=O)N1CCC1CNC(=O)CC1(CO)CCCC1 2173,C12(NC(C=C(CCC)C)=O)CCCC1(F)CN(C(=O)CCCN(C)C(=O)C1CC1)C2 2174,N1(C(c2cnc(OC)s2)=O)CC(C)CN(C(=O)Cc2ccc(F)c(F)c2)C(C)C1 2175,N1(C(c2cc(OC)no2)=O)CCC(F)CC1C(=O)Nc1cc(C)cc(O)c1 2176,c1(OCC(N2C(CC=C)CCCC2)=O)nccc(C)c1C(=O)OC 2177,C(=O)(CC(C)C(C)(C)C)N1CC(C=CC)C(C(=O)NC2CN(CCC)C2)C1 2178,c1(C(N2C(C3CCN(C(CC4CC(SC)C4)=O)C3)CCC2)=O)cncc(Cl)c1 2179,c1(OC)ccc(C)c(C(N2CCC(C(C)NC(=O)CCN(C)C(C)=O)C2)=O)c1N 2180,N1(C(c2n(C)ccn2)=O)CCC2CC(NC(=O)CCCc3cnn[nH]3)CCC2C1 2181,c1(C(=O)NC2C(OC)CN(C(=O)Cn3nccn3)C2)cc(C#N)c(F)cc1F 2182,CCCCCC(C)CC(=O)NC1CN(C(C2CC(C)(c3ccccc3)C2)=O)CC1C 2183,C1(C(=O)NOCC2(C)CCC2)(CC)CCN(C(c2c[nH]c(=O)cn2)=O)C1 2184,CCC(C(=O)N(C1CCN(C(=O)Cc2cc[nH]n2)C1)C)c1ccccc1 2185,c1(C(C)NC(COCCC(c2n(CC)nnn2)NC2CCC2)=O)ccccc1Cl 2186,c1(C(=O)NCC2(NC(C3CCCCC3F)=O)CC2)c(F)ccc(F)c1Cl 2187,C1(NC(C2CCCC2)=O)CC2CC1N(CCc1ccncc1)C2 2188,c1(CC)onc(C)c1CNC(=O)CCC1CCN(C(=O)CC2(C)CCC2)CC1 2189,Cc1c(NC(=O)Cn2nc(Br)cc2CN2CCC(C)C2)cccc1Cl 2190,Cc1nc(-c2nc(-c3cnn(CCN(C)C)c3)nn2CCC2CCCC2)ccc1F 2191,C1(CC)CC(C(=O)N(C2CN(C(c3nn(C)cc3Cl)=O)C2)C)CCO1 2192,N1(C(C(C)=CC)=O)CC(S(=O)(=O)N2CCN(C(=O)C(C)N(C)C)CC2)C1 2193,c1(C(=O)NCCC2CN(C(C(CC#C)C)=O)C2)ccc(SCC)c(F)c1 2194,c1(CC)cnc(O)c(C(=O)NC2CN(C(c3csc(C(F)(F)F)c3)=O)CC2C)c1 2195,c1(C(=O)NC(C(C)NC(c2c(C)cnn2C)=O)CO)cccc(Br)c1Cl 2196,C(=O)(CC(C)CC)NCC(=O)NC(C(=O)NCC(=O)N(CCCOC)C(C)C)C 2197,c1(CC(=O)NC(C2C(C(N3C(COC)CCCC3)=O)C2)C)cccc(F)c1F 2198,c1(C(N(C2CN(C(=O)C=CCn3cncn3)C2)C)=O)ccc(C#N)s1 2199,CC1CN(C(=O)CCn2cnnn2)CCN(C(=O)C2CC2)C1.C12CCCN1C2=O 2200,N1(c2cc(CC)nc(CC)n2)CC2CCN(C(=O)Cc3cccnc3)CC(C2)C1 2201,N1(C(C=CCN(CC)CC)=O)CC2(CC2)CC1C(=O)NC(C(C)C)C1CCC1 2202,C1(CNC(c2c(OCC)scc2)=O)CCC(C)(C)CN1C(=O)C(C)CF 2203,c1(NC(C(c2ccccc2C)OCCCCCC)=O)ccc(SC2CC2)c(F)c1 2204,N1(C(c2ncn(C(C)C)c2)=O)CC(C(N2CC(OCC(F)F)C2)=O)C(C2CC2)C1 2205,C(C)(CCC(=O)NCCC1CC(NC(c2cccc(F)n2)=O)C1)OCC 2206,N1(C(c2cncc(NC)c2)=O)CCOCC12COCCN(C(=O)C=C(C)C1CC1)C2 2207,N1(C(CC=CC(C)(C)C)=O)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CC2C1 2208,c12ccc3nc(oc3c1)S2.Cc1cc(CNC(=O)NCCn2ccnn2)cnc1Cl 2209,N1(C(C=CC=CCC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CC1C(F)F 2210,c1(C(=O)NCC(CC(=O)N(CC(CSC)OC)CC)OC)ccc2[nH]ccc2n1 2211,C=CCCC(F)(F)C(=O)N1CC(NC(=O)CC2CCC2)C(c2ccccc2)C1 2212,N1(C(C=C(CC)C)=O)CCC(C)(C)C1CNC(c1coc(CSC)n1)=O 2213,C1(CC)OCCC1C(=O)NCc1cc(C(=O)NC(C23CC(CO2)C3)C)n[nH]1 2214,c1(C(=O)NC(C)C(CO)NC(=O)CCC2CCCO2)cc2n(c1)CCCC2 2215,c1(C(N2CC(CNC(c3ccc(C(C)(C)C)s3)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 2216,C(=O)(CC1=CCOCC1)N(CCOCCN(C(C(CC#C)(C)C)=O)C)C 2217,C(CCN=C(NC(C)C)NC1CC1(C)C)N(CC)CC 2218,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2219,C(=O)(C(O)CC(F)F)NCCC1(O)CN(C(C(C)(C)CF)=O)C1 2220,C1(CNC(c2c(CC)n(C)nc2)=O)CN(c2cc(C)nc(SC)n2)CC(C)(C)O1 2221,c1(C(N(c2nc3ccccc3o2)CCOC)=O)cc(C)nc2c1nc(C)n2C 2222,CC(C)(C(=O)NC1CC2(C1)CC(NC(C1CC3(CCC3NC(N)=O)C1)=O)C2)C(N)=O 2223,Cc1cc(C(F)(F)F)cc(CCN2CC(C(=O)N(C)C)OC(C)C2)c1 2224,c1(C(N(CCO)CC)=O)cnn(CCNC(=O)C(O)Cc2cnc[nH]2)c1 2225,c1(C(=O)NC(C(C)NC(CSCCC)=O)(C)C)ccc2cc(F)ccc2n1 2226,c1(C(=O)NCC(CNC(C(c2c(C)noc2C)CC)=O)C)ccc(C)c(F)c1N 2227,C(=O)(C(C)(C)C(=O)N1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C(CCOC)C1)NC 2228,c1(CCC(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncnc1 2229,N1(C(CCC2CCCN(C)C2)=O)CCC(F)(CNC(c2ccsc2C#N)=O)CC1 2230,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2231,C(=O)(CCCCCC(C(=O)NCc1cccs1)N1CCC(c2cccnc2)C1)OC 2232,c1(CN2CCOCC(NC(C3OCCN(C)C3)=O)C2)cnc2ncccn12 2233,c1(C(=O)CC23CCN(C2)C3=O)[nH]c2c(c1C)CCCC2.c1(CC(=O)OC)cscn1 2234,C1(CC)CCCCCCN1C(=O)CC(C)C(C)(C)NC(c1cccc(O)c1F)=O 2235,C(=O)(CC1=CCCC1)N1C2C(C(=O)NC(C3CCOC3)CO)C(C2)C1 2236,CCS(=O)(=O)c1ccc(CN=c2ccnc(NCc3cc4c(s3)CCC4)[nH]2)cc1 2237,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OCC)nn1)=O)CO 2238,N1(C(C2(OC)CCSC2)=O)CCC(F)(F)C(CNC(=O)CC2CC3(CC3)C2)C1 2239,C1(CO)C(=O)N1.CC(C)CCO.C1(C)C(=O)N1.C(C(=O)NCCF)N 2240,c1(C(N2CC(C)N(C(C34CC=CC(C3)OC4)=O)CC2)=O)cc2nccn2c(O)n1 2241,Cc1nn(CCN2CCCCC2)c(C)c1I.N12CCCC1C(=O)OC(C)C2=O 2242,CCC(C)C(F)C(=O)NCCCCC(CO)NC(=O)Cc1csnc1C 2243,CCC(CC)CCC(=O)NCC1(NC(=O)CCC2CC2(Cl)Cl)CCOC1 2244,c1(NC(c2ccc(CNC(CCC(C)OC)=O)cn2)=O)ccc2c(c1)OCC2 2245,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2246,N1(C(c2n(C=C)nnc2)=O)CCOC2(CCN(C(=O)CC(C)(O)COC)C2)C1 2247,c1(C(=O)NCC2C3CN(C(CCC(=C)Cl)=O)CC32)cc(C)c(=O)n(C)c1 2248,C(CCC(N)=O)(C(=O)NCC1CCN(C(c2cc(O)n(C)n2)=O)CC1)NC(C)=O 2249,C(=O)C(C)(C)CC#N.C(CC(COC)NC(=O)C=CCF)OCC 2250,c1(C(=O)Nc2ccc(OC(F)(F)F)cn2)ccnc(CNC(C2(O)CCOC2)=O)c1 2251,N1(C(C(C)NC(CC)=O)=O)CCc2ccccc2C(NC(=O)CSc2ccco2)C1 2252,N1(C(CCC=CC)=O)CCN(C(c2csc(-c3cnc[nH]3)n2)=O)C(C)C1 2253,Cc1ccc(C(N2CCN(C(=O)C(c3cscn3)N(C)C)CC2C)=O)c(C)n1 2254,C(=O)(CS(=O)C(F)(F)F)NCC1(O)CN(C(Cc2ccc(CC(C)C)cc2)=O)C1 2255,O(C1CCCc2c(C(F)(F)F)cccc21)C.c1(OC)cccnc1CC=O 2256,Cc1cc[nH]c(=N)c1C(=O)N(C)CCNC(c1cnn(-c2cccc(F)c2)c1)=O 2257,C(CC(C(=O)N1CCC(CCF)CC1)NC(c1ccccc1)=O)OC 2258,c1(C(=O)NC(CC)CNC(c2cn(C)nc2O)=O)cc(C)cc2c1CCC2 2259,N1(C(CCc2ccn(C)n2)=O)CC(CNC(C2(C#N)CC3CC3C2)=O)C(C)(C)C1 2260,C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(c1c(C)cc(C)nc1S)=O)C 2261,c1(C(N(CCN(C(=O)CC2CC2(C)C)C)C)=O)cccnn1 2262,N1(C(Cn2nc(C)c(Cl)c2)=O)CCN(C(=O)Cc2ccns2)C(CCO)C1 2263,C(=O)(CC(CC)C(C)C)N1CCCC(CC)C1C(=O)NC(C)C(C)(C)OC 2264,C1(C(=O)NC(CC2CN(C(c3cc(C)c(Cl)cc3)=O)C2)C)CCc2nnnn2C1 2265,c1(C(=O)NC2C(CNC(CCCc3onc(C)n3)=O)CCC2)cc(F)ccc1N 2266,c1(C(=O)NCCCCCN(C(c2c(SC)snn2)=O)C)[nH]cc2c1CCCC2 2267,N1(C(c2nc(C)n(C)c2)=O)CCC2CCC(C1)N2C(C1CN2CCCC1C2)=O 2268,C(C(C)C(C)C(=O)NCC1(CNC(C23CCC(CC2)C3)=O)CCCC1)OC 2269,c1(SCC(=O)NC2CCCCC2NC(=O)Cc2cc[nH]n2)ccccc1F 2270,C=C=CC(C)C(=O)NCc1ccc(C(=O)NCCC2CCCCC2)cc1 2271,N1(C(CC(C)n2cccn2)=O)CCC2(CCN(C(=O)CC3CCC(C)(C)O3)C2)C1 2272,c1(C(C(=O)NCCN2CCOCC2)N(C(C)C2CC2)CC)cccc(F)c1Br 2273,C(=O)(CCC(=O)N1CCCC1(CCOC)CN)NC 2274,n1(CCOCC)ncc(CNC(=O)CCN2CCN(CC)CC2)c1C 2275,FC1(F)C2C3CC(NC(CCCc4ccccc4Cl)c4ccccc4)C3CC12 2276,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2277,CC(CC(=O)N1C2CCC1(CNC(=O)CC1CC1(C)C)CC2)C(F)F 2278,C1(NC(c2c(CC)occ2)=O)CCCCC1CNC(c1nc(Cl)oc1C)=O 2279,c1(CNC(CNC(CN(C)C)=O)=O)cccc(CNC(c2sc(F)cc2Cl)=O)c1 2280,N1(C(CCC(=C)Cl)=O)CC2(COC(CNC(C3CCCC(CC)CC3)=O)C2)C1 2281,c1(CNC2C(C(=O)NCC3(C)CCC3)CCCC2)ccc(O)c(O)c1 2282,C1(C(=O)NC(CCC)C)CN(C(=O)CCCF)CCC1(C)C 2283,c1(C(=O)NCCN(C(=O)Cn2cccnc2=O)CC)c(C)ncn1O 2284,c1(OC)cc(C)ccc1C(=O)NC1C=CCN(C(C2(C#N)CC3CC3C2)=O)C1 2285,c1(C(=O)NCC2(CNC(c3cc(COC)no3)=O)CC2(F)F)cnc[nH]c1=N 2286,c1(N(CCN(C(C)C)OCN2CCCC2=O)C)cc(Br)n(C)c1 2287,c1(C(N2CCOC(C(N)=O)C2)C(=O)NCC(=C)C)c(C)cnn1CC 2288,C1(NC(C(n2cc(Cl)cn2)C)=O)CN(C(c2cc(F)c[nH]2)=O)CC2(CCC2)C1 2289,c1(CC)[nH]ccc1C(=O)NCCCCC1CN(C(=O)Cc2cnc(C3CC3)s2)C1 2290,c1(C(N2CC(N(C)C(C3CC4C=CC3CC4)=O)C3(C2)CC3)=O)ccc(S(C)(=O)=O)[nH]1 2291,C(=O)(C(C)(C)CC(=O)NCC1CN(C(=O)C(CCc2ccccc2)OC)C1)OC 2292,C(CNC(=O)Cc1ccncc1)(CC(F)(F)F)NC(C(CC)n1nccc1C)=O 2293,N1(C(c2csc(Cl)c2)=O)CCCN(C(=O)C(O)C2CCC2)C(CO)C1 2294,O=C(C1NCCc2ccccc21)NCC(C1CCCCC1)=O 2295,c1(C(=O)NCC2N(C)CCN(C(C(C(C)C)C)=O)C2)cncc([N+](=O)[O-])c1 2296,CCC(F)(C(=O)OC)C(=O)OCc1cc(Cl)cc(Br)c1 2297,c1(CC)nc(C2CCCN(CCOc3ccccc3)C2)n(-c2c(C)noc2C)n1 2298,c1(C(NNC(c2n(C)cc(CNC(=O)OC(C)(C)C)c2)=O)=O)nccc(F)c1Cl 2299,c1(CNCC2(NC(N(C)C)=O)CCOC2)cc(C2CC2)n(C(C)(C)C)n1 2300,C(C)(C(C)COC)(c1n(CCC)nnn1)NCC(C)(C1CC1)OC 2301,C1(NC(Cn2c(C)nnn2)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)C(C2CC2)C1 2302,c1(C(N(CCC(=O)NCCC2ON=C(C)C2)CCO)=O)cncc(F)c1C 2303,c1(C(=O)NCC(C)CNC(c2cc[nH]n2)=O)cc(OC(F)F)ccc1F 2304,n1(CCC(=O)N(CC#C)CC=C)ccc2cccnc12.C1(=O)CC(CC=C)N1 2305,C1(CC(=O)NCCOCC(C)C)CCCC(=O)N1 2306,CC1CN(C)CC1C(=O)NCCCNC(c1ccc(OCC2CC2)cc1)=O 2307,C1(OC)CCCCN(CC(=O)NC2CCOCC2NC(c2cccnn2)=O)C1=O 2308,c1(C(=O)NC2CCCC(NC(=O)COC3CC(CO)C3)C2)ccc2cc[nH]c2n1 2309,Cc1cc(NC(N2CCCC(C(N3CCC(O)C3)=O)C2)=O)c2c(C)nn(C)c2n1 2310,C(C(O)CC(=O)NC(C)(C)CNC(c1ccc(C(=O)NS(C)(=O)=O)nc1)=O)N(C)C 2311,c1(NC23C(CN(C(C(CC)C(C)C)=O)C2)CCC3)ncc([N+](=O)[O-])cc1C(N)=O 2312,CC1=CCC(C(=O)NCC(C)(C)OCCNC(c2cnn(CCF)c2)=O)CC1 2313,C1(C(N(CCCNC(CC2(C)CCCO2)=O)C2CC2)=O)CCCC1(F)F 2314,N1(C(c2c(C)nc[nH]2)=O)CCC(NC(C2CC(C)CO2)=O)C12CCC2 2315,CCC(CCC(=O)NCCOCC1CCCC1)NC(=O)CS(=O)CC 2316,c1(NC(=O)NNC(=O)c2ccccc2O)ccc2cc[nH]c2n1 2317,c1(NC(C=CCC(C)(C)NC(C=CCCC)=O)=O)ccc(CC)nc1 2318,C1(N(C)C(C2CC2C(C)(F)F)=O)CCC(C(=O)NC2(c3ccccc3C)CC2)CC1 2319,C1(C(=O)NC(CC#C)C(=O)NC(CO)C(O)CC)CC2C(C1)C2(F)F 2320,CC1(C)C(NC(=O)N(c2ccon2)CCCC2CCC2)C12CC2 2321,N1(C(CC2CC(OCC)C2)=O)CCC2(CC2)CC1C(N1CC2CC2C2CC12)=O 2322,Cc1noc(Cl)c1CC(N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1)=O 2323,N1(C(CN(C)C)=O)CC2(C1)CN(C(=O)C(Cc1ccccc1Cl)NC=O)CC2CO 2324,c1(C(C)C(F)(F)F)nc(C2CCCO2)nn1-c1ccn(C)n1 2325,Cc1ccc(C(=O)NCC2CCN2Cc2ncn(C)n2)[nH]1 2326,c1(OC)ccc(Cl)c(NC(=O)CC2CCCN2Cc2ccc(C#N)c(F)c2)c1F 2327,C=CCC(C)C(=O)NC1CC(F)(CNC(c2nccnc2SCC)=O)C1 2328,c1(OC)cc(C(N2CC(CC(C)NC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 2329,c1(C(=O)NCC(CC)(C)NC(C2CCCC23CC3)=O)cnn(CC)c1Cl 2330,Cc1nn(CCC(=O)NC2CC2CN(C)C)cc1Br.C12CCCN(C1)C2=O 2331,CC(C)(C(=O)NC1C2CCN(C(=O)CN3CCC(F)(F)C3)CC12)C(N)=O 2332,C1(CNC(CCc2c(C)n(C)nc2)=O)CCCCCN1C(=O)Cn1nnc(=O)[nH]1 2333,C(=O)(CCC1=CCCCC1)NCC(C)CNC(=O)CC(C)O 2334,N1(C(C(C)OC(C)=O)=O)CC(CNCCCOCCOCCO)CC(F)C1 2335,S(=O)(=O)(c1cccc2ccccc12)N1C2CN(C(C(C)OCC=C)=O)C(C2)C1 2336,CON(CCC(=O)N(C(C)C(F)F)C)C(=O)C1(CCSC)CC1 2337,c1(C(c2n(C3(C)CC3)nnn2)NCCC(O)CCO)cc2ncccn2n1.NC 2338,N1(C(c2nc(-c3cc(C)cc(C)c3)sc2)=O)CCN(C(=O)CO)C2CCCCC12 2339,CC1CC(NC(=O)Cc2cc(F)ccc2O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 2340,C12(C(=O)NCC(c3ccccc3)NC(C(CC)OC)=O)CC(C(C)=O)(C1)C2(F)F 2341,C1(C(=O)NC2C(NC(c3cncc(SC4CC4)c3)=O)CC2)CC(F)(F)C1(F)F 2342,C1(CCNC(=O)Cn2ncnn2)CCCCN1C(=O)CC1(O)CCC1 2343,C=CC(C)(C)C(=O)NCC1OCCC1C(N1CC(C2CCCO2)C1)=O 2344,C1(CC)CN(C(=O)CC(C)COc2ccccc2)CCN1C(=O)C(C)CC1CC1 2345,c1(C(=O)NC2(CCNC(c3ccnnc3S)=O)CCC2)ccc(Cl)cc1Cl 2346,Cc1cc(P(C)(C)=O)oc1C(N1CCC(C(C)NC(c2ccoc2Cl)=O)CC1)=O 2347,N1(C(C2CCN(C(C34CCC(C)(OC3)C4)=O)CC2)=O)Cc2cncnc2C1 2348,C(=O)(C(C)(C1CCC1)N(C)C)NC1(CN(C(=O)C(C)(C)C2CCCCC2)C)CC1 2349,c1(CNC(CCN(C)C(C2CCCN2C)=O)=O)ncc(Cl)cn1 2350,c1(C(=O)NC2(CO)CN(C(C3CCCC(C)CC3)=O)C2)cccc2nn(C)cc12 2351,c1(OC)ccccc1CC(c1ccc(C)cc1)(F)C(N)=O.C1C(=O)O1 2352,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)C(n2ccnc2C)C)CC1)NC(C)=O 2353,N1(C(C2C(COC)CCC2)=O)CC2CN(C(=O)CN3CCCS3(=O)=O)CC2(C)C1 2354,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(c1ccn2c1CCC2)=O 2355,CC1=C(C(=O)N2CCCC2CCNC(c2cnc(O)c(Br)c2)=O)CCO1 2356,C1(C(=O)NC(C(=O)N(C)CC)C)CCC=CC1NC(C12CCN(CC1)C2)=O 2357,Cc1ccccc1C(C)NC(=O)C(C1(O)CCC1)NC(=O)COCC(C)C 2358,C=C(C)C1CN(C(=O)CC2CCN2C(c2cc(C)c(=O)n(C)c2)=O)CCO1 2359,c1(C(N(C2CCCC(NC(C(COC)O)=O)C2)C)=O)ccnc2ncc(C)cc12 2360,N1(C(=O)CNc2nccs2)CCC(NC(=O)C=CCN2CCOCC2)C(CO)C1 2361,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2362,CC1(S(C)(=O)=O)CCCN(C(C23CSC(C2)C3)=O)C1 2363,CCC(C)C(C)C(=O)NCCCCn1cc(-c2cn(C)nc2C(=O)OC)nn1 2364,c1(Cc2c(C(=O)OCC)scc2)ccc(N2CCCCC2)cc1 2365,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(=O)Cn1ccccc1=O 2366,c1(C(=O)OC)cn(C)nc1C(=O)N(C(C)CNC(=O)CC12CCCC1C2)C 2367,Cc1cc(C)c(C(N2CC(N3CC(NC(=O)CC(C)CF)CC3=O)C2)=O)s1 2368,Cc1cc(C(=O)NC(CC2CCCC2)C(=O)NCCCCCC(C)C)nc(O)c1 2369,c1(N(C2CCC2)C(C2CCC2)=O)nc(N2CCC(CC3CC3)C2)c2ncsc2n1 2370,C=CCCCC(C(=O)NCCSCCOC)NC(=O)Cc1csc(C)c1 2371,CS(=O)(=O)c1sccc1C(=O)NCC1CC(CNC(=O)Cn2ncnn2)CO1 2372,CS(=O)(=O)C12CCN(CC1)C2.C(O)(C(F)(F)F)C1(C(=O)NC2C3CCCC23)CCC1 2373,N1(C(C(C)=C2CCC2)=O)CCC(C2CC2)(CNC(c2ncnc3c2CCC3)=O)C1 2374,C1(NC(CCC(=C)C)=O)COC2(CNC(c3cnccc3OC)=O)CC1C2 2375,N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(=O)Cc2conc2C)C2CC12 2376,N1(C(C2C(C)OCC2)=O)CCC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 2377,c1(C(N2CC(CNC(CCOC)=O)OCC2)=O)cc(Cl)c(F)cc1OC 2378,c1(NC(C2CCCC2NC(C2CC23CCOC3)=O)=O)c[nH]ccc1=O 2379,C1(NC(c2cc(SC)oc2)=O)CC2CN(C(=O)Cc3c(C)noc3Cl)CC12 2380,c1(C(=O)NC2CN(C(c3cc[nH]c3C3CC3)=O)C2)ccnc2cnsc12 2381,c1(C(N2C3CN(C(C(C)n4cnnn4)=O)C(C3)C2)=O)ccc2c(O)nnc(O)c2c1 2382,c1(C(=O)NC(C)CCNC(c2cc(Br)ccn2)=O)ccc([N+](=O)[O-])cn1 2383,C1(CC(=O)NCC(CC)NC(c2n[nH]c(C)c2Cl)=O)OCCCC1(C)C 2384,Cc1cc(Cl)cc(C)c1C(=O)NCC=CCNC(=O)CCOC1COC1 2385,C12(CNC(c3n(CC#C)ccc3)=O)CN(C(=O)COC3CC3)C(CO)(C1)C2 2386,C1(O)(C(C)NC(=O)CC2NC(=O)NC2=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1 2387,C1(C(=O)NCc2cncc(OC)n2)CN(C(=O)COCCC(C)C)CCC1C 2388,N1(C(C(=O)OCC)C)CCN(C(C2(NC(C)=O)CCCC2)=O)CC1 2389,C(C(C)C(F)C(=O)N(CC(C)O)CCF)NC(CC1(OCC)CC1)=O 2390,C1(C(=O)NCC2C=CC(CNC(Cc3cc(COC)on3)=O)C2)CCC(C)CC1 2391,C1(C(N(C)CC2(CNC(C(C3CCOCC3)OC)=O)CC2)=O)CCCCO1 2392,C1(CC)C(NC(C2CCOC2)=O)CCCN1C(c1cnc(C(F)F)s1)=O 2393,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)C=CC2)=O)ncnc2ccsc12 2394,N1(C(C2N(CCC)CCC2)=O)CCC(C)(CNC(C2(N(C)C)CCC2)=O)C1 2395,CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CNC(N)=O)CC(CO)C1 2396,Cn1ncc2ncnc(N3CCN(C(C4CCSCC4)=O)CC3CO)c12 2397,N1(C(CCNS(CC)(=O)=O)=O)CCCC1CNC(=O)CCn1ccnc1 2398,Cn1c(O)nc2c(C(=O)NC3CCN(C(c4cnc(O)s4)=O)CC3F)cccc12 2399,c1(SC)cc(C(=O)NCC2CCN(C(=O)C(O)c3ccsc3)CC2)oc1C 2400,c1(C(N(CC(C)CNC(=O)Cc2cccnc2Cl)C)=O)ccnc2c1CC(=O)N2 2401,n12nnnc1C2.c1(C(C(=O)NCCC2CN(C(C)C)C2)OC(C)=O)ccccc1 2402,N1(C(C(C(=C)C)(C)C)=O)CC(NC(=O)C(C)(C2CC2)OC)CC2(CCC2)C1 2403,c1(C(=O)NC2CCCN(C(=O)CCc3ccccc3O)C2)ccc([N+](=O)[O-])s1 2404,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)N(C(C)C)Cc1nnc(CC)o1)C 2405,C1(NC(=O)C(O)CC2CC2)CCCCC(F)(F)C1 2406,C1(C(N2CC(CNC(C3CCC(=O)O3)=O)C2)=O)CCC2CC2CC1 2407,N1(C(C(C)OCC)=O)CCCN(C(c2cnc(C(F)F)nc2)=O)CC1C 2408,C1(CN(C(Cn2cc(CNC(c3scc(C)c3)=O)nn2)=O)C2CC2)CCCC(C)C1 2409,N1(C(c2n(C)nc(C)c2Cl)=O)CCC2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2C1 2410,C1(CN(C)C(c2cnoc2-c2ccoc2)=O)CCCN1C(c1ccnnc1)=O 2411,CCC(C(=O)NCC(Cc1ccccc1)N(C)C(C12CC(CO1)C2)=O)N(C)C 2412,C(=O)(C(F)C1=CCCCC1)N(CCCN(C(c1ncc(CC)s1)=O)C)C 2413,Cn1cnc(CCC(=O)NCCSCC(N2CC(OCC(N)=O)C2)=O)c1 2414,Cn1ncc(CN2CCCC2C(O)C(F)(F)F)c1F 2415,C1(C)(NC(C=C(C)Cl)=O)CCN(C(C2CCN(C(C34CC(C)C3C4)=O)CC2)=O)C1 2416,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C)N(CC)CC)=O)C(C)C1 2417,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2418,N1(C(c2cc(C)cc(C)n2)C(=O)NCc2ccccc2Br)CCCC(F)(F)CC1 2419,CCC(C(=O)N1CCCC(CC(N2CC(Cn3ccnn3)C2)=O)C1)C(C)(C)CC 2420,C(=O)(C1CNC(=O)c2ccccc21)NC1C(CC(=O)OCC)C2CCC1C2 2421,C1(C(C(N2C(CSC)CCC2)=O)C)CCCN(C(c2cc(C)c[nH]2)=O)C1 2422,CC(CCCCNC(c1cscc1Cl)=O)NC(c1cscc1C(F)(F)F)=O 2423,C1(C(C)NC(C23CC(CC(F)F)(C2)C3)=O)CCCCN1C(=O)Cn1cc(Cl)cn1 2424,C1(NC(C23CC2C3)=O)COC2(CNC(C(C)OCCC=C)=O)CC1C2 2425,c1(C(N2CCC(CN(C(=O)CC(O)C3CC3)C)C2)=O)ccccc1-n1cnnn1 2426,c1(C(N2C(C(=O)NC3(CC#C)CC3)CC2C)=O)ccc(C)c(F)c1 2427,C1(C(=O)NC2(C)CN(C(CC3C(C)CCC3)=O)C2)(CO)CCCCO1 2428,c1(NC(N2C(C(=O)Nc3ncn(CC)n3)CC2)=O)cc(OC)c(F)cc1F 2429,c1(C(=O)NCC2(O)CC(NC(CCCC3C(C)C3)=O)C2)cccc2occc12 2430,C1(C2CCN(C(=O)CCC3CCC3)C2)(NC(C(C)(C)Oc2ccccc2)=O)CC1 2431,N1(C(c2nc(C)[nH]n2)=O)CC2CCN(C(c3cc(C4CCCC4)no3)=O)C2C1 2432,Cc1oc(C(C)C)cc1C(=O)NCCC(O)CNC(C1CCC1c1ccccc1)=O 2433,C(CCC(=O)NCCNC(c1c[nH]cc1CC1CC1)=O)=C(C)C 2434,C12(C(N(C)CC3(NC(C4C(c5n(C)ncc5)C4)=O)CC3)=O)CC1COC21CCC1 2435,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2436,c1(NC)c(C(N2CCCC(NC(C3(C)CCC3)=O)C2C)=O)cccc1N 2437,C12(C(N3CCC(NC(c4sncc4Br)=O)C(F)C3)=O)CCC(F)(CC1)CC2 2438,Cc1nscc1CN1CCCCC1.C12CCC(C1)NC2=O.C12(CC1)C(=O)NC2 2439,N1(C(C=CSC)=O)CCOC(C(=O)NC2(CCO)CCOCC2)CC1 2440,C1(C(C(=O)NCC(C)C)N(C2CCCCC2)CC(C)C)CCN(C)C1 2441,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2442,c1(C(N2CCC(NC(CC=C(C)C)=O)C2C)=O)ccc2c(c1)CCC(C)N2C 2443,C1(NC(c2cc(C(N)=O)oc2)=O)C2CN(C(c3nn[nH]c3Cl)=O)CC12 2444,N1(C(C(C)(C)SC)=O)CCC(C(C)(C)NC(=O)C(=O)NCC(F)(F)F)CC1 2445,c1(CC=C)ccccc1C(=O)NCC(CCOC)NC(=O)CC1OCCC1(C)C 2446,S(=O)(=O)(c1ccc(F)c(COC)n1)NC(CC)(C)C(=O)OC 2447,c1(C(=O)NCC(CNC(c2coc(Cl)c2)=O)OC)ccc2ccn(C)c2c1 2448,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CC 2449,C=C(Cl)CC(C(=O)N(C1CCCC1C)C)NC(C1CNC(=O)O1)=O 2450,c1(NC(C)CN2CCSCC(C)C2)ncc(C2CC2)cc1F 2451,C1(NC(CC(C)C)=O)CN(C(=O)C(n2cccc2C=O)C)CC1(C)C 2452,C(CN=C(NCc1cccc(F)n1)NCc1cc(F)ccc1O)SC 2453,C12(C(=O)NC(C)CCNC(=O)Cc3cccc(O)c3F)CCC(CC1)C2(C)C 2454,C1(C(N2C(CN(C(c3cc(CC)on3)=O)C)CCCC2)=O)CN2CCN1CC2C 2455,CCC(COC)C(=O)NCC(CC1CCCC1)C(=O)N(C)CC1(CC(C)C)CC1 2456,C1(CNC(C(CC2CCOCC2)NC(=O)OC(C)(C)C)=O)CCCCC(O)C1 2457,C1(C(N2CCC(n3ccc4ccccc34)C2)=O)CC2(CCC2)C12CCC2 2458,c1(N(CC(=O)NCC)C)ccc(S(=O)(=O)NC(CO)C2CC2)c(Br)c1 2459,N1(C(c2ccc(C(=O)OC)o2)=O)CCN(C2CN(C(c3cc(C)sn3)=O)C2)CC1 2460,c1(C(=O)NCCCCC(C)NC(=O)CN(CC(C)(C)C)C)cccc(C#N)c1Br 2461,C1(NC(c2c(C(C)(C)C)noc2)=O)CC(F)CN(C(=O)Cc2cncs2)C1 2462,c1(C(=O)NCCCCN(C(=O)Cn2cnnn2)C)sccc1Cl 2463,CC1CN(C(CC2CCC3CC23)C(=O)Nc2ccccc2Cl)CC(=O)N1C 2464,N1(C(CNC(=O)COCCCOCCSC)=O)CC(C(=O)NC)C2(CC2)C1 2465,c1(CCC)c(C(N2CC(CNC(c3onc(C)c3C)=O)CC2C)=O)nnn1CC 2466,N1(C(C2(CC=C)CC2)=O)CCN(C(c2sc(C)cc2OC)=O)CC2(CC2)C1 2467,c1(C(N2CCOC(CCCNC(=O)C3CC3)C2)C(=O)NC)ccc(C2CC2)cc1 2468,c1(CNC(c2ccc(NC(C3CCC(F)C3)=O)nc2)=O)cc(Cl)ccc1[N+](=O)[O-] 2469,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)Cc2nccnc2C)csc1C 2470,N1(C(c2nc(CC)oc2C)=O)CCN(C(C2CC(O)C2)=O)CC2CCCCC12 2471,C(=O)(C1=CCC2CCC1N2C(=O)C(C(=O)OC)C(C)(C)C)N1C(CC)CC1 2472,C12CN(CC1C)C(=O)C2.C1(C(N(C2(SCCC)CC2)C)=O)CCC(=O)N1 2473,N1(C(C2N(C(C(C)(C3(C)CC3)OCC)=O)CCC2)=O)CC=C(C(C)C)CC1 2474,N(C(=NCCC1CCC1)N1CCC(C(=O)N(C)C)CC1)CC(C)N(C)C 2475,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(CC(=O)Nc2cc(OC)cc(Cl)n2)CC1 2476,c1(CN(C(c2ncc(C)o2)C(=O)NCC2CCOC2)C)ccccc1Br 2477,C1(NC(C(C)Cc2ccnn2C)=O)COCCN(Cc2ccc(F)cc2F)C1 2478,c1(C(=O)NC2(C)CC(NC(C3ON=C(CC)C3)=O)C2)cnn(C)c1COC 2479,Cc1cnc(NC(C2CC23CN(C(c2cnc(Cl)cn2)=O)C3)=O)cc1F 2480,c1(OCC(=O)NC(CN(C)C(C2CS(=O)(=O)C2)=O)(C)C)cccc(Cl)c1Cl 2481,C1(C(=O)OC)CC(n2cc(C3CCC3)nn2)CN1C(=O)CC(C1CC1)C1CC1 2482,c1(CC)nn(C)c(CSc2nc(-c3ccn(C)n3)nn2C(C)CCC)c1Cl 2483,c1(C(N(C(c2cn(CCC=C)nn2)C)C)=O)cccc2c1cnn2C 2484,c1(C(=O)NC2C3C(C)N(C(Cn4ncc(C)c4)=O)C2C3)cnc2[nH]cncc1-2 2485,c1(C(N2CCC(CNC(C(C(C)O)C)=O)C2(C)C)=O)nccc2c1CNC2=O 2486,C1(NC(c2ccc(=O)oc2)=O)CCC(O)CN(C(=O)CC2(O)CCCC2)C1 2487,O=C1CC(NC(=O)CC2CCN(C(C3(O)CCC3)=O)CC2)CCN1 2488,C(=O)(C(F)(F)C1=CCOCC1)N(C1C(O)CCN(C(C=COCC)=O)C1)C 2489,CCCCC(CCCC)NC(=O)CC(C)(C)N(C(=O)Cc1cccc(C#N)c1)C 2490,N1(C(=O)NC2CCC3SCCSC23)Cc2ccccc2OC2(C1)CN2 2491,C(=O)(C1=NNC(C(F)(F)F)C1)NC(CN(C(C1(OC)CCCCC1)=O)CC)C 2492,c1(C(=O)NC(CC)CNC(=O)CC2CC2C)ccc2nnnn2c1 2493,c1(OC)ncc(C(=O)NCCCNC(C2(C)CNC(=O)C2)=O)nc1C 2494,N1(C(CCC=C(C)C)=O)CC2CC1(C(=O)NC1(C)CS(=O)(=O)C1)C2 2495,c1(C(N(CCNC(C(C)(C(C)C)SC)=O)C(C)C)=O)cnc2c(C)cccn2c1=O 2496,C1(C(=O)NCC(C)OC)C2CCC(C2)N1C(c1onc(C)c1C)=O 2497,C(CC(=O)NCC1(NC(C2CC2CC(C)C)=O)CC1)OCC 2498,Cc1coc(C(C)C)c1C(=O)NCC1CC1CNC(C1CC(F)(CO)C1)=O 2499,c1(C(N(CCCNC(CCOCCCOC)=O)CCO)=O)c(Cl)ccnc1F 2500,CCC(CC(=O)NC(C1CN(c2ncccc2C(=O)OC)CCS1)C)C(C)C 2501,N1(C2CN(C(=O)C(COC)OC)C2)CC(NC(c2c(OCC)c[nH]n2)=O)CC1=O 2502,C#CC1CN(C(=O)CC2CCCN(C(=O)CNC=O)C2)CC1OC 2503,C#Cc1ccc(C(=O)NCC2(NC(=O)C(c3ccccc3)C)CC2)nc1 2504,N1(C(C2CCC(C)O2)=O)CC2C(NC(C3(C)CCC3)=O)C2C1 2505,CC(CC(C)(C)C)C(=O)NC(c1ccccc1)C(=O)NC1CCN(C(C)(C)C)C1 2506,CCC(CCOC)C(=O)NCC1(C(=O)NC2Cc3nccn3C2)CC1 2507,c1(CNC(C(CSC)NC(=O)C(c2cnn(C)c2)C)=O)nnc(C)n1C 2508,C(c1cc(C)no1)=CC(=O)NCC(C)N(C(CN(S(CC)(=O)=O)C)=O)C 2509,N1(C(CC(C)CNC(=O)CC2(C)CCCO2)=O)CC2(CCOC2)C1 2510,C1(C(N2CC(CNC(CCc3onc(CC)n3)=O)C(C)C2)=O)CC(S(C)(=O)=O)C1 2511,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2512,C(=O)(C(C)c1ccco1)N(CCCNC(=O)COCCN(C)C)CC 2513,C1(CC=C)(NC(c2cc(C(F)(F)F)ccn2)=O)CCN(C(=O)C(C)(O)CSC)C1 2514,C1(SCCOC(c2ncc(OCC)nc2)=O)CN(C(c2ccnn2C)=O)CC1(F)F 2515,CCCC(C)C(=O)NCC1CC1NC(c1coc(N(C)C)n1)=O 2516,C12(NC(c3scc(C)c3)=O)CCCC1N(C(C1CC(=O)C1)=O)CCC2 2517,c1(SCC)cnc(O)c(C(N2CC(NC(c3cccc(CO)n3)=O)C(F)C2)=O)c1 2518,N1(C(C2C(C#N)C2)=O)CCCC(NC(=O)C(c2ccc(Cl)cc2)(F)F)CC1 2519,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCC1CC1)C 2520,C(N=c1cc[nH]c(=NCCn2cc([N+](=O)[O-])cn2)[nH]1)c1nc(O)sc1 2521,C(CCNC(C1(Cl)CC1(C)C)=O)(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O 2522,N1(C(c2ccc(SC)s2)=O)CCC(C)C(NC(=O)CCC(F)F)C1C 2523,CC1(C2CCCN(C(=O)CC3CCCN(C(c4cn[nH]c4)=O)C3)C2)CC1 2524,N1(C(CNC(C2C=CS(=O)(=O)C2)C)=O)CCCC2(C1)NC(=O)N(C)C2=O 2525,C1(C(C)C)C(NC(c2cncc(C3CC3)c2)=O)CCN1C(=O)COCC1CCOC1 2526,c1(C(=O)NC(CCC(N2CCCC(C(=O)OCC)C2)=O)C)cccc(C)c1O 2527,C1(Nc2ccc(-n3c(CC)c(C(=O)O)nn3)cc2)CCNC2(CCC2)C1 2528,N1(C(COC)=O)CC(C2CCCN(C(=O)CC3OCCCO3)C2)C1 2529,C1(SC(C)C)CCC(C)CN1C(=O)CC1(CNC(=O)C(C)NCCC#C)CC1 2530,C1(NC(=O)NC(c2nnnn2C2CC2)C)CCCCN1C(C)C 2531,c1(C(=O)NC2(C)CCCN(C(CCC(=O)NCCC)=O)C2)cccc2cccn12 2532,C(=O)(CC(C)NC(=O)NC1CCOCC1)N(CC(C)CNC(C1CCCC1)=O)C 2533,c1(C(N(C(CN(C(CC(=C)C)=O)C)C)C)=O)ccc(=NC)[nH]c1 2534,C(=O)(CC(F)(F)C(C)C)N1CC(CCNC(C2N(CC)CCCC2)=O)OCCC1 2535,c1(N2CC(NC(Cc3c(C)cc(C)cc3O)=O)(CO)C2)ncnc2scc(C)c12 2536,O=C(CCC(F)(F)F)NC1CCC(NCCSCC2CSC2)CC1 2537,C=Cc1cncc(C(=O)NCC2CC3CCC2N3C(C23CCC(F)C2CC3)=O)c1 2538,CN1CCC(C(=O)NCC2CCC(NC(=O)Cc3nnc(O)s3)C2)CC1=O 2539,c1(CN2CCCC(NC(c3ccc(CN(C)C)cc3)=O)C2)ccc(F)c(C#N)c1 2540,C1(C(=O)NCCC(=O)NCCNC(c2nc(C)oc2)=O)CCc2ccccc2O1 2541,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C1CC1 2542,c1(C(=O)NCC2C(NC(c3ccc(CNC(C)=O)o3)=O)CC2)csc(C#N)c1 2543,N1(C(C(C)(CO)NC(c2ccc(CC)o2)=O)=O)CCN2CC(O)CC2C1 2544,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2545,CC(C)C(C)C(CNC(C1CN(C)C1)=O)NC(c1cn(C)nc1C(F)F)=O 2546,N1(C(c2scc(C)c2)=O)CCCCC2(CCN(N3CCCC3CN(C)C)C2)C1 2547,CCC(C)CCCC(=O)N1CC2(CC2)CC1Cn1cc(CC(C)C)nn1 2548,C(CCCC(C)NC(C1CC1C#N)=O)NC(C1C(COC)C1)=O 2549,C1(NC(COC(C)C)=O)CC2CC1CN(C(=O)CCc1ccc(O)nn1)C2 2550,C=C(C)C1OCCCC1NC(=O)N(C)C(c1cc(C)cc(C)c1)C 2551,C(=O)(CC(O)C(Cl)(Cl)Cl)NCC1CCC(NC(c2c(C)nns2)=O)C1 2552,C1(C(=O)NC(CC=C)CNC(c2cscn2)=O)(CO)CCCCO1 2553,N1(C(=O)NCC2(C(=O)NCCOCCOCCOC)CC2)CCOC(C)(C)CC1 2554,C1(C(N2CCC(C(C)(C)O)CC2)=O)N(C(C2CCCOC2)=O)CC12CCCC2 2555,c1(CC)n[nH]c(CC)c1CC(=O)NC12CC(CNC(=O)C(C)(C)C)(C1)C2 2556,C(=O)(C(C)(C)CC#N)N(C)CC=CC(N1CCCOCC1)=O 2557,C#Cc1cn(C)nc1C(=O)NC(CNC(=O)C(C)(C)Cc1ccc(Cl)cc1)C(C)C 2558,c1(NC2CCC(NC(C3CC4(CCO3)CC4)=O)CC2)ncnc2[nH]cnc12 2559,C1(CNC(CCc2nnc(C(C)(C)C)o2)=O)(NC(C2C3CCCC23)=O)CCOCC1 2560,N1(C(C(CC)OC)=O)CCC(O)(C2(NC(=O)C(C3CCCCC3)OC)CC2)CC1 2561,C1(C2(C)CC2)CN(C(C23CC(NC(C4CC(=O)N4)=O)(C2)C3)=O)CCO1 2562,c1(C(C)NC(CCC2CCN(C(CCCOCCOC)=O)C2)=O)c(C)n[nH]c1C 2563,C(=O)(CC(C)C(C)C)NCC(CCCC)NC(c1scnc1C1CCCCC1)=O 2564,C1(CC(=O)NC2CCC(N(C)C(c3cc(CO)[nH]n3)=O)C2)CC2CCC1CC2 2565,CN1CCN(C(=O)C=Cc2ccc[nH]2)C(C(=O)NCC2C=CCCC2)C1 2566,CC1(C)OCC2CC12NC(=O)CCC1(NC(c2ncccc2Cl)=O)CCC1 2567,C1(CNC(CCc2cccc(OC)n2)=O)CCCCN(C(=O)CCS(C)(=O)=O)C1 2568,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2569,C1(C(C)C)C(=O)N2CCC(O2)C(=O)N1.C(CC(=O)OC)OCCOC 2570,Cc1c(C(=O)NC2CCC23CN(C(C2COC(=O)C2)=O)C3)oc2ccc(F)cc12 2571,Cc1c(NC(=O)CN2CCN(C(c3ccccc3O)=O)CC2)cnn1C 2572,C1(NC(C2(C)CC3(CC3)C2)=O)CCCC(C(N2CC([N+](=O)[O-])C2)=O)CC1 2573,C1(C(=O)NC2(CC=C)CC2)CN(C(c2c(C)cccc2C)=O)CCC1(C)C 2574,c1(NCC(C)(C2CC2)NC(c2ncn3c2CCC3)=O)ncnc(Cl)c1C#N 2575,C=C(C)CCCC(=O)N1CC(CNC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2576,CCC1=C(C(=O)N(C(CNC(=O)Cn2ncc(O)nc2=O)C2CC2)C)CCCO1 2577,c1(C(=O)NCC2(C(=O)NCC3=CCCC3)CCCC2)ccnc(O)c1 2578,c1(NC(Cc2ccc(OCC=C)cc2)=O)ccc2cc(OC)ccc2c1 2579,S(=O)(=O)(C1CN(C(=O)OC(C)(C)C)C1)NCCc1onc(C(C)(C)C(F)F)n1 2580,N1(C(Cn2c(C)ccn2)=O)CCC2CN(C(C3COCCO3)=O)CC12 2581,c1(OC)ccc(F)cc1CN1CC2(CC2CNC(c2cc3sccc3s2)=O)C1 2582,c1(N(CC(C)C)C)ccnc(C(N2CCC(NC(c3ccc(Cl)s3)=O)CC2)=O)n1 2583,C1(C)(NC(C(C)N(C(c2cn(CC=C)nc2)=O)C)=O)CN2CCC1CC2 2584,c1(C(C)=O)c(C)[nH]c(C(=O)NC2(c3nccs3)CCC2)c1C 2585,C=CCC(C(=O)N1CC(C(=O)NC2(CC(N)=O)CCC2)OC(C)C1)C(C)C 2586,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2587,C1=CCC(CNC(c2nnnn2CCOC2CC2)c2ncco2)CC1 2588,C1(NC(CC2CCC(OC)CC2)=O)CCN(C(c2nonc2N)=O)CC1C 2589,C1(CN(C)C(c2ncccc2O)=O)CN(C(=O)Cn2ccccc2=O)CC12CC2 2590,Cn1ccc2c(C(=O)NC3CCCCN(C(C4CC4C#N)=O)C3)[nH]cc2c1=O 2591,C1(CNC(CCCC=C)=O)(OC)CCN(C(c2ccnn2CCF)=O)CC1 2592,C1(C(=O)OC)C(F)CCC(C(=O)OCCCC(C)C)N1C(=O)OC(C)(C)C 2593,N1(C(c2nc(CNC(C(CC)C(C)C)=O)oc2)=O)CC(C)CC(C)(C)C1 2594,C1(C(=O)NN(CC(=O)N(CCCOCC)C(C)C)C)(CC)CC1 2595,N1(C(c2cn(C)cc2C(F)(F)F)=O)CCCN(C(C2CCCCC2C(N)=O)=O)CC1 2596,c1(NC(C(C)(C2CCC2)NC(c2cc(C(C)C)[nH]n2)=O)=O)sccc1C#N 2597,C1(C)(CC)C=C(C(=O)N2CC(CNC(C3(CS(C)(=O)=O)COC3)=O)C(O)C2)C1 2598,N1(C(c2nccc(C#C)c2)=O)CCC(C(=O)NCC(F)(F)CO)=C(F)C1 2599,C1(OCC#C)CCN(C(=O)C(C)(C)NC(=O)CC2CCC(=O)C2)CC1 2600,CC(=O)CCC(=O)N1CCN(CCN(C(=O)CCC2CCC(C)O2)C)CC1 2601,N1(C(c2ncn(C)n2)=O)CC(O)CC1CNC(c1cc(C2CC2)n(C)n1)=O 2602,C1(CNC(C2CC(C)=C(C)CC2)=O)COC(C)(C)CN1C(c1coc(C(N)=O)c1)=O 2603,C1(CC(=O)NC2C3CN(C(c4c(C)oc(C5CC5)n4)=O)C2C3)CC2CCC1CC2 2604,c1(CC(=O)N(C)CCOCCNC(C2COCCO2)=O)ncc(F)cc1F 2605,C1(OC(c2ccc(-n3cnnn3)cc2Cl)=O)CCOC2(CCCC2)C1 2606,C12(NC(c3nc(C(C)=O)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2607,c1(C(N2CC(C(C(=O)N(C)Cc3c(CC)con3)OC)C2)=O)ncncc1C 2608,C(C)(CO)(C(=O)N1CC(C(N)=O)(CNC(c2cnn(C)c2Cl)=O)C1)OC 2609,c1(NC(CNC(CC)CN2CCCC2)=O)cc(-c2ccnn2C)ccn1 2610,c1(C(=O)NCC)cnn(C(C)(C)C)c1C.C1(C)C(=O)NCC1CNC(=O)OCC 2611,c1(C(=O)NCC(CNC(=O)CS(=O)(=O)C(C)C)OC)cccc2ccc(O)nc12 2612,C(=O)(CCN=c1cc[nH]cc1S(=O)(=O)NCCN1CCCC1=O)NC(C(C)C)=O 2613,c1(OC)ccc2c(c1)OCCN2C(=O)NC1CC(S(C)(=O)=O)C1 2614,c1(C(=O)NCC=CCNC(CCNC(C2C(C)C2)=O)=O)ncc(F)c2ccccc12 2615,N1(C(C(CC2CC2)OC)=O)CC(F)(F)CC1CNC(c1cocn1)=O 2616,Cc1cc(C)c(C(=O)NC2COCCC2NC(c2conc2C)=O)c(O)n1 2617,C(C(=O)NC1CCN(C(=O)CN2CC(=O)NC2=O)CC1O)(C(C)(C)C)NC(C)=O 2618,CC(O)CCCCNC(C1(CNC(=O)C(C)C2CCOC2)CCCC1)=O 2619,CC1(C)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1NC(=O)Cc1n[nH]cc1Br 2620,C(=O)(C1CCCCc2ccccc21)NCCN(C(=O)C(C)C#N)CC 2621,CC1(C)CN(C(c2csc(C(C)(C)C)n2)=O)CC(CNC(=O)CNS(C)(=O)=O)O1 2622,c1(Cn2cc(C(C)NC(CC(N)(C)OC)=O)nn2)cc2ccccc2[nH]1 2623,C(=O)(CC(C)C(=O)O)NC1CCCN(Cc2cn(CCCCC)nn2)C1 2624,C(=O)(CC1=CCCC1)NC1CCN(Cc2ccccc2)C1.CC12CC(C1)C(=O)N2 2625,c1(C(N2C(C)CC(NC(c3cc(F)ccc3F)=O)C2)=O)n[nH]c2c1CN(C)CC2 2626,C1(C(=O)NC2C(CNC(c3n(CC)ncc3Cl)=O)CC2)CC2(CCOCC2)C1 2627,N1(C(C=Cc2c(C)ncs2)=O)CC2CC(NC(c3snc(Cl)c3Cl)=O)CC2C1 2628,C1CCN(C(C)=O)C1.C(CCNC(=O)NC(=O)OCC)O 2629,C(CCC)(C(=O)NC(c1ccnn1C)C(=O)NCCOCC1CCC1)=CC 2630,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(=O)CCCc2cccc(CC)c2)C1 2631,N1(CCCC2(NC(C(CC(C)(C)C)OC)=O)CCCC2)CCC2(COC(=O)N2)C1 2632,C(C(=O)NC(C)C(=O)N(C)C1CC1)(C(C)CC)NC(CCCCOCC)=O 2633,C(CCC(=O)NC(C(=O)NCCCn1cccn1)c1cccs1)=CC(C)C 2634,c1(C(=O)NCC2COCC2NC(C2CC2C2CCC2)=O)nccc2[nH]ccc12 2635,C12(COC)CC(C(=O)NC(C)CCCNC(=O)CCc3nccs3)(CO1)C2 2636,C(CC1CCC1)(C(=O)NCC(N1CC(C)(C)C1)=O)NC(C)C 2637,C=C1CCC(NC(=O)NC(Cc2ccccc2)C(=O)N2CCCCC2)CC1 2638,Cc1cc(F)cc(C)c1C(N1CC2CCC1CN2CC1CCS(=O)(=O)CC1)=O 2639,c1(CC(C(=O)NC2C(CC)N(C(=O)C=CBr)CC2)C)ccc(C)cc1C 2640,N1(C(C(C)c2ccco2)=O)CC(C)(C(=O)N(C2CC(F)(F)C2)CCO)C1 2641,CC1=C(C(=O)NC2CC2NC(=O)CNC(C2CCCC2)=O)CCS1(=O)=O 2642,CC1(C)CCN(C(c2nc(NCc3c(F)cccc3Cl)no2)=O)CC1 2643,C#CC1(O)CC(C(=O)NC(c2cn(C)nn2)C(=O)NCc2nn(CC)nc2C)C1 2644,C(=O)(C1=NNC(=O)C1)NC(C1(O)CCN(C(C(=Cc2ccccn2)C)=O)C1)C 2645,c1(NC)cnc(C(N2CCC(C)(CNC(c3ncccc3C3CC3)=O)C2)=O)nc1 2646,C1(C(=O)NC(c2cn(C)nc2)C(=O)N2CC(c3ccn(C)c3)C2)CC(=O)CCO1 2647,CC1(C)CCN(C(=O)CCc2nccs2)C1CC(N1CCOCC1CC(N)=O)=O 2648,C1(F)(CNC(C2C=CC(NC(C(C)NC(CC)=O)=O)C2)=O)CCCCC1 2649,N1(C(c2cccc(C(=O)OC)n2)=O)CCC(NC(C2(C(F)(F)F)CC2)=O)C(O)C1 2650,c1(C(N2CCN(C(CC(C)SC)=O)C(CF)C2)=O)c[nH]c2c(F)cccc12 2651,C1(C(=O)NC2(CNC(c3ccc(C#N)[nH]3)=O)CCCC2)CCCCC1C1CC1 2652,N1(c2cc(NCC3CSCCO3)nc(C)n2)CCC(C)C(C)(C)C1 2653,C1(C(N(CCCn2cc(C(C=C)(C)O)nn2)C)=O)CCc2ccccc2C1 2654,c1(OCC(=O)N(C(C)C(=O)NC2C=CC(CC(C)C)C2)CC)ccccc1F 2655,c1(C(=O)OC)cc(NC(C2CCCCC(F)(F)C2)=O)cc(Cl)c1F 2656,C12CCCCCCN1C2.C(=O)(C(CC(F)F)c1ccccc1)NC 2657,c1(CNC(C(CC=CC)C)=O)n[nH]c2c1CN(C(C13CC=CC(C1)OC3)=O)CC2 2658,c1(CC)ccc(CC(C(=O)OC)NC(=O)COc2ncccn2)cc1 2659,C1(NC(c2n(CC(C)C)ncc2)=O)CCCC(N(C(=O)C(F)CC2CC2)C)C1 2660,C(C)(CO)(C(F)F)NC(C(C)N(C(c1ncoc1C)=O)CC)=O 2661,C(=O)(CCC(=O)NC1CCCCO1)N(CCNC(=O)CSCc1cccnc1)C 2662,CCC(C)(O)C(=O)NCC1(C)CC(NC(=O)CCc2nc(CSC)no2)C1 2663,C12C(c3ccccc3)CN1C2=O.C1(C(=O)OCC)OCCC1C 2664,c1(SC)ccsc1C(=O)N(CC(C)NC(c1ncn(C)n1)=O)C.c1ccccc1 2665,C1(NC(CC2CCC(C)CN2C(c2cnn(C)c2N)=O)=O)CCn2nnnc2C1 2666,CCCC(O)CC(=O)NCC(C)(C)CN(C(=O)C(C)NC(=O)OCC)C.C(C)(C)C 2667,N1(C(C2(CNC(C(C)C3(O)CCC3)=O)CC23CCC3)=O)CCC2(CCCCC2)C1 2668,Cc1cc2[nH]c(C(=O)NCC(C3CCOC3)NC(c3ccc(O)c(N)n3)=O)cc2o1 2669,C1(NC(C(C)OCCC#C)=O)CCCCC12CCCN(C(c1ccc(C)o1)=O)C2 2670,C(CC(C(C)(C)C)NC(=O)CC1(O)CC1)N(C)C(c1cnccn1)=O 2671,C=C(C)CCC(C)OC(c1ccc(-c2ccncc2C)s1)=O 2672,c1(C(C)=O)ncc(C(N2CCC2CNC(=O)CC(C)c2cnn(C)c2)=O)s1 2673,C(CN=c1nc2ncn(C)c2c(NC(=O)OC(C)(C)C)[nH]1)NCC(C)CCO 2674,C1(c2ccn(C)n2)CN(C(=O)CCCCN)C(C)(C)C1 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2836,C(c1cccnc1)=CC(=O)N(C1CCN(C(C2COC(=O)O2)=O)C1)CC 2837,Cc1ccc(C(=O)NCC(CO)NC(c2c(C)ccn2C)=O)c(Br)c1 2838,C1(CN(C(c2n(CC)ccc2)=O)CC)CCCCN1C(=O)Cc1cnccc1C 2839,c1(CN2CCC(CC)(NC(c3cscn3)=O)C2)ccc2nccn2c1 2840,c1(NCC2(NC(CC3ON=C(C)C3)=O)CCCCCC2)cc(C)c(F)cc1N 2841,N1(C(C(=O)OC)COC)CCC(N(c2ccccc2)C)CC1.C(=O)CN1CCC1 2842,c1(NC(NCC(C)OC(F)F)=NCc2cnn(C)c2)ccc(Cl)c(C(F)(F)F)c1 2843,c1(COC)nc(NCC2(C)C=CCCC2)cc(NCc2cc(Br)cnc2F)n1 2844,c1(C(N2CCC(N(C(c3cc(=O)cc[nH]3)=O)CC)C2)=O)c(C)ccc(F)c1N 2845,c1(C(N2C(C)CC2)=O)cnc2c(c1)N(C(CSC(F)(F)F)C(=O)O)CCO2 2846,C1(CNC(C(C)(C)OC)=O)(CO)CCN(C(=O)COCC(C)C)CC1 2847,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CC2CC23CC3)C2(CCC2)C1 2848,C1(C(=O)NC2C(NC(C3CC(C)C3)=O)CCOC2)CCC(N=[N+]=[N-])CC1 2849,CCCC(C)(CO)NC(=O)Cn1cc(C(C)Oc2scc(C)c2C)nn1 2850,c1(-c2c(CCC)csc2)cnc2cc(C(=O)Nc3cccnc3C)ccn12 2851,N(C1CCCn2nccc21)C(C(C1CCC1)NC(C(C)(C)CCC#N)=O)=O 2852,c1(CC(N2C(CNC(C3CCCS3(=O)=O)=O)CC2)=O)ccc(F)cc1 2853,C1(CNC(C=Cc2n(CC)ncc2)=O)C2CCCC1N(C(=O)CCSC)C2 2854,N1(C(c2cc(C)nn2C)=O)CCC2CCCC12C(=O)NCCN1CCCC1 2855,C1(C(=O)NCC#CC)CC2(CCC2)CN1C(c1cc(F)ccc1C)=O 2856,C1(C#N)(C(=O)NC2C(CNC(c3cnc(C)nc3C3CC3)=O)C2)CCS(=O)(=O)CC1 2857,C(C(CNC(c1cnn(-c2ccc(Cl)cc2)c1)=O)C(F)(F)F)NC(=O)C=CCF 2858,C12(C(N3CC(CC(C)NC(C4N(CC)CCCC4)=O)C3)=O)CCCC1OCC2 2859,C1(NC(C(CC)SC)=O)Cc2ccccc2N(C(=O)CCN2CCOC2=O)C1 2860,c1(OCC(=O)NC2CCN(C(c3ccc(OC)nn3)=O)C2)ccc2c(c1)CCC2 2861,Cc1cc(=NCCSC(F)F)[nH]c(=NCNC(=O)COC2CCc3ccccc32)[nH]1 2862,C(N=c1cc[nH]c(=NCC)[nH]1)c1cc(C)c(CCN2CCCC2)c(C)c1 2863,C1(C)(C(=O)NCCC2CCN(C(CCC(=C)Br)=O)C2)CC(OC)CN1C 2864,C(=O)(C1OC(=O)c2ccccc21)N(CC(C)NC(C1SC2C=CC1CC2)=O)C 2865,CCCCC(CC)C(=O)NCCCN(C)C(C1CC1C(C)(F)F)=O 2866,C1(CNC(c2cnc(C3CC3)s2)=O)CC2CCCC2N1C(=O)CN1CC2CC2C1 2867,C1(C#N)(NC(C2C(CNC(C(C)(C)OC(C)C)=O)OCC2)=O)CC1(C)C 2868,C#CC1CN(C(=O)CCN(C(=O)CN(C)C(N)=O)CCO)CC1O 2869,c1(C(=O)NC2C3CN(C(C=C(C)C(F)F)=O)C2C3)ccc(F)cc1C(F)(F)F 2870,c1(C(=O)NCC2(OCC)CN(C(=O)CCc3nccs3)C2)cc(C(C)C)nc(O)c1 2871,C(=O)(CC1=NNC(=O)C1)NCC1(O)CCN(C(CCc2cc(C)on2)=O)C1 2872,C1(C)(CNC2CCC(OCC)CC2)CCC(O)CC1 2873,CC(C)CC(C)CC(C)C(=O)O.CCCC(C)CO 2874,CC(CCCCCO)NC(=O)CCCN(C)C(C1CC(=O)OC1(C)C)=O 2875,N1(C(c2nc(C(=O)NCC=C)sc2)=O)CCC2C(C1)CN2C(=O)CCCCOC 2876,C123CC1CN(C2)CC3=O.C1(CCNC(=O)Cc2nc[nH]n2)(CC)CCCC1.C=O 2877,c1(CC(N2CC(C)C(NC(C3CC3C#N)=O)CC2)=O)ccc2c(c1)CCN2C 2878,C1(CC)CN(C(C2CC(OC)CCN2C(c2cc(C3CC3)on2)=O)=O)CCN1C 2879,C(=O)(CC(CC)CC)NC(C(=O)NC(CCCCC)C)C(C)OC 2880,Cn1c(=O)c2ccc(C(=O)NC3(c4nnnn4C)CC(CO)C3)cc2n(C)c1=O 2881,N1(C(CCc2c(C)nccc2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C(O)C1 2882,N1(C(c2cc(C)oc2)=O)CC2COCCC2(NC(c2cccc3[nH]ncc23)=O)C1 2883,C1(NC(C2(SCC)CCC2)=O)COCCN(C(c2c[nH]n(COC)c2=N)=O)C1 2884,CC1CC(C(=O)NCCCNC(=O)OC(C)(C)C)CN1C(=O)CCCCN(C)C 2885,C1(CC=C)(NC(=O)C(O)C(=C)C)CCN(C(c2cccc(OC)c2N)=O)CC1 2886,C(=O)(C1=CS(=O)CCC1)NCC(C)NC(c1cc(Br)cs1)=O 2887,CC1=C(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC3CC23)CCO1 2888,c1(C(N2CC(NC(C3CC(N(C)CC)C3)=O)C2)=O)cnn(-c2ccccc2)c1C 2889,c1(CC)[nH]c(C)nc1C(=O)N(C(C)CN(C(=O)CC1CC(=O)NC1=O)C)C 2890,C1(NC(C(=O)NCCC(C=C)C)=O)CC12CCOCC2 2891,CCC(C)CCCC(=O)NCC1(CNC(=O)C(CC)n2ccnc2)CCCCC1 2892,C1(C(N2C(C(C)NC(c3n(C=C)ncc3)=O)CCC2)=O)CCc2cnnn2C1 2893,N1(C(c2cn(CCOC)nc2)=O)CC(NC(c2cnn[nH]2)=O)C2(CCC2)C1 2894,c1(C(=O)NCCCN(C(=O)CC2CCCOC2)CC)c(C)nnn1C 2895,c1(NCCC2CN(C(C=CC(C)(C)C)=O)C2)ccc(OC2CCC23CCC3)cc1 2896,C1(C(N2CCC(COC)(N(C(=O)C=CCF)CC)CC2)=O)Cc2cccnc2C1 2897,c1(CC)ccc(C(=O)NCCOCCNC(=O)C(C)NC(N)=O)c(F)c1Cl 2898,N1(C(C(C2CN(C(C3CCCC(C)C3)=O)C2)OC)=O)CC2CCCC(C1)N2C 2899,c1(CC)nc(N2CCN(c3ccc(C(C)(F)F)cn3)C(C)C2=O)c(C#N)cc1C 2900,c1(C(=O)NCC(=C)CCNC(=O)C(F)=C2CCC2)cncc(P(C)(C)=O)c1 2901,C(C)(CO)(C(=O)NC1CCN(C(=O)CSc2ncccc2N)C1C)OC 2902,n1(CC#C)ccnc1C(=O)N(CCC)CCNC(C1CC(CC2CC2)C1)=O 2903,N1(C(C2(C#N)CCCO2)=O)CC(C2CCCN(C(=O)CCCN=[N+]=[N-])C2)C1 2904,N1(C(C(n2ncc(C)c2)C)=O)CCC(O)(CNC(=O)Cc2cn(C3CC3)cn2)C1 2905,C1(CC(=O)NCCC)CCCN(C(C23COC(CF)(C2)C3)=O)C1 2906,Cc1ncsc1C=CC(=O)NCCC1(O)CCN(C(=O)Cc2ccccc2)C1 2907,C(=O)(C1CCCCn2ncnc21)NC1C(CC)N(C(c2ccsc2)=O)CCC1 2908,C1(CN(C(c2ccc(=N)[nH]c2)=O)CC)CCN(C(=O)C(C)CF)CC1 2909,c1(CC(N(CCCC2C=NOC2)CCC)=O)c[nH]c2ncccc12.C1CCC(=O)O1 2910,c1(C(N2CCC(C)(C(N3C(C)CCCCC3)=O)C2)=O)nccc2cc[nH]c12 2911,C1(CNC(c2c(C)non2)=O)CC(F)CN1C(=O)C(C)Cc1cnn(C)c1 2912,C1(CC#C)(NC(=O)CCOC(C)(C)C)CCN(C(C2(COC)CCC2)=O)CC1 2913,c1(CCC)nc(C)c(C(=O)NC(C2CCCN2C(=O)Cc2cnc[nH]2)C)s1 2914,C1(C(=O)NCC(C)CNC(c2cc3sccc3[nH]2)=O)Cc2ccccc2C(=O)O1 2915,C(=O)(C1=CCN(C(c2ccc(F)cn2)=O)CC1)N(CC(C)(C)C#N)C 2916,c1(C(N2CCC(N(C(c3nncc(CCC)c3)=O)C)C2)=O)cc(OC)ccc1N 2917,C1(NC(CC2N(CC)C(=O)CC2)=O)CC12CCN(C(=O)C1=CCCC1)CC2 2918,n1(CC(=O)NC2CCCC(NC(c3oc(CC)c(C)c3)=O)C2)nc(O)ccc1=O 2919,C1(NC(CCC=C(C)C)=O)CCOC(C(=O)NCCc2c[nH]nc2O)C1 2920,CCC(CCC(=O)N1CCC(CN(CC(=O)OC)C=O)CC1)OC.C(C)(=O)NC 2921,N1(C(CCC#CC)=O)CCC(NC(c2ncccc2OC)=O)C(C)C1 2922,N1(CC(N2CCCC(CCOC)C2)=O)CCC2C(=O)NCC2C1 2923,c1(NC(C2(CNC(=O)COc3ccsn3)CC(=C)C2)=O)cccc2sccc12 2924,C(C(C)(O)CC(=O)NC1CCCCN(C(=O)CC2CCSCC2)C1)OC 2925,c1(C(N2CCC(NC(c3c(C(C)C)c[nH]c3)=O)C(C)C2)=O)cc2ccccn2c1 2926,C1(=O)C#CCO1.CCC(CN(CC(F)(F)F)CC)OC 2927,c1(C(=O)NC(c2nnc(C)o2)COC)ccc(Cn2ccnc2C)o1 2928,C(C(=O)O)(C1CCOC1)NC(=O)NCCSC(F)(F)F 2929,C12CCCN1C(=O)c1cn(cn1)CCn1cc2nn1.C1(COCC)CC(C)(F)C1 2930,C(=O)(CN1C(=O)COc2ccccc21)N(C)Cc1cn(Cc2ncon2)nn1 2931,c1(C(N2CC(CNC(=O)CN3CCCC3=O)C2)=O)cccc(Cl)c1 2932,C1(C(=O)NCC2C(CNC(C3CCCO3)=O)C2(F)F)CCCCCCC1 2933,C1(C(N(CCCCCNC(=O)CCc2cccc(O)c2)C)=O)CC12CCCCC2 2934,CCCS(=O)(=O)C(C)C(=O)NC1CCCC(NC(c2nccc3occc23)=O)C1 2935,C#Cc1cnc(C(=O)NCC2CCN2C(=O)Cc2cnc[nH]2)c(C)c1 2936,C1(NC(c2cn[nH]c2)=O)CC2(C1)CC(C(=O)NC1(CO)CC(F)C1)C2 2937,CC(C)C(O)C(F)(F)C(=O)N(C)CC1COCCN1C(c1ccc2c(c1)CC2)=O 2938,N1(c2ncc(C)cn2)CC2(CN(C(=O)Cn3ccnc3C)CC2CO)C1 2939,CCC(CC(=O)NCCCC1(NC(c2coc(C#N)c2)=O)CC1)SC 2940,c1(CC)noc(CNC(C)CC#CCOCCO)n1 2941,C12CCN(CC1)C2=O.C(=O)(CCCc1cccnc1)CCCN(C)CCO 2942,C1(NC(C(C)=C(C)C)=O)CC2CC(C1)CN(C(C1CCCN1CC(F)(F)F)=O)C2 2943,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)sc2sccc2c1Cl 2944,c1(C(N(CCNC(c2cc(C(N)=O)c[nH]2)=O)CC)=O)csc2c1CCC(C)C2 2945,c1(CC(=O)NCC2CCN(CC(=O)Nc3cccc(Cl)c3)C2)ccc([N+](=O)[O-])cc1 2946,C12CN(CCN1OC(C1CC3CCC3C1)=O)C2=O.c1(CC)noc(C(C)(C)C)n1 2947,c1(NCC(N2CCC(C)(C(=O)NCCc3ncc[nH]3)C2)=O)cc(O)nc(O)n1 2948,CC1(NC(=O)CN2CCCC2)CCN(C(c2sccc2C(F)F)=O)CC1 2949,c1(C(C)NCc2ncnn2CC(F)(F)F)ccc(NC2CC2)cc1 2950,C(=O)(C(C(C)(C)C)NC(N)=O)NCCCN(CCCc1cscc1Cl)CC 2951,C(c1ccc([N+](=O)[O-])cc1)=CC(N1CCN(C(C(C)O)=O)CC1C)=O 2952,C(=O)(CCC(=O)N1CC2C(N(C)C(C3CCCOC3)=O)C2C1)N(C)C 2953,c1(C(C)=O)c(C)[nH]c(C(N2CC(C)(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)=O)c1C 2954,C(=O)(C(C)(C)Cn1cc(C2(C)CN(C(=O)CC=C(Cl)Cl)C2)nn1)OCC 2955,C(CCCCC(=O)N1CC(CONC=O)C1)n1cc(COC)nn1 2956,C(CCC(=O)NC(C)CC(C)NC(c1occc1-c1cnn(C)c1)=O)OCCC 2957,c1(NC(c2ccccc2CO)=O)ccc2nc(O)oc2c1.C12(CCC1)CC(=O)N2 2958,C12(C(N(C3CCN(C(C4CCC5(CCC5)O4)=O)CC3)CC)=O)CCOC(C)(C1)C2 2959,N1(C(C(C)=C2CC2)=O)CC(NC(=O)Cn2nc(C)c(Br)c2C)CC(F)C1 2960,C1(OCC)(CNC(c2sccc2C(F)F)=O)CN(C(=O)CCCC2CCC2)C1 2961,CCCC(CCC)C(=O)N1CC(CNC(=O)C=C2CCN(C)CC2)(COC)C1 2962,N1(C(=O)CCc2ccsc2Cl)CC2CCCC(C1)N(C(c1cnco1)=O)C2 2963,c1(OC)nc(C)cc(=NC2CC23CC(NC(=O)CCc2cn(C)nc2C)C3)[nH]1 2964,C1(C(=O)OCCCC2CCCC2)CC2(COC2)C1 2965,c1(OC)cc(C(=O)NCC2CN(C(c3ccnc(F)c3N)=O)CC2C)cc(C)n1 2966,C#Cc1cncc(C(=O)NCC23CCC2CN(C(=O)C(C(C)C)NC=O)C3)c1 2967,CN1CC(C)(C(N2CC3(CCN3C(=O)CC3CSCCS3)C2)=O)CCC1=O 2968,N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCC2(C)CC2)C(C(F)F)C1 2969,N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)C=C1CN2CCC1CC2)C3 2970,C(=O)(C1CCCc2nn[nH]c21)C(C)(C)C.C1CCC(C)OC(=O)CONC(=O)O1 2971,Cc1ccc(CC(=O)NCCN(C(C2C(C)(C)C2(F)F)=O)C2CC2)cc1Cl 2972,N1(C(CCCC#C)=O)CCC2(CCC2NC(=O)CC2OCCC2(C)C)CC1 2973,c1(C(=O)O)cc2oc(C(N3CCC4C(O)CCC34)C3CC3)cc2[nH]1 2974,N1(C(C(CCSC)O)=O)CCCC(NC(C2CCN(C(N)=O)CC2)=O)CC1 2975,NS(=O)(=O)c1ccc(S(=O)(=O)N2CCCOC2)cc1 2976,N1(C(C(CC=C)C(C)C)=O)CCC(C2CN(C(c3c(SC)cccc3F)=O)C2)C1 2977,C1(C(=O)NC(=O)C(C)COC(C)C)C2CC3C(C2NC(C2(SC)CC2)=O)C13 2978,Fc1ccc2c(c1)C(c1nc(Cc3ccno3)nn1Cc1ccccc1Cl)CCO2 2979,Cc1nc(C(=O)NCCOC2CC2)cs1.C12CC1CC(=O)NC2 2980,CC1CCC1CNC(=O)CN(C(=O)C=CC1CC1)C 2981,c1(C(=O)NCC2N(C(CC3C(C)(C)CCO3)=O)CC2)cccc2nsnc12 2982,Cc1cc(C(=O)NCC23CC2CN(C(=O)C=CBr)C3)nn1-c1ccccc1 2983,Cc1nn(C)cc1CC(N1CC(CN(C)C(C2SC3C=CC2C3)=O)C1)=O 2984,c1(C(N2CC3N(C(C4(CO)COC4)=O)C3C2)=O)ccc(F)c2ccccc12 2985,Cc1ccc(NC(=O)CN)cc1.C(=O)(C(C)n1ccnn1)NC(CNC(N)=O)C1CC1 2986,c1(C(C2CC2)NC(c2n(C(C)(C)C)nnn2)c2cc(I)cs2)ccc(CO)cn1 2987,C(CCC[Si](C)(C)C)OC(C(Cc1ccccc1)SC)=O 2988,n1(C(C)C2CC2)ccc(C(=O)C2CC2)n1.C12CC1(C)CCNC(C1CC1)C2 2989,C#CCCCCC(=O)NC1CC(CCNC(C23CCCN2CCC3)=O)C1 2990,c1(C(N2C3C(CNC(C(COC)C)=O)CC(CC3)C2)=O)cccc([N+](=O)[O-])c1N 2991,c1(C(N(C(CCNC(CC=C)=O)C)C)=O)cc2cccc(O)c2[nH]1 2992,c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3C(C2)C3(F)F)=O)CC1O 2993,N1(C(C2(C)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCCCNC(N)=O)C1 2994,C12CC3CC1CN(C3)C(=O)CC1(C(C)C(=O)N2)CC1.C1(OC(C)(C)C)CCCC1 2995,Cc1ncnc(N2CCC(C)(CNC(=O)Cn3cccn3)CC2)c1Br 2996,C(C1CCCN1C(c1csc(Cl)c1)=O)=CCC(=O)NCCSC 2997,C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3c(C)noc3CC)=O)CC2C1 2998,C1(C(=O)NCC(C)O)CCCCCC1NC(=O)C=CCO 2999,c1(CC)cccnc1C(=O)NC1(C2CCCCN2C(c2snc(O)c2Cl)=O)CC1 3000,n1(CC(N2CC(CCNS(C)(=O)=O)C2)=O)cc(-c2ccn(C3CCCC3)n2)nn1 3001,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(C)C1.C123CC(CO1)(C2)C(=O)NC3.C1C(=O)N1 3002,N1(C(C(=O)NCCNC(C)=O)=O)CC=C(c2cccc(Cl)c2C)CC1 3003,C(=O)(CCCC(C)(C)OC)N1CCC(C(N2CC(C(CC)CC)C2)=O)OCC1 3004,CN=c1ncc(-c2cnc(N3CCN(Cc4ccc(OC)o4)CC3)nc2)c[nH]1 3005,C(=O)(C(C)(O)C(C)(C)C)NCC1CN(C(c2c(C)sc(O)n2)=O)C1 3006,Cc1c[nH]cc1C(=O)N(CC(=O)NCCC(C)(C)C1CC1)CC(C)C 3007,c1(COC)[nH]nc(OC)c1Cl.N12CCC(C1)N1C=C2C1.C(=O)(C=CCOC)NCC 3008,Cc1nc2c(s1)CN(C(C13CCC(CC1NC(C1CC(=O)NC(=O)C1)=O)C3)=O)C2 3009,C1(C(N(CCN(C(Cc2cc(CC)no2)=O)C)C)=O)CC12CCC(=O)CC2 3010,Cc1ccc(NC(C2C(NC(=O)CCN=[N+]=[N-])C2(C)C)=O)c(C)n1 3011,C(C(=O)NC1(C2CCCN2C(c2nccnc2N)=O)CC1)(C(C)C)SCC 3012,C(=O)(C(O)CC(C)(C)C)NCC(CNC(CC(C)(C)N(C)C)=O)O 3013,CCCCC(O)C(C)C(=O)NC(C)C=CC(=O)NCCC(C)C(F)F 3014,c1(OC)c(F)cc(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CC2C)cc1Cl 3015,N1(C(C2CCC(CNC(c3cc(COC)co3)=O)C2)=O)CC(C)(C)C12CCC2 3016,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3017,C1(C(N(C2CCCN(C(C3CCCC4CC34)=O)CC2)C)=O)CS(=O)(=O)CC(=O)N1 3018,C(=O)(CCCCC#N)NCCC1CN(C(CN(CC)CC)=O)CC1C 3019,N1(C(CC)C(C)C)CC2COCC2(C(=O)NC2CN(Cc3cccs3)C2)C1 3020,CCCC(CCCS(C)(=O)=O)C(=O)NCC1CC(NC(C2(C)COCCO2)=O)C1 3021,N1(C(C(C(CC)C)N(C(=O)CCN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3022,N1(C(c2c(C)coc2)=O)CC2CN(C(=O)C=CC(C)C)CCC2(CO)C1 3023,C1(C(N2CC(CC(C)NC(=O)C(c3ccn(C)n3)C)C2)=O)OC2CCC1CC2 3024,CC1C(C)C(C)CN1C(=O)C(=O)NCC(F)(F)F.c12ccc(c(F)c1)NC2 3025,CCC(CCC(=O)NCCN(CC(F)F)C)NC(c1cc(C)ns1)=O 3026,Cc1cc(NC(c2nnnn2C2COC2)C2CCC(C)C2)c(C)s1 3027,c1(C2C(CNC(=O)NC(C3CCOC3)COC)CC2)ncc(C)cn1 3028,CC(C)CC(F)C(=O)N(C1CCCN(C(=O)CCOCC2CCC2)C1)CC1CC1 3029,C(CC(C)C)(C(=O)NCC(=O)N(C)OCC)NC(C=CC(CC)C)=O 3030,c1(CCOC(C)=O)ccc(C(=O)NCC2C(NC(=O)CCCF)C2(C)C)cc1 3031,c1(C(=O)NCCN(C(CCCn2c(C)ncc2)=O)CC(C)O)c[nH]c(=S)cn1 3032,CCCC(C)CC(=O)N(CCCC(=O)NCCOC1CCOC1)C 3033,c1(OC)ccc(NC(C2CCN(Cc3ccnc(Cl)c3)CC2O)=O)cc1Br 3034,C(=O)(CC1OCc2ccccc21)N(CCNC(C(=O)NC)=O)CCOC 3035,Cc1nnc2n1CCN(C(=O)Nc1nn(C)cc1S(N)(=O)=O)C2C 3036,c1(C(N2C3CCC(CNC(C(CC)N(C)C)=O)(C3)C2)=O)cccc2ccn(C)c12 3037,CC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1NC(=O)Cn1ccnn1 3038,N1(C(c2c(CNC(CC(=O)OC)=O)cnn2C)=O)CC(C)CCCC1C 3039,C1(C(N(CCC)CCNC(c2cc(Cl)c[nH]2)=O)=O)(CCOC)CCCC1 3040,C(C(CC(C)C)C(=O)N(CCC(C)C)C)NC(c1onc(C)n1)=O 3041,c1(C(=O)NCC(CC=C)NC(=O)Cn2ccnn2)cn2cccc(C)c2n1 3042,C12(NC(c3cncc(-n4cnnn4)c3)=O)CC1CN(C(C1CCC13CCC3)=O)C2 3043,N1(C(C2(CC)CC2)=O)CC2(CNC(C3CC(C(F)(F)F)C3)=O)CC(F)(C1)C2 3044,CN1C(=O)Cc2cc(NC(C3CCN3Cc3c(Cl)ccc(F)c3F)=O)ccc21 3045,S(=O)(=O)(c1ccc(N2CCS(=O)C(C)C2)c(F)c1)N1Cc2c(ccc(OC)c2)C1 3046,C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(CNC(C(C)(C2CC2)OC)=O)CCC1 3047,N1(C(C=C(COC)C)=O)CCC(CN(C)C(C2CC2(F)F)=O)C1 3048,c1(OC)ccccc1C=CC(=O)NC1CCCC1NC(=O)Cc1c(C)noc1C 3049,C1(NC(C2(C)CN(C(=O)CC3(O)CCOCC3)C2)=O)CC2(CNC(=O)O2)C1 3050,CC1CCN(C(c2cc(Cl)c[nH]2)=O)C(C(=O)NCCCc2ncc[nH]2)C1 3051,Cc1cc(CC(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(O)n1 3052,C1(CNC(C(C=CCCC)O)=O)CN(C(=O)C(C)(C)CF)CCO1 3053,C(C(O)CN(C)C(C1CCN1C1CCCC1)=O)N(C)C(C1(O)CC1)=O 3054,C(N=c1[nH]nc(-c2ccon2)s1)C1CC(NC(c2cc(N3CCCC3)ccn2)=O)C1 3055,c1(C(=O)NC(C(C(C)C)NC(=O)CC(C)(C)C)C)nc2ccccn2c1F 3056,Cc1nn(CC(=O)NCCN(C2CCCCCC2)C(=O)C(O)C2CC2)cc1[N+](=O)[O-] 3057,N1(C(Cn2ccc(C)n2)=O)CCC(F)C(NC(c2cc(C)nn2CC(F)F)=O)C1 3058,CC1CCN(C(c2cncnc2)=O)CC1NC(=O)C(C1CCCCCC1)=O 3059,N1(C(CCCCCOCC)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)CC12 3060,C(=O)(C(C)(C)CN(C)C(C1COCC(C)O1)=O)N(CC(CC)OC)C 3061,c1(N2CCCCC(OC)C2)ncnc2scc(Br)c12 3062,c1(C(=O)NCC(CNC(=O)C=CCO)O)cc(Cl)cc2c1CCC2 3063,Cc1cccc(OCC(=O)NCCC2(NC(=O)CCS(C)=O)CC2)c1C 3064,c1(N2CC3N(Cc4c(C)cccc4Br)C3C2)ncnc2[nH]c(C)nc12 3065,C1(CNC(Cc2n(C(C)C)ncc2)=O)CN(C(C2C3CCC(=O)C23)=O)CCCO1 3066,c1(C(=O)NC(CNC(CCCCC)=O)CCCC)cc(C2CC2)ccc1F 3067,C(C(CC(C)C)C(=O)NCC1CN(C(c2ccc(Cl)c(F)c2)=O)CC1C)OC 3068,C1(CN(C)C(C2CCCCS2)=O)CCN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1 3069,c1(C(=O)NC2CC(N(C(C=CSC)=O)C)C2)ccc(NC(=O)N(C)C)cc1 3070,N1(C(CCOC)=O)CCCC1CCNC(C1CCNC1=O)=O 3071,C1(C(N2CC(O)(CNC(c3scc(C(C)(C)C)n3)=O)C2)=O)CCCC12CCC2 3072,N1(C(CC2C(C)(C)C2)=O)CCCCC1CCNC(=O)CCC1(O)CCCC1 3073,c1(OCCC(=O)N(CC(CC)NC(=O)C=C2CC2)CC#C)ccc(Cl)c(Cl)c1 3074,CC1CC(C)(C(N2CCCC(O)(CCNC(=O)C3=CCC3)C2)=O)CC(C)O1 3075,c1(CN(C(c2ccc(OCCCC)cc2)C(=O)NCC)C)c(C)cc(C)cc1C 3076,c1(CC(N2C(CNC(C3(N(C)C)CCC3)=O)C=CC2)=O)ccc(Cl)c(Cl)c1 3077,c1(OC)nc(C)cnc1NC(C1CC(CNCc2n[nH]cc2Cl)C1)=O 3078,c1(NC(=O)NC(C(=O)N2C(C)CC2)CCc2ccncc2)cc(N)nc(Cl)c1 3079,C(=O)(CCCNC(N)=O)NC(CN(C)NC(C1CC1(C)C)=O)(C)C 3080,c1(C(N(C)C(C2CC3CCC2C3)c2ccccc2)=O)cccnc1-c1nncn1C 3081,N1(C(C2C(C)CC(C)O2)=O)CCC(C2CC2)C1CNC(=O)C=CBr 3082,c1(NC(C(=O)Nc2ccc(C)c(N3CCCC3)c2)=O)ccnc2c1c(C)nn2C 3083,C(=O)(C(C(C)CC)N(C(=O)Cn1cccn1)C)NC(CCC)(C)CC 3084,c1(C(=O)NCC(CO)NC(=O)COCCCF)cnc(-c2cccs2)nc1 3085,Cc1ccnc(O)c1C(=O)NCC(C)NC(c1cn(C)c(-c2ccccn2)n1)=O 3086,c1(C(=O)NC(C(=O)OC(C)C)C)ccc(CNC(c2nonc2N)=O)cc1 3087,C1(C(N2CC(N(C)C(c3ncn(C)n3)=O)C2)=O)CCCC2CC12 3088,N1(C(c2ncn(C(C)C)n2)=O)CCC2CC2(NC(=O)CC=C(Cl)Cl)CC1 3089,C1(CC(=O)NCCC2CCN(C)C2)CCNC1(C)C 3090,c1(N2C(CNC(C3N(C(C)C)CCC3)=O)C(C)CC2)nc(Cl)ncc1C(F)(F)F 3091,N1(C(C2(CC#C)CC2)=O)CC2CC(C1)C2NC(=O)CNC(=O)OCC 3092,C1(C(C)NC(c2ccccc2C2CC2)=O)C(C)CCCN1C(=O)CC1CSC1 3093,c1(C(=O)NC2CCCC(CNC(c3[nH]cc(CC)c3)=O)C2)ccc2c(c1)CCCS2 3094,N1(C(CNS(CC)(=O)=O)=O)CCCC2(C1)C(NC(=O)CO)CCN2C 3095,C1(NC(C23C(CN(C(c4c(OC)cccc4)=O)C2)C3)=O)CCC(C)(C)OC1 3096,c1(C(=O)NC23C(CN(C(CCCC(=C)C)=O)C2)C3)ccc2cnnn2c1 3097,n1(CCCC(=O)NC)c(C(C2CC(F)(F)C2)N)nc2ccccc2c1=O 3098,C1(NC(CC2(C=C)CCC2)=O)CCN(C(=O)CC2CC(=O)C2)C(C)C1 3099,N#Cc1cnc2c(Cl)cccc2c1NC(C1CC1NCc1ccc(Br)cc1Cl)=O 3100,N1(C(C=C(C)CNC(=O)Cc2scnc2C)=O)CCCC1C(C)O 3101,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3102,C1(N(C)C(C2CC2C2CCC2)=O)COC2(CCN(C(=O)C(C)(C)Cl)CC2)C1 3103,CCC(C)(C)C(C)CC(=O)NC1CN(CCNC(c2ncc3[nH]ncc3n2)=O)C1 3104,CCCC(C)C(=O)N1CCCC1CN(C(=O)Cn1cccc1)CC 3105,c1(OC)cc(C(=O)NC2CN(C(c3ccccc3C#N)=O)CC2C)ccc1Cl 3106,C1(NC(C2CC(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)CNC(=O)N(C)C 3107,c1(C(=O)NC(CC(C)NC(c2ccnn2C)=O)C)ccc(-c2cnnn2C)cc1 3108,N1(C(c2c(SC)n(C)nc2)=O)CC2COCC2(C(=O)N(C)Cc2ccco2)C1 3109,C1(NC(C(C)C2(O)CCC2)=O)COCCC1NC(=O)C(C1CCOCC1)F 3110,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3111,C12CCC(O)CN1C2=O.c1(SCCCN2CCCC2)cccc(Cl)c1 3112,C1(C(N(C)CC2CC(=C)C2)=O)CCN(C(C2CCCCCN2C)=O)C(C)(C)C1 3113,C(=O)(C(=O)CC(C)C)N(CCCC(N1CCCC(CCC)C1)=O)CCO 3114,C(=O)(C(C)CC(C)CC(C)C)N(CCNC(CNC(CCC(C)C)=O)=O)C1CC1 3115,c1(-n2cc(C(CC)NC3(C(=O)OC)CC(F)C3)nn2)ccc2c(c1)NC(=O)CO2 3116,C1(CNC(C2(COC)CCCC2)=O)CCCCN1C(C)=O.C12(CC1)C(=O)NC2 3117,C1(CC)CN(C(=O)CC(CC)OC)CC1C(=O)NC1(c2ccccc2)CCC1 3118,C1(C(=O)NC2CCN(C(CCCSC)=O)C2C)CC12CCC(F)(F)CC2 3119,C(=O)(CCP(C)(C)=O)NCCC(C(=O)NC1CCCC(C(N)=O)C1)OC 3120,Cc1ncc(NC(=O)C(CC2CC2)NC(=O)C(C2(O)CCCC2)F)c(C)c1C 3121,c1(C(=O)NCC(N(C(C2(CCOC)CC2)=O)C)C2CC2)c[nH]nc1F 3122,c1(CC)cc(C(=O)NC2CCN(C(=O)C(C)(C)n3cc(Cl)cn3)C2)ccn1 3123,C(=O)(C(F)C(C)CNC(=O)C(C)(C)CF)NCc1c(OC)cccc1 3124,C12(C(=O)NCc3cnc(C)s3)CC1CN(C(C1CCO1)=O)C2 3125,N1(C(C(C)=C2CC2)=O)CCC2CC(NC(c3ccco3)=O)CCC2C1 3126,c1(CC(=O)NCC2(CNC(CNC=O)=O)CC2)cncs1 3127,Cc1nc2cc(NC(=O)Nc3ccccc3C#N)ccc2o1 3128,C(CNC(=O)C(F)(F)C(F)F)(CC(F)(F)F)NC(C1CN(S(CC)(=O)=O)C1)=O 3129,C1(OC(=O)OC)CCN(C(=N)NCCNC2(c3ccc(Cl)cc3)CCC2)C1 3130,N1(C(CCc2ccc(OCCC)cc2)=O)CCc2ccccc2C1CC(=O)OC 3131,C1(C(N2C(C)C(NC(C3CCCC34CC4)=O)CC2)=O)CC2(CC(=O)C2)C1 3132,C1(CNC(c2ccn(C(C)C)n2)=O)CCCN(C(C2(C)CC2(C)C)=O)C1 3133,C1(c2n(CC)nc(Cn3cccn3)n2)CCn2c(C)cnc2C1 3134,C(=O)(CCCCCc1cn(C(C)(C)C(=O)O)nn1)N(c1cc(C)nn1C)C1CC1 3135,Cc1ccc(C(=O)NC(C)Cn2cc(-c3cncs3)nn2)cc1[N+](=O)[O-] 3136,N1(C(CN(C2CCC2)C)=O)CC(NC(C2C=CC=CC=C2)=O)C(c2cnn(C)c2)C1 3137,C1(C#N)(C(=O)NC)CCN(C(=O)C(N)CC2CCC(=O)NC2)CC1 3138,C1(NC(C(CC=CC)C)=O)CC2CCC1C(NC(=O)CNC(N)=O)C2 3139,CCCC(C(=O)N1CC(C)(NC(c2nccn3ccnc23)=O)C1)C(C)C 3140,CC1(NC(c2cnc(Br)s2)=O)CCN(C(C2(O)CCC2)=O)C1 3141,CC(C)(C#N)CCCC(=O)NCc1csc(CNC(C2CC23CCSCC3)=O)n1 3142,c1(CCC)cc(C(N2CC(F)CC2CNC(=O)C(C)O)=O)sc1C 3143,c1(OC)ccc(Br)cc1C(c1nnnn1C)NC(=O)C(C(C)(C)C)SC 3144,c1(C2(CC(=O)NC(C)CC(C)O)CC2)ccccc1C(F)(F)F 3145,C1(CNC(C(C(C)C)(C)C)=O)CC2(CCN(C(c3ccns3)=O)CC2)C1 3146,c1(N(C(=O)C(C)C2CCC2)CCCN)cc(C(F)(F)F)cc(O)c1.CC 3147,c1(C(=O)NC(CC(N)=O)C(F)(F)F)nc(Br)n2c1CNCC2 3148,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3149,N1(C(=O)NCc2csc(-c3ccc(Br)cc3)n2)CCN2CC(O)CC2C1 3150,C12CCC(CC1)C(=O)NC2=O.C(=O)(CCc1ncc[nH]1)N(C(C)CC(N)=O)C 3151,C(=O)(C(C)(C)C(C)C)N(CC(N1CCC(CSCC)C1)=O)CC#C 3152,C1(NC(CC(C)N(C)C)=O)CC(C(=O)NC(CO)CCC2CC2)C1(C)C 3153,c1(OC)ccc(Br)c(C(=O)NCC(C)NC(C2CC3(C2)CC(O)C3)=O)c1 3154,C(=O)(C1=NN(C2CC2)C(=O)CC1)Nc1c(F)ccc(Oc2ccc(OC)cc2)c1 3155,C(=O)(CCCCCF)NCCN(CCOC)C(C1CC1C1CCCC1)=O 3156,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(N1CC=CC1CF)=O 3157,CC(CNC(c1csc(O)n1)=O)C(F)C(=O)NCC1(C)CCOC1 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3194,CCCCCCCCC(=O)NCC(C(C)C)NC(=O)CC(C)(C)C1CC1 3195,C(=O)(C(C)(C)C(=O)OC)NCC(=O)NCCOCC(N1CCN(CCCC)CC1)=O 3196,N1(C(c2cscn2)=O)CCC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3197,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3(CSC3)C2)=O)CC1 3198,C1(OC)CN(C(c2ccc(CO)cn2)=O)C(C)(CNC(c2c[nH]c(C#N)c2)=O)C1 3199,Cc1cc(C(N2CCC(CF)(NC(C3CCC3c3nc[nH]n3)=O)C2)=O)c(C)s1 3200,Cc1nc2ccc(C(N3CC(NC(C4SCCCS4)=O)C(C)(C)C3)=O)cc2s1 3201,C1(C(=O)NCCCCCN(C(COCC(C)C)=O)C)CC(S(C)(=O)=O)C1 3202,c1(C(=O)NC(C2CCCN2C(C2CCC(C(F)(F)F)O2)=O)(C)C)cncc(F)c1 3203,C1(C(C(=O)NC2CCN(Cc3cccc(Cl)c3F)CC2)O)CCCCCCC1 3204,Cc1cc(C(=O)NCC(C2CCOC2)NC(c2nccnc2N)=O)cnn1 3205,c1(C(N2C(CC)(CC)CC(NC(=O)C3=CCCCO3)C2)=O)cn2cnnc2cn1 3206,C(=O)(C(C)COC)NCCNC(=O)OCC.C(=O)(CCC1CC1)N.C1COCC1 3207,C1(C2N(C(Cc3cc(C)on3)=O)CCC2)CCN(C(c2ccc(Cl)cc2)=O)CC1 3208,C1(N(C(C(C=C=C)C)=O)C)CCC2CN(C(C34CCC(OC)C3C4)=O)CC12 3209,C1(C(N2CC3C(NC(C4N(C(C)=O)CC(O)C4)=O)C3C2)=O)CC2(C1)CC1(CC1)C2 3210,c1(NC(CC(CC)NC(C(CCC)=CCC)=O)=O)c(C)[nH]c(C)cc1=O 3211,c1(C(=O)NCC2(C)N(C(C=CC(CC)=CC)=O)CCC2)ccc2[nH]c(C)c(C)c2c1 3212,C(=O)(NNC(=O)CCc1cccc(Cl)c1)c1ccc(C)cc1 3213,c1(CC)cc(C(=O)NCC2CCCN(C(=O)C(F)CC)C2)nn1-c1ccccc1 3214,c1(-c2cn(SC3(CC(N4CC(C)SCC4)=O)CC3)nn2)cc(F)cc(F)c1F 3215,c1(C(=O)NC(CC)CN(C(=O)C(O)c2ccco2)CC)ccnc(C(F)(F)F)c1F 3216,CCCCCCN(C(c1cc(-c2ccccc2)no1)C(=O)NCC1CC1)C 3217,N1(C(CC=C)=O)CCCC(C)(CNC(=O)CSCC)C1 3218,N1(C(c2c(C)[nH]cc2)=O)CCOC2CCN(C(=O)CC(O)C3CCCC3)CC12 3219,N#Cc1ccc(C(=O)NC2CC(n3cc(NC(=O)C4=CCCS4)nn3)C2)o1 3220,c1(C(N(CC(CNC(CCC(=C)Br)=O)O)C)=O)c(C)cccc1Cl 3221,N1(C(c2ccc(Br)cc2Br)=O)CC2CCN(Cc3cccc(F)c3O)C2C1 3222,C=CCC(C)C(=O)NC(C)Cc1cn(-c2cccc(CC(=O)OCC)c2)nn1 3223,c1(C(=O)NCC2(O)CCN(C(=O)CCc3cn[nH]c3)CC2)ccc(=O)n2c1CCC2 3224,CCC(C(=O)OCC)C(=O)N1CCC(C(=O)NCC2(O)CN(C)C2)C1 3225,CCCC(C(=O)NCC(Cn1cc(-c2ccc(=O)n(CC)c2)nn1)OC)C(C)C 3226,C(N=c1[nH]c(Cl)ncc1C1CC1)C1CN(Cc2cccc(C(C)C)n2)CC1C 3227,c1(C(N2CCC(O)(C(N)=O)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Cl)c1Cl 3228,c1(C(=O)NC(C(C)NC(C(C)OC)=O)C)ccccc1Oc1ccncc1 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3265,c1(CC(=O)NCC2(O)CN(C3CCCC3CCC3CC3)C2)c(F)cccc1Cl 3266,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3267,C(=O)(C1=NOC2(CCN(C(=O)Cc3ccc(C)o3)CC2)C1)Nc1scc(C)n1 3268,c1(C(N2CC(C(C)NC(c3c(C)onc3)=O)C2)=O)cn2c(n1)CCC2 3269,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)CC3C)=O)ccc2O1 3270,N1(C(C2(C#C)CCOCC2)=O)CCC2CN(C(c3cnsc3)=O)CCC2C1 3271,CC1COC(C(=O)NCC2CC2C(=O)N(C)C(C)C2CC2)C1 3272,c1(CC(C)C)c[nH]c(C(=O)NC2CC(NC(=O)CCc3nnc(C4CC4)o3)C2)c1 3273,C1(OC)COCCC1CC(=O)NCCCCN1CCC(OCCn2cccn2)CC1 3274,c1(-c2nc(C3(C(CN(C)CCC(C)(C)C)(C)O)CC3)on2)c(C#N)ccc(Cl)c1F 3275,C1(CN2CC(c3c(OC)ccc(Cl)c3)OCC2)Cc2ccccc2C1C 3276,Cc1[nH]c(C#N)cc1C(=O)NC(CNC(=O)C(C)c1cc[nH]n1)CO 3277,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3278,C1(NC(C(c2c(C)cccc2)(C)C)=O)CC2CCC1C(NC(=O)C(F)F)C2 3279,N1(C(C2(C)CC3C=CC2C3)=O)CC2(CC(NC(c3cc(C(F)F)no3)=O)CO2)C1 3280,C1(CC=C)(C(=O)NCC[Si](C)(C)C)CN(C(=O)C(O)c2ccco2)C1 3281,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3282,C1(CC(=O)NCCC2CC(C(=O)NCc3c(C)noc3)C2)C(C)(C)C1(C)C 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3336,C1(NC(C=C(CC)CC)=O)CN(C(C2CCCC=CC2)=O)C2CC12 3337,C1(Nc2nnn(C)n2)CCN(C(=O)CCCc2cccc(Cl)c2)CC1(C)C 3338,C1(CCCC)CCC(C(=O)NCC(O)CSC)CC1 3339,c1(C(N2CCN(C(C=C(C)C)=O)CC2c2ccncc2)=O)ccc2c(c1)CCC2 3340,N#Cc1c(C(N2CC3(CCN(Cc4ccc(F)nc4)C3)C2)=O)cccc1F 3341,C1(CC)CN(C(c2cccc(CO)c2C)=O)CCN1Cc1ccc(Cl)nc1OC 3342,c1(OC)cc(CN(C)C(C2(C3CCCN3C(=O)Cc3cscc3Cl)CC2)=O)on1 3343,Cc1oc2ccccc2c1C(=O)NCC1CCCC1NC(c1cc(O)nn1C)=O 3344,N1(C(c2ccc(CNC(C3CCCN3C3CC3)=O)o2)=O)C2COCC1C2 3345,c1(C(N2CCC(C)(CNC(C3C(C)C3(F)F)=O)C2)=O)n[nH]c2cccnc12 3346,N1(CC(C2CC2)OC)CCC(=O)N(CC(c2nccs2)C)C1=O 3347,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)N(C)Cc1ccccn1 3348,CC(N=c1[nH]c(N(CCCNc2ccncc2)C)nc2c1CCC2)c1ccsc1 3349,c1(-n2cc(C3(F)CCN(C(C4CN(CC)C(=O)C4)=O)C3)nn2)ccc(F)c(N)c1 3350,c1(OC)cc(O)ncc1C(=O)NCCC1(O)CN(C(c2ccc(N)c(N)n2)=O)C1 3351,c1(NC(C2CN(C(c3occc3C3CC3)=O)C2)=O)cc(C(F)F)cc(F)c1 3352,N1(C(=O)NC(C2CC2(Br)Br)C)CC2(C(=O)NCc3ccccc3)CC1(C)C2 3353,c1(C(N)=O)cccc(OCC(N2CCN(C(C3CC=CCC3)=O)CC2)=O)c1 3354,C1(C(=O)NCC(CNC(C2C(C(C)C)CCO2)=O)CO)CCC(F)(F)CC1 3355,c1(C(=O)NC2CN(C(c3ncnc(C)c3C)=O)CC2C)cc2scc(C)c2[nH]1 3356,N1(Cc2ncnc(OC)c2C(C)=O)CCCC(C)(C)C1CNC(=O)CCCC(C)C 3357,c1(CC=O)ccnc(NCC23COC(CNC(=O)C(O)c4ccsc4)(C2)C3)c1 3358,C=C1CC2(C1)CC(C(=O)NC(CCNC(C13C(=O)C4CC1C3C4)=O)C(C)C)C2 3359,C1(CNC(C2(CC)CC2)=O)CC2COCC2N1c1ccncn1 3360,CC1CCCN1CC(=O)NCCC1CC1.C(=O)(COCCO)NCCO 3361,C1(O)(CNC(CCc2nc(C)c(C)o2)=O)CC2CCC(C1)N2C(=O)C=CBr 3362,CC1CC(CNC(c2csc(CO)n2)=O)CCN1C(=O)CCCc1ccccn1 3363,N1(C(C(C)Cn2cccn2)=O)CCC(C)(C)C(C(=O)NCC2CCC3(CC3)C2)C1 3364,C1(C(=O)NCCC2CC(NC(c3noc(CC)c3C)=O)C2)CCc2n[nH]cc2C1 3365,N#Cc1c[nH]c(C(N2CC3C(CNC(=O)CCCc4ccncc4)C3C2)=O)c1 3366,CC(C(=O)N1CC(CNC(=O)CSS(C)(=O)=O)C1)C1(O)CCC1 3367,N1(C(c2ccncn2)=O)CC2OCCN(C(c3cnncc3O)=O)C2C1 3368,c1(C(=O)NCC(CC2CC2)OC)cccc(C#N)n1.C1(=O)C(C(C)OC(C)C)N1 3369,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)N(C1(C)CC1)C)C2 3370,C=CC(CC)CC(=O)NC(C1CN(C(c2nnc(CC)s2)=O)CCO1)C 3371,CCCC(C(=O)NC(C(=O)NC1CC1(C)C)C(C)OC)N(C)C 3372,N1(C(C(c2nc(C)sc2)=O)=O)CC(NC(c2ccc(C(C)C)nc2)=O)C(C)(C)C1 3373,N12CCC(CC1)Cn1cc(nn1)C2.N1(CCOCCCC)CCCC1CSC 3374,CN1CC=C(C(=O)NCC2CC2CNC(C23CCCN2CCC3)=O)C1 3375,c1(CN2CC(C(F)(F)F)(C3CC3)C2)cnn2c1OCC2 3376,C(c1cccc(Cl)c1)=C(C(N1C(CNC(C(C)(C)OC(C)=O)=O)CC1)=O)C 3377,CCCCC(=O)NC(Cc1cc[nH]n1)C(=O)NCCCCSC 3378,C1(NC(=O)CO)CCN(C(=O)CCc2cnn[nH]2)CCC1(F)F 3379,N1(C(c2c(CC)cccc2)=O)CCC(N=[N+]=[N-])(C(=O)NC2(C)CCOCC2)C1 3380,N1(C(C(C)C)=O)CCN(C(=O)CCc2nnc(C3CC3)o2)CC1C 3381,c1(C(=O)NC2C(CNC(C3=CC(C)CC3)=O)COC2)ccc([N+](=O)[O-])cn1 3382,c1(C(N2C(CN(C)Cc3c(C)cco3)CCCC2)=O)cnc2c(c1)CCCC2 3383,CC1CC2(C(=O)NC(c3ccn(CCNC4CN(CCF)C4)c3)=O)CC12 3384,CC1CCCN(C(C2CCS2(=O)=O)=O)C1CNC(=O)CCN1CCOC1=O 3385,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3386,C1(CNC(CCSC(C)C)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3387,C(=O)(C1=CC2CCCCCCC12)N(C)CCN(c1ncc(C(N)=O)cc1Cl)C 3388,c1(C(N2CC(OCC)(CNC(=O)Cc3cc(C)no3)C2)=O)cn(C)nc1C(F)F 3389,N1(C(c2cc(CNC(C3(C)CC(=C)C3)=O)on2)=O)CCC(CO)C(O)C1 3390,C=CCCC(C)(C)C(=O)NCCC(C)(C)NC(C1CCCC(C(F)(F)F)C1)=O 3391,N1(C(COC2(C)CN(C(=O)CN3CCCCC3=O)C2)=O)CCc2ccncc2C1 3392,CC1CCC(NC(c2ncoc2C(C)(C)C)=O)CN1C(c1cccc(Cl)c1N)=O 3393,C=C(C)C(CC(=O)NCC1N(C(=O)C=Cc2ccccn2)CCC1)OCC(C)(C)C 3394,C1(CC(=O)NCCn2cc(CNC(C3(C)CC3(C)C)=O)nn2)(CC)CCOCC1 3395,c1(NC(C(c2ncc(C)o2)NCC(c2ccccc2F)F)=O)c(C)cc(C)cc1C 3396,c1(N(CCC(C)O)C)nc(N2CCOC(C)(CCO)C2)nc2c1CSC2 3397,C(=O)(C1=CC2CCCC12)N(C1CCC(NC(c2ccc3nc[nH]c3n2)=O)CC1)C 3398,C(=O)(CCCCC(=O)OC(C)(C)C)N1CCN(C(CCCON)=O)CC1C=C(C)C 3399,CCC(F)(F)C(=O)NC1CCN(CCNC(C2CC(F)(F)CS2)=O)CC1 3400,CC1(C(=O)NCC2(O)CCC2)CCCN1C(c1ccc(Cl)s1)=O 3401,C1(NC(C(CC#C)C)=O)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)CC12CC2 3402,C1(N(C(CN(CCOC)C(C2CCS2(=O)=O)=O)=O)C)COC(C)(C)C1 3403,c1(NC(C(=O)N(C2CCN(CC)C2)C)=O)cc(F)ccc1NC1CCNCC1 3404,N1(C(C(C)C(F)F)=O)CC(CN(C2CCC2)C(=O)C2CC2)C2(CC2)C1 3405,N1(C(C(=O)NCC(C)CNC(C2(CS(N)(=O)=O)COC2)=O)C)Cc2ccccc2C1 3406,C1(C(=O)N)C2CCCC(=O)C12.C12CCCCN1CC1(CC1)N(C)C2=O.CO 3407,Cc1ncc(C(=O)NCC2CN(C(c3ccns3)=O)CC23CC3)c(C)n1 3408,CCCC(CNC(=O)CCc1cccn1C)C(=O)NCC1CCN(CC)C1 3409,c1(COC)nnc(OC)c(OC)c1OCN1C(C(=O)NCC)CSC1 3410,C12CCN(CC1)C(=O)c1cnn2n1.c1(OC(C(=O)OC)C)cnn(C(C)C)c1 3411,Cc1cc(=O)ccn1CC(=O)NCC1CCN1C(c1coc(C2CCC2)n1)=O 3412,C12(CNC(=O)COC3CCOC3)CC(CO1)N(C(C1CCC3(CCC3)O1)=O)C2 3413,c1(NC)nc(C)ccc1C(N1CCCN(C(C2CC(OC)C2)=O)CC1)=O 3414,Cc1cc(S(=O)(=O)NCCC(=O)NC2CCCCN(C(=O)CC(C)(F)F)C2)cn1C 3415,C=CCC(CC)C(=O)N1CCOC(C)(CNC(c2cc(C(=O)OC)cs2)=O)C1 3416,C1(N(C)C)C2CN(C(C3CCC(NC(C4CC5(CCC5)C4)=O)CC3)=O)CC12 3417,N1(C(c2nc(Cl)cs2)=O)CCC(N(C(C2(O)CCC2)=O)CC2CCCCO2)CC1 3418,c1(CNC2(n3cc(CC(=C)CCCC=C)nn3)CCOC2)c(Cl)cc(Br)cc1Cl 3419,OC1(NCc2ccn(CC3CC3)n2)CCCC1 3420,c1(OC)ccc(O)cc1C(N1CC2CC1CC2NC(c1ncc(C)cc1C)=O)=O 3421,N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)COCC2CCCOC2)C(CO)C1 3422,C(=O)(C1=CCN(C)C1)NCC(C)C(=O)N1CCCC1CC1CCC1 3423,Cc1ncc(NC(C2CCCCN(C(=O)Cc3cccnc3F)C2)=O)cc1C#N 3424,Cc1cccc2c1OCCC2NC1CCCCC1CN1CCC(C)CC1 3425,N1(C(C(C)(C)NC(N)=O)=O)CC2(C=C(C(=O)NC(C)CC3CC3)CO2)C1 3426,C(CCNC(=O)Cc1cccnc1O)(C(=O)N(C(C(CO)OC)C)C)OC 3427,Cc1c(F)cc(C(C)NC(=O)NCCNc2c(F)c(F)c(C)c(F)c2F)cc1F 3428,c1(CCC(=O)NCCNC(C(C)(C)c2cccnc2)=O)ccc2c(c1)OCCO2 3429,C(CO)(CCCCNC(C1CC(C(F)F)C1)=O)NC(c1cscc1Cl)=O 3430,CCCCCCCC(=O)N1CCCC(CNC(c2cccc(Cl)c2F)=O)C1 3431,C1(C(=O)NCCCN(C(=O)CCn2cnccc2=O)C)CN2CCN1CC2 3432,C1(C(N(CC=CC(=O)NCC(COCC)O)C)=O)CCC(C)O1 3433,C1(NC(C2N(C(COCCC#C)=O)CCC2)=O)CC2C(C1)C2(F)F 3434,c1(C(=O)NC(C)(C)CCCNC(=O)C=CC(=O)N2CCCC2)ccc2cc[nH]c2c1 3435,c1(C(N2CC(O)(CCNC(C3=NNC(=O)C3)=O)C2)=O)cc(=O)n2nccc2[nH]1 3436,c1(C(=O)NC(C(C)(C)NC(C=CC)=O)C)cc2[nH]nc(C)c2cn1 3437,N1(C(C=CC)=O)CCN(C(C2CCCN(C)C2)=O)C(C2CCCC2)C1 3438,CCCC(C(=O)NCC1(C)CCCN1C(=O)CC1CSCCS1)NC(N)=O 3439,C1(NC(C(C(C)NC(=O)CC(C)=C(C)C)C)=O)CCC2(CCC2)CC1 3440,c1(COC)ccc(C(N2CCC(CNC(=O)C(F)=CC3CC3)(OC)C2)=O)cc1 3441,CC1(CNC(C2C3(CC3)C23CC3)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1 3442,C=CCCCC(C(=O)N1CCC1CCC)NC(=O)C(=O)C(C)CC 3443,Cc1nn(C)c2c(N3CCc4nocc4C3)nc(=NCc3cnn(C)c3)[nH]c12 3444,C(CNC(=O)CC1CCN(CCF)CC1)(C(C)C(C)C)NC(c1cc(C)[nH]n1)=O 3445,C1(NC(C(CC#C)O)=O)CN(C(=O)C=C2CCC2)CCC1(C)C 3446,C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCN1C(c1cc(OC)ccn1)=O 3447,c1(OCC(=O)NC2(CNC(c3n(C)ccn3)=O)CC2)cccc(F)c1F 3448,N1(C(C23N(C(C4C(C)CC4)=O)CC(C)(C2)C3)=O)CC(C)C12CCOCC2 3449,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCN(C(=O)COC3(C)CCC3)C2)C1 3450,C1(CN(C(C(C)(C)OC)=O)C)CCCCN1C(=O)CCCc1ccccc1 3451,c12c(cc([N+](=O)[O-])cc1Cl)CN2c1ccccc1C(C)C.C(C(F)(F)F)S.CCO 3452,Cc1cc(C(N2CC(C(=O)O)C3(C2)CN(C(=O)C(O)CF)C3)=O)c(C)cc1Cl 3453,N1(CC#CC)CCN(C(=O)C(CC2CC2)N(C(C2CNC(=O)C2)=O)C2CC2)CC1 3454,CN1CCCC(C)(C(=O)N(CC(O)CNC(=O)CC2OCCC2(C)C)C)C1 3455,N1(C(CNC(=O)OCC=C)=O)CC(O)CC1C(=O)NCC=C1CCC1.C 3456,c1(OCC(=O)NC2(F)CC(NC(COCC)=O)C2)cccc(CCC(C)OC)c1 3457,c1(OCC(N2C(CNC(=O)COc3cccnc3)CC2)=O)cnc(O)nc1O 3458,N1(C(=O)OC(C)(C)C)Cc2ccc(COC)nc2C1.C1(=O)CC(C2CCC2)N1 3459,CC1CN(C(=O)CC2(CO)CCC2)CC1C(N1CCC(N2CCCC2)C1)=O 3460,CC1CN(C(c2ccc(F)cc2Cl)=O)CCCN1C(c1ccc(C2CC2)nc1)=O 3461,N1(C(=O)Cc2ccco2)CCOC(CC(N2CCCOCC2)=O)C1 3462,c1(C(=O)NC(CCOC)CNC(=O)C(C)CSC)cnc(C#N)s1 3463,N1(C(Cc2c(C)cccc2)=O)CC2(CCN(C(C3(C)CC=CCC3)=O)CC2)C1 3464,C1(C(=O)Nc2cn[nH]c2)(NC(c2ccc(C(F)F)o2)=O)CCSC1 3465,S(=O)(=O)(c1ccsc1C(=O)NCCCCC(C)NC(=O)C(F)(F)CO)NC 3466,Cc1nn(C)c(C(=O)NCc2cc(O)nc(CNC(=O)C(C)O)n2)c1Cl 3467,C(=O)(C(C)(C)CC(C)C)NC1C(C)CN(C(=O)C(=O)NCC2CC2C2CCC2)C1 3468,C1(CCC=C)(C(=O)NCc2cc(COC)on2)CN(C(=O)CCc2cnc[nH]2)C1 3469,C1(NC(C=C(COC)C)=O)CCC2(CC1)CC2NC(=O)Cc1cncc(O)c1 3470,c1(NC(=O)NCc2n(CC)ncn2)cnc2c[nH]nc2c1 3471,C1(C#CC(=O)NC2CC3CC(NC(c4csc(Cl)n4)=O)CC23)(CC)CC1 3472,c1(C(C)C)noc(CCCC(=O)N2CCC(CNC(=O)Cc3cnnn3C)C2)n1 3473,CN1CC=C(C(=O)N(C)CC2CCCN2C(=O)C=CBr)C1 3474,N1(C(CCC(=O)OC(C)(C)C)=O)CCN(C(C2CCC(F)C2)=O)CC12CCC2 3475,C(C(CCC)C(=O)NCC(CNC(=O)OCC)OC)OC(C(=O)N)(C)C 3476,N1(C(C2C(NC(C3CCCC3F)=O)CCOC2)=O)C2C=CCC1CCC2 3477,C(=O)(CS(C)(=O)=O)N(CC(=O)NCCN(C)C(c1cnn[nH]1)=O)CC1CC1 3478,Cc1cc(C(N2CCCC2C(C)(C)NC(=O)CCc2cnc[nH]2)=O)cc(C)c1F 3479,c1(C(=O)NC(CNC(C2(CC#C)CCCCO2)=O)C)cc(F)cc(Cl)c1O 3480,C1(C(=O)NC2(C)C(NC(c3c(C)cccc3N)=O)CCC2)CC2C=CC1C21CC1 3481,c1(OC(CC)C)cc(NCC2(O)CCN(C(C3CCCC3C)=O)CC2)nc(C)n1 3482,c1(C(N2CC(NC(CSCC)=O)C(O)CC2)=O)cc2c(C)sc(C)c2s1 3483,c1(CN2CC(CNC(=O)OC(C)(C)C)N(C)CC2)ccc2c(O)nccc2n1 3484,CC1OC(=O)NC1C(N1CC(O)(CCNC(=O)Cn2cnc(C#N)n2)C1)=O 3485,Cc1ccc(-c2nnc(S)n2CC(=O)NC2CCN(C(C)C)C2C2CC2)cc1 3486,c1(C(=O)NCc2ccoc2)ccc(C(N2C(CN(C)C)CC(OC)C2)=O)cc1F 3487,N1(C(c2cc(C)c(O)cc2)=O)CC(C)(CNC(C2CCC(=O)N2)=O)CC1(C)C 3488,CC(C)CC(Cn1cc(CCCCc2ccccc2)nn1)NC(c1cccs1)=O 3489,N(C1CCc2ccccc21)(CC(=O)OC)C(=O)COCCNC(=O)NCC.CCC.CC 3490,C1(C(C)C)C(NC(C2CC2c2ccccc2)=O)CCN1C(c1cc(Cl)ccn1)=O 3491,CC1CN(C(=O)CSCCC#N)CCC1CNC(=O)Cn1ccccc1=O 3492,N1(C(c2cc(CC)oc2C)=O)CCC2(CC(NC(=O)CN3CCOCC3)CO2)C1 3493,N1(C(=O)OC(C)(C)C)CCOCC2(COCCN2c2ccc(N(C)C)nn2)C1 3494,c1(C(N2CC(O)CC(NC(C=CSC)=O)C2)=O)cc2cc(Br)ccc2o1 3495,c1(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2(C)C)ccc(C#N)cc1 3496,N1(C(CC(CC)(F)F)=O)CC2(CC(C(=O)NC34CCC(CC3)C4)CO2)C1 3497,c1(SC)ccc(C(N2CC(F)(CNc3ncc(Br)c(C)n3)C2)=O)cc1F 3498,C(CC1=CCN(CC2CCCC2)CC1)NC(C1CCCCCC1)=O 3499,c1(OC)ncnc(N(CC(CSC)C)C)c1NC(CC)C1CCC1 3500,c1(C(=O)NCC2C(C)CN(C(C34CC5CC3C4C5)=O)CC2)ccn2ccnc2c1 3501,N1(C(N2CCC3C(CCN3Cc3ccccc3)C2)=O)CC(C(=O)O)c2ccccc21 3502,N1(C(C(C)C)=O)CCCCC(NC(=O)Nc2ncccc2N(C)C)C1 3503,C(CCCC(C)NC(C1CCCSC1)=O)NC(c1ccn(C(CC)CC)n1)=O 3504,N1(C(CNC(C(C(C)C)=O)=O)=O)CC(NC(=O)CCc2ccoc2)C2CC2C1 3505,c1(CC(=O)NC(C)CC(C)NC(=O)CNC(=O)N(C)C)cc(Cl)ccc1Cl 3506,C#Cc1cccc(C(=O)NCC2CC(C)N(C(c3nnn(C)c3N)=O)C2)c1C 3507,c1(C(=O)NC2CC(C)CN(C(C3(O)CCOC3)=O)C2)ccc(S(N)(=O)=O)c(F)c1 3508,Cc1cc(C(=O)NC(CCN(C)C)C(N2CC3CC=CC2C3)=O)cc(O)n1 3509,c1(C(C)OC)nc(Cl)cc(=NCC2(C)CCC(NC(C3C=CC=CC=C3)=O)CC2)[nH]1 3510,C12(CC)CN(CCS1=O)C(=O)N2.C1(CNS(C)(=O)=O)CC1(F)F.COC 3511,N1(C(C(C)(C)CF)=O)CCC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(F)(F)C1 3512,C1(C(=O)NCC2CC(NC(C(c3nccc(C)c3)(C)C)=O)C2)CCCS(=O)(=O)C1 3513,Cc1nc2n(n1)CC(C(=O)OCC(c1ccccc1)N(C)C)CC2 3514,N1(C(CN(C(C(C)OC)=O)C)=O)CCN(C)C(C(C)C)C1.C(=O)OC 3515,C(=O)(CCC(=O)NCCN(CCOCCO)C(C1CSC(C)=N1)=O)NC 3516,c1(C(=O)NC2C(CC)CN(C(C3CNC(=O)N3C)=O)C2)cc(C#N)ccc1N 3517,c1(C(=O)NCC2(F)CC(NC(C(CCC)CC)=O)C2)c(C)nc(C)nc1C 3518,CCC(CC(=O)N1CCC(CN(C(c2ncoc2C(C)C)=O)CC)CC1)C(C)C 3519,c1(C(=O)NCC2N(C(C(C=C)OC)=O)CCCC2)cc(C#N)n(C)n1 3520,C1(NC(C(c2ccc(OC)cc2C)C)=O)CN(C(=O)C(N)=O)C2(CCCC2)C1 3521,N(C(=NCCc1cc(Cl)ccc1Cl)NC1CC1C1CC1)CC(C)(C)F 3522,C1(C(=O)NCCF)CCCS1(=O)=O.c12cccc(c1)C1(CCC1)NC(=O)N2 3523,C(C(=O)NCCC(=O)NCC)(C(C)(C)C)NC(C(C(C)C)O)=O 3524,Cc1cc(C(=O)NC2CC(CNC(c3[nH]ncc3C#N)=O)CC2O)nnc1O 3525,C1(SCC(N2CSCCSC2)=O)CNCC2(CCC2)O1 3526,C1(C(C)NC(=O)NCC(C2CCCO2)O)CCN(C)CC1 3527,C#CCC(C(=O)N1CC(N(C(=O)C=CCn2cncn2)C)C1)C1CC1 3528,Cc1cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2O)ccc1Cl 3529,C(CC1CCCC1)(C(=O)NOCCF)NC(CNC(CC)=O)=O 3530,S(=O)(=O)(c1cccc(N)n1)N(C(CCC)C(=O)O)C.c1(CO)ccccc1CC 3531,c1(C(=O)OC)cc(NC(=O)NC(c2cccc(OC(F)F)c2)C)ccc1F 3532,N1(C2(c3ncc(NC(=O)OC(C)(C)C)[nH]3)CC2)CC(C(=O)O)C2(CC2)C1 3533,C(C(N)=O)(C(C)(C)C)NC(C(C)(C1CCC1)NC(CC)=O)=O 3534,N1(C(c2cc(CNC(CC(C=C)(C)C)=O)nn2C)=O)CCC2(CCC(OC)C2)C1 3535,n1(CC#C)cccc1C(=O)NC1(C(=O)NCC2CN(C(C)C)C2)CCSC1 3536,N1(C(C(Cc2ccccc2)OC(C)C)=O)CCc2c(C(=O)O)csc2C1 3537,c1(CC(N2C(CCC)(CCC)CCC2)=O)cn2ccccc2n1 3538,c1(NC(CCC=CC)=O)ccc(NC(c2cc(O)nc(C)n2)=O)c(C)c1 3539,C(=O)(C1=NN(C)C(=O)CC1)N1CC(CNC(c2c(CC)cns2)=O)C(O)C1 3540,C1(CNC(CNC(=O)Cn2cccc2)=O)C2CN(C(=O)CCC3CCOC3)CC12 3541,c1(OC)ccc2c(C)c(C(=O)NC3CCN(C(=O)C(C)C)CC(C)(C)C3)[nH]c2c1 3542,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3543,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2ccon2)=O)C1 3544,N1(C(=O)Cn2ccc(C3CC3)n2)CCCC2CCN(C(=O)C3=COCC3)CC12 3545,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)O)CC2)CC1 3546,c1(CCCN(C)C(C2CC2(C)C)=O)cn(CCN(C)C)nn1 3547,S(=O)(=O)(c1c[nH]ccc1=NC(CF)CF)NC(c1cc(C)no1)C 3548,C1(NC(C2(C)COCCO2)=O)CCCCCC1C(=O)NC(C(O)CO)C1CC1 3549,c1(C(=O)NC2CCN(c3nccc(C(=O)OC)n3)C2)cc(F)ccc1C 3550,C1(C(=O)NCCCCCC=C)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3551,C(=O)(C(C)(CC)CCC)N1CCC(CC=C)(C(=O)NCc2snnc2C)C1 3552,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(=O)CCc1nncn1C 3553,C(=O)(C(CNC(=O)OC(C)(C)C)NCCC1CNC(=O)C1)OCC 3554,C1(C(=O)NC)CCN(C(=O)CC(C2CC2)N(C(C2CNC(=O)C2)=O)C2CC2)C1 3555,C1(C(=O)NCC(C)NC(=O)C(CO)NC(N)=O)COCCN1CC(F)F 3556,c1(C(=O)NCC23CC(NC(C4(C#N)CCCC4)=O)(C2)C3)ccc2occc2n1 3557,N1(C(CC(C)(F)F)=O)CC2(CCC(NC(=O)CC3NC(=O)NC3=O)CC2)C1 3558,C1(C)(C(=O)NCCC2(OC)CN(C(c3cc(CC)[nH]n3)=O)C2)CCCC(F)(F)C1 3559,C1(CNC(c2n[nH]c(C)c2O)=O)CN(C(c2ccccc2F)=O)CCN1C 3560,C(=O)(C1CCc2nccn21)N(C(CNC(c1c(C)nsc1C)=O)C1CC1)C 3561,CC1=C(C(=O)NC2CCC2NC(=O)Cn2cncn2)CCS1(=O)=O 3562,N1(C(CC2CCC(NC(C3(SC)CC3)=O)CC2)=O)CCN2C(=O)OCC2C1 3563,c1(-c2n(CCOC)c(N3CC4(CCC4O)C3)nn2)nn(C)c2c1CCC2 3564,c1(CC)nc(O)c(C(=O)N(C)CCNC(c2oc(Br)nc2C)=O)cc1C 3565,C(CC(F)(F)CN(C)C)NC(c1c(CC)occ1)=O 3566,C1(C(N2CC3CN(C(COCCC#C)=O)CC3C2)=O)COc2ccccc2O1 3567,CCC(CN(C)C)CC(=O)NCC12CC1CN(C(C1CSCC(=O)N1)=O)C2 3568,C(=O)(CCN(CCO)Cc1cnon1)NC(C)C 3569,C1(CCNC(CCc2scc(C)n2)=O)CCCN(C(c2sc(C)nc2C)=O)CC1 3570,Cc1cnc(NC(=O)NCC2CC23CNC3)nc1O 3571,C#CCCCCC(=O)NCc1ccc(COCC2(C)CC2)cc1 3572,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3573,c1(C(=O)NC2C(NC(c3n(C)nc(O)c3)=O)COC2)cnn2c(=O)cc[nH]c12 3574,C(=O)(CC(C)CC(C)(C)C)NC1CCN(C(C(c2c(C)noc2C)C)=O)C(C)C1 3575,C(CCC)(C(O)C(=O)N1CC(OC)CC(O)C1)NC(CC(CC)OC)=O 3576,N1(C(c2c(OC)csc2)=O)CCCN(C(c2ccnn2CC(C)C)=O)C(CO)C1 3577,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3578,C(CC(=O)N1CCC1CNC(=O)CCc1cncnc1)OC 3579,c1(SCC)ccc(C)c(C(N2CC(C3(NC(=O)CC4CCCCC4)CC3)C2)=O)c1 3580,C(=O)(CCS(=O)(=O)Cc1ccncc1)N1CC(N(C(=O)C2=CCSC2)C)C2(C1)CC2 3581,N1(C(CN(CC#C)C(C2CCC(F)(F)C2)=O)=O)CCC2(CC1)CC2C#N 3582,C1(CNC(C2(C(C)=O)CC2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3583,C(=O)(C1=C2CCN=C2NC=C1)NC1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3584,C(N=c1nc(Cl)[nH]c(C)c1C#N)C1CCN(C(c2c(CCC)occ2)=O)C1 3585,c1(CC(=O)NCC=CCNC(C2C(CC)N(C)CC2)=O)ccc(Cl)nc1F 3586,CC1CC(c2nn[nH]n2)CC(C)N1CC(C)(C)CO 3587,Cc1ccc(C(=O)NC2CCC(NC(=O)CCN3CCOCC3)C2)cc1C1CC1 3588,c1(CC)cccc(C(=O)NC2CC2NC(=O)COc2ccc(C)cc2)c1C 3589,N1(C(CCCC(=C)Cl)=O)CCC2(CCN(C(=O)C(C)(C)COCC)C2)C1 3590,C1(CC(=O)NC(CC)C)CN(C(c2cc(O)cc(=O)o2)=O)C(C)(C)C1 3591,N1(C(COCC(=O)NC)=O)CCC(C(=O)NC2(C(N)=O)CC2)C1C 3592,c1(C(N(C2CCN(C(c3cc(C(N)=O)cn3C)=O)C2)C)=O)cnc(O)n1C 3593,c1(C(N2C(CNC(c3cc(C(F)(F)F)ns3)=O)CCC2)=O)cccc[n+]1[O-] 3594,c1(NC)ccc(C(=O)NCC(C)N(C(=O)COC2(C)CCCC2)C)cn1 3595,CN1CCC(C(=O)NCC=CCNC(C23CCCC2C3)=O)CC1=O 3596,c1(SC)ccc(C)c(C(N2CCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3597,C(C(C)(O)CC(=O)N1CCC(CNC(=O)CC2(C)CCCCC2)C1)OC 3598,c1(CC(=O)OC)ccc(C2CCC2)cc1.C1C(C)C(=O)OC(=O)C(=O)N1 3599,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3600,C(=O)(C(C)(C)C(C)(C)O)N1C(CCNC(c2cccc(COC)c2)=O)CCC1 3601,c1(NC2CC(O)CC(O)C2)nc(N2CC(c3nncs3)C2)nc2ccccc12 3602,c1(C(=O)NC(C2(C(=O)NC3CCCC3C)CC2)C)nsnc1O 3603,Cc1nc(C(N2CCC(F)(C(=O)Nc3ccc(N)cn3)C2)=O)ccc1Br 3604,C(CC(CC)C(=O)NC1C=CCC(C(=O)NCC(N2CCCCC2)=O)C1)=CC 3605,C1(CNC(C2C(C(C)C)OCC2)=O)CCC2CN(C(C3CN(C)CCO3)=O)CC12 3606,C(=O)(C(CNC(=O)CC12CCCC1C2)C(C)(C)C)N(C)Cc1cnnn1C 3607,N1(C(CC(C)(C)NC(C2CC(N(C)CC)C2)=O)=O)CC2(CCCCC2)CC1C 3608,C(=O)(CN=c1cc[nH]cc1)N1CCC=C(CNC(=O)CC2CCOC2=O)C1 3609,C=CC(O)(C(=O)NCCC1CC(F)(F)CN1C(=O)CCCCC#N)C(F)(F)F 3610,c1(CC)cc(C)c(C(=O)NCC(C)(CSC)OCCNN2CCCCC2CO)o1 3611,C1(NC(c2n[nH]c(CC)c2C)=O)CC(OC)CN(C(=O)C(C2CCOC2)OC)C1 3612,C1(C(C)NC(CC=CC)=O)CN(C(c2ccnc(OC)n2)=O)CCO1 3613,n1(C(CC)C)ncc(C(=O)NC23CC(NC(=O)CN4CC(C)C4)(C2)C3)c1COC 3614,CCC(CNC(C1CN(C(=O)CCC(C)(C)C)CCN1C)=O)CC(C)C 3615,C(=O)(CC(C)c1ccco1)OC(C1CN(C(CC2CC(OCC)C2)=O)C1)=O 3616,N1(C(=O)CCCCCBr)CCC2(CC1)CC(F)CO2 3617,C1(NC(C2N(C)CCCC2)=O)CCN(C(=O)COc2ccsc2Cl)CCC1CO 3618,C=CCC(CNC(c1cn[nH]c1)=O)C(=O)NCc1ncccc1F 3619,N1(C(C(C)SC(F)(F)F)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC12 3620,c1(C(=O)NC2C(CNC(Cc3nc(C)sc3C)=O)CCCC2)cccc(Cl)c1N 3621,C1(NC(c2ccc(CC)nc2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3622,C(CC(O)C(F)(F)F)C(=O)NC(CC=CC)C(=O)N1CCCC1C1CCOCC1 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3641,c1(C(=O)NC(C2N(C(c3ccc(C)o3)=O)CCCC2)C)ccc2c(c1)nnn2C 3642,c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)coc2c(Cl)cccc12 3643,Cc1nc2cccc(C(=O)NCC3(NC(c4cc5sc(C)nc5[nH]4)=O)CC3)n2n1 3644,CCC(C)C(O)C(C)C(=O)NC(c1ccc(OC(C)C)cc1O)CN1CC=CC1 3645,N1(C(c2cc(CC)no2)=O)CCCC(CNC(C2CN(S(C)(=O)=O)C2)=O)(OC)C1 3646,c1(C(N(CC(C)(C)CNC(=O)Cc2nncn2C)C)=O)cnc2c(c1)ncn2C 3647,N1(C(C2(N(C)C)CCC2)=O)CCN(C(c2scnc2Br)=O)C2CC12 3648,C1(C(N(C(CNC(c2cnc(CC)s2)=O)C)C)=O)(OC)CCC(F)(F)CC1 3649,Cc1cc(C)c(C(=O)NCCN(C(=O)Cc2cn3ccsc3n2)C)cc1C 3650,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=CC2CCCO2)CC2(CCC2)C1 3651,N1(C(c2ccc(COC)cc2)=O)CC(CNC(C2CC(C)(O)C2)=O)CC(C)(C)C1 3652,c1(OCCC(=O)NCCN(C2CC2)C=O)ccc(Br)cc1.C(=O)(CC1CCC1)N 3653,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3654,c1(C(=O)NC(COC)CNC(=O)Cc2c[nH]nc2C)ccc2n[nH]cc2c1Cl 3655,n1(CC(=O)NC(C)CCc2ccc(F)cc2F)ncc2cccc(Br)c2c1=O 3656,c1(C(N2C(CNC(=O)CCc3cnc[nH]3)CC(OC)C2)=O)c(Cl)c(C)nn1C 3657,N1(C(=O)OC(C)(C)C)CCC(CC=O)CC1.c1(C(F)CO)ccc(O)cc1 3658,C(=O)(C(O)CCS(C)=O)N(CC)CC.C1(=O)CCCC(=O)OCC2CCN1CC2 3659,N1(C(CN(C)C(c2ccco2)=O)=O)CCN(C(C2CCCS2)=O)CC1 3660,c1(CS(=O)(=O)NC(C2CC(NCCC(C)C)C2)=O)cnc2n1CCCC2C 3661,N1(C(CCSC)=O)CCC2CCCC12C(=O)N(CC(N1CCCC1)=O)C1CC1 3662,C1(CNC(=O)COC(F)F)CC2CCC1N2C(=O)CCc1cscn1 3663,C(=O)(C(CNC(=O)CCc1cnc(C)o1)CC1CCCC1)NC1C(CC)CCC1 3664,N1(C(C2(CC)CCCCC2)=O)CCC(O)(C(C)NC(=O)Cc2cncnc2)CC1 3665,Cc1ncccc1C(N1CCC(C(C2CCC2)N(C)Cc2ccc(Br)cc2)C1)=O 3666,C(=O)(C#CC1(C)CCCO1)NC(C1CC1C(=O)NC1(C)CCCCC1(C)C)C 3667,CC1(C)CCCN(C(c2c(F)cc(F)cc2F)=O)C1CNC(C1OCCO1)=O 3668,N1(C(CCCC)=O)CCC(C)(CC(=O)N(C)CC2CCCOC2)C1 3669,C1(NC(C(CC)(C)F)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3670,N1(C(C(C2CCOC2)OC)=O)CC2C3CCC(C2C1)N(C(C1(OC)CC1)=O)C3 3671,c1(NC(c2c(C(N3CC4CC4C3)C)occ2)=O)[nH]cnc1C#N 3672,C(=O)(C(C(=O)NCC1CCCN1C(c1cc(C2CC2)oc1C1CC1)=O)OC)OCC 3673,N1(C(c2ccc(SCC)nc2)=O)CCN(C(c2ncc(C)cc2F)=O)CC1CO 3674,C(=O)(CC1CCc2ccccc21)NCCOCCC(=O)NCCCOC1(CF)CC1 3675,c1(C(C2CCCOC2)NC(c2n(SCC(=C)C)nnn2)=O)cc2cc(Cl)cnc2o1 3676,CC1CCCN(C(=O)CC(C)(C)c2cn(CO)nn2)C1CNc1ccc(Cl)cc1 3677,N(C1CN(C(C2CCCN2C)=O)Cc2ccccc21)C(c1noc(C)c1C)=O 3678,Cc1cc(F)cnc1C(=O)NC(C1CCCCCC1)C1CCNC1 3679,C1(NC(CCC=C)=O)CC2C(NC(=O)C(C)(C)n3cnnn3)C2C1 3680,c1(N2CCC(NC(c3c(C)ccs3)=O)C(C)C2)nc2ccc(Br)cc2o1 3681,c1(COCC(=O)NC(CNC(c2c(OC)n[nH]c2)=O)(C)C2CC2)nnc(S)n1C 3682,C1(C(N(CC(CNC(c2c(CC)cns2)=O)C)C)=O)(CO)CC(C)(C)C1 3683,Cn1ncc(C(=O)NCCOC(C)(C)CNC(C2C(C)(C)C2(F)F)=O)c1Cl 3684,n1(CC(=O)OC)ccc(Br)cc1=O.C1(COC)CCC1C(=O)OCC 3685,CC(C)(C(=O)NCC1CC1CNC(=O)COCP(C)(C)=O)n1cccn1 3686,N1(C(C=CCC2(C#C)CC(=O)C2)=O)CCCC(C(=O)N(CC(C)C(=O)OC)C)CC1 3687,C=CCCCC(=O)N(C)CC1(O)CN(C(c2occc2C(=O)NCC)=O)C1 3688,N1(C(C(CC)OC)=O)CCC(O)C(NC(C2CNC(=O)N2)=O)C1 3689,C1(CC(=O)N(c2cccc(C)c2OC(C)C)c2ccc(F)cc2)CS(=O)(=O)C2CNCC12 3690,C(=O)(CCS(=O)(=O)N(C)C)N(C1CCCN(C(=O)C(=O)CC)C1)CC#C 3691,O(NC(=O)C(C(C)NC(c1cn2ccccc2n1)=O)C(C)C)CCOC 3692,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3693,N1(C(C=Cc2cc(C)no2)=O)CC(CNC(=O)CC2COCCO2)CC(C)(C)C1 3694,C(CCCC(C)C)(C(=O)NCCCNC(=O)OC(C)(C)C)N(c1ccnc(C)n1)C 3695,N1(C(COC(C)=O)=O)CC2(CCC(CNC(=O)C(C)(C)C(C)(F)F)O2)C1 3696,c1(-c2cn(CCCNC(c3cc(C4(C)CC4)n[nH]3)=O)nn2)ccc(O)nn1 3697,c1(C(=O)Nc2ccncn2)cc(O)c2c(-c3cnn4ccccc34)cnn2c1 3698,c1(C(C)CC(=O)NC2CC(CNC(C3CC(C)(F)C3)=O)C2)cc(F)cc(F)c1 3699,N#Cc1cc(CN2CC3C(C2)N3C(c2ccncn2)=O)ccc1Cl 3700,N1(C(C23CCC(OC)C2C3)=O)CC2CCCC(C1)N2C(=O)CCCSC 3701,c1(OC)ccc(C)cc1NC(C1CCN(C(=O)C2=COCC2)C1(C)C)=O 3702,C=CC1(C(N2CCN(C(c3cc(C)ns3)=O)C(CCC)C2)=O)CCOCC1 3703,CC(CC(=O)N1CC(C)(C)CCC1C)C(C)(C)NC(=O)CN1CCOCC1 3704,C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CCN(C(C2(C(=O)NC)CCC2)=O)CC1 3705,N1(OCCOC)CCN(C(=O)CCc2cnn(C)c2)CC1 3706,c1(SCC(=O)NCCCCNC(c2ccn(C)n2)=O)cc2ccccc2[nH]1 3707,c1(C(=O)NC(c2ccc(I)cc2)C(=O)NCC#C)ccc(OC)c(F)c1F 3708,c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)c2ccco2)cc(C(N)=O)c[nH]1 3709,C=CCCN=C(NCc1cc(Cl)cn1C)NC1CCOC(C2CC2)C1 3710,C1(NCC#C[Si](C)(C)C)CCOC2(CCC2)C1 3711,C=CC1CCN(C(C2(NC(C3CC4CC4C3)=O)CC(O)C2)=O)C1 3712,c1(OC)ccc(C(=O)NCC#CCNC(C2CCCC(O)C2)=O)nc1 3713,C(=O)(CC(C(F)(F)F)n1cccn1)N1C(CN(C)C(C2CNC(=O)N2)=O)CCC1 3714,C1(C(=O)Nc2cccc(OC)c2)CCCC(N=c2ccc([N+](=O)[O-])c(O)[nH]2)C1 3715,N1(C(CCC(=C)C)=O)CCC(F)(CNC(C2CCC(=O)N2C2CC2)=O)CC1 3716,C1(CCNC(C(C)NC(C=CCOC)=O)=O)CCN(C)C1 3717,CC1CN(C)CC(C(=O)NC(C)C(N2CC(O)(CC(N)=O)C2)=O)O1 3718,CCC(CC)C(C(=O)N1CC(O)CC1CNC(C1(COC)CC1(F)F)=O)OC 3719,C12(C(=O)NCC3N(C(C(c4ccc(CC)s4)=O)=O)CC3)COC(CF)(C1)C2 3720,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3721,N1(C(=O)Cc2coc3ccccc23)C2CCC1CN(C(C1C3COCC13)=O)CC2 3722,c1(C(=O)NCCC2N(C(C3(C)C=CCC3)=O)CCC2)ccc2ocnc2n1 3723,C12(NC(C(CCSC)OC)=O)CC1CN(C(c1coc(C)c1)=O)C2 3724,c1(NC(C2CCC(NC(c3c(OC)ccs3)=O)CO2)=O)cc(Br)cn2ccnc12 3725,c1(CC)cnccc1C(N1CCC1(C)CC(=O)NCC1(N(C)C)CC1)=O 3726,c1(C2(CC(=O)Nc3cn(CC)nc3)CC2)ccc(C(=O)C(Cl)(Cl)Cl)cc1 3727,c1(OC)cccc(OC)c1C(=O)NCCC1CCCN(C(=O)C(C(C)C)OC)C1 3728,c1(OCC)ccc2nc(N3CCC4(CCC(CNC(=O)CC5CC5)O4)C3)sc2c1 3729,CN1C2CCC1CC(=CC(=O)NCC1CCN(C(c3cnccn3)=O)CC1O)C2 3730,c1(C(=O)NCC2CCC(C(N(CC)Cc3ccco3)=O)O2)c(C)noc1C 3731,c1(-n2cc(CCN(C(=O)C(C)O)CCOC)nn2)ccc(C(C)C)cc1 3732,c1(NC(=O)CSN2CCC2)cc2n(n1)CCN(C(=O)Cc1ccccc1F)C2 3733,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3734,C1(CC(=O)N(C)CCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3735,c1(C(N(C2CCN(C(=O)CCC3CC(C)C3)C2)CC#C)=O)ccc2nc(O)[nH]c2c1 3736,C12C3C(CN1Cc1ccc(nc1Cl)NC2=O)C3(C)C.c1(OC)cncc(CO)c1 3737,c1(COC)ccc(C)cc1C(=O)NCC=CCNC(=O)CCCc1nccs1 3738,C(=O)(C1CCc2c[nH]nc21)N(C1CCN(C(C(CCCC)O)=O)CC1)CC1CC1 3739,C1(N(C(=O)CCC2CC(NC(C3CCCCS3)=O)C2)C)CNC(=O)OC1 3740,c1(C(N2CCCC23CCOC3)C(=O)NC)ccc(F)c(C)c1F 3741,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCCC(C)c3cn[nH]c3)C1CC2 3742,C1(F)(C(=O)NCC2OCC(CNC(=O)COCCCF)C2)CCC2(CC1)CC2 3743,c1(C(C)=O)ccc(OCC(=O)NC(C)CN(C)C(c2ccc(F)s2)=O)cc1 3744,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3745,C1C(CC(C)C)C(=O)N1.N1(C(C2(OC)CCOC2)=O)CCCCC(CO)C1 3746,c1(OC)cc(OC)cc(S(=O)(=O)NCc2cc(-c3n[nH]c(C4CC4)n3)on2)c1 3747,C#CCC1CC(=O)NCC(C)(C)OC(=O)CC(=O)N1.C(C)(C)(CC)OC 3748,Cc1nn(C)c2nc(C(=O)NCC3(CNC(=O)Cn4cnnc4O)CC3)ccc12 3749,C1(NC(C(CC)CCOC)=O)CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 3750,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3751,C1(C(=O)NCCNC(C(c2cccnc2)SC)=O)CC(O)C(O)CO1 3752,c1(C(N(CC(C)NC(=O)CC(C)C(=O)OC)CC)=O)ccc2ccnc(Cl)c2n1 3753,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3754,CC1(C)COC(CC(=O)NC2(CO)CCCN(C(=O)COc3cccnc3)C2)CO1 3755,C1(COC)(NC(c2sccc2C#N)=O)CCCN(C(=O)CCn2cc(C)cn2)C1 3756,c1(CC)cc(C(N2CC(=C(F)CNC(=O)C(C)COCC)C2)=O)c(C)nn1 3757,c1(N(C)C)cc(NCC2(O)CN(C(C3CC(Cl)(Cl)C3)=O)C2)ccc1[N+](=O)[O-] 3758,C1(CN(C)C(C23CC(C)(C2)C3)=O)CN(C(=O)C(F)(F)C2CCCC2)CCO1 3759,Cc1ccc(C(C)N(CC(C)C)CCC2(O)CCOCC2)cc1C#N 3760,C=C(C)CC(C(=O)N1CC2CC(C)C2C1)NC(=O)C(O)CCC 3761,c1(CC(=O)OC)ccc(NC(=O)CCC(C)C)cc1.c12ncc(s1)CNC(=O)C2 3762,C(C1CSc2ccc(Br)cc21)C(c1ccccc1)C.C12CCCN1C(=O)C(=O)N2 3763,CC1CC2(CCN(c3ccnc(N(C)Cc4ncc[nH]4)n3)C2)CO1 3764,C1(C(=O)NC2C(C(=O)OCC)CC=CC2)CCCC12OCCO2 3765,C(CCCC(C)C)(c1n(CC=C)nnn1)Nc1sc(C)nc1CC 3766,N1(C(=O)Cc2ccco2)CC2CCCC(C1)N(Cc1ccc3nonc3c1)C2 3767,c1(C(N2C3C(NC(=O)Cc4cscn4)C(CC3)C2)=O)sc2ccccc2c1Cl 3768,N1(C(=O)CCc2ccccc2)C2CCC1CC(C(N1CCCc3n[nH]cc31)=O)C2 3769,c1(C(N2CC3(N(C(C(C=C)(C)O)=O)CC3)C2)=O)ccc2ncn(C)c(=O)c2c1 3770,N1(C(c2cnc(F)c(Cl)c2)=O)CCC2CCN(c3nc(C(F)(F)F)ns3)CC2C1 3771,N1(CC2(C)CCN(Cc3ncn(CC)c3)C2)CCC2C(C(=O)OC)C2C1 3772,C1(NC(CCCNC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3773,C1(NC(=O)NC(c2cc(Br)no2)C)CCN(C)C(c2ccccc2)C1 3774,C1(C(=O)NCCCCN=[N+]=[N-])CN(C(=O)CCOCC2CCC2)CC12CC2 3775,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc(OC)n2)=O)C1)C)OC 3776,CC(C)C(O)C(F)(F)C(=O)N(C1CN(C(C2CC2c2ccncc2)=O)C1)C 3777,n1(C(C)C)ccc(C(=O)N(CC(O)CN(C(=O)CN(S(C)(=O)=O)C)C)C)n1 3778,C(N=c1[nH]c(N(C)CCc2cccnc2)nc2c1CSC2)C1(OC)CCOCC1 3779,CC(C(=O)NC12CC(CNC(C34CCCC3(C(N)=O)C4)=O)(C1)C2)C(F)(F)F 3780,CC1CN(C(C2C3CN(Cc4ccnn4C)CC23)=O)CCS(=O)C1 3781,C1(C(=O)NCC2CCN(C(C(C=C)C)=O)C2)CCC(C2CC2)C1 3782,C(=O)(C(C)CC(=O)N1CCC(CNC(c2ccc(C(C)C(C)C)cc2)=O)C1)OC 3783,c1(C(=O)NC(CN2CCN(C(C3C(OC)CC3)=O)CC2)C)cccc(=S)n1O 3784,C1(C(C)NC(c2cnc(C3CCCC3)s2)=O)CCCN(C(C2CNC(=O)N2)=O)C1 3785,N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCC2(CCN(C(=O)C(=O)N(C)C)C2)C1 3786,c1(C(=O)NC2C(OC)CN(C(=O)CCc3csc(=N)[nH]3)C2)cc(C)nc(C)n1 3787,CC(C)(C)C(C)(C)C(=O)N1CC2C(CNC(=O)CC(O)CCn3cnnn3)C2C1 3788,Cc1ccc(CCC(=O)NC(C)CCNC(C2C(C)C2C)=O)c(C)c1 3789,C(C)(C1=CCCOC1)NC(C(CC1CCOCC1)NC(c1[nH]cc(C)c1)=O)=O 3790,c1(C(N(C2CCCC(NC(=O)CC34CC(C3)C4)C2)C)=O)cc(=O)n2nccc2[nH]1 3791,C1(C(=O)NCCCN(C(=O)CSC(F)F)C)CC(=O)N(c2ccccc2F)C1 3792,CCC1=C(C(=O)NC2CCCC2CNC(c2ccc(SC)nc2)=O)CCCO1 3793,c1(C(=O)NCC2(F)CCN(C(C(CC)OC)=O)C2)cnc(C)cc1C 3794,c1(C(=O)NC2CC3(C(NC(CCNS(CC)(=O)=O)=O)C3)C2)cc(Cl)ccc1F 3795,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3796,CC(=O)CCCC(=O)NC(C12CC(C)(CO1)C2)C(=O)NCCOCC(F)F 3797,n1(CC)cc(C(N2CCCC2C(C)(C)NC(c2cc[nH]c2)=O)=O)c(C)n1 3798,c1(N(C(C)C)C(C)C)nc2ccccc2cc1-c1nnnn1CCCF 3799,c1(COC(C)C(=O)NCC2CCN(C(c3cncs3)=O)C2)ccccn1 3800,c12cc(nn1C)C1(CC1)C(=O)N(C)C2.c1(C2C(C)C2)cn(-c2ccccc2)nn1 3801,CCC(C)(C)CCCC(=O)NC(CNC(c1cc[nH]c1C1CC1)=O)CO 3802,c1(CC(=O)N(CC(=O)NCCSCCCO)C)cncnc1 3803,c1(C(C)NC(C2(C)CCC2)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1.C12CC1C(=O)N2 3804,C1(C(N2CC(C)OC(C)C2)C(=O)NCCOCC)CC2CC1C1CC21 3805,C(C)(CO)(C(=O)N(CCCCC(=O)N(C1CCC(CO)CC1)C)C)OC 3806,CC1CN(C(=O)CSCC(F)F)CCC1CNC(c1ccnn1CC#N)=O 3807,c1(OC)cccc(C(N2CCN(C(C)CNC(=O)C(C)CS(C)=O)CC2)=O)c1C 3808,C#Cc1ccc(F)c(C(N2CC3(CC3)CC2CNC(C2CC23CCOC3)=O)=O)c1 3809,N1(C(CCC(=O)N(C(C)C)C)=O)CC2CCC1CN2C(=O)C=CC1CCOCC1 3810,CN1CC=CCC1CC(N1CCC(CC(=O)NCC2CCCN2C)C1)=O 3811,N1(C(=O)Cc2cnsc2)CCCC(C2CCCN(C(=O)Cc3nc[nH]n3)C2)C1 3812,N1(C2c3ccc(s3)NC2=O)CC(C)(C)C(O)C(C)(C)C1.O=CNCCC1CC1 3813,CC1CN(C(C2CC2C#N)=O)C1C(=O)NCC(C)(C)C#N 3814,C#Cc1ccc(C(=O)NC2CCN(C(c3nnc(Cl)cc3N)=O)CC2O)cn1 3815,c1(C(=O)NC2CC(CCNC(C(N3CCSCC3)C)=O)C2)ccc2ccoc2c1 3816,c1(CNc2cccc(C3CC3)c2)cnc2n1CCCCC2 3817,N1(C(C(=O)NCCS)c2cccs2)CCOC(C2CC2)CC1.CCO 3818,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3819,c1(OC(F)F)c(C(=O)OCC(=O)NCCCOC)ncnc1C 3820,C(=O)(C(C)COC)NC(C(=O)N(CCC)CC)c1cccs1 3821,c12ccc(F)cc1C2.C1(CC)CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3822,C1(N(C(=O)C(C)C2CC2)CC)CCN(C(c2csc(C)c2Br)=O)CC1 3823,C12(NC(CN(C)C(C3(S(N)(=O)=O)CC3)=O)=O)CC1CN(C(=O)OC(C)(C)C)C2 3824,c1(C(N2CCC(F)(CNC(CCOCC(C)C)=O)C2)=O)cc2ccncc2s1 3825,N12CCCC(C1)NC(=O)CCC1(CC1)C2=O.N1(NC(C23CC(F)C2C3)=O)CCOCC1 3826,N1(C(C(C)OCC2CCCO2)=O)CCC2(CCCN2c2ccnc3ncnn23)CC1 3827,n1(CC(N2CCC(O)(CN(C(C3C(C)C3C)=O)C)CC2)=O)ccc2cccnc12 3828,CC(C)CC(F)C(=O)NC1(C2CN(C(c3cc(-c4ccco4)on3)=O)C2)CC1 3829,C1(NC(C(c2cccnc2)C)=O)CC2CC(NC(=O)CCc3cccn3C)C2C1 3830,C=CCCC(C)NC(C1CCCC1CNC(C1CN(C)C1)=O)=O 3831,C(=O)(C(N=[N+]=[N-])C(C)C)N1C(C)(CCCN(OC)C)CC(O)C1.C12CCN1C2=O 3832,Cc1nc(NC2(C(CN(C)CC3CCOC3C)=O)CC2)sc1C(=O)NC1CC1 3833,c1(SCC)ccc(Br)c(C)c1O.c12oc(C(F)(F)F)cc1C(=O)NC2 3834,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CC1 3835,CC#CCC(C(=O)Nc1ccc(CC)nc1)NC(=O)CCn1cncn1 3836,CCCCCC(O)C(=O)N1CCC2CC2(C(=O)NOc2ccc(CO)cc2)C1 3837,N1(C(COCCC)=O)CC(CC(N2CC(C3CCCO3)C2)=O)CC1(C)C 3838,C(=O)(C(C(=O)NC(C)(C)C(C)NC(c1occc1CN(C)C)=O)OC)OCC 3839,c1(C(=O)NCCC2CCC(NC(COCCOC)=O)C2)cc([N+](=O)[O-])ccc1N 3840,C1(C(=O)NCCC(=O)NC2CCCOC2)CCCNC12CC2 3841,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3842,Cc1cc(C)c(C(=O)NCC(N2CCC(NCc3ccccc3C)C2)=O)c(Cl)n1 3843,CC1(C)OC(=O)CC1C(=O)NCCOCCNS(=O)(=O)NC1CC2(CCC2)CO1 3844,c1(NC(CC(CC)NC(=O)C(C)CC(C)C)=O)cccc(Br)c1OC 3845,Cc1onc(CO)c1C(=O)N(C(CNC(=O)C(C)C1CCCO1)C1CC1)C 3846,C(=O)(C#CC1CCOC1)NCC1C(C)CCN(C(=O)C=CC=C(Cl)Cl)C1 3847,CC(C)C(C(=O)NCC1(NC(C2CN(C)C2)=O)CCOC1)c1cnn(C)c1 3848,C1(C(C)C(=O)NCC(CO)NC(c2cnns2)=O)CCC(=O)N1 3849,CC(C)C(CCNC(c1nnn(C)n1)c1nnnn1CSc1ccccc1)N(C)C 3850,c1(OC)ccc(C)cc1C(N1CC(CNC(c2ncc(C)cn2)=O)C2(CC2)C1)=O 3851,C1(C(N2CCC(N(C(=O)C(c3cccnc3)O)C)C2)=O)CCc2ccccc2C1 3852,C12(CNC(c3ccc(C(C)C)o3)=O)CC(CN1C(C1CCCCO1)=O)C2 3853,C1(CNC(c2cn(C3CC3)cn2)=O)CC2(CC2)CN1C(C1CCCN1C1CC1)=O 3854,Cc1ccccc1NC(C1C(NC(C2CCC2C#N)=O)CCO1)=O 3855,c1(C(=O)NCCOCCCNC(Cn2c(C)cc(CO)n2)=O)cc(O)nc(Cl)c1 3856,C=CC(C)(CC)C(=O)NCc1ccc(C(=O)NCCCOC(C)=O)nc1 3857,c1(CO)ccccc1.C(=O)(CC)N(CCCC)CCOC.C12(CC1)C(=O)NC2=O 3858,C12(CNC(=O)CNC(C3CCCCC3)=O)CCC1CCN2C(=O)Cc1cccs1 3859,C(=O)(CCCCN=[N+]=[N-])N1CC(C(N(C)CC2CCC(C)CC2)=O)N(C)CC1 3860,C1(C(=O)NCC(C)NC(c2ccc(-c3cccc(Cl)c3)s2)=O)(CC)CCNC1=O 3861,Nc1cccnc1C(=O)NCC1CCCC1C(=O)NCCn1cc(CO)nn1 3862,C(=O)(CC(C)C(F)F)NCCCCNC(CC(CC)O)=O 3863,C=CCC(CNC(C1(C(F)(F)F)CCCC1)=O)NC(=O)CN(C)C(C)=O 3864,C1(CNC(CC2OCC(C)(C)C2)=O)CN(C(=O)CC2CCCCC2)CCCO1 3865,C(CC(C(=O)N(CCC(=O)NC(c1ccccc1O)C1CC1)C(C)C)OC)OC 3866,c1(CC)c(C(=O)NC2CCN(C(c3csnn3)=O)CC2O)sc2ccccc12 3867,C=CCC(C)(CNC(C1(C)CCCN1C(=O)COC1CCCCC1)=O)CO 3868,c1(CC)cccc(C(=O)N(CCNC(=O)CCc2ccn(C)n2)C2CC2)c1 3869,C#CC1CCCN1C(=O)COCCCCCN=[N+]=[N-] 3870,N1(C(C(COCC)C)=O)CCSCC1CCNC(=O)Cc1ccnn1C1CC1 3871,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3872,C1(SCC(=O)NCC2N(CC(=O)NCC3(Br)CC3)CC2)CCCCO1 3873,Cc1nsc(NC(C)CNC(C2(CF)CCOCC2)=O)c1C#N 3874,N1(C(=O)NC2CN(C)CC2F)CCCC(OCc2ccccc2)CC1 3875,N1(CC(CC)NC(=O)CS(=O)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 3876,C1(NC(c2cn(-c3ccc(O)cc3)nn2)=O)CCCCN(C(c2nc(Cl)cs2)=O)C1 3877,Cc1c(F)cc(C(N2CCC(C(N3CC(C#N)C3)=O)C(O)C2)=O)cc1F 3878,N1(C(CSCC(=O)OC)=O)CCC2CCCN(C(c3c(C)nn(C)c3C)=O)C2C1 3879,C1(C(N(C)Cc2nnn(C)n2)=O)COCCN1C(C1CCCN1S(C)(=O)=O)=O 3880,c1(OC)cc(C(=O)NC2(CNC(=O)C(c3cccc(C)c3)=O)CCOC2)n(C)n1 3881,c1(C(N(CCN(C(C(C)OCC)=O)CC)C)=O)cc(Cl)cnn1 3882,CC1=CCCCC1.N1(CCCCCNC(=O)C)CCN(C(=O)CNC=O)CC1 3883,C1(C(=O)NCC(=O)N(C2CCCC2)CC)CCCN(C(=O)Cc2nc[nH]n2)CC1 3884,c1(N2CC(CC)N(C(C3CC3N)=O)CC2)ncnc2ccc(F)cc12 3885,N1(C(C(C)n2cnnn2)=O)CCCC(N(C(=O)C(F)OC(F)(F)F)CC2CC2)C1 3886,C(CCCCC(=O)NCC(O)CC1CCC1)NC(c1cnnc(C)c1C)=O 3887,S(=O)(=O)(c1ccccc1NC(=O)N(C)CC1(O)CCC(C)(C)C1)N(CC)CC 3888,C(=O)(CCCCCCCCCO)NCCC1N(C(=O)C=CCF)CCCC1 3889,C1(C(=O)NCC(C)CNC(=O)COCC2CCCO2)CCS(=O)(=O)C1(C)C 3890,C#CC1CN(C(=O)C(CCOC)NC(c2cnn(CC)n2)=O)CCO1 3891,N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CC(NC(=O)C(C)(C)CF)C2)C1 3892,c1(OC)cc(F)c(NC(=O)NCC2COCCC2C)c(F)c1 3893,c1(CCC)ccccc1C(=O)NC1CC(NC(=O)Cc2ccc(C)o2)C(O)C1 3894,C1(C(N2C(CNC(CC(CC)OC)=O)CC(F)C2)=O)CNc2ccnn2C1 3895,C#CCC(CC#C)C(=O)NCC1CCCC(NC(C2(c3cc[nH]c3)CC2)=O)C1 3896,C1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)C)Cc2c[nH]cc2S1(=O)=O 3897,C1(N(C(=O)CCNC(=O)NC)CCC)CCCN(C(=O)CP(C)(C)=O)CC1 3898,Cc1nnc2ccc(C(N3CCCC3C(C)NC(c3cncs3)=O)=O)cn12 3899,Cc1c(F)ccc2nc(C3CCN(c4cc5ccccc5c(O)n4)CC3)[nH]c12 3900,c1(OC(C(C)Cn2ccnc2)=O)cccc([N+](=O)[O-])c1 3901,CCC(O)C(C)C(=O)N1CC(CNC(C2CCS(=O)CC2)=O)C(C)(C)C1 3902,C1(CC(C)C)C(=O)NCCN1C(=O)CC1(C)CCN1C(C1COCCN1C)=O 3903,C1(CNC(C#CC(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)NC1=O 3904,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(NC(C)C)cc2)=O)CCC1C 3905,c1(C(=O)NCCCNCCNC(C2C(OC)CCC2)=O)cccnc1Cl 3906,O=C(CCCn1cc(CC2CCCCO2)nn1)NCCCN1CCCC1 3907,C1(NC(C(c2ccccc2C)COCC)=O)CCCN(C(C)(C)C)C1=O 3908,C(C)(CC(C)(C)CO)NC(C1(C(C)C)CCN(C(C=C(CCC)CCC)=O)C1)=O 3909,CC(C)(CC#N)C(=O)N(CCF)CCNC(=O)Cc1ccc(C#N)cc1 3910,c1(C(=O)NCCCN2CCC(NC(C3(C#C)CCC3)=O)C2)cc(CC)ccc1C 3911,CCC(CC(=O)N(C1CCCN(C(=O)CCN(C)C)C1)C)NC(C1CCC1)=O 3912,C1(NC(C2CCN2C2CCCC2)=O)CN(C(=O)C2=CCCOC2)CCC1C(F)(F)F 3913,C(=O)(C(CCOC)OC)NC(C=CC(=O)NC(COC)(C)CO)(C)C 3914,N1(C(CCC)=O)CCC(O)(CCNC(=O)Cc2n[nH]c(=NC)s2)CC1 3915,CC(N=c1[nH]nc(C2CC2)s1)c1ccnc(F)c1 3916,O=C(CN=c1cc(F)c(Br)c[nH]1)Nc1cnn(Cc2ccncc2)c1 3917,C1(NC(C(C)(C)N(C)C)=O)CCCCCN(C(c2c[nH]nc2C2CCCO2)=O)C1 3918,C=Cc1cc(C(=O)N(CC(N2CCC(C(=O)CC)C2)=O)CC)cc(F)c1 3919,c1(C(N2CC(COC)N(Cc3ncccc3C)CC2)=O)c(F)ccc(F)c1Cl 3920,c1(OC)ccc(F)c(C(=O)NC2CC(NC(=O)CC3CCCN(C)C3)C2)n1 3921,N1(C(=O)CCCc2ccsc2)CCCN(C(=O)CC23CCC(CC2)C3)C(CO)C1 3922,C1(C(c2ccccc2)C)CCN(C(=O)CSc2ccc(F)cc2)CC1O 3923,C=CCCC(O)CNC(=O)CC(O)CNC(c1csc(C)c1C)=O 3924,C1(NC(C(Cc2cc[nH]n2)NC(CN(C(C)C)C)=O)=O)CCCC2(CCC2)C1 3925,c1(-n2ccc(C(=O)NCC3(O)CCCC3)n2)ccc(F)cc1.C12CC(C1)NC2=O 3926,C1(NC(=O)CC2CN(C(=O)C3=COCCC3)CC23CC3)CCN2CC(O)CC2C1 3927,N1(C(C(C)CC2CCCCC2)=O)CCC(C(C)NC(c2ncc[nH]c2=O)=O)CC1 3928,C1(C(=O)NC(C(C)O)C)CC2(CCN(C(=O)CC3CCCCC3)C2)C1 3929,N1(C(c2ccc(N(C)C)nn2)=O)CC=C(CNC(c2cnn(C3CC3)c2)=O)CC1 3930,CC1(C)CC(NC(c2csc3nccn23)=O)CN1C(=O)Cc1ccncc1Cl 3931,c1(NC(CC(C2CC2)NC(CC(C=C)C)=O)=O)cc(O)c(C)cc1C 3932,CC1C(O)CCCN1C(C1(CSc2ccc(F)cc2F)CCC(=O)C1)=O 3933,Cc1[nH]nc(C(F)F)c1C(=O)NC1CCC(CNC(C2CCC(F)C2)=O)CC1 3934,C(=O)(CCCC(F)(F)CO)NCC1(C)C(C)CN(C(=O)CCn2cc(Cl)cn2)C1 3935,c1(OC)cc(C(N2CCC(O)(CNC(=O)C(c3cccc(C)c3)F)C2)=O)ccn1 3936,N1(Cc2c(C(=O)NC(C(=O)OC)CC(F)(F)F)scc2)CCC2C(O)CCCC2C1 3937,CC(Cc1cccc(F)c1)CC(=O)N(CCCC1C=CCC1)CCc1cn(CCF)nn1 3938,CCC(CCC(=O)NC(C)C1CC1)NC(=O)C(C)CCO 3939,N1(CC(C2CCCO2)OC)C(=O)CN(Cc2csc(-c3cccs3)n2)C1=O 3940,C12(C(=O)NC34CC3CN(C(c3cnc(SC)[nH]3)=O)C4)C3C4C1C1C2C3C41C(N)=O 3941,c1(N2CC3CN(C(CN(C)C(N)=O)=O)CC3C2)nc2cc(F)cc(F)c2o1 3942,N1(C(c2cc(C)on2)=O)CCCC(C2CCN(C(=O)C=C3SCC(=O)N3C)C2)C1 3943,C(=O)(C(CC)(CC)C(=O)OC)NCCOCC(=O)NCCCC(=C)C 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4016,C(CCC(C(=O)Nc1ccccc1)N(C1CCN(C)CC1)C)=CC 4017,CCC(C)CC(C(=O)NCc1cc(C#N)n(C)c1C)NC(C)=O 4018,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(Cc2ccc(CC(C)C)nc2)=O)CC1 4019,N1(C(CN(CCCC=C)C(=O)C=C(C)CCC)=O)CCC(CC)(CC)CC1 4020,c1(OC)noc(C)c1C(N1CCC(CN(C(=O)CC2(C)CCCCC2)C)C1)=O 4021,N1(C(CC=CCC)C(=O)NC2CC(C(=O)OC)C2)CC2(C1)CC2(F)F 4022,C(=O)(C(=O)CCCC)N(CC(C)NC(=O)CCc1cnc(C(C)(C)C)o1)CC 4023,N1(C(C(CC=C)CC)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 4024,c1(CNC(=O)NCC2CCOCO2)cc2c(nc1O)CCCCC2 4025,c1(C(=O)NCC2CN(CC3CCCC3(F)F)C2)ccc2c(n1)OCCO2 4026,C1(O)(CN(C(c2nn(CC)c(C)c2)=O)C)CCCN(C(=O)C(F)=C(C)C)C1 4027,C1(NC(C(C)N(CCSc2ccccc2)C)=O)CN(C(=O)C(=O)N(C)C)CC1O 4028,c1(C(N(CCCCN(C(c2nccc(CC)c2)=O)C)C)=O)nc[nH]c2ncnc1-2 4029,c1(-n2c(C(C)(CCCOC)NCC=CCC)nnn2)ccc(Cl)cc1F 4030,N1(CC(=O)N(CC)CC)CC2(CC2)CC1CSc1csc(-c2ccccc2)n1 4031,c1(-c2cn(C(N3CC4CC4(C(N4CC(C(N)=O)C4)=O)C3)=O)nn2)cnccc1Cl 4032,C1(CNC(c2n(CCC)ncc2)=O)CCN(C(C2CSCN2C)=O)C12CCC2 4033,N1(C(C2(OC)CCCOC2)=O)CCN(C(=O)CSCCC(C)C)C(CO)C1 4034,C(C(CC(F)(F)F)NC(c1cc(F)cc(F)c1)=O)NC(CC1CC(OC)C1)=O 4035,C1(NC(CCCC=C)=O)CCCC(NC(C2CC(=O)C2C)=O)CC1 4036,C(CCC(C)C)(C(=O)NC(c1ccccn1)C)NC(c1c(CC)nccn1)=O 4037,C(=O)(C(C)(O)C(F)(F)F)N1CCC(CN(CC(c2ccc(C)c(Cl)c2)=O)C)CC1 4038,c1(N2CCC(OCC)C2)nc2ccc(F)cc2s1.C12(CC1)C(=O)NCCO2 4039,C1(NC(C(CC=C)NC(C)=O)=O)CCCC2CN(C(=O)C(O)CCS(C)=O)CC12 4040,N1(C(C2CN(C(C3CCC(NC(C)=O)CC3)=O)C2)=O)CCCC(C)CC1 4041,C(=O)(C(C1=CCCSC1)N1CCOC(C(C)(C)C)C1)NCC=C 4042,N1(C(c2nc(OC)cc(OC)n2)=O)CC2(CCC2)CN1C(c1cncc(Cl)c1)=O 4043,N1(C(c2c(N)cc(F)cn2)=O)CC=C(CC(=O)NC2CC2O)CC1 4044,C1(NC(C2N(C(C3CC(CC)(CC)C3)=O)CC(OC)C2)=O)CC2(CC(OC)C2)C1 4045,C(CCC(=O)N(CC1CN(C(=O)CC2CC(F)C2)C1)Cc1ccccc1)OC 4046,C1(N(C)C(c2cnc(-c3ccoc3)[nH]c2=N)=O)CS(=O)(=O)CC1N(C1CCC1)C 4047,C(C(C)(CO)CO)N(C(=O)C(C1CC1)N(C(=O)CC(=O)N(C)C)C)C 4048,C1(C(N(C(C)C)CCF)=O)CN(C(=O)Cn2cnnn2)CC1(F)F 4049,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4050,c1(SCC2(C(=O)NCC3N(C(CC(C)(C)C)=O)CCC3)CC2)cc(F)cc(Cl)c1 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4069,c1(C(N2CC3C(CNC(c4n(CC)ccc4)=O)(C3)C2)=O)cnc2c(C)nccn12 4070,c1(C(=O)OCC)ccnc2c1CCCN2C(=O)C(=O)NCCC1CCCSC1 4071,C1(CN(C(C2CCOC2)=O)CC)COCCN1C(=O)CN1CC2CC2C1 4072,N1(C(C2(C)CC(NC(C3CCN(CC)C3)=O)C2)=O)C2CSCC1C2 4073,c1(N(CCCN(C(CSCCC(C)C)=O)C)C)ncc2c(Br)cccc2n1 4074,Cc1cc(Br)cnc1C(=O)NC(CNC(=O)COC(F)(F)F)CO 4075,c12nc(Cl)c(Cl)nc1NC2=O.N1(C(C2CC2OCC)=O)CCC(OCC)C1 4076,CC1=C(C)CC(C)(C(=O)N(CCNC(=O)CC#N)C(C)C)CC1 4077,c1(C(N2CC(OCCC(=O)NCCOCCC=C)C2)=O)ncsc1C 4078,c1(NCc2c(Cl)nccc2)ccc(S(=O)(=O)NCc2ccns2)cn1 4079,Cc1nc(N2CC3(CCC3)CC2CNC(C2CCSC2)=O)c2ccsc2n1 4080,C1(C)(C(N2CC(NC(c3ccc(C)c(C)c3O)=O)C2)=O)CC(C(C)(C)C)=NO1 4081,C1(CNC(CSC(C)C)=O)C2CN(C(c3cc(C4CC4)cs3)=O)CC12 4082,N1(C(c2nc(CNC(CSCC)=O)oc2)=O)CCC2(CCCN2C)C1 4083,c1(N2CC(=O)N2)ccccc1C(CNC(C)=O)OC.C(C(C)SC)CC 4084,Cn1cnc(CNC(=O)CC2(NC(C3CCCCS3)=O)CCC2)n1 4085,c1(C(=O)NCC2CCCC(NC(C(CC)(C)CO)=O)C2)ccc2cnoc2c1 4086,Cc1ncc(Br)cc1C(=O)NCCN(C(=O)COC(C)C)CC1CC1 4087,Cc1cnc(CN(C(=O)C=CC(C)NC(=O)CCCn2cccn2)C)o1 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4106,CCCS(=O)(=O)CC(=O)N1CC(C(C)O)(CNC(=O)CCc2ccc(Cl)nc2)C1 4107,Cc1nc(CN2CC(C)CC2C(=O)NC2CC3(CCC3)C2)c(C)o1 4108,CC1CC(C(=O)N(CCCCN(C)C(c2c(Cl)noc2C2CC2)=O)C)CC(C)C1 4109,N1(C(c2c(C)cnn2C)=O)CCC2(CC1)CC2NC(c1cc(C#N)ccc1F)=O 4110,N1(CC(=O)Nc2ccc(F)nc2)CC2(CCN(Cc3cccnc3)C2)C1 4111,c1(CC)c(C(N2CCCC(NC(=O)C(C)c3ccsn3)C2)=O)cnn1CCC#N 4112,C(=O)(C(CO)C(C)C)NCCOC1CCN(C(CCC(=O)OCCC)=O)C1 4113,N1(C(CC2ON=C(CC)C2)=O)CC2CC1CC2NC(c1cc(-c2ccco2)on1)=O 4114,c1(C(N(C)CC2(NC(C3N(CCC)CCC3)=O)CC2)=O)nc2ccccc2s1 4115,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4116,c1(C(N(CCCCCNC(C(C(C)OC)O)=O)C)=O)ccc2nnn(C)c2c1 4117,C1(CNC(c2c(C)sc(Cl)n2)=O)CC2CCC1N2C(C1CC2CCC2C1)=O 4118,c1(OCC(=O)Nc2ccccn2)ccnc2c1CCO2.C12CC13CCN(C3)C2=O 4119,C1(CN(C(=O)CN2CC(C)(C)C2)CC)CCN(C(=O)C(C)CC#N)CC1 4120,C=C=CCCC(=O)NC(C1CN(C(=O)C=C(CCC)CCC)C1)C 4121,Cc1ncc(Br)c(C(N2CCC(NC(c3cc(Cl)n(C)n3)=O)C(C)C2)=O)n1 4122,C1(S(C)(=O)=O)(OCCCC)CCCCC1.c12ccc(o1)C=CC(=O)OC2 4123,C1(CNC(c2nn(C)c(O)c2)=O)(CO)CCCN(C(C2CC3C(C2)C3(C)C)=O)C1 4124,C1(NC(C2CCc3n[nH]cc3C2)=O)CCC2(CC1)CC2Nc1ccncn1 4125,c1(C(N2CC(C(=O)NCC3CCC(F)(F)CC3)C(F)C2)=O)ccc2n[nH]cc2c1 4126,N1(C(c2c(C)cc(O)nc2)=O)CCC(CNC(C2CC(=C3CCC3)C2)=O)C(C)C1 4127,S(=O)(=O)(c1cccc(Cl)n1)N1C(CNC(c2cnccc2CO)=O)CCC1 4128,C(CCCCCN=c1nc2ncn(C)c2c(NCCCC2CC2(F)F)[nH]1)OCC 4129,CC1(C)C(=O)CCCN1C(=O)CCOCCO 4130,N1(C(CCOCCCNC(C2CCCC2C(F)F)=O)=O)CCOC2(CCC2)CC1 4131,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CN(C(C2CCC2C)=O)CC12CCC2 4132,c1(C(=O)NC2C=CCN(C(c3nnn(C)c3C(F)F)=O)C2)ccc(C2CC2)nc1O 4133,Cc1cccc(C)c1CC(=O)NCC(c1ccc(F)cc1)NC(C1CCOC1)=O 4134,C1(C(N2CCC(N(C(=O)CCF)C)CC2)=O)COC2COCC12 4135,C1(NC(CCCC=C)=O)CN(C(=O)CN2CCN(C3CC3)C2=O)CCC1CO 4136,N1(C(C2(C)CN(C)C(=O)C2)=O)CC2CCC(CNC(C3CN(C)CCO3)=O)(C2)C1 4137,O=C(C1CCc2nccn21)N1CCCC1c1ccccc1 4138,Cc1c(C(N2CC(NC(C3CCOC3)=O)C(C)C2)=O)cccc1Cl 4139,c1(C(N2C(C)CN(C(c3ccc(C)n3C)=O)C(C)C2)=O)nccc2ccccc12 4140,C(=O)(C1=CC2(CCOCC2)C1)N1C(C(C)NC(=O)CSCCC#N)CCC1 4141,c1(COC)cncc(C(=O)NC2CCC(NC(=O)C(c3ccccc3Cl)C)C2)c1 4142,C1(C(N2CCN(C(CC3CNC(=O)O3)=O)C(CO)C2)=O)CC2C=CCC(C1)C2 4143,N1(C(c2ccc(C(C)(C)C)cc2)=O)CCCCC(NC(C2(n3cnnn3)CC2)=O)C1 4144,C1(CC(=O)NCC2(NC(C3(OCC)CCC3)=O)CCOC2)C(=O)NN=C1C 4145,c1(CCC)nc(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CC)cs1 4146,c1(OCCOC(=O)CCF)cccc(C2CCC2)c1 4147,C1(O)(CCNC(c2nncs2)=O)CN(C(=O)CC2CCC2(F)F)C1 4148,C(=O)(C1=COCCO1)N1C(CN(C(=O)CN=S(C)(C)=O)C)CCCC1 4149,c1(NC(C2(F)CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)nc2ccc(Cl)cc2[nH]1 4150,n1(CC(=O)NCC(C)OC)cc(C2CCC2)nn1.c12cn(nn1)CC(=O)N2 4151,c12cc3ccccc3nc1C(=O)NC2.c1(CC)noc(CS(=O)(=O)F)n1 4152,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)CCc2scnc2C)n1 4153,c1(CNC(C2C(C(=O)NC(C3CCOC3)COC)C2)=O)ocnc1C(N)=O 4154,C1(CCCNC(c2c(C)con2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4155,C1(CNC(c2coc(CC3(CC#C)CCC3)c2)=O)(CC(=O)N)CCOCC1.OC 4156,C(C(=O)N=S1(=O)CCC2OCCNC2C1)c1c(OCCCC)ccc(SC)c1 4157,N1(C(c2c(CC)ncs2)=O)CCC2CCCC12C(=O)N(CC(F)(F)Cl)C 4158,Cn1ncc(C(=O)NCC(C2CC2)NC(=O)C(O)Cn2cncn2)c1Cl 4159,c1(CC(=O)NCC(CNC(c2cnc[nH]2)=O)OC)ccc2ccccc2c1 4160,c1(OC)ccncc1NC(=O)C=C(C)CNC(=O)Cc1ccncc1Cl 4161,C1(CC(=O)N(CC)CC)CCCN1C(=O)C(F)n1ccnc1.C=C(C)C 4162,N1(C(c2cncc(C)c2)=O)CCC(F)(F)C(CNC(c2ncc(Cl)s2)=O)C1 4163,O=C(N=c1[nH]nc(Cl)cc1Br)C1CC(O)CN1C(=O)Cc1cn2cc(F)ccc2n1 4164,C(=O)(CCC(F)(F)C(F)F)N1CC(NC(C(c2cccc(Cl)c2)C)=O)C(O)C1 4165,CCC(CC)CCCC(=O)NC(CNC(=O)C=C(C)C)CC(C)C 4166,c1(C(C(=O)NCCCN(C(CCCOC(C)=O)=O)C)C)ccc(C)cc1 4167,c1(CONC(C2CCCN2C(=O)Cc2cc(C(C)C)no2)=O)ccccc1Br 4168,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4169,C1(CC)CCN(C(C2CC=C(C)CC2)=O)C1C(=O)NCCC1(OC)CCC1 4170,Cc1ccc(OC(C)C(=O)NCC2CN(C(=O)CCC=C(C)C)C2)c(C)c1 4171,C=CC(CC)C(=O)NC1COCCC1C(=O)N(C)CC1CCC(=O)N1 4172,C(=O)(C(O)CCC(F)(F)F)N1CCC(N(CCC)C(c2cnn[nH]2)=O)CC1 4173,c1(CCC(=O)C(CNC(C(C)C)=O)=O)c[nH]c2ccccc12.C12C3CC1N(C3)C2 4174,CCCC(CCC)C(=O)NCC1(NC(C2CCCC(O)C2)=O)CC(F)(F)C1 4175,C1(NC(c2cc(Br)co2)=O)COCCC1NC(C1(C2CCC2)CC1)=O 4176,c1(C2(C(=O)NC3CC(CNC(c4n(C)nnc4)=O)C3)CCC2)ccc(Cl)cc1 4177,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4178,C(C(=O)NC1CC(NC(c2cccc(-c3ncon3)c2)=O)C1)(C(C)(C)C)N(C)C 4179,C=CC1OCCC1C=O.N12CCCCC1CN2N(C)C(=O)C1CC1.C1CCC1 4180,C1(N(C)C)CCCN(CC(=O)NCC2(NC(C3CN(C)CC3O)=O)CCC2)C1 4181,N1(C(c2cn(CC=C)nn2)=O)CCC2CCC(NC(=O)CCCC(=O)N(C)C)C12 4182,C1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CC2(COC(=O)N2)C1 4183,c1(C(=O)NC2(CC)CN(C(c3oc(SC)nc3C)=O)C2)cccc2nn(C)nc12 4184,C1(NC(CNC(CNC(C=C(CCC)C)=O)=O)=O)CCCC1(C)CO 4185,C1(C(N(C2CCN(C)C2)CCOC)=O)CN(C(=O)CCCc2cc[nH]n2)C(C)(C)C1 4186,C1(COC(CC(c2cccc(C(F)(F)F)c2)C)=O)CC(F)(F)CO1 4187,c1(C(=O)NCC2(OC)CCN(C)C2)nc2ccccc2n1C1CC1 4188,Cc1cc(C(=O)NC2(c3cn(-c4ccc(Br)cc4F)nn3)CCC2)cc(O)c1 4189,CC1CC(CNC(=O)CCNC(=O)CO)CN1C(c1ccccc1SCC#N)=O 4190,c1(N(C(c2cccc(F)c2)C)C(=O)NC2CCOC2C(F)(F)F)cccc(Br)c1 4191,c1(C(=O)NC23C(CN(C(COCC(C)C)=O)C2)C3)ccc(-n2cncn2)cc1F 4192,N1(C(C(C)OC)=O)CCC(F)(C(=O)NCCc2cnn(C)c2C)C1 4193,S(=O)(=O)(c1cncc(C(=O)NC2C3CC2CN(C(=O)CCC(C)(F)F)C3)c1)NC 4194,c1(C(=O)NC2CCC2NC(c2ccncc2)=O)cncc(-c2cc[nH]n2)c1 4195,c12cccc(c1)C(=O)N2.c1(C2N(CC(=O)N(C)C)CC2)cccc(O)n1 4196,c1(C(=O)NCCCOCCNC(C(C(CC)O)(F)F)=O)ccc([N+](=O)[O-])cc1N 4197,C1(C(C)C)CCC(C(=O)NC2CCC2NC(c2ccc(C(F)F)cc2)=O)CC1 4198,CC1(C)CCN(CC(=O)Cc2ccc(F)cc2)C(CO)C1 4199,c1(C(=O)NCC2(CCCNC(=O)Cn3cncn3)CC2)coc2c1C(O)CCC2 4200,c1(CC)cc(C(=O)NC2CCC(NC(C3CC4CC4C3)=O)C2)cc(O)n1 4201,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2SCCS2)C2CC(O)C1C2 4202,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4203,CCC(C(=O)NC(CNC(=O)C(C)(C)OC)CC(F)(F)F)C(C)(C)CC 4204,c1(C(=O)NC2COCC2NC(C2CC2F)=O)cc2occc2[nH]1 4205,c1(-c2ccc(C(N(C(C)(C)C)CC)=O)cc2)ccc(F)c(C)c1 4206,S(=O)(=O)(c1ccc(Br)cc1NCC(C(F)F)c1ccccc1)N(C)CCOCCO 4207,Cc1ccc(C=C(C#N)C(=O)N(C(C)CNC(=O)C(C)OC2CCOC2)C)cc1 4208,C(CC(C(=O)N1OC2CCC1CC2)NC(c1cncnc1C)=O)=CC 4209,Cc1nc2cc(C(N3CC4CC3C4NC(=O)CC(C)(C)N(C)C)=O)[nH]c2s1 4210,N1(C(C2C(C)C2)=O)CCN(C(c2cnc(Br)s2)=O)C(C)C1 4211,C1(C(N(C(C(=O)NC)C)C)=O)CCC(C)(C)N(C(=O)CC2CC2)C1 4212,CC(CC(F)F)C(=O)N1C(C(=O)NCC(=O)NCC2CC2)CCC1C 4213,N1(C(C(C)N(CC(F)(F)F)CCO)=O)CCN(C(c2ccncc2)=O)CC(C)(C)C1 4214,c1(C(=O)NCC2CCN(C(C3CCC(=O)N3)=O)C23CCC3)cn2ccccc2n1 4215,N1(C(=O)NC2CC2)CCC2(CC(C(=O)NCC3CCC(C(=O)O)CC3)=NO2)C1 4216,c1(C(=O)NC2CCN(C(CCOCCOC)=O)C2C(C)C)cc(C)c(F)c(C)c1 4217,C1(C(=O)OC(C)(C)C)C2CCC(C2)C1NC(N(C1CC(C(N)=O)C1)C)=O 4218,c1(C(=O)NC(C(C)C)CCN(C)C(c2cc3n(n2)CCO3)=O)nc2ccccc2s1 4219,C(C(CC(=O)NC1CCN(c2ccc(Cl)cc2)CC1)C(F)F)OC(C)C 4220,c1(CSCCCCC(C)=O)c[nH]c2ccc(F)cc12 4221,S(=O)(=O)(c1cc(F)ccc1C)NC(c1c(C)cc(F)c(C(C)C)c1)=O 4222,C1(NC(CN2C(C)CCC2)=O)CC=C(C(=O)NCC(=O)Nc2ccncc2)C1 4223,c1(OC(F)(F)F)ccccc1CNC(c1nnnn1C1CCCCC1)C1CCSC1 4224,c1(CC(=O)N(C2CCN(C(C(n3ccc(Br)n3)C)=O)C2)C)c(Cl)cncc1Cl 4225,c1(CNCCCC(=O)NC(c2ccccc2)C)cc2ncc(Br)cc2o1 4226,C(C)(C)(CCC(=O)NC(C)C=CC(=O)NC1CC(CCO)C1)OC 4227,c1(C(=O)NCCCCCNC(Cc2nc(C)[nH]n2)=O)ncnc2sccc12 4228,S(=O)(=O)(c1ccc(N(C)CC2(C)CSC(C)=N2)c2cnccc12)NC 4229,C1(OC)CN(C(=O)C2CC2)CC1CO.C1(CNC(=O)CCNC(=O)CO)CC2CC2C1 4230,N1(C(C(C)OCCOC)=O)CCCC(N(CCO)C(c2ccnn2COC)=O)C1 4231,Cc1nn(C)c(C(=O)NCc2nc(CNC(C3CCC(=O)N3)=O)cs2)c1Cl 4232,CCC(CC(F)(F)F)C(=O)NCC(CNC(=O)C=Cc1cc(F)ccc1F)CO 4233,N(C(=NCCCCl)NCC(C(C)C)c1ccnn1C)Nc1cccc(SC)c1.CC 4234,C(C)(C(=O)N1CCN(c2nc(C)c(Br)s2)CC1)(C(C)(C)C)NC(C)=O 4235,c1(C(=O)NCC(C2CCCC2)NC(CSCCC(C)C)=O)csc(N=S(C)(C)=O)n1 4236,C1(C(=O)NC(c2occ(C(N(C3CCOC3)CC)=O)n2)C)CC(C)N(C)C1 4237,C1(C(=O)NCC(CC)(C)NC(c2cnn(CCOCCO)c2)=O)CCCN(C)C1 4238,c1(CC(=O)NCC2C(NC(CCc3cc(OC)no3)=O)C2)ccccc1C 4239,c1(OCOC)cccc(NC(c2nnnn2CC(F)F)c2ccns2)c1 4240,C(=O)(CCCCC(N)=O)NC(CC(C)NC(c1cnncc1C(F)(F)F)=O)C 4241,C(=O)(CC1=NN(C)C(=O)C1)NC1CC(C)(NC(C(CCSC)N(C)C)=O)C1 4242,Cc1cccc(F)c1C(=O)NC1CCCC(NC(c2ccc(Br)cc2N)=O)C1 4243,N1(C(C(COC)C)=O)CCCC12CCN(C(C1CCC(=O)C1)=O)CC2 4244,c1(CC)ccc(OC)c(NC2CC3CC2(CO)C3)c1 4245,c1(C(=O)NC2C(CO)CCN(C(C3NC(=O)OC3)=O)C2)cnn2c1OCCC2 4246,[N-]=[N+]=NCCCC(=O)NCC(=O)NCC(c1ccncc1)=O 4247,N1(C(C2C(C=C)C2)=O)CCC(C2(NC(=O)Cc3cc(C(F)(F)F)n[nH]3)CC2)CC1 4248,c1(C(N2C(CCNC(CC(C)n3cccn3)=O)CCC2)=O)nc(Br)ccc1N 4249,C1(NC(c2c(CC)n(C)nc2)=O)CCN(Cc2cc(Cl)ccc2Cl)C1(C)C 4250,c1(C(=O)NCCC(=C)CNC(=O)CC23CCC(CC2)C3)ccc2ncncc2c1 4251,N1(C(C(N2CCNC2=O)C)=O)CC2CC2(CNC(=O)CC2(CO)CC2)C1 4252,N1(c2cc(C)nc(Cl)n2)CC2CC1CCC2NC(=O)CC(C)C1CCCCC1 4253,CC1CC(C(=O)N(C(C)CNC(C2CCC(C(F)(F)F)O2)=O)C)CC(C)C1 4254,C1(C(=O)NCC(CC=C)NC(c2csc(NC=O)n2)=O)CCc2ccccc2O1 4255,C12(CNC(CC=C)=O)COCCN1C(=O)CN(C(C1CC1C#N)=O)C2 4256,c1(NC(c2scc(-c3ccc(OCOC)nc3)c2)=O)ccc(Cl)nc1Br 4257,C1(CC(=O)NC(C)CCNC(c2cnnn2-c2ccccc2)=O)COCCN1C 4258,N1(C(C(CC2CC2)NC(Cc2nc(C)oc2)=O)=O)CCSCCC1C 4259,n1(CC)nnc2c(N(C)C(C3CCC(C(=O)OC)O3)=O)ncnc12 4260,N1(C(COc2ccc(C)cc2)=O)CCC(C)(C)C1CNC(=O)CC1C(C)C1(F)F 4261,c1(C(N2CCC(C(C)NC(C3(CO)CCCO3)=O)C2)=O)cc2c(cn1)OCCC2 4262,c1(C(N2CCC(NC(c3ncc(CC)nc3)=O)C2)=O)cncc(F)c1C(F)(F)F 4263,CC1CN(C(C2CCC3(CCC3)O2)=O)CCN(C(C2CCCN2N=O)=O)C1 4264,C(=O)(C#CC1(C)COC1)NC(C)CC(C)NC(C1CC1C1CCOCC1)=O 4265,c1(CC(=O)NC(C(C)(C)NC(c2c(C)con2)=O)C)cc(F)cc(F)c1 4266,S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(=O)NC(C(C)C)C2CC2)C2CCC1C2 4267,c1(C(=O)NC2C(CC)N(C(c3csc(C)n3)=O)CC2)cc(F)cnc1O 4268,C1(C(C)NC(=O)CCCC2CCC2)CCCCN1C(=O)CSCc1csc(C)n1 4269,CC1(C)C(C(=O)NNC(C2COC3CC2C3)=O)(O)CCO1 4270,N1(C(C2ON=C(C)C2)=O)CCC(CN(C(=O)CCc2nccs2)C)CC1 4271,CCCC(O)C(=O)N(CC)CC1CCCN(C(=O)C(C)CC2CCCCC2)C1 4272,CCCCC(O)CNC(=O)CCN(C(=O)C(C)OCOC)C(C)C 4273,N1(C(c2[nH]n(C)c(=O)n2)=O)CCC2(C1)CN(C(=O)C(C)(F)C(C)(C)F)CCO2 4274,C1(NC(N(C)C)=O)CCCCN(N(CCCO)C2CC2)C1 4275,C(=O)(CCP(C)(C)=O)N(C(Cc1cccc(Cl)c1)C(=O)N1CCC(CSC)C1)CC 4276,N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(=O)CCC2CCCOC2)C(CO)C1 4277,c1(C(=O)NC(c2ccccc2Cl)C)cc(F)ncc1NC(c1occc1Br)=O 4278,CC1(CNC(=O)C(C2(O)CCCC2)F)CCN(C(C23CC(F)C2C3)=O)C1 4279,N1(CCC(=O)NC(CC2CN(C(C(C)NC(CC)(C)C)=O)C2)C)CCCCC1 4280,c1(C(=O)NCc2ccc(OC)nc2)c(C)nn(CC)c1Cl.N12CC(F)CC1C2=O 4281,N1(C(C(CCCC)O)=O)CC2CCC1C1CN(C(c3cc(C4CC4)no3)=O)CC21 4282,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4283,c1(C(=O)NCCN(CCC)C(c2ccc(O)c(O)c2)=O)cc2cc(C)ccc2s1 4284,CC1COCC(C(=O)NCC(C(=O)N2CCC2c2ccccn2)N(C)C)O1 4285,C1(C(N(CCC(=C)C)C)=O)CCC2(CC1)CC(NC(=O)OC(C)(C)C)C2 4286,c1(OC)cc(C(N2CCCCC2CNC(=O)C(O)C(C)OC)=O)ccc1F 4287,c1(C(=O)NCC2CC(OC)CN2C(=O)CN(C)C(C)C)ccc2c(c1)N(C)CC2 4288,C(CCCCC=O)N(C)C(C1C=CCS1)=O.C(C(F)(F)CO)N 4289,c1(CNC(C)CCCc2cccc(Cl)c2)cccc2c1OC(C)C2 4290,n1(CC(N2C(CN(C)C(C3CC(N(C)C)C3)=O)COCC2)=O)cnc([N+](=O)[O-])c1 4291,c1(CN(C)C(C2CCN2C(C2CCCC2O)=O)=O)nccn1C 4292,C=CCC(C)C(=O)N1CC(NC(c2cn(CC3CCCO3)nn2)=O)CC1CCO 4293,Cc1ccc(C(=O)NC2(CCNC(c3cccnc3N)=O)CCC2)c(Cl)c1 4294,N1(C(C2C(NC(C(C3CCC(=O)N3)C)=O)CCCC2)=O)CCC12CCCSC2 4295,Cc1n[nH]cc1C(N1CCC1CNC(c1c[nH]nc1-c1ccnn1C)=O)=O 4296,Cc1nc(N2CCCC(N(C)C(C3CC(CF)C3)=O)CC2)cc(N)n1 4297,C(CCCCC1CC1)NC(C1(n2cc(-c3csc(C(=O)O)c3)nn2)CC1)=O 4298,N1(C(COCC)=O)CC2CCCCC2(NC(c2cccc(OCC)c2C)=O)C1 4299,N1(C(c2nc(CC)oc2C)=O)CC2CC1CN(C(C1(C(F)(F)F)CCC1)=O)C2 4300,C(=O)(CC(c1ccccc1)C1CC1)NCC(C)(C)N(C(CCNC(C)=O)=O)C 4301,N1(C(CN2CCC(C)CC2)=O)CCC(NC(=O)Cc2ccc(Cl)s2)C(C(C)C)C1 4302,N1(C(CN2CCCC(OC)C2)=O)CCCC2(NC(=O)C3=CCOCC3)CC2C1 4303,c1(CC(N2CCC(F)C2)=O)cnn(-c2ccccc2)c1.C12CC(C1)C(=O)N2 4304,c1(CC(C(=O)NCC(C)NC(=O)CCC(N)=O)C)ccc(O)cc1 4305,CCC(C)CCC(O)CC(=O)NC1(CNC(C2CCCN2CC(C)C)=O)CCC1 4306,C#Cc1cc(C(C(=O)NCC2CCOC2)N(C(C)CSC)CC)cc(Br)c1 4307,N1(C(C(C)=C(C)C)=O)CCC(C)N(C(c2ccc(N(CCO)CCO)cc2)=O)CC1 4308,C(C(CC1CC1)C(=O)N1CC(CO)CC1CO)NC(C1CC(N(C)C)C1)=O 4309,c1(CC)ccc(C(=O)NC2CC2CNC(=O)C(CO)NC(N)=O)cc1S(C)(=O)=O 4310,c1(OC)cccc(F)c1CC(=O)NCc1csc([N+](=O)[O-])c1 4311,c1(C(=O)NC2CC(F)(CNC(C3CCC4CCC3O4)=O)C2)c[nH]cc(F)c1=O 4312,CCCCCC=CCC(=O)NCCOC1CN(C(c2cc(C)no2)=O)C1 4313,N1(C(CCC(C)OC)=O)CCC2(CC1)COC(CNC(=O)C(F)n1cccn1)C2 4314,Cc1ccc(C(N2CCC(C(C)C(=O)NC3CCCCC3)C2)=O)cc1C#N 4315,C1(NC(=O)C=Cc2ccc(C(F)F)o2)CN(C(=O)C#CC2CC2)CC2(CCC2)C1 4316,C(CC(C)(C)CO)NC(c1n(C(CC)C)nnn1)c1cnn(C2CC2)c1 4317,C(=O)(CC(=O)O)NC(C1CCN(C(c2sccc2CO)=O)C1)C 4318,CC1CCC(C(=O)Nc2csc(C(N)=O)c2)N(C(C2CN(C3CC3)C2)=O)C1 4319,CCCC(CNC(=O)C(C)(C)CSC)C(=O)NC(c1ccncc1)C 4320,Cc1nn(C)cc1CC(=O)NCC1COCCN1C(C1CC(CC(F)(F)F)C1)=O 4321,C(=O)(C(C)(C)Cn1cccn1)NCC1CN(C(C(C)c2ccsc2)=O)C1 4322,C1(NC(CC=C)=O)CC(CO)N(C(c2cncc(-c3cccc(F)c3)c2)=O)C1 4323,C1(C(=O)NC2CCN(C)C(=O)C2)CC12CCN(C(C1C=CCC1)=O)CC2 4324,c1(C(C)C)ccc(COC)cn1.C(C(=O)NCCN(C)CC)OCCOCC 4325,C(=O)(CCCN(C)C(c1cc[nH]c1)=O)NCCSC 4326,N1(C(CN2C(C)CN(Cc3ncccc3Cl)CC2)=O)CCC2(CC1)C(F)(F)C21CC1 4327,C(=O)(C(C)(C)S(C)(=O)=O)N(C)CCN(C1CCCO1)C(c1cc2c(s1)CCC2=O)=O 4328,C#CC1(O)CCCC(NC(=O)NC(c2ccnc(F)c2)C)C1 4329,c1(CC(=O)NCC(F)CNC(c2coc(Cl)n2)=O)cccc(N2CCOC2=O)c1 4330,c1(C(=O)NCC(C)NC(C2CCCN2C(=O)C2CC2)=O)n[nH]c2ccccc12 4331,c1(NC(C2C(NC(C(CC)O)=O)C2)=O)cc(Cl)c(Cl)c(Cl)c1 4332,c1(C(=O)NC2C(NC(c3cnc(C(C)OC)s3)=O)CC2)c(C)cc(O)cc1C 4333,c1(C(=O)OC)ccc(NC(=O)NCC(C)=CCNCc2cccs2)cc1 4334,Cc1c(C(=O)NC2CN(C(=O)CCc3nc(=N)[nH][nH]3)C3CC23)c(C(F)F)nn1C 4335,c1(N(CCCNCCF)C(CC2C(C(=O)OC)CCCC2)=O)ccc(C#N)nc1 4336,C1(N(C)C(c2cc(F)ccc2F)=O)CN(C(=O)CN2CCS(=O)CC2)CC1(C)C 4337,CC1(C)CC=CCN(C(C23CCC(C2)N(C(=O)CC2CC4C=CC2C4)C3)=O)C1 4338,c1(C(N2CCC(O)(CNC(c3c(CC)n(C)nc3)=O)C2)=O)c(C)ccc(C)c1C 4339,CC1CCC(C2CCC2)CN1C(=O)NCCCc1cccc(Cl)c1 4340,C1(C(=O)Nc2cn(C(C)CN)nn2)CCOCCN1C(C1CCCOC1)=O 4341,C(CC(C(F)F)c1ccccc1)N(c1nnnn1C1COC1)CCC(C)C 4342,c1(SCC)nc(Cl)cc(=NCC(C2CCCC2)NC(=O)CSC)[nH]1 4343,C(CCC(C)C(=O)NCC12CCC(CC1)N2C(=O)CCC1CC1(C)C)OC 4344,C1(CNC(c2c(COC)onc2)=O)(NC(=O)COCCCF)CCCCC1C 4345,c1(C(=O)NCC2C3CN(C(C(c4cn(C)nc4)O)=O)CC32)ccc(F)c(F)c1N 4346,c1(SC)ccc(NC(C2CC23CC(NC(c2cc(COC)[nH]n2)=O)C3)=O)cc1C 4347,c1(CC(=O)NC2CC(C(=O)Nc3c(C(=O)OC(C)C)ccs3)C2)ccnc(Br)c1 4348,C1(C(=O)NCCSCC(=O)NC(C=C)(C)CC)CCC(COC)CC1 4349,c1(SCCNC(c2c(C)occ2)c2nnnn2C)ccccc1F 4350,C(CN=c1ccnc(NCCc2cccc(F)c2)[nH]1)NC(c1cncs1)=O 4351,c1(C(C(=O)NC(C)C)N(CC(C)C)CC)cn(CC(F)F)cn1 4352,c1(CN2C(C(=O)NC(c3ccccc3)C)CC(C)C2)c(Cl)cc(O)cc1Cl 4353,C1(C(N2CCC(Cl)C2)=O)CC2OCCC2N(C(c2ccccc2)=O)C1 4354,N1(C(CC(C)N(C)C)=O)CCCOC(CNC(=O)C(C)(C)C(=O)N(C)C)C1 4355,Cc1cccn2c(C(=O)NC(C3CCN(C(c4coc(O)n4)=O)C3)C)cnc12 4356,c1(N2C(C)(C)C(NC(=O)CCC[N+](=O)[O-])CC2)ccc([N+](=O)[O-])cc1CO 4357,C1(=O)CCCCCCCC23C(C(=O)OC)(CN1C2)C3.C(C)(C)(C)NC(=O)OC 4358,CC1(C)COCCC1Sc1cccc(-n2cc(-c3nccs3)nn2)c1 4359,c1(OC)ncccc1C(N1CC(F)CC1CNC(C1CC2(CC2)CO1)=O)=O 4360,Cc1cc(=O)oc2cc(OCCN(c3cccc4c3SCCC4)C)ccc12 4361,C1(CNC(=O)Nc2ccc(CNC(CNC=O)=O)cc2)CC2CC1CC2O 4362,CCC(CC)CCCC(=O)NC(C)CCCCNC(=O)CCCCN(C)C(C)=O 4363,C1(NC(c2ccc(C)c(O)n2)=O)CC2CCC1N(C(c1coc(C#N)c1)=O)C2 4364,C=C1c2ccccc2C(=O)N1C(C)C(=O)NC(C)CN(C)C(C1(C)CC=CC1)=O 4365,C1(C)(C(=O)OC)C=CCN1C(=O)C(CCSC)NC(=O)C=Cc1ccn(C)c1 4366,C1(CNC(C(CNC(CN(CC)CC)=O)C)=O)CC1C1CCCC1 4367,CCC(C)CC(C)C(=O)N(CC(CO)(CO)NC(c1ccnc(OC)c1F)=O)C 4368,C12(C(=O)NCC(CC(C)C)(C)NC(=O)CSC3CC3)CCCN1S(=O)(=O)CC2 4369,C1(COC)(CNC(C2CCC2C#N)=O)CN(C(=O)Cn2[nH]cnc2=N)C1 4370,CC(CC(=O)NCCN(C(C1CC1C(F)(F)F)=O)C1CC1)n1cc(Br)cn1 4371,CCCC(CCC)C(=O)N(C)CC1CCN(C(=O)CNC(c2cccnc2)=O)C1 4372,N1(CC(=O)NCC(C2CCC2)NC(=O)CSCC2CCCO2)CCC(=O)NC1=O 4373,Cc1c(NCc2cn[nH]c2)ncnc1N1CCN(c2cccnc2)CC1 4374,N1(C(C(C=C)O)=O)CC2(CCN(C(C3CC(C(F)(F)F)C3)=O)CC2)C1C(C)C 4375,c1(SC)cccnc1C(N1CC(O)(C(C)(C)CNC(c2ccccc2F)=O)C1)=O 4376,N1(C(CCCN(C)C)=O)CC2CCC(C1)N2C(c1cc(=O)n(C)o1)=O 4377,c1(OCCC(=O)NC2CC(CO)N(C(=O)CCCC3CC3)C2)cccc(Cl)c1 4378,N1(C(CC(COC)C)=O)CCC2CCC(C1)N2C(=O)CC(C(C)C)OCCOCC 4379,N1(C(COCCN(C(=O)CC2OCCO2)C)=O)CCC2CCCC2CC1 4380,C(CC(O)C(=O)N1CCCCC1CN(C)C(c1cccc(C2CC2)n1)=O)SC 4381,N1(C(CNS(N(C)C)(=O)=O)=O)CC2COCC(C1)C2NC(C1CCC(=O)N1)=O 4382,C1(C(N2C(CCNC(c3ccon3)=O)CC(F)(F)C2)=O)CC2COCC(C1)C2 4383,CC1=CCSC1C(=O)NC1(C)CC(C(=O)NC(CCC2CC2)CO)C1 4384,C(=O)(CCS(C)(=O)=O)NC1CC(NC(CC(C)C2CCCC2)=O)CC1O 4385,C(C1CCCCC1)=CC(=O)N(C(C(=O)N(C(C)CC(N)=O)C)C1CC1)C 4386,N1(C(c2cn(CC)nc2C)=O)CC(F)(F)CC1CNC(c1cc(F)ccc1F)=O 4387,c1(C(N2CCC(NC(C3(C)CSC3)=O)C(O)C2)=O)c[nH]c2ccncc12 4388,C1(COC)(NC(C2Cc3nnsc3S2)=O)CCC(C)(C)CC1 4389,Cc1ccc(CSC(C(N2CCOC(CSCCC#N)C2)=O)C)cc1 4390,c1(C(=O)NCC(CNC(CC2(C)CCCCC2)=O)F)nccc2c1CNC2=O 4391,C(=O)(NNC(=O)C(C)(C)CCCCNC(C(CC)C(C)C)=O)C1(SC)CC1 4392,c1(N2C(C)CC(CNC(=O)CC3CCC(O)C3)C2)ncnc2[nH]ccc12 4393,C1(NC(c2[nH]cc(CC(C)C)c2)=O)CN(C(c2cc(=O)n(C)o2)=O)C2(CCC2)C1 4394,C1(C(=O)NC(C(C)(C)C)CNC(=O)CNC(=O)C2CC2)CCC2C(CC1)C2(F)F 4395,Cc1ccc2ncc(C(N3CC(F)(CNC(=O)CC4CCCCC4O)C3)=O)n2c1 4396,CN=c1nc(C(N2CCN(C(c3conc3C3CCC3)=O)C3CC23)=O)cc(C)[nH]1 4397,c1(SCC(N2CCCCC2)=O)nnc(-c2ccsc2)n1C1CC1 4398,N1(C(CC(C)C)=O)CCC(CNC(C2(CN(C)C)CCOCC2)=O)C(C)C1 4399,N1(C(C2(CC)CC(C)(C)C2)=O)CCN(C(C2(C)CCCS2)=O)CC1CC 4400,CCCC(CC)CCC(=O)NC1C=CCC(C(=O)NCc2ccc(O)cc2)C1 4401,C1(NC(C(c2n(C)ncc2)(F)F)=O)C2CCC1N(C(=O)C(CCO)N(C)C)C2 4402,c1(C(=O)NCC2C(NC(C)=O)CC2)cc(C)c2n[nH]cc2c1 4403,Cn1c(C(N2CCN(C(c3cccc(CO)n3)=O)CC2)=O)cnc1O 4404,c1(C(C)C)nn(C)cc1C(=O)NCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 4405,C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(=O)Cc2c(F)cccc2Cl)CC1 4406,S(=O)(=O)(c1ccc(Br)c(C(=O)OC)c1)NC(CCCCC=C)=O 4407,c1(CC(N2CCC(NC(=O)CC3CC4CC4C3)C2)=O)cccc(Br)c1Cl 4408,N1(C(c2c(C)cccc2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC2(CCC2)C1 4409,c1(C(=O)NCC2C(CNC(C3(C(C)(C)O)CC3)=O)C2)ccnc2[nH]c(O)nc12 4410,N1(CC(=O)N(C2CCCCC2)CCNC(C2CCC(CC)O2)=O)CCNC(=O)C1 4411,C1(NC(Cc2nnc(C)s2)=O)CCC2CN(C(C3CCS(=O)(=O)C3)=O)CCC2C1 4412,c1(C2(C(N(CC(C)NC(CCCOC(C)=O)=O)C)=O)CC2)ccc(Cl)c(F)c1 4413,N1(C(C#CC)=O)CC2CN(C(=O)Cc3ccc(OC)c(O)c3)CC2C1 4414,c1(C(=O)NC)ncccc1NC(c1cn(CC(F)F)nn1)=O 4415,c1(C(C)NC(CN(C(C2CC(OCC)C2)=O)CCO)=O)nccc(O)n1 4416,N1(C(CN2C(C)CC2)=O)CCC2(C1)CN(C(c1ccc3nccn3c1)=O)CCO2 4417,N1(C(C(C)OC)=O)CCC(C(C)(C)NC(C2CC2C)=O)CC1 4418,C1(NC(C(C)SCCCC)=O)CCN(C(c2cc(=O)c(OCC)c[nH]2)=O)CC1C 4419,C12(NC(CN(C(=O)OC)C)=O)CCC(CC1NC(c1sc(C)nc1C)=O)C2 4420,C(=O)(CCC(C)=O)N.C1(C=O)(SC)CN(N2CC(C)(C)C2)C1 4421,CC1(C#N)CCCN(C(C2CCC=CC2NC(c2cncs2)=O)=O)C1 4422,c1(C(N2CC(N(C)C(c3ccc(C(N)=O)cc3)=O)C2)=O)ccc(=O)n(C)c1 4423,CC1(C)CCC(NC2CCC3(CC2)CN(C(=O)C(N)=O)CCO3)c2ccccc21 4424,N1(C(C2CCCC2)=O)CCN(C(C23CCN(CC2)CC3)=O)CC1CF 4425,Cc1cc(NCCCn2cncn2)nc(N(C)CCF)n1 4426,c1(CNC(CC(C)NC(C(CC=C)C)=O)C)ccc(Br)c(C(=O)OC)c1 4427,N1(C(Cc2cc(C)no2)=O)CC2(C1)CN(C(C1CCC(C)(C)CC1)=O)C2 4428,C(=O)(C(CC)C(=O)OCC)N1C(C(=O)NCC(=C)CC)(COC)CCC1 4429,C(=O)(C(C)C(C)(C)C)NCC1(O)CC(NC(C(C)C2CCC2)=O)C1 4430,Brc1cccc2[nH]c(CCc3nc(-c4cc5c(s4)CSC5)no3)nc12 4431,C1(NC(c2cnc(Cl)[nH]2)=O)CCN(C(c2nccnc2C(N)=O)=O)CC1F 4432,c1(CN2C(C(N(C(C3(C)CC3)C)C)=O)CC2)cc(I)ccc1O 4433,C1(C(=O)NC(CCC=C)C)CCC(NC(=O)C(O)CN2CCCC2)CC1 4434,N1(C(CN(C(=O)Cc2nncn2C)C(C)C)=O)CCC(CO)C(O)C1 4435,n1(CC(N2CC(CC)C(NC(=O)CNS(N)(=O)=O)C2)=O)nc(Cl)ccc1=O 4436,N1(C(C(C)OCOC)=O)CC2CC(N(C)C(c3cc(C)ccc3Cl)=O)C1C2 4437,C1(C(=O)NC(C)(C)C(=O)N2CC(C(N3CCCC3)=O)C2)(CC)CNCCO1 4438,CCS(=O)(=O)CC(=O)N1CC(C)CCC1C(=O)NCCC1CC=CCC1 4439,C1(C(=O)NCC2(F)CC(CNC(c3c(C)con3)=O)C2)CCCCC1F 4440,c1(CCC(=O)N(C2CCN(C(c3[nH]cc(C)c3C)=O)C2)CC)ccc(F)cc1F 4441,N1(C(C2(NC(C3CCOC3)=O)CC2)=O)CCC(CSCC)CC1C 4442,C1(C(N2CCC(OC)(CNC(c3cncc(CO)c3)=O)C2)=O)CC(=O)NC(=O)N1 4443,CC1(C)CCC(CC(=O)NCC(=C2CN(C(=O)Cn3ncnn3)C2)F)OC1 4444,Cc1cc(NC2CCC(NC(=O)C(C3CCC(=O)N3)C)CC2)n2nc(C)nc2n1 4445,N(C)(S(=O)(=O)N(C)C)CC(N1CC(CC)(NC(c2ncsc2C(F)(F)F)=O)C1)=O 4446,CCC(CNC(c1cccc(O)n1)=O)(CC)C(=O)N1CCC(N(C)C)C1 4447,N12CCCC(C1)SCC2=O.C1(C=O)CCC(c2ccccc2)CC1.O=CC1CC1 4448,C(CCCC(C)(C)C(=O)NNC(=O)C12CCCC1C2(F)F)NC(CC)=O 4449,c1(N2CCC(n3c(C)ccc3C)CC2)[nH]c(=NC(C)C(C)F)nc2sccc12 4450,C(=O)(C(C(C)C)C1CCC1)NC1(CC=C)CN(C(c2cnc(N(C)C)o2)=O)C1 4451,Cn1ncc(C(=O)NCc2ccc(Br)cc2Cl)c1C#N 4452,c1(C(=O)NC(C)C(N2CCN(C(c3cncnc3)=O)CC2)=O)ccc(F)cc1F 4453,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3cnnc3O)C2)=O)CCCCC1 4454,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4455,C1(CNC(C2C(OC)CCC2)=O)CC(C)N(C(=O)Cc2cnn(C)n2)C1 4456,c1(C(=O)NCC(C)NC(CCC(C)c2ccccc2)=O)cc2ccccc2n1C 4457,C(=O)(C(C(C)(C)O)NC(=O)C(C)=C1CCCC1)NCCC(CC)C 4458,c1(CC(=O)N(CC(CC)NC(C2(CCCC)CC2)=O)C)cnc2ccccn12 4459,C1(C2CCN(C(c3cn(C)nc3O)=O)CC2)(NC(C(CC(C)C)NC(C)=O)=O)CC1 4460,c1(CC(=O)NCC(CN(C)C(C2CCC(=O)N2)=O)O)cncn1C 4461,CC(C)C(CCN(C(=O)CC1C(C)C1(F)F)C)NC(c1cnc(S)n1C)=O 4462,c1(OC)cncc(C(=O)NC23CC2CN(C(c2cccc(N(C)C)n2)=O)C3)n1 4463,C(N=c1ccnc(N2CCCC3(CC2)CC3)[nH]1)c1c(C)n[nH]c1 4464,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CN(C(c1ncccc1N)=O)CCO2 4465,c1(NC(C)=O)ccc(C(=O)NCC2CC2(C)CNC(c2cc(Cl)c[nH]2)=O)cn1 4466,O=C(C1CCCc2ccnn21)NCC1CN(C(c2cnc(O)nc2Cl)=O)CCO1 4467,N1(C(C2C(C(=O)OC)CC2)=O)CCOC(CCNC(=O)C=Cc2cocn2)C1 4468,c1(C(=O)NC(C2CCOC2)CNC(C(C)(C)C(N)=O)=O)csc2c(F)cccc12 4469,CC1CCN(C(=O)C(N2CC3CCC2C3)C)CC1CNC(c1cc(Cl)c[nH]1)=O 4470,c1(NCc2c(O)cccn2)[nH]c(=NCCC2CCC(F)(F)C2)nc2scnc12 4471,C1(C(N2CCC(CN(C)C)C2)=O)CN(C(C2CCC(=O)O2)=O)CC(C)(C)C1 4472,N1(C(CC2C(=O)NCCC2)=O)CCCC(Cl)(O)CC1 4473,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4474,CN1C2(CCN(C(c3cnnc(O)c3)=O)CC2)C(C(C23CCC2C3)=O)CS1(=O)=O 4475,C1(C(=O)NCC(C2CCC2)NC(c2cc(C)sc2)=O)COCCN1C(N)=O 4476,C(=O)(C(CCC(C)C)NC(=O)C=C(C)C(C)(C)C)N1C(CC)CCC1 4477,N1(C(C(Cc2ccsc2)NC(c2cnnn2C2CC2)=O)=O)CCC12CCCC2 4478,n1(CC(N2CC(C(=O)N(Cc3onc(C)n3)C3CC3)C2)=O)nc(C)cc1C 4479,CCC(C)(CO)NC(=O)COC1CC(NC(=O)CC2CCC(=O)N2)C1 4480,c1(N2CCC(c3cc(F)c(OC)c(F)c3)C(C)CC2)ncc2cc(Br)cnc2n1 4481,N1(C(CCNC(=O)OC(C)(C)C)=O)CCC=CC1NC(C12CCCC1C2)=O 4482,Cn1nc(C(N2CC3CCC(C2)N3C(c2ccc(Cl)s2)=O)=O)c2cc(Br)ccc12 4483,c1(C(N2CC3CCC3(C(=O)NCC3(F)COC3)C2)=O)ccc(F)cc1[N+](=O)[O-] 4484,C1(C2CCN(C(=O)OC(C)(C)C)C2)(NC(=O)CNC(N(CC=C)CC=C)=O)CC1 4485,C1(CCC(=O)NCC(CO)NC(=O)CSc2nncn2C2CC2)CCC(O)CC1 4486,C1(COC)(CNC(=O)Cc2cnn(CC)c2)CCN(C(c2nc(C)no2)=O)CC1 4487,N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3cc(-c4ccc(F)cc4)sn3)C2)C1 4488,Cc1cnc(C(=O)NC2CN(C(c3cnnc(O)c3)=O)CC2F)c(Br)c1 4489,N1(C(C2=NOC(C)C2)=O)CCC2(C1)CN(C(=O)CCC1CCCCO1)CCO2 4490,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2(CC3CC3)CC2)=O)CC(C)C1 4491,C(=O)(CCCC(=O)C(C)(C)C)N(CC(C)NC(C1(CF)CC1)=O)C 4492,c1(C(N(CCNC(C(C)P(C)(C)=O)=O)CC2CC2)=O)cnc2ncnc(O)c2c1 4493,c1(NC(CC2C(NC(C(CCSC)O)=O)CC2O)=O)cc2n(n1)CCO2 4494,N1(C(C2(C)CCN2C(=O)C(N2CCOCC2)O)=O)CCCNC(=O)CC1 4495,CCCC(CCCNC(c1ncccc1C(F)(F)F)=O)NC(C1(F)CCC1)=O 4496,C1(C2CCN(C(=O)C(F)(F)C3(O)CCCC3)CC2)(NC(C(C(CC)C)O)=O)CC1 4497,C1(CNC(C2(COC)CCCO2)=O)CC2COCC2N1c1nc(Cl)ncc1F 4498,C1(N=[N+]=[N-])(C(N(C(C#C)(C)C)C2CC2)=O)CCN(C(=O)CN2CCSCC2)C1 4499,c1(NC2CC(SC)C2)cc(NC(=O)C(C)(C)C2CCCCC2)ccc1Cl 4500,c1(-n2ncc(CN(C)C(=O)Nc3ncc(C(F)(F)F)s3)c2)ccccc1O 4501,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4502,N1(C(C(C)CCc2ccccc2)=O)CCN(C(c2cnn(C)c2)=O)CC(C)(F)C1 4503,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4504,C(=O)(C1=CCCC1(C)C)N1CCC(C(C)(C)NC(c2n(CC)cnn2)=O)C1 4505,C1(NC(c2c(CC)noc2)=O)CCCN(C(=O)CCC(=O)N(C)CC)CC1F 4506,CC(N=c1cc(NCc2nnc(O)o2)nc(C(F)(F)F)[nH]1)c1ccccc1 4507,CC(C)C(C(=O)NCCc1ccncc1)C(C)NC(C1CC(=O)C1)=O 4508,C(=O)(CCN(OC)C(=O)C(C)N(C(=O)C(C)C#N)C1CC1)OC 4509,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4510,CC1(C)OC(=O)CC1C(N1CCN(C(=O)Cc2ccc(Cl)s2)C(CF)C1)=O 4511,Cc1ccsc1C(=O)NCc1cc[nH]c1C(=O)NC(C12CC(CO1)C2)C 4512,c1(NC(c2c(C)scn2)=O)ccc2ccnc(NC(=O)C(C)(C)F)c2c1 4513,c1(CC(N2CCCC(CNC(c3c(C#N)nc[nH]3)=O)C2)=O)cc2ccccc2o1 4514,n1(CC)c(C(=O)NCCC(O)CNC(=O)C(C2CCCCC2)OC)cnc1O 4515,C(=O)(CCCCCNC(c1cn(C2CC2)cn1)=O)NCC(CCCC)O 4516,C1(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C2CC1CN(C(c1cncn1C1CC1)=O)C2 4517,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)Cc2cnc[nH]2)C1(C)C 4518,c1(CC(C)OC)nc(-c2ccc(C3CCOC3)cc2)n(C2CS(=O)(=O)C2)n1 4519,N1(C(C(C)(O)C(F)(F)F)=O)Cc2ccc(O)cc2C1 4520,C=CCC(C)C(=O)NCC1(C)CC(NC(C2CCCC(C(F)(F)F)C2)=O)C1 4521,C(N=C(NCC1(C)CCCS1)NC1CCCC1)C1CCN(C(C(C)(C)C)=O)C1 4522,c1(CC)cccc(C(N2CCC3C(NC(c4csnc4C)=O)C23)=O)n1 4523,C1(C)(NC(C=CC=CCC)=O)CC(NC(=O)C=CC(=O)OC)C1 4524,CCC(CNC(=O)C(C1CCOC1)NC(c1ccc(Cl)s1)=O)CCO 4525,C(CC(=O)N1CCC(C(=O)NC(CO)C(C)O)O1)OC(C)C 4526,N1(C(c2cn(CCCC)nn2)=O)CCOCC(CNC(=O)C(O)C(C)(C)C)C1 4527,N1(C(c2nc(CCC)sc2)=O)CCC2(CCCN2C(=O)CCC2CCCCO2)C1 4528,C12(C(=O)NC(CC3CN(C(C(=O)NCCOC)=O)C3)C)CCCC1C2(F)F 4529,C1(C(=O)O)CC12CN(C(c1cccc(Cl)c1)c1ccccc1)C2 4530,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCOC3)=O)C1C2 4531,Cn1ncc2cccc(CN(C)CC#N)c12.C12CCC(OC1)C(=O)N2 4532,c1(NC(CCC)CO)cc(F)cc(I)c1 4533,n1(C(C)C)nncc1C(=O)NCC(C)NC(=O)C(C)(C)c1ccsc1 4534,C1(NC(c2ccc(Cl)cc2)=O)CCCC12CCN(C(c1ncc(F)cn1)=O)C2 4535,C(=O)(C1=C(C)OCC1)NCC1(CNC(C2C(CC)C2)=O)CCOCC1 4536,N1(C(C(CC)OC)=O)CCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 4537,N1(C(c2cscc2Cl)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(CCO)C1 4538,N1(C(Cc2cn(C)nc2Cl)=O)CCCC(NC(=O)C(C)(C)C2CCC2)CC1 4539,c1(C(=O)NC(CC2(C)CN(C(=O)CN)C2)=O)ccc(O)c(C(N)=O)c1 4540,Cc1sc(Cl)c(C(=O)NC(C2(CNC(=O)CCCC#N)CC2)C)c1C 4541,N1(C(C(C)(C)OCC)=O)CC23CCCCC2(C1)CN(C(c1cscc1Cl)=O)C3 4542,Cc1ccc(C(C(=O)NCC(C)(C)CNC(c2cc(Br)n[nH]2)=O)C2CC2)cc1 4543,C(C)(C)(C(C)CC(=O)NCC(O)C(F)F)NC(C(N1CCOCC1)C)=O 4544,C1(N(C)C(C2(C)CC2)=O)CCCC1CNC(c1cncn1C1CC1)=O 4545,C(=O)(CS(C)(=O)=O)C(CSCC(=O)N(C(C)(CN)C1CC1)C)=O.c1(N)ccccc1Cl 4546,C(=O)(C1CCc2ccccc21)NCCCCNC(=O)CC1CC1C(F)(F)F 4547,c1(C2(C)C(C(=O)NCC3(C)CCCS3)C2)cccc(Br)c1 4548,C1(NC(c2c(C)noc2)=O)C=CCCC1C(=O)NCC(F)(F)Cl 4549,C1(C(=O)NCCC2CN(C(C3N(C)CCC3)=O)C2)CCC(NS(C)(=O)=O)CC1 4550,CC1(C)CCN(C(C2(C(N)=O)CCC2)=O)CC1CNC(C1CCC=CCCC1)=O 4551,c1(C(N2C(CNC(C(C(C)(C)C)OC)=O)C(C)(C)CC2)=O)cc2n(n1)CCCC2 4552,N1(C(C2(CC)CCNC2=O)=O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1C 4553,c1(NC(C(CO)NC(CC2C(CC)C2)=O)=O)cnc(C)c(C#N)c1 4554,C1(NC(C#CC2(C)CC2)=O)CN(C(c2ccc(CSC(F)F)o2)=O)CCC1F 4555,c1(OC)ccc(Cl)c(C)c1C(=O)NC1CCCCN(C(c2ccc(F)o2)=O)C1 4556,c1(OC)cc(C(=O)NCC2CC(C)N(C(=O)C(O)CSC)C2)cc(F)c1F 4557,N1(C(c2c(NC(c3n[nH]c4cccnc34)=O)c[nH]n2)=O)Cc2cccc(Br)c2C1 4558,C#Cc1cncc(NC(=O)C(CNC(=O)C(c2ccccc2)C)CC=C)c1 4559,C1(CNC(Cc2c(C)noc2)=O)C2CN(C(c3cccc(C(C)(C)C)c3)=O)CC12 4560,C(=O)(CCNC(=O)C(C)NC1CC1)N(C(=O)C=CC1CCC1)CC 4561,Cc1cccc(Br)c1C(=O)NC(C)C(=O)N(C)Cc1ccc(Cl)nc1 4562,c1(OC(C)C)ccc(Cl)cc1C(=O)NCC(O)CNC(=O)CC12CCC(CC1)CC2 4563,c1(C(C(=O)NCC(C)N(C(=O)CC2CCCCN2C)C)C)cccc(F)c1 4564,C(=O)(C(C)(CC)CCC)NC(CCC)C(N1CCOC(CC)(CC)C1)=O 4565,c1(C(N(CC(CN(C)C(c2ccc(O)nc2)=O)O)C)=O)ccc2oncc2c1 4566,Cc1sncc1C(N1CC(c2ccccc2)(NC(C2CCCN2C)=O)C1)=O 4567,N1(Cc2n(CC)nnc2C)CCc2ccccc2C1CNC(=O)C(C)CC1CC1 4568,N1(C(C(C)(O)C2CCC2)=O)CCCC(NC(=O)C(F)CC2CCCC2)CC1 4569,c1(C(=O)NC2CN(C(C3C(C(C)C)CCC3)=O)CC2(C)C)cnc2ccoc2c1 4570,N1(C(C(C)C#N)=O)CCC(C(F)(F)F)CC1CNC(c1ccnc(S)c1)=O 4571,C1(C)CC(O)C12CCC2.N1(C(C(C)=C(CC)C)=O)CC2(C1)CC(=O)N2 4572,CCC(C)CCC(O)CC(=O)NCCCN(C)Cc1cn(C)ccc1=O 4573,c1(CNC(C=CCCC)=O)cccc(Oc2ccc(C(C)(C)C)cc2)n1 4574,CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)CCc2nncn2C)C1 4575,C1(C(N2C(C)CC(CCNC(C3CCC3)=O)CC2)=O)CCc2nnnn2CC1 4576,N1(C(C2CC(=C)C2)=O)CCOCC1CN(C)C(C1(C(N)=O)CC1)=O 4577,c1(C(=O)NC2CN(C(C3CCO3)=O)CC(O)C2)nc2ccc(Br)cn2c1Cl 4578,N#Cc1cccc(NC(C2C(C(N3CCC3c3ccccc3)=O)C2)=O)c1F 4579,C(CCCC(C)c1ccccc1)SC.N12CCCC1CN(C1CC1)CC2=O 4580,C1(c2n(C)ncc2)CN(C(=O)CSS(C)(=O)=O)CCN1C(=O)CC12CC(C1)C2 4581,c1(CC(N2CCC(C(C)NC(C3CCC4CC34)=O)CC2)=O)ccc2n[nH]cc2c1 4582,C1(C(=O)NCCC(C)C)CCC(NC(C2CCN(C)C2)=O)CC1 4583,c1(C(=O)NC2C(CNC(c3ccc(C(C)(C)C)cc3)=O)C2)ccc2cnnn2c1 4584,c1(C(N(CC(=O)NC(C)CCC=C(C)C)CCOC)=O)sc(F)cc1C 4585,Cc1nc([N+](=O)[O-])cn1CCC(=O)C(N1CC(C)C2(C1)COC2)=O.C(C)(C)(C)O 4586,C(=O)(C(O)C(C)(C)C)N1CC(C)C(n2cc(-c3ccc(Cl)s3)nn2)C1 4587,C1(NC(c2c(C)nccc2)=O)CN(C(=O)C=Cc2ccc[nH]2)C2(CCCC2)C1 4588,C1(NC(c2n(C)c(C#N)cc2)=O)CCCC12CN(C(=O)Cc1cnccn1)C2 4589,C(CC1=CCN(C(C2(O)CC2)=O)CC1)NC(c1cnn(CCC)c1CC)=O 4590,C1(NC(c2c(C)oc(CNC(C3C(C)(C)C3(F)F)=O)n2)=O)CCC(N=[N+]=[N-])CC1 4591,C(=O)(C(C)(C)C(F)F)N(C)CC1N(C(C(C)CCO)=O)CCCC1 4592,C1(c2ccccc2)(C(=O)NCC(CC)NC(=O)C(O)C(C)SC)CCCCO1 4593,CCCC(C(=O)OC)N(C)N1CC(C)CC1CNC(=O)OC(C)(C)C 4594,N1(C(C2(CC=C)CCC2)=O)CCC(CNC(c2cnc(C)nc2CC)=O)C(C)C1 4595,c1(C(=O)N(C2CCOC2)CCN(C(CN(C)C)=O)CCCN(C)C)nonc1N 4596,c1(C(N2C(C(=O)Nc3cc(C)c(Br)cc3F)CSCC2)=O)ccc2c(c1)OCO2 4597,C(CCCCCN)N1C(=O)CSC1.C(=O)(CC(C)(C)C)NC(C(=O)OC)CO 4598,c1(CC(=O)NC2CC(C)(NC(=O)CC3(O)CCOC3)C2)ccc(F)c(F)c1 4599,c1(CC)ncc(C(=O)NC2CCN(C3CCN(C4CCOCC4)C3=O)C2)c(C)n1 4600,C=C(CNC(c1ccoc1CC)=O)CCNC(c1cscc1F)=O 4601,c1(CNC(C2CCN(CCCN3CCC(C(=O)O)C3)CC2)C)n[nH]c2ccccc12 4602,N1(C(=O)OC)CC(CNC(c2cc(C)c(-c3ccccc3)s2)=O)C(O)C1 4603,c1(SC)cc(C(N2CCCC(N(C(=O)Cc3[nH]cnc3C)CCF)C2)=O)ccn1 4604,C1(CNC(C2CCOC2)=O)CN(C(=O)CSc2ccccc2)CC1CC(F)(F)F 4605,N1(C(c2cc(C(C)C)nn2C)=O)CC2CC1CC2NC(=O)Cc1ccc(Cl)nc1 4606,c1(C(=O)NC2CCN(CCNC(C(CC)(C)O)=O)CC2)cc(C)cc(O)c1 4607,C(=O)(C1=CCCC1)NCC(c1ccccc1)N(C)C(C12CC(C)(CO1)C2)=O 4608,c1(NC(=O)NCC(CCC)CCO)cc2cccnn2c1 4609,C1(=CC(=O)NCC(CN(C(C(C)(C)OC(C)C)=O)C)O)C2CC3CC(C2)CC1C3 4610,N1(c2snc(CN(C)C)n2)CCCN(Cc2cccc(C3CC3)c2)CC1 4611,C1(C(=O)OC)(C(=O)NC2(C3CCCCO3)CC2)CN(C(=O)CC2CCC(=O)C2)C1 4612,C1(NC(c2cncc(C#C)c2)=O)CC2CC(NC(c3ccc(O)nc3)=O)CC2C1 4613,C1(C(=O)NCC(C)N(C(=O)CN2CSCC2=O)CC)CC(=O)C1(C)C 4614,c1(SCC(=O)N(C(C)CNC(c2c[nH]nc2C2CCCO2)=O)C)ccc(Cl)cc1 4615,CCS(=O)(=O)c1ccc(C(=O)NC2CC2NC(c2cc(OC(C)=O)ccn2)=O)cc1 4616,C1(NC(Cc2ccccc2)C2CC2)CC(N(C)CC)C12CCC2 4617,c1(C(N2CC3N(C(C(C(C)C)OCC)=O)CC(C3)C2)=O)cn2cc(Cl)cnc2n1 4618,CC1CCCN(C(=O)CCC(F)F)C1CNC(C1CCN(CC2CC2)CC1)=O 4619,C=CCC(C)(C)C(=O)N1CC(CNC(c2cccn2C(C)C)=O)C(O)C1 4620,c1(N(CCN(C2CCN(C3CC3)C2)C)C)ccc2c(Cl)nc(C3CC3)nc2c1 4621,c1(C(C)C)c(C(=O)N(C)C(C2CCN(C(=O)C3=CCOC3)C2)C2CC2)cccc1F 4622,N1(C(CC(C)(C)C)=O)CCCC2CN(C(c3cc4c(s3)CCC4)=O)CCC12 4623,N1(C(CCC#CC)=O)CCCC(N(C(=O)COc2ccccc2)C)CC1 4624,c1(C(N2CCC(N(C(=O)CCN3CCC(O)CC3)C)C2)=O)ccnc2c1CCO2 4625,CCCCCC(F)C(=O)NC(C)CCCC(=O)N1CC(=O)NC(C(C)C)C1 4626,C1(NCC2CC(S(C)(=O)=O)C2)CN(C(=O)C=CC(F)(F)F)C2(CCOC2)C1 4627,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CC(O)C(C)C)C)cnc1C(F)(F)F 4628,c1(C(N2C(C)CC(NC(COCCC=C)=O)C2)=O)nsc2ccccc12 4629,C1(CNC(=O)Cc2nncs2)CCC2(CCC2)C1NC(c1cnc(C2CC2)o1)=O 4630,N1(C(C2CCN(C(c3ccc(C#C)o3)=O)CC2)=O)CC2OCCOC2C1 4631,C1(NC(CCN(C(=O)C(C)C(C)C)CC)=O)CCC(=O)NC1C 4632,Cc1cccc(CCC(=O)NCC(C)(O)CNC(=O)C(C2CC2)C2CC2)c1 4633,CC(C)CC(O)C(=O)NC1CN(C(=O)C=Cc2ccc(C(C)(C)C)cc2)CC1C 4634,C(=O)(C1=CCN(C(C2COCCO2)=O)C1)NC(C(C)C)C1CCC1 4635,C(=O)(C(F)(CNC(C1CC(C)(C)CO1)=O)C(C)C)N1CCCC(CC)CC1 4636,N(C1CCc2ccc(Cl)cc21)C(c1cccc(F)c1Br)c1n(CCC)nnn1 4637,N1(Cc2c(C)cc(Br)cc2)CCN(C(c2cnc(C(F)(F)F)cn2)=O)C(C#N)C1 4638,c1(C(N2CC(CCC)N(C(=O)COCC)CC2)=O)cc(C)c(OCCF)c(Cl)c1 4639,Cc1ccc(C(=O)NCCC(C)CCNC(=O)C(=O)C(C)(C)C)nc1O 4640,C1(NC(C2CCCCS2)=O)CCN(C(c2ccc(CO)c(Cl)c2)=O)C12CCC2 4641,C1(C)(NC(CN(C2CC(C#N)C2)C(CCc2cnc(C)o2)=O)=O)CCCC1(C)C 4642,c1(SC)ccccc1CC(N1CCC(C(C)NC(=O)Cc2csnc2C)CC1)=O 4643,CC1(C)CN(C(C2(C3CCCN3C(c3cn[nH]c3)=O)CC2)=O)CCCO1 4644,c1(C(N2CCCC3(NC(c4sc(C)c(O)n4)=O)C2C3)=O)cc2cnccc2[nH]1 4645,C=CC1(CCC(=O)NC2CCC2CC(=O)OC)CCCCC1 4646,N1(C(CCOC)=O)CC(CNC(=O)C(C)NC(C)=O)C(F)(CO)C1 4647,N1(C(C2(C)CCN(C(=O)Nc3ccccn3)CC2)=O)CCC2(CCCO2)CC1 4648,c1(OCC(=O)N(C)CC2N(C(C(CN(C)C)O)=O)CCC2)nc(O)nc(O)n1 4649,c1(COCC)nc(C)cc(=NC2CCCN(C(c3cscc3C(F)(F)F)=O)C2)[nH]1 4650,C(=O)(C1=C(C)C(C)(C)OC1=O)N(C)CCN(C)C(C12CC(C1)C(C(F)(F)F)O2)=O 4651,C1(C(N(CCCC=C)C)=O)(NC(c2snnc2CC)=O)CCCC1C 4652,c1(C(=O)NCC2CN(C(c3[nH]cc(CN(C)C)c3)=O)C(C)C2)ccc(N)cc1Cl 4653,C1(F)(C(N(CCNC(C(C)C(=O)N(C)C)=O)CCOC(C)(C)C)=O)CCS(=O)(=O)C1 4654,C(=O)(CC(C)N(C(=O)C(c1cnn(C)c1)NC(N)=O)C)NC(CCOC)C 4655,N1(CC(N2CCN(Cc3ccc(C)cc3)CC2)=O)CCCC2(CCCCO2)CC1 4656,CC1CCC(NC(=O)Cc2ccc(N(C)C)cc2)CN1C(=O)Cc1cc[nH]n1 4657,c1(NC(C2CCN(c3ccccc3F)C2=O)=O)cccnc1C(N1CCOCC1)=O 4658,CC(C)P(=O)(CC(=O)NC1CC2CCC1(NC(=O)CCc1cnoc1)C2)C(C)C 4659,n1(CC(=O)N(CCN(C(=O)CC2CCC(C3CC3)O2)CC)CC)ncc(Cl)c1C 4660,c1(C(=O)NCC2N(C(C(CC)OC)=O)CC=C2)cc2sc(C)cc2[nH]1 4661,Cc1cc(C(=O)NCC2CCN2C(c2ccc(Cn3ccnc3)cc2)=O)cn1C 4662,Cc1ccc(C(=O)NCC2(C(=O)N(C)C)CCCOC2)c(-n2cc(CO)nn2)c1 4663,CN1CCCC(CCNCc2cnn(-c3cccnc3)c2)C1=O 4664,C(C(Cl)C(C)(F)F)NC1(c2n(CC)nnn2)CC(OCc2ccc(Cl)s2)C1 4665,N1(C(C)=O)CCOC(CNC(=O)CCC2CCCC2)C1.c12csc(n1)C[NH+]([O-])C(=O)C2.O.C 4666,N1(C(C2CCN(C)C(=O)C2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC12CCC2 4667,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)C(CNC(C2CC23CCC3)=O)C1 4668,Cc1cc(CCNC(C2(CO)CCN(C(C3CC3C(N)=O)=O)C2)=O)n(C)n1 4669,N1(C(=O)CC2CCOC(c3ccccc3)C2)CCc2nnc(C3CCC3)cc2C1 4670,n1(CC(=O)NCCCCCCNC(C2(Cl)CC2(F)F)=O)nnc2ccccc2c1=O 4671,C(C1=CCN(C(=O)CC(O)CNC(C2CCOC2(C)C)=O)CC1)OC 4672,N1(C(CC=C)=O)CCC(O)CC1C(=O)Nc1cscc1C 4673,c1(C(=O)NC(CC#C)C(=O)NC2CCCN(C)C2C)ccc2[nH]ccc2n1 4674,C1(CC(=O)NCCC2COCCN2C(c2cc(CO)on2)=O)CN2CCN1CC2 4675,c1(C(=O)NCC2CCC(C(=O)NCCCCCCC)C2)cc2cccn2cn1 4676,CCC(C(=O)OC)C(=O)NCCNC(=O)CC1CCC(C)(C)CC1 4677,C1(SC(CCC)C(C)C)=NC(=O)C2(CCC2)CN1 4678,c1(C(=O)NC2(C)CC(NC(c3nocc3C3CC3)=O)C2)cc(N)nc(Cl)c1 4679,C1(CNC(C=CCN(CC#C)C)=O)CCCC(CNC(=O)CC2(C)CCC(=O)N2)C1 4680,N1(C(CN(C(C)C)C(c2csc(Cl)c2)=O)=O)CCCC(O)C1C 4681,C1(NC(Cc2cccc(OCC)c2)=O)CCN(C(C2CC(=O)N2)=O)C12CCCC2 4682,C1(NC(CN(C)CCO)=O)CS(=O)(=O)C2CN(C(C3C(C)(C)OC3(C)C)=O)CC12 4683,C1(CC)CN(Cc2cn(CCCn3ncc(Br)n3)nn2)CCO1 4684,CC1CCN(C(=O)CCCCN(C)C)CC1CC(=O)NCCN=[N+]=[N-] 4685,C(N=c1[nH]c2c(c(=NCc3snnc3C3CC3)[nH]1)CC(C)CC2)c1nc(C)sc1 4686,c1(C(C)(C)C)cc(C(N2CC(O)(C(N3CC(C(N)=O)C3)=O)C2)=O)no1 4687,C1(NC(c2n(CC(C)C)ncc2)=O)CC2CCC(C1)C2NC(=O)C1=CCCO1 4688,N1(C(c2cnc(C)c(N)c2)=O)CCCC2CN(C(=O)C3=CCN(C)C3)CC12 4689,C(=O)(CCCCC(=O)OC)N1CCCC(C(=O)OCC)CC1.c12cnc(s1)C2 4690,C(=O)(C(C)(C)C(C)C)N1CCC(N(C(=O)CN2C(C)CCC2C)CCC)C1 4691,N1(C(c2ccc(N)c(F)c2)=O)CCC2C(NC(C3CCCC3)=O)C2CC1 4692,c1(C(N(C)CC2CCN(c3nccc(C)n3)C2)=O)cnn2cc[nH]c(=O)c12 4693,C(=O)(C(=O)N(O)C(C)C)N1CC(c2cn(-c3c(C)noc3C)nn2)C1 4694,N1(C(c2cc(Cl)cnc2Cl)=O)CCCC2(CCCN(Cc3ncccc3O)C2)C1 4695,c1(C(N2C(CN(C(=O)CC(C)COC)CC)CCC2)=O)cc(N)nc(Cl)c1 4696,N1(C(CCS(=O)(=O)NC)=O)CC2OCCN(C(=O)Cn3nnc(C)n3)C2C1 4697,c1(CN2CCC(N3C(=O)CCC3=O)CC2)nc2cc(Br)ccc2o1 4698,c1(CCC(=O)NC(C2CCCC2)CNC(C2CC(N(C)C)C2)=O)cc(F)cc(F)c1 4699,c1(OCC)nccc(C(=O)NCCCCCCNC(=O)Cc2cc(C)no2)c1F 4700,CC(C)CC(Cc1ccccc1)C(=O)NC1CN(C(C2(C)CCCO2)=O)CC1C 4701,N1(C(CNC(=O)OCC)=O)CC(NC(c2nc(C)ccc2F)=O)CC(O)C1 4702,C1(CN(C)C(C2(n3cc(-c4ccc(Cl)cc4Cl)nn3)CC2)=O)CCC2CC1C2(C)C 4703,C(C)(C(C(=O)NCC(=O)NCCO)C(C)C)NC(c1cn(CC)nc1)=O 4704,CC1CCN(C(C2COC2)=O)CC1(C)CNC(c1ccnc(OCC(F)F)c1)=O 4705,C12(CNC(CC3C(C)CCC3)=O)CCCC1CN(C(C1CCCC1F)=O)C2 4706,N1(C(CCC(C)(C)OC)=O)CC2(CCC2)CC1C(=O)N(C1CCCC(C)(C)C1)C 4707,Cc1ccnc2sc(C(=O)NCC3CCCCC3C(=O)O)c(C)c12 4708,O=C(CN=c1ccc(Br)c(Br)[nH]1)Nc1cnn2c1OCCC2 4709,C1(CN(C)C(c2ccc(CO)nc2)=O)COCCN1C(=O)CNS(=O)(=O)C1CC1 4710,c1(OC)nc(C)ccc1C(C)NC(C1CCCN(c2ccc(F)cc2)C1=O)=O 4711,c1(CNC(C2N(C(c3cncc(COC)c3)=O)CCC2C)=O)cccc(C)c1F 4712,Cc1cc(C)nc(N(C2(C#N)CCNC2)C(C2CCC(=O)NC2)=O)n1 4713,N(C1CCOc2c(F)cc(F)cc21)C(c1c(OC(C)C)cccc1)=O 4714,c1(C(N(CCCCNC(C(n2ccc(C3CC3)n2)C)=O)C)=O)csc(Cl)n1 4715,N1(CC#CCOC)CCCCC(NC(c2cnnn2-c2ccccc2)=O)C1 4716,C1(CC=C)(NC(=O)CCC#N)CCN(C(c2cnc(C3CCCO3)s2)=O)C1 4717,S(=O)(=O)(c1cccc(Cl)c1F)N1CCN(C(c2ccc(C)c(F)c2F)=O)C2C1C2 4718,C1(CC(=O)NCCCN(C(C2(n3cc(Br)nn3)CC2)=O)C2CC2)CC2CC2C1 4719,n1(CC)ncc(C(=O)NC2(CO)CCN(C(=O)C(C)CSC)C2)c1C 4720,CCCCCC(=O)Nc1ccccc1.C(=O)(COCC(F)F)NC(C1CC1)C1CC1 4721,Cc1cc(C(N2CCOC(C(N(CCCc3ccccc3)C)=O)C2)=O)nn1C 4722,C(=O)(C1=CSCCO1)NC(CCN(C(c1c(C)nns1)=O)C)C 4723,C1(C)(CC)CC(NC(=O)Cc2cc(C)[nH]n2)CN1C(C1(NC(N)=O)CC1)=O 4724,n1(CC=C)c(N(CC(F)(F)Cl)C)nnc1C1=Cc2cc(Cl)ccc2OC1 4725,CC1CC(C(=O)NCC2C3CN(C(C4CC(C)(C)CN4C)=O)CC23)=NO1 4726,C1(NC(c2c(CC)ncs2)=O)C2CC1N(C(=O)CCSc1cccc(Cl)c1)C2C 4727,C(CN=c1cc(F)nc[nH]1)(C1CC1)NC(CC(C(C)C)c1ccccc1)=O 4728,N1(C(c2ccccc2Br)C(=O)Nc2ccc(Cl)cc2)CCC2(C1)OCCO2 4729,C1(C(CC)O)CN(C(=O)C(=O)N(C2CC(COC)C2)C)C1 4730,c1(C(N2C3CN(C(C(CC)C(C)O)=O)C(C3)C2)=O)onc2ccccc12 4731,Cc1noc(C)c1S(=O)(=O)N1CCC2CN(C(=O)CC#N)CCC12 4732,C1(C(N(CC(C)NC(C=CC(CC)NC(C)=O)=O)C)=O)CCC(NC(C)C)CC1 4733,c1(NC)ccc(C(N2CC3CCCC23)=O)cc1[N+](=O)[O-] 4734,C(=O)(C1CCc2cc(F)ccc21)N1CCC(F)(CNC(=O)Cn2ncnn2)C1 4735,c1(C(=O)NC2CN(C(c3n[nH]cc3Br)=O)C3CC23)cccc(F)c1O 4736,c1(NC(Cc2cncc(OC)c2)=O)ccc2c(c1)C(=O)NCC2 4737,C1(C(N(C(C#C)C)C)=O)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4738,N1(C(CCNC(C)=O)=O)CC(O)CC1CNC(C1CC2(CSC2)C1)=O 4739,CC(C)(C)CCCC(=O)N1CCC(NC(C2C3CCCCCC23)=O)C12CC2 4740,C1(C(=O)NCc2cc(O)cc(F)c2)CC2(CCN(C(c3cc(F)c[nH]3)=O)C2)C1 4741,CC1(C(=O)NCC(F)CNC(=O)CSc2ccccn2)CCCC1 4742,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4743,Cc1cc(C(N2CCC(N(CCO)C(C3(C)CCC(=O)NC3)=O)C2)=O)ccc1F 4744,N1(C(CC(C)(C)OC)=O)CCCCC(CNC(=O)Cc2ccc(F)c(F)c2)C1 4745,c1(OC)cc(C(=O)NCCNC(c2c(C3CC3)cnn2C)=O)cc2cn(C)nc12 4746,C(CCCCC(=O)NC(=O)C(F)(F)c1cnn(C)c1)c1cn(CCSC)nn1 4747,N1(C(C2C(C)(C)C2CNC(C2CC2C(F)F)=O)=O)CCC2(CC1)CSC2 4748,C1(SCC(C2CCCN2C(=O)OC(C)(C)C)C)CCCN(c2ccccn2)C1 4749,c1(OC)ccc(C(=O)NCCCC(N)c2ccccc2)cc1C#N 4750,C=C(C)C1OCCC1C(=O)NC1CCN(C2CCN(CCOC)C2)CC1 4751,C1(C(N(CC(=O)NC(C)CO)CC2CC2)=O)C2CN(C)CC12 4752,c1(OC)cccc2[nH]cc(CCN3CCN(C(=O)C=CC(C)(C)C)CC3)c12 4753,C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(C)C(c2cc(C3CC3)ccc2Cl)=O)C1 4754,C=CCC(C)(C)CNC(=O)CC1CCN(C(=O)CP(C)(C)=O)C1 4755,CC1C(NC(=O)Cc2cnsc2)CC2CCC1N2C(=O)C(F)(F)c1cnccn1 4756,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)CC2(CO)CC2)CC1c1cn[nH]c1 4757,N1(C(=O)COCCO)CC2CCCCC2(CN=c2[nH]nco2)C1 4758,c1(C(C)C)cc(NC(=O)C(=O)NCCCN2CCOC2=O)cc(C(C)C)c1 4759,c1(C(=O)OC)c[nH]ccc1=NC(=O)C(N)Cc1ccc(C#N)cc1 4760,C(c1cc(Cl)ccc1Cl)=CC(N1CCN(C(=O)CCN2CCC2)CC1)=O 4761,C1(C(=O)NC(C2(O)CN(C(Cc3nc(C)sc3)=O)C2)C)CCC2(CC1)CC2(F)F 4762,c1(C(=O)NC2C(CNC(c3ccc(F)cc3Cl)=O)CC2)ccc2ncncc2c1 4763,c1(C(=O)NCCCCNC(=O)COCC(F)(F)F)snc(Cl)c1Cl 4764,C(C(C(=O)NC1CC1)N(C1CCCC1)CC1CC1)(C1CCC1)OC 4765,CCC(C)CC(=O)C(=O)NC1(CN(C)C(c2ccc(CN(C)C)o2)=O)CC1 4766,C1(CNC(C2N(CC(C)C)CCCC2)=O)CC12CCN(C(C1CC1CF)=O)CC2 4767,c1(N(C(C)=O)C)ccccc1C(=O)NCC(CNC(C1CC(N=[N+]=[N-])C1)=O)CO 4768,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4769,CC1CN2CCCC2CN1C(=O)C(C)(C1CC1)N(C(=O)Cn1ccccc1=O)C 4770,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CC2CC1CN2 4771,C(CCCCCNC(C1CSCN1C(=O)N(C)C)=O)NC(c1c(C)snn1)=O 4772,c1(C(N(C(C)C(=O)NCC(F)Cl)CC)=O)cc(C#N)cs1 4773,Cn1cncc1CC(=O)NCCCC(=O)NC1CC(CF)C1 4774,N1(C(CC(=O)NC)=O)CCC2CC1CN2C(=O)CNC(c1cccc(C)n1)=O 4775,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(NC(C3CC3C(N)=O)=O)C2)s1 4776,C1(NC(c2c(CC(C)C)cccc2)=O)CCC2(CCN(C(c3ccoc3)=O)C2)C1 4777,CC(C)C(CC(=O)NCC(F)CNC(c1cocn1)=O)c1ccccc1 4778,CCC(CC)CC(F)C(=O)NC1CC2CC1N(C(=O)Cc1csnc1C)C2 4779,Cc1cccc(CCNC(=O)NCC(c2ccc(C(F)(F)F)cc2)F)c1F 4780,C1(CC2CC2)CN(C(=O)OC(C)(C)C)C(C)(C)C1.C12N(CCC1(C)C)C(=O)NC2C 4781,C1(C(=O)NCc2cn(CC)nn2)CN(C(C2CC(C)(C)CCO2)=O)CC12CC2 4782,c1(C(=O)OCC)cc(NC(=O)Nc2ccccc2-c2nn[nH]n2)c(O)c(C)c1 4783,CCCCC(C(=O)NCc1ocnc1CC)NC(c1cc(C)c(C)[nH]1)=O 4784,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4785,C1(CNC(C(C#C)(C)C)=O)CCC(C)N(c2nccc(C)c2C(=O)OC)C1 4786,CCC(C)CC(CO)NC(=O)CC(CC)N(C)C(C1CC(=O)N(C)C1)=O 4787,Cc1nc2ccc(C3CCN(C(c4cc(C)c(=O)n(C)c4)=O)CC3)cc2o1 4788,C(=O)(C#CC1CCCCO1)N(C(CNC(c1cncc(C=C)c1)=O)C)C 4789,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(CC4CCCCO4)c3)=O)C2)s1 4790,c1(OC)cncc(C(N2CC(NC(=O)CN(C)C3CC3)C3CCCC23)=O)c1C 4791,N1(S(CC)(=O)=O)CCCCC1C(N1CC=CC(NC(=O)C#CC2CC2)C1)=O 4792,C1(NC(CCCC(C)C)=O)CCN(C(c2ccnc(Cl)c2)=O)C12CCCC2 4793,C1(CNC(c2ccc(OC)s2)=O)CC12CCN(C(C13CCC(CO1)C3)=O)CC2 4794,c1(C(N2CCOC(C3CCOCC3)C2)=O)[nH]cc2c1CCC2 4795,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4796,c1(OC)cccc(C)c1C(=O)NC1CN(C(=O)C(C)NC(C)=O)CC1F 4797,c1(C)cc(OC)c(OC)cc1-c1ccc(CNc2nc3ccncc3o2)cn1.OC 4798,N1(C(CC(C)SC)=O)CCC(F)(F)C(CNC(C2(C)CC(C)(C)C2)=O)C1 4799,C1(NC(=O)CCN2CCCS2(=O)=O)CC2CCC1N(C(C1CC3CCC1C3)=O)C2 4800,C1(CNC(c2c(C)cco2)=O)CC2COCC2N1C(c1cc2cccnn2n1)=O 4801,C12(C(=O)NC(C)C(C)n3cccn3)CC(C)(CN1C(=O)CN(C)C(N)=O)C2 4802,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC12 4803,c1(C(=O)NC(C2(O)CN(C(=O)CC3CCCO3)C2)C)ccnc2c1CC(=O)N2 4804,c1(C(=O)NCCC2CCCN(C(C3(C)CC3(Cl)Cl)=O)C2)cc(O)nc(C2CC2)n1 4805,C=CCC(C(=O)N(C(C)CCNC(C1(n2cccn2)CCCC1)=O)C)C(C)C 4806,C(CC(C)C(=O)NCC1CCN1C(=O)CCN1CCCCC1)OC 4807,C1(OC)CCCC(C(=O)OCCOc2ccc(F)cn2)C1 4808,CC1CN(C(=O)CCC(C)NCCc2ccccc2)CCc2ccc(O)cc21 4809,N1(C(C2CC(C)C2)=O)CCOCC12COCCN(C(C1C3CCCCCC13)=O)C2 4810,N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)C(F)C3CC3)C2)C1 4811,C(CCCCC(=O)NC1CCC(NC(=O)CC2CNC(=O)C2)C1)OCC 4812,c1(NC(N(CC(C)(C)C)CCNC(C)=O)=O)cnc(C)c(C)c1 4813,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)c1 4814,S1(=O)(=O)c2ccc(cc2)C2(CC2)N1.c1(C(=O)OC)ccc(C(=O)OC)cc1 4815,c1(OC(C)C)ncc(C(=O)NCC2(CC3CCCCC3)COC2)cc1Cl 4816,CC(C)CCCCCC(=O)NCC12CCCCC1N(C(=O)C1=C(C#N)CCC1)CC2 4817,n1(CC(=O)NC(C(=O)N(C)Cc2cnn(C)c2)C2(O)CCC2)[nH]cnc1=N 4818,C(=O)(CCCC(N)=O)Nn1ccnn1.CC(CC(C)c1cccnc1)N1CC(C)C1 4819,CCCCCC(O)C(=O)N(C(C)C=CC(N1CC(c2ncc[nH]2)C1)=O)C1CC1 4820,c1(OC)cc(N2CCC(NC(c3ccc(C(=O)NCCSC)nc3)=O)C2)ncn1 4821,c1(N(CC(=C)C)C)nc(NCC2CCC3(CO2)CC(O)C3)c2ncn(CC)c2n1 4822,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4823,c1(N2CCCC(C=C)C2)nc2c(c(=NCc3nc(O)cc(O)n3)[nH]1)CCC2 4824,c1(C(N2C(CC(=O)Nc3c(C)nc(C)s3)CCC2)=O)c(C#N)c(C(F)(F)F)nn1C 4825,C1(NC(CN2C(C)CCC2)=O)CCC(NC(=O)C(O)c2ccsc2)CC1 4826,c1(CCC(N2CCCC(NS(CC)(=O)=O)CC2)=O)cccc2ccccc12 4827,C(=O)(CC1OCCc2ccsc21)N(CC(C)N(C(c1n(CC)nnc1)=O)C)C 4828,C1(C(N2C(C(=O)NCCCOC)C=CC2)=O)CCCC(=O)C1 4829,C(C(CC(=O)NCc1cnn[nH]1)C1CCC1)NC(C(C1CCCCC1)C)=O 4830,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)CCn3ccnc3)CC2C1 4831,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4832,N1(C(CCOCCOC)=O)CCC(C(F)F)(CNC(=O)Cc2sccc2C)C1 4833,Cc1noc(C)c1CC(C)C(=O)NCCC(C)(C)NC(C1C2CCC(=O)C12)=O 4834,c1(C(N(CC(CC)NC(c2ccc(OC(C)C)cn2)=O)CC)=O)nnc(S)n1C 4835,N1(C(CC(CC)C2CC2)=O)CC(N(C)C(C2CCN(OC)CC2)=O)C2(CC2)C1 4836,CC1CC(c2cn(-c3ccncc3)nn2)CCN1CC(N1CCC(O)CC1)=O 4837,C1(C(=O)NC2CN(C(c3cccc(C#N)c3)=O)C2)CCc2ncnn2C1 4838,S(=O)(=O)(c1cccc(N2Cc3cncnc3C2)n1)NC(c1n(C)c(Cl)cn1)C1CC1 4839,C12(CC)CN(C(=O)O)CC(CO)(C1)C2.c12ccnc(c1)C(=O)NC2 4840,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4841,CC(C)S(=O)c1ccc(C(N2CC3(CCC(CNC(C4(C)CC4)=O)O3)C2)=O)cc1 4842,N1(C(=O)NCc2snc(O)c2Cl)CCC(C2CC2)CC1 4843,n1(CCOC(C)C)c2nnc1nc1[nH]n2C=C1.c1(OC)ccc(Cl)c(O)c1 4844,c1(C(C)(C)C)ccc(S(=O)(=O)NC(C2CCCN(Cc3cncs3)C2)=O)cc1 4845,C1(CCC)(NC(=O)CCN(CC)CC)CCCN(C(C2(CC(C)C)CC2)=O)C1 4846,N1(C(CC(C=C)CC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4847,c1(C(N2CCC(N(C(=O)CSC(C)C)CC)CC2)=O)nccc2ccccc12 4848,N1(C(C=C(CC)C)=O)CC2CC(CNC(c3ccc(CS(C)(=O)=O)o3)=O)C2C1 4849,c1(NC(C2(CC=C)CCCN2C(=O)C(CCC)=CCC)=O)cccc2cccnc12 4850,c1(C(N2CC(C(C)NC(c3cnn(C)c3N)=O)OCC2)=O)cc2cscc2s1 4851,c1(C(N2CCCCC(NC(C(CC)(F)F)=O)CC2)=O)cc2c(cn1)NC(=O)CO2 4852,C(CC)(CCCC(=O)NCC(C)(F)C(C)(C)F)NC(C1(COC)CC1)=O 4853,c1(C(=O)OC)noc2c1CCCC2NCc1nnnn1C 4854,C(C1=CCCN(C(C)(C)C)C1)NC(=NCC=C)NC1CC(OC(=O)OC)C1 4855,Cn1cc(C(=O)NC2CCCN(C(=O)CC3CCCO3)C2)c(O)nc1=O 4856,c1(C(=O)OCC(c2cnn(C)c2)OC)cc(C)c(Br)o1 4857,CC1CCC(C)(C(N2CCCCC2CCNC(=O)Cc2cccnc2F)=O)CC1 4858,c1(N(C)C)ccc(N(C2CCN(CC3CC3)CC2)C(=O)CCCOC(N)=O)cc1 4859,c1(C(N2CC(OC)C(NC(=O)C=CS(C)=O)C2)=O)ccc(C)c(CO)c1 4860,C1(CNC(C(CC)(C)O)=O)CC(C(=O)N2CC(O)(CO)C2)=NO1 4861,c1(-c2n(C(CC)CC)nc(C3CCOC3)n2)ccc(C)c(Br)c1 4862,Cc1c(Cl)cc(C(=O)Nc2c(Br)ccnc2Br)cc1Cl.C12C3CN(CC13)C2=O 4863,CCS(=O)(=O)c1ccc(C(N2CCC(C(F)F)C2)=O)cc1 4864,C12(C=O)CC1(C(=O)OCC)C2.C(=O)(C(C)N(C1CCCC1)C)N.C(C=CC)OCF 4865,N1(C(c2ccc(CCC)[nH]2)=O)CCC12CN(C(=O)CSC)C2 4866,c1(N(CCNC(C2N(CCC)C(=O)CC2)=O)C(C)C)ncc2ccccc2n1 4867,c1(N(CC)CC)ccc(C(CCC)(C)NC2(Br)CC2)cc1 4868,CCCCC(CC(=O)NC(C)CC(C)CC)NC(=O)CC1(C)CC1 4869,N1(C(C2(C)CC(OC)(OC)C2)=O)CC2(CCC(CNC(=O)C(O)C(C)C)O2)C1 4870,c1(NC(c2ccc(-c3ccsc3)cc2)=O)cc(C(=O)O)cnn1 4871,C1(NC(c2c(CC)ccs2)=O)CCCCN(C(C2CCCC(C)CC2)=O)C1 4872,c1(OCC)ccc(C)nc1C(=O)NCC(F)CNC(C1CC1C(F)(F)F)=O 4873,c1(C(N2CCCC(CN(C)C)C2)C(=O)NCCCF)cc(Br)ccc1F 4874,c1(SCC(N2C(C3(NC(Cc4c(C)con4)=O)CC3)CCC2)=O)c(C)cccc1Cl 4875,C1(CC(=O)N(CCCNC(=O)CCn2ccnc2)CCO)CCCCCC1 4876,C1(F)(C(=O)NC2C(OCC)CC2)CCCN(C(=O)C(C)CC2CCC2)C1 4877,N1(C(=O)NC)CCC(C(N2CCCC(C(C)NC(=O)CN(S(C)(=O)=O)C)C2)=O)CC1 4878,CN1CCN(C)C(C(=O)NC2C(NC(=O)CC#N)CC2)C1 4879,c1(-c2ccc(C)cc2C#N)cc(NC(c2c(F)cccc2F)=O)c2cc[nH]c2c1 4880,CC1(C(N2CCCC(NC(c3coc(C4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4881,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(=O)C2CC2)C(c2ccncc2)C1 4882,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3cc(CCOC)on3)=O)CC2C1 4883,c1(C(N2CC3C(NC(c4n(C(C)C)cnc4)=O)C3C2)=O)c[nH]c2cccnc12 4884,N1(C(c2cnc(C)s2)=O)CC2CCC(NC(c3cccc(F)c3Cl)=O)CC2C1 4885,Cn1c(C(N2C(C(=O)NC3(CO)CC3)CC3CC23)=O)ccc1C#N 4886,c1(OC)ccc(CO)cc1O.C1(C=O)CC(F)CCN1C(C1C2CCC(C2)C1C)=O 4887,C(=O)(C(O)CC(N)=O)N(CCC(=O)NCc1cnc(C)o1)CCO 4888,C#CCC(O)C(=O)N1CCC(C(=O)N(C)CCN2CCOCC2=O)CC1 4889,C1(NC(C(C)(N(C(C2CSCC(=O)N2)=O)C2CC2)C2CC2)=O)CC(O)C12CCC2 4890,C1(NC(C(N2CCC(O)CC2)C)=O)CCCC(CNC(=O)CCN(S(C)(=O)=O)C)C1 4891,C(C(C)C(=O)NCCC1(C(=O)N(C)CCc2ccccn2)CC1)OCC 4892,C1(C(=O)NCC2(C(=O)NC(c3ccncc3)C)CC(C)(C)C2)CCC(C#N)CC1 4893,C1(C(=O)NCC23CCCC(CN2c2nnco2)C3)CCC2(CC1)CC2(F)F 4894,N1(C(CS(=O)(=O)NC)=O)CCCC(N(C(=O)Cc2cnc(C)s2)CCO)CC1 4895,C(=O)(CCCCCN=[N+]=[N-])NC1(CC=C)CN(C(C2CCN(CCSC)C2)=O)C1 4896,Cc1nn(C)c(C)c1CC(C)C(=O)NCC(CO)NC(=O)CN1CCCCCC1 4897,c1(C(C)C)conc1C(=O)NC1(CCNC(=O)CC2(C#N)CC2)CC1 4898,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4899,c1(C(=O)NCCCCCCN(C(COCCN(C)C)=O)C)cc2n(c1)CCSC2 4900,c1(C(=O)NCC2OCC(CNC(c3cc(CC)no3)=O)C2)c(F)cc(Cl)cc1Cl 4901,N1(C(C2CN(C(C3C(C(=O)OC)C3)=O)CC2C(C)C)=O)CCCC(N=[N+]=[N-])CC1 4902,CCCCC(O)C(=O)N(CCNC(c1ccc(OC)cc1F)=O)C(C)C 4903,N1(C(CCc2n(C)ncc2)=O)CCOC(CCNC(C2CC2(C)C(F)F)=O)C1 4904,c1(OCC=C)cccnc1C(=O)NCCN(C(C1CN(C)C(=O)N1)=O)C1CC1 4905,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4906,CC(C)C(CN(C)C)C(=O)NC12COC(C1)C(NC(c1nn(C)cc1Cl)=O)C2 4907,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4908,Cc1cc(C#N)c(O)nc1C(=O)NC(C1CCCN(C(C2CC2(F)F)=O)C1)C 4909,c1(-c2onc(C(C)OC(c3ccc(SC)cc3)=O)n2)cccc(F)c1 4910,CC1CCCCC1(CNC(c1cocn1)=O)NC(=O)CCNS(C)(=O)=O 4911,c1(C=O)cccnc1.C1(C(=O)NCC(=O)N(CCCNC2CCC2)C)CCCSC1 4912,N1(C(C(=O)NC(CCCN=[N+]=[N-])C)c2ccoc2)CC(=O)NCC1C1CC1 4913,N1(C(C=CC)=O)CCCCC(CNC(c2cncc(N3CCCC3)n2)=O)C1 4914,C1(NC(=O)C(F)Cc2ccc([N+](=O)[O-])cc2)CN(C(C2COC2)=O)CC12CCC2 4915,N1(C(c2cncc(C#C)c2)=O)CCC2CCN(C(c3nc(C)ccc3F)=O)C2C1 4916,c1(C(=O)NCC(CC)(C)NC(=O)C(C)NC(=O)NC)cc2cncn2c(O)n1 4917,CCCCS(=O)(=O)NC(C)C(N1CC(C(=O)Nc2[nH]ccc2C)C(O)C1)=O 4918,N1(C(C(CCC)O)=O)CCN(C(=O)CCc2cn(C)cn2)CC1c1cnn(C)c1 4919,C(=O)(CC(C)(C)C(F)F)NC1C(CCNC(C2(C)CCN(C(C)=O)C2)=O)CCC1 4920,c1(C(N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)=O)cnc2c(Cl)cccn12 4921,C1(C(=O)NC(c2nc(C)sc2)C)C=CCN(C(=O)C(F)CC2CCOC2)C1 4922,N1(C2C(=O)O2)CCCOCC1.N1(C(c2ccccc2)C(=O)OCC)CCCC1C#N 4923,N1(C(C(=O)NC(C2CCC(C)CC2)CC)=O)CC2CCC1C(O)C2O 4924,c1(C(N(CC(CN(C(c2onc(C)c2C)=O)C)O)C)=O)cncc(S(C)(=O)=O)c1 4925,C(=O)(C1CCC(Nc2ncccc2OC(F)F)c2ccccc21)OC 4926,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1nc(Cl)ccc1F)=O)=O 4927,N1(C(C2CC3(CCC3O)C2)=O)CCC2C(C1)CN2C(c1cnn(CC2CC2)c1)=O 4928,N1(C(C2OCCC(NC(c3c(COC)cc[nH]3)=O)C2)=O)CCCC2(CCCO2)C1 4929,CCCCC(C)C(=O)NCC1COC(C(N2CC(OC(=O)NC)C2)=O)C1 4930,C1(CCNC(=O)C=COOc2ccccc2)(OC)CN(C(=O)CCNC(N)=O)C1 4931,c1(CN2C(C(=O)NCc3cccc(Cl)c3Br)CNCC2)ccc(Br)c2nsnc12 4932,c1(CC(=O)NCCCCCN(C)C(C23CC2CCC3(F)F)=O)cccc(F)c1F 4933,c1(COC)cc(C(=O)NCC2(CCNC(c3oc(CO)nc3C)=O)CC2)c(C)o1 4934,c1(OC(C)C)ccc(C(=O)NCCCN(CCO)C(c2cn(C)nc2Cl)=O)cc1 4935,N1(C(C2OCCO2)=O)CCCC(O)(CCNC(=O)C(F)(F)Cc2ccccc2)C1 4936,c1(C(=O)NCC(CSC)OC)n[nH]c2c1CN(C(c1ncc(C)cc1F)=O)C2 4937,CC1=C(C(=O)N2CC(NC(C3CC3c3cncn3C)=O)CC2(C)C)CCCC1 4938,c1(C(=O)NCC(C(C)C)NC(c2c(Cl)nc(OC)s2)=O)ccc(=O)n2c1CCC2 4939,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)C1=NOCC1 4940,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4941,c1(NC)ncccc1C(=O)N(C)CCOCCN(c1ncc(C)n1C)C 4942,c1(C(=O)NC(CNC(CC(C=C)(C)C)=O)C(C)C)cc(C)nc2c1cnn2C 4943,C(=O)(C1CCCn2nccc21)NC1C(C)N(C(c2nncs2)=O)CCC1 4944,N1(C(c2nc(C(C)OC)sc2)=O)CCCCCC1CNC(C1CC=CC1)=O 4945,C(C)(CCC(C)C)NCC1CC(C)C1 4946,N1(C(C(C)CNC(C2CC2(F)F)=O)=O)CC2CN(C)CC2C1 4947,c1(C(=O)NC23C(CN(C(COCCC=C)=O)C2)C3)ccc(F)c(O)c1 4948,c1(NCCCCC#CC)[nH]c(=NC2CSc3ccccc32)nc2sccc12 4949,CC(CN(C)C)CC(=O)N1CCC(NC(c2cccc(C(=O)NC3CC3)c2)=O)C1 4950,C1(C2CCN(C(=O)C(F)(F)c3cscc3C(F)(F)F)C2)(NC(C=NOC)=O)CC1 4951,CC(=O)CCCC(=O)NC1CC12CC(NC(=O)CCc1cc(C)[nH]n1)C2 4952,C1(C(N2CC3C(C(=O)NCCOCC(=C)C)(C3)C2)=O)CCC2OCCC2C1 4953,C12(NC(c3ccnn3CC3CC3)=O)CCCC1N(C(c1cncc(Cl)n1)=O)CC2 4954,CN1CCN(C(=O)CC(C)(C)NC(C2CNC(=O)N2)=O)C(CO)C1 4955,C1(C(=O)NCCCNC(=O)CC2CCC3(CCC3)OC2)CC2C=CCC(C1)C2 4956,c1(C(=O)NCC2CN(C(CCC(C)C)=O)C2)cn2c(n1)C(C)CCC2 4957,C1(C)(NC(CC2(NC(c3cc(OC)no3)=O)CCC2)=O)CCCC1C 4958,C1(C2CCC2)(NC(C2CN(C(=O)Cn3cccnc3=O)CCO2)=O)CC1 4959,Cc1cc(C(=O)NC2CN(C(c3ccc(Br)cc3)=O)C2)nnc1C 4960,C1(CC=C)(NC(=O)C(c2cc(Br)cs2)C)CCCN(C(=O)C(C)=CC)C1 4961,Cc1cncc(C(N2CCCCC2CN(C)C(C2(c3cc[nH]n3)CC2)=O)=O)c1C 4962,c1(C(N2C(CCNC(CC(C=C)CC)=O)C(C)CCC2)=O)ccnc2c1CCC2 4963,C1(NC(C2(CC=C)CC2)=O)COCCN(C(c2cccc(OC)c2Cl)=O)C1 4964,c1(OC)cc(C)ccc1C(C1CCN1C)(CC)NC(c1cnc(C(C)(C)C)s1)=O 4965,C1(CNC(C)=O)CCN(C(=O)CC2(CCNS(CC)(=O)=O)CCCCC2)CC1O 4966,C1(CNC(C=CC)=O)CCN(C(c2c(C)noc2-c2ccccc2)=O)C12CCC2 4967,Cc1cnoc1Cn1cc(CCCCNC(c2[nH]nnc2-c2ccccc2)=O)nn1 4968,C(=O)(CC(C)(C)n1cc(-c2ccc(Cl)cn2)nn1)NC(C)COC1CCCC1 4969,C12(C(=O)NCC(CN(C(=O)CN3CSCC3=O)C)(C)C)COCC1CN(CCF)C2 4970,N(C)(C1CCc2ccccc21)CC(=O)N(C1CCC(C)C1)N1CCOC1=O 4971,C1(NC(=O)OC(C)(C)C)CC(NC(=O)COC2(C(=O)OC3COC3)CC2)C1 4972,C(=O)(CC(C(F)(F)F)c1ccon1)NC1CCN(C(COCCN(C)C)=O)C1 4973,c1(CCN2CC(CCNC(C(C(C)C)OC)=O)C2)cccc(F)c1N 4974,C(=O)(CC(O)c1cnc(Cl)s1)N(C(CNC(C1(CCC=C)CC1)=O)C)C 4975,C(C(C(=O)NOCCC(F)(F)F)NC(C1CC2(CCO1)CC2)=O)OC 4976,CC1(C(=O)NCC(CO)NC(C2CCCCO2)=O)Cc2ccccc2C1 4977,C1(CC2NC(=O)N(C(c3cc(Cl)ccc3F)=O)C2=O)CCC2(CCCNC2=O)O1 4978,c1(OCCC(N2C(C)(CNC(CCC=CC)=O)CCC2)=O)cccc([N+](=O)[O-])c1 4979,c1(CCNC(=O)NC(C2CCS(=O)(=O)C2)C)cccc(C(C)(C)C#N)c1 4980,C1(CC(N2CC(NC(C)=O)C2)=O)CC2(C1)CN(C(c1ncc(Cl)cc1Cl)=O)C2 4981,N1(C(c2cn(C)nn2)=O)CC2CCC(NC(c3ccn(C4CCCC4)n3)=O)(C2)C1 4982,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)Cc2ccco2)C1 4983,c1(C(=O)NC2CCCN(C(C3CCC(=O)NC3)=O)C2)cc(Cl)cc2cccnc12 4984,N1(C(C(C)C(C)(C)O)=O)CCC(CNC(=O)CCCN2CCCC2)C(C2CC2)C1 4985,C(=O)(C(C)(C)CO)NC1C(CNC(Cc2cc(C)no2)=O)C1 4986,C(=O)(C(F)C1=CCCCC1)N1C2(CNC(=O)COC3CCOC3)CC(C1)C2 4987,c1(S)ccccc1C(C(=O)N(C(C)C)CCc1nn[nH]n1)C 4988,c1(C(C)C)ccccc1NC(=O)CCN(C(=O)CC1CCN(C)C1=O)C(C)C 4989,c1(CCC)ncoc1C(=O)NC(C)(C)C=CC(=O)Nc1ccsc1C 4990,c1(C(=O)NC(CC=CC)C(=O)N2CCC(CC)C2C)ccc(C)cc1C 4991,C1(NC(C2CC(OCC)C2)=O)CC2C(NC(c3ccc(C)cc3)=O)C2C1 4992,c1(OC(C)C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)ccc(O)cc1 4993,N1(C(CC2C(C)(C)C2)=O)CCC(C2(NC(=O)Cc3nc4c(s3)CCCC4)CC2)C1 4994,C(=O)(C1CCc2c[nH]nc21)N1C(CNC(c2cccc3nccn23)=O)C=CC1 4995,C1(NC(C2C3(CC(OC)C3)C2)=O)CCCCCC1NC(C1COCCN1C=O)=O 4996,c1(C(N2CC(CC(C)NC(C(CC)C(C)C)=O)C2)=O)cc([N+](=O)[O-])cnc1N 4997,C1(C(N(CC(N2C(C(=O)OC)CC2C)=O)CC2CC2)=O)CC2(CCC2O)C1 4998,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 4999,CC(C)CC(C)(O)CNC(=O)C(C1(C)CC1)NC(c1cccc(Cl)c1O)=O 5000,N12CCCC(C)(C)C1C2.N1(C(C(=O)NCc2ncc(C)s2)=O)CCCNC(=O)C1 5001,CCCCCCC(=O)NCC1CC2(C1)CN(C(=O)C(CCSC)NC(C)=O)C2 5002,C(C)(CNC(C1(C)CCSCC1)=O)(C(C)C)NC(COCc1onc(C)n1)=O 5003,C(=O)(C1=C(C)CCOC1)NC(CCNC(c1ccc(C#C)cn1)=O)(C)C 5004,C1(CNC(C(C)n2ccnc2)=O)CCCCN(c2nnc(CC3CC3)o2)C1 5005,c1(C(=O)NCCCN(C(C(CC)OC)=O)CC)cccc(Cl)c1C(F)F 5006,C(N=c1[nH]c(C)nc(C)c1F)C1(NC(C(CCOC)C)=O)CCCCC1C 5007,c1(CC)cc(N)c(C(=O)NCC(C)CNC(c2ncc(C)cc2F)=O)c(F)c1 5008,C(=O)(CC(C)COC)N1CCCC(N(C(c2ccnn2CC(F)(F)F)=O)CC)C1 5009,CCC(C(=O)NCCCCN(C(=O)Cn1ccc(Br)n1)C)N(C)C 5010,c1(NC(C2CC(F)CN(c3ncc(C4CC4)cn3)C2)=O)cccc(F)c1O 5011,Cc1cc(C#N)nc(NC2CC2CNC(=O)Cc2cc(-c3cccs3)on2)n1 5012,C1(NC(C2OCC(CNC(COC(C)C)=O)C2)=O)CCC12CCC2 5013,Cc1cc(C(N2CCN(C(c3nccnc3Cl)=O)C(C)C2)=O)cc(C)c1O 5014,C1(NC(C(CC)N(C)C)=O)CCN(CCc2cnn(COC)c2)CC1(C)C 5015,N1(C(C2CC(C(C)C)C2)=O)CCN(Cc2ccc(C(F)(F)F)cc2Br)C2CC12 5016,n1(CCCC(=O)NCC(CNC(c2cnn(C)c2C)=O)OC)nc(C)cc1C 5017,C(CC(=C)Cl)(C(=O)NCCC1COCC1O)NC(C(CC=C)NC(C)=O)=O 5018,C(=O)(C1=NN(CCO)C(=O)CC1)NCCC1CC(NC(C(C(C)O)C)=O)C1 5019,CCCCC(C)C(=O)N1CC(OC)CC1CNC(=O)C=NOC 5020,C(=O)(CC(C)(F)F)NC(C1(CNC(C2CC2c2ccc(F)cc2)=O)CC1)C 5021,CCCC(CCC)CC(=O)NCC1(F)CCCN(C(=O)CCc2ccncn2)C1 5022,CCCCC(C)CCC(=O)NC(C)CN(C(C1CCC1)=O)CC 5023,c1(C(=O)NC(CCSC)C(=O)NO)ccc2c(c1)OCO2 5024,CCCC(CNC(=O)C(C)(C)c1ccno1)C(=O)N(C)CC1CC1(C)C 5025,c1(C(=O)NC(CC)CNC(c2cnc(C)[nH]2)=O)cc2c(C)c(C)ccc2[nH]1 5026,C1(NC(C=NOC)=O)(CO)CCN(C(c2c[nH]nc2-c2ccccc2)=O)CC1 5027,C(CCC)(C(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C)=CCC 5028,C1(OC)CCCCC1C(=O)NC1CCC(NC(C2CC3CCC2C3)=O)C1 5029,C(=O)(C1=C(F)CN(C(C23CC(F)(C2)C3)=O)CC1)N(C1CC2CCC1CC2)CC 5030,N1(C(COCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5031,C1(N(C(=O)C(F)CC2CC2)C)CCN(C(c2ncoc2C(F)(F)F)=O)CC1 5032,O=C1NC2(NC(=O)C(F)(F)F)CC3CC1C2C3.N12CCCN(CC1)C(=O)C2 5033,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(CNC(C=C(C)C(C)C)=O)CC1(C)C 5034,CCC(C)C(C(=O)NC(C)(C)CN(C)C)N(C(=O)C(F)C1CCC1)C 5035,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)CCOc2ccccc2F)CCO1 5036,C1(C#CC(=O)N2CCN(CCNC(=O)CCC(C)O)CC2)(CC)CC1 5037,C1(N(C)C)CCC(NC(=O)NC(C2CCCN2C(C2(O)CCCC2)=O)=O)CC1 5038,c1(OC)cccc(C(=O)NCC2CCN(C(=O)Cn3nnc(C)n3)CC2C)c1F 5039,c1(C(=O)NCC(=O)N(C2CCN(C(=O)CC3CCCC3)C2)CC)cc(F)cc(F)c1 5040,c1(-c2ccc(C)cc2)nc(=NC2CC3CN(C(=O)C(C)OCC(C)C)CC23)s[nH]1 5041,c1(CC)ccc(C(=O)NC2CN(C(=O)C(CC)SC)CC2(C)C)cc1C#N 5042,Cc1nc2c(C(C)NC(=O)CC3CC(C)(C)CO3)cccc2o1 5043,C1(Nc2nc(Cl)nc(C)c2F)CC2(CCN(C(C3CC(C)CO3)=O)CC2)C1 5044,C1(CNC(C(C)CC2CC2)=O)CCCCN(C(=O)CN2CCCCCC2=O)CC1 5045,CCCCC(O)C(=O)NC(CNC(c1c(C#N)cnn1C)=O)CC 5046,C1(C(=O)NCCCC2CC(NC(c3cc(C)ns3)=O)C2)CC2(CC2)C(=O)O1 5047,Cn1ncc2ncnc(N3CC4CCCN(C(c5cc(C(N)=O)cs5)=O)C4C3)c12 5048,CC1CCCN(C(c2ccn(C(F)F)n2)=O)C1CNC(c1ccc(Cl)s1)=O 5049,C1(C(=O)NC(C2CCCCO2)CCOC)CC2(CC2)C(=O)O1 5050,C=C1CC(C(=O)Nc2ccnc(C3CC3)n2)N(C(C2CCC(CO)CC2)=O)C1 5051,C(=O)(CCCCC(=O)OC(C)(C)C)N1C2CCC(CCNC(C=CCC)=O)(C2)C1 5052,CN1CCCCC1CCC(=O)NC1CC2(C1)CC2NC(c1cc(O)cs1)=O 5053,Cc1cccc2c1CCOC2C(=O)NCC(CCOC)NC(C1CCCSC1)=O 5054,C(Cc1cn[nH]c1)(C(=O)NCC1COC(=O)N1)NC(CC=CCC)=O 5055,n1(CC(=O)NCC2CC3(CCN(C(=O)C=CCO)C3)CO2)ccc2c(O)cccc12 5056,C1(O)(C(C(N2CCC(C(C)NC(c3c(NC)scn3)=O)C2)=O)(F)F)CCCCC1 5057,c1(C(=O)NCC(CO)NC(c2ccc(C#C)o2)=O)cc2cc(C)cc(C)c2[nH]1 5058,CCCC(CCC)C(=O)N1CCC(NC(=O)C(C)Cc2ccc(C#N)cc2)C1 5059,CC1CN(C)CCCN1C(=O)CC(C(C)(C)C)NC(=O)CC1CCC(=O)CC1 5060,C1(C#N)(OC)CC(C(N2CC(F)CC2CNC(c2cn(C)nc2C(F)F)=O)=O)C1 5061,c1(C(N2CCC(N(CCOC)C(C3CC(C)CO3)=O)CC2)=O)cc(C)c(F)cn1 5062,C1(OC(C)(C)C)CC2(COC(C)C2)C1.Cc1nc(C)oc1C(=O)O.C1(=O)CO1 5063,C(=O)(C(CC(C)(C)C)NC(=O)C(F)OC(F)(F)F)NCc1c(O)ncc(C)c1 5064,C1(CC=C)(NC(c2c(-c3ccsc3)noc2C)=O)CCN(C(C2CCCO2)=O)C1 5065,Cc1nn2cc[nH]c(=O)c2c1C(=O)NC1CCCN(C(=O)C(C)(C)C)CC1 5066,N1(C(C(CC)COC)=O)CC(C(=O)NCCCn2cc(C)cn2)C2(CCC2)C1 5067,Cc1nc(NC2CCCC(NC(=O)Cc3cccnc3Cl)C2)c2scc(C)c2n1 5068,N1(C(CS(CC)=O)=O)CCOC2(C1)CN(C(=O)C(C)COC1CCOCC1)C2 5069,c1(C(N2CCCCC(NC(C3C(C(=O)OCC)CC3)=O)C2)=O)cc([N+](=O)[O-])ccn1 5070,c1(N(C(C)(Cc2cccs2)N(C)C)C)nc[nH]c1C(C)(C)C 5071,C=CCC(CNC(=O)CCC(C)CN(C)C)C(=O)Nc1cnn(CC2CC2)c1 5072,c1(C(=O)NC(C)CCCNC(=O)C(F)(F)C(C)(C)O)nn(C)c2ccc(O)cc12 5073,C1(C)(CC)CCCN(C(C2(SC)CN(C(C3CNC(=O)N3)=O)C2)=O)C1 5074,N1(C(CCc2cc(OC)no2)=O)CCN(C(c2nnn(C)c2C)=O)C2CCCC12 5075,C(N=c1[nH]c(C)cc(=NC(C)c2c(C)ccnc2OC)[nH]1)c1n(CC)cnc1 5076,c1(C(N(CCNC(C2CC(CS(C)(=O)=O)C2)=O)CC)=O)cccc2ccnn12 5077,C1(C2CC(=C)C2)CCC(C(=O)NC(C)CCNC(=O)COC2CCC2)CC1 5078,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CNC(=O)CCOC1CCC1 5079,CCC(C)(C#N)C(=O)NCC(C1CCCCC1)NC(c1c(OC)noc1C)=O 5080,C(CC(=O)NC1CC(CCN(C2CCCO2)C)C1)OC.C1C(=O)N(C)CCO1 5081,c1(C(N2CC(C(C)NC(c3ccc(Cl)nn3)=O)C2)=O)cc(N)cc(O)c1F 5082,C1(Cl)(C(N2CC(N(C)C(c3cnn(C4CCOC4)n3)=O)C2)=O)CC12CCC2 5083,c1(OC)ccccc1C(C)NCc1cc(C(=O)Nc2cc(O)ccn2)ccn1 5084,Cc1ccc(NC(c2ccc(C(C3CC=CCC3)CO)cc2)=O)cc1C 5085,c1(CNC(c2nnnn2CSC2CCOCC2)C2(CCO)CC2)cc(Cl)no1 5086,C12(C(=O)NCC(CNC(c3cc(CC)nn3C)=O)O)CC(C)(C1)OC2C 5087,C1(C)(CNC(CN2CCN(C)CC2)=O)CN(C(C2CC(F)C2)=O)C(C)(C)C1 5088,C1(CC(=O)NC(C2CCN(C(c3c(C(C)C)noc3)=O)C2)C)CCCCC1O 5089,C1(C(N2C(C)CC(CC(N3CC(COC(C)=O)C3)=O)C2)=O)Cc2ccccc2N1 5090,CC(C)(C(=O)NCC=CCNC(=O)CC1CCC(=O)N1)CCC(F)(F)F 5091,O(NC(=O)C(O)CNC(=O)C(F)CCCC)C(C=C)C 5092,C(CCN=c1[nH]c2c(c(=NC3CC4C=CC3CC4)[nH]1)COC2)N(n1ccnc1)C 5093,C(=O)(CCCCCc1cccs1)N1CC(C(C)NC(C(c2cccnc2)C)=O)C1 5094,N1(C(c2ccc(OCCO)cc2F)C(=O)NCCSC)CCN2C(=O)CCC2C1 5095,C1(CC(=O)N(C(C)C(=O)NCCCc2cccnc2)CCC)COCC(C)O1 5096,N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(C2CN(C(c3cccnn3)=O)C2)C1 5097,c1(C(N2CCC(n3cc(COCC)nn3)C2)=O)cc2n(n1)CCCCO2 5098,C=CCC(C(=O)N1CCC(CNC(=O)C(CO)OC)(COC)C1)N(C)C 5099,C(CC(C(C)C)NC(=O)C(C)N(C)C)NC(c1n(C(C)C)ccn1)=O 5100,C1(CC(N2C(CO)CC(NC(CCC=C=C)=O)C2)=O)CN2CCN1CC2 5101,N1(C(c2c(CC)scn2)=O)CC(C)CN(C(c2ns[nH]c2=O)=O)CC1C 5102,c1(C(N(CCNC(C(C)NC(=O)NC)=O)C2CC2)=O)cc2c(nc1O)CCCC2 5103,c1(C(C(=O)NC2(C)CC2)N(CC=C)CCCOC)ccc(F)s1 5104,Cc1cc(C)c(C(=O)NCC(F)CNC(=O)Cn2cnc(=N)[nH]2)cc1Br 5105,n1(CC(=O)NC(C2CN(C(c3cnc(C4CCCO4)s3)=O)C2)C)cccnc1=O 5106,CCC(C)(C)C(O)C(=O)NCC1C2CN(C(c3cc(N)c(C(=O)OC)s3)=O)CC12 5107,N1(C(c2nccc(Cl)c2Br)C(=O)NCCOC)CC(CO)OC(C)(C)C1 5108,N1(C(CNC(=O)NC)=O)CC2CC(C1)C(=O)N2.c1(CC(=O)NC)cc(SC)co1 5109,C12(CNC(=O)CCc3ccsc3)CCC1CCN2C(=O)CCCC1CCCCC1 5110,C1(NC(CC(C=C)CC)=O)(CNC(c2nn(CC)nc2C)=O)CC2CCC1CC2 5111,N1(C(C2CC2c2ccccc2C(C)=O)=O)CC2CN(C(C3CNC(=O)O3)=O)CC12 5112,C1(OC)CC2CCC1N2C(=O)NC1(Cc2ccc(Cl)cc2F)CCOC1 5113,c1(C(=O)NCC(CNC(CC2CCN(C(C)C)CC2)=O)O)nsc2ccccc12 5114,C=Cc1ccc(CN2CCN(C(=O)CC(=O)N3CCOCC3)C(CC)C2)cc1 5115,N1(C(CCOC)=O)CCC(CCNC(C2(C(=O)N(C)C(C)C)CC2)=O)CC1 5116,Cc1cc(C)nc(SCC(=O)NC2CC(O)(CNC(c3cnccc3Cl)=O)C2)n1 5117,c1(C(C(C)C)=O)c[nH]c(C(N2CCC(N(C(=O)Cc3cnn(C)c3)C)C2)=O)c1 5118,c1(C(=O)NC(C(=O)NCC2CC(C)C2)C)ccncc1OC 5119,c1(OC)ccc(SCC2CC(F)(F)C2)c(Br)c1 5120,C1(CNC(C2C3CCCC23)=O)(CO)CC12CCN(C(=O)CC(F)(F)Cl)CC2 5121,N1(C(CC2ON=C(CC)C2)=O)CCN(C(=O)CCCCCNC(C)=O)CC1CO 5122,N1(CCC)CCCC1C(=O)NC1CC(C)(NC(=O)C(c2ccc(C)s2)C)C1 5123,C1(C(N(CCN(C(c2cnn(C3CC3)c2)=O)CC)CC)=O)CCNC(=O)C1 5124,C1(NC(CC2C(C)CCO2)=O)CC2(CCN(C(c3ccoc3C3CC3)=O)CC2)C1 5125,C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(C1CCS1(=O)=O)=O 5126,Cc1nn(C)c(Cl)c1C(N1CCN(S(=O)(=O)C(F)(F)F)CC1)C(=O)NCCC#N 5127,CC1OC(C)(C)OC1(C)C(=O)NCCCC(C)(C)NC(=O)CN(C)C(=O)C1CC1 5128,Cc1ccc(Cl)c(F)c1C(N1CC(O)(C(C)NC(=O)Nc2cccc(F)c2)C1)=O 5129,c1(CN2CC(c3n(C(C)C(N4CCC(C)C4CO)=O)cnn3)C2)ccc(=O)n(C)n1 5130,C1(Cl)(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CC1(C)C 5131,c1(CNC2CC(NC(c3ccc(C(=O)OC)c(C)c3)=O)C2)c(C)ccc(Br)c1C 5132,c1(-c2c(OCC#N)ccc(F)c2)ccc2c(C(=O)Nc3nccs3)n[nH]c2c1 5133,c1(OC)ccc(Br)c(CCN(C(=O)C(N)Cc2c(O)cccc2F)C2CC2)c1 5134,C(C)(CO)(C(=O)NCCC1CCCC(C)C1)NC(C1C(OCC)CC1)=O 5135,Cc1ccc(C(=O)NC23CCC(CC2NC(=O)Cn2ccc(C)c2)C3)cc1O 5136,N1(CC(=O)N(CCC(C)NC(=O)CC2(OC(=N)O)CC2)C)CCCC(C(N)=O)C1 5137,S(=O)(=O)(CCC(F)(F)F)Nc1c(C(=O)Nc2c(OC)nccn2)c(F)ccc1 5138,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5139,N1(C(C(C(C)O)N(C)C)=O)CC(C)(C)CC1CNC(c1sccc1-n1cccc1)=O 5140,C(=O)(C1Cc2ccc(F)cc21)N1CC(OCCNC(=O)Cc2sc(O)nc2O)C1 5141,C1(C(=O)NC(c2nc(C)sc2C)C)CCN(C(c2cc(Cl)n(C)n2)=O)CC1C 5142,CC(C)(CCCNC(C1CCC(=O)N1)=O)C(=O)N1CCN2CCCC2C1 5143,C(=O)(C(=O)CC(C)C)N1CC(CC)(NC(=O)Cc2cnsc2)C1 5144,CC(C)C(C)(CNC(C1CC1C(C)NC(=O)C=Cc1cncn1C)=O)C(C)C 5145,C1(CNC(c2ccc(C)s2)=O)CC2(CCN(C(=O)C(C)S(=O)(=O)C(C)C)CC2)C1 5146,C1(C(=O)NC(C)C(C)C)(CC)CCCN(C(c2csc(CO)n2)=O)C1 5147,c1(C(=O)NC2CC(NC(c3nc(OC)c(F)cn3)=O)C2)ccc(C#N)cc1F 5148,C1(NC(C2C(C)CCC2)=O)CCOC12CCN(C(=O)C(C)(C)CCCO)CC2 5149,c1(CC(=O)NCC2(OC)CN(C(C3CC3(C)C)=O)C2)ccc(F)cc1C 5150,C(CCC(F)(F)F)(c1ccccc1)NC(=O)NCc1cccc(OC(C)C)n1 5151,C1(OC)CCC(CC(=O)NCCNC(c2cnn(-c3ccccn3)c2C)=O)CC1 5152,Cc1ccc(C(=O)NC(CNC(=O)C(c2ccc(C)nc2)(F)F)C(C)C)c(N)n1 5153,c1(N2CC(C)OC(CO)C2)ncc(S(=O)(=O)NCCc2ccncc2Br)cc1Cl 5154,Cc1cnn(C)c1C(=O)N(C)CC1CCCN1C(=O)CCC(C)NC(N)=O 5155,c1(C(=O)NC2CCN(C(c3c(C)cccc3O)=O)C2)ccc2cnccc2c1Cl 5156,C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(CSCCC)=O)CC12CC2 5157,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5158,C(CC(C)(C)CC(=O)NC1CC(O)(CNC(=O)C(C)(C)C2CCCO2)C1)OC 5159,CC1CCC(C)N1CCNC(C1(F)CCN(OC(=O)NCc2ccccc2)C1)=O 5160,N1(C(Cc2c(C)noc2C)=O)CC2CN(C(=O)CCC3CCCC3)C2C1 5161,N1(C(CCCSC(C)(C)C)=O)CCC(C2CCN(C(=O)C(F)(F)C(F)(F)F)C2)C1 5162,Cc1c(C(N2CC(C)(NC(=O)CCn3cnnn3)C2)=O)oc2c(Cl)cccc12 5163,c1(C(=O)NC(C(C)C)CCNC(c2cc3n(c2)CCC3)=O)ccc2nncn2c1 5164,CCCCS(=O)(=O)CC(=O)NCc1ccc(CNC(=O)CC#N)cc1F 5165,c1(OC)ccc(C=CC(=O)Nc2ccc(S(=O)(=O)CC(C)C)s2)cc1F 5166,C1(NC(C2OCCN(C)C2)=O)CC2CN(C(=O)C(O)CF)CC2C1 5167,c1(NC(C(N2CCN(C(c3c(C)ccs3)=O)CC2)C)=O)cc(Cl)cc(Cl)c1Br 5168,CON1CC(C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)CC1=O 5169,C=CCCCC(C(=O)NC1C2CCCCCC12)NC(=O)C(C)SC 5170,N#Cc1cccc(C(=O)NC2CC3CC(NC(C4CCCC4)=O)CC23)c1F 5171,N1(C(c2n(C=C)ncc2)=O)CCC(C)CC1CNC(=O)CC 5172,Cc1cccn2cc(C(N3CC(CNC(=O)CSC(C)C)C(F)C3)=O)cc12 5173,Cc1sncc1C(=O)NC(C)C=CC(=O)N(CCS(C)(=O)=O)C 5174,c12cccc(Br)c1[nH]s2.CC(Cc1ccccc1)C(=O)N(C)Cc1ccccc1 5175,C(=O)(CCCCC(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5176,CC1(NC(C2CCC3CCC2O3)=O)CCN(C(=O)CC2CC=CCC2)CC1 5177,C(Cn1cncn1)(C(=O)NC1CC1CCCCO)NC(c1cc[nH]c1)=O 5178,N1(C(c2ccc(SC)o2)=O)CC(C)CCC1CNC(=O)COc1cnn(C)c1 5179,c1(C(N2CCC(NC(c3cncc(OCC)c3)=O)C2)=O)cc(C)ccc1O 5180,c1(C(C(=O)N(CCCCCNC(C(CCC)F)=O)C)O)ccc(F)cc1C 5181,Cc1cnccc1NC(c1cnn(CCNC(N)=O)c1C)=O 5182,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(c3cnnn3C)=O)C(C)C1)=O)C2 5183,C(CC(C)C)(C(=O)NCCCCCN(C)C(C1CC12CC(C)(C)C2)=O)NC(C)=O 5184,C(=O)(C1=CC2CCCCCCC12)N1C(C)CN(C(C2(CF)CC2)=O)CC(C)C1 5185,C1(C(=O)NC(CNC(c2c(C)ncn2C)=O)CC(F)(F)F)CCC(N=[N+]=[N-])CC1 5186,c1(N2CCN(N(Cc3nc(CC)sc3)CC)CC2)ccc2nccc(N)c2c1 5187,CC1OC2(C(=O)N(CCCN(C(=O)CCSc3ccccc3)C)C)CC1C2 5188,CC(C)(C)CC(=O)OCC(C(C)(C)C)=O.C1CC(O)CNC(=O)C=CCN1 5189,CCCC(CC)C(=O)N(C1CCN(C(=O)C(C)(C)COC(C)C)CC1)C 5190,CC1c2ccccc2OC1C(N1CC(NC(=O)COCCF)C(C)C1)=O 5191,N(C(=NCC1CCOC1)NCC1(CC(=O)OC)CC1)C(C=C)C 5192,CC(C)CN=C(NCC(n1cccn1)C)NCC1CCCN1C1CCOCC1 5193,N1(C(C(C)OCC)=O)CCC2CN(C(c3ccoc3Cl)=O)C(CO)C2C1 5194,c1(CCN(C)C(C2CCC2)=O)cn(CCCC(=O)NC)nn1.C(=O)(COC1CCC1)O 5195,CN1N=C(C(=O)NC2CN(C(C3CC(F)(F)CCC3(C)C)=O)CCC2O)CCC1=O 5196,C1(C(=O)NCC(C(C)O)O)CCC2(CC2)N1C(c1cccc(CO)n1)=O 5197,c1(C(=O)NCc2ccc(-c3c(CC)cccc3)cn2)ccnc2[nH]c(C)nc12 5198,C(=O)(N(CCC(=O)N1CCC(n2cnnn2)C1)OC)C1CC(C#C)(O)C1 5199,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)s2)=O)C1 5200,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(c1cc(C)c(O)c(C)c1)=O 5201,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5202,C1(C(=O)NCC(c2ccsc2)C)CC=CCN1C(c1cccc(CO)c1)=O 5203,c1(C(N2CCC(O)(CNC(Cc3c(C)nsc3)=O)C2)=O)ncc(C2CC2)cc1F 5204,N1(C(C(CCCC)(C)F)=O)CC2(CCCN(C(c3ccnn3CCF)=O)C2)C1 5205,CC1SCCN(C(C23CC(CN2C(=O)C(C)(C)CN(C)C)C3)=O)C1C 5206,c1(C(C(=O)NCC(CSc2cn(C)nc2)O)O)ccccc1F 5207,N1(C(CC=C=C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5208,N1(C(Cc2c(C)cco2)=O)CC2CCOC2(CNC(c2ccnc(Cl)c2F)=O)C1 5209,N1(C(CCC)=O)CCC2(CC1)CC(C(=O)Nc1c(C)cccc1C)C2 5210,c1(CC(=O)Nc2scc(CC(=O)NC3CCN(CC)C3)n2)c(O)ccc(F)c1F 5211,C(=O)(C(CC(C)C)N(C)C(c1c(C)cnn1C)=O)NCCOC(CC)(C)C 5212,Nc1ccccc1C(=O)NCC(=O)NC1CC12CC(NC(C1(COC)CC1)=O)C2 5213,S(=O)(=O)(c1cc([N+](=O)[O-])c(N)cc1[N+](=O)[O-])N1CCN(C2CN(C)CC2O)CC1 5214,C1(NC(CCC#C)=O)CN(C(c2ccncc2N(C)C(C)=O)=O)C(C)(C)C1 5215,C1(CNC(CC(C)CF)=O)COCCN(C(c2ccsc2Br)=O)C1 5216,Cc1cc(C(=O)NCCC(O)CNC(C2(CCCF)CC2)=O)nn1CC(F)(F)F 5217,N1(C(=O)CC2CCCCN2C(=O)C(O)c2ccsc2)CC2(CCOCC2)C1 5218,CC1CC(C(=O)NCCC2CCCCC2O)N(C(c2ncncc2Cl)=O)C1 5219,C(C(CC)(CC)NC(C1CC(F)C(=O)N1)=O)NC(C=CCC)=O 5220,C1(CC=C)(NC(=O)C(C)=CCC)CC2CCC(C1)N2C(c1snc(C)c1N)=O 5221,C(=O)(CC(C)CC(=O)NCC(O)C(=O)NC1CC(C(C)O)C1)OC 5222,C1(OCC)CC(NC(=O)CC(=O)NC)CN(C(=O)Cn2ccnn2)C1 5223,C1(CC=C)(NC(=O)CC(C)C=C)CC2CCC(C1)N2C(=O)Cc1cc[nH]n1 5224,C(=O)(CS(=O)(=O)CC(C)C)N1C(CN(C(C(CC(C)=O)(C)C)=O)CCO)CCC1 5225,CC1CCN(C(c2cc[nH]c2)=O)C(CNC(C2CCOC2=O)=O)C1 5226,C12=NC(Cl)=CC(=NC(=O)C3CC3N1)N2.c1(OCC)cc(-c2ccncc2)ccn1 5227,N1(C(C2CC(OCC)C2)=O)CCC2(CNC(=O)Cc3ccccc3O)CCCC12 5228,C1(CNC(C2(CSC)CCC2)=O)CC12CCN(C(=O)C#CC1CC1)CC2 5229,C(CCCC(=O)NCC(C1CCOC1)O)N(C(=O)Cn1cnc(C#N)n1)C 5230,CCC(C)(C)C(C)(O)c1nnc(-c2cc(C)nn2C)n1Cc1cccs1 5231,c1(C(N2CCN(CCNC(c3ccn(C)n3)=O)CC2)=O)ccc(C(F)F)c(F)c1 5232,C(=O)(C(C)CC(N)=O)N(CCN(C(=O)C(C)Oc1cccc(N)c1)CC)CC.CC 5233,C1(C(=O)NS(CC)(=O)=O)C(C)(C)CN(C(=O)CCC(C)SC)CC1(C)C 5234,N(C1CCCOc2ccccc21)C(=O)NC(Cc1c(C)ccs1)N(C)C 5235,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5236,N1(C(c2c(COC)nn[nH]2)=O)CC2CC(C(=O)NC(C)(CO)CC(C)C)C(C2)C1 5237,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5238,c1(C(N(C2CCCN(C(C3CCS3(=O)=O)=O)C2)CC)=O)ccnc2c1CC(=O)N2 5239,c1(OC(C2CCCN(C(N3CCN(C)C(=O)C3)=O)C2)=O)ccc2c(n1)OCCO2 5240,C1(C2CC2)(CNC(CCP(C)(C)=O)=O)CCN(C(c2cncc3nc[nH]c23)=O)C1 5241,c1(C(N)=O)cnn(C)c1.N1(C2(C(=O)NCCCN)CC2)CCCC1.C1C(=O)N1 5242,C(=O)(C(C(C)CC)NC(=O)C=CCCC)NC(CC#C)C 5243,Cc1nn(C)c(Cl)c1C(N1CC(C(=O)Nc2cc(C(C)C)nn2C)C1)=O 5244,CCC1=C(C(=O)NCC2(C)CC(NC(c3cc4n(n3)CCCC4O)=O)C2)CCCO1 5245,N1(C(CCC=C(C)C)=O)CC(CN(C(=O)C(O)C(C)(C)C)C)C2(CC2)C1 5246,CCC(CCOC)C(=O)N1CC(OC)CC1CNC(C1(CO)CCOCC1)=O 5247,c1(C(N2CCC(F)(C(=O)N(CCn3c(C)cnn3)CC)C2)=O)ccc(C)nc1O 5248,CC1CC(NC(=O)C(CCOCCO)NC(c2ccncc2)=O)CC(C)C1 5249,N1(C(COCCC(C)C)=O)CC2CC(C1)C2NC(c1ncoc1-c1ccon1)=O 5250,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(C)n2C)=O)cc2n(c1)CCOC2 5251,c1(OC)ccnc(C(=O)NCC2(NC(=O)CC3CC(C)=NO3)CCC2)c1 5252,C1(CC(N2C(C(=O)O)CCC2C2CC2)=O)CCN(C(=O)CC2CCC3CC23)CC1 5253,c1(C(c2n(CC)nnn2)NC2(c3cccc(Cl)c3)CC2)c(F)ccc(Br)c1Cl 5254,C1(C(C)C2CC2)CCCN1C(=O)C(O)CNC(=O)CC1CC=CC1 5255,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)(NC(c2nnn(C)c2N)=O)CCCCC1 5256,c1(C(N2CCC(C)(NC(C3CN(CC)C(=O)C3)=O)C2)=O)ncnc2cc[nH]c12 5257,c1(COC)cccc(C(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5258,c1(C(C)(C)NC(C(C)Sc2ccccc2)=O)ccccc1.C12(CCOC1)C(=O)O2 5259,c1(C(=O)NCCCCNC(C2(CCCC)CCOC2)=O)cc(-n2ccnc2)ccn1 5260,O=C(C1=CCCC1)NC1(c2n[nH]cc2Br)CC1.C12CCCN1C2=O 5261,CC1CN(C)CC(C(=O)NC2CC2NC(=O)COc2cccc(O)c2)O1 5262,c1(C(=O)NCCN(CCC)C(C2CCSC(C)C2)=O)cccc2[nH]cc(Cl)c12 5263,c1(COC(C2C(NC(C(CCC)(C)C)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] 5264,c1(OC)cccc(C(=O)NCC23CC2CN(C(c2nccs2)=O)C3)c1I 5265,N(C(=NCC1CCOC1)N1CCC(SCCN(S(C)(=O)=O)C)C1)Cc1ccccc1 5266,C1(C)(C(=O)NC(C)CN(C)C(C2(C)CCCC2(F)F)=O)CCC(C)(C)CC1 5267,N1(C(C(C)CSCC#N)=O)CC(NC(=O)CCC2CCOCC2)C(C)C1 5268,CC1CN(S(=O)(=O)N(C)Cc2ccccc2)CCN1C(=O)CC(C)(C)C 5269,C1(COC)(NC(c2nn(C)cc2Cl)=O)CCN(C(c2nccc(C)n2)=O)CC1 5270,c1(CN(C2CC3CC2CN3)CCc2cc(C)[nH]n2)ccc(Cl)cc1 5271,c1(CC)cccc(C)c1C(N1CCN(C)C(CCNC(C2CC(OC)C2)=O)C1)=O 5272,c1(C(N2CCCN(C(=O)C(C3CC3)C3CC3)CC2)=O)cc2c(nc1O)CCOC2 5273,Cc1cnc(C#N)nc1N1CCCC1CNC(C1(C)CCCS1(=O)=O)=O 5274,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1ncccc1Br)=O 5275,c1(C(=O)NCC2N(C(c3cnc(COC)s3)=O)CC2)ccc(Br)nc1O 5276,C(=O)(CC(F)(F)Br)N(C1CCN(C(C2CCN(C)C2C)=O)C1)CC 5277,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)oc(C)c2C)=O)CC(F)(F)C1 5278,C1(C(=O)NC2CCN(C(=O)C(O)C3CCC3)CC2)CCCc2ccccc2C1 5279,Cc1cnc(N2CCC(CCCO)C2)c(S(=O)(=O)N(CCCC(C)C)CCO)c1 5280,CC1(C)CN(C(c2cnc[nH]2)=O)CCC1NC(C1CC2(CC2)CO1)=O 5281,C(C#Cc1cccnc1)NC(C(COCC)NC(C1CN(C)CCN1C)=O)=O 5282,N1(C(C2CC(C)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5283,N1(C(C(C)OC(C)(C)C)=O)CCN(C(c2ccnn2CCF)=O)C(C2CC2)C1 5284,C1(C(=O)NCCOCC(C)C)COCCN(C(C2CC(F)C2)=O)C1 5285,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5286,c1(C(N(C2CCN(C(C3CC3OC)=O)C2)CC)=O)ncccc1C(C)(C)C 5287,c1(COC(C)C)cccc(C(=O)NCCNC(=O)CN2C(=O)CCC2=O)c1 5288,C1(C(N2CC(Cc3nccc(OC)c3)C2)=O)CC12CCCOC2 5289,CCC(CC(C)C)C(=O)NCCC(C)N(C)C(c1ccsc1C#N)=O 5290,Cc1nc2n(c1CCC1CCC(CNC(=O)OC(C)(C)C)CC1)CCCC2 5291,n1(CC=C)cc(C(=O)NCC(C)N(C)C(C2CCN(c3nccn3C)C2)=O)cn1 5292,C1(NC(C2CCN(CCC)C2)=O)CCC2CN(CCCc3cnn(C)c3)CC2C1 5293,c1(NC(C2C(CNC(CN(C(CC)C)C)=O)C2)=O)cc(OC)ccc1F 5294,N1(C(CN(C2CCCC2)C)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5295,c1(C(=O)NCC23N(C(CC(=C)C)=O)CCC2CC3)noc2c1CC(C)(C)CC2 5296,CCC(C)C(C(=O)NCC1COC(C)(C)C1)NC(=O)CN(C)C1CC1 5297,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CC)CCN(C(C2CNC(=O)C2)=O)CC1 5298,CCCCCCC(F)C(=O)N1CCCC1CN(C)C(c1cncc(OC)c1)=O 5299,c1(N(C(C)C2CC2)Cc2ccc(F)cc2)nccc2nn[nH]c12 5300,C=CCC(CNC(c1ccnc(O)c1)=O)C(=O)NC1(CO)CC2CCCC12 5301,N1(C(CCC(C)OC)=O)CC2CN(C(=O)C=Cc3cn(C)nn3)CC2C(F)(F)C1 5302,N1(C(CCCC#C)=O)CC(C)N(C(c2cnc(C3CCC3)o2)=O)CC1C 5303,N1(CC(C)C)CCC(c2nc(CC3CC4CCC3C4)n(-c3ccnc(F)c3)n2)CC1 5304,C#CCC(CC(=O)N(C)CC1(OCC)CC1)NC(C1CCN1CC)=O 5305,C1(CC#C)(C(N2CC(n3ccnc3)C2)=O)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5306,Cc1cnc(C(N2CCC(CN(C)C(C3CC3CF)=O)CC2)=O)cc1C#N 5307,C1(C(N(CCC#C)CCO)=O)CN(C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 5308,Cc1cc(C(C)N(C)C)cc(C)c1F.C12CCN(C1)C(=O)N2 5309,c1(C(N2CC3CC(CNC(c4n(C)c(S)nn4)=O)C3C2)=O)cc2cccnc2[nH]1 5310,c1(CC(=O)NCCN(C(c2c(CC)cco2)=O)C)csc2nccn12 5311,N12CCCN(CC1)C(=O)OC(=O)C=CC=C(OCC)C(CC)N2C 5312,c1(C(=O)NC(C2(CNC(C3CC3C(F)F)=O)CC2)C)cnc2ccccn12 5313,Cc1nn(C(C)C)cc1C(=O)NCCC(C)NC(C1CCC(=O)N1)=O 5314,c1(N2CC(CC(=O)OC(C)(C)C)OCC2)c(Br)cncc1[N+](=O)[O-] 5315,c1(C(=O)NCC2C(CNC(Cn3ncc(C)c3)=O)C2)ncccc1Br 5316,c1(C(=O)NC2(CNC(c3ncncc3Cl)=O)CCOC2)cn2ccccc2n1 5317,CC(CNC(=O)C=C=C(C)C)C(F)C(=O)NCCCc1ccnn1C 5318,c1(CCC)cc(C)ccc1CN1CCNC(=O)C1c1cccc(Cl)c1 5319,C1(CC(N2CCC(N(C(C3CC(F)C(=O)N3)=O)CC)CC2)=O)CC2(CCO1)CC2 5320,C(=O)(C#CC1CCCC1)NCC1N(C(Cc2c(C)noc2Cl)=O)CC2(CC2)C1 5321,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2CC(c3cccnc3)C2)=O)C1 5322,c1(C(=O)O)nccc2c1CN(CC(N1CCCC1c1ccccc1F)=O)CC2 5323,c1(C(N(CC(CNC(c2c(C)ccc(C)n2)=O)O)C)=O)cc2cc(F)ccc2o1 5324,C1(OCC(=O)NCC2CN(C(C3SCCCS3)=O)C2)CCCOC1 5325,C(=O)(C1Cc2ccc(Cl)cc21)NC(C)C(C)(C)NC(c1cn(CCO)nn1)=O 5326,N1(C(c2c(CCC)n[nH]c2)=O)CCC2(CCN(C(C3(CC(F)F)CC3)=O)C2)C1 5327,CCCCCC(CC)C(=O)NC1CCCN(C(c2cc(N)cc(F)c2)=O)C1 5328,c1(C(N(C2CCCN(C(C34CC(F)C3C4)=O)C2)CC)=O)noc2c1CCCCC2 5329,CC1CC(N(C)C(C2CCN(c3ccnn3C)CC2)=O)CCN1 5330,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5331,C1(C(=O)NC(CC(=O)NC)C)(COC)CCN(C(=O)C=Cc2cocn2)C1 5332,C(C1=CCCCC1)(C(=O)O)NC(=O)NCc1cc(CC)no1 5333,C1(F)(CNC(c2cnc[nH]2)=O)CC2CCC(C1)N2C(c1noc2ncccc12)=O 5334,C(=O)(C(F)C(C)C)NC(C(=O)N(CCN(C)CC)CC)C1CCCC1 5335,CC(C(C(=O)O)NC(=O)Nc1nc(COC(C)(C)C)no1)c1ccccc1 5336,C1(NCC(=O)N(C(C)C(c2ccccn2)=O)C)CCNCC12CC2 5337,C(CCCCO)N(C)C(c1cc(CNC(=O)CCc2cccn2C)cs1)=O 5338,C1(NC(C(C)C2CCCC2)=O)CN(C(C2CCCCC2O)=O)CC2(CC2)C1 5339,C1(CNC(c2c(C(C)C)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5340,N1(C(C(CC=C)C(C)C)=O)CCN(C(=O)CCS(N)(=O)=O)CC(C)(F)C1 5341,c1(C(C)CCC(F)(F)F)ccccc1C(=O)NC(CNC(=O)NC)(C)C.C1CC1 5342,N1(C(CSCC(=O)OC(C)(C)C)=O)CC2CC2(CNC(C2CC2(C)C)=O)C1 5343,CC1CC(NCC(C)(C)F)CN(C(c2ccc(Cl)cn2)=O)C1 5344,N1(C(C(=O)Nc2cc(C(=O)OC)n(C)c2)=O)CCS(=O)(=O)C2(CCCC2)C1 5345,n1(CC)cc(CCCC2C(NC(=O)OC(C)(C)C)CC2)nn1.C12(CC1)C(=O)N2 5346,CC(F)(F)CC(=O)NC1CCC1NC(=O)COc1ncccc1C(F)(F)F 5347,N1(C(C(C)NS(C)(=O)=O)=O)CC(O)CC1CNC(C1CCC(CO)CC1)=O 5348,Cc1cncc(C(=O)NC2CN(C(c3cn(C)nn3)=O)CCC2C(F)(F)F)c1C 5349,c1(CC(=O)NC2C(NC(CCN3CCN(C)CC3)=O)C2)ccc(C(N)=O)cc1Cl 5350,c1(CCC)cc(C(=O)NCC2CCN2C(c2c(OC(C)=O)c[nH]c2C)=O)cc(O)n1 5351,CCCCC(C(=O)NC(c1cnn(C)c1)C(=O)NC(Cn1cncn1)CC)OC 5352,c1(C(C(=O)N(CC=C)CCF)N(C(=O)OC(C)(C)C)C(C)C)cncnc1 5353,N1(C(CCc2cccc(OC)n2)=O)CCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 5354,C1(CCC)CCCN(C(c2ccc(CNC(c3ccoc3)=O)o2)=O)CC1 5355,N1(CCC(=O)NC2CCC(NC(C3(F)CC3Br)=O)CC2)CCNC(=O)C1 5356,Cc1cccc(CCC(=O)NCC(C)(C2CCC2)NC(c2ccnc(C)c2)=O)c1 5357,CC1(C)CCC2(CCCN2C(c2cccc(S(=O)(=O)NCCO)c2)=O)CC1 5358,C1(C(=O)NCCC(C(C)C)NC(C2CC2C)=O)CN2CCN1CC2 5359,c1(C(=O)NC(C2CCCN2C(=O)CCCF)(C)C)c[nH]c2ncccc12 5360,n1(CC)ncn(NC(=O)CN(C(c2cc3n(n2)CCC3)=O)C2CC2)c1=O 5361,CCC(C)C(C)C(=O)NCC1(C)CCN(C(c2cn(C)nc2O)=O)C1 5362,N1(C(C2N(C(c3csnn3)=O)CCC(=C)C2)=O)CCN2CCCCC2C1 5363,CCCCC(C(=O)NC1CCCN(C(c2cc(C)ncc2C)=O)C1C)C(C)C 5364,CN=c1cc(C(=O)NCc2cc(C(=O)NC3CNC(=O)C34CC4)n(C)n2)cc[nH]1 5365,c1(OC(C)C)ccc(COC(=O)CC2(NC(=O)C(C)N=[N+]=[N-])CC2)cc1 5366,Nc1c(C(N2CCCC2CNCc2ccc(F)c(O)c2)=O)nc(O)nc1O 5367,C1(O)(C(N2CCCC(CCNC(CCC=C)=O)C2)=O)CCCC(C)(C)C1 5368,C(=O)(C1CC=CC1)NCc1ccc(C(=O)NCCC(=C)C)s1 5369,C1(C(N(CC(CC)NC(c2cc(C)ccc2N)=O)CC)=O)CCc2nncn2C1 5370,Cc1nc2ccc(-c3nc(C4CCCC4(F)F)nn3C3(C)CCS(=O)(=O)C3)cc2[nH]1 5371,C1(NC(=O)CCc2cnccn2)COC2(C1)CN(C(C1CCCO1)=O)C2 5372,c1(C(N2CC(NC(C3(CC)CC3)=O)C(OC)C2)=O)ccc(O)c(CCOC)c1 5373,c1(C(N2C(C3(NC(c4n(CC)cc(Cl)c4)=O)CC3)CCC2)=O)n[nH]c2c1CC1CC21 5374,CCCCC(C)CCC(=O)NC1CC(NC(=O)C(C)c2ccsc2)C1 5375,c1(OCCC(=O)NC2CCC2NC(c2cc(Cl)no2)=O)ccc(Br)cc1F 5376,CCC(C)CC(C)C(=O)N1CCC(N2CCC(NC(C3CC3C(C)O)=O)CC2)C1 5377,C1(C(N(C)C)=O)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 5378,c1(C(C)=O)cc(C(=O)NCC2CCC(NC(=O)CCOC3CCOCC3)C2)cs1 5379,C=CCN=C(NCCCC1CC1(Cl)Cl)N1CCC(NC(=O)C(C)C)CC1 5380,N1(C(CCC(=C)Cl)=O)CCC2CCN(C(=O)Cn3cc(C(C)=O)nn3)C2C1 5381,N1(C(c2c(C)cco2)=O)CC(NC(=O)CCc2cncc(Br)c2)C(F)(F)C1 5382,N1(CC(CC)OC)CCCN(c2cc(NC(=O)C(F)C(C)C)ncn2)CC1 5383,C1(CN(C)C(c2cccc(C3CC3)n2)=O)CN(C(=O)C2=C(Cl)CCC2)CC12CC2 5384,S(=O)(=O)(c1ccc2c(c1)OCC(=O)N2C)N1CCC(NC(N2CCC(C)CC2)=O)C1 5385,c1(C(=O)NC(C(C)C)CNC(c2cnoc2C2CC2)=O)cccc2nncn12 5386,N(C1CCc2ccc(Br)cc21)C(C(N1CCCC(CCC(C)O)C1)=O)=O 5387,N1(C(c2c(C)cnnc2)=O)CC2CCCC(CNC(C3(C)C=CCC3)=O)(C2)C1 5388,C(=O)(CC(C)(O)C(F)(F)F)NCC1OCCN(C(C=C(C)c2ccccc2C)=O)C1 5389,c1(NC(C2CC(NC(c3cncc(C)c3)=O)C2)=O)ccc(Br)c(Cl)c1F 5390,c1(C(=O)NC(C)C(C)NC(c2cncc(C(N)=O)c2)=O)cnc(N(C)C)c(Cl)c1 5391,c1(OC)ccc(NC(C2(C)CCCN(Cc3cccc(F)c3)C2)=O)c(F)c1 5392,C1(NC(CC)=O)CC2CCC1N2C(=O)C(O)CC1CCCC1 5393,CCCCC(C(=O)NC1CCC(NC(c2ccc(F)cn2)=O)C1)C(C)C 5394,C1(CCNC(CCOCC#C)=O)CC(F)(F)CN1C(=O)C(CC)NC(N)=O 5395,CCC(C)CC(C(=O)NCc1cncc(F)c1)NC(c1c[nH]cc1C)=O 5396,C(=O)(CC(C)(C)CNC(=O)CN1CCOCC1)NC1(C)C(C)CCC1 5397,N1(C(C)C(=O)NCc2cccn2C)CC(c2cc[nH]n2)C(C)C1 5398,C1(F)(CNC(C(C)OCC)=O)CCCN(C(C2(CO)CCCCC2)=O)CC1 5399,C1(NC(C2(OCC)CCC2)=O)CC(O)CN(C(=O)CC2CCC3(CCC3)O2)C1 5400,C1(C(=O)NCC(CCNC(=O)C=CCF)OC)CCc2nn[nH]c2C1 5401,CC12CC(C(=O)NC3CN(C(C4(O)CCSCC4)=O)CC34CC4)(C1)C(C)(C)O2 5402,N1(C(C(CC=C)(C)C)=O)CC2(CCN(C(C3C=CCS3)=O)C2)C1 5403,C1(NC(c2nc(COC)sc2)=O)CC2(C1)CC2NC(=O)C(c1ccc(C)s1)C 5404,N1(C(CC2C(CC)C2(F)F)=O)CCC(=CC(=O)NCC2CC(=O)N2)CC1 5405,CC1CCN(C(=O)C(C)Sc2ccc(Cl)cc2Cl)CCN1C(C1CC1C#N)=O 5406,CC(C)C(C)C(=O)N(C(=O)CN1CC(c2ccccc2)C(O)C1)CCO 5407,C(=O)(CN=c1[nH]c(C)cs1)N(C)CC1(O)CN(C(c2c(OC)ncc(C)c2)=O)C1 5408,CCC(CC)C(C)C(=O)N1CCN(C(=O)C(=O)NCC2CC2)CC1CC 5409,CC12CCC(C(=O)NC3CC(O)CN(C(c4cc(F)c[nH]4)=O)C3)(CC1)CO2 5410,C(=O)(CC1=CSC2=NCCN12)NCCCC(C)NC(C1COC(=O)C1)=O 5411,N1(C(c2ccnc(C)n2)=O)CC2CCN(C(c3ccoc3C3CC3)=O)CC2C1 5412,c1(C(N2C(CN(C(CCOC)=O)C)COCC2)=O)cccc(Cl)c1SC 5413,C1(C(=O)NCCNC(c2cnn(CCC)c2C2CC2)=O)CCC2C1C2(F)F 5414,c1(C(N2CCCCC2COC)C(=O)NCC)ccc2c(c1)C(=O)NC2=O 5415,CC1(C#CC(=O)N2CCC(NC(=O)CSC3CC3)C2)CCCO1 5416,c1(C(N(C2CCCN(C(C3(OCC)CC3)=O)C2)C)=O)nc2c(cc1Cl)OCCO2 5417,c1(C(N2CC(C)C(CNC(=O)CCS(N)(=O)=O)C2)=O)cc2c(cnn2C)nc1O 5418,C1(NC(C2C(CC)OCCC2)=O)CCSC12CN(C(c1cncn1C(C)C)=O)C2 5419,C1(C(CNC(C=CSC)=O)(C)O)CCCN(C(c2ncsc2C)=O)C1 5420,CCCS(=O)(=O)c1ccccc1C(N1Cc2nnc(O)n2CC1CC)=O 5421,c1(CNS(C)(=O)=O)cn(C)nc1C(C)NCC(C)Cc1n(CCCOC)nnn1 5422,C#Cc1ccc(C(=O)NC)nc1.c12c(C)nn(C)c1[nH]c(=O)[nH]2 5423,C1(C(=O)NCCCN(C)C(C2(C#N)CC(C)C2)=O)CS(=O)(=O)CC12CC2 5424,CCN=C(NCC12CC(CCO1)C2)NC1CCCC(C(C)C)C1 5425,c1(C(=O)Nc2scc(CN3CCN(CCC)CC3)n2)ccc(S(C)(=O)=O)nc1 5426,N1(C(Cc2ncc(C)s2)=O)CC(=O)NC1c1ccccc1 5427,N1(C(c2c(CC)n(C)nn2)=O)CC2(CCN(C(=O)C(C)(C)c3cc[nH]n3)CC2)C1 5428,C1(C(N2CCC(NC(CNC=O)=O)C(O)C2)=O)CN2CCCCC2CO1 5429,C1(CC)CCCCC1NC(=O)C(CCNC(=O)CCc1ccncc1)NC(C)=O 5430,Cc1c(C(=O)NC2CC23CC(NC(C2C4CCC(F)(F)C24)=O)C3)cccc1Cl 5431,CC(CCCC(=O)N1CCOC(C(C)(C)C)C1)NC(=O)COc1ccsc1 5432,C1(C(N(CCCNC(C(C)OC)=O)CCO)=O)CC(=O)NC(=O)N1 5433,C1(NC(CC2(OC)CCCC2)=O)C(C)CN(C(c2cc(C)sn2)=O)CC1C 5434,N1(C(c2cncc(CC)c2)=O)CCC2(CC1)CC(C)N(C(=O)C(F)C1CCC1)C2 5435,N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2ns[nH]c2=O)=O)CC12CCC2 5436,c1(C(N(C2CCN(C(C(C)C(F)F)=O)C2)CCO)=O)ccc2cccnc2c1 5437,C(C1CN(C(c2n[nH]cc2[N+](=O)[O-])=O)Cc2ccccc21)NC(C1=NOC(C)C1)=O 5438,N1(CCC(=O)NC(C)Cn2cc(C(C)(C)CC3CC3)nn2)CCC(C(N)=O)CC1 5439,c1(N2CC(F)CC(OC)C2)nc2cc[nH]c2c(=NCc2ccc(Cl)cn2)[nH]1 5440,c1(C(N(C2CC(NC(C3CCCC4(CC4)C3)=O)C2)C)=O)cc2c(cn1)COCC2 5441,CCC(C)(CNC(=O)CC(C)N(C)C)C(=O)NCC1(CO)CC12CCC2 5442,C(=O)(C(C)(C)C1CCCN1C(C1CC(C)(O)C1)=O)N(CCOCC#C)C 5443,C1(N(C)C(c2ccc(C3CC3)s2)=O)CCC(NC(C2CC(=C3CC3)C2)=O)CC1 5444,C1(C(N2CC3COCC3C2)=O)C2CCC(C2)N1C(C12CC(CO)(C1)C2)=O 5445,S(=O)(=O)(c1ccc(C#N)c(NCC2CCC(CC)O2)c1)NCC(C=C)(F)F 5446,c1(SCC(=O)NCC=CCNC(C2=C(C#N)CCC2)=O)ccc2c(c1)OCCO2 5447,N1(C(CN2CC(CC)C2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5448,CC1CCCc2c(C(C(Cc3cn(C4NC(=O)CC4(C)C)nn3)C(=O)O)=O)cnn21 5449,N1(C(c2cccc(C(C)=O)c2)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 5450,C(=O)(CCCS(N)(=O)=O)N1C(C(N2CCC(CCOC)(CC)C2)=O)CC(OC)C1 5451,C(=O)(C(O)CNC(=O)CC1CC1)N(CCC)CC1CC1 5452,Cc1ccccc1CC(=O)N(CC(C)CNC(c1ccc(SC(F)(F)F)s1)=O)C 5453,C1(NC(CCCSC)=O)CC2CCC(C1)N2C(c1cccc(Cl)c1F)=O 5454,c1(C(N2CCC(C)C(NC(=O)CSS(C)(=O)=O)C2)=O)cc([N+](=O)[O-])cnc1N 5455,c1(CNC(=O)NC(C2CCC2)C)cccc2cccnc12 5456,Cc1nn(C)c2ncc(S(=O)(=O)NC(CSC3CCCCC3)C3CC3)cc12 5457,c1(C(=O)NC(CNC(c2c(C)con2)=O)(C)CC)cc2c(C3CC3)cccc2[nH]1 5458,C(N=C(NCCC(F)(F)C(F)(F)F)N1CCC(O)CC1)c1n(C)ccn1 5459,Cc1nnc2n1CCCC2C(=O)N1CCC(CNC(=O)C2=CCCC2)C1 5460,N1(C(C=CC=CCC)=O)CC(C)C(NC(=O)COc2c(C)ncnc2C)C(C)C1 5461,C(=O)(CC(C)(C)C(=O)OC)NC1(C(=O)NCc2cnc(CC)s2)CCC1 5462,c1(C(=O)OC)cc(=NCCCCNC(c2c(C)nn(C)c2C)=O)[nH]cn1 5463,C(=O)(CCCCCNC(=O)C(c1nc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5464,CN1CCN(C(C)(C)C(=O)NC2CC(NC(c3cc(O)nc(CO)n3)=O)C2)CC1=O 5465,Cc1cc(F)cnc1C(=O)NCCC1CCCCN1C(C1C(C)OC(C)C1C)=O 5466,N1(C(C2C(C)(C)C2C#N)=O)CC23CCCC2(C1)CN(C(=O)CCOC1CC1)C3 5467,N1(C(C(COC(C)C)NC=O)=O)CCCN(C(c2coc3c2CSC3)=O)CC1CO 5468,C12(CNC(C(C)N(C)C(C3CC(CC4CC4)C3)=O)=O)CCCCC1C2 5469,C(C(C(=O)N1CC(OCC)C1)OC1CN(C(=O)Cc2ccccc2)C1)NC 5470,N1(C(CN(C)N2CCCCC2CCF)=O)CCC(C2CCC2)CC1 5471,N1(c2ncc(Br)c(C)c2F)CCC(OC(F)F)C(F)(F)C1 5472,C(=O)(C(F)(F)C1CCOCC1)NCCCN(C(C1C(CCC)C1)=O)C 5473,c1(OCC)ccc(S(=O)(=O)N2CCCC(CNC(c3ccc[n+]([O-])c3)=O)C2)cc1 5474,C(=O)(C(Cl)=CCl)NCCN(C(C)C)C(c1cn(C2CCCCC2)nn1)=O 5475,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5476,c1(C(c2nnnn2CCCNCC2CC2)NCC(C)(C)C(F)F)ccc(F)cc1Br 5477,c1(C(N2C(CN(C(=O)C(C)(O)c3ccccc3)C)CCC2)=O)ncccc1Cl 5478,N1(CCN2CCC(NC(C(C)Cc3ccccc3)=O)CC2)CCc2ccccc21 5479,N(C(=NCCCOc1ccccc1OC)N1CCC(F)(F)C(C)C1)CCOC 5480,c1(NCc2ccc(OCCC)cc2)c(OC)ccnc1F 5481,c1(N(C)C(C2CC2C(=O)Nc2ccn3ccnc3c2)=O)cc2ccccc2n1C 5482,c1(CC)ccoc1C(=O)N(CCCCNC(=O)C(C)(C)c1cccnc1)C 5483,C1(CNC(CCOC(C)C)=O)CCCCC1C(=O)N(CCCCOC)C 5484,c1(C(=O)OCC(c2ccccc2)NC(C2CC(C(=O)O)C2)=O)cncc2nc[nH]c12 5485,c1(CC)cc(C(N2CCC3CC23C(=O)NCc2noc(C)n2)=O)c(C)o1 5486,N1(C(c2cc(F)cnc2O)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5487,C(=O)(C1=NOC(C)(C)C1)N(CC(CNC(c1cc(COC)[nH]n1)=O)(C)C)C 5488,CCC(C)C(O)CC(=O)NCCCOCCC(=O)NC1CC(=O)N(C)C1=O 5489,N1(C(C=C(C)C(F)F)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5490,C=CC(C)(C)CCN=c1nc2sccc2c(N(CC(C)Oc2ccccc2Br)C)[nH]1 5491,CC1CCN(C(=O)CCOCc2ccccc2)CCN1C(=O)Cc1sccc1Cl 5492,C1(C(C)C)CCC(C)CC1C(=O)NCCC1CC(NC(=O)CN=S(C)(C)=O)C1 5493,C1(CNC(=O)C=Cc2ncc[nH]2)CN(C(C2(C3CCC3)CC2)=O)CCC12CCC2 5494,c1(C(N2CC(NC(Cn3c(C)ccc3C)=O)C(C)C2)=O)cc(Cl)c(Cl)n1C 5495,N(C1CCS(=O)(=O)c2ccccc21)C(c1ccc(C)cc1)c1nnnn1C 5496,CC1CCCC(CC(=O)NCCOC2CCN(C(c3cnc(N)cn3)=O)C2)C1 5497,C1(N(C(Cc2c(CC)noc2CC)=O)C)CN(C(c2ccc(C)s2)=O)CCC1C 5498,C(CN=C(NCC(c1ccncc1)OC)N(C)C(C)C)c1cc(OC)ncc1 5499,N1(C(C2CCCC(NC(c3ccccc3)=O)CC2)=O)Cc2cccc(O)c2C1 5500,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ccc2F)CC)ccc(N)cc1F 5501,C1(C(N2CCC23CCCCC3)=O)CCN(C(=O)Cn2ccnc2)O1 5502,N1(C(=O)NCC(CCC)CCC)CC2CC3CC2C1C3O 5503,N1(C(C2C=CCN2C(=O)CN2CSCC2=O)=O)CCC2(CCOC2=O)C1 5504,Cc1cc(C2CC2)ncc1C(=O)NC1CC(CCNC(C2(C)CCCN2C)=O)C1 5505,N1(C(c2ccc(C)o2)=O)CC2CCC1CN(C(=O)C(C)C1CC1)C2 5506,c1(C(N2CC(CC(CNC(CC3ON=C(C)C3)=O)(C)C)C2)=O)cc(C)nc(O)n1 5507,c1(C(N(CC(=O)NCC2CC23CC3)CC#C)=O)cccn1CCC 5508,C(=O)(C(C)(C)C(C)(C)C)NCC1C(C)CN(C(=O)Cn2cnnc2)CC1 5509,C1(CCNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O 5510,C1(NC(C(N2CCOCC2)C)=O)CN(C(=O)CC23CCCC2C3)CC12CCCC2 5511,CC1CN(C(c2csc(Cl)n2)=O)CCC1NC(C1(c2cnco2)CC1)=O 5512,N1(CC)CCN(CCC(N2CCC3C(NC(c4ccc(N)cn4)=O)C23)=O)CC1 5513,C1(C(N(c2nc(N3CCC(COC)CC3)nc(C)c2)C)=O)Cc2ccncc2C1 5514,c1(C(=O)NCCCOCCOCCNC(C2C(=C)CC2)=O)ccoc1CC 5515,C=C1CC(C(N2CC(CC(=O)N(CCN(C)C)C)(OC)C2)=O)(C(=O)NC)C1 5516,C12C3CC1N(C3)C(=O)c1cc([nH]n1)NC2=O.C1(CN(C)C)(CO)CC1 5517,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(c2ccncc2)=O)C1(C)C 5518,c1(C(=O)NC(CCCNC(C(C)SCC)=O)(C)C)ccc2cnc(C)n2c1 5519,CCC(C)(O)Cc1cn(CC2CCN(C(=O)CC3CC(=O)C3)C2)nn1 5520,c1(OCC)ccc(Cl)nc1C(=O)NCc1cccnc1CNC(=O)C(F)(F)CO 5521,c1(CCC(=O)N(C)CC=CC(N2CC(O)(C3CCCC3)C2)=O)cncc(O)c1 5522,C(CC(C(=O)NCCOCCNC(c1csc(Cl)n1)=O)OC)OC 5523,c1(CNC(CN(C(C(C)n2cccn2)=O)CCO)=O)ccnc(N(C)C)c1 5524,c1(CCN2CC(O)(CNC(CN3CC(C)(C)C3)=O)C2)oc2ccccc2c1Cl 5525,C1(CNC(C(C)=C2CC2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)CC1(F)F 5526,c1(C(N2CC(OCCNC(=O)Cn3cccnc3=O)C2)=O)cnc2[nH]nnc2c1 5527,N1(C(c2nc(-c3c(CC)cccc3)[nH]n2)=O)CCNC(=O)C1c1ccccc1 5528,C=CCCC(F)(F)C(=O)NCC1CN(C(=O)CN2CCCNC2=O)CCC1C 5529,C1(NC(C2N(C(C)=O)CCC2)=O)CC2CC1N(C(=O)Cc1ccccc1O)C2 5530,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CC3CC(F)(F)C3(C)C)CCC12 5531,c1(C(N2CCC(C(C)NC(=O)C3=CCOC3)C2)=O)coc2ccc(Cl)cc12 5532,c1(COC)ccoc1C(=O)NC1CCCC1CNC(=O)CC(=O)NC 5533,Cc1ccc(NC(=O)C(=O)NC2C3CN(C(=O)C(C)OCC4CC4)CC23)cc1 5534,N1(C(c2c(C)cns2)=O)CCN(C(=O)C#CC(C)(C)C)CC(O)C1 5535,N1(Cc2cc(OC)c(I)cc2)Cc2[nH][nH]c(=NC(=O)c3cnn(C4CC4)c3)c2C1 5536,C1(C(F)(F)F)(NC(=O)C2CC2)CCN(C(C23CCCC2CC3)=O)CC1 5537,CC1CCC(C)CN1C(=O)C(=O)NC(c1ccccc1F)c1nnc(CO)s1 5538,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCNC1(NC(CCOC)=O)CCCC1 5539,C1C(CC(C)C)C(=O)N1.C(CC)(CC(=O)OC)NC(C=CC(CC)C)=O.OC 5540,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)c1ccccc1 5541,c1(C(N2CC(C)C(NC(c3ccc(CO)cn3)=O)CC2)=O)cccc2cnsc12 5542,C(CC(F)F)(C(=O)N(CC(O)C(C)(C)C)C)NC(c1c(C)non1)=O 5543,c1(C(=O)NCC(Cc2ccc(C)cc2)F)cc2c(Br)cncc2[nH]1 5544,Cc1cccc(C(N2CC=CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)n1 5545,n1(CC)ncc(C(N2CCC(COC)(NC(=O)CCCN3CCCC3)C2)=O)c1C 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5564,c1(CNC(=O)NCCOCC(=C)C)c(C)c(Br)c(C)c(C)c1C 5565,C(=O)(C(C)CNC(C1(N(C)C)CC1)=O)NC(C)C(F)F 5566,CC1CC2(CCO1)CC2C(=O)NCC1CCN(C(c2c[nH]ccc2=O)=O)CC1C 5567,N1(N(C)C)CCC(F)(C(=O)NC2C3CN(C(=O)CSc4ccccc4)CC23)C1 5568,O=C1CCCC(c2ccccc2)(COCCCF)N1 5569,N1(C(C(C#N)=CC(C)C)=O)CC2(CCN(C(C3CCC4CC3C4(C)C)=O)CC2)C1 5570,C(C(O)C(=O)NC(C(=O)Nc1cc(C)[nH]n1)C1(O)CCC1)SC 5571,C12(CNC(=O)CC3CCC34CCC4)CCCC1N(C(=O)CN1CCCC1)CCC2 5572,c1(C(=O)NC(C)CN(C(=O)CN2CC3CC3C2)C)ccc(Cl)c(N)c1Cl 5573,C1(C(=O)NCCC(=O)NC(c2ccco2)C#C)CC2C=CC1C2 5574,C1(NC(C(CC)NC(=O)C(C2CCOCC2)F)=O)CC2OC(=O)CC12 5575,C(=O)(C(=O)CC(C)C)NCC1(C(C)NC(Cc2cn(CC)nc2)=O)CC1 5576,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)C)=O)cncc(Cl)c1C 5577,C1(NC(C=C(C)Cl)=O)CCCC(NC(=O)CCn2ccnc2)C1 5578,c1(C(N2CC(CN(C(=O)CC(C)(C)O)C)C2)=O)ccnc(C(F)F)c1 5579,c1(C(N2CC(NCCCOC)OCC2)=O)ccc2c(C3=CCOC3)n[nH]c2c1 5580,Cc1nc2nc(=S)[nH]n2c(C)c1CC(=O)NC(C)C(C)NC(=O)C(F)F 5581,C12(NC(C(C)CN3CCOCC3)=O)CCC(CNC(=O)C(C)C3CC3)(C1)OC2 5582,N1(C(CCCc2cc(C)no2)=O)CCC(NC(C2SCCCS2)=O)C(O)C1 5583,c1(C(C)=O)ccc(N2CCOC(C(C)NC(c3snc(Cl)c3Cl)=O)C2)nc1 5584,c1(CNC(C(C2CCCN(C(CCSC)=O)C2)(C)C)=O)cnc(F)cc1C 5585,C(=O)(CC1=CCN(C(c2cc(O)cc(=O)o2)=O)CC1)NCc1cccc(C)c1C 5586,Cn1nnnc1C(c1ccc(C(F)F)s1)NCC1CC(F)C1 5587,CC(C)CCCC(C)CNC(=O)CC1C2CN(C(=O)CC34CCCC3C4)CC12 5588,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5589,C1(NC(c2cnn(CC)n2)=O)CC(C)CN(C(=O)C=C(C)I)C1 5590,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5591,N1(C(Cc2c(C)cnn2C)=O)CCCCCC1C(N1CCC2CCCC12)=O 5592,C1(F)(CNC(C2C(c3n(C)ncc3)C2)=O)CCC(CNC(=O)COC2CC2)CC1 5593,C(C(=O)OC)(C(C)(C)O)NC(C(CC)COC)=O 5594,C1(NC(c2c(C)onc2C2CC2)=O)CCN(C(c2ccc(N)c(Cl)c2)=O)CC1F 5595,Cc1c(C(=O)NC(C(N2CC(O)(CC(C)C)C2)=O)C2(C)CC2)ccn1C 5596,N1(C(C(=O)NCC)=O)CC2(CC2)CC1CNC(=O)CC1COC(=O)C1 5597,C(=O)(C1=CC2(CCN(C(C3CCOCC3)=O)CC2)OC1)N1CCCC(OCC)CC1 5598,N1(C(c2n(C)nc(O)c2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(O)C1 5599,CC1(C)CC(O)(CC(=O)NCC(C2CC2)NC(C23CC(C)(CO2)C3)=O)CO1 5600,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 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5619,C(c1ccc(F)c(F)c1)=CC(N1CCC(C)(NC(c2c(C)con2)=O)C1)=O 5620,C1(NC(c2c(C)nns2)=O)CC2CCC1(N=c1[nH]c(C(C)C)nc3[nH]cnc13)C2 5621,c1(OC)cc(C(N2CCC(NC(=O)Cc3coc(C)n3)C(C)C2)=O)ccc1Cl 5622,c1(C(=O)NCC(CC)(CC)NC(C2CCCC(C)C2)=O)nc2cccnc2s1 5623,c1(NC(C(C)NC(=O)OC(C)(C)C)C2CCC2)cnccc1Cl 5624,N1(CC)CCOCC1C(=O)NCC1C2CN(C(=O)Cc3c(C)n[nH]c3C)CC12 5625,c1(CN(C2CCCC2)C(=O)CN2CCC(O)(CO)CC2)cc2cc(Cl)cnc2o1 5626,c1(C(N2CC(CNC(=O)Cn3cccc3)C3(C2)CC3)=O)cc2ccccc2[nH]1 5627,CCN=c1[nH]c(C(N2CCCC2CCNC(=O)CN(C2CC2)CC)=O)cs1 5628,c1(C(N2CCC(N(C(C(C)OCC=C)=O)C)C2)=O)ccc(OC)cc1OC 5629,C(=O)(C(C)(C)C1CCOC1)NCCOC(CNC(C(=O)N(C)C)=O)(C)C 5630,c1(C(N(C(CCNC(Cc2cccc(C)c2F)=O)C)C)=O)cc2c(o1)CCCC2 5631,C(=O)(C(Cc1ccccc1)N(C(=O)CCCCN)C(C)C)OC 5632,C1(C(=O)NC2CCN(Cc3nc(-c4ccccc4)no3)C2)CC2CCC1O2 5633,C(=O)(C(C)(O)CNC(=O)CCC1CCCN1C(=O)CC1(C#N)CC1)OC 5634,c1(C(N2CC(O)(CC)C2)=O)cncc(C(=O)OC(C)(C)C)n1.C1(=O)N(C)N1 5635,c1(C(N(CCOC)CCNC(C2CCC(C)CC2)=O)=O)ncc2ccccn12 5636,C(=O)(C(C)(CC)CCCC)NCCC1(C(C)(C)C)N(C(CCCCOC)=O)CCC1 5637,c1(C(N2CCC(NC(c3cc(OCC)no3)=O)C(C)C2)=O)cccc2sncc12 5638,c1(-c2nn(CC3CC(C)C3)c(C3CC4C(C3)C4(F)F)n2)ccc(Cl)cc1O 5639,C1(C#N)(C(=O)NC(C(C)NC(=O)CC2(C)CCCC2)C)CCCC1 5640,N1(C(CC=C=C)=O)CCOCC(CNC(c2cnc(-c3ccc(Cl)cc3)s2)=O)C1 5641,N1(C(C2(SC)CN(C(=O)C(c3cccn3C)=O)C2)=O)CC(=O)N(C)CC1C 5642,C(CCN=C(NCCc1ccc(C)o1)N1CCN(c2ccc(F)cc2)CC1)OC 5643,N1(C(CC(C)c2cnn(C)c2)=O)C2CCC1C(CNC(c1ccsn1)=O)C2 5644,N1(C(C(C2CCOC2)OC)=O)CC=C(C(=O)NC2COCCC2O)CC1 5645,c1(C(=O)NC2C3CC2N(C(=O)COC2CCCCC2)C3)ccc2c(n1)CCC2=O 5646,N1(C(C(=O)N(CC(C)NC(c2coc(C3CCCC3)n2)=O)C)C)CCNC1=O 5647,n1(COC)ncn(NC(=O)c2cc3ccc(-n4cccn4)cc3[nH]2)c1=O 5648,N1(C(CCc2ncn(C)c2)=O)C2CCC1C(NC(=O)CCN1CCOC1=O)C2 5649,C1(CN(CCC(F)(F)F)C)CC2(C1)OCCO2.c12cncc(c1)N(CC(=O)O)C2 5650,C1(O)(C(C)NC(CCn2ncc(C)c2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 5651,C1(O)(CC(=O)Nc2ccc(C#N)cc2)CCN(CCNS(C)(=O)=O)CC1 5652,c1(C(=O)OC)sc(NC2CONC2=O)cc1-c1ccccc1 5653,c1(C(=O)NCC2(NC(c3cc(C(C)C)no3)=O)CCCC2)cc(N)cc(F)c1 5654,C(=O)(C(C)(O)C(F)(F)F)NCCCN(C(c1c(F)ccc(CC)c1)=O)C(C)C 5655,C(=O)(CC(O)C(C)C)NC1CC(CC(N2CC3C(CC)C3C2)=O)C1(C)C 5656,CC1(C(=O)NCC2(CNC(=O)CCF)CCC2)COC(=O)OC1 5657,c1(C2CN(CCOC(CCC#C)=O)C2)ccc([N+](=O)[O-])cc1Cl 5658,C(CC)(c1ccccc1)=CC(N1CCN(C(c2coc(N(C)C)n2)=O)C(C)C1)=O.CN 5659,c1(C(N2C(C(N(CC(C3CCC3)OC)C)=O)CC(O)C2)=O)cc2cccnn2c1 5660,Cc1nccc(NC(N2CCCC2c2n[nH]cc2NC(c2csc(C)c2)=O)=O)n1 5661,C12(CCCCC1)CN2.C1(c2ccc(F)cc2)(CNC(C)=O)CC2(CC2)C1 5662,c1(C(=O)NC2C(CNC(c3cnc(OC)c(C)c3)=O)C2)ccc(Cl)c(C)c1Cl 5663,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5664,c1(C(=O)NC2C(NC(CCCC#C)=O)CC2)cc(S(=O)(=O)CC)ccc1Cl 5665,c1(OC)ccc(CN2CCN(Cc3cc(Br)cs3)C3CC23)c(C)c1C 5666,CC(C)(C)CC(C(=O)N1CC(c2ncc[nH]2)C1)NC(C1(C)CC2C=CC1C2)=O 5667,c1(NC(C2CC(NCc3ccnc(Cl)c3)C2)=O)ccc(Cl)cc1F 5668,Cn1cc(S(=O)(=O)N2CCC(C(=O)NCC3CC(O)CN3C(=O)CNC=O)C2)cn1 5669,C#Cc1ccc(C(=O)NC(CCC=C)C(=O)NC(C)CCC=C(C)C)nc1 5670,c1(N2CCC(NC(C(CC)SC)=O)C(F)C2)c(Br)cccc1[N+](=O)[O-] 5671,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1cscc1Cl)=O 5672,CCCC(C)(CC)C(=O)NCC1CCC(C)CN1C(=O)Cc1ccc(Cl)cn1 5673,N1(C(c2cc(C(=O)OC)cs2)=O)CCN(C(c2scnc2Cl)=O)CC1CC(=O)OC 5674,N1(C(c2cc(C)c(Cl)c(N)c2)=O)CCC2(CC1)CN(C(=O)CC1CC3CC3C1)C2 5675,C1(NC(=O)CCc2ccncc2)CCCCC1NC(=O)Cn1cc(Br)cn1 5676,C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC(CC)NC(=O)CC1CC(=O)C1 5677,CCCCC(CC)C(=O)NCCOC.C1CN(C(=O)COCC(=O)NCO)C1 5678,CC(C(=O)NC1(CCCCNC(C2CC(C)(O)C2)=O)CC1)C(F)F 5679,CCC(CC)(CCNC(=O)Cc1cc(C)cc(C)c1)NC(C12CCC(=O)C1C2)=O 5680,C12(C3N(CC)CCC3)CCC(CC1)CN2C(c1csc(-c2ccnc(C)c2)n1)=O 5681,CCCCC(CN=c1nc(SC)[nH]s1)NC(c1ccc(C2CCCCC2)nc1)=O 5682,N1(C(c2c(CC)cco2)=O)CC(NC(=O)Cc2cc(C)cc(F)c2)C2(CCC2)C1 5683,c1(C(=O)NC23CCN(C(C4(CC)CC4)=O)CC2C3)cc2c(nc1O)CCCC2O 5684,C1(C(=O)N(CC(N)=O)CC2(CN(C(CCCC)=O)C)CC2)CNC(=O)N1C 5685,c1(OC)cccc(Br)c1C(N1CCC(O)C(C(=O)NC(CO)C(F)(F)F)C1)=O 5686,Cc1cc2ccc(Cl)cc2cc1NC(=O)Nc1ccc(-n2cnnn2)cc1 5687,N1(C(C2(SC)CC2)=O)CCN(C(=O)C(N2CCNC2=O)C)C2CCCCC2C1 5688,C(C1=NOC2CN(C(C3(C4CCC4)CC3)=O)CC12)NC(=O)CNc1nccs1 5689,Cc1nc(C(F)(F)F)ccc1C(=O)NCC1(NC(=O)Cc2cnc[nH]2)CC1 5690,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(COC)CC2)=O)CC1C)=O 5691,CCC(C(=O)N(C1CCN(C(C2(CCCF)CC2)=O)C1)C)c1cnc(C)s1 5692,c1(C(N2CC3CC(C2)N3C(c2ccc(C(F)(F)F)cn2)=O)=O)ccc([N+](=O)[O-])nc1 5693,c1(OC)ccc(CNC(=O)CC2CCCC2)cc1C(N1CC2CC1C2C(=O)OC)=O 5694,c1(OC)ccc(F)cc1-c1nc(Cc2cccs2)nn1C1CCCCC1 5695,c1(C(=O)OCC(c2ccc(Cl)c(F)c2)=O)cc2cc(F)ccc2nc1Cl 5696,c1(C(=O)NCC2(C)CCN(C(c3ccc(O)nn3)=O)C2)ccc(C#N)c(Cl)c1 5697,N1(C(c2c(C(C)C)scn2)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 5698,CC1(C)Oc2ccc(C(N3CCC4C(CCN4C(=O)C(O)C(F)F)C3)=O)cc2O1 5699,N1(C(c2c(C)oc(Br)c2)=O)CC(NC(c2ccco2)=O)CC(C)C1 5700,N1(C(c2cc(C)ns2)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CCC1C 5701,c1(CC(=O)NCC(=O)NCC(N2CCOCC2)=O)cncc(O)c1.C12CN(C1)C2=O 5702,C(CC(C)C(=O)NC1CCC(N(C)CCn2nccn2)CC1)=CC 5703,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(=O)C2CC(c3ccccc3)S2)CC1C 5704,C(CNC(=O)C(C1CCC1)C1CCC1)(C(C)C(C)C)NC(c1c(C)cno1)=O 5705,c1(C(=O)NCC2CCN(C(C(COC)OC)=O)CC2)cccn2nccc12 5706,c1(CNc2cccc(CCC(=O)OC)c2)cn2c(n1)CCCC2C 5707,Cc1ccc(Br)c(S(=O)(=O)NC2CCCC(NC(c3nnc4n3CCC4)=O)C2)c1 5708,c1(C(=O)NCC2N(C(CCc3n[nH]c(=N)s3)=O)CCC2)cc(Cl)nnc1Cl 5709,c1(C(N2CC3C(NC(C(C)SC(C)C)=O)C3C2)=O)cccc(Cl)c1OC(F)(F)F 5710,C(=O)(CC(C)C(=O)N1CCC(C(=O)NCc2cnn[nH]2)C1C)OC 5711,Cn1cc(C(N2CCC(NC(C3CCS3(=O)=O)=O)C2)=O)c2cc(F)ccc12 5712,C(CCC(CC)CC)N(C(C(CC1CN(C(=O)NC2C(=C)C2C(C)C)C1)F)=O)C 5713,C(=O)(C(C)(C)CC(C)C)NC(COC)CC(=O)N(C)CCC1CCCCC1 5714,C1(NC(C2CCOC2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)C2(CCC2)C1 5715,N1(C(Cc2c(COC)cccc2)=O)CC(NC(C2CCOCC2)=O)CC12CCC2 5716,C1(O)(C(N(CCCCN(C(CCN(C(C)=O)C)=O)C)C)=O)CC1(C)C 5717,N1(C(C2CCC(CC)O2)=O)CC2(C)CN(C(C3CNC(=O)N3)=O)CC2(C)C1 5718,c1(C(=O)NC2(C#N)CCN(Cc3cc[nH]n3)C2)cc([N+](=O)[O-])c(F)c(F)c1F 5719,c1(C(N2CCN(C(c3cnccc3F)=O)C3CCCC23)=O)n[nH]c2ccccc12 5720,N1(C(CCCC#CC)=O)CC2CC(F)(F)CCC2(NC(=O)COCC)C1 5721,S(=O)(=O)(CC(=O)NC(C1CN(C(c2cccc(OC)n2)=O)CCO1)C)NCC 5722,c1(C(=O)OC)ncoc1CC(N1CCOCC1)=O.C1COCCOCCN1 5723,C(c1cccc(OC(F)F)c1)=CC(=O)NCC1(NC(CCC2CCC(=O)N2)=O)CC1 5724,C(c1ccnn1C)=CC(=O)NCCCC(C)NC(C1CN(C(C)=O)C1)=O 5725,N1(C(COC2CC(NC(C3C(C)CCOC3)=O)C2)=O)CC(F)CC(F)C1 5726,C(=O)(CCCCN(C)C)NCC(c1ccccc1F)NC(CCN(C)CC)=O 5727,c1(C(C(=O)NCC(=C)C)N(CCOCC)C2CC2)cccc(OCCCCl)c1 5728,C(C(=O)NCC1CCCCC1CNC(C1CCC(=O)NC1)=O)(C(C)C)OC 5729,C1(CNC(COCCOCCOC)=O)CCCCCCN1C(c1ccc(O)cc1)=O 5730,c1(OC)ccc(Cl)cc1NC(N1CC(c2ocnc2COC(=O)C(F)(F)F)C1)=O 5731,C1(O)(C(C(=O)NCCCCCC)NC(=O)C(C)(CO)OC)CCCCC1 5732,N1(C(c2cc(CCC)[nH]n2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5733,c1(NCC(=O)N(C2CC2)Cc2cn(C3(C)CCCC3)nn2)cnn2c1CCCC2 5734,N1(C(Cc2nc(C)c(C)s2)=O)CCN(C(=O)C(C)CC(C)C)C(c2cn[nH]c2)C1 5735,CCC(C(=O)N1CCN(CC(O)COc2ccccc2)CC1)C(=O)O 5736,Cc1ccc(C(=O)CCC(=O)OC(C2CCNC2=O)C)c(C)c1 5737,c1(CC)noc2ncc(C(=O)N(C)CCN(C)C(c3nnc(C)s3)=O)cc12 5738,c1(C(=O)NC2C(NC(=O)C#CC3CCC3)CS(=O)(=O)C2)c[nH]c2nccc-2c1 5739,N1(C(c2nc(C(C)(C)C)sc2)C(=O)NCC2CC2)CCCN2CCCC12 5740,CC(CCCCCO)NC(C1CCCC1CNC(=O)Cc1cn[nH]c1)=O 5741,C(C(COC)CC(=O)NC1CCN(C(=O)C(C2CC2)SC)C(C)C1)OC 5742,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5743,N1(C(=O)Cc2ccc(OC(F)F)cc2)CC2CN(C(c3ccsc3Cl)=O)CC2C1 5744,C#Cc1ccc(NC(C2CC(C)CN(C(c3[nH]nnc3C3CC3)=O)C2)=O)c(C)c1 5745,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5746,c1(NC(CN(C)C(c2ccc(Cl)cc2F)=O)(C)C2CC2)ncnc2[nH]ccc12 5747,Cc1cc(N2CCOC(C(N3CCC3CO)=O)C2)nc(C)n1 5748,c1(OC2CN(C(C(=O)NCCC3CCOC3)=O)C2)ccccc1 5749,N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CCl 5750,C1(C2CCCCC2)(C(=O)NC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5751,C1(NC(C=CCOC)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1O 5752,N12CCOC(C1)C(=O)N(CC#C)CCC2=O.C1(CN(C)C)CCCC1 5753,c12ccc(nc1)NC2.c1(C2C(CS(C)(=O)=O)CC2)nnnn1CC(F)F 5754,c1(C(=O)NC(CNC(c2ccc(CC)c(CC)c2)=O)CO)ccc2occc2c1 5755,C(=O)(C(CC)CC(C)C)N1CC(C2CC2)(C(=O)NC(C2CCCCC2)C#C)C1 5756,c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C(C2)C3)n[nH]c2c(C)cccc12 5757,N1(C(C2COCCN(C(C(C)CC(F)F)=O)C2)=O)CC2OCC(CO)C2C1 5758,c1(N(C)C)cnc(C(=O)NCC2CCCN2C(C2CCN(C)C2)=O)cn1 5759,N1(C(CS(=O)(=O)NCC)=O)CCOCC(F)(CNC(=O)CN(C)C)C1 5760,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 5761,C12C3CCN(CC13)C(=O)CN2.C1(N(C)C(C2CC2Cl)=O)CCCCCC1 5762,N1(C(C(CCOCCO)NC(C(C(C)O)(C)C)=O)=O)CCC12CCCOCC2 5763,C(CCSC)(C(C)C)NC(CN(CCC#C)C(=O)Cc1csnn1)=O 5764,C(C)(C1=CCN(C)CC1)NC(C1C(CC)OCCC1)=O 5765,C1(C(=O)NC2CCCN(C(c3cc(C)cc(O)c3)=O)CC2)CC2(C1)CS(=O)(=O)C2 5766,N1(c2ncnc(NC(CC)CC)c2C)CCc2c[nH]nc2C1 5767,c1(C(=O)NCC2C(NC(c3cc(NC(C)=O)ncc3)=O)C2)nn(C)c(C)c1Cl 5768,c1(OCC)nn(C)cc1NC(C1CC(C)N1C(C1CN(C)CCO1)=O)=O 5769,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)COCCOCCO)C1 5770,CCC(C)(F)C(=O)N(C)CCN(C)C(C1(N2CCCCC2)CCCCC1)=O 5771,C1(NC(c2n[nH]c(C)c2O)=O)CCC2CN(C(C3CC(OC(F)(F)F)C3)=O)CC2C1 5772,c1(C(=O)NCC(c2ccc(Br)cc2)(C)C)ccc2c(c1)NC(=O)C2 5773,S(=O)(=O)(c1ccc(NCc2cc(C)ccc2F)nc1)N1CCC=C(C)C1 5774,C#Cc1ccnc(C(=O)NC2CCCN(C(c3coc(O)n3)=O)CC2)c1 5775,c1(NC(c2scc(CNC(CC=C=C)=O)c2)=O)cccc(F)c1C 5776,N1(C(=O)NCc2ccc(C3(C(=O)OC)CC3)o2)CC(S(C)(=N)=O)C1 5777,Cc1cc(C(=O)NCCCNC(C2(CF)CC2)=O)cnc1C(F)(F)F 5778,c1(C(N2CCC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cc(S(N)(=O)=O)cn1C 5779,N1(C(CNC(C)=O)=O)CC2CN(C(c3ccc(Cl)cc3N3CCCC3=O)=O)C2C1 5780,c1(C(N(C(CN(CCC)CCN(C)C)=O)C)C)sc(C2CC2)nc1C 5781,CC(C)C(Cc1ccccc1)C(=O)NCC(c1ncnn1C)N(C)C 5782,C(CS(=O)(=O)C1CC1)NC(=O)CC1CCCN1C(C1CC(F)(CF)C1)=O 5783,OCCC(N=c1cc(NCCOC2CC2)nc(C(F)(F)F)[nH]1)c1ncnn1CO 5784,c1(C(=O)NCC#CCN(C)C)ccc(CNC(C2(C#N)CCC2)=O)cn1 5785,C1(CN(C(=O)COC(C)(C)CNC(C2CCCCC2O)=O)C)CCCC2CC12 5786,C(=O)(CC1=NNC(=O)C1)NC1CCC(NC(CN(CC)CC)=O)C1 5787,c1(C(=O)NCCN(C(C=CC)=O)CC)cccc(C2CCCOC2)c1 5788,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(c1ccc(F)cn1)=O 5789,C12CN(CCO1)C(=O)C(=O)NC2.c1(C(=O)OCC)cc(C(C)C)[nH]c1C1CC1 5790,C12(CNC(C(C=C)O)=O)CC(CO1)N(C(C1(N3CCOCC3)CCCCC1)=O)C2 5791,Cc1cccc(OCC(N2CC(OCCCS(N)(=O)=O)C2)=O)c1 5792,c1(C(=O)OC)n[nH]c2c1CCN(CC1CCC(C(F)(F)F)O1)C2 5793,S(=O)(=O)(c1cccc(=NCc2cc[nH]c(=N)n2)[nH]1)N(CC(C)OC)CC 5794,Cc1cc(S(=O)(=O)NCc2nocc2Cl)sc1C#N 5795,C1(C(=O)NC2C(c3ccn(C)n3)C2)CCC2(CC2)N1C(C1(O)CCOC1)=O 5796,C1(NC(CC2(C)CCOC2)=O)CCC2(CC1)CN(C(=O)CCCCC#N)C2 5797,C1(S(N)(=O)=O)(C(N(C2CCC(NC(C=C(C)Cl)=O)CC2)C)=O)CCC1 5798,c1(C(=O)NC2CCN(C(CCC(C)OCC)=O)CC2)ccc2nc(S)[nH]c2c1 5799,CC(C)(F)C(C)(F)CNC(C1CC1c1ccc(OC(F)F)nc1)=O 5800,C1(NC(CNC(CCCCC)=O)=O)CCC(C)(C)CC1CNC(C1CC(OC)C1)=O 5801,c1(NCC2C(C)(C)CCO2)[nH]c(=NC2CCS(=O)(=O)C2)nc2scnc12 5802,c1(CC(C)C)ccc(C(N2CCC(CF)C2)C(=O)NCCN(C)C)nc1 5803,O(N(CC)C(=O)CNC(=O)CC(C)(C)CN(C)C)CCn1ccc(CC)n1 5804,C1(NC(CN(C2CC2)CC)=O)CCCC(NC(c2ccnc(C3CCC3)c2)=O)C1 5805,C(=O)(C(C#N)C(C)C)N1C2C(NC(COCCC)=O)C(C2)C1 5806,C1(CNC(COCCC#C)=O)CCCCN(C(c2csc(-c3ccsc3)n2)=O)C1 5807,C(=O)(C1=COc2ccccc2O1)NC1C(CNC(C(C(C)C)C)=O)CC1 5808,CC1CCN(C(c2cc(Cl)cn2C)=O)CC1NC(c1ccn(C)n1)=O 5809,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5810,c1(C(N2CC(C)N(C(=O)CNS(=O)(=O)C3CC3)CC2)=O)ccn2cccc2c1 5811,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(=O)C=CC(=O)OC(C)C)C2C1 5812,n1(CC(=C)C)c(N(C2CCCC2C#N)C)nnc1-c1ccc(SC)s1 5813,C1(C(N(C2COC(C)(C)C2)C)=O)CN(C(=O)Cn2cncn2)CC12CC2 5814,c1(C(=O)NCC(C2CCC2)NC(CCC2C(C)(C)C2)=O)ncc2[nH]ncc2n1 5815,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1COC(=O)N1)=O 5816,C(=O)(CC(CCCC)NC(=O)Cn1ccnc1C)N1C(C#C)COCC1 5817,c1(C(=O)NCCN(C(=O)C=Cc2cc[nH]n2)C(C)C)ccc(O)c(CO)c1 5818,Cc1c(F)ccc(C(N2CC(NC(C3(C)CC4(CC4)C3)=O)C2)=O)c1C 5819,c1(C(N(c2ccc(-c3scnc3C)cc2)CCC)=O)coc2ccccc12 5820,C12(NC(C(CC)O)=O)CCC(C1)N(C(C1(C(F)(F)F)CCCC1)=O)C2 5821,c1(SCCC(=O)NC(CNC(Cc2cn(CC)nn2)=O)C2CC2)ccccc1Cl 5822,C1(C(N(C)CC2N(C(CC(CC)OC)=O)CC(F)C2)=O)OC2CCC1CC2 5823,C1(C(=O)NCCCCN(C(C2(CCOCC)CCC2)=O)C)OCCCC1(C)C 5824,c1(C(C)NC(c2n(CC)nnn2)C)cccc(OCC(F)(F)F)c1 5825,CC1CN2CCN1CC2C(=O)NC1C=CCN(C(c2ccc3snnc3c2)=O)C1 5826,n1(CC(N2CC3C(C(=O)Nc4cc(O)cc(F)c4)(C3)C2)=O)cc([N+](=O)[O-])cn1 5827,CC(C)CCCCC(=O)NC1CC(OCC(N2CCC(CCO)C2)=O)C1 5828,C12(C(=O)NC3C(NC(c4ccc(CO)nc4)=O)COCC3)CCC(CO)(CC1)C2 5829,C=CC(C)CCN=c1[nH]c(=NCC2(C)CCOC2)c2sccc2[nH]1 5830,N1(C(c2c(C(C)C)ccs2)=O)CCC(C(C)NC(=O)CN2CCS(=O)CC2)CC1 5831,CCCCC(CNC(=O)CC=CCOC)NC(=O)CCC(=O)N(C)C 5832,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5833,C1(O)(CNC(CCCOC(C)(C)C)=O)CCCN(C(C2CC3C=CC2CC3)=O)C1 5834,N1(C(COCCC=C)=O)CC(O)CC1CNC(c1c[nH]nc1CCC)=O 5835,Clc1cccc(C2(NCC=CCC3CC3)CCC2)c1 5836,N1(c2n(CC(=C)C)c(C(C)F)nn2)CCN2C(=O)CCC2C1 5837,C1(C(N2CCCN(C(c3cnccn3)=O)CC2)=O)COc2cc(Br)ccc2O1 5838,C1(C(=O)NCC#CC(F)(F)F)CC(O)CCN1C(c1cscc1Cl)=O 5839,CCCC(O)CC(=O)NC(C)(CNC(=O)Cn1cc(C2OCCO2)cn1)CO 5840,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN(C(=O)CC1CC3(COC3)C1)C2 5841,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5842,N1(CC(=O)N(CCCN(C(C(C)CC2CCCO2)=O)C)C)CCCNC1=O 5843,N1(C(C(=O)N(C(C)C)CCc2cccc(Br)c2)=O)CCCC2(CCCNC2=O)C1 5844,C1(C(=O)NC(C)CNC(=O)C=Cc2cnc(C)s2)(CC)CCC(O)CC1 5845,C1=CCCC(Nc2ncc(-c3ccccn3)s2)CCC1 5846,C(CC(C)(C)CC(=O)N1CCCN(C(c2c(C)nn(C)c2Cl)=O)CC1)OC 5847,N1(C(c2ccc(CN(CC)CC)o2)=O)CCN(C(c2cc(F)cs2)=O)CC1C1CC1 5848,C1(CC=C)(C(=O)NCc2nc(C3CC3)n[nH]2)CCN(C(c2ccccn2)=O)C1 5849,C1(CNC(C2CC(CF)C2)=O)CC2CN(C(C3(Sc4ccccc4)CC3)=O)CC12 5850,N1(C(Cn2nnc(C)n2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CCOC2)C1 5851,c1(-c2scc(C(C(=O)NCc3nc(C)c(C)[nH]3)(C)C)n2)cc(Cl)ccc1F 5852,C1(C(=O)NCC2CCCN(C(C)CN(C)C)C2)CN(C)CCN1C 5853,CCCCCC(O)C(=O)Nc1cnc2occc2c1.C12CCC(C)N(C1)C2 5854,c1(N2CCC(O)(CNC(=O)Cc3cnccc3Cl)CC2)ncnn2cccc12 5855,c1(C(N2CCC(NC(C3(C)CCCS3(=O)=O)=O)C2)=O)cc2c(Cl)nccc2o1 5856,c1(C(=O)NC2C3CN(C(C4CC(OCC)C4)=O)C2C(O)C3)sc2cccnc2c1Cl 5857,C1(CNC(c2cnoc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5858,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5859,CC1(C)C2CCN1C2=O.c1(C2CC(CNC(=O)CC#N)O2)ccccc1 5860,N1(C(=O)OC(C)(C)C)C2CCC1CN(C(=O)NC1CCCN(S(C)(=O)=O)C1)C2 5861,N1(C(C(C)=CC)=O)CCC2CN(C(c3cnn(CCO)c3N)=O)CCC2C1 5862,C1(CC(=O)NCC2N(C(c3ccn(C)c3)=O)CCC2)CCC(C)(O)CC1 5863,C=Cc1cc(C(=O)NCC(CO)NC(=O)CC2CCCS(=O)(=O)C2)cc(F)c1 5864,N1(C(CCC(C)OC)=O)CCC(F)CC1C(=O)NCc1cn(C)nc1C 5865,CCCCC(C(=O)NCCNC(=O)CCCc1cnc[nH]1)NC(N)=O 5866,c12cccc(c1C)CN1CCN2CC1.c1(C(=O)OC)nc(C2CC2)oc1C 5867,N1(C(c2cc(N)c(N)nc2)=O)CCN(C(=O)C2=CCOCC2)C2CCCCC12 5868,c1(CCC)nc(=NC2CC(C)N(C(=O)CCn3ccnc3)C2)s[nH]1 5869,N(C(=NCCc1nn(C)c2c1CCCC2)N1CCCC(CSC)C1)CCOC 5870,c1(CNC(=O)CSc2ccccn2)cnn2c1CN(C(=O)C=CC1CCC1)CC2 5871,C(=O)(CCCCC(F)(F)F)NCCN(CC(C)O)C(c1c(C)nn(CC)c1C)=O 5872,N1(C(C(C)OC2CCC(=O)N2)=O)CCCCC1NC(C1CCCCCC1)=O 5873,c1(OC)nscc1C(=O)NC1COCC1NC(C1(C)CC1)=O 5874,C(=O)(C(F)(F)C(F)(F)F)N1C(CN(C(=O)CC2(C)CCS(=O)(=O)N2)CC)CCC1 5875,c1(CC)ccc(C(C(=O)NC(c2ncc(C(=O)OC(C)(C)C)o2)CC)OC)cn1 5876,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2sc(C)cc2OC(F)F)=O)C(C(F)F)C1 5877,CC(=O)CCCC(=O)NC(C(=O)NCCCOC1CCCC1)C(C)C 5878,C(=O)(C(O)CC(C)C)NCC(c1ccccc1)N(C(CN(C(COC)=O)C)=O)CC 5879,N1(C(c2ncnc(C)c2C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCS(C)=O)C1 5880,CCC(CC)C(C(=O)NC(C)CCC(=O)NCC(=O)NOC(C)CC)OC 5881,O=S(=O)(c1cnc2ccsc2c1)N1CC(O)C1c1ccccc1 5882,N1(C(C2CC(=C)C2)=O)CC2CC2(NC(=O)Cn2ccnn2)C1 5883,C1(CNC(C2C(CC)OCC2)=O)CCCN(C(c2cnc(C(C)O)s2)=O)C1 5884,Cc1ccc(O)c(CNC(=O)C(c2ccccc2)NC(C2CCN(C)CC2)=O)n1 5885,N1(CCCOCC=C)CC(C2CN(C(=O)C(C)NC(=O)NC3CC3)C2)C1 5886,C1(C(=O)NCC(n2cc(CN3CC4CC4C3)nn2)C)CCC(=O)C(C)C1(C)C 5887,C1(CC(C)NC(C2(C)CCCS2)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 5888,N1(C(c2cc(C)no2)=O)CCCC(O)(CNC(c2cc(Cl)ncc2N)=O)C1 5889,C1(CN=C(NCCOC(C)C)NCC(=O)Nc2ccccc2)CCCCC1(F)F 5890,N1(C(c2c(CC)nn[nH]2)=O)CCC(C)CC1CNC(=O)CCOCCOCCO 5891,S(=O)(=O)(c1ccc(Nc2nnc(C)n2C)c(Cl)c1)N1CCC(CNC(C)=O)CC1 5892,C12(NC(CN(C)C(N)=O)=O)CCCC1N(c1nccc(C#N)n1)CCC2 5893,n1(CC(=O)NCCCCCNC(=O)COC2CCOC2)ncn2nccc2c1=O 5894,C(=O)(CC(C)C(=O)N1CCC(CN(C(=O)COC2CCCC2)C)C1)OC 5895,c1(CCC)nc(C(N2CCC(COC)C2)=O)cs1 5896,CC(C#N)CN=C(NCC1CCN1Cc1cccc(Cl)c1)NC(C)(C)C 5897,Cc1c(C(=O)NC2CC(CNC(c3csc(C(F)F)c3)=O)C2)cnn1C 5898,C(CC(C(=O)N(C(C)C(C)OC)C)NC(=O)CSC1CC1)OC 5899,CC12CCN(CC1)CC2C(=O)NC12CC(NC(C34CC(F)C3C4)=O)(C1)C2 5900,N(C1CCCc2c[nH]nc21)C(C(CCNC(CN(C(C)C)C)=O)O)=O 5901,c1(C(N2C(CNC(C(C)Cc3ccco3)=O)C=CC2)=O)cc2n(c1)CCC2 5902,C(N=c1nc(NCC2(SC)CC2)c2c([nH]1)CCOC2)C1(CC)CCC1 5903,S(=O)(=O)(c1cnccc1NCC1(CCO)CCC1)NCC1N(C)CCC1 5904,c1(C(=O)NCC2N(C(C)=O)CCC2c2ccccc2)cc2ncncc2s1 5905,c1(CN(C)C(C23CC(n4cc(C5CC5)nn4)CCC2C3)=O)cc(F)c(F)cc1N 5906,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCCN(C)C)CC 5907,C1(C2CCN(C(=O)CCC(F)(F)F)CC2)(NC(C2CC(C)(C)OC2)=O)CC1 5908,C1(NC(C2C(C)(C)C2NC(=O)C(=O)C(C)(C)C)=O)CCCOC12CCC2 5909,c1(CC)ccc(Br)cc1C(=O)NC(C)CCN(C)C(C1C(C)(C)C1(C)C)=O 5910,CN1CC(NC(=O)NC(C23CC(CN)(C2)OC3(C)C)=O)Cc2ccccc21 5911,c1(C(=O)NCC2CCN(C(=O)CCC3CCOC3)CC2)nc2n(c1Cl)CCCC2 5912,C1(C)(NC(CCN(C(c2nn(CC)c(O)c2)=O)C(C)C)=O)CCC(C)(C)C1 5913,c1(CNC2(CC(=O)Nc3cncnc3O)CCC2)ccc(Cl)c(F)c1 5914,C1(NC(c2c(C)scc2)=O)CN(C(c2cc3n(n2)CCC3)=O)CC12CCC2 5915,N#Cc1cncc(C(=O)NC2(CF)CCN(C(=O)Cc3sccc3Br)C2)c1 5916,c1(CC(C(=O)NC(C)CCCNC(=O)CNc2nccs2)=O)ccc(F)cc1 5917,Cc1ncc(Cl)cc1C(N1CC(N(C(=O)CC2CCCCC2(C)C)C)C1)=O 5918,N1(C(C(c2n(C)ncc2)O)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)C12CC2 5919,S1(=O)(=O)C2=CC=CC(=NCCCOC3CCN1C3)N2.C=CCOC(C)C 5920,c1(CC)cnoc1C(=O)N(CCC(C)NC(=O)C(C)OCC1CCC1)C 5921,c1(CC(N2CCC(NC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)ccc(S(N)(=O)=O)s1 5922,c1(C(=O)NCCC(=C)CNC(C2(c3ccno3)CCC2)=O)cn(C(C)C)nc1C 5923,c1(OC)cc(C(N2CCC(C(=O)Nc3cccnc3C(F)(F)F)C2)=O)cc(Br)c1 5924,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2sc(Cl)cc2s1 5925,N1(C(CCC)=O)CCC(OC2CN(C(C3CCCN3C(C)=O)=O)C2)C1 5926,CC(C(C)C(=O)N1CC(OCCNC(=O)CC(=O)N(C)C)C1)C(C)(C)C 5927,c1(CC)cccc(C(=O)NCC2CCC(C(=O)NC3CC4CCC4C3)CC2)n1 5928,c1(OC)ncnc(N2CCN(C(c3ccc(C(C)(C)C)nc3)=O)C(C)C2)c1C 5929,O(NC(=O)C(C1(O)CCC1)NC(c1ccc(O)cc1)=O)CC=CC 5930,C1(c2nnc(C)o2)CCN(C(=NCC2CCCO2)NC(C)C2CC2)CC1 5931,c1(-n2c(C3C(C)C3C)nc(CCSC)n2)ccc(F)c(F)c1 5932,CC1CCN(C(=O)CC(c2ccon2)C2CC2)C1CNC(=O)CC1OCCC1C 5933,C1(C)(C(N(C)CC2(O)CCN(C(=O)CC3CC3(C)C)CC2)=O)CC(C(C)(C)C)=NO1 5934,C12(CNC(=O)Cc3ccccn3)CC(CNC(c3ncsc3Br)=O)(CO1)C2 5935,c1(C(=O)NC2C(NC(=O)CCc3nccs3)CC2)ccc(-c2ccco2)nc1 5936,c1(C2C(C(=O)NC(CC=C)CNC(=O)Cn3cncn3)C2)ccc(OC)cc1 5937,c1(C(C)OC2CCCOC2)ccc(-c2cccs2)cc1.N12CC(C)(C1)NC2=O 5938,c1(C(=O)NCC2C(NC(c3n(CC)nc(C4CC4)c3)=O)C2)cccc2c1C(=O)NC2 5939,C1(N(C(CCC#C)=O)C)CN(C(=O)C(CC)CC)CCC1C 5940,S(=O)(=O)(c1cnn(C)c1)NC(N1CC(C(=O)OC)OC(CO)C1)=O 5941,CC1CC(C(=O)N2CCCC2C=CC(=O)NCC2CCN(C3CC3)C2)=NO1 5942,c1(CNC(C2CCCCN(C(C3(OCC)CC3)=O)C2)=O)nn(C)c2c1COCC2 5943,CC#CCCCC(=O)NCC1CN(C(=O)CC2CCCN2C(C)=O)CC1C 5944,c1(C(n2cc(C3CCN(C(C4COCCO4)=O)C3)nn2)C)ccccc1F 5945,C1(CC(=O)NC2C=CCN(C(Cc3nnc(C)s3)=O)C2)Cc2ccccc2C1 5946,C(=O)(C(F)(F)CC(C)C)N1CC(CCNC(=O)C2=CCCOC2)(OC)C1 5947,c1(NC(C2CN(C(c3c(OC)cncn3)=O)C2)=O)c(C)cccc1[N+](=O)[O-] 5948,C(=O)(C(CC(F)F)C1CC1)N(C1CCN(c2cn[nH]c2)C1=O)CCC 5949,C1(CC)(NC(C2CSCN2C)=O)CCOCC1.C12(CCOCC1)C(=O)NC2 5950,c1(OCC)ccc(OCC)c(NC(=O)NC2CCNC2C)c1 5951,CC(C(=O)NCCOC(C)(C)CNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5952,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(SC)s1)=O)OC 5953,C(=O)(C1=CS(=O)CCC1)NCCN(C(C(CC=C)C)=O)C1CC1 5954,c1(CNCCN(CCC)C)ccc2c(c1)NC(=O)C2 5955,C(C(=O)N1Cc2ccccc2CO1)C1CC(NC(C(C)=CCC)=O)C1 5956,Cc1ccc(NC(=O)CC2CCCN2C(C2(CC3CC3)CCC2)=O)c(C)c1 5957,c1(OC(C)=O)cc(Br)cc(F)c1C#N.c12ccc([nH]1)C(=O)N1CC(C1)NC2=O 5958,c1(N2CC(CC=C)(N(C(=O)CCN3CCCCC3=O)CCC)C2)ncncc1C 5959,N1(C(C(CO)N(C)C)=O)CCC(CNC(C23CC(CO2)C3)=O)CC1(C)C 5960,N1(C(c2ccc(C)[nH]2)=O)CCOCC1CC(N1CC(F)(F)C1C1CC1)=O 5961,c1(C(=O)NCCC2CCC(NC(c3cnns3)=O)C2)c[nH]ccc1=O 5962,C(=O)(C1=NN(C(C)C)C(=O)CC1)NCCCN(C(C(C)(C1CC1)OC(C)C)=O)C 5963,C(=O)(C1CCCn2nccc21)N1CC2N(C(c3cc(C)cc(Cl)c3)=O)C(CC2)C1 5964,C(N=c1[nH]c(NC2CCC3CCC23)nc2cccnc12)c1c(C)n(C)nc1 5965,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 5966,CC(C)CC(C(=O)O)NC(C1CCCN(C(c2ccnn2C)=O)C1)=O 5967,c1(CNC(C2CC(C(F)(F)F)(OC)C2)=O)nc(CNC(=O)COC)cc(O)n1 5968,c1(NC(=O)NCc2csc(C3CC3)c2)cc2c(nc1O)CCC2 5969,c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc(-n2cccn2)nc1 5970,N1(C(Cc2c(C)nc(C(F)(F)F)s2)=O)C2CCNCC1CC2 5971,C1(NC(C(CSC)C)=O)COCCN(Cc2ccc(F)c(F)c2)C1 5972,CCC(O)C(C)(C)C(=O)NCC(C)CN(c1nc(C(C)C)cc(C)n1)C 5973,c1(SCC(=O)N(CCCN(C(C(CC)F)=O)C)C)nc(C)c(C)c(C)c1C#N 5974,C1(N(C(=O)CSC(C)C)CCC)CCN(C(c2cn(C(C)(C)C)nc2C)=O)CC1 5975,N1(C(C2C=C(C)CS2)=O)CC(CC(=O)NCC(=O)N(C)O)CC1(C)C 5976,C(=O)(CCCC(=O)NC)OC1CCN(c2n(CC)c(C(C)CF)nn2)CC1C 5977,C1(C(=O)NCCCCNC(=O)C=Cc2cccnc2)CCC(=O)N2CCCC12 5978,N1(C(CCN(C)CC)=O)CC2C(C(=O)Nc3cccnc3)C2C1 5979,c1(OC)cc(CNCC2CCC(CC(F)(F)F)CC2)ccc1Br 5980,Cc1nc(C(N2CCC2CNC(C2(n3ccnn3)CC2)=O)=O)c2ccccn12 5981,c1(N(CC(C)C(F)F)C)cccc(S(=O)(=O)N2CCSC(C)C2)n1.C(CO)N 5982,CCCCC(C(=O)NC1CC1)N(C)CC1(C#N)CCOCC1 5983,C(CCCCC(=O)NCC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 5984,C1(NC(c2cncc(C)n2)=O)CCCN(C(c2cc(Br)sc2Br)=O)CC1 5985,c1(C(N(C(=O)NCC(C=C)C)C)C)cnccn1 5986,S(=O)(=O)(c1c(F)cc(F)cc1F)Nc1scc(C(=O)Nc2cccc(Br)c2F)n1 5987,CCCCC(C(=O)NCc1cc(C2CC2)no1)NC(C1OCCC1(C)C)=O 5988,n1(CCCN2CC(NC(C(C(CC)C)OC)=O)C2)c(C)cc(C)nc1=O.C(C)=O 5989,c1(C(=O)NC2CN(C(C(C)O)=O)CC2F)cn2ccc(Br)cc2n1 5990,C1(O)(CCNC(C(C)SCC)=O)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 5991,C=CCC(C(=O)NCCCOCCCNC(=O)Cn1nnnc1C)NC(C)=O 5992,c1(C)cnn(C)c1C(=O)N.C1(CCNC(c2nc(CC)oc2)=O)CC2C=CC1C2 5993,N1(CC)CCC(C(N2CCCC2(CNC(=O)C#CC(C)C)COC)=O)CC1 5994,Cc1cc(C2CC2)ccc1C(=O)Nc1ccc(NC(=O)Cc2cnc[nH]2)cc1C 5995,N1(C(c2n(C(C)C)ncc2)=O)Cc2cccc(CNC(=O)C(C)(C)C(N)=O)c2C1 5996,Cc1nc(C(=O)NCCC2CCCN2C(=O)CO)ccc1Br 5997,N#Cc1ccccc1NC(C1CC1NCCO)=O.c1(N)ccc(C(F)(F)F)cc1O 5998,c1(C(=O)NC2CCN(C(CC(C)SC)=O)C23CC3)coc(S(C)(=O)=O)c1 5999,C1(NC(C2=CCN(C(CN3CCC(C)CC3)=O)C2)=O)CCn2ncnc2C1 6000,N1(C(C2CC(CC)OCC2)=O)CCCCC2(C1)CN(C(c1n[nH]c(C)c1O)=O)C2 6001,c1(C(N(CC(C)CNC(=O)CC2CCNC2=O)C)=O)cc2sccc2[nH]1 6002,c1(C(=O)NC2C(NC(C(C(C)C)NC(N)=O)=O)COC2)nn(C)cc1[N+](=O)[O-] 6003,CCCCC(CNC(=O)Cc1nncn1CC)NC(=O)C(N(C)C)C1CC1 6004,C(N=c1nc(N2CC3(C2)NC(=O)NC3=O)c2[nH]ccc2[nH]1)c1ncn(C)n1 6005,c1(C(=O)NCC2CC(CNC(c3cnc(C)s3)=O)OC2)c(C)cccc1Cl 6006,N1(C(CONC(c2ccc3nccc(N)c3c2)=O)=O)CCCC2(CC(O)C(=O)CC2)C1 6007,Nc1c(F)c(F)cc(C(N2CCN(C(c3ns[nH]c3=O)=O)C3CCC23)=O)c1Cl 6008,CC(CCC(=O)Nc1cncnc1O)NC(c1ccncc1Cl)=O 6009,c1(OC)ccc(C)nc1C(=O)NCC1(F)CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1 6010,c1(C(N2CCCN(C(C3CCN(OC)CC3)=O)CC2)=O)cc2ccc(F)cc2s1 6011,Cc1ncc(C(=O)N(C)C)n1-n1cccc1.C1CCOCCN1C 6012,C1(C2CC2)(C(=O)NCCCCN(C(=O)CCN2CCOCC2)C)CCC1 6013,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6014,c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)ncc(Br)cc1O 6015,C1(C(N(CCNC(c2ccc3nncn3c2)=O)C2CC2)=O)CCc2nnnn2C1 6016,O=C(C(F)C1=CCCCC1)N1CCN(C2CN(CC3CCCS(=O)(=O)C3)C2)CC1 6017,c1(OC)ncc(Cl)c(C)c1C(=O)NC(C)CCNC(C1CC1C(=O)NCCO)=O 6018,c1(OC)nccc(C(=O)NCCC2CCCN2C(c2cc(Cl)ns2)=O)c1F 6019,Cc1nc(CO)ncc1C(N1CCC(NC(C2C=CCCC2)=O)C1(C)C)=O 6020,c1(C(=O)NCC(C2CCOC2)NC(CCC(N)=O)=O)cnc2ccccn2c1=O 6021,C(=O)(C1=CC2(CCOCC2)C1)NCC1CC(C)N(C(=O)C=C2CCCCC2)C1 6022,S(=O)(=O)(c1cccnc1N1CCCOCC1)N(C)CC12CC1CCC2(F)F 6023,C1(C)(CNC(c2c(CNC(c3c(C)c[nH]n3)=O)ocn2)=O)CCN(C)C1 6024,C1(C(=O)NC23CC(NC(c4n(CC)nc(C)c4)=O)(C2)C3)CCN(CCO)C(=O)C1 6025,C=CCCCCCCCC(=O)N1CC2CC1CC2NC(c1ccc(C)cn1)=O 6026,N1(C(c2n(C)nc(Cl)c2)=O)C2CCC1CC(CNC(=O)C(F)=C1CCC1)C2 6027,c1(CC(=O)N(CC(C)NC(C(C=C)(C)CC)=O)C)cnn2c1OCCC2 6028,c1(-n2cc(OCCN(CC(OCC)OCC)C)nn2)cccc(F)c1Br.OCC 6029,N1(C(C(c2cn(C)nc2)=O)=O)CCC(C(=O)NC2CCSC2)C1C(C)(C)C 6030,C(=O)(C(CNC(c1c(C)[nH]c(C)c1C)=O)CC(C)C)NC(c1cc(C)on1)C 6031,C1(CNC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccc(C(F)(F)F)cn1)=O 6032,Cc1nn(CCN2CCOC(CCNC(C3(C)CCC(=O)N3)=O)C2)cc1Br 6033,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6034,C(=O)(C(F)(CNC(C1CC(C(=O)OC)C1)=O)C(C)C)N(c1cccc(CC)c1)C 6035,N1(C(C=C(CC)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1CC 6036,N1(Cc2cccc(OCC(=O)NC)c2)CCOC(C)(CNC(C)=O)C1 6037,C(=O)(C(C)(C)C(=O)N1CCCC1c1ccc(F)c(F)c1)N1CC(C)C(CO)C1 6038,c1(C(CC)C)ccc(C(=O)NC2CCC2CNC(C2(O)CC2)=O)c(O)n1 6039,c1(NC(=O)NCC2(OC(C)(C)C)CC2)n[nH]c(=N)[nH]1 6040,C1(C2CC2)(NC(C2C(NC(COCC=C)=O)C2)=O)CCCC1 6041,c1(NC(c2ccc(OC(F)F)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6042,c1(C(N2C(C3(NC(C(COCC)C)=O)CC3)CCC2)=O)cc(OC)nc(Cl)c1 6043,CCCCC(CN1CCCC(NC(c2n[nH]cc2C)=O)CC1)CC 6044,CP(C)(=O)C1(C(N2CCOC(CCNC(=O)CC3CCOC3)C2)=O)CC1 6045,N1(C(C(CC2CCC2)NC(C2CN(C3CC3)C2)=O)=O)CC2(CCC2)C1 6046,CS(C)(=O)=Nc1nc(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C23CC3)cs1 6047,C1(NC(CCC(C)OC)=O)CC2CCC(C1C)N2C(=O)C1=CCCCO1 6048,C1(CC(N2CCC(CN(C(Cc3c(C)occ3)=O)C)C2)=O)CCC1C1CC1 6049,CC1=CCSC1C(=O)NC(C1CCN(C(=O)CC2CCCC2O)C1)(C)C 6050,C1(NCc2c(Cl)nc(N(C)C)s2)(CO)CCN(C(c2cnc(Cl)s2)=O)CC1 6051,C1(N(C(=O)C(=O)NCc2cn(C3CCOC3)nn2)C)CS(=O)(=O)C12CCOCC2 6052,N(C1c2ccccc2CC1NC(C12CCC(CC1)CC2)=O)C(C(C)C1CCC1)=O 6053,CCCC(CC)C(=O)NC1CN(C(=O)C2=NNC(=O)C2)CC1CC 6054,C1(NC(C(CC)Cc2ccccc2)=O)CC2CN(C(c3n[nH]c(C)n3)=O)CC2C1 6055,N1(C(C(C)N(C(CC2CC(SC)C2)=O)CCO)=O)CCOC2C(O)CC12 6056,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6057,C=CCCC(C(=O)N1CC(CO)(OC)C1)NC(=O)C(C(C)(C)C)N(C)C 6058,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6059,N1(C(COCC=C)=O)CCC(CNC(c2cccc(C)c2)=O)C12CCC2 6060,CC1(C)C2CC1CN(C(=O)CC(=O)NCCOCC(F)(F)F)C2 6061,C1(CNC(CC2C(=C)C2)=O)(CNC(c2cc(C)n(CC)n2)=O)CC12CCC2 6062,S(=O)(=O)(CC(=O)NC(C)(C)C)CNC(C1(CCF)CCN(CCOCC)C1)=O 6063,C1(C(=O)Nc2cnn(CCC)c2CC)C2Cc3c(Br)cccc3C12 6064,C1(CNC(CSCCCC)=O)CCC2(CN(C(=O)Cc3cnccn3)C2)O1 6065,N1(C(c2c(C)noc2)=O)CC=CC(NC(=O)CC2(c3cccc(F)c3)CCC2)C1 6066,Cc1ccnc(C(N2CC(C(N)=O)(CNC(=O)CN3CCCCCC3)C2)=O)c1N 6067,Cc1cn(C)cc1C(=O)NCCCCNC(c1cccc(NS(C)(=O)=O)c1)=O 6068,C(CCCCCN(C(=O)CCn1ncn(C)c1=O)C)NC(C1(CC)CC1(F)F)=O 6069,C(=O)(CCN1C(=O)COc2ccccc21)N1C(C)CCCC1C 6070,N1(CC)C(C)(C(=O)OCc2cc(Br)c(C)n(C)c2=O)c2cc(C(=O)O)ccc21 6071,N1(C(C2CC(OC)C2)=O)CCOC2CN(C(c3nccc(Cl)c3O)=O)CC12 6072,N1(C(C(C)n2cccc2)=O)CCC2(CC2)CC1C(=O)NCCN1CC=CC1 6073,O(NC(=O)C(O)C1(O)CN(C(c2ccc(=N)[nH]n2)=O)C1)CCCOC 6074,C#Cc1ccc(CNC(=O)C(C)C(C)NC(=O)CCN2CCOCC2)cc1 6075,n1(CC(=O)NC(C(C)NC(CC(C)F)=O)(C)C)c(=O)cnc2ccccc12 6076,N1(C(C(CC)NC(=O)C(=O)NCC2CC2)=O)CCOC(C)(C)C1C 6077,Cc1sccc1C(=O)NC(CC(C)OCC)C.c1(S)cnc(Cl)s1 6078,N1(C(c2cc(F)c[nH]2)=O)CC2CN(C(c3ccnc([N+](=O)[O-])c3)=O)CC2C1 6079,c1(NC(CC(CNC(=O)CSC2CCCCO2)O)=O)cccc(Cl)c1O 6080,C=CC(C)(C)CC(=O)N1CCC(CCC(=O)NCCCN(C)CCOC)C1 6081,c1(NC(C2C(C(=O)Nc3c(C)ncc(C)n3)C2)=O)ccc2c(c1)OC(C)(C)O2 6082,C1(C)(C(N(C)CC2CCN(C(C3(C)CCCO3)=O)C2)=O)CCCNC1=O 6083,n1(CCC)ncc2c(C(=O)NC(C3CCCCC3)COC)cc(C)nc12 6084,c1(C(=O)NCCN(C(C(C)Oc2ccc(C(C)=O)cc2)=O)C)cnc(C)c(Cl)c1 6085,C=CC(C)(C)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 6086,Cc1cc(C(=O)NC(c2ncc(-c3nn[nH]n3)c(C)n2)C)n2ncc(CO)c2n1 6087,Cc1cc(NC(=O)NC2CCCC23CC3)cc(Br)n1 6088,c1(C(=O)NC(CN(C(c2cc(OCC)ncc2)=O)C)C)cc(F)c(N)cc1F 6089,Cc1nccc(C(=O)NC(C2CCCN2C(=O)CCc2cccn2C)C)n1 6090,C12(C(N)=O)CCCC1(C(=O)NCC(F)CNC(c1cccc(OCF)n1)=O)C2 6091,C1(NC(c2cn(C3CCOC3)nn2)=O)CC2CC1CN(C(=O)C(F)(F)C1CC1)C2 6092,c1(N2CCC3(C(C(N4CCCC4)=O)C3)C2)ncnc2cccnc12 6093,C(CC(C(=O)N(C)C)NC(=O)CCc1nc[nH]n1)=CC 6094,CC1CCCC=C1C(=O)N1CCCC(F)(C(=O)NC(c2cncn2C)CO)C1 6095,CCCCCS(=O)(=O)Oc1ccc(NCc2cccc(C)c2OC)cc1 6096,C1(NC(c2cc(OC(C)C)no2)=O)CCN(C(c2ccc(Cl)cc2)C)C(C)C1 6097,c1(OC(C)C(=O)NC2CC2CNC(=O)Cc2ccc(O)nc2)ccc(Cl)c(Cl)c1 6098,N1(C(C2C(C(C)C)CN2C(=O)Cc2ccn(C)c2)=O)CC2CC(CO)C(C2)C1 6099,C1(C)(C(N(C(C)CCNC(=O)CCCc2cccs2)C)=O)CC2CCC(C1)S2 6100,N1(C(C(CCC)N)=O)CC2(CC(NC(c3c(C)cccc3N)=O)C2)C1 6101,C1(CNC(c2nc(C)oc2)=O)CN(C(=O)C(n2ccc(C3CC3)n2)C)C(C)(C)C1 6102,CC1(C(=O)NCCSCCO)CC12CCN(C(c1cccc3c1CCC3)=O)CC2 6103,C1(C(N2C(C(=O)OC)CC2)=O)CCCC(NC(=O)C(=O)N(C)C)C1 6104,C1(NC(Cc2ncc(C)o2)=O)CCCC(NC(=O)CCNC(=O)C=CCl)C1 6105,C1(CNC(C(c2ccccc2)C)=O)CN(C(C2CCC3CC3CC2)=O)CCC1(F)F 6106,N1(C(c2c(OC)c(F)ccc2F)=O)CCCC2(CCN(C(=O)CCCC#N)C2)C1 6107,N1(C(=O)C=C2CCC2)CCN(CC(=O)N(CC(F)(F)F)CC2CCCC2)CC1 6108,CN1CC=C(CC(=O)NC2CCC2NC(c2cc(Cl)c(Br)[nH]2)=O)CC1 6109,C1(OC)CN(C(=O)CC(C)CNC(=O)C(O)C(F)(F)F)CCC1OC 6110,CC(C)(C(=O)NC(CNC(c1conc1C1CC1)=O)(CO)CO)C1=CCSCC1 6111,N1(C(CS(CC)(=O)=O)=O)CC2CCCC(NC(=O)COCCCF)C2C1 6112,CCC(O)C(C)C(=O)NC1CCCC1NC(c1cccc(OC)c1O)=O 6113,C1(C(=O)NC(C=C)(C)CC)CCN(C(c2cccc(OC)c2O)=O)CC1(C)C 6114,CC(C(=O)N(CCCO)CCO)(C1CCC1)NC(c1cnn(CCF)c1)=O 6115,C#Cc1cn(C)nc1C(N1CCCOC(CCNC(=O)C(C)NC(=O)C2CC2)C1)=O 6116,CN1C(=O)CCCC1Cn1cc(-c2cc(Cl)ncc2N)nn1 6117,Cc1cc(C(N2CC(NC(=O)CC3CC3)C3CC3C2)=O)c(C)n1-c1ccccc1 6118,C1(NC(CCOCC#C)=O)COCCN(C(=O)CC(CC)NC(=O)OCC)C1 6119,C(C1C(C(=O)NC2(C)CC(NC(=O)COc3ccsn3)C2)C1(C)C)=C(C)C 6120,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)Cc2cc(C)ns2)CCC12CCC2 6121,n1(CC(=O)NC2CC(C)(NC(CC=C=C)=O)C2)nc(C)c([N+](=O)[O-])c1C 6122,Cc1cnc(C(N2CCCC2CN(C)C(C23CCC(C2)OC3C)=O)=O)c(F)c1 6123,C(CCCCCC(=O)O)NC(=O)NCc1cnc(C)[nH]1 6124,Cc1ccc(C(=O)NCC(O)CNC(=O)C2=C(Cl)CCOC2)c2cccnc12 6125,c1(CC(=O)NCCC(C)N(C(c2nc(OCC)oc2)=O)C)ccc(F)cn1 6126,C(=O)(CC(CC)CCCCC)NCCC(=C)CNC(=O)CSC(F)(F)F 6127,N1(C(C(C)NS(C)(=O)=O)=O)CC2CCN(C(c3cn(C)c(O)n3)=O)C(C2)C1 6128,c1(C(=O)OC)c[nH]ccc1=NCC1(CNC(C2CCCC(C)C2)=O)CCCC1 6129,C#Cc1cc(C(=O)N(C)CCN(c2snc(C)c2C#N)C)cc(F)c1 6130,CCCCCCN(C1CC1C(C)(C)C)C(C1CC(CNC(C2CCC2)=O)C1)=O 6131,CCCCC(O)C(C)C(=O)NCC(C)CNC(=O)C(C)=CCO 6132,c1(CCNC(=O)C(N2CCC(N3CCCOC3=O)CC2)=O)ccc2c(c1)CCO2 6133,C(=O)(CC(F)(F)C(F)(F)F)S(CCCOC)(=O)=O.C(C)(C)(CN)N.C1C(=O)NCCO1 6134,c1(NC(N(CC(O)CNC2CNC(C(F)(F)F)C2)C)=O)ccccn1 6135,c1(CCC(=O)N(C)CC2CCN(C(CC(=O)OC)=O)C2)cc(C)cc(C)c1 6136,C(C1(O)CCOc2ccccc21)NC(=NCCOCC)NC1CC1C1CC1 6137,N1(C(CNC(CCOC)=O)=O)CCC(C)CC1C(=O)Nc1ccc(OC)s1 6138,c1(OC)c(C)csc1C(N1CCC(CN(C)C(C2(C)CCOC2)=O)C1)=O 6139,C(C(C)(O)CC(=O)NCc1cc(C(N2CCC3(CC2)CC3)=O)co1)OC 6140,C12(C(N(CC(=O)NCC(CSC)OC)CC(C)C)=O)CCC(CC1O)C2 6141,n1(CCCC)ccc(C(=O)NCCC2(NC(=O)Cc3ccccc3)CC2)n1 6142,N1(C(c2ccc(CN3CC(OCC)C3)nc2)=O)CCC2CCCCC2C1 6143,C1(C(=O)NCC(C)(C)CCO)CCOCCN1C(C1CC(C)(C)C1)=O 6144,Cc1c(C(=O)NCC2CCC(C)CN2C(=O)CC2CC=CC2)sc2cc(F)ccc12 6145,N1(C(C)=O)Cc2n[nH]cc2C1C(=O)N(C)CN.C=C1CC1C(=O)OC 6146,Cc1cc(C)n(C2CCCN(C(c3nnc(C(C)C)s3)C(=O)NCC(C)C)C2)n1 6147,CCCCCCC(=O)NC(c1nc(C(=O)NC(CC)CC(F)(F)F)co1)C 6148,Cn1ccnc1CC(=O)NCC(C)(F)CNC(C1CC(OC(F)(F)F)C1)=O 6149,c1(N2CC(C(C)NC(c3ccc(C)nc3)=O)OCC2)ncc([N+](=O)[O-])cc1C#N 6150,c1(CCC(=O)NCCCC(N2C(CC)CN(CC)CC2)=O)coc2ccccc12 6151,C1(C(=O)OC)(NC(=O)C(=O)NCc2cc(OC)c(O)c(Br)c2)CCC(F)(F)CC1 6152,Cc1noc(C)c1CN1CC2CC1C2C(=O)NCC(F)CO 6153,N1(CC(N2CCC(CCNC(c3cc(C)on3)=O)C2)=O)CCC(F)(F)C1 6154,Cc1ccc(C(=O)N(CCN(C)C(c2coc(Cl)n2)=O)C(C)C)nc1 6155,Cc1cccc(F)c1CC(=O)NC1CC(N(C)C(c2c(C)ncn2C)=O)C1 6156,Cc1noc2ncnc(NC3CCCN(C(C4CCCN4S(C)(=O)=O)=O)C3)c12 6157,C1(C(N2CC(C(C)NC(C(C)SCCCC)=O)OCC2)=O)CC2(CC(OC)C2)C1 6158,c1(NC(C)=O)cc(C(=O)NC(C)(C)CCCNC(=O)C=C2CCC2)ccc1F 6159,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)CNc2cnn(C)c2)C1 6160,Cc1cncc2cc(C(N3CCCOC(CNC(=O)Cc4csnn4)C3)=O)sc12 6161,N1(C(c2c(C)nsc2C)=O)CCCN(CCNC(C23CCCC2C3)=O)CC1 6162,O=C1CCC(C(=O)N2CCC(NCc3cc(C(F)(F)F)cc(Cl)c3)C(F)C2)=NN1 6163,C1(NC(CNC(CN(C)C)=O)=O)COC2(CO)CC1C2.C12CC1CNC2=O 6164,N1(C(c2c(OC)cc(N)cc2)=O)CCC2CN(C(C3CNC(=O)N3)=O)CC2C1 6165,C1(NC(C2CC3(C2)CC32CC2)=O)CCCCN(C(c2cc3occc3[nH]2)=O)C1 6166,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(=O)Cc2csnn2)C1 6167,N1(C(CCCSC)=O)CCC2(CCCN2C(C2CCCN2C(C)C)=O)C1 6168,C1(CNC(C(C)C)=O)(NC(=O)CC2C=CCC2)CCCCC1 6169,C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N1CC(CSC)C1 6170,C(CCCCCC(C)C)NC(C1C(CNC(c2cc(C)ncn2)=O)OCC1)=O 6171,c1(C(=O)NCCN(C(=O)C(n2ccc(C3CC3)n2)C)CC)ccc(C)c(C)c1N 6172,c1(C(CNC(c2nnc(C)s2)=O)NC(c2c(CC)con2)=O)ccccc1F 6173,C1(CC)CC(O)CN1C(=O)C(COC)NC(=O)Cn1ncccc1=O 6174,N1(C(c2ccn(CCNC(c3c(C)cc[nH]3)=O)c2)=O)CCC(CO)(CO)C1 6175,C=CCCC(=O)NCC(C1CCC1)NC(C1CN(C2CCOC2)C1)=O 6176,CCCCCCC(C)C(=O)N(C1CN(C(c2c[nH]c(=NC)o2)=O)CC1O)C 6177,C(=O)(C#CC1CCCO1)N(CCNC(c1c(C)nn(-c2ccccc2)c1C)=O)C 6178,c1(C(N2CC(N(C(CSC(C)=O)=O)C)C2)=O)cc(C)ccc1Br 6179,C1(NC(CN(C(COC)=O)C)=O)CCCC(CNC(c2csnc2C)=O)C1 6180,c1(C(=O)NC2CCCC2NC(C(C(C)C)N(C)C)=O)cc2c(O)cc(Cl)cc2[nH]1 6181,C(=O)(C(CO)C(C)C)N1CCC(CCNC(Cn2nc(C)oc2=O)=O)C1 6182,C(CC(C(C)C)NC(c1cscc1C(=O)OC)=O)N(C(CCC)=O)C 6183,N1(Cc2cc(CNCc3cccc(OC)c3F)ncc2)CCCC2(CCC2)C1 6184,c1(C(=O)NC2CC3CC(NC(C(C)SCCCC)=O)C3C2)cc2nccnc2[nH]1 6185,N1(C(C2(CSC)CC2)=O)CC(C)CN(C(=O)Cc2nsc3ccccc23)C(C)C1 6186,c1(CCC(=O)NC(C2CC(NC(=O)C(C3CCCC3)OC)C2)C)cccnc1 6187,C1(NC(c2nc(CCC)oc2)=O)CC12CCN(C(c1ccoc1C1CC1)=O)CC2 6188,N1(C(CC2CC(C)(C)N(C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)CC2CSCC2(C)C1 6189,c1(C(=O)NC2C(NC(COC(C)C)=O)C2)ccc(C(N)=O)o1 6190,N1(C(CN(CC)CC)=O)CCN(C(=O)CCc2cccc(C)c2)CC1C1CC1 6191,C(=O)(C1=CCCCC1P(C)(C)=O)OCC(OC)OC1CC1 6192,CCCCCC(C)(CC)C(=O)N1C(CC)C(COC)OC1=O 6193,N1(NC(C2(C)C(CC)CCC2)=O)CCC(C)C(CC(=O)N(CC(CC)CC)C)C1 6194,C(CNC(=O)C(N1CCOCC1)C)(CCNC(c1ccc(Cl)o1)=O)OC 6195,C(CC(=O)NCCSCCCO)(C(F)(F)F)NC(=O)C(c1ccccc1)F 6196,CCC(C)(CNC(=O)CSC)CN(C)C(C1CC=CCC1)=O 6197,C1(C(=O)NCC2C(NC(Cc3c(Cl)cn(C)n3)=O)CCCC2)CCCCC(F)(F)C1 6198,C(=O)(C(O)Cc1cnn(C)c1)N(CC(C)N(C(=O)C(C)NC(C(C)(C)C)=O)C)C 6199,Cn1nncc1C(=O)NCC1(NC(=O)CCN2CCCC2=O)CCOC1 6200,c1(C(c2nnnn2CCOC)NC(CC)(CC)CC)cc(Cl)ncc1F 6201,c1(C(=O)NCC(C2CC2)NC(c2cccnc2S)=O)cc2ccsc2s1 6202,N1(CC)CC(C(=O)NC2CC3CCC2(NC(c2ccnc(C)c2)=O)C3)CCC1=O 6203,c1(C(=O)NC2C(NC(CC(CC)CC)=O)CC2)cnc2ccoc2c1 6204,C=CCCCCC(=O)NCCC=C.C1(CCSC)C(=O)N1 6205,N1(C(C(C)C2CCCO2)=O)CC(NC(c2sc(Br)cc2F)=O)CC1C 6206,c1(C(=O)NC2CC(O)(CNC(C(c3cn(C)nc3)O)=O)C2)cccc2oncc12 6207,CC(CCF)N=c1nc(N2CCC(O)C(F)C2)c2cc(C(F)(F)F)ccc2[nH]1 6208,C=C(C)CCC(=O)N(C1C2CN(C(=O)CN3CC4CC4C3)CC12)C 6209,Cc1cc(C(=O)C(=O)NC2CCCCC2NC(=O)Cc2cnn(C)c2)ccc1F 6210,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CN(C(=O)C(C)CSc3ccccc3)C2)c1C 6211,C(=O)(CC(CC)CC)NC(C1CN(C(=O)CCOc2ccc(OC)cc2)C1)CC 6212,O=S(=O)(c1ccc(Cl)c(F)c1F)N1CCCC1CC(c1ccccc1)O 6213,c1(CNC(N2CCC(OC)C2)=O)ccc(N2C(=O)CCC2C)cc1 6214,CCC(CC)C(C)C(=O)NCC(C1CCN(C(c2nc(C)n(C)c2C)=O)CC1)F 6215,C1(C(C(=O)NCCC#N)N(C)CC2CC(F)(F)C23CCC3)Cc2ccccc2C1 6216,Cc1ccnc(C=CCOC(C2CCN(c3ccccc3)C2)=O)c1 6217,N1(CCC(=O)N(c2nnnn2CCC2CCCCC2)CC)CCCCCC1 6218,c1(NCC)ccc(Cl)cc1C(=O)NCC(F)CNC(C1CC2CC1CO2)=O 6219,N1(C(C2CC=CCC2)C(=O)N(c2c(C)cccc2)C2CC2)CCS(=O)C(C)(C)C1 6220,C(=O)(CC=C(Cl)Cl)NCCC(C)N(C(=O)Cc1ccccc1OCC#N)C 6221,CSC1=C(C(=O)NCC(C2CCOC2)NC(=O)CC2=NNC(=O)C2)CCCC1 6222,N1(C(Cc2ccc(C)o2)=O)CCCC(O)(CNC(C2CCN(C)C2=O)=O)CC1 6223,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CC3)CCCO1)=O)C2 6224,c1(C(N2CCC(C(C)O)C2)C(=O)NCCC)cc2ccc(OC)cc2o1 6225,C(N=c1ccn(C(C)(C)C)[nH]1)C1CCC(C)(C)C1 6226,c12ccc(c(C)c1)S(=O)(=O)N2.C1(C(=O)OC)C(Cl)(Cl)C12CC2 6227,c1(C(N(CCCN(C(=O)CCCF)CCO)C)=O)cc(C2CC2)ccn1 6228,N1(C(c2c[nH]cc(Cl)c2=O)=O)CC2CN(c3cc(C(F)(F)F)ncn3)CC2C1 6229,C1(CCCNC(c2nnnn2C(C)C)CCC)CCCCCC1 6230,C(C(C(=O)N(CCNC(=O)C(C)(C)c1cnn(C)c1)CC1CC1)OC)OC 6231,c1(N2CCC(NC(C3(O)CCOCC3)=O)C2=O)cccc(Br)c1F 6232,c1(CC)cc(C(=O)NC(C2CCCC2)CNC(C2CC3CCC3C2)=O)cc(O)n1 6233,C12(CC)CC(C(=O)NC(CNC(c3coc(COC)n3)=O)CO)(CO1)C2 6234,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C2N(C)CC(O)C2)=O)CC1O 6235,c1(C(=O)NC(CC(=O)NC(CC=C)(C)C)CC)cc(Cl)ccc1O 6236,N1(C(C2CCOC2)=O)CCN(S(=O)(=O)Cc2cncs2)CC1.N12CCC(C1)C2=O 6237,Fc1ccc(C2CCCN2Cc2cscc2Cl)cn1 6238,C(=O)(C1=COCC1)N.C1(C(C)(C)C)CC(C(=O)NCCN(CCC2CC2)C)C1 6239,CCCC(C(O)C(=O)N(OC)C(C)(C)C)NC(c1nccs1)=O 6240,c1(C(=O)NCC(=C2CN(C(=O)CSC3CCCO3)C2)F)cnc(C(N)=O)cn1 6241,Cc1nnc2n1CCCC2C(=O)NCC1(F)CCN(C(=O)CNC(N)=O)CC1 6242,c1(CCC)ccc(S(=O)(=O)N2CCC2C(=O)Nc2c(C)ccc(OC)c2C)cc1 6243,CC(CC1CCC1)N=c1[nH]c(=NCc2cc(Br)cn2C)[nH]c2c1CCC2 6244,C1(NC(CC(C)n2ccnc2)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C1(C)C 6245,C1(C(=O)NCc2cccc(N(C(CNC(=O)OC)=O)C)c2)CCCCN(C)C1=O 6246,C1(C)(NC(C(C)CN(C(=O)CCCCN(C)C)C)=O)CCC(C)C1(C)C 6247,c1(OCCC(N2CC(NC)C2)=O)ccc(Cl)cc1Cl.N12CCCC(C1)NC2=O.CO 6248,c1(C(N2CCC(CCNC(=O)Cc3ccco3)C2)=O)ccc(F)c(F)c1 6249,CCC(CC)(CC(=O)OC)C(=O)NC1CCCN(C(=O)CCN2CCCC2)CC1 6250,c1(C(N2C(CNC(c3ccc(CO)cn3)=O)CCC2)=O)cn2cccc(Br)c2n1 6251,c1(CCC(=O)NCC(C)(CO)NC(Cc2n(C)ncc2)=O)nnc(S)nc1O 6252,CC1(NC(=O)CCC2CC2)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 6253,c1(CC(N2CCN(C(C3(Br)CC3)=O)CC2CO)=O)ncc(F)cc1F 6254,Cc1cc(Cl)c(C(=O)NCC2(CNC(C3CNC(=O)CC3C)=O)CC2)cc1N 6255,C(=O)(C(C)C(C)NC(=O)CCC1OCCO1)N(CC(=O)NCCC)C 6256,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6257,C1(c2nnnn2C2CCOC2)(NCC2CC(=C)C2)CCN(C(=S)NCC)CC1 6258,N1(C(CC2CC(C)C2)=O)CC2CC1C2NC(c1ccnc(N2CCN(C)CC2)c1)=O 6259,CC(F)(F)CCC(=O)NC1CC(NC(C2CC3CCC2CC3)=O)C1(C)C 6260,C1(N(C(c2cnn(C)c2I)C(=O)NCC(F)F)C)C2CC3CC(C2)CC1C3 6261,C(=O)(CCS(C)(=O)=O)NCCC1(C(=O)NCCC=C=C)CCC1 6262,N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)C(=O)NC2CC2)CC1c1cnn(C)c1 6263,c1(SCC(=O)NC(CC)CNC(c2cnn(C(F)(F)F)c2)=O)cccc(Br)c1 6264,C(C1=NOC2CN(C(=O)C=CCO)CC12)NC(c1ccc([N+](=O)[O-])cc1O)=O 6265,Cc1cccc(CN2C(=O)NC(CCCc3ccsc3)C2=O)c1F 6266,C1(CC=C)(NC(c2csc(C(C)(C)C)n2)=O)CCN(C(=O)C(C2CC2)OC)CC1 6267,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6268,C1(CC(=O)NCC(C2CC2)NC(C=C(CC)CC)=O)CCCOC1 6269,c1(C(=O)NC(C2CN(C(=O)CCN3CCCCC3=O)C2)C)cnc2[nH]cncc1-2 6270,C1(CC(=O)NCC(C)(C2CC2)NC(=O)C(=Cc2cn(C)cn2)F)(OC)CCSCC1 6271,N1(C(C(C(CC)(F)F)(C)C)=O)CC2CC(C1)C2N=c1cc[nH]cc1[N+](=O)[O-] 6272,Cc1cn(CC(N2CC3C(C2)N3C(=O)Cc2cccc(F)c2)=O)nc1C(F)(F)F 6273,C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6274,C(=O)(C(F)(F)c1ncccn1)NCCCCNC(c1ccoc1C1CC1)=O 6275,C1(CCC)CN(C(=O)CC2C=NN(C)C2=O)CCN1C(=O)Cc1ccc(C)s1 6276,CC1CCN(C(=O)CNC(C2CCCC2O)=O)C(CNC(C2CCC(=O)N2)=O)C1 6277,c1(CNC(C2C(C)(C)CO2)=O)nc(CNC(C2(CCO)CC2)=O)cc(O)n1 6278,C1(N(C(c2cc(CC)no2)=O)CC2CC2)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6279,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6280,N1(C(c2cnc3cc[nH]c3c2)=O)CC23CCCCC2(C1)CN(C(C1CC1F)=O)C3 6281,Cc1ccc(C(=O)NC(C)CN(C)C(C2CC(=O)NC2(C)C)=O)cc1N 6282,CCCCC(F)C(=O)NC1CCCCC1C(=O)NCc1cc(C)nn1C 6283,C1(OC)CC(F)CN(C(C2CCC(C)N2C(=O)Cn2cnccc2=O)=O)C1 6284,C1(NC(N2C(c3n(C)ccn3)CCC2)=O)CCC(F)(F)CC1 6285,c1(OC)cc(N2CC(OC)CC2CNC(=O)COc2cn[nH]c2)nc(C(N)=O)n1 6286,C(=O)(CC(C)(O)C(F)(F)F)N1C2CC(NC(CCCCC#C)=O)CC1CC2 6287,C(C(C)(C)CC(=O)NCC(C(C)C)NC(c1ccn(C2CCC2)n1)=O)OC 6288,C1(CC=C)(NC(C2CCC(N(C)C)CC2)=O)CCN(C(=O)C(O)CC)C1 6289,Cc1c(C(=O)NC(CNC(=O)C(C)Oc2cccnc2)C(C)C)ccn1C(C)C 6290,c1(C(=O)NC2C(NC(c3c(COC)cc[nH]3)=O)CC2)ccc2c(c1)NC(=O)CS2 6291,N1(C(C(C)OC(C)=O)=O)CCC(C)(CC(=O)NCC(C)CC2CCC2)C1 6292,N1(CCNC(COC(CCC)=O)=O)CCN(CCc2cccnc2OCC)CC1 6293,CC1(C)COCC1C(=O)NC(Cc1ccoc1)C(=O)Nc1cn(CCF)nn1 6294,c1(NCC2CN(C(c3c(C)n[nH]c3)=O)C2)ncnc(N(C)C)c1[N+](=O)[O-] 6295,c1(OC)ccc(OCCCC(=O)NCC2CC2)cc1.C12CCC1C(=O)N2 6296,N1(C(C(F)=CC)=O)CC(NC(=O)Cn2cnc(Br)n2)CC(O)C1 6297,C(=O)(C(C)(C)CCC#N)NCc1cncc(C(N(C2CC(O)C2)C)=O)c1 6298,N1(C(C(F)=CCC)=O)CCCC(CCC)(NC(=O)C(C)Cc2ccc(F)cc2)C1 6299,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CCCCC2)CC12CCC2 6300,N1(C(C2N(CC)CC2)=O)CCN(C(C2CCN(C)CC2)=O)CC1c1ncc[nH]1 6301,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6302,C1(NC(CC(C)(C)OC)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C(C)C)cc1 6303,C1(C(C)C(=O)Nc2cn(-c3ccccc3)nn2)CCCN(C2CCC2)C1 6304,c1(CC(=O)N(CC(CNC(c2c(OC)n[nH]c2)=O)C)C)cn2cc(C)sc2n1 6305,c1(C(N(CCCN(C(=O)CCc2ccccn2)C)C)=O)cc(F)c(F)c(N)c1Cl 6306,N1(C(c2c(C(C)C)noc2)=O)CC2(CCN(C(=O)CNC(c3cccs3)=O)C2)C1 6307,N1(C(=O)Nc2ccc(OC(C)C)cn2)CC2(CC2)c2ccc(Br)cc21 6308,N1(C(CC2C(OC(C)(C)C)CC2)=O)CCC(F)(CNC(=O)C(F)(F)C(F)F)CC1 6309,c1(N2CCN(C(C(CCC)NC(N)=O)=O)CC(O)C2)nc2ccc(F)cc2o1 6310,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6311,C1(NC(c2c(NC)nccc2)=O)CCN(C(=O)CC(F)(F)F)C(C)C1 6312,CN1CCc2cc(C(N3CCN(C(=O)C(C)(C)CO)CC(CO)C3)=O)sc2C1 6313,c1(NCc2ccn(CC#C)n2)cn(CC(=O)NCC#N)c2cccnc12 6314,Cc1ncnc(C)c1CC(=O)NCC(CNC(C1CCCCS1)=O)C(F)(F)F 6315,c1(C(=O)NC2C(C(=O)Nc3c(I)ccc(OC)c3)C2)ccc2cccc(Br)c2n1 6316,c1(C(N(CC(COC)O)C)=O)oc(CNC(C2CCCS2)=O)nc1C 6317,CC1CCC=C1C(=O)NC1(C(=O)NC(C)(CO)C2CCC2)CCSC1 6318,CC1CN(C(c2nccnc2C(N)=O)=O)CC1NC(C1C2CCCCC12)=O 6319,c1(NC(c2ccc(C(=O)NCc3ccsc3)[nH]2)=O)ccc(NC2CCCC2)c(F)c1 6320,Cc1cc(CNC(=O)Cc2cc(-c3ccc(CC(C)C)cc3)nn2C)ccc1F 6321,Cc1cc(CC(=O)NC2CC2C(=O)NCCc2csc(S)n2)no1 6322,N1(C(c2c(SC)cn(C)n2)=O)C2CC=C(C(=O)N3CCC(C(C)(C)O)C3)C1CC2 6323,C1(C(C)C(=O)NCc2coc(C(F)F)c2)CCN(C(=O)CC2COC(=O)N2)CC1 6324,C1(NC(CC(C(C)C)O)=O)CCN(C(C23CCCCC2C3(F)F)=O)C12CCCC2 6325,N1(C(=O)CSCC2C3CC4C(C3=O)C24)CC2(CCCC2NC(c2cccs2)=O)C1 6326,CCCCC(C)CCC=O.C1(=O)CC(C)(N)C1=O.NNC 6327,C1(CNC(CCN(C(C)=O)C)=O)(OCC(=O)O)CCOC1.C1C(=O)N1C1CC1 6328,c1(C(N(C(C)C(C)C)CC)=O)cc(COC)no1.C1(=O)C(OC)N1 6329,c1(C(N2CCC(C)(CNC(C3C(C)(C)C3C#N)=O)CC2)=O)ccccc1N=[N+]=[N-] 6330,N1(C(C2C(OCC)C2)=O)CCC(F)C(NC(c2sc(C(C)OCC)nc2C)=O)C1 6331,C=CC(O)(C(=O)NCCC1(NC(=O)CC(C)C2CCCCC2)CC1)C(F)(F)F 6332,N1(C(C(C(C)NC(c2c(C)nsc2N)=O)C)=O)CCC2CCCC12 6333,N1(C(C(CO)SC)=O)CCCC(C)(CNC(c2c(C)csc2Cl)=O)C1 6334,c1(CNCc2nc(-c3cccc(Cl)c3)on2)ccc2cnccc2c1 6335,N1(C(CCN(C(C(CCCC)=O)=O)CCO)=O)CCC2(CCCC2)C1 6336,C1(CC=C)(NC(c2cc(CC)on2)=O)CCN(C(C2COCCC2C)=O)CC1 6337,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C=CC=CC)=O)CC1CCOC 6338,c1(OC)cc(C(C(=O)NC2(C)CC2)N(C2CC3(C2)CC(F)C3)C)cc(F)c1Br 6339,C(=O)(C(F)(F)C(C)O)NC(COC(C)C)C(=O)NCCc1ccncc1 6340,N1(C(C2C(C(=O)OC)C=C2)=O)CCC2(CC1)CC(NC(c1cc(O)ncn1)=O)C2 6341,Cn1ncc(CN(C)CC2CCN(C(C3(C#N)CCCO3)=O)CC2)c1Cl 6342,C(CCC(C)C)(C(=O)NC12CC(C(N)=O)(C1)C2)NC(c1cccc(CC)n1)=O 6343,c1(CC(=O)NC(C)CCNC(c2scnc2Cl)=O)ccnc(O)c1 6344,c1(NC)ccc(C(=O)NCCN(CCCN(C)C)C(c2c[nH]nc2F)=O)nc1 6345,CS(=O)(=O)C1(Cn2cc(CCNC(=O)CCC3CCCN3C)nn2)CCC1 6346,CCCCC(C)C(=O)NC1COCCC1NC(C12CC(F)(C1)C2)=O 6347,Cc1nccnc1C(=O)NC1CC(C(=O)NCCCC2CCCO2)C1 6348,C1(N(C(CN(CCC)C)=O)C2CC2)CN(C(=O)CCc2ccc(C)s2)CCCO1 6349,N1(C(CC(=O)N(C)C)=O)CCC(NC(=O)CN(C)S(=O)(=O)N(C)C)C(CO)C1 6350,N1(C(CCC(C)NC(=O)CS(=O)(=O)N(C)C)=O)CCC(CO)(CO)CC1 6351,c1(C(N(CCC)CCNC(=O)C(F)CC2CC2)=O)c(Br)ccc(F)c1C 6352,CC1Sc2ccc(C(N3CC4CCC4(CC(=O)O)C3)=O)cc2NC1=O 6353,C#CC1(F)CN(C(c2ncoc2CNC(=O)C(C(C)C)OC)=O)C1 6354,C1(CNC(=O)CC2CC2)CN(C(=O)C(F)c2cnco2)CCCO1 6355,C(=O)(CCC(C)(C)C)N1C(C)CC(CNC(Cc2ccc(C)cc2)=O)C1 6356,C1(OC)CCCN(C(=O)CC2CCN(C(C3CC4(CC4)C3)=O)C2)C1.CC(=O)O 6357,C1(C(=O)NC(c2n(CC)cnn2)Cc2ccc(F)cc2)CCC(C)(C)O1 6358,c1(C(C(=O)NC)N(C2(C#N)CC(C)(C)C2)C)cccc(OC)c1Cl.n1(CC)ccnc1 6359,C1(F)(CNC(c2n(C)nnc2)=O)CCCN(C(=O)C(C)(C)CF)C1 6360,C1(C(=O)OC)CCCC12CN(Cc1ccc(F)c(C)c1F)C2 6361,C1(NC(=O)CCc2ccncc2)CCCCC1C(=O)NCC(=O)OCCC=C 6362,C(=O)(C(COCC)N=[N+]=[N-])NC(CCC)CNC(=O)Cc1ncccc1F 6363,c1(C(N2C(CC(=O)Nc3c(Br)cc(C)c(C)n3)CCC2)=O)ccc2c(n1)OCCO2 6364,C1(C(=O)NCC(=O)NC(C)C)CCCC(NC(C2(C#N)CCOC2)=O)CC1 6365,C1(CNC(c2c(OC)nccn2)=O)CN(C(c2cnc(N)c(N)c2)=O)CCCO1 6366,c1(CC(=O)NC2N(C(COCCCCC)=O)CCC2)ccc2nc[nH]c2c1 6367,C(CCN=c1nc2c(c[nH]1)CCCCC2)NC(c1cc(CC(F)(F)F)on1)=O 6368,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCCN(C(c1n(CC)nnc1)=O)C1CC1 6369,Cc1cc(C(=O)NC2CCC2CNC(=O)C(C)C2CC2)sc1Cl 6370,O=C(N=c1[nH][nH]c2c1CN(C(c1cnnc(Cl)c1)=O)C2)c1cc(F)c(F)cc1F 6371,N#CC1=C(C(=O)NCCC2(O)CCN(C(C34CCC(CC3)CO4)=O)C2)CCC1 6372,C(C(O)CC(=O)NC1C=CCN(C(C2CCCN2c2nccs2)=O)C1)N(C)C 6373,N1(C(c2nc(OC)oc2)=O)CC2CC3CC2C1C3NC(c1cc(C)oc1C)=O 6374,Cc1[nH]c(C#N)cc1C(=O)NCCCCCN(C(=O)COCc1nc[nH]n1)C 6375,C(=O)(C(C)C(C)NC(=O)CC1CNC(=O)O1)NCc1c(C(C)(C)C)n[nH]c1 6376,C1(NC(N(C(C)CO)C(c2ccccc2)COC)=O)CCC2CCOC1C2 6377,CC(CC(=O)NC1CCCOC1)C(C)(C)NC(c1ccc([N+](=O)[O-])[nH]1)=O 6378,S(=O)(=O)(c1cc(F)ccc1OC)NC1CC2(CC(NC(c3c(OC)nsc3)=O)C2)C1 6379,N1(C(=O)C=CC2CC2)CCCCCCC1C(N1CC2(CO)CC2(CO)C1)=O 6380,C=CCC(F)(F)C(=O)NCC(C1CC1)N(C)C(c1cc(Cl)cnc1OC)=O 6381,C(=O)(CS(=O)(=O)CC(=O)NCC1CCC(NC(C2CCS(=O)(=O)CC2)=O)C1)OC 6382,N1(C(c2c(OC)ccs2)=O)CCCC(C2CCN(C(=O)Cc3nnc(C)o3)C2)C1 6383,C1(CNC(CCC(=C)Br)=O)C(C)CCCN1C(=O)Cc1ccc(F)cc1 6384,C1(NC(Cc2cn(C)nc2)=O)CCCN(C(=O)CC(F)(F)Cl)C1 6385,C1(C)(CC)COCCN1C(c1ccc(O)c(F)c1)C(=O)NC1CCC1 6386,C(CCS(C)(=O)=O)(C(=O)NCCN(C1CCCOC1)C(C)=O)OCC 6387,CC(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCC12CCC2)S(N)(=O)=O 6388,c1(CCN)cc(-c2ccccc2)ccc1F.C1(c2n(C)nnn2)CCCCC1CN 6389,CC1=CCN(C(=O)C(C)NC(=O)CC2CCCCC2)CC1 6390,C(CCCCC(=O)NC1CCC(C)(CNC(c2cc[nH]c2)=O)C1)=CC 6391,C1(NC(c2cccc(C)n2)c2n(CCCOC)nnn2)C(C)CCC1C 6392,N1(C(C2CC3(CN(C(C)C)C3)C2)=O)CCC2(C1)C(=O)NC(=O)N2C 6393,N1(C(c2nccc(CNC(C(C(C)O)O)=O)c2)=O)CCN(CCO)C(=O)C1 6394,C(=O)(CC(C1CC1)NC(=O)C(C1CCCCC1)F)N(C)CCC1CCCO1 6395,c1(C(N2CC(C)(NC(c3cccc(C)c3C)=O)C2)=O)cc(Cl)c(F)cc1O 6396,c1(C(=O)NCCN(C(c2cn(C3COC3)nn2)=O)CC)csc(I)c1 6397,Cc1ccc(F)c(N2CCCC(C(=O)NCC3CN(C(=O)C(F)C(C)(C)O)C3)C2)c1 6398,CC#CCCC(=O)NC(C)(CNC(=O)C(C)n1cncn1)C(C)C 6399,C(C(CC1CC1)C(=O)NCc1ccncn1)NC(C1(C)CC(=O)C1)=O 6400,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCC2CC2(F)F)CC12CCCC2 6401,c1(C(=O)NC(CCNC(C)=O)C(C)C)cc(O)nc2c(Br)cccc12 6402,C(=O)(C(O)C(F)(F)F)NCC1(NC(C2CCN(C3CCN(C)CC3)CC2)=O)CC1 6403,N1(C(c2ccc(NC(C)=O)c(F)c2)=O)CC2OCCN(C(=O)CC(C)C)C2C1 6404,C(=O)(C(C)C(O)CC)OC(CC(=O)NCC=C)SC 6405,N1(C(c2c(C)ocn2)=O)CCC(C)C(CC(=O)N(C2CNC(=O)C23CC3)C)C1 6406,C(=O)(CC1COCc2ccccc21)NCCN(C(Cc1ccc(C)s1)=O)C1CC1 6407,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6408,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3CCC3)COC1C2 6409,C1(C)(C(=O)NCCC=C=C)CCN(C(=O)C(C)C2CCCC2)CC1 6410,c1(C(=O)NCC2C(C)CCCN2C(C2CCCN2C)=O)cnc2ccnn2c1N 6411,c1(C(C)(C)C)cccc(CNC(=O)CC2CC(F)CN2C(=O)CC2CNC(=O)O2)c1 6412,N1(C(COCC)=O)CCN(C(c2cc(SC)oc2C)=O)C2CCCCC2C1 6413,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6414,CN1CCOc2c(C(N3CCC(NC(C4(C)CC4(F)F)=O)C3(C)C)=O)cccc21 6415,c1(NC(C(C(C)C)NS(=O)(=O)c2cnn(C)c2)=O)cccc2c1OC(C)(C)C2 6416,c1(NC(COC(C)(C)C)=O)cc(N2CCOC(CF)C2)ncn1 6417,c1(CC(=O)NC(C#C)C)cn2cc(-c3c[nH]nc3C)ccc2n1 6418,CC1CC(C(=O)NCC2(C(=O)N(C3(c4cc[nH]n4)CC3)C)CC2)CN1C 6419,N1(C(CC2(NC(=O)OC)CCOCC2)=O)CCC2CN(C(=O)CC)C2C1 6420,N1(C(c2c(C)c(O)cc(N)c2)=O)CCC(C)C(NC(C2CCCCCC2)=O)C1C 6421,C12(C(N3CC4CC4(NC(c4snc(O)c4Cl)=O)C3)=O)CCCN1CCC2 6422,c1(C(N(C2CCCN(c3ccccc3)C2=O)C)=O)cc2cccc(F)c2s1 6423,C1(NC2CC(C(=O)Nc3c(C(=O)OC)nccn3)C2)CC2(CCC2OC)C1 6424,c1(C(=O)NC2CC(NC(c3cccc(C4CC4)c3)=O)C2)cnn2cccc(Cl)c12 6425,Cc1cnccc1C(N1CC(O)(CCNC(c2csc(Cl)c2Cl)=O)C1)=O 6426,c1(CCOCCOC)noc(C)n1.N12CC(C1C)C2=O.c1(O)ccccc1.C(C)C 6427,C1(OC)CN(C(=NCCCSC)NCc2cn(Cc3cccs3)nn2)CC1OC 6428,C(=O)(CCCCCc1cccs1)NCC(C)(CNC(=O)NCC#N)OC 6429,CCCCCC(O)CC(=O)NCCCC(C)(C)NC(=O)Cc1ccc(Br)cc1 6430,C1(CC)CCN(C(=O)C(CCOC)OC)CC1n1nnc(N2CCNCC2)n1 6431,C1(C(N2CCCC2CC(F)(F)F)C(=O)NCCn2ccnn2)CC12CCC2 6432,C(CCC(C)C(=O)NCCC1(OCC(=O)NC2CC2)CCC1)OC 6433,N#Cc1cc(S(=O)(=O)NCCC(O)C(F)(F)F)ccc1NC1CN2CCN1CC2 6434,C(=O)(C1=CC2CCC1C2)N1CCCC(NC(C=Cc2cccc(C)c2)=O)(CO)C1 6435,C12(NC(C(C3CC3)OC)=O)CCCC(CN(C(=O)Cn3cc(C4CC4)nn3)C1)C2 6436,Cc1cc(N)c(C(=O)NC2CN(C(c3coc(Cl)n3)=O)CC23CCC3)cc1C 6437,c1(C(=O)NCCC(C)(C)NC(C2CCc3n[nH]cc3C2)=O)ccc(F)c2ccoc12 6438,c1(NC(COC(c2c(CC)n[nH]c2)=O)=O)nsc2ccc(C)cc12 6439,CN1Cc2ccc(OC)c(c2)C(=O)NC2N1CC(C)(C)C2.C1(CCC)CC1 6440,CC1CCCC(C)N1CCC(=O)NCC1(C)CCN(C(c2sccc2F)=O)C1 6441,C(=O)(C(O)C(C)(C)C)NCC1(C(=O)Nc2nccc(C(C)(F)F)c2)CC1(F)F 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6459,C(CNC(=O)C(N1CCCCC1=O)C)(CC(C)C)NC(c1c(C)csc1)=O 6460,c1(C(=O)NCCOC(CNC(CC(CCC)C)=O)(C)C)ccc2c(c1)CCOC2 6461,C1(NC(N2CCC(n3c(CNC(C)=O)ncn3)C2)=O)CCc2ncccc2C1 6462,N1(C(c2ncc(F)cn2)=O)CC(F)(F)CC1CCNC(C1CCCCC1)=O 6463,c1(OCCC)c(OC)cc(C(=O)NCC(C)(CO)NC(=O)C(C)CF)cc1Cl 6464,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1nccnc1O)=O 6465,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6466,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(=O)Cc3conc3C)CC12 6467,c1(N2CC(CCN3C(=O)C3)C2)ccnc2ccnn12.c1(NC(N)=O)cccnc1 6468,c1(C(N(CC(C)N(C(C(CC)n2cccn2)=O)C)C)=O)cn(C)nc1COC 6469,c1(CNC(C2(CSC)CC2)=O)nc2c(s1)CCN(C(c1ccn(C)c1C)=O)C2 6470,CCC(C)C(CC(=O)NCC(C)(F)C(C)(C)F)NC(c1cccc2ccnn12)=O 6471,c1(CCN2CCC(N(CCC)C(c3ncccc3F)=O)C2)ccccc1[N+](=O)[O-] 6472,N1(C(CCC(=O)N(C)C)=O)CC2CCCN(C(c3cccc4c3CCC4)=O)C2C1 6473,Cc1cccc(CN2CC3CC2C3C(=O)Nc2cccc(O)c2O)c1O 6474,c1(C(=O)NCC2N(C(C3CC(C)N(C)CC3)=O)CCCC2)ccc2cccnn12 6475,C(C)(C)(C(=O)NC1CC(CNC(c2coc(C(F)F)n2)=O)C1)N(C)C 6476,N1(C(C(C)C)C(=O)NCC2CCCO2)CCCCCC(N)C1 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6495,C12(CNC(CCCCC)=O)CCCC1N(C(=O)C(F)=C(C)C)CCC2 6496,C(C(=O)NC1CN(C(c2cc(O)nn2C)=O)CC1C(F)(F)F)(C(C)C)SCC 6497,N1(C(CCN(C(c2ccc(C(C)=O)o2)=O)C)=O)CCC(NC2CC2)CC1C 6498,C12(C=O)CC(CN(C(=O)CCCCCF)C1)C2.C(=O)CCC1CCOC1 6499,N1(C(c2ccc(F)cc2Br)C(=O)NCCOC)CCOC2(CCSC2)CC1 6500,c1(C(=O)NCC(CNC(=O)CC2(N3CCCC3)CC2)OC)ncccc1F 6501,c1(C(=O)NC(CC)C#N)ccc(=NCc2cc(F)ccc2Br)[nH]c1 6502,Cc1cn(C)cc1C(=O)NCC1(F)CN(C(=O)CC2CCC(C)C2)C1 6503,N1(CC(=O)NC(c2cc[nH]n2)=O)CC2(CCC(C)CC2)C1.Cc1ccc(OCC)cc1 6504,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2F)=O)c(Br)c1 6505,Cc1ccc(C)c(C(=O)NC(CNC(c2cn[nH]c2)=O)C(C)C(C)C)c1 6506,C12(O)CCCN(C1)C2=O.n1(CC(=O)N(C2CC(NC(C)=O)C2)C)nc(C)oc1=O 6507,N1(CC(C)OC(C)=O)CCN(C(=O)CC(C)NC(c2ccccc2)=O)CC1 6508,c1(C(=O)NC2CCN(C(CCCCCOCC)=O)C2)ccc2c(c1)COC2 6509,C1(CCC)CN(C(c2cc(C)n(C(F)F)n2)=O)CCN1C(=O)C(C)C1(O)CCC1 6510,c1(NC(C2C(CNC(c3cc(CC)oc3C)=O)CCCC2)=O)ncc(Cl)cc1Cl 6511,c1(N(C2CC(N)C2)C(c2cccnc2Br)=O)ncnc2ccc(I)cc12 6512,C(=O)(C(CC(F)F)N(C)C(c1ccnc(C)n1)=O)NCc1nc(CC)on1 6513,O=C(C1=NOC2(CCC2)C1)NCCC1(NC(=O)C(c2ccccc2)F)CCOC1 6514,C1(C(=O)NCC(CN(C(C(C(=O)OC)(C)C)=O)C)(C)C)CCC2CCC(=O)N12 6515,C1(O)(NC(=O)COC(=O)CC2CCS(=O)(=O)C2)COCCC1O 6516,C12(NC(=O)C(C)CCOc3ccccc3)CC(CO)(CO1)C2.CCC1CN1C 6517,c1(C(N2C(C)(C(=O)Nc3ccc(CCC)cc3)CCC2)=O)cccc2c1OCC2 6518,N1(C(C2CCCC2C(=O)O)=O)CCCC(c2cn(CC3(F)CCOC3)nn2)C1 6519,Cc1csc(CCCC(=O)NCCC2CCN(C(=O)CC34CCCC3C4)C2)n1 6520,N1(C(Cc2cc(C)on2)=O)CC(C(=O)NCCc2ncc(C)o2)OC(C)C1 6521,C1(CNC(c2c(C)nn(CC(F)F)c2)=O)CC2(CC2)CN1C(=O)C(C)CCO 6522,N1(C(C(=O)CC2CCC2)=O)CCC2(C1)CN(C(=O)C(O)Cc1cnc[nH]1)C2 6523,C12(C(N(C(C(N3C(C(=O)OC)CCC3)=O)C3CC3)C)=O)CCCC1C2(F)F 6524,N1(C(=O)NCC(C)S(C)(=O)=O)CCC(C(=O)OC(C)(C)C)C(F)C1 6525,c1(OC)ncc(C(N2CCC(CNC(c3cc(=O)n(C)o3)=O)C23CC3)=O)cc1Cl 6526,C1(COCC(=O)NC2CC2)CN(C(=O)CNC(C2C=CC(C(F)F)C2)=O)CCO1 6527,CC1(NC(C2CC2(F)Cl)=O)CN(C(=O)CCCNC(CNS(C)(=O)=O)=O)C1 6528,c1(C(N2CCC(NC(c3c(SC)n(C)nc3)=O)C2C)=O)ccc2c(c1)nnn2C 6529,c1(C(N(C2CN(C(=O)CC#N)C2)C)=O)ccc2c(c1)OC(F)(F)O2 6530,N1(C(c2c(CC)ccc(C)c2)=O)CCC2(COC(CNC(=O)C3=CCCC3)C2)C1 6531,CCCCC(F)C(=O)NC1CC2CC1CC2C(=O)NCC1(O)CCC1 6532,C1(c2n(C3(CNc4cc(C)ncn4)CC3)nnn2)(OC)CCCSCC1 6533,Cc1ccc(NC(=O)C(=O)NCCCN2CCCS2(=O)=O)nc1C 6534,c1(CNC(c2nn(C)c(I)c2)=O)cnc2cnccn12 6535,C1(NC(C(C)N(C(c2c(COC)non2)=O)C2CC2)=O)CCS(=O)CC1 6536,CC1(C(F)F)CN(C(=O)C(c2ccc(F)cc2)=O)CCO1 6537,C(=O)(CCCCNC(=O)OC(C)(C)C)NC(C(C)NC(=O)CN(C)C(C)C)CO 6538,C(=O)(CC(O)CC(C)(C)C)NC(CC)(CC1(NC(=O)C2CC2)CCCCCC1)CC 6539,c1(CC#C)cccc(C(=O)NCCCOCCCNC(C2(N(C)C)CCC2)=O)c1 6540,CCCCCCC(C)CC(=O)N1CC2ON=C(CNC(=O)C3=CCCCC3)C2C1 6541,c1(C(N(C2C(NC(C(C)=CC)=O)CCCC2)C)=O)n[nH]c2ccc(O)cc12 6542,CCC(C(=O)NCC(CNC(c1ccc(CSC)s1)=O)OC)C(F)(F)F 6543,Cc1cc(C(=O)NCCCN(CCOC)CC2CCS(=O)(=O)CC2)ccc1F 6544,CCCCCC(CC)C(=O)NC12CCC(CC1)N(C(=O)C(C)CSC)C2 6545,c1(OC)ccc(C(=O)NCC2(F)CN(C(=O)C(F)C3CCOC3)C2)c(F)c1 6546,c1(C(N2C(CN(C(=O)CC3CC3C3CC3)C)CCC2)=O)cc2cccn2cn1 6547,C(C)(C(=O)NCCCCC1CN(C(c2ccoc2)=O)C1)=C(C=C)O 6548,C1(CN(C)C)CCCCN1C(c1conc1CNC(=O)C=CC1CC1)=O 6549,CC1(C)OC(C)(C)C1C(=O)NCC1CN(C(C2CC=CCO2)=O)CC1(F)F 6550,c1(-c2cn(CC(C(C(c3ccc(CO)cc3)(C)NC=O)=O)=O)nn2)ncc(Br)cn1.N 6551,N1(C(=O)C=CI)CC2CCCC(Nc3ncnc4c3nnn4CC3CC3)C2C1 6552,C#CCCCCCCCC(=O)NC12CCC(CC1n1cc(-c3cnsc3)nn1)C2 6553,c1(CC(=O)NCC23CC(CN2C(=O)CC2CCC2(F)F)C3)nc(F)c(F)cc1F 6554,N1(C(c2cc(C)nnc2)=O)CC2(CCCN(C(=O)CC3CCCC3O)C2)C1 6555,C#CCCCCCC(=O)N1CC(F)(F)CC1CNC(=O)CC1COCC(C)O1 6556,CC(CCC(C)(C)C)C(=O)N(C1CCCN(C(=O)CS(=O)(=O)C2CC2)C1)C 6557,c1(C(N2C(SC(c3cn(C(C)C)nn3)C(C)C)CC2)=O)ccc(F)cc1C(F)F 6558,N1(C(CSCC(C)C)=O)CCC(N(CCO)C(C23CCC2C3)=O)C1 6559,Cc1n[nH]cc1CC(=O)NCC1(CO)CN(C(c2coc(CC3CC3)n2)=O)C1 6560,c1(C(c2n(C(CC)C)nnn2)NCC2(CF)CCC2)ccnc(SC)c1 6561,CCCC(C)(C)C(=O)N1CCC(CC(C)NC(C2CC2c2ccco2)=O)CC1 6562,N1(C(CC(CNC(C(CCOC)OC)=O)O)=O)CC2(CC(OC)CO2)C1 6563,CC1CN(C(C2C=CC=CC=C2)=O)CCCN1C(c1cc(O)nc(Cl)c1)=O 6564,C1(CC(=O)N(C2CN(C(C3CCN(C)CC3)=O)C2)C)CCCOCC1 6565,N1(C(C(c2ccccc2)N(c2ccc(F)c(Cl)c2)C=O)=O)CC(O)CC12CCC2 6566,c1(C2c3n(nnn3)CCCN2)ccnc(C(=O)OC)c1.C(CCS(C)=O)OC 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6602,CC1(C)CCN(C(c2cc(F)ccc2F)C(=O)NCc2ccco2)CCS1=O 6603,CCCCC(CCCC)C(=O)N1CC(COC)CC1CNC(C1CCCO1)=O 6604,Cc1oc2ccccc2c1CC(=O)NC1(C)CCN(C(C2CC23CCC3)=O)CC1 6605,C=CCC(CC(F)F)NC(C12CC1CN(C(c1ccn(C)c1)=O)C2)=O 6606,CCC(CC1CC1)CC(=O)N1CCCC(C(N)=O)(CNC(C2NCCC2)=O)C1 6607,C(=O)(CCCCCSC)NC(CN(C(c1cnn(C2CC2)c1)=O)CC)C 6608,c1(C(=O)NC(CCCC)CNC(=O)CCCc2ccsc2)cc2n(c1)CCSC2 6609,CCCC(C(=O)NCCC1CCN(C(c2nocc2C)=O)CC1(F)F)C(C)C 6610,S(=O)(=O)(CC(=O)NC1CCC(CC(=O)NC2CCCN(C(C)=O)C2)CC1)NC 6611,N1(C(C(C)SCC)=O)CCCC1CCNC(=O)C(C)n1cccn1 6612,C1(CCN(CC=O)C(C)(C)C)CCC2(CC1)CCC2O.C(CC(=O)O)N(C)C(C)=O 6613,N1(C(c2c[nH]c(=N)o2)=O)CCC=C(CNC(C2CCCN2C2CC2)=O)C1 6614,CN1CCc2[nH]nc(C(=O)NC(C)(C)CNC(C3CC4CC3C3CCCC43)=O)c2C1 6615,CCC(C)CC(C(=O)NCCc1nc(C)no1)NC(c1nccc2[nH]ccc12)=O 6616,C1(NC(C(CC)(C)CO)=O)CC2CCC1N(C(=O)CCc1cncc(F)c1)C2 6617,c1(OC)ccc(C(=O)NC(C)CNC(C2NC(=O)OC2C)=O)c(Br)c1 6618,Cc1ccn(CC(=O)NCCC(C)N(C(=O)C(C)SC(C)C)C)n1 6619,Cc1ccc(C)c(C(N2CCC23CN(C(=O)C(C)Oc2ccccc2F)C3)=O)c1 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6691,c1(C(N2C(CNC(=O)C(O)C3CCC3)CC(O)C2)=O)nnc(O)cc1O 6692,N1(C(C2C(C)SCC2)=O)CC2COCC2(C(=O)NCc2ccc(Cl)cc2)C1 6693,C1(CCC)CN(C(=O)C(c2ccccc2F)(C)C)CCN1C(=O)CS(=O)CC 6694,Cc1cn2cc(C(N3CCC(NC(=O)CSCC(F)(F)F)CC3C)=O)nc2s1 6695,N1(C(CCCn2c(C)cc(C)n2)=O)CCCCC(N(C(=O)C=CCF)C)C1 6696,C(C(=O)N1CC(C)(C)C1C(=O)O)(C(C)(C)C)N(C)C(c1ccccc1F)=O 6697,N1(C(COCCCC)=O)CCN(C(c2ccc(F)c(C(F)F)n2)=O)C2COCC12 6698,c1(C(C(=O)NCCCC)N(C(C)C(F)(F)F)C)cccc2nc(CC)sc12 6699,N1(C(CC(OCC)OCC)=O)CC(C)(C)CC1NC(=O)Cc1cc(O)nnc1O 6700,N1(C(c2nc(OC)c(F)cn2)=O)CC2CCC1C(NC(=O)COC(F)(F)F)C2 6701,c1(OCC(N2C(CNC(c3c[nH]ccc3=O)=O)C=CC2)=O)cccc(Cl)c1 6702,n1(CC(C)(C)C)cc(CC(O)Cc2ccccc2)nn1.C1C(=O)N1CCO 6703,C(=O)(C1=NNC(=O)C1)NCC1CN(C(CCc2cnn(C)n2)=O)C1 6704,c1(C(C)C)cc(C(=O)NC(C)(CNC(=O)C(C)n2ccnc2)CO)on1 6705,c1(CN(C(C(C)N(CCC)C(C2CC(CC)C2)=O)=O)C)nnnn1C 6706,c1(C(N2C(C(=O)Nc3ccc(CO)nc3)CC(C)C2)=O)cc2c(ncn2C)[nH]1 6707,Cc1[nH]nc2ccc(C(=O)NCC(C)CNC(=O)COCC3CCCO3)c(Cl)c12 6708,C1(C(=O)NC2CCCN(C(c3cnn(C4CC4)c3)=O)C2)Cc2nncn2C1 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6727,C1(CNC(C=C(C)Cl)=O)CC(NC(c2cnn(CCC(F)(F)F)c2)=O)C12CCC2 6728,N1(C(CCN(CC#C)C(c2occc2COC)=O)=O)CCC2(CCCN2C)C1 6729,c1(C(N2CC=CC(NC(c3cnn(CC)n3)=O)C2)=O)ccc(F)c(C#N)c1 6730,c1(SCC(C)NC(C(=O)NCC(C)N(C(C)=O)C)=O)ccccc1 6731,CCC(C)C(C(=O)N1CC(C(C)C)CC1C)N(C)C(c1ccnn1CC)=O 6732,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(O)(CNC(c2n(C)ncc2C2CC2)=O)C1 6733,C(CC(=O)NC(CCO)C(F)(F)F)(C(F)(F)F)NC(CN1CCC(OCC)C1)=O 6734,C=CCCCCC(C(=O)NC(CC(C)C)C(=O)OC)N1CCCCC1CSC 6735,Cc1ccc(OCC(=O)NCC2CN(C(C3CCS3(=O)=O)=O)CC2C)cc1C 6736,c1(C(N2CCC(O)(CCNC(C(C)(CO)OC)=O)CC2)=O)cc(F)c(C)cc1F 6737,c1(C(N2CCC(CC=C)(NC(=O)CC(=O)OC)CC2)=O)ccc(S(C)(=O)=O)o1 6738,C=CC(O)C(=O)N1CCC1CNC(c1cc(-c2ccccn2)ns1)=O 6739,c1(C(=O)NC(C2CCOC2)CNC(c2nc(C)oc2)=O)ccc([N+](=O)[O-])n1C 6740,N1(C(COC(CNC(CCC=C)=O)(C)C)=O)CC(COC)CC1(C)C 6741,C(CCN=c1[nH]ncs1)N(C(c1cccc(CC(C)C)c1)=O)C.C1(N)CC1 6742,C(=O)(C(C)(C)CC(C)(C)C)N(CC(CC)NC(c1cnc(C)c(C#N)c1)=O)C 6743,C(CN=C(NCCSCCO)NC12CCCC1C2)c1ccccc1 6744,N1(C(COC)=O)CCC(C2CC2)C1CNC(=O)CCn1ccc2cccnc12 6745,Cc1oc2ccccc2c1CC(N1CCC(NC(C2(CCF)CC2)=O)C(F)C1)=O 6746,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(NC(C(N2CC(C)C2)C)=O)C1 6747,C(=O)(NNc1ncnc2[nH]cnc12)c1c(NCC(C)CCl)nn(C)n1 6748,n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CC2NC(=O)CNC(=O)C2CC2)n1 6749,CC(CNC(=O)C(c1ccccc1)Sc1cscc1C1CC1)(CO)NC(N)=O 6750,c1(OC)cc(CC(=O)NCC(n2cc(-c3ccnc(C)c3Cl)nn2)C)ccc1Br 6751,N1(C(c2ccn(CC)n2)=O)CCC(O)C(N(C(=O)C(C)CSC)C)C1 6752,CC(C(=O)NC1CCCN(CCCNC(=O)CC2OCCC2(C)C)C1)S(N)(=O)=O 6753,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)co2)=O)C1 6754,C1(C(C)C(=O)NCC(C2CC2)NC(=O)C(C)(C)NS(C)(=O)=O)CCC(C)(O)CC1 6755,CC1(O)CN(C(C2(C)CCCN(C(c3ccc(Cl)s3)=O)C2)=O)CCC1O 6756,C(=O)(C1=NOC(C)C1C)NCCn1cc(CNC(CSCCC)=O)nn1 6757,CCC(C)C(C(=O)NC1(C(C)O)CC1)N(C)C(C1CCCCN1C)=O 6758,c1(C(N2CC(C)C(C(=O)Nc3cc(S(N)(=O)=O)cs3)C2)=O)csc2ccccc12 6759,C=CCCC(C)NC(=O)NCCNC(c1occc1F)=O 6760,c1(OCC(=O)NCC(C)NC(c2ccc(F)cn2)=O)ccc(C2CC2)cc1 6761,C(CCCCC(=O)NC1(C(=O)NCCSCCCC)CC(CO)C1)=CC 6762,C12OCCC13CN(C3)C2.C1(C)(C(=O)OC)CCCN(Cc2noc(C)n2)C1 6763,C1(NC(C(C)CCc2ccc(F)cc2)=O)N(C(=O)C2CC2)CCCC1(C)C 6764,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6765,CC1(C)OC(=O)CC1C(N1CCC(C)(CC(=O)NCC2(C)CCCCC2)C1)=O 6766,C1(NC(C(C=C)O)=O)CCC2(CC1)CC2.C12CCCCC1CNC2=O 6767,C1(NC(C(CC=CC)C)=O)CC2(C1)CC(C(=O)NCC1(C3CC3)CCCO1)C2 6768,Cc1cc2ccc(C(=O)NCC3(C)CN(S(=O)(=O)c4cccc(Cl)n4)C3)cc2[nH]1 6769,c1(CC(=O)NCC2N(C(CCc3c(C)nn(C)c3)=O)CC2)ccc(Cl)cc1F 6770,c1(C(=O)NCC2CCCCN2C(c2cnc(C3CC3)o2)=O)cc2cccc(Cl)c2o1 6771,c1(CC(C)(C)CO)nc(C2(C3CCCNC3)CC2)n(-c2ccccc2)n1 6772,CCC(CC(=O)NC1CC(CNC(c2ccn(C3CC3(F)F)n2)=O)C1)C1CC1 6773,c1(NC(C(CCO)NC(=O)OC(C)(C)C)=O)coc2c1C(=O)NCCC2 6774,C1(N(C(C(C)NC(CC)=O)=O)C)CCCCN(C(=O)CCC=C(C)C)C1 6775,C1(C)(C(N(C)OCC(F)(F)F)=O)CCCN(C(c2c[nH]c3ncccc23)=O)C1 6776,C(=O)(C1=C(C)OCCC1)N(C1CCC(CNC(c2c(OC)scc2)=O)CC1)C 6777,c1(CC(=O)NCCCN(C(=O)CSCc2ccccc2Cl)C)ccc(O)nc1 6778,CC1CCN(C(=O)CCN(C(c2ccc(C3CC3)o2)=O)C2CC2)CCS1 6779,c1(C(=O)OC(c2c(OC)cccc2)NC)cc(C)c(O)nn1 6780,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)ccc([N+](=O)[O-])cc1Br 6781,N1(C(c2cn(C)nc2)=O)CCC(NC(c2cn(-c3ccccc3)nn2)=O)C12CC2 6782,CCCCCCCCCC(=O)NCC1CCN(C(=O)COCC(=O)OC)CC1C 6783,C1(C(=O)NC2(CC(=O)OCC)CC2)CC2(CC2)CN1C(=O)C=Cc1ccn(C)c1 6784,C1(NC(c2c(OC)noc2C)=O)CCCCN(C(=O)CC(C)c2cccnc2)C1 6785,C(C1C(C(=O)NCC2(F)CC(NC(=O)COCC(F)(F)F)C2)C1(C)C)=C(C)C 6786,C1(F)(C(N2CC(C)(CCC)C2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 6787,C1(C(C(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)O)CCS(=O)(=O)CC1 6788,C1(O)(CC(=O)NC2C(NC(c3c(C)nc(-c4cnn(C)c4)[nH]3)=O)C2)CCCCCC1 6789,C1(NCC)(C(=O)NC)CCN(C(c2cnc[nH]2)=O)C1.C(C)=C 6790,c1(OC)ccc(CNC(=O)CC23CCCC2C3)nc1.C12CCCN1C2=O 6791,c1(CCN(C)C)ccc(C(=O)NC2CCC(NC(C3(CO)CCCO3)=O)C2)cc1 6792,C(=O)(C1=CCCCC1C)N(CCNC(CCC(CC)O)=O)CC1CC1 6793,CCC(CC(=O)N1CCC(CF)(NC(=O)CCCCC2CC2)C1)OC 6794,N1(C(N(C)CC2CCC=CO2)=O)CC2CC1C1CC21 6795,c1(CNC(C2CCC2CF)=O)ccc(-n2ccnc2O)cc1.C12(CC1)N(C)C2=O 6796,c1(NC(N(C2CCC(C(N)=O)C2)C)=O)ccc2c(Br)cccc2c1 6797,c1(C(=O)NCc2cccc(C(N(CC(C)C)CC)=O)n2)cccc2ccoc12 6798,n1(CC(=O)NC2(CNC(=O)CC3CC4CC4C3)CCC2)ncc2ncccc12 6799,c1(OCCNC(COC(CC)(C)C)=O)ccc(Cl)cc1.c12cccc(c1)CNC2=O 6800,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(=O)CCc1cncc(O)c1)CC 6801,n1(CCC(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)c(C)cc(O)cc1=O 6802,CCCCCC(C)(C)CNC(=O)C(C)N(C(=O)C(F)CC1CCCCC1)C 6803,c1(N2CCCC(C(C)NC(CCC=C)=O)C2)cc(OC)nc(OC)n1 6804,C1(NC(c2nc(COCC)sc2)=O)C=CCN(c2nccc(CC)n2)C1 6805,N1(C(C2CC(CNC(C(C)OCC)=O)C2)=O)CCC2(CCCN2C)C1 6806,C1(CCNC(c2ccc(Cl)o2)=O)CCCN(C(c2cc(O)ncn2)=O)CC1 6807,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6808,c1(C(=O)NCC(C2CCC2)NC(C(C)NC(=O)OC)=O)ccc2c(c1)CCCS2 6809,N1(C(CN(CCC)C)=O)CC(NC(C2(O)CCSC2)=O)CC2(CC2)C1 6810,N1(C(C)C)C(=O)CCC1C(N1CC(NC(c2csc(F)c2)=O)C(F)C1)=O 6811,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C2CN(C(Cc3cccc(OC)c3Cl)=O)CC21 6812,c1(COC)ccc(S(=O)(=O)N2CCC(c3nc(-c4cccs4)cs3)CC2)c(F)c1 6813,C(CCN(C)C(C1(C(=O)OC)COC1)=O)(C(C)(C)C)NC(C(CCC)OC)=O 6814,N1(C(CN(C(=O)OC)C)=O)C2CCC1CC(C(C)NC(=O)CC1CCCOC1)C2 6815,N1(C(Cc2ccn(C)n2)=O)CCC(C(=O)O)CC1(C)C.C(C)(C)(C)OC(=O)N 6816,c1(C(N2CCCC(NC(CC3(C)CCCO3)=O)C2)=O)ccc2ncncc2c1 6817,c1(CC)nn(C)cc1C(=O)NCCCNC(c1cc(N2CCCCC2=O)no1)=O 6818,c1(C(=O)NCC2(CNC(CCC(=C)Cl)=O)CCC2)ccc(Cl)c(CC)c1 6819,C1(CC(=O)NC(C(=O)N(C)Cc2nc(CC)sc2)(C)C2CCC2)C=NN(C)C1=O 6820,N1(C(C2(C#N)CC=CC2)=O)CC(NC(C2CC(F)(CO)C2)=O)C(N=[N+]=[N-])C1 6821,CCC(CCO)NC(C1CC1CNC(=O)C(c1cnn(C)c1)=O)=O 6822,C1(NC(c2c(CC)onc2)=O)CCCN(Cc2cc(F)ccc2F)CC1 6823,N1(C(=O)OC(C)(C)C)CCOCC2(CC(C(N3CCCC3(C)C3CC3)=O)CO2)C1 6824,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6825,N1(C(CN2CCN(CC)CC2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO 6826,C(=O)(C1=CCN(C)C1)NC(C(C)C)C(N1CCCC2(C1)N=N2)=O 6827,C(=O)(CC(C)CC(C)(C)C)N1C2(C(=O)NC(CCCC)(C)CO)CC(C1)C2 6828,c1(C(=O)NCCc2cnn(-c3ccccc3)c2)nnc(C(C2CC2)NCCO)o1 6829,C1(C)(C(=O)OC)COCCN1C(=O)C(Cc1cn(C)nn1)OC1CCCC1 6830,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6831,Cc1ccc(C(=O)O)cc1NS(=O)(=O)Cc1cc(F)n(C)n1 6832,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2ccn(CCC)n2)=O)CCCC1 6833,CCCC(C(=O)N(C1CCC(n2cc(C(C)=O)nn2)CC1)C)c1ccccc1 6834,Cc1ccc(C(=O)NC2(CNC(c3ccsn3)=O)CCCC2)c(C2CC2)n1 6835,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6836,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1ccn(C2CCC2)n1)=O 6837,CC(CCCCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(=O)C=CC(=O)N(C)C 6838,N1(CC)CCC(CC(=O)OC(C2CC2C(=O)OCCN2CC3(COC3)C2)=O)CC1 6839,CC1CCCC1N=c1[nH]c(NC2CCc3c(Cl)cc(Cl)cc32)nc2c1CCCC2 6840,C1(C(=O)NC(C(=O)NC(CCSC)CO)CCOCCO)CN2CCN1CC2 6841,C(=O)(CCC(O)C(C)(C)C)N(CC(C)NC(=O)CC1(C)CC(F)(F)C1)C 6842,C1(C(=O)NC(C)CC2CCOCC2)CCN(C(=O)COC2CCCC2)O1 6843,c1(C(=O)NCCCN(C(=O)CON=C2CCCCCC2)C)nccn2ccnc12 6844,N1(C(c2c(NC)cccc2)=O)CCC2(CC(NC(=O)C(F)CC3CC3)C2)C1 6845,C1(C(=O)OC)(CC)CCCN(C(=O)C(Cc2c(C)nn(C)c2C)NC(=O)CCF)C1 6846,c1(C(=O)NC(CNC(C(C(=O)OC)C)=O)(C)CO)cccc2ncnn12 6847,C(C(=O)NCC1CCN(c2cccc(C(F)(F)F)n2)CC1C)(C(C)(C)C)OC 6848,CC1(C)C(CO)OCCN1C(=O)Nc1ncc(C(=O)OCc2ccccc2)[nH]1 6849,Cc1cc(=NCC2C3CCCC23)[nH]c(N(C)Cc2cccnc2O)n1 6850,C1C(F)C(=O)NC2CC12.C(CC(C)Cc1cn[nH]c1)NC(N1CC(COC)C1)=O 6851,C1(NC(C(C)n2ccnc2)=O)CN(C(=O)C=Cc2ccc(O)cc2)CC1(C)C 6852,C(CC(N)=O)(C(=O)NC(c1cnsc1)C)NC(Cc1nc(C)sc1)=O 6853,C1(CCC(=O)NCC2CCC(C(=O)OCC)C2)CC2CCC1C2.N12CCC1C2=O 6854,CC1COCC(CC(=O)NC2(CO)CCN(C(c3sccc3CO)=O)C2)O1 6855,N(C1CCC2(CC2)Oc2ccccc21)C(=O)NCCOCc1cccc(C)c1 6856,c1(CC)cc(Cl)ccc1C(=O)NC1CCN(C(C2CC(C(=O)OC)C2)=O)C1 6857,N1(C(c2cccc(-c3cccc(SC)c3)c2)C(=O)NCCC#N)CC(O)C(O)C1 6858,CC1(C)CC(CC(=O)NC2CN(C(=O)C(C)(C)C)CC2F)NC1=O 6859,N1(C(C)=O)CC(F)CC1C(=O)NCC1CCCC1NC(=O)CNC(N)=O 6860,C1(NC(C(C)(C)F)=O)CCCC12CCN(C(=O)C#CC1CCOCC1)C2 6861,Cc1nc(S(=O)(=O)Nc2ncc(-c3ccc(F)cc3)cn2)ccc1Br 6862,C(=O)(C1=CCCCCC1)NCC1(C(C)NC(C2CCCNC2=O)=O)CC1 6863,CCCCCC(O)CC(=O)NCC(O)CC(N1CC(=O)NCC1CC)=O 6864,C1(NC(C2N(C)CC(C)(C)C2)=O)CCC2CC1CN2C(=O)C1=CCOCC1 6865,C(CCCCCNC(=O)C(C1CCN(C(=O)C(CO)NC(N)=O)C1)F)N(C)C 6866,N1(C(C(=O)NCc2ccccc2CCc2ccccc2)=O)CCCC2(CCCO2)C1 6867,c1(OC)ccc(Cl)c(C(N2CCC(CF)(NC(c3sncc3C)=O)C2)=O)n1 6868,CC(C)(CCC(=O)N1CCC(NC(C2CCC(C)(C)CC2)=O)C12CCC2)[N+](=O)[O-] 6869,CC1(C)CCC(C(N2CCC(NC(=O)CSc3cccc(F)c3)C2)=O)OC1 6870,N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)Cc1nc(C)c(C)[nH]1)C2 6871,C1(NC(C2(C)CCCN(C)C2)=O)CCCCCN(C(c2cc(F)n[nH]2)=O)C1 6872,c1(C(=O)NCCN(C(C(CC)(C)OC)=O)C)cc(N)cc(C)c1F 6873,c1(CCC(=O)NC(C(C)NC(Cn2c(CCC)ncc2)=O)CO)c(C)nn(C)c1C 6874,N1(C(CC2(NC(C(C)N(CC)CC)=O)CC2)=O)Cc2c[nH]nc2C1 6875,C12(C(N3CCC3c3cccc(O)n3)=O)CC(CCO1)N(C(=O)C(F)C1CCCC1)C2 6876,c1(C(=O)NCC(C2CCCN(C(COC)=O)C2)(C)O)cccc2nsnc12 6877,C1(CNC(C(C)(F)F)=O)CC2CN(C(c3cncc(C(F)(F)F)n3)=O)CC12 6878,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6879,C1(NC(C2C(CC)CCO2)=O)CC(O)CN(C(=O)CCc2cc(Br)co2)C1 6880,C1(C2CC2)(NC(CCC(C)(C)F)=O)CCN(C(c2cc(Cl)ccc2Cl)=O)C1 6881,C1(CNC(c2n(C=C)nnc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6882,N1(C(C2C(C)SCCC2)=O)CCOC(C)C1C(N1CC2(CO)CC2(C(=O)O)C1)=O 6883,C(CC(=O)NOCC(C)C)(C(F)(F)F)NC(C(C1CCOCC1)OC)=O 6884,c1(NC(=O)Nc2c(C)cc(C(F)F)o2)ccccc1S(=O)(=O)C(C)C 6885,N1(C(CCCCCOC)=O)CCN(C(C2CC(C)CC(=O)N2)=O)C(C)C1C 6886,CC1CCN(C(=O)C(O)Cc2cn(CC3CCC3)nn2)C(C(C)CN(C)C)C1 6887,N1(Cc2ccc(CC)cc2)CCN(C(C2CCN(C)C2)=O)CC1c1cn[nH]c1 6888,CC1(C)CCC(NC(C2COC(CNC(=O)CC3CC4C=CC3CC4)C2)=O)CC1 6889,C1(NC(C2C(C)C2C2CC2)=O)CN(C(=O)CC2CC3(CCO2)CC3)C2(CCCC2)C1 6890,Cc1ccc(Br)cc1C(C)NC(Cn1ccnc1)C(C)C 6891,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6892,C(=O)(CN=c1cc[nH]cc1)NCCOCC(=O)NC(C)CCn1cncn1 6893,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6894,N1(c2n(CC=C)c(C(c3ccccc3)C)nn2)CCC2COCCC12 6895,C(=O)(CC1CCOc2ccccc21)NC(CCNC(CCC(=O)N(C)CC)=O)C 6896,c1(OC)cc(C(=O)NCC=CCNC(=O)C(c2cnccn2)C)n(C)n1 6897,CC1CN(C(C2CC3(CC(NC(C4C=CCC4)=O)C3)C2)=O)CC(C)(C)O1 6898,N1(C(CCCCOCCC=C)=O)CCN(C(=O)CCC(C)SC)CC1CC(F)(F)F 6899,C1(C(C)C)(C(=O)N(CC(=O)NC2(C)CCOC2)CC2CC2)CCCC1 6900,C(=O)(C(O)C(C(C)C)OC)N1CC(CC)C(NC(c2cnn[nH]2)=O)CC1 6901,C(C)(C(=O)N1CC(C(C(=O)NCC)OC)C1)SCCCC.C(COC)(CC)C1CC1 6902,C1(F)(C(=O)NCC2(CCNC(c3c[nH]nc3F)=O)CC2)CCOCC1 6903,CN1CC(O)CCC1C(=O)NCCN(C1CCCCC1)C(C1C=CC=CC=C1)=O 6904,Cc1cccc(C(=O)NC2(CF)CCN(C(=O)COCc3ccccc3Cl)C2)c1 6905,CN(C)S(=O)(=O)N1CCC(C(N2CC3CC(C2)C3N)=O)CC1 6906,N(C(=Nc1ccccc1)N1CCC(OC)C1)Cc1c(C#C)cccc1 6907,S(=O)(=O)(c1cccc(F)c1)NCCC(N1CCCC1Cc1ccc(Br)s1)=O 6908,CC1(C)CCN(C(C2CCC(F)CC2)=O)CC1CNC(c1c[nH]ccc1=O)=O 6909,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6910,N1(C(CN(C(C)C)C(C2CN(C(=O)N(C)C)C2)=O)=O)CCC(C(N)=O)C1 6911,N1(C(c2cc(C)sc2)=O)CC2(CCC2)CCC1CNC(=O)CC1COCC1O 6912,c1(OC)c(Cl)cc(NC(C2CC2NS(=O)(=O)c2cn[nH]c2)=O)cc1Cl 6913,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2C=CC=CC=C2)=O)C(CO)C1 6914,C(C)(CNC(=O)Cc1nccn1CC)(CC(C)C)NC(CSCCCCCC)=O 6915,Cc1nc(Cl)[nH]c(=NCC23CCC(NC(=O)C4=CCCS4)(CO2)C3)c1F 6916,c1(C(C(=O)N(CCNC(c2csc(S)n2)=O)CC)C)c(C)n[nH]c1C 6917,N1(C(C(C2CCN(C(c3ccnc(Br)c3)=O)CC2)C)=O)CCc2ncccc2C1 6918,C1(O)(CCNC(C(CC=C)C)=O)CCCN(C(c2cnc(C(C)C)o2)=O)C1 6919,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1CC(C#C)C1)COC 6920,CC(C)(C(=O)NC1CCCC1NC(=O)CCNC(=O)CO)C1CC1c1ccccc1 6921,c1(CN(C(=O)CC(O)C2CCC2)CC(C)C)ncc(F)cn1 6922,Cc1[nH]nc(C(N2CCC(N(C(=O)C(C)CCN(C)C)C)CC2)=O)c1[N+](=O)[O-] 6923,n1(C2(OC(C)C)CCC2)cc(C#CCNC(c2nccc3[nH]ccc23)=O)nn1 6924,N1(C(CN(C2CCC(=O)N2)C)=O)CCC(CNC(c2ccco2)=O)C1 6925,C1(COC(C2(C(=O)OCC)CCC2)=O)CCC(C)c2ccccc2C1 6926,CC1CC(F)(F)CN1C(C1CC2CCC1N2C(C1CCC(=O)N1)=O)=O 6927,CC(C)C(F)(F)CC(=O)NC(C)CCN(C)C(c1cn(CC(F)F)cn1)=O 6928,c1(OC)cc(C(N2CCN(C(=O)C(C)(C)C3CCCO3)C(C)C2)=O)c(F)cc1N 6929,C1(C(=O)NCC2(OC)CC2)CN(C)CCN1C(c1cc(C)n(C)c1C)=O 6930,C1(C(=O)NC2(CN(C)C(C3(N(C)C)CCC3)=O)CC2)CC(C)(CO)C1 6931,C1(NC(CCc2cn(C)nn2)=O)CC(F)(F)CC1NC(=O)C=Cc1cn(C)nn1 6932,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 6933,Cc1ccc(F)cc1CC(=O)NCC1CC(NC(c2cc(=O)n(C)o2)=O)C1 6934,O=C(CCCc1ccsc1)NCCN(C(c1cccs1)=O)Cc1nc[nH]n1 6935,N1(C(c2c(C)nns2)=O)CC(NC(c2occc2F)=O)CC(O)C1 6936,Cc1cc(C(=O)NC(C2CN(C(C)C(=O)NCCOC)C2)C)n(C(C)(C)C)n1 6937,c1(OC)c(C(=O)NC(C)CCCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6938,C1(NC(C(C)COCc2cccc(C)c2)=O)CCCN(C(=O)C(C)(F)F)CC1 6939,Cc1c(F)ccc(F)c1C(N1CCC(CC(N2C3CSCC2C3)=O)C1(C)C)=O 6940,N1(Cc2ccc(C(=O)OC)[nH]2)CCC(CO)(NC(c2cccc(=O)n2C)=O)CC1 6941,Cc1c(Cl)ccnc1NNC(=O)CN1CCCCC1c1ccc(F)cc1 6942,n1(CC)nc(C)cc1C(=O)NC1C=CCN(C(c2ncoc2C)=O)C1 6943,c1(CC)c(C(=O)NCC2CCN2C(c2cc(C(N)=O)ccn2)=O)nnn1CC 6944,C1(Cc2ncc(C(=O)NCCN3CCC4(CCC4)CC3)s2)CCC2(CCCC2)CC1 6945,n1(CC(=O)NCCNC(=O)CC2(CO)CCCO2)ccc(Br)n1 6946,c1(C(N2CC(NC(CCOC(C)=O)=O)C2)=O)cc(F)c(Br)cc1F 6947,N1(C(C(C)c2ncco2)=O)CCN(C)CC1C1(NC(=O)CC(=O)N(C)C)CC1 6948,C1(C(=O)NC(C2CCCC2)CC)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6949,c1(C(=O)NC2(CN(C(CC3C(C)C3)=O)C)CC2)c[nH]c2c(F)c(Cl)ccc2c1=O 6950,Cn1ccc2c(C(N3CCC4(C3)CN(C(c3ncccn3)=O)C4)=O)ncnc12 6951,C1(c2n3c4c(cccc4)c(n3)n2)CC(=O)NC1(C)C.c1nncn1C(F)(F)F 6952,c1(C2(C(=O)NCC(=O)N(C3CCCO3)C)CCC2)ccccc1 6953,C1(CNC(c2n(C(C)C)ncc2)=O)CCN(C(c2ccc(F)cc2O)=O)C1(C)C 6954,C(C(CC(=O)N1CCC(NC(=O)C2=CCCOC2)C(O)C1)C(F)(F)F)N(C)C 6955,C12CCC(CC1)C(=O)N2.C1(NC(CC(=O)N(CC)CC)=O)CC(=O)N(C)C1 6956,C1(C(N2CCC(CNC(CCn3c(C(C)C)ncc3)=O)C2)=O)COC2COCC12 6957,N1(C(c2nnc(CC)s2)=O)CC2(COC(CNC(=O)Cc3c(C)noc3C)C2)C1 6958,C(=O)(C(O)CCCNC(C1CCC(O)CN1C)=O)NCc1cc(C)ns1 6959,CCC(C)(C#N)C(=O)N(C1CCCN(C(c2nccnc2C)=O)C1)CC1CC1 6960,N1(C(C(CC(C)C)N(C)C)=O)CCCC(NC(c2cn[nH]c2)=O)CCC1 6961,c1(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCCC2CC2)ccc(Cl)nc1 6962,N(C(=NCC1(C)CCNC(=O)C1)N1CCN2C(CCS2(=O)=O)C1)C(COC)C 6963,C(C)(CNC(=O)Nc1ccc(Cc2ccccc2)o1)(CSC)OC 6964,C1(CCC#C)CCCN1C(=O)CCC1CCN(C(=O)CC2CCCSC2)C1 6965,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)N(C)C(c1ncc(F)cc1F)=O 6966,c1(OC)cc(CN2CCOC(C(=O)NCc3ccn(C)n3)C2)ccc1C 6967,CC1CC(NC(=O)C(F)=C2CCC2)CN1C(c1cccc(Cl)n1)=O 6968,Nc1cnccc1CNCC1CCNC1 6969,C1(CNC(C(C(CC)(C)C)O)=O)CCC2(CCC2)CN1C(=O)CN1CC(C)(OC)C1 6970,C1(NC(C(c2cncnc2)C)=O)CCN(CC(=O)Nc2ccncc2)CC(O)C1 6971,N1(C(C(COCC)C)=O)CCN(C(c2cc(OC)cnc2F)=O)CC1CC(F)F 6972,c1(-c2c(C(=O)Nc3ncc(-c4ccccc4)cn3)csc2)ccc2sccc2c1 6973,c1(SC)cc(C(=O)NCCCCC2(NC(=O)CN3CCOC3=O)CC2)n(C)n1 6974,CC1(C)CN(c2cc(C(=O)NCC3(CO)CC3)[nH]c(=N)n2)CC1c1ccccc1 6975,C(=O)(C(C1=NOCC1)N1CC(=O)NCC1)NC(CC)C.C(C)(C)(C)OC 6976,N1(C(C2CC3(CC(NC(=O)C4CC4)C3)C2)=O)CC2(CCC2)CC1CO 6977,Cc1cnoc1C(=O)NCC1(C(=O)N(C2CC2(C)C)C)CCCC1 6978,N1(C(COC(CC)(C)C)=O)CCC(C(=O)Nc2cnc(O)c(F)c2)C(O)C1 6979,C12(NC(=O)OC(C)(C)C)CCOC(CNc3ncccc3C3CC3)(C1)C2 6980,c1(C(=O)NCCC2CCN(C(c3cnns3)=O)C2)cc(F)c(Cl)cc1F 6981,c1(CCNC(=O)NCCc2ccc(N3CCN(C)CC3)cc2)c(F)cccc1F 6982,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 6983,C(CS(=O)(=O)CC(=O)NC1CCCN(C(c2cc(C)[nH]c2C)=O)C1)OC 6984,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(=O)C(C)(F)F)CC12CCC2 6985,c1(CC(=O)NC(C2N(C(CCCCSC)=O)CCC2)C)cccc(F)c1O 6986,C(CNC(C1C2COCC12)=O)(CC(F)(F)F)NC(c1c(SCC)nccn1)=O 6987,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 6988,CC(C)(C(=O)NCCNC(c1cn(-c2ccc(Cl)cc2)nn1)=O)C(F)(F)F 6989,N1(C(C(=Cc2cnc[nH]2)C)=O)CCOCC(F)(CNC(c2cc(C(N)=O)co2)=O)C1 6990,CCC(C)(C#N)C(=O)NC1(CCC(=O)NCCc2cnn(CC)c2)CCC1 6991,S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1CC2CC(CC(CNC(C(C)C)=O)C2)C1 6992,C1(C)(C(=O)N(CC(C(C)C)NC(c2cn(C)nc2O)=O)CCO)CC=CCC1 6993,C1(C(F)F)CCCN(c2cc(N3CCN(CC4CCC4)CC3)ncn2)C1 6994,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 6995,c1(OC(C(=O)NCCN(C(C(C)SCC(C)C)=O)C)C)ccccc1Cl 6996,C1(NC(C2CCCS2)=O)CCSC12CN(C(=O)CCc1nc3ncccn3n1)C2 6997,CC#CCCCC(=O)NCC1C=CCN1C(c1ccc(SC(F)F)cc1)=O 6998,c1(N(C)Cc2cccc(CC)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 6999,Cc1cc(=NCc2csc(C(C)C)n2)[nH]c(Sc2nn(C)cc2[N+](=O)[O-])n1 7000,n1(CC)cc(CC(=O)NC2(CC)CCOC2)cn1.C12CC(C1)CCNC2=O 7001,c1(CC(=O)N(C(C)C)CCN(C)C)ccc(F)c(F)c1.C12CCN(C1)C2 7002,Cc1onc(C(=O)NC2CC2CNC(=O)CSc2ccccc2)c1Br 7003,C1(CNC(C2CC(=C)C2)=O)COC(C)(C)CN1C(=O)Cn1cnnc1O 7004,C(=O)(CC(C)CC)NCCCN(C(c1cn(CC(CC)O)nn1)=O)CCO 7005,Cc1oc(C)c(C(=O)NC(c2cccc(O)c2)CNC(=O)C(F)C2CCCC2)c1C 7006,C1(C(=O)NCCC(=O)NC2CC(CO)(NC(C3CC3F)=O)C2)CCc2nc(O)[nH]c2C1 7007,c1(OCCC(=O)NC2(CNC(N)=O)CCC2)cccnc1.C12(CC1)C(=O)N2 7008,Cc1nn(CC(=O)Oc2ccc(CN)cc2)c(C)c1[N+](=O)[O-] 7009,C1(CCC)(NC(c2cc(C(C)(C)C)no2)=O)CCCN(C(C2CC23CCC3)=O)C1 7010,C1(CNC(C2NC(=O)OC2)=O)CN(C(=O)C=Cc2ccccn2)CCCO1 7011,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7012,C1(NC)CCCC2NCCC12.N12CCN(CC1)C1(CCC1)C2=O 7013,C1(CNC(C(c2n(C)ncc2)(F)F)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CCO1 7014,Cc1cnncc1C(=O)NCC(C)(C)CN(C(=O)COCC(=O)N(C)C)C 7015,N1(C(C=CC(C)C)=O)CCOC(C(C)NC(c2ccc(Cl)n2C)=O)C1 7016,c1(CNC(C(=O)NCCC(=O)OC)=O)nccc(CC#N)n1 7017,N1(CC)CC(C(=O)N(C)CC2CCCCN2C(=O)CCSC)CC1=O 7018,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7019,C1(C(N2CC(CCNC(CCC=C)=O)OCCC2)=O)CCc2nccn2C1 7020,N1(C(C2C(C(=O)OC)CC2)=O)CCC2C(CNC(C3CCSCC3)=O)C12 7021,C#Cc1ccc(C(=O)NCCCCC2CN(C(=O)C(O)Cc3ccccc3)C2)nc1 7022,C(CCC(CO)SC)NC(=O)CC(CC)c1ccc(-c2n(CC)ccn2)s1 7023,C1(C(N(CC(=O)N(C)CCN(C)C)C(C)C)=O)CCCSC1C 7024,CN1CCN(C(C2CCCC2)=O)C(c2ccccc2)C1.C1(C(=O)NC)C2CNC(=O)C12 7025,C(CCCC(=O)NCCCO)N(C)C.CC(C)(C)NC(=O)CCC1(C)CC1 7026,C1(NC(c2cnc(CC)s2)=O)CCN(C(=O)COCCCN(C)C)CC1F 7027,Cc1cc(C)c(C(N2CC3CC(C(=O)NC4(CC(N)=O)CC4)(C3)C2)=O)cn1 7028,C1(=CC(=O)NCCOC2CN(C(c3ccc(CSC)cc3)=O)C2)CCCCC1(C)C 7029,CCC(C)(CNC(C1CC1C(N)=O)=O)NC(=O)C(C)(C)c1cc[nH]n1 7030,c1(OC)cc(CC(N2CCN(CCNC(C3(O)CCCC3)=O)CC2)=O)ccc1C 7031,N1(C(C(C)OC)=O)CC2CN(C(c3ccc(C(C)(C)C)cc3)=O)CC12 7032,c1(C(=O)NC2CCCCN(C(c3cc(C)cc(O)n3)=O)C2)[nH]cc2c1CCCC2 7033,C1(C(=O)NCC2C(C(N3C(C#C)CCC3)=O)C2(C)C)CC2COCC2C1 7034,c1(C(=O)NCCCCN(C(C(CC)C)=O)C)cn2c(C)cccc2n1 7035,C(=O)(C(F)(F)C(F)(F)F)NCC(C)(C(C)C)NC(c1ccnc(C)c1F)=O 7036,c1(CC)[nH]c(=N)sc1C(=O)NC1CC(CCNC(c2cnc[nH]2)=O)C1 7037,N1(C(C23N(C(C4(C(N(C)C)=O)CC4)=O)CC(C2)C3)=O)CCCCCCC1C 7038,N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(c1ccsn1)=O 7039,c1(NC(COC(C)C)=O)cnc(OC(=O)N(CCCN(C)C)C)cn1 7040,O(NC(=O)C(C1=[SH]NSC1)NC(c1coc(C)c1)=O)CCCC#C 7041,C(C)(CO)(C(=O)N1CC(c2n[nH]c(C)n2)C1)OC.C12CCC1C(=O)NC2 7042,N1(C(c2nc(C(C)=O)sc2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7043,c1(NC(c2nccs2)C)nccc(N2CCC(N3CCOCC3=O)CC2)n1 7044,N1(C(C(C)=CC)=O)CCOC(CNC(=O)CCc2n[nH]c(=N)s2)C1 7045,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7046,C(CN=C(NCc1c(F)cccc1Br)NCC1CCN(C)C1=O)SC 7047,c1(NC(C2C(CNC(C3CC(C)(C)C3)=O)CCCC2)=O)cc2sccc2cn1 7048,N1(C(c2n(C)ncc2Cl)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(O)C1 7049,Cn1ccnc1C(=O)NCC(=O)NCC(C)(Cn1cccn1)NC(=O)CC(F)F 7050,N1(C(CCSCC)=O)CCCOC(CNC(=O)Cn2ccc(C)n2)C1 7051,Cc1c(C(=O)NC2(CO)CCN(C(=O)C(F)(F)c3ccccc3)C2)cnn1CO 7052,CCCC(C)C(=O)NC(C1CN(C(C23CC(CO2)C3)=O)C1)C 7053,c1(OC)cc(C(=O)NC2CCN(S(=O)(=O)c3cccnc3)CC2F)ccc1C#N 7054,CCC(C)(C)CCCC(=O)NC1CCCC1NC(c1c(C)ccc(F)c1O)=O 7055,c1(C(C(=O)N(CC(C)CNC(C2CC2C2CC2C)=O)C)C)noc2ccccc12 7056,N1(C(CCOC(C)(C)C)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7057,C1(C(=O)OC)CC(S(=O)(=O)N2CC(C(=O)OC(C)(C)C)CC2(C)C)C1 7058,S(=O)(=O)(c1ccn(C)n1)N(C)Cc1c(F)cccc1F 7059,C12(CC(C)(C)C1)C(=O)NC2.C1(CN(C(C(C)c2ccsc2)=O)C)CCCC2CC12 7060,C1(C(=O)NCCN(CC(F)(F)F)C)CC2CCC1O2.C1(=O)CC(=O)N1 7061,n1(CC)cnc(C(=O)NC2(CNC(=O)C(O)CSC)CCOC2)n1 7062,C(=O)(C(CCC1CCC1)OC(F)F)NCCOC1(C)CC(C)C1 7063,c1(C(N(C2CCN(C(C3CCCS3)=O)C2)CCC)=O)cnn2cccc(Cl)c12 7064,c1(CC(N2CCC(F)(CNC(C(CCC#C)O)=O)C2)=O)ccc([N+](=O)[O-])cc1F 7065,c1(SC)nccnc1C(N1CC(O)CC1CNC(=O)C(O)CN1CCCC1)=O 7066,C1(C)(C(=O)NC23CC(OC)(C2)C3)CCN(C(C2CCN(CCC)C2)=O)C1 7067,CC(C)CC(C)C(=O)N1CCC(N(C)C(C2CC3C=CC2CC3)=O)CC1 7068,C(=O)(CC(=O)NC(C)C(=O)NCC(c1cscn1)O)OC 7069,Cn1ccc2c(C(=O)NC3CCN(C(=O)CSC(F)F)C34CCC4)cccc12 7070,c1(C(=O)NC2CCC(CCNC(Cc3n[nH]c(=N)s3)=O)C2)cc2c(nn1)CCC2 7071,N1(C(C2CC2NCc2ccccc2-c2ccc(F)cc2)=O)CC2C(C1)C2(F)F 7072,N1(C(CN(C(C)=O)C)=O)CCC2(CC(NC(C34CC(CCO3)C4)=O)CO2)C1 7073,C(C1=NOC(C)C1)NC(CC1C(CNC(c2c(C)ocn2)=O)C1)=O 7074,CCCCCC(O)CC(=O)N(C1CCN(C(=O)CCC(F)(F)F)C1)CCO 7075,c1(C(C(=O)OC)N(C(=O)CSC)CC(=O)NC)cncn1C 7076,c1(C(N(CCCN(C(=O)CCc2cncn2C)C)CCO)=O)cc(N)cc(F)c1 7077,C1(OC(c2ccc(-c3ccccc3)o2)=O)CC2CC2C1 7078,c1(CC)cccc(C(N2CC(N(C(=O)C(F)C(F)(F)F)C)C3(CC3)C2)=O)c1N 7079,C1(NC(C(C)OCCC=C)=O)CCN(C(c2cc(OC)no2)=O)CC1F 7080,C1(C(N(c2c(C)cccc2)C)=O)CCN(C(=O)C(CC(N)=O)NC(N)=O)O1 7081,c1(CCC)ncc(C(=O)NC(CNc2ccc(SCC3CC3)s2)C2CC2)s1 7082,C1(C(=O)NCCN(C(C2N(CC)C(=O)CC2)=O)CC2CC2)CN(CP(C)(C)=O)C1 7083,C1(CCNC(C(C)Cc2cnn(C)c2)=O)CN(C(c2ccc(Cl)[nH]2)=O)CCO1 7084,C(c1ccco1)=C(C)C(=O)N1CCC1CC(=O)NCC(c1nccs1)C 7085,c1(C(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)cccn(C2CC2)c1=O 7086,C(=O)(CC(F)(F)F)NCC(CN(C(C(CC)N(c1nc(=N)[nH][nH]1)C)=O)C)O 7087,c1(CNC(C(C2CC(NC(C3(C)CC3(F)F)=O)C2)F)=O)ccccc1O 7088,N1(C(C2C(C)(Br)C2)=O)CC(F)CC1CNC(=O)C(c1ccc(Cl)cc1)(F)F 7089,Cc1nn(C)cc1C(=O)NC1(CCNC(c2ccccc2C(F)(F)F)=O)CCC1 7090,Cc1c(NC(C2C(NC(=O)C(O)C3CCCC3)CC2)=O)cc(C2CCCC2)n1C 7091,C(C(C)(C(=O)NC(C(=O)N1CCC(F)(CO)C1)C(C)O)OC)OC 7092,N1(C(C(c2cc(C(N(CCN(CCOC)C)C)=O)no2)=O)=O)CCCS1(=O)=O.OC 7093,C=CC(CC)CC(=O)NC1(C(=O)Nc2cnn(CC3CC3)c2)CC1(C)C 7094,C1(C(=O)NCC(C)Cc2cn[nH]c2)(CC)CCCN1C(=O)Cn1nc(C)nc1C 7095,c1(C(N2CCCC(O)(CCNC(=O)C3=COCC3)C2)=O)ccc2nnc(O)n2c1 7096,c1(OCC)ccc(Cl)nc1C(N1CC2C(C1)N2C(=O)COC)=O 7097,N1(C(C(C)OCC2CCCO2)=O)CC2CC1CN(C(c1nncs1)=O)C2 7098,c1(C(=O)NC2(C)CCN(C(CC(C)C3CC3)=O)C2)ccc2c(c1)CCCCC2=O 7099,c1(C(N(CC(CNC(CC(CC)O)=O)O)C)=O)cccc2cnnn12 7100,C1(C(=O)Nc2ccc(C)cc2)CCN(C(=O)C(c2ccccc2)F)C12CC2 7101,c1(C(CO)NC(=O)Cc2csc(C(N3CC4CC4C3)=O)n2)cccnc1F 7102,c1(CC)cccc(CC)c1CC(N1CCCC(c2ccccc2)(C)C1)=O.C1CC1 7103,C(CN=c1[nH]c(N(C)CCOCC2CC2)nc2ccsc12)(SC)SC 7104,c1(C(c2nnnn2CC2CC2)NC(C2CCOCC2)CC)ccc(F)nc1C 7105,CCCC(O)C(=O)N1CC(N(C)C(c2c[nH]nc2-c2ccc(Cl)cc2)=O)C(O)C1 7106,CCC(CC)(CO)C(=O)NCC(F)CNC(=O)C(C)n1cccc1 7107,C1(NC(C(=O)NCC2(OCCC)CCOC2)=O)CCCCC1CCC(C)C 7108,c1(C(=O)N(C(CCC)C(=O)N2CC(C)(N(C)C)C2)CC)ccc([N+](=O)[O-])o1 7109,CC(CN=c1[nH]cnc(Cl)c1F)NC(c1cn(-c2ccccc2)nn1)=O 7110,N1(C(c2ccn(CC)n2)C(=O)NC)CCCC2(CCCO2)C1 7111,N1(C(C2CCCC(NC(Cn3c(C)ncc3)=O)CC2)=O)CCC2CCN(C)CC12 7112,CCCCC(CN=c1ccc(C(C)=O)c[nH]1)NC(c1c(C(=O)OC)cno1)=O 7113,C12(C(=O)NCCCC(C)(C)C)CCC(CN(C(c3cc(=N)[nH][nH]3)=O)C1)C2 7114,N1(C(c2c(C)ncs2)=O)CCCC1(C)Cn1cc(Cn2cc(C(N)=O)nn2)nn1 7115,N1(C(c2nc(C)sc2)=O)CCCCC12CC(NC(c1coc(Br)n1)=O)C2 7116,c1(C(=O)OC)cc(F)c(Cl)c(NC(=O)N=c2[nH][nH]c(C)c2C)c1Cl 7117,C1(CNC(c2[nH]cc(C(N)=O)c2)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCOC2 7118,c1(C(N2CC(CNC(C(CSC)C)=O)C(F)(F)C2)=O)cc(C)c(Cl)c(C)c1 7119,c1(OCC)cccnc1C(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 7120,C#Cc1ccc(C(=O)NC2CC(CNC(C34CC(OC)C3C4)=O)C2)c(C(F)(F)F)c1 7121,c1(C(=O)NC(C(=O)N2C(CC(=O)NC)CC2)c2ccoc2)cnc(O)o1 7122,N1(C(c2ccc(C)s2)=O)CCCC(C)(CNC(C2(C)CCOC(C)C2)=O)C1 7123,Cn1ncc(C(=O)NCC2(C)CCCN2C(=O)CSc2n[nH]c(O)n2)c1C#N 7124,c1(CN(C)C(=O)OCCNC(c2ncccc2F)=O)ccc(OC(F)F)cc1 7125,CCCCC(CNC(c1c(C)noc1C)=O)NC(c1cc(C(C)(C)C)n[nH]1)=O 7126,c1(CCC(=O)NCC2C3CN(C(C(=C(C)C4CC4)F)=O)CC32)cccc(Cl)c1Cl 7127,N1(C(c2ncn(C)n2)C(=O)NCc2c(OC)cccc2)CCc2cc(Br)ccc21 7128,N1(C(COCC)=O)C2CCC1CC(CC(C)NC(c1c(F)cccc1Cl)=O)C2 7129,Cc1nn(CC(C)C)c(C)c1CC(=O)NC(C)CNC(c1cc(C(C)=O)cn1C)=O 7130,Nc1cccc(Cl)c1C(N1CCCC(N(C(=O)C#CC2CC2)CCF)C1)=O 7131,c1(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1N 7132,N1(C(C(C(C)C)C2CCCCC2)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C12CC2 7133,n1(CCC(N2CC(C(=O)OC)(C(N3CC(C(C)OC)C3)=O)C2)=O)cccnc1=O 7134,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1CC(OCC)C1)C 7135,C(C(C)N=c1[nH]c2c(c(=NCC=CCl)[nH]1)COC2)c1c(C)nn(C)c1C 7136,n1(CCC)c(N(CC(C)C)CC)nnc1C(c1ccc(F)cc1)O 7137,CCCCS(=O)(=O)N1CCCCC1C(=O)NC1CC1CNC(=O)CC1(C)CC1 7138,CCC(C)(CO)C(=O)N1CCC(C(C)NC(c2cccc(C3CC3(C)C)c2)=O)C1 7139,C1(COC)(NC(=O)CC(C)CF)CCN(C(=O)Cc2ccc(OC)cc2)C1 7140,c1(C(=O)NC(CC)(C)CNC(=O)C=Cc2cnns2)ccn2ncnc2c1 7141,C1(N(C(CC=CC)=O)C)CCCCN(C(=O)C(c2cccc(OC)c2)C)C1 7142,C1(C)(NC(C2N(CCC)CCC2)=O)CCC(NC(C2C3CCCCC23)=O)CC1 7143,CCCCC(C)(F)C(=O)NCC(CO)NC(C1CCC(CC)C1)=O 7144,C1(NC(=O)CSNc2ccccc2)CC12CCCC2 7145,n1(CC2CC(NC(CN(C)CC)=O)C2)cc(C2CCCO2)nn1 7146,c1(C(=O)NC(CCCC)CNC(=O)Cc2c(C)cnn2C)nnc(Cl)cc1N 7147,C1(NC(=O)Cn2cnnc2O)COCCC1NC(c1ccn(C(F)F)n1)=O 7148,c1(SC)ccc(C)c(C(=O)NCC2COCCN(C(=O)Cc3cc(C)ns3)C2)c1 7149,c1(C(=O)OC)ccnc(C(N2CC(OCCNC(=O)C(C)O)C2)=O)c1 7150,N1(C(C(C2CCC2)SC)=O)CCCC(C2(NC(c3cc(=O)n(C)cn3)=O)CC2)C1 7151,N1(C(=O)CSCc2cccs2)CCC(NC(c2cc(=O)cc(Cl)[nH]2)=O)C(CO)C1 7152,C(C(=O)N1CCC(C)(CCNC(=O)CC2(C)CC2)C1)(C(C)C)NC(COC)=O 7153,C(C(C)(CC)OC)N(C(C(C)N(C(=O)CCc1nccs1)CCC)=O)C 7154,c1(COC)cc(NNC(=O)NCCc2c(C)n[nH]c2C)ncn1 7155,C1(C(N2CCC(CCNC(c3n(C)cnn3)=O)CC2)=O)CCc2nc(O)[nH]c2C1 7156,C(=O)(C1CCN(C)c2ccccc21)N1CC(N(C(CC2C(C)C2)=O)C)C1 7157,c1(NC2CCCOC2)cn(CNC(=O)NCC2(C(N)=O)CC2)nn1 7158,c1(C(=O)NCC2N(C(c3ccc(CC)cn3)=O)CC=C2)c(Cl)ccnc1F 7159,N1(C(C2CN(C(C(C=C=C)C)=O)CC23CC3)=O)CCc2ccccc2C1 7160,CC1CC(CCN(C(c2ccc(Br)c(F)c2)C2CC2)C(=O)NC(C)(C)C)CC(C)N1 7161,CC1(C)COC(CC(=O)N(CCCNC(C2CCO2)=O)C2CC2)CO1 7162,c1(CNC(C2CC(CNC(=O)CN3CC=CC3)C2)=O)ncc(F)cn1 7163,Cc1cc(CC(=O)NCc2cc(C(=O)NCC(F)Br)cs2)on1 7164,c1(C(N(CC(C)NC(C2CCCN(CC)C2)=O)CC)=O)cc(C)nc(O)c1 7165,C1(c2nnnn2C)(Cc2c(CCC)cccc2)CCCN2CCSCC12 7166,C1(C(=O)NCCCN(C(C2C(=C)C2)=O)C2CC2)CCc2nc[nH]c2CC1 7167,C1(CNC(C(C)(C)O)=O)CN(C(C2CCN(C3COC3)C2)=O)CCCO1 7168,N1(C(CN(CCC)C)=O)CCC(NC(=O)C(c2cccnc2)OC)CC1 7169,c1(CC=C)ccccc1C(=O)NC12CC(C1)N(C(=O)C(F)C(C)C)C2 7170,N1(C(Cn2ccc(C)c2)=O)CCOC(C(=O)OC)CC1.N1(CC)CC(c2ccon2)C1 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7472,N1(C(CNS(CC)(=O)=O)=O)CCC(C2CC2NC(C2CC=CCC2)=O)CC1 7473,C1(C(=O)NC(CC)CN(C(=O)CCc2ccnc(Cl)c2)C)CN2CCCN1CC2 7474,C12(C(=O)NC(CNC(c3ccc(N)c(O)c3)=O)CO)CCCCC(=O)N1CCC2 7475,CCC(C)(CCNC(C1CC(=O)N(C)C1)=O)NC(=O)CSC 7476,C(N=c1[nH]c(=NC2CCC2C#N)[nH]c2c(F)cc(F)cc12)c1ncc(C)cc1Br 7477,N1(C(=O)NCc2ccc(C)cc2C(=O)O)CCC2CC(NC(C)(C)C)CCC2C1 7478,N1(C(c2c(Cl)sc(C)c2C)=O)CCC2(CC1)COC(CNC(c1cn[nH]c1)=O)C2 7479,C(CNC(C1CC12CCCC2)=O)(CC(=O)N1CCOC(CO)C1)OC 7480,C1(C(N(C2(C#C)CC2)C)=O)CCC(O)CN1C(=O)COC1CCCC1 7481,N1(C(C(=O)NCC(C)N(C)Cc2ccc(C3CC3)nn2)C)C(C)CCC1C 7482,C1(CNC(Cc2nc(C)[nH]n2)=O)C2CN(C(C3CSCCS3)=O)CC12 7483,N1(C(C=CC)=O)CC2(CCN(C(c3ccsn3)=O)CC2)CC1C 7484,C1(C(=O)NCC(C(=O)OC)OC)CCN(C(=O)CCOCC(F)F)C(C(C)C)C1 7485,c1(C(C)C)cc(CNC2CC(NC(c3ncc(F)cn3)=O)C2)ccc1F 7486,N1(C(C(C2CCCN(C(C(CC)(C)C)=O)C2)C)=O)CCC12CCCSC2 7487,Cc1cc(Cl)ccc1C1(NC(=O)NCC(C)(C)c2cn[nH]c2)CC1 7488,CCCCS(=O)(=O)CC(=O)NC(C1CCN(C(c2cc(C3CC3)n(C)n2)=O)C1)C 7489,C1(C(=O)NCCCN(C(=O)CC2=CCOCC2)CC)CCCCC12CC2(F)F 7490,C1(NC(c2c(SC)csc2)=O)CC2(C1)CC(NC(c1coc(C3CC3)n1)=O)C2 7491,O=C(CC1=CCCCC1)N1CC2CCCC1C2c1cn(-c2ccccc2[N+](=O)[O-])nn1 7492,Cc1ccc(NC(=O)CCC2CCC(NC(c3c[nH]c(C)c3)=O)C2)cc1CO 7493,C(Cc1cn[nH]c1)(C(=O)NC(CNC(=O)CCc1nncs1)CO)OC 7494,c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCN(C)CC3)=O)C2)cc(F)cc1F 7495,c1(CC(=O)NC(C2(O)CCN(C(c3c[nH]nc3F)=O)C2)C)c[nH]ccc1=O 7496,C(C1c2ccsc2CCN1C(=O)CCCc1ccc(I)cc1)OC 7497,C(=O)(C(CC(C)C)n1ccnc1)N1C(CN(C(C=CCC)=O)C)CCCC1 7498,N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 7499,N1(N(C)C(N2CCOCC2)=O)CCCN(C(c2ccccc2)C(=O)CCN)CC1 7500,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(C2CC3CCC2C3)=O)C1C 7501,N1(C(C(CC)(C)COC)=O)CC2CS(=O)(=O)CC2(CNC(c2nocc2C)=O)C1 7502,C1(C(=O)NCCCCCN(C(=O)CC(C)(F)F)CC)CCCC(F)C1 7503,c1(C(N(C)CC2OCCN(C(C(CCCC)C)=O)C2)=O)ccc2nnn(O)c2c1 7504,N1(C(c2nnc(CC)o2)=O)CCC(C(=O)NC(c2cn(C)nn2)(C)C)=C(F)C1 7505,C12(C(=O)NC3(CCNC(=O)C4=CSCCO4)CCC3)CCCC1CS(=O)(=O)C2 7506,C1(C(N(CC(CNC(c2cc(C)[nH]n2)=O)O)C)=O)CCCN1C(=O)OC(C)(C)C 7507,C1(NC(CCc2c(C)ncs2)=O)CC2C(NC(=O)COCCCF)C2C1 7508,N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 7509,c1(OCC(N2CCN(C(CCC)=O)CC2)=O)cnc(O)n(-c2ccccc2)c1=O 7510,C(CC(C(C)(C)C)NC(=O)CC1CC=CCC1)N(C)C(c1sccc1CO)=O 7511,C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCN(C(=O)C(C)Cn2ccnc2)C1 7512,N1(C(C(CC2CCOCC2)NC(C2CCC(OC)CC2)=O)=O)CC2C(C1)C2(F)F 7513,C1(C(N2CC(C)(CF)C2)=O)CC2CN(C(c3csnc3Cl)=O)CC2C1 7514,c1(Cc2n(CC)c(N3CCOC(CF)C3)nn2)ccc(Cl)cc1F 7515,N1(C(c2ccc(CC3CC3)o2)=O)CC(O)CC1C(=O)NCC1CCCNC1=O 7516,c1(C(=O)NCC2CCCC(CNC(C(C)N3CCC3)=O)C2)noc2c1CCCC2 7517,N1(C(C(C2CCCC2)SC)=O)CCCC(C)(C)C1CNC(C1(C(F)F)CCC1)=O 7518,N1(C(Cn2c(C)ccc2C)=O)CCOC(c2cn(Cc3ccn(C)n3)nn2)CC1 7519,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CC)C(NC(c2ccc(S(C)=O)cc2)=O)CC1 7520,C(C(=O)NC1CC1CNC(=O)COCC)(C(C)C)NC(=O)OCC 7521,N1(C(C(C(C)C)OCC)=O)CCC2(CCC(NC(=O)C3=C(Cl)CC3)CC2)CC1 7522,CCC(C(=O)NC1CC(C(=O)Nc2ccc(CO)c(F)c2)=CC1O)C(F)(F)F 7523,Cc1nn(C)c(NC2CC(C)CC(C)C2)c1C#N 7524,N1(C(c2ccc(COC)o2)=O)CC(CNC(=O)CSCCC(C)C)CC1(C)C 7525,N1(C(c2cc3sccc3s2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C(CO)C1 7526,CCC(C)(CS(=O)(=O)Nc1ccccc1)NC(C)CCc1ccc(O)cc1F 7527,c1(C(=O)NC(C2CN(C(CS(CC)(=O)=O)=O)C2)C)cnc2c(C)cnn2c1 7528,C1(C(N2CCC(C)C2)=O)(CNC(=O)C(C2CCC(=O)N2)C)CCOCC1 7529,C12(C(N3CC(C)N(C(=O)Cc4ccoc4)CC3)=O)CC3CC(C1)CC(O)(C3)C2 7530,C1(NC(CCSCC)=O)C=CC(C(N2CC(c3cnccn3)C2)=O)C1 7531,C1(NC(C(CC)n2ccnc2)=O)CC1C1CCCN(C(=O)C(C)(C)C(C)C)C1 7532,Cc1ccc2c(c1)CN(C(c1nc(F)ccc1F)C(=O)NCCC#N)CCO2 7533,N1(C(c2n(CC)nnc2)=O)CCCC1CNC(=O)C(C(C)C)Oc1cccc(Cl)c1 7534,CC1CCC(NC(c2cncn2C(C)C)=O)CN1C(=O)CCC(C)(C)F 7535,N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCc2ccc(O)nn2)C(C)(C)C1 7536,C1(C#N)(C(=O)NC(C)CCN(C)C(c2cc(C3(O)COC3)on2)=O)CCSCC1 7537,N1(C(Cn2ncn(C)c2=O)=O)CCC2CC1CN(C(=O)CCc1cc(Cl)no1)C2 7538,C1(COC(CCN(C2C(=O)NC2)CC)=O)CCN(CC)C1.OC 7539,c1(C(=O)OC)ccc(C(=O)CN2CC(CC(=O)O)C(O)C2)cc1 7540,c1(-n2cc(C(C)NC3C(c4c(C)noc4C)CCCC3)nn2)ccc(C#N)nc1 7541,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)COCCOC)C(C2CC2)C1 7542,c1(C(=O)NCCC(C)NC(C2CN(CCOC)C(=O)CC2)=O)ccsc1S(N)(=O)=O 7543,S(=O)(=O)(c1cnn2ccc(=NCC3CCSC3)[nH]c12)N1C2CC(CC)CC1CCC2 7544,C12(C(N(C(C)C)CCO)=O)CCCC1N(C(=O)CC1CCN(C)CC1)CCC2 7545,N1(C(c2c(C(C)C)c[nH]n2)=O)CC(NC(C2CC3(CCC3)C2)=O)C2(CCC2)C1 7546,c1(C(N2CC(CNC(=O)CC3CCCC3)OCCC2)=O)cc2c(Cl)cccn2n1 7547,C1(C(N2CC(OCCC(=O)N(CC(F)F)CCC)C2)=O)CCCC(CC)C1 7548,C1(CNC(=O)Cc2cccs2)CCN(C(C2CC3CC2C2CC32)=O)CCC1(F)F 7549,C1(CC(=O)NC(CCCCNC(c2ccc(C)cn2)=O)C)CC(C)CC(C)(C)C1 7550,n1(NC(C)(C)C)ncc2c1CCCC2NC(=O)NOCC(c1ccccc1)C=O 7551,C(=O)(C(C)S(C)(=O)=O)N(C(c1ccccc1)CNC(c1cc(C)ncn1)=O)C 7552,C1(S(C)(=O)=O)(C(=O)NC(C2CCCC2)CNC(c2[nH]cc(CC)c2)=O)CCCC1 7553,C12(CN(C(CCCSC)=O)C)CC(NC(=O)Cc3cn[nH]c3)(CO1)C2 7554,N1(C(C2C(C)C2)=O)CCCC(C2CN(C(=O)CN3CCN(C)C(=O)C3)C2)C1 7555,C(=O)(C#CC1(C)CC1)NC(C1CCN(C(c2cnn[nH]2)=O)C1)C(C)C 7556,C1(CC(=O)NC2CCC(N(C(CCCC)=O)CC)CC2)C(=O)N(C)N=C1C 7557,N(C(=NC1CCOCC1)NCC(C1CCC2(CC1)OCCO2)C)C(C)CC(F)(F)F 7558,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CC2)C1 7559,N1(C(c2c(-c3c(OC)c(F)ccc3)c(F)ccc2)=O)CCCc2sc(OC)nc21 7560,c1(NC(=O)CC2(OC)CCCC2)cccc(COC)c1.C12(CC=C)CN(C1)C2=O 7561,c1(CN2CCC(C(=O)NCc3c(C)cc(Br)cn3)C(O)C2)cc2ccncc2[nH]1 7562,CCC(C(=O)NC1CCN(C(c2cc[nH]c2)=O)C12CCC2)C(F)(F)F 7563,N1(C(C(CCC2CCC2)NC(c2c(C)ocn2)=O)=O)CCC2CN(C)CC2C1 7564,C(=O)(C(CNC(=O)CC(O)C1CCCC1)CC1CC1)N(CCCC)C 7565,C(=O)(C1=CCCN(C(=O)CC(F)(F)F)C1)NCC(COC)(F)F 7566,Cc1ccc(C(c2nnnn2C2CC2)NCC2CCCO2)cc1C 7567,CCN=c1[nH]c(CNC(=O)N(C2CC(O)C2(C)C)CC)cs1 7568,N1(C(C(N2CCNC2=O)C)=O)CC2C(C(=O)NCCc3cnn(C)c3)C2C1 7569,N1(C(C2CCC(C)(CC)O2)=O)CC2CC(NC(c3ccc(C)c(F)c3)=O)C2C1 7570,C(=O)(C(CC)CC(F)F)NC1(CN(C(c2cc(CC)c(F)cc2)=O)C)CC1 7571,Cc1cc(C(=O)NC2CC(N(C)C(C3CCC3)=O)C2)[nH]c1C 7572,C(Cn1cncn1)(C(=O)NOCC1CCCO1)NC(C(C(C)C)SC)=O 7573,c1(C(c2n(CC=C)nnn2)NC2CCCCC2CO)c(C)cccc1[N+](=O)[O-] 7574,n1(CC(=O)NCCN(CC(C)O)C(C2OCC2(C)C)=O)cnc(Br)n1 7575,CC1(C)CCC(CS(=O)(=O)NC(C(N2CC(C)C2)=O)=O)OC1 7576,N1(C(Cc2cncc(C)c2)=O)CCC2(CCC2)C(NC(C2CC2C2CCC2)=O)C1 7577,c1(NC)ncccc1C(=O)NCC1(F)CC(CNCc2cc(C(F)(F)F)n[nH]2)C1 7578,c1(C(=O)NCCn2cc(CC(C)(C)NS(C)(=O)=O)nn2)cc[nH]c(=N)n1 7579,CC1C(C)N(C(=O)CCOCC2CCCO2)CCN1C(C1C2CCC1CC2)=O 7580,c1(C(N2CCCC(C(C)NC(C3C(CCOC)C3)=O)C2)=O)cnc2cc[nH]c2c1 7581,C1(CNC(c2nnnn2CCCSC2CC2)C(C)C)CCC=CO1 7582,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7583,Cc1nc(N(C2CNCC2O)C(C2(CCF)CCOCC2)=O)c(Cl)cc1[N+](=O)[O-] 7584,C1(NC(COCCOC)=O)CCCN(C(=O)CCc2cnc(C)nc2O)CCC1 7585,CC1C(NC(=O)Cn2[nH]c(=O)[nH]c2=O)CCN1C(=O)CC1CC1C(F)(F)F 7586,C(C1CCOCC1)=CC(N1C(CC(=O)Nc2cnn(CCF)c2)CCCC1)=O 7587,CCCC(O)CCNC(=O)CCN(C(=O)CNC(C)=O)C1CCC1 7588,Cn1ccc(=O)c(C(N2CCC(O)(CC(=O)NCC3CC(F)(F)CO3)CC2)=O)c1 7589,c1(C2CC(NC(CSc3onc(C)n3)=O)C2)cccc(F)c1.n12cc(nn1)C2 7590,N1(C(C2CCCN(C)C2)C(=O)NC2CC(F)(F)C2)CCc2cccc(F)c2C1 7591,C1(C(C)C(=O)NCCn2cnnn2)CCCN(C(C2SCCS2)=O)C1 7592,c1(N(CC(C)NC(COCCCC)=O)C)cc2n(n1)CCCCC2=O 7593,c1(OC)cc(Br)cc(CN2CCCC(C(=O)Nc3ccsc3)CC2)c1O 7594,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7595,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7596,N1(C(c2ccc(CNC(c3nnn(C)c3N)=O)o2)=O)CCC2(CC1)CC2(F)F 7597,c1(C(N2CCCOC(c3ccccc3)C2)=O)cnc2c(Br)c[nH]c2c1 7598,c1(N2CCCC(C(C)(C)NC(CCSC)=O)C2)cc(-c2ccco2)nc(C)n1 7599,Cn1cnc(I)c1N1CCC(CNC(N2CCCCC2c2ncccn2)=O)CC1 7600,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(C)CC2CCCCC2)=O)C1C 7601,C1(NC(C(CC)C(C)O)=O)C(C)CCN(C(=O)CC2C(=O)ON=C2C)C1C 7602,c1(SC(N2C(CC(=O)NC3COCCO3)CC2)=O)cc(F)c(F)cc1Br 7603,C1(C(=O)NC(c2nn[nH]n2)CC)(NC(=O)CC2(C3CC4(CC4)C3)CC2)CCCC1 7604,C1(NC(Cc2cccc(OCC)c2)=O)CCSC12CN(C(=O)C(O)C(F)(F)F)C2 7605,c1(OC)ccc(F)c(C(=O)NCC(C)(C)NC(C2OCCC2C(C)C)=O)c1 7606,n1(CCOC(C)C)nc(-c2cc(Cl)ccn2)nc1-c1c[nH]c(=O)cn1 7607,c1(C(N(CCOC)CCNC(=O)Cc2cccs2)=O)cc(N)c(Cl)c(O)n1 7608,c1(C(=O)NCC2C3CN(C(c4snc(O)c4Cl)=O)CC23)cn2cccnc2n1 7609,C(CC(=O)NC(C1CC(NC(c2cnn[nH]2)=O)C1)C)OCCOC 7610,CC1(C)CCC(C(=O)NCC2CCCN2C(c2cc(O)cs2)=O)C1 7611,c1(OC)ccc(C(=O)N(CCCCN(C)C(C2(C)CC3C=CC2C3)=O)C)cc1N 7612,Cc1ccc(C(N2CC3CC2CC3NC(=O)Cn2ncnn2)=O)c(N=[N+]=[N-])c1 7613,c1(OC)cncc(C(=O)NCC(O)CN(C(=O)CC2CCC(=O)N2C)C)c1C 7614,Cc1ccc(C)c(C(=O)NCC2CCN(C(c3cn[nH]c3)=O)CC2C)n1 7615,CCCCCC(F)C(=O)N1CCCC(C)C1CNC(=O)C(F)(F)CC 7616,c1(N(CC=C)C)ccc(C(N2CC(CCNC(=O)C(F)C(C)C)C2)=O)cc1 7617,C1(NC(CCC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCO1)CCO2 7618,c1(C(N2CCC(F)(CNC(C(C3CCC3)OC)=O)C2)=O)sc([N+](=O)[O-])cc1Cl 7619,c1(C(N(c2ncccn2)CCC)=O)cc2nccnc2cc1C 7620,CC(C)CS(=O)(=O)CCC(=O)Nc1cccc(CC2COc3ccccc32)c1 7621,c1(CC(N2CC(NC(CCC(C)OC)=O)(CF)C2)=O)ccc(Cl)c(C)c1 7622,N(C1CCCc2c(Br)cccc21)C(c1n(CCCSC)nnn1)c1ccc(I)s1 7623,N1(C(C2CCC(NC(C3(COC)CCC3)=O)CC2)=O)CCC(O)C(C)(CO)C1.CO 7624,C1(CC)CCN(C(C)=O)C(C(=O)NCc2ccc(=N)[nH]n2)C1 7625,CCCCC(O)C(C)C(=O)N1CC(N(C(=O)COCCCC(C)C)C)C1 7626,C1(NC(c2c(CCC(=O)OC)cccc2)=O)CN(C(=O)CC2CC2)CCC1(C)C 7627,C(N=c1cc(N(C)Cc2csc(CO)n2)nc[nH]1)C1(OC)CCOCC1 7628,C1(=O)C(C)(C)CC(C)(C)C(N(C(CN(C)CCO)=O)C)CCCC(C)N1 7629,N1(C(=O)COc2ccc(Cl)nc2)CCC(O)(C(N2CCC(n3cccn3)CC2)=O)C1 7630,C(=O)(C1CCCc2nn[nH]c21)NCC(C1CCC1)NC(c1c(C#N)ccs1)=O 7631,N1(C(=O)OCC)CC2CCC(C1)N2C(=O)Nc1ncsc1C(F)(F)F 7632,N1(C(c2ccc(C#C)cc2)=O)CCCC2CN(C(=O)C(n3ccnc3C)C)CC12 7633,N1(C(C(CNC(C(CC)(CC)OC)=O)C(C)C)=O)C2CCC1CC(=O)NC2 7634,c1(N2CCC=C(C(=O)OC)C2)ncnc2c1ncn2C(C1CCCC1OC)CO 7635,N1(C(C(c2c(CC)cccc2)(F)F)=O)CC(NC(=O)C=CCF)CC(O)C1 7636,C=CCCCC(=O)NCC12CC(CN1C(=O)CCc1cnn(C)c1C)C2 7637,Cc1cc2[nH]c(C(N3CCN(C(=O)COC4COC4)CCC3C)=O)cc2s1 7638,Cc1c(C(N2C3CCC2CN(C(=O)CS(C)(=O)=O)C3)=O)sc2ccnc(O)c12 7639,CCC(Cc1nc2ccccc2s1)(CC)C(=O)NC(c1cccc(F)c1)C 7640,c1(C(=O)NCC(C2CCC2)NC(C2CC2(F)F)=O)ncccc1Br 7641,C1(NC(C2CC23CCC3)=O)COCCC1NC(C1CCS(=O)CC1)=O 7642,N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(c2ccc(O)nn2)=O)C2CC12 7643,C(C1=CCN(C(=O)CC2CCOCC2)CC1)=CC(N1CCC(C(N)=O)C1)=O 7644,Cc1cc(F)sc1C(=O)NC(C(=O)NCC(O)CCC1CC1)C1CCCC1 7645,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cc(O)c2cnn(C)c2c1 7646,N1(C(C(C)NC(COC)=O)=O)CCCCC1C(N1CC2CC2(CO)C1)=O 7647,CCC(CC(=O)NCC1CCCCCN1C(c1c(COC)nccc1)=O)C(C)C 7648,c1(OC)ccccc1CC(C)(C)C(=O)N(CC(O)CNC(=O)C(C)C1CC1)C 7649,C(=O)(CC(CC#C)C1CC1)N1CCCC(N(C(=O)CC2(N(C)C)CC2)CC#C)C1 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7740,c1(C(C)=O)cc(C)ccc1NC(N1CC(CO)OC(C(F)(F)F)C1)=O 7741,C1(F)(C(N(CCNC(CCNC(=O)OCC)=O)CC2CC2)=O)CCCCC1 7742,N1(C(CCOCCC)=O)CCN(C(=O)C(C(C)(F)F)c2ccccc2)C(CC)C1 7743,NC(=O)CCCC(=O)NCC1CCCCN1C(=O)CCNC(=O)Cc1ccoc1 7744,N1(C(COC2N(CC(=O)OC3CC34CC4)CC2)=O)CCc2sccc2C1 7745,C1(NC(C(CC)N2CCCC2=O)=O)COC2(CCN(C(=O)Cc3csnn3)C2)C1 7746,c1(C(N2CC(O)(C(C)NC(CC(=C)C)=O)C2)=O)cc(C)c(F)c(S(C)(=O)=O)c1 7747,c1(C(=O)NCC2(O)CCN(C(C(C)C#N)=O)C2)c(C2CC2)nc2sccn12 7748,Cc1nccnc1C(=O)NCC(C(C)C)NC(=O)C(c1ccccc1)=O 7749,C(C(C)(C)CCCNC(=O)C(C)NC(=O)C1CC1)OCCOCC 7750,c1(CN(C)C(c2ccc(-c3ccc(SC(F)F)cc3F)o2)=O)ccc(F)c(F)c1 7751,N1(C(C2(COC)CCC2)=O)CC(CNC(=O)C(C)Cc2cnn(C)c2)C(C)C1 7752,Cc1cc(C)c(NC(C2CCC(NC(c3cccc(I)c3C)=O)C2)=O)c(C)c1 7753,C(=O)(CCCCCCS(N)(=O)=O)NC1C2(CN(C(C(CC#C)C)=O)C2)CC1 7754,C1(C(=O)NCCCOCC=C)(NC(=O)C(C)CC2CCC2)CCN(C)C1 7755,c1(C(=O)NC2CCC(CNC(c3n(CC)nnc3C)=O)C2)cc(OC)ccc1Cl 7756,c1(C(=O)OC)sc(NC(c2cc(NC(C34CCN(CC3)C4)=O)cs2)=O)nc1C 7757,C1(CC=C)(C(=O)N(CC)Cc2nccs2)CCCN1C(=O)CC1CC2(CCC2)C1 7758,N1(C(C(COC)N(C)C)=O)CCCN(C(C2CN3CCN2C(C)C3)=O)CC1C 7759,N1(C(c2cc(C)sc2)=O)CCOC(C(C)NC(=O)Cc2cnn(C)c2C)C1 7760,N(C(=NCC(C)(C)C(F)(F)F)N1CCN(C(c2cccc(F)c2)C)CC1)C(C)C 7761,C(C(=O)NC1CC(CCC2COC(C)(C)O2)C1)(C(C)C)c1cn(C(C)C)nn1 7762,c1(C(C)=O)cc(S(=O)(=O)N2CCCC3C(Br)C23)c(F)cc1C 7763,N1(C(C2C3CCN(C(CC(CC(C)C)O)=O)CC32)=O)CCC2CCN(C)CC12 7764,CCC(CC(C)C)C(=O)NCC1(NC(c2cnc(SC)s2)=O)CCOC1 7765,c1(COC(C(C)CCNc2ccccc2)=O)nnc2n1CCNC2=O 7766,c1(C(C)=O)cc(C(N2CCCC(C)(CNC(=O)C(O)C(C)C)C2)=O)ccc1C 7767,N12CCCN(CC1C)C(=O)C1(CC1)CC2=O.c1(OC)cc(C(C)(F)F)on1 7768,c1(C(=O)NC2C(NC(C(C)(C)n3cccn3)=O)CCC2)cc2ccccn2c1 7769,C(C(CC(C)C)C(=O)N(CCC(=O)N(C)CCN1CCCCC1)C)OC 7770,C1(NC(c2ccc(C(C)C)cn2)=O)CN(C(c2cnc(S)[nH]2)=O)CCC1F 7771,Cc1nc2c(o1)CCN(C(=O)CC(C(C)(C)C)NC(=O)C=Cc1cn(C)nn1)C2 7772,c1(COC)ncn2cc(C(N3CCC4CNC(=O)NC4C3)=O)ccc12 7773,N1(C(c2c(CC)nns2)=O)CC(Nc2ncc3c(n2)CCCC3)CC2(CCC2)C1 7774,C1(C(=O)N=c2[nH]nc(-c3cccnc3)s2)CC2CCNCC(C1)C2 7775,N1(Cc2n(C)ncc2I)CCN(C(=N)NCC(F)F)CC1 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7794,N12CC(C1)C2=O.C1(=O)C(C2CC2)NCCN1C.C1(C(=O)NC)(C(N)=O)CC1 7795,c1(NC(C(C(=O)OC)C)=O)ccc(C)c(CO)c1.C12CCN(C1)C2=O 7796,N1(C(C(C)OC)=O)CC(O)CC1CNC(C1CCC(=O)N1C(C)C)=O 7797,C1(CC)CCOC1C(=O)NCCCC(=O)NCC1(C)CCCO1 7798,C1(CC(=O)NC2(CO)CN(C(c3ccc(C4CC4)o3)=O)C2)CCOCC1 7799,N1(C(C=C(CCN(C)C)Cl)=O)CCC(C2CC2)C1CNC(c1snnc1C)=O 7800,N1(C(=O)CC2CC2)CCC2CCCN(C(c3ccccc3C3CCC3)=O)C2C1 7801,C(CNC(=O)C=Cc1cnn(C)c1)(CC(=O)N1CCCCCO1)OC 7802,N1(C(C(=O)N(C)C)=O)CC2C3CCC(C2C1)N(C(=O)CC(C)(O)C(F)(F)F)C3 7803,C(=O)(CCC(F)(F)C(F)F)NCC1CC(NC(CCC2CCCC(=O)N2)=O)C1 7804,C#CCC(CC(=O)OC)NC(c1ccc(CNC(=O)C=C(C)CSC)s1)=O 7805,N1(C(C(C)CN(C)C)=O)C2CCC1CN(C(=O)CCNS(C)(=O)=O)C2 7806,c1(OC)cc2c(cc1C(c1nnnn1C(C)C)NC(C)C(C)C)OC(F)(F)O2 7807,C1(N)(C(=O)OC)CCS(=O)(=NC(=O)Cn2cc(-c3cccc(Br)c3)cn2)CC1 7808,N1(C(C2CCC23CCOCC3)=O)CCCC2(CC(NC(C3(O)CC3)=O)C2)C1 7809,C(CC(C(=O)N1CC(CO)C(O)C1)NC(c1ncc(F)cn1)=O)SC 7810,C1(CN(C(=O)CN2CCCCC2=O)CC)CCN(C(C23CCC2C3)=O)CC1 7811,CC1CCCCC1(CNC(C1CC(N=[N+]=[N-])C1)=O)NC(C1(CO)CCC1)=O 7812,C=CC(C)(CC)C(=O)N1CC(C)(NC(=O)C(CC(=C)C)OC)C1 7813,Cc1c[nH]nc1C1(C(=O)N(C2CC(NC(=O)Cn3ccc(C(N)=O)n3)C2)C)CC1 7814,N1(C(CCCc2n(C)cnn2)=O)CCCC(C(C)(O)CNC(=O)COC2CC2)C1 7815,C1(NC(C=CC)=O)CC2CC(NC(C34CC(C3)C4)=O)C1C2 7816,Cc1cc(Cl)ncc1C(=O)NCCNC(C12CC(NC(=O)OC(C)(C)C)(C1)C2)=O 7817,CCC1=NOC(C(=O)NC(C)CNC(=O)CCCN(CCC)C(C)C)C1C 7818,Cc1nc(C)n(CC(=O)NC(CN(C)C)C(=O)NCCCN=[N+]=[N-])n1 7819,c1(C(N2CCC(CC(C)NC(C3(C=C)CC3)=O)CC2)=O)ccc(F)c(Cl)c1N 7820,C1(NC(c2ccoc2)=O)CN(C(=O)CCn2ccnc2)C2CCCCC12 7821,C(c1ncc[nH]1)=CC(N1CCC(OCCNC(=O)CC2(O)CCCC2)C1)=O 7822,C1(c2ccccc2)(C(=O)OCC)C(COC)CC1NC(N1CCN(OC)CC1)=O 7823,c1(C(=O)NC(CCC=C)C(=O)N2C(CC)CCC2C)cccn2nccc12 7824,N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CC(F)(F)C(F)F)CC12CCC2 7825,C1(C(N(C(CC(=C)Br)=O)C)C)CCN(C(C2CCCC(OC)C2)=O)CC1 7826,c1(NC(=O)NCC2C(C)(C)COC2)cc(F)cc2ncoc12 7827,Cn1c(O)nc2cc(C(c3nnnn3CC3CC3)NC(C)(C)CCO)ccc12 7828,c1(CC)ccsc1C(=O)NCC(C1CC1)N(C(=O)CCc1cn(C)cn1)C 7829,N1(C(c2cc(SC)oc2)=O)C2CCCC1CN(C(C1CCCCN1C)=O)C2 7830,n1(C(CC)CC)nccc1C(=O)N(CC(C)(C)NC(=O)C(CO)N(C)C)C 7831,c1(C(=O)NCCC2N(C(C3N(C)C(=O)OC3)=O)CCCC2)n[nH]c2c1CCC2 7832,C1(CC(=O)N(CC(C)N(C)C(c2cc3sccc3s2)=O)C)CCC(C)(C)CO1 7833,c1(CC)cccc(C(=O)NC2CN(C(C3CCCC3CC)=O)CC2O)n1 7834,c1(NC(=NCC#C)NCC2(F)CC2)sc2ncn(C)c(=O)c2c1C 7835,C=CCC(C)C(=O)NCC(CCCC)NC(=O)C(C)NC(C1CCCCC1)=O 7836,Cc1c(F)ccc(C(=O)NC23CC2CN(C(c2ccc(C(F)(F)F)[nH]2)=O)C3)c1Cl 7837,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7838,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(c3ccsc3)=O)C4)cc2o1 7839,N1(C(c2cccc(OC)n2)=O)C2CCC1C(NC(C1CC3CN(C)CC13)=O)C2 7840,C(CCN=c1ccc(NC(Cc2cccc(Br)c2)CO)c[nH]1)OC 7841,Cc1nc(N2CCC(F)C(NC(C3CC4CC4C3)=O)C2)c(C)c(C)n1 7842,N1(C(c2ccc(CNC(c3c(C)n(C)cn3)=O)cc2)=O)CC(C)OCC(C)(C)C1 7843,c1(C(N2CC(F)(CNC(C=C(CCC)C)=O)C2)=O)ncncc1Cl 7844,C1(C(C)(CNCCCOCCO)OC)CCOCC1 7845,CC(CN(C)C)CCC(=O)N1CC(CNC(c2cccs2)=O)CC1(C)C 7846,N1(C(CC2C(C)CCN(C(CCC=CC(C)C)=O)C2)=O)CC(C)(CO)CC1(C)C 7847,C1(NC(c2cccc(F)c2)=O)CN(Cc2ccc(OCC(O)CO)cc2)CC12CC2 7848,N1(C(C(COC(C)C)NC(C)=O)=O)CC2CCC1CN2c1ccnc(CO)n1 7849,C1(NC(c2cc(OCC)ncc2)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1C 7850,C(=O)(C(C)CC(F)F)NCC(CC=C)NC(c1ccnc(OC(C)CC)c1)=O 7851,Cn1c(C(N2CC(O)(C(F)C(=O)NC3CC(=O)N(O)C3)C2)=O)ccc1C#N 7852,CC1CCCC1C(N1CC(CCCCNC(=O)CNC(c2ccsc2)=O)C1)=O 7853,c1(C(=O)OCC)ccc2cc(C(C(=O)NCC(C)C)N(C)C3CC3)ccc2n1 7854,C1(OC)CCC12CC(C(=O)NC13CC(NC(=O)CC4CCOC4)(C1)C3)C2 7855,C(c1ccc(F)cc1)=CCN(C(CC(C)C)CO)CC1CC1CN=[N+]=[N-] 7856,C(=O)(C(C)S(N)(=O)=O)N1C(C(N2CC(CO)C2)=O)(COC)C=CC1 7857,N(C(=NCCC(=C)C)NC1CCN(c2ncccc2F)CC1)C(C=C)COC 7858,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7859,c1(C(N2CC(C)C(CNC(=O)Cc3ccno3)C2)=O)ccc2c(O)ncnc2c1 7860,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7861,c1(CNC(=O)CSC2CC2)nc(CNC(C2CCC3(C2)N=N3)=O)cc(O)n1 7862,c1(CC)cnc(C(=O)NC(C)CC(C)C)nc1.C12CCC(C1)CCC(=O)N2C 7863,Cc1cc(=NC(=O)C(=O)NC2CCCN(C(c3cscc3N(C)C)=O)CC2)[nH]o1 7864,C=CCS(=O)(=O)CCn1nc(C(C)CC)nc1-c1ccc(OC(C)(C)C)cc1 7865,C1(NC(C2CC(C)(F)C2)=O)CC2CCCC(C1)N2C(=O)C#CC1CCCO1 7866,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)NCC1CC2CCC(C1)O2 7867,N1(Cc2cc(-c3ccc(OC)c(F)c3)ncc2)Cc2ccc(O)cc2C1 7868,C1(C(C)NC(C2C(CC)CCO2)=O)CN(C(c2c(Cl)cnn2CC)=O)CCO1 7869,c1(N2CCN(C(=O)NC(N(C3CC(=O)NC3)C)=O)CC2)ccccc1[N+](=O)[O-] 7870,N1(C(c2cnc(CCCC)s2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7871,c1(C(=O)NCCN(C(CC(C)SC)=O)CC(C)O)cc(F)c(F)c(N)c1Cl 7872,c1(SCC(=O)NC(CO)CCCCNC(C2COCCO2)=O)nc2ccccc2o1 7873,N1(CC)CC(NC(=O)C(C(C)(C)C)NC(c2nc(C)oc2C)=O)CCC1=O 7874,C12CCC(CC1)NC(=O)n1cc(nn1)C(=O)NC2.C1(N)CC12CCC2.C(F)F 7875,C(=O)(C(CCC1CC1)ONC(c1cccn1SCC)=O)NCC1CC(=C)C1 7876,N1(C(c2c(C)[nH]nc2-c2cccs2)=O)CC(=O)NC(C)C1 7877,N1(C(COCC#C)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7878,N1(C(=O)COC2CCCCC2)CC(COc2cn(-c3nccs3)nn2)C2(CC2)C1 7879,C(=O)(C(CC(C)C)NC(=O)C(C#N)CC1CC1)NCCCC(=C)Cl 7880,c1(NC(=O)CC2CS(=O)(=O)CCO2)nc(F)c(Br)cc1F 7881,C1(O)(C(N2CCCC(CNC(=O)CC3CC4CC4C3)C2)=O)CCCCCC1 7882,C1(N(C(c2ccc(CC)s2)=O)C)CCCC2CN(C(=O)C=Cc3cc[nH]c3)CC12 7883,c1(C(=O)NC(CCCNC(CCOC)=O)C)csc(C)c1C 7884,c1(CC)ccc(F)cc1C(=O)NCC(C)(CO)NC(c1cc(F)ccc1O)=O 7885,N1(C(C(C)SCC)=O)CCN(C(=O)CCOC(C)=O)CC1CC(F)F 7886,C12(C(N3CC(CNC(C(C)OCCN(C)C)=O)C(C)C3)=O)CCC(C1)C(C)(C)O2 7887,c1(C(N2C(CN(C(CCCOC)=O)C)CCC2)=O)ccc2nc(O)[nH]c2n1 7888,N1(C(C(c2cn(CC)nc2)(F)F)=O)CC=CC(NC(c2cnc(Cl)s2)=O)C1 7889,C(CC(C(C)(C)C)NC(C1CCCN1C1CCCCC1)=O)N(C(C1C(C)C1)=O)C 7890,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7891,N1(C(CNC(C(C)(C)C)=O)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(O)CCCOC2)C1 7892,C1(SC)COCC1n1cc(CC2CN(C(C3CC(O)C3)=O)C2)nn1 7893,C1(NC(CN(CCC#C)C)=O)C2CN(C(c3cc[nH]c3C3CCCC3)=O)CC12 7894,c1(C(N2CCC(C)C(NC(C3CC(C)(C)C3)=O)C2)=O)nc(O)nc(O)c1N 7895,Cc1cc(C(N2CCC(NC(=O)CC(C)C)CC2)=O)c(Br)cc1F 7896,CCC(C)C(O)CC(=O)NC(CN(C(=O)C=C(C)C)C)CC 7897,C1(NC2C(COC)C2)CCC(NC(c2ccc(C)o2)=O)C1 7898,c1(OC)ccc2cc(C(N3CCC(NC(=O)Cc4cnc(C)o4)C3C)=O)[nH]c2c1 7899,C=CC(O)C(=O)N1CCC(C2CCCN2C(=O)CCc2cnccn2)C1 7900,N1(CC)CC(C(=O)NCCNC(=O)CC2CCCO2)CCC1=O 7901,N1(C(C(C(C)C)F)=O)CCC12CN(C(C1(c3ccc(O)cc3)CCC1)=O)C2 7902,C1(C)(CNC(c2nc(NC(C)=O)oc2)=O)CCCN1C(c1cnn(C)c1C)=O 7903,NC1CN(c2nc(=N)nc(N3CCOC(C4CC4)C3)[nH]2)C2(CCOCC2)C1 7904,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1C(CNC(c2cc(C)c(Cl)cn2)=O)C1 7905,C(=O)(C1=CC(C)(C)C1)N(C)CC1CCN(C(c2cnc(C)nc2)=O)C1 7906,C(=O)(C(C)(C)C(=O)NCCNC(c1cn(C2CCCCCC2)nc1C)=O)NC 7907,CC1(C)CCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1C(=O)NCC12CCCC1C2 7908,c1(CNC(c2ccc(C)[nH]2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7909,C1(O)(CNC(C2C(c3n(C)ncc3)C2)=O)CCN(C(c2ccc(F)s2)=O)C1 7910,C(C1=CCN(C(c2cc(-c3ccccn3)no2)=O)CC1)NC(C(C=CC)O)=O 7911,C1(C(=O)NCC(C)C(F)(F)F)C2CC3C(C2NC(c2cc(O)nc(O)c2)=O)C13 7912,C(=O)(C1=CC2CCCC12)NCCC1CN(C(=O)CCc2ccco2)C1 7913,CC(CC(N)=O)C(=O)NCCCCCN(C)C(C1(C(F)(F)F)CC=CCO1)=O 7914,c1(C(=O)NC2CC3CC(NC(=O)Cn4cccn4)C3C2)ccn2nncc2c1 7915,N1(C(C(C)Cn2cccn2)=O)CC2OCC(NC(=O)NCCCCl)C2C1 7916,c1(C(N2C3CCC2CC(C(N2CCC(CO)C2)=O)C3)=O)c(F)cc(Cl)cc1Cl 7917,N(C(=NCc1cnsc1)Nc1ccccc1-c1ccc(F)cc1)C(c1ncccn1)C 7918,C=C(Br)CCC(=O)NCC(CC=C)NC(=O)C(COC)N(C)C 7919,C(N=c1ccnc(C2CCCC2)[nH]1)C1(NC(C2CC(S(N)(=O)=O)C2)=O)CCCC1 7920,c1(C(N2C3CC(NC(=O)C=C4CCCC4)(C3)C2)=O)ccc2nc(O)nc(O)c2c1 7921,c1(OCCC(=O)NCCC2(OC)CN(C(C3CCO3)=O)C2)c(C)nn(C)c1C 7922,c1(-c2c(C(N(CCC(C)NC(C3CC3(C)C)=O)C)=O)c[nH]n2)ccccc1Br 7923,C(=O)(CCCCC(F)(F)F)N(C1CC(N(C)C(c2cnc(O)c(F)c2)=O)C1)CC(N)=O 7924,c1(NS(COC)(=O)=O)cnsc1C.C1CCCO1 7925,N#Cc1ccc(Cl)nc1NC(C1C2CN(C(C3CC3(F)F)=O)CC12)=O 7926,C=Cc1ccc(C(=O)NCC2C(CNC(c3cc(SC)nc(Cl)c3)=O)C2)cc1 7927,S(=O)(=O)(c1cccnc1NCC1CC(C)OC(C)C1)NCCS(CCC)(=O)=O 7928,c1(N(CC(C)O)CCNC(C2CNC(=O)N2C)=O)ncnc2c1ncn2C 7929,c1(C(=O)NC(C(C)NC(c2cc(C)c(C)o2)=O)C(C)C)nc2ncc(C)cn2n1 7930,C(=O)(C1CCCn2ccnc21)NC(CC)(CC)CCNC(=O)C(C(C)C)C1CC1 7931,N1(C(=O)CCNS(=O)(=O)CC2CC2)CC2CCN(C(c3cnc[nH]3)=O)CCC2C1 7932,N1(C(C(C)OCCCC)=O)CCCCC1CNC(=O)CSC1CC=C(C)CC1 7933,Cc1ccc(Cl)c(OCC(=O)NC2CC(C)N(C(c3cnnc(O)c3)=O)C2)c1N 7934,N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(c3ocnc3C(F)(F)F)=O)C2C1 7935,N1(CC(=O)N(C)CCN(CCO)C(c2ccc(Cl)s2)=O)CCc2ccccc21 7936,C(=O)(C(CO)NC(c1cn(C)cn1)=O)NCC(C)NC(=O)OC 7937,c1(C(=O)NC2CCN(C(C(C)(O)C3CCC3)=O)CC2O)ccc2cncn2c1 7938,c1(C(N2CCN(Cc3cc(OCC)cc(F)c3)C3C2C3)=O)ccc2cnoc2c1 7939,C1(NC(C2(C)CCCN(C(C(C)(C)CO)=O)C2)=O)CC2(CCCCO2)C1 7940,C1(C(N2CCC(NC(=O)C=Cc3cscn3)C(O)C2)=O)CCC2C(C1)C2(F)F 7941,C(=O)(C(C)(F)C(C)(C)F)NCC1CCC(N(C)C(C2CC3CC3C2)=O)CC1 7942,c1(C(=O)NCCC2CSCCN2C(C2CCCCS2)=O)ccc2c(c1)OCO2 7943,Cc1nc(NCC2CCCCC2NC(C2(C)CNC(=O)C2)=O)cc(Cl)n1 7944,C1(CNC(c2c(C)c(Cl)ccn2)=O)CN(C(=O)CC2CCCOCC2)CC(C)(C)C1 7945,N1(C(CCC2(C)CC2)=O)CC(C2CC2)(C(N)=O)C1.c12ccc(o1)C(=O)NC2 7946,C1(C(N(CCCCCNC(c2cc(CCCO)on2)=O)C)=O)CCC(C)(C)OC1 7947,c1(OC(N2CCN(c3ccc(Cl)cc3)CC2)=O)cccnc1O 7948,N1(Cc2cn(CCCNC(CN3C(=O)OCC3)=O)nn2)CCC(F)(F)CC1 7949,Cc1cc(C(=O)NCC(C)CNC(c2cnc(-c3ccoc3)s2)=O)cc(N)c1O 7950,C1(C(=O)NCCN(C(=O)CSC(F)(F)F)CC)CC2CC(OC)C2C1 7951,Nc1cc(C(=O)NC23CC(CNC(=O)Cc4cncnc4)(C2)C3)ncc1Cl 7952,N1(C(C(C)OC2CCCCC2)=O)CCCC(C2CCN(C3CCN(C)C3=O)C2)C1 7953,c1(C(N2C(CN(C(c3ccnn3C)=O)CC)CCC2)=O)ccnc2ccnn12 7954,N1(C(c2nc(N)c(Br)cc2)=O)CC2(CCN(C(c3ccnn3C3CC3)=O)C2)C1 7955,c1(N2CCC(NCc3c(OCC)cc(Cl)cc3)CC2)nc(C)c(C)cn1 7956,CCC(C)CCC(=O)Nc1ccc(NC(C2(C)CCOC2C)=O)cc1C 7957,N1(CC)CCC(C(=O)NC2CC(C(F)Cn3cc(C(C)(C)C4CC4)nn3)C2)C1 7958,C(=O)(C(CNC(C1CC1C(C)C)=O)CC(C)C)N(C)Cc1c(C)nn(C)c1 7959,Cc1ccsc1C=CC(N1CC(O)(C(C)(C)CNC(=O)C=CC2CC2)C1)=O 7960,C1(CC)(NC(c2ccc(C#N)o2)=O)CCN(C(c2ccccc2NC(N)=O)=O)C1 7961,n1(CC)cc(CN(C(=O)CN(C)CCN(C(=O)Cc2cc[nH]c2)C)C)cn1 7962,c1(C(=O)NC2(CO)CN(C(c3ccnc(C4CC4)c3)=O)C2)cnc2[nH]cnc2c1 7963,C1(C)(CNC(c2c(CC)c[nH]n2)=O)CCC(NC(=O)CCc2cccc(Cl)c2)C1 7964,C#CCCCCCCCC(=O)N1CC(CNC(=O)CCC(=O)OC)C(C)C1 7965,CCCCC(C)CCC(=O)NCC1(CNC(=O)CSC(C)C)CCCC1 7966,CC(C)S(=O)(=O)C(C)C(=O)N1CC(C)(C)OCC1CNC(C1(CC2CC2)CC1)=O 7967,C(=O)(C1=C(CC)OCCS1)NCCN(C(=O)C(c1ccc(Cl)c(Cl)c1)O)CCC 7968,N1(C(C2C(CC)C2)=O)CCC(C)C(NC(c2cc(-c3ccco3)on2)=O)C1 7969,C(C)(C(=O)N1CC(O)CO1)C(CC)CC(=O)N(C1CN2CCN1CC2)C 7970,C1(CC(=O)NC(C2CCCCC2)CNC(c2cc(C)no2)=O)(OC)CCCCC1 7971,Cn1cnc2c(N3CCCC(N4CC(O)C4)C3)nc(S(C)(=O)=O)nc12 7972,C1(COC)CN(C(c2c(C)noc2C)=O)CCN1C(=O)C=Cc1cccn1C 7973,C1(CNC(C=CC=CCC)=O)CCC(C)CN1C(=O)Cc1ccc(C)s1 7974,Cc1ccc2ccccc2c1NC(C1CC(C)CN(c2ncnc3n[nH]cc23)C1)=O 7975,CC(C)C1=NOC(C(=O)N(CC(=O)NCC(C)(O)C2CCCC2)CC2CC2)C1 7976,c1(C(=O)NC2CC(NC(CCNC(=O)CO)=O)C2)cc(C2CC2)cs1 7977,C1(NC(CC2(C)CC2)=O)CCCN(C(c2cc3cccnc3[nH]2)=O)CC1F 7978,C(CCCC(C)(F)F)(C(=O)O)NC(c1cncc(C(C)C)n1)=O 7979,Cc1nncn1CCCC(=O)NCC(C(=O)NC1CCOC1)N(C)C 7980,C1(CN(C(C2(C)CSC2)=O)CC)CCN(C(=O)CC2(N(C)C)CC2)CC1 7981,CC(CN(C)C)CCC(=O)N1CCC1CNC(c1ccc(Cl)cn1)=O 7982,C1(CNC(CCC)=O)N(C(C2CC(C3CCC3)C2)=O)CCCC1(C)C 7983,C=C(C)CCN=c1[nH]c(N2CCN(C3CCSCC3)CC2)nc2cc[nH]c12 7984,C1(C2CC2)(NC(c2c(CC)ocn2)=O)CCN(C(=O)COCC(C)C)C1 7985,CC(C)CC(C(=O)O)NC(C1(CO)CC1C(F)(F)F)=O 7986,C1(C(NOCC(CC)C)=O)C2CCC(C2)N1C(=O)Cc1ccon1 7987,Cc1cc(F)ccc1C(N1CC2CCC1C2NC(=O)C(C)Sc1ccccc1)=O 7988,C(C(C)CN=c1ccnc(C)[nH]1)NC(c1cccc(OC)n1)=O 7989,C#CCC(CC(F)F)C(=O)NCc1ccsc1C(=O)NCC(=O)NC(C)C 7990,C#CCC(C)(CC)C(=O)NC1CCC1NC(C1CCN(CC(F)F)CC1)=O 7991,n1(CC(=C)C)c(Cc2ccccn2)nnc1-c1[nH]nnc1C 7992,C12(NC(COC)=O)CC1CN(C(C1(CC3CC3)CC1)=O)C2 7993,FCCCN=C(NCCCN1CCCCC1)NCC(c1ccccc1)C1CCC1 7994,c1(-c2ccc(CCCCCC)s2)ccc(SCOC)cc1O.C1(=O)C(CCC2CC2)N1 7995,CC(=O)CCCC(=O)NCCNC(C1CN(C(c2ccc(F)o2)=O)C1)=O 7996,N1(C(C2CC(C)(C)CN2C(=O)CC2(O)CCOCC2)=O)Cc2ncsc2C1 7997,C(=O)(CCCCCC(C)C)OC(C1(C(N(CC(C)(C)OC)C)=O)CC1)=O 7998,C1(NC(C2C(c3n(C)ccc3)C2)=O)CCCCC1NC(=O)C(N(C)C)SC1CC1 7999,Cc1cccc(CC(=O)NCc2ncoc2CCNC(c2csc(CO)n2)=O)c1 8000,c1(OC)cc(Cl)c(CC(=O)C(=O)OC)cc1Cc1cnn(CCl)c1C 8001,C1(C(N2CC(CNC(=O)COCC(F)(F)F)C(O)C2)=O)(OCC)CCSCC1 8002,c1(C(N2CCCC(O)(CNC(c3cncc(C)n3)=O)C2)=O)cnc2[nH]nnc2c1 8003,c1(C(N2C(CNC(Cc3c(C)ccnc3)=O)C=CC2)=O)ccc([N+](=O)[O-])s1 8004,CC1(C)COC(CC(N2CCCC(Cn3cc(-c4ncc(Cl)cn4)nn3)C2)=O)CO1 8005,N1(C(CS(=O)(=O)NCC)=O)C(C(=O)NCCc2ccco2)CC2CCCC12 8006,C(C1c2ccccc2CCN1C(=O)C1=CCOCC1)NC(c1n(C=C)nnc1)=O 8007,C(C(C)(CCO)NC(=O)CC1CCN(C(c2ccc(CC#N)cc2)=O)C1)OCC 8008,N1(CC(=O)NCC(CN(C(c2c(C(=O)OC)[nH]nn2)=O)C)C)CC(=O)NC1=O 8009,CCCC(C)CCCC(=O)N1CCN(CCNC(=O)C(C)S(N)(=O)=O)CC1 8010,N1(C(CCC(=O)NCCC)=O)CC2CCCC2(C(=O)NC23CCC(C2)OC3C)C1 8011,N1(Cc2ccc(C#N)cn2)CCC2(CCN(C(=O)CC3CCOC3)C2)C1 8012,c1(COCC)cn(CCCNC(c2cc(COC)no2)=O)nn1 8013,C(=O)(C(CO)C(C)(C)C)NC1(C)CCC1.C12CC(C1)NCC(=O)N2 8014,N1(C(=O)Cn2cc(Cl)cn2)CCN(C2CCC(NC(=O)Cc3ccon3)C2)CC1 8015,Cc1ccc(CCCN(c2ccc(F)cc2)C2CCOC2)c(C)c1 8016,c1(CC=O)ccc(F)cn1.c1(C(=O)OC)cc(C(=O)NCCNC(C)=O)c[nH]1 8017,c1(CC(C)C(=O)NCC2CN(C(c3ncc[nH]3)=O)CCO2)ccccc1Cl 8018,N1(C(COCCCOC)=O)CCC2(CC2)CC1C(=O)N(C)Cc1scnc1C 8019,c1(OC)ccnc(C(N2CCC(C)C(C)C2)C(=O)NCc2ccc(F)cc2C)c1Br 8020,C(C(CC(=O)NCc1cnc(C)o1)NC(C1CN(CC(C)C)C1)=O)OC 8021,CCCC(CNC(=O)CCC1CCOC1)C(=O)NCP(C)(C)=O 8022,C(=O)(N=c1[nH]ccnc1C1CC1)C1C(NC(=O)Nc2cc(C)nn2C)C1 8023,C1(C)(NC(CCCN(C)C)=O)CCN(C(C2CCOC2c2cccnc2)=O)CC1 8024,Cc1c(C(=O)NC(C)CNC(C2CCC(C)O2)=O)sc2ccc(Cl)cc12 8025,N1(C(c2nc(OCC)sn2)=O)CCCC(CCCCNC(c2cccnc2C)=O)C1 8026,C1(CNC(C(C)OC(c2ccc(C)nc2)=O)=O)Cc2ccccc2C1 8027,C1(NC(C2C3COCC23)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 8028,C(=O)(CS(=O)(=O)C1CC1)NCC1(C)N(C(c2n(C)c(S)nc2)=O)CCC1 8029,C1(C(=O)NC(C2CCCOC2)CC)(NC(=O)COc2ccccn2)CCOCC1 8030,c1(NC2CCCN(C(c3cccc(C)c3)=O)C2)nc(Cl)nc2c1ncn2C 8031,c1(C(C(C)C)C(=O)OCC(N2CCCC2)=O)cccc(C#N)c1 8032,N1(C(C(C)[SH](c2ccccc2)CC#N)=O)CCCC(N=c2[nH]ncs2)CC1 8033,N1(C(CCOCCC)=O)CCC2(CC1)CC2C(=O)NCC1CCC(C2CC2)CC1 8034,c1(N(C(CN2CC(NCC)C2)=O)Cc2cncs2)nc(C)cs1 8035,Cc1nnc(C)cc1C(N1CCCC(CCC(=O)NCCN2CC(C)(O)C2)C1)=O 8036,c1(C(CO)NC(C2CCC(NC(c3ccncc3F)=O)C2)=O)cccc(F)c1 8037,c1(S)csc2ccccc12.c1(OC(C)(C)C)ccc(Cn2ncc(C=O)c2)c(F)c1 8038,c1(C(=O)NC2CCCN(C(CCCSC)=O)C2C)c(O)nnc(C)c1C 8039,c1(C(N2CC(CC(=O)OCC)OCC2)C(=O)NCC(F)F)cc(F)cc(Cl)c1 8040,Cc1cc(C(N2CCC(CC(=O)NCC(C3CC3)C3CC3)CC2)=O)[nH]c1C 8041,C1(N(C)C(c2cnn(C3CC3)c2)=O)CN(C(c2nonc2N)=O)CC1F 8042,C(C)(C)(C(c1nnnn1C1CCC1)NCCCOC(=N)O)N(C(C)=O)C 8043,C1(C(=O)NC2CC(NC(c3c(CC)sc(=N)[nH]3)=O)C2)C2CCCCCCC12 8044,C(c1nnn(C)n1)=CC(=O)N(CCN(C(COCCOCC#C)=O)C(C)C)C 8045,C(CN=C(NC(=O)N(C(C)C)C(C)(C)C)NCC1C=CCCCC1)SC1CC1 8046,C1(COC)(CNC(=O)CC2C=CC(NC(C3CC(CF)C3)=O)C2)CCCC1 8047,c1(C(C(=O)NC(C)C)N(C(C)C)CC)cnn(-c2ccccc2)c1 8048,C1(CC)CN(C(=O)Cc2c(F)cncc2Cl)CCC1NC(C1CCSCC1)=O 8049,c1(C(N(CC(CC)NC(=O)CCC2CCCC2)CC)=O)nc(OC)ccc1C 8050,Cc1cc2[nH]c(C(N3CC(NC(C4(O)CCCCC4)=O)C(C)C3)=O)cc2s1 8051,c1(CC)nn(C)cc1C(=O)NCC1CCCC1NC(=O)COc1ccsn1 8052,C1(CC)CN(C(C2CC2c2nc[nH]n2)=O)CCN1Cc1ccc(C)cn1 8053,Cc1[nH]nc(C(F)F)c1C(N1CCC(CCNC(C2CN(C)CC2C)=O)CC1)=O 8054,N1(C(C(C(C)OC)N(C)C)=O)CCC(CC(=O)NCC2COCCN2C)CC1C 8055,C1(NC(c2c(NC)scn2)=O)C(C)(C)C(NC(C2SC3C=CC2CC3)=O)C1(C)C 8056,C12(C(=O)NCCCN(C(C3(COC)CCCC3)=O)C3CC3)CCCCN1CCC2 8057,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CNC(c2cccnc2C(N)=O)=O)C12CC2 8058,CC1(NC(=O)CNc2cc[nH]c2)CCC(NC(=O)CC(F)(F)F)CC1 8059,c1(C(C)C)ccc(C(N2CC(NC(c3ncccn3)=O)CC2C)=O)cc1[N+](=O)[O-] 8060,S(=O)(=O)(c1cc(F)c(F)cc1F)N1CCn2c(C)nnc2C1 8061,N1(C(c2c[nH]c(=NCC=C)s2)=O)CCN(C(=O)C=CCF)CC(O)C1 8062,N1(C(COCCC)=O)CCCOC(CNC(c2csc(Cn3cccn3)c2)=O)C1 8063,C(=O)(CCC(C)NC(c1coc(N(C)C)n1)=O)N(CCOC)CCO 8064,c12cccc(c1)C(=O)NC(NC(COC(CC)(C)C)=O)CNC2=O.C1(NC)CC1 8065,c1(C(=O)NC2CCC(NC(=O)CO)CC2)ccc(=O)n(CC2CCCO2)n1 8066,N1(C(c2c(C(C)(F)F)cccc2)=O)CC(NC(=O)CCn2cccc2)CC(O)C1 8067,O=C(N1CC(O)CCO1)c1ccc(Br)c(Br)c1 8068,c1(OC)ccc(CC(=O)NCC(C)CN(C(=O)C(O)C2CC2)C)c(Cl)c1 8069,N1(C(c2c(CC)non2)=O)CCCC2(CNC(c3ccnn3CC)=O)CCCC12 8070,C(C(C)N=c1cc(-c2ccccn2)nc(S(C)(=O)=O)[nH]1)(NS(CC)(=O)=O)OC 8071,CC1CN(C(=O)C(C2CCN(C(c3[nH]ccc3C3CC3)=O)CC2)C)C(C)C1C 8072,C1(NC(=O)NCCCOCCC(=O)NC2CCC2)CC2CC1CC2O 8073,C(C)(N=c1[nH]c(Cl)ncc1F)C1N(C(C(CCC)CCC)=O)CCCC1 8074,C=Cc1cc(C(=O)NC2CCC2NC(c2c(C3CC3)noc2C)=O)cc(F)c1 8075,C=CCC(C1CC1)NC(C1CCN1C(=O)CSC)=O 8076,C1(NC(CC(C=C)C)=O)CN(C(c2cccc3ccccc23)=O)CC2(CCC2)C1 8077,N1(C(CCC2C(C)C2)=O)CCOCC1CNC(C1CN(C)C1)=O 8078,N1(C(c2cncc(C)n2)=O)CC(Nc2ncc3ccsc3n2)CC(C)(C)C1 8079,c1(CC)c(C(=O)N(CCCNC(=O)C=CCn2cncn2)CC)cnn1CSC 8080,C1(C(=O)NCC2CC3CC(NC(c4ccns4)=O)CC32)CCC2CC1CO2 8081,N1(C(C2N(C(c3coc(C4CC4)n3)=O)CCC(=C)C2)=O)CCC12CCCSC2 8082,C=CCC(C(=O)N1CCCC(N(C(=O)CCCCCCSC)CCO)C1)C(C)C 8083,CP(C)(=O)C(C1CC1)NC(=O)C(O)c1ccco1.C12(CC1)CC(=O)N2 8084,C#CC1(NC(=O)C(F)C2CC(NC(C3(C(C)(C)O)CCC3)=O)C2)CCCOC1 8085,C1(C(=O)NC2C(C)N(C(=O)CCOC3CCCCC3)CC2)CC2(CC2)CN1C 8086,C(=O)(C(CSC)CC)NCC1(C(=O)N(C(CC)CC)C)CC(=C)C1 8087,c1(NC(c2cc(C)on2)=O)nc2ccccc2nc1Cl 8088,N1(C(c2ccc(SC)o2)=O)CC2CCCC2(C(=O)NCC23CSCC2C3)C1 8089,C#Cc1ccc(C(=O)NCC2CC(CNC(c3ccc(C)cn3)=O)C2)cn1 8090,c1(C(=O)NCCN(C(C(C)OC)=O)C)ccnn1C1CCC1 8091,C1(CNC(CCOC)=O)CN(Cc2c(F)cc(F)cc2Br)CCC1(F)F 8092,C(CCC(C)(F)F)NC(c1cccc(F)c1)c1n(C(CC)C)nnn1 8093,CCCC(C)CCNC(=O)CCNC(=O)C(C)(C)C1CCOC1 8094,c1(C(N2C3(C(=O)NCC(CO)OCC)CC3CC2)=O)cccc2ccccc12 8095,C=C(CCC(=O)OC(C)C)C(=O)NC(C)CC(=O)NC1CC1 8096,Cc1cc(CC(C)C(=O)ONC2CCC(C)N(C(=O)OC(C)(C)C)C2)ccc1N 8097,c1(N(C)C)ccc(SNCc2n[nH]c(C(F)(F)F)n2)cn1 8098,C12(CNC(C(C(C)(C)C)NC(C)=O)=O)CCC(CC1)N(C(C1C3(CC3)C13CC3)=O)C2 8099,c1(C(N2CC(C)(NC(C3CCCCCC3)=O)C2)=O)ccc(N)c(Cl)n1 8100,Cc1ccnc(C(N2CC(F)(CNC(=O)C(C(C)C)NS(N)(=O)=O)C2)=O)n1 8101,c1(C(N2CCC(CCNC(C(C=CCCC)O)=O)C2)=O)cn2cccnc2n1 8102,c1(CC(=O)OCCSc2ccc(NC)cc2)c[nH]c2cccc(C)c12 8103,N1(C(C=C(C)C2CCCCC2)=O)CCC(NC(=O)Cc2conc2C)CC(O)C1 8104,C1(C(=O)OC(c2c(C)nsn2)C)CCc2ccccc2NC1=O 8105,CC1CCSCCN1C(c1ccc(-c2cn(-c3cccnc3Br)nn2)cc1)=O 8106,C1(C(=O)NCC(C)CN(C)C(C2(O)CCSC2)=O)CC2(CCC2)C1 8107,C(C)(C)(CC(=O)NC(c1ccc(F)cc1)CNC(=O)CC1CSC1)SC 8108,N1(CC(C)C)CC(C(=O)NC(C)(C)C(C)NC(=O)CCc2ncc[nH]2)CC1=O 8109,N(C1CCCc2occc21)C(c1n(C(C)C)ncc1Br)=O 8110,c1(OCC)ccccc1CC(=O)N(C)CCNC(=O)CCCSC(C)(C)C 8111,N1(CC(=O)NC2CN(C(CCCc3nnc(C)n3C)=O)C2)CCc2sccc2C1 8112,c1(CC(=O)NCC(CN(C(CCC(CC)C)=O)C)C)ccc2c(c1)ncn2C 8113,Cn1c(O)nc2cc(C(=O)Nc3c(I)cnnc3O)ccc12 8114,CCCC(C)OCCC(=O)N(CCCNC(=O)C(O)C1CCCC1)C(C)C 8115,C12(NC(c3ccc(C)cc3F)=O)CCCCCC1N(C(=O)C(C)C)CC2 8116,c1(C(N(CC(C)NC(=O)Cc2cncnc2O)C)=O)ccnc(Cl)c1Cl 8117,N1(C(CC2(C=C)CCCCC2)=O)CC2CCN(C(C3SCCS3)=O)C2C1 8118,c1(-c2cn(CC(=O)NCC3CC3)nn2)ccc(C(F)(F)F)cc1 8119,C(=O)(C(CC)C(=O)N1CCCC(NC(c2ccc(C)cn2)=O)C1)OCC 8120,N1(C(c2cn(C)nc2)=O)CCN(CC(=O)NCCN2CC=CCC2)CC1 8121,c1(C(=O)NC23CN(C(C(CCCC)F)=O)C(CC2)CC3)c[nH]c2c(F)cccc12 8122,C1(C(=O)NC(COCC)C)C2CC3C(C2NC(c2cc(C)nnc2C)=O)C13 8123,N1(C(C(C(C)C)SC2CC2)=O)CC2(C1)CN(C(=O)CC1(O)CCOC1)CC2CO 8124,Cc1c[nH]nc1C(=O)N(CCCOCCN(C)C(c1cnc(C(C)(C)C)o1)=O)C 8125,C=CC(C)(C)C(=O)N(CC(O)CN(C)C(C1(CC)CCOC1)=O)C 8126,C12(NC(CC3CC(=C)C3)=O)CCCC1CN(C(c1ccc(F)c(O)c1F)=O)C2 8127,c1(-c2oc(CNC3(CNC(=O)OC(C)(C)C)CCCC3)c(C)c2)cccc(Cl)c1 8128,c1(OCC)ncccc1NC(c1csc(CNC(=O)C(C)C2(O)CCC2)n1)=O 8129,c1(OC)ncc(C(=O)NC2CC2NC(c2c(C)nn(C3CC3)c2Cl)=O)cc1C 8130,C1(C)(C(=O)NC2(C)CC(NC(c3n(CCC)ccc3)=O)C2)CCC(=O)N(C)C1 8131,CC1CN(C(=O)CN(S(C)(=O)=O)C)CCCN1C(C1C2COCC12)=O 8132,C1(NC(Cn2nnc(=N)[nH]2)=O)CCN(C(=O)COC2CCCCC2)CC1 8133,c1(C(N(CCOCCNC(=O)C(F)(F)CC)C)=O)nc(SC)cc(C)n1 8134,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CCN(C(c1ccc(I)c(O)c1)=O)C2 8135,C(CNC(C1(C)N=N1)=O)(C(=O)NCCC1COCCO1)N(C)C 8136,c1(C(=O)NC2C(NC(C(=C(C)C3CC3)F)=O)CCC2)cccc(CCN(C)C)c1 8137,C1(C(N2CC(CNC(=O)Cn3cc(C(F)F)cn3)C2)=O)CC1C1CC(F)(F)C1 8138,N1(C(C(C)SC)=O)CCC(NC(c2cnc(C(C)(C)C)nc2)=O)C(F)(F)CC1 8139,CC1(C)COCCN(C(C2CC(O)CN2C(=O)CC2CC2C2CC2)=O)C1 8140,Cc1nnc2n1C(C(=O)NC1CCc3nc(NC4CC4)sc3C1)CC2 8141,C1(C(=O)NC(C(=O)OCC)CC)CN(C(C2(Cl)CCC2)=O)CC12CC2 8142,C1(NC(C(CCC)F)=O)CCC2(CCN(C(C3(C)CCCC3(F)F)=O)C2)C1 8143,C1(O)(CNC(C2CCCOCC2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1 8144,Cc1cnn(C)c1C(=O)NCC=CCNC(C1CCCN(c2ncccn2)C1)=O 8145,C1(C(=O)OCC)CCC(F)(CNC(c2ccccc2I)=O)CC1 8146,C(C(C(=O)NCc1cc(C)no1)C(C)(C)C)NC(C(C)(C)SC)=O 8147,c1(OC)nc(C)cc(C)c1C(N1C(C)(C(=O)OC)CCC1)=O 8148,C(C)(C)(CCCC(=O)Nc1cnn(C)c1C)NC(CCn1ccc(C)n1)=O 8149,C12(C(=O)NC(CNC(C(C=C)(C)C)=O)C(C)(C)C)CCC(CC1)C(C)O2 8150,C1(NC(c2cncnc2-c2ccccc2)=O)CC2CC1N(C(c1cccs1)=O)C2 8151,c1(C(=O)NCCCN(C(c2ccc(C#C)cn2)=O)CC)ccc2c(c1)CCC2 8152,N1(C(c2c(C)scn2)=O)CCC2(CC1)COCC(CNC(=O)CCCF)O2 8153,N1(C(=O)NC2CN(C3CCCCC3)C2)CCC(C2CCCC23OCCO3)C1 8154,c1(C(c2nnnn2C)NCC(=O)NCC)c(CC)cccc1C 8155,N1(C(c2coc(Br)n2)C(=O)OC)CC2CC1CS2=O.C12CC(C1)NC2=O 8156,N1(C(C(Cn2cccn2)NC(COCCSC)=O)=O)CCCN(C(C)C)CC1 8157,Cc1ccnc(C(N2CCN(CCNC(C3(C)CCCC3C)=O)CC2)=O)c1O 8158,CC(C)(C#CC(=O)N1CCCC1CCO)CNC(c1ccc(F)c(C)c1)=O 8159,C=CCC(C)(C)CC(=O)NC12CCOC(CNC(=O)CC3CCN(C)C3)(C1)C2 8160,c1(CCN(C(C(N2CCC(C)C2)=O)=O)C)c[nH]c2cccc(Cl)c12.[nH]1cncn1 8161,N1(C(CCC#N)=O)CCN(CC2(NC(=O)CC(O)CN(C)C)CCCC2)CC1 8162,c1(C(C(=O)NCCC(C)NC(=O)CCOCCOC)OC)ccccc1F 8163,C1(COC)(COCc2ccncc2)CN(C(=O)CCc2nc(SC3CC3)no2)C1 8164,c1(C(=O)NCC2CCC(CNC(=O)C(F)F)CC2)cc2cccc(Br)n2c1 8165,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8166,C1(CCNC(c2ccccc2)=O)CCN(Cc2ccc(F)s2)C1 8167,c1(NC(C2COCCN2C(C2C3COCC23)=O)=O)ccc(Cl)c2cc[nH]c12 8168,C1(CNC(C(C)SC)=O)CCC2(CCN(C(=O)Cn3ncnn3)CC2)CO1 8169,C(=O)(CCC(=O)NCC1COCCN1CC1CC1)NCc1nnc(C)s1 8170,C(C(C)(C)N=c1[nH]nc(C#N)s1)N(C)C(c1nnc(C2CC2)c2c1CCC2)=O 8171,C12(CNC(Cc3c(C)[nH]nc3C(F)(F)F)=O)CCCCC1CN(C(=O)CC#N)C2 8172,N1(C(c2ccc(NC(C)C)cc2)=O)CCC2(CNC(=O)C(O)CF)CCCCC12 8173,c1(C(N2C(C)CC(NC(C3(CC)CC3)=O)C2)=O)cc(C)cnc1OC 8174,C(CC(C)C)(C(=O)N1CCC(CCO)CC1)ONC(c1cn(CC=C)nc1)=O 8175,N1(C(c2cnn(C)c2N)=O)CC2(CCC(CNC(=O)CC3CC4CCC3O4)O2)C1 8176,C1(C(=O)NCCCC(=O)NCCCOCC=C)CC(=O)OC1(C)C 8177,C(=O)(C1=C(F)CN(C(C2CC23CCCCC3)=O)CC1)N(C(C#C)C)C 8178,c1(N2CCOCC(NC(C(C)OCC#C)=O)C2)cc(OC(C)C)ccc1[N+](=O)[O-] 8179,c1(C(N2CC(OC(C)(C)C)CC(C)C2)C(=O)NC)cc(C(C)C)ccc1F 8180,N1(C(Cc2c(C)nsc2)=O)CC2CC(C1)CN(C(C1(C3CCCO3)CCC1)=O)C2 8181,C1(CNC(c2c(C)cc(C)s2)=O)CCC12CCN(C(C1CCCOC1)=O)CC2 8182,N1(C(c2cc(I)cn2C)C(=O)NCCCC)CCOc2cccc(F)c2C1 8183,N12CC=CC1(C(N1CCCC1)=O)COC(C)C2=O.C1(COCC)(OC)CCCC1 8184,c1(CNC(c2sc(C)cc2Br)c2n(CCOC)nnn2)cnc(OC(C)=O)cn1 8185,c1(C(=O)NC2CCC(CNC(COCCC)=O)C2)cc(-c2cccnc2)n(C)n1 8186,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8187,C(=O)(C1CCc2c(Cl)cccc21)N1CCC(CNC(C2CC(=C)C2)=O)C12CCC2 8188,c1(OC)ccccc1C(O)C(=O)NCC1CCC1NC(c1cc(CO)nn1C)=O 8189,C1(CCC(=O)NC2CCCC2CNC(C2CC(O)C2)=O)CCCCO1 8190,C(=O)(CC(C)CNC(c1occc1CNC(=O)CC1C(=O)NN=C1C)=O)OC 8191,c1(C(=O)NCC2CCCN2C(=O)C2=CCCS2)cnc2nccnc2c1 8192,Cc1cn(C)nc1C(N1CCC(CN(C2CCC(Cn3ccnc3)C2)CC)CC1)=O 8193,C(=O)(C(C)(C)c1cccnc1)NCCN(CCC)C(c1nocc1C(C)(C)C)=O 8194,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8195,c1(NCCNC(=O)OCC)[nH]c(=NCC2CCCC(F)(F)CC2)nc2ncn(C)c12 8196,C(C(C)(C(=O)N(CCCCC(=O)NCC(O)C1(Cl)CC1)C)OC)OC 8197,C1(C(N2CC(NC(c3cncnc3)=O)C3(C2)CC3)=O)CC2CC1CC2(F)F 8198,c1(N2CCC(CNc3cc(OCC)ncn3)CC2)nc(=O)cc(N)[nH]1 8199,c1(CC(N2C(CNC(Cn3ncc(C#C)c3)=O)CCCC2)=O)ccc(Cl)c(F)c1 8200,c1(C(N2CC(C3N(C(CN4C(C)CC4)=O)CCC3)(O)C2)=O)ncc(Cl)cc1Cl 8201,CC1COCC(CC(=O)NC(C)(C(=O)N(C2CCCC2)CCO)C2CCC2)O1 8202,C1(C(N(CCN(C(C)=O)C(C)C)C)=O)C2CCC(C2)C1Cc1ccccc1 8203,c1(C(C(=O)NC(C)CNC(c2c[nH]nc2F)=O)(C)C)ccc(Cl)cc1Cl 8204,C(=O)(C(Cc1cn(CSC2(F)CCC(C)CC2)nn1)CC(F)(F)F)OC 8205,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)C)NC(CC#CC)CO 8206,c1(C(=O)NCC(CNC(C(C2CCCC(F)(F)C2)OC)=O)O)cnnc(C)c1C 8207,C=CCC(CC=C)C(=O)N1CCCC(C)(CNC(=O)CCOC)C1 8208,Cc1nc(-n2cccc2)sc1C(=O)NC1(CNC(c2cnn(C)c2Cl)=O)CC1 8209,CC1CCC(NC(=O)CCCN2CCCC2)CN1C(=O)CN(C)CCO 8210,O=S(=O)(c1ccccc1)C(F)(F)F.c1(N)nccc(=NCC2CC2C2CC2)[nH]1 8211,C1(CNC(C(F)=CCC)=O)CC(NC(c2coc(CC3CC3)n2)=O)C1(C)C 8212,C(CC(C)(C)C(F)(F)F)NC1(NC(=O)OC(C)(C)C)CCCC1 8213,NC(CCNCc1csc(C(F)(F)F)n1)C(F)(F)F 8214,C(CCCN(CCCNC(c1ccno1)=O)C)NC(C1(C(F)(F)F)CC1N)=O 8215,C(CS(=O)(=O)CC(=O)N1CCC(C(C)C(=O)Nc2ccn(C)c(=O)c2)C1)OC 8216,N1(C(C2(C)CC(C)C2)=O)CCN(C)C(CNC(C2(C)CCCS2)=O)C1 8217,C(CN=c1cc(C2CCCC2)nc[nH]1)(C1CC1)NC(c1cc(C2CC2)[nH]n1)=O 8218,C1(NC(CCC=C)=O)CC2CCCC(C1)N2c1cc(C(F)F)ncn1 8219,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(c2ccc(C)cn2)=O)C1 8220,CCCCC(C(=O)NCC1CCCN(C(c2ncccc2CO)=O)CC1)C(C)C 8221,C(CCCCCCCO)=CC(=O)NC1CN(C(C(CSC)(C)C)=O)CC2C1C2 8222,C1(NC(C2(CC#C)CCC2)=O)CN(C(c2ccc(CC(C)C)cn2)=O)CC1C 8223,c1(C(N2CCCC(F)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8224,N1(C(=O)CCOc2cccc(Cl)c2)CCCC(C2CCCN(c3ncns3)C2)C1 8225,C1(C(=O)NCC=CCNC(C2(CC)CCOC2)=O)CC2(C1)CC(C)C2 8226,C1(CCNC(c2ccco2)=O)(C(=O)NCC2COCCO2)CCCC1 8227,c1(C(=O)NC2(C(=O)OCC)CC2)cccnc1CC.C12(CC(O)C1)C(=O)N2 8228,c1(OC)cc(OC)cc(C(=O)NC(C2CCN(c3nncs3)C2)C)c1 8229,C1(C(=O)NCC(C2CC2)OC(C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8230,c1(CC=C)cccc(C(N2CCC(C(C)C(=O)NCCCN3CCC3)CC2)=O)c1 8231,C1(C(=O)NCCN(C(COCCC=C)=O)CCOC)CC2C=CC1CCC2 8232,c1(C(N2CC3CC(NC(C4CC(F)(F)C4)=O)CC3C2)=O)cc2cccc(F)c2s1 8233,CN1CCC(=CC(=O)NCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8234,C(=O)(C(C)(C)C(F)F)NC(CNC(C1(CC)CCC1)=O)(C)Cn1cccn1 8235,c1(N2CCCC(CS(N3CC(C)OC(CC#N)C3)(=O)=O)C2)ccc2ccccc2n1 8236,N1(Cc2cc(Br)ccn2)CCC(O)CC1C(=O)OCc1ccc(C)cc1 8237,C1(CC)C(=O)NCCCN1C(=O)CCOCCN(C(=O)CN1CC(=O)NC1=O)C 8238,C12(CNC(COCCCOCC)=O)CC(NC(C3COCCO3)=O)(C1)C2 8239,C1(CNC(C(C)CN(C)C)=O)CC2CCC(C1)N2C(c1cccc2c1COC2)=O 8240,Cc1ccsc1C(=O)NCC1C=CC(NC(=O)C(O)CC2CCCC2)C1 8241,c1(OC)ccc(-c2cn(CCCNC(=O)CSC(F)F)nn2)cn1.c1cn(CC)nn1 8242,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8243,N1(C(C2C(NC(=O)NCCCl)C2)=O)CCC(CC2CCCCC2O)CC1 8244,N1(C(C2N(C)CCOC2)=O)CC2CCC2(CCNC(c2cc(CO)n(C)n2)=O)C1 8245,c1(C(=O)OC)cncc(-n2cc(CONC(c3ccnnc3O)=O)nn2)c1 8246,N(C(=NCCC(C)NC(=O)OC(C)(C)C)NCC(C)(C)C)C1CC(OC)C12CCC2 8247,Cc1ccc(CC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8248,C1(C#N)(C(N(C)CC2N(C(COCCN(C)C)=O)CCCC2)=O)CCCOC1 8249,C1(CC(=O)NC(C)C(C)n2cccn2)C(NC(=O)Cc2cncs2)CC1O 8250,N1(C(C(C)(C)OC)=O)CCC(C)C1C(=O)NCCc1cnc(C)[nH]1 8251,c1(CC)ccc(C)c(C(N2CCC(CCNC(C3SCC=C3C)=O)CC2)=O)c1 8252,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8253,C1(CC(=O)OC)CCCN1C(N(C1(C(=O)OC(C)(C)C)CCC1)C)=O 8254,c1(NC(c2nnnn2Cc2nnn(C)n2)C)ncc(C(F)(F)F)cc1Br 8255,N1(C(CCCc2c(C)ccs2)=O)CCC(C)C1CNC(c1ccccc1CO)=O 8256,Cc1cnc(C(=O)NC2C3CC4C2C4C3C(=O)NC2(CCCF)CC2)c(C)c1 8257,c1(C(=O)NC2(CC)CCCN(C(CCC)=O)C2)ccc2nnn(C(C)(C)C)c2c1 8258,N1(C(c2cc(C3CC3)ccn2)=O)CC2OCCN(C(c3sccc3Cl)=O)C2C1 8259,N1(C(CCOCC)=O)CCC(O)C1C(=O)N(CC(C)(C)OC)C 8260,C(C(CC(=O)NCc1cncc(Cl)c1)C1CCC1)NC(C(=O)N(C)C)=O 8261,N1(C(c2ccc(CNC(C(CCCC)=O)=O)o2)=O)CCC2(CCCOC2)C1 8262,c1(C(N(C2CCN(C(=O)C(C(C)C)SC)CC2)CC#C)=O)cnc2cc[nH]c2c1 8263,C1(C(=O)NCCNC(C(C)c2cccs2)=O)CC(C)(C)CO1 8264,C12(CNC(=O)CC(F)(F)F)CCCCC1N(C(=O)CN1CCSCC1)CC2 8265,C(=O)(C(C(=O)N1CC2CCCC1C2CNC(=O)C(N)=O)C(C)(C)C)OCC 8266,c1(C(=O)OC)ccnc(-c2cccnc2)c1.C12CCCC(C1)C(=O)N2 8267,c1(C(=O)NCCN2CCN(C(CC3C(C)C3)=O)CC2)csc2c1CCCC2 8268,N1(C(C2(OC)CC(C)C2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8269,C(=O)(C(C)(C)C1CCCC1)NC(C)C=CC(=O)NCc1csnn1 8270,C1(CNC(CC2(C)CC2F)=O)C2CN(C(c3ccc(C(N)=O)nc3)=O)CC12 8271,N1(C(C2N(C(CC(C)O)=O)CCOC2C)=O)CCC2(CC1)CN(C)C2 8272,c1(OC)c(CC2CN(C(=O)C#CC3CC3)C2)cccc1Cl 8273,C1(C(N(CCCCCC)C)=O)CC(NC(=O)CC2C=NN(C)C2=O)C(O)C1 8274,c1(C(=O)NC(CCCCNC(COC(C)=O)=O)C)ccc(N)cc1C(C)C 8275,C1(CC(=O)N(CC(COC)C)C)CN(C(c2csnc2OC)=O)CCC1C 8276,C(=O)(CC(C)(C)C#N)NC(C(C(C)C)NC(=O)CCc1cccs1)C 8277,N1(C(C(C)(C)SC)=O)CC2(CCCN(C(=O)C(C)(C)SC)C2)C1 8278,N1(C(c2nnnn2C)Cc2c(OC)cccc2)CCCOC(C(C)C)C1 8279,C1(C(=O)NC2C(NC(=O)CCc3ncccn3)CCCC2)CCc2nc(O)[nH]c2C1 8280,C(=O)(CC(C)(C)CC(=O)NC(c1cc(C)ccc1OC(F)F)C)OCC 8281,N1(C(c2ncsc2C(F)(F)F)=O)CC2(CCN(C(C3(O)CC4CCC3C4)=O)C2)C1 8282,CC(C)C(O)CC(=O)NCC1CN(C(=O)CCNC(N)=O)CC1C(F)(F)F 8283,CC(C)CC(O)C(C)C(=O)N(C)CCOCCNC(=O)CCC[N+](=O)[O-] 8284,C(=O)(C#CC(C)(C)CNC(=O)C(C1CCOCC1)F)NC(c1c(C)nccc1)C 8285,N1(C(C=C(C)c2ccsc2)=O)CCCC(CCO)(C(=O)O)C1 8286,C1(CNC(CNC(C(CC)CC)=O)=O)CN(C(=O)CCN2CCC2)C2(CCC2)C1 8287,CC(C(=O)NC1C(C(N2CCN(C)CC2C)=O)CCCC1)C(C)(C)C 8288,C(=O)(CN=c1cc[nH]cc1)N1CC(C)C(C(N2CC[Si](C)(C)C2)=O)C1 8289,c1(CNC(=O)Nc2cccc(OCCN(C)C)c2)cc2cccnc2[nH]1 8290,Cc1cc(Br)cc(C(=O)NC2CC(NC(=O)CCS(C)=O)C2)c1F 8291,C1(C(=O)NC(C2CCN(C(=O)C(Br)=C(C)C)CC2)C)CC2(CC2)CO1 8292,Cc1onc(Br)c1C(=O)N(CCN(C)C)CC1CCNCC1 8293,N1(C(Cc2ncc(CC)[nH]2)=O)CCCC(C2CCN(C(=O)CC3CC3)CC2)C1 8294,N1(C(C2CCCC3(CCC3)C2)=O)CCCC2(C1)CN(C(=O)C(F)(F)C(F)(F)F)C2 8295,c1(C(C)C)ccc(NC2CC(n3cc(-c4c(Cl)cccc4Cl)nn3)C2)c(Br)c1 8296,C1(C(N2CC(CC)C(F)C2)=O)CCC(NCS(C)(=O)=O)CC1 8297,CC1CN(C)CCC1N(C(=O)CC1CC(NC(c2cc(O)ncn2)=O)C1)C 8298,CCCCCC(C)CC(=O)NC1CCN(C(c2cccc3c2CCC3)=O)C1(C)C 8299,C1(C(N2CC(C(N3CC(COC(C)=O)C3)=O)OCC2)=O)CC2(CCC2O)C1 8300,NC1CSC(CC(=O)NCc2ccccc2I)C1 8301,N1(C(C2(OCF)CCC2)=O)CCC(CC(N)=O)(Nc2ccnc(COC)n2)CC1 8302,c1(OCCC)cc(OC)cc(CC(=O)N(CCCNC(C2COC(C)C2)=O)C)c1 8303,c1(CNC(=O)NCC(C=C)(F)F)ccncc1-c1cccc(CC)c1 8304,c1(C(N(C)CC2CCCN2C(=O)CSc2cnc[nH]2)=O)ccc(CO)cn1 8305,CN1CCC2CN(C(C3CCN(Cc4nc(Br)cs4)CC3O)=O)CC12 8306,c1(CC(=O)NCCCCNC(C(C)NC(CC)=O)=O)ccccc1Br 8307,CCC(O)C(C)C(=O)NCCC1(OC)CN(C(C2CC2F)=O)C1 8308,CC1(C)Cc2[nH]nc(C(N3CCC(O)(CNC(=O)C(F)C4CCCC4)C3)=O)c2C1 8309,CCC(C(=O)NCCCCCN(C(=O)C(C)c1cccs1)C(C)C)C(C)C 8310,N1(C(c2ccn(COC)n2)=O)C(CC(=O)NCC2CNC(=O)CO2)C2CCCC12 8311,C1(C(N(CCC(=O)N(CC)Cc2ccnn2C)C)=O)CCCCC1C 8312,C1(CNC(c2cccc(CC)c2)c2nnnn2CC)CCCCCCN1 8313,n1(CC)cc(C(=O)NCCN(C(C2CC2C2CC2)=O)CC2CC2)c(C(F)(F)F)n1 8314,c1(C(N2CC(CNC(C3CN(C(C)=O)C3)=O)CC2(C)C)=O)c(F)ccc(N)c1F 8315,c1(C(=O)NCCCCCN(C(C(COCC)C)=O)C)cc(OC)n(C)n1 8316,Cc1cc(C(=O)NC2CC(CCNC(C3(O)CCC(C)CC3)=O)C2)nc(C)n1 8317,c1(C(N2C3C(CNC(c4cc[nH]c4)=O)CC(CC3)C2)=O)cc2n(n1)CC1(CC1)C2 8318,N(C(=NCC(=C)C)NCC(=O)NC(C)C)C(c1ccccc1)C#C 8319,C(=O)(C1OCCc2c(Br)cccc21)N(C)CC1(NC(c2cocn2)=O)CC1 8320,Cc1cc(C(=O)N(CCCNC(=O)CCC2CCCN(C)C2)C(C)C)cc(Cl)c1 8321,c1(C(N(CC(O)CNC(C2(O)CCOCC2)=O)C)=O)onc2ccccc12 8322,C1(CNC(COCCCC(C)C)=O)(NC(=O)C(F)n2cccn2)CCCCCC1 8323,Cc1cc(C(N(c2ncc(C)c(C)c2)C2CCNCC23CC3)=O)cnc1C 8324,N1(C(c2ccc(SC)o2)=O)CCC2(CC2NC(=O)CCCCOC(C)(C)C)C1 8325,N12CC3CC(CC3C1)NC(=O)c1nc(C)[nH]c1C2=O.C1(C)CC(F)C1(Cl)Cl.CC 8326,c1(NC2C(CCC)CN(C(=O)OC)C2)cc(Br)c(F)cc1F 8327,c1(C(N2CC(N(C(=O)C(c3ccc(Br)cc3)O)C)C2)=O)cc2c[nH]nc2s1 8328,c1(C(=O)NC2CCC(N(C(=O)CC34CCC(CC3)C4)C)C2)cnn2c1OCCC2 8329,CCC(=O)CCC(=O)N1CC=CC1(C)C(=O)NC1CNC(=O)C1(C)C 8330,C=CC1(CC(N2CCC(C)C2CNC(c2cc(C)cc(C)c2)=O)=O)CCCCC1 8331,C1(CNC(C(C)OCC#C)=O)COC(C)(C)CN1C(=O)C=Cc1ccnn1CC 8332,C1(NC(CN(C)C)=O)CC12CC(NC(c1cc(C(c3ccccc3)=O)cs1)=O)C2 8333,O=C1CCC(C(=O)NCC2(C(N)=O)CCN(C(=O)Cc3nnc(O)s3)C2)CN1 8334,Cc1ccc(Cl)cc1NC(=O)CC1CC(C)(C)CN1C(=O)C(C)N=[N+]=[N-] 8335,C1(C(N(CCNC(CC(C=C)C)=O)C2CC2)=O)CC1C1CCOCC1 8336,CCCC(C)(CCC)C(=O)NCc1nc(O)c(C)s1 8337,CC(CS(C)(=O)=O)NC(c1ccc(CNC(=O)CN(C)C(N)=O)nc1)=O 8338,c1(CC(=O)N(CCCNC(CCC)=O)CC2CCCC2)cnc2ncccn12 8339,C1(C2CCN(C(C3CC34CC(O)C4)=O)C2)(NC(CN(c2ccc(F)cc2)C)=O)CC1 8340,N1(C(C(CC)(C)O)=O)CC2(CC(C(=O)NCCCOC(=N)O)CO2)C1 8341,Cc1cc(=O)cc(CNC(C23CC(CNC(=O)C(O)C(C)C)(C2)C3)=O)[nH]1 8342,N1(C(c2cn(CCC)nc2C)=O)CCC(NC(c2cnncc2O)=O)CC1C 8343,CC(C)(C)C(C)(C)C(=O)NCC1(C(F)F)CCN(C(C2CNC(=O)C2)=O)C1 8344,c1(OC)ccc(NC(=O)CC2(NC(C3CNC(=O)C3)=O)CC2)cc1C 8345,c1(CNC2C=CC(C(=O)Nc3ncc(Br)nc3I)C2)ccc(Br)c2cccnc12 8346,Cc1cc(CC(=O)NC(C(=O)NCC=CCO)C2CCOC2)nn1C 8347,N1(C(c2cc(CNC(C3C(C)=CCS3)=O)ncc2)=O)CCC2(CNC(=O)C2)C1 8348,C1(NC(C(F)=CCC)=O)CCCCCN(C(=O)C(c2c(C)noc2C)C)C1 8349,CCCCCCCCCCCC(=O)NCC1CC(F)(CNC(=O)C=NOC)C1 8350,c1(COC)cc(C(=O)OCC(=O)NCCc2ccccc2)n[nH]1 8351,C1(N(C(CC(=O)NCC#C)=O)C)CCC2CN(C(=O)C(c3cccnc3)C)CC12 8352,c1(OC)cnc(C(N2CC(O)(C(=O)NCc3ccc(C)cc3OC)C2)=O)c(F)c1 8353,C(CCCCNC(=O)CC(C1CC1)NC(c1coc(SC)c1)=O)N(C)C 8354,C=CCC(CC=C)C(=O)NCC1COCC1NC(C12CCC(CC1)CO2)=O 8355,c1(NC(C(=O)NCCC(C)N)=O)cncc(N2C(=O)NCC2C)c1 8356,c1(C(=O)NCC2(CNC(C(COC)N(C)C)=O)CC2)ccc(C(C)=O)cc1C 8357,C1(NC(C2CCCCCC2)=O)C2CCCC1c1ccccc1C2 8358,C(=O)(C1CS(=O)(=O)c2ccccc21)NCC1N(C(C(CC)C#N)=O)CCCC1 8359,C1(=CCNC(C2CCCCO2)=O)CCN(C(c2cccnc2)=O)CC1 8360,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)Cn2nccc2N)C1 8361,C12(C(N3CCC(CC(C)NC(C(C4CC4)OC)=O)CC3)=O)CCC(CC1)CO2 8362,c1(C(N(C2CCC2C(=O)NC(C)(C)C)C)=O)csc(C2CCCO2)n1 8363,C(CCCCCC)=CC(=O)N(C(CCN(CCCCC)CCC)=O)C 8364,CC(C)CC(C)(O)c1cn(CC2CCCC2NC(=O)CN(C)C)nn1 8365,N#CC1(C(N2CCC(CNC(=O)Cc3nc(C4CC4)n[nH]3)CC2)=O)CCCOC1 8366,C1(NC(c2c(OCC)c(F)ccc2)C)CCNCC(C)(C)C1 8367,C(=O)(C1=CC2C=CC(C1)C2)N1CC(C)C(NC(c2ccc(SC(F)(F)F)nc2)=O)C1 8368,c1(C(N(C)CCN(C)C(C2CC3COCC3C2)=O)=O)cnc2[nH]c(O)nc2c1 8369,CCCC(C(O)C(=O)NCCC(C)C(F)F)NC(C1(c2cc[nH]n2)CC1)=O 8370,Cc1noc(N)c1C(=O)NCC(C)C(=O)NCc1cncc(F)c1 8371,c1(C(=O)NCCN(C(C)C)C2CC2)c(NC(=O)CC2CCOC2C)cccc1Cl 8372,N1(C(c2n(CC)ccc2)=O)CC(C(=O)NCc2nc(CC)cs2)C2(CC2)C1 8373,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8374,N1(CC)CCC(NC(=O)C(C)(C)NC(c2cn(C3CC3)cn2)=O)CC1 8375,C(=O)(CS(=O)(=O)CCOCCCNCCOCCNC(C(C(CC)C)=O)=O)NC 8376,N1(C(CCCCCC)=O)CC(NC(=O)C(C)Oc2ccccc2)C(O)C1 8377,N1(C(c2c(CC)noc2)=O)CCC(O)(C(C)NC(=O)CN(C2CCC2)C)CC1 8378,C1(CNC(C2CC(F)(F)C2O)=O)CCN(C(=O)CC2(O)CCC2)CC1 8379,C1(NC(C(C)CF)=O)CCCN(C(c2ccc(CNS(C)(=O)=O)o2)=O)C1C 8380,C1(CNC(c2ccc(C(F)F)nc2)=O)CC2(CC2)CN1C(C1CCCOC1)=O 8381,Cc1cc(S(=O)(=O)N2CC(N3C(=O)CCC3=O)C2)sc1C 8382,CCCCCC(F)C(=O)NC(COCC)C(=O)NC(C)COC 8383,C(=O)(CC(C)P(C)(C)=O)N1C(CN(C)C(C2(N3CCCCC3=O)CC2)=O)CCC1 8384,O=S(=O)(NCc1ccccc1F)N1CCC(c2ncc(Cl)cn2)CC1 8385,N1(C(C2(CCOC)CCCC2)=O)CC(NC(=O)CCC2CCCN(C)C2)C(C)C1 8386,c1(C(N2CCCC(F)(CNC(c3nncs3)=O)C2)=O)ccc2ccoc2c1 8387,c1(C(=O)NC(CNC(C2C(C)C2(F)F)=O)(C)C2CC2)cncc(-n2cccc2)c1 8388,N1(C(c2c(OC)ccs2)=O)CC2CN(C(=O)C(=Cc3ccccn3)C)CC2C1 8389,c1(C2(C(=O)NC(C(=O)NC(C)C(C)n3cncn3)C3CCC3)CC2)ccccc1 8390,N1(C(C2CC(C)N(C(=O)OC(C)(C)C)C2)=O)CCCC2(C)CCCCC12 8391,c1(C(N2C(C)CC(CNC(c3cc(C)cc(O)c3)=O)C2)=O)ccc2nnnn2c1 8392,C1(CC)C(C(=O)NCCC2CN(C(c3ccc(C(C)C)cn3)=O)C2)CCN1C 8393,Cc1ccc(CC(=O)NCc2nc(C(F)F)no2)o1 8394,C1(CN2CC(C(=O)NC(CN(C(C3C(=C)CC3)=O)C)C)C2)CCCCC1 8395,CC#CCCCC(=O)N(C1CCN(C(=O)C(C)C2(O)CCC2)C1)CC 8396,C(CCCCN=c1[nH]c(=N)[nH]c(=NC2CC2C)[nH]1)N(C)C.C(C(F)(F)F)N 8397,C(=O)(C#CC1CCC1)NC(C1CCN(C(C23COC(C2)C3)=O)C1)C 8398,C1(CC)(OC)CN(C(C2(C)CN(C(=O)CCC3CCCO3)C2)=O)C1 8399,c1(C(=O)NCC(C)NC(=O)Cc2cncs2)cc(Cl)ccc1OCC(N)=O 8400,N1(C(CCCSC)=O)CC2(CCC2)CC1CNC(C1CCCCC1N=[N+]=[N-])=O 8401,N1(C(c2cc(CC)nc(O)c2)=O)CCC2(CNC(=O)C(=O)N(C)C)CCCCC12 8402,c1(C(=O)OC)ccc(C(=O)NC(C)C(C)NC(c2c(F)cncc2Br)=O)cc1O 8403,C1(C(N(CC(C)NC(=O)CCSC(F)(F)F)C)=O)CCC2(CCCC2)C1 8404,Cc1cc(C(=O)NC2(CNC(=O)C(C3CCCCCC3)O)CC2)oc1C 8405,N1(CCNC(=O)Nc2c(C)nn(-c3ccncc3)c2)CCc2ccncc2C1 8406,C1(O)(C(=O)NCC2(CCNC(c3ccc(-c4ccco4)s3)=O)CCC2)CCOC1 8407,C1(NC(c2c(C)oc(Cl)n2)=O)C2CCC1CN(C(c1ccc3nccn3n1)=O)C2 8408,N1(Cc2cnc(CCCC)s2)CC2CN(C(c3sccc3OC)=O)CC2C1 8409,C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2)N(C)C)(CC)CC1(F)F 8410,Nc1cnc(Cl)cc1C(=O)NCCC1(NC(=O)COC2CCCC2)CCC1 8411,c1(C(N(C(CNC(C(C)=C2CC2)=O)C)C)=O)c(O)ncc(Br)c1C 8412,c1(CNC(=O)CCC2CCC(N3CCCC3)C2)ccc2oc(O)nc2c1 8413,C1(C)(C(=O)NC(c2ccc(Cl)s2)CC)CCCN(Cc2cc(SC)oc2C)C1 8414,C1=CCC2(CCN(c3ncnc(-c4ccccc4)n3)C2)CCC1 8415,N12CCc3cc(ccc31)NCCC2.N1(C)CCC(c2nc[nH]n2)C1.CO 8416,C1(NC(C(C)CO)=O)(CO)CCN(C(=O)COCCCF)C1 8417,N1(C2CC(N(C)C(=O)OC(C)(C)C)C2)CC2CC2C1C(=O)OCCOC 8418,Cc1ccc2c(=NC3COC3C)[nH]c(=NCc3cc(Cl)c(Cl)cc3C)[nH]c2c1 8419,N1(C(C(CCN(C)C)O)=O)CC2CC(C(N(C)Cc3cccc(CO)c3)=O)C1C2 8420,C(CCCCC(=O)NC12CCCC1OCC2)N(C(=O)CC1CCCCC1)C 8421,CC(C)CC(C(=O)N1CC[Si](C)(C)C1)N(C(=O)CC(C)(C)C1CC1)C 8422,C1(NC(=O)NCCC(C)CCN(C)C)CC2CCCC(C1)N2C(=O)OC(C)(C)C 8423,C(=O)(CC(CC)NC(C1CC2C=CC1O2)=O)NCC1(SCC)CC1 8424,Cc1c(C(N2CC(O)CC2CNC(C2CC2C(F)(F)F)=O)=O)c(Cl)nn1C 8425,N1(C(C2C(NC(C(C)CC(F)F)=O)CC=CC2)=O)CC(C)(C)OCC1C 8426,C(=O)(CP(C)(C)=O)N1C(CC(=O)NC(CC)CNC(C)=O)CCC1 8427,N1(C(C2CC(OC)C2)=O)CCOCC1CNC(C1(CO)CCOCC1)=O 8428,N1(C(C(C)CF)=O)CCC2C(CCCN2C(c2ccc(OC(F)F)cc2Cl)=O)C1 8429,c12coc(n1)NC1CC1NC2=O.c1(NC(CN(C)CC)=O)ccccc1 8430,c1(CN(C2CC2c2ccccc2)CC2CCC(C(=O)OCC)C2)cc(Br)ccn1 8431,C=CC(CC(=O)NC(COC)CO)c1ccco1 8432,c1(C(=O)NC)cccc2c1CN(C(=O)CN1CCN(S(C)(=O)=O)CC1)CC2 8433,Cc1cc([N+](=O)[O-])ccc1NC1CCCC(NC(=O)C(F)C(C)(C)O)C1 8434,C(=O)(CCC(C)(C)N(C)C)NC(C1CCN(C(C2C(C(C)C)C2)=O)C1)(C)C 8435,N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CC(F)C2)=O)CCC2(CCN(C)C2)C1 8436,c1(CNC(CCOCC)C2CC2)ccc(OC)c(C)c1Cl.c12nnnn1C2C1CC1 8437,Cc1cc(N2CCC(NC(c3cn(CCO)nn3)=O)C2(C)C)ncc1C#N 8438,C1(C(=O)NC(C(=O)NC(C#C)C(C)C)(C)C)CN(C)CCN1C 8439,N1(S(C)(=O)=O)CCCC1NC(=O)C(Cc1cn[nH]c1)NC(=O)CCn1cccn1 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8655,C12(C(=O)NC3(C)CCN(c4cc(CC)ncn4)C3)CCC(C(F)F)(CC1)CC2 8656,c1(C(N2CCC(C3CC3)(NC(CCCC)=O)C2)=O)cnc2ncnn2c1C(C)C 8657,O=S(=O)(c1c(C2CC2)cccc1Cl)N1CCOCC1.C12(CCOCC1)CS(=O)(=O)N2 8658,N1(C(c2c(C(C)C)cnn2C)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)C(C)(C)C1 8659,c1(CN2C(CN3CCN(CCC)CC3)CC3(CC3)C2)cc(OC)c(O)c(Br)c1 8660,c1(OC)ccc(C(=O)NC(C)CC(C)NC(=O)Cc2cnc(C)o2)cc1C(F)F 8661,N1(C(c2c(C)scn2)=O)CCC2(NC(c3cnco3)=O)CCCCCC12 8662,N(C(=NCCNCc1ccc(CO)cc1)NCS)c1ccc(OCC)s1.C(C)(C)(C)O 8663,C1(NC(c2c(C)nco2)=O)CCCCC1NC(c1ccccc1NC(=O)N(C)C)=O 8664,N1(C(=O)NCCC(=O)OCC)CCC2CN(C(=O)Nc3ccc(F)c(Cl)c3)CC12 8665,C12(NC(=O)Cn3cnc(Br)n3)CC(C1)N(C(=O)CC(=O)NC1CC1)C2 8666,C1(NC(C2(C(=O)NC)CCC2)=O)CC2CC(C1)N(C(=O)Cn1cc(Cl)c(C)n1)C2 8667,c1(-n2cc(C(N(CC(O)CNC(C3CC(C#N)C3)=O)C)=O)nn2)ccccc1Cl 8668,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8669,C1(NC(CN(C)CCO)=O)CN(C(C2CCN(C)C2=O)=O)CCC12CCC2 8670,C1(C2CCCN(C(C34CC(CN3C3CC3)C4)=O)C2)(NC(CN(C)C)=O)CC1 8671,c1(-c2ccc(OC)cc2)ccc(=NCc2ccc(COC(C)C)cc2)[nH]c1 8672,c1(OCC=C)ccccc1CNC(C1C2CC1N(C(=O)CN1CCSCC1)C2)=O 8673,c1(OC)ccc(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)nc1N 8674,C=C1CCC(C(N2CCCCC2C(=O)NCC2=COCCO2)=O)CC1 8675,C12CC(C1)CC(=O)N2.C(CC(C)(C)C1CCCO1)N(C(CC=C(C)C)=O)C1CC1 8676,C1(C(=O)NCCCCCN(C(CN(CCC)C)=O)C)CC2CCC(C1)O2 8677,N1(C(CC2C=CC(NC(C3CCN(C)C3=O)=O)C2)=O)CCC2(CCCCO2)C1 8678,c1(N2CCN(C(C(=O)NCC)CC3CCCO3)CC2)ccc2ccccc2c1 8679,N1(C(CC(C)(C)n2cc(SC(C)Cn3ccnc3)nn2)=O)Cc2ccccc2C1 8680,c1(NC(C2CC(F)(F)CN2C(c2cccc(O)n2)=O)=O)cc(C(F)(F)F)cnc1Br 8681,C(=O)(C1=C(C)OCC1)N(CC(C)NC(C1(c2cncnc2)CC1)=O)CC 8682,CC(N=c1cccc(S(=O)(=O)NCC23CCCC2C3)[nH]1)c1cccnc1 8683,c1(N2CCCC(CC=C)(NC(C3(C#N)CCCO3)=O)C2)nc(Cl)nc2sccc12 8684,N1(C2c3c(Br)ccc(c3)NC2=O)CCc2cc(F)cc(F)c2C1.C1(CSC)CC1 8685,N1(C(C(n2ccc(C)n2)(C)C)=O)CCN(C(c2cn(C)nn2)=O)CC2(CC2)C1 8686,C(CN=c1[nH]c2c(cc1C#N)C(=O)CCC2)(C1CCCCC1)NC(C(C=C)C)=O 8687,c1(C(=O)NCC23CN(C(c4n(C)nnc4)=O)C(CC2)C3)c(S(C)(=O)=O)cnn1C 8688,N1(CCn2cc(C(=O)OC(C)C(=O)NC3(C)CCCCC3)nn2)CCS(=O)(=O)CC1 8689,c1(C(C)C)noc(CCC(=O)NC2CCCC2NC(C2(CF)CC2)=O)n1 8690,N1(C(C(F)=CCC)=O)CC2CC(C1)CN(C(C1CC(=O)N(c3cn[nH]c3)C1)=O)C2 8691,C(N=c1nc2ncn(C)c2c(NCC2(CO)CCCO2)[nH]1)c1nnn(CC)n1 8692,c1(NC(CC(CNC(CSCC#C)=O)C)=O)cn(C)c(C)cc1=O 8693,c1(C(N2CC3CCN(C(C(CC)C#N)=O)CC3C2)=O)cc2c(nn1)c(C)nn2C 8694,C(=O)(C1CCc2c[nH]nc21)NCCCOCCN(C)C(C1CC1(Cl)Cl)=O 8695,c1(C(N2CCN(C(COCC)=O)C(CO)C2)=O)cc2cc(Br)ccc2c(=O)o1 8696,C1(C(N(C)CC)=O)CCCN(C(=O)Cn2cc(Cc3cnn(C)c3)nn2)C1CC 8697,c1(C(=O)NCCN(C(=O)CCOC(C)CC(C)C)CC)ncoc1C1CCCCC1 8698,C1(NC(=O)CSC(F)(F)F)COC2(CCN(C(C3CC34CCSCC4)=O)CC2)C1 8699,CC(C)C(O)C(=O)NCC(C1CCCCN1C(=O)CS(=O)(=O)N(C)C)(C)O 8700,Cc1ccc(F)c(C(=O)NCC(C)CN(C)C(C23CCC(C2)OC3C)=O)c1 8701,c1(C(=O)NC2C(NC(c3nc(C(C)(C)C)oc3)=O)CC2)ccc(OCCF)cc1Cl 8702,c1(NC(C)=O)ccc(C(=O)NCc2cnn[nH]2)cc1.C12(CC1)C(=O)N2 8703,Cc1nc(O)c(Br)cc1C(=O)NCCC(C)NC(=O)Cc1ccc(O)nc1 8704,C1(=O)C(F)(CC)C(=O)c2coc(c2CCCCOC)C(=O)NCCN1CC 8705,c1(SC)ccc(C(=O)NCC(C(C)C)NC(=O)CCc2cn(C)cn2)c(Cl)c1 8706,N1(C(=O)NCc2ncc(C(C)(F)F)cn2)CCOC(C2(C)N=N2)C1 8707,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(C1(C(N)=O)CC1)=O 8708,N1(C(CCCOC)=O)CC=C(CNC(=O)CCC2(C)CC2)CC1 8709,c1(NC2CCN(C(C(C)=C(CC)C)=O)CC2CO)c(Cl)cccc1[N+](=O)[O-] 8710,c1(SC)nc(=N)[nH]c(=NCC(C)n2cnc(C(C34CCC(C)(CC3)CO4)=O)c2)[nH]1 8711,Cc1sncc1C(=O)NC1(C(=O)NCc2noc(C(N)=O)n2)CC(CO)C1 8712,N1(C(C2(CNC(C3CN(CC)C(=O)C3)=O)CCC2)=O)CC2(C1)NC(=O)NC2=O 8713,c1(C(=O)NCCNC(C(C)(O)Cn2ccccc2=O)=O)ccc2c(c1)CCCO2 8714,Cc1nnccc1C(=O)N(C)CC1CCCN(C(C2CC(C)(C)O2)=O)C1 8715,c1(C(=O)NCc2cccc(CNC(=O)C3=COCC3)c2)nsc2c(Cl)cccc12 8716,C1(C(=O)NC2C(C)(COC)C2)COCCN1C(C12CC1C2)=O 8717,c1(CCC(=O)NC(C(C)C)CNC(C2CN(S(C)(=O)=O)C2)=O)ccc(Cl)nc1 8718,c1(NC(C(COC)Oc2ccccc2Cl)=O)cc(Cl)nn(C)c1=O 8719,Cc1ccnc(CCC(=O)N(CC(O)CNC(=O)C(F)(F)c2cscn2)C)c1 8720,C(=O)(C1=NNC(=O)CC1)NCCN(C(Cn1c(C)ncc1)=O)Cc1ccccc1 8721,N1(CC(=O)N(C)Cc2ncc[nH]2)CCC(C2CCCO2)CC1 8722,CCC(CC(F)F)C(=O)NCC(C)CNC(c1c[nH]c(=N)o1)=O 8723,CC(O)CCCCCC(=O)N1CCC(n2cc(C3(F)CCCCC3)nn2)C(C)C1 8724,CC(C)CCC(N)C(=O)NC1(c2ccc(I)cc2)COC1 8725,C#CCCC(O)C(=O)N1CCCC1C(C)NC(=O)CCc1cncn1C 8726,C1(NC(C(C(C)C)=O)=O)CN(C(c2ccc(C(N)=O)cc2)=O)CCC1(F)F 8727,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8728,C1(c2scc(C)n2)CN(C(c2cnn(CCC3CCOCC3)c2N)=O)CCO1 8729,C(=O)(CC1=CCCC1)NCCCOCCN(C)C(c1ccc(SCC#N)cc1)=O 8730,C1(CC)(CNC(C2OCCC2CNC(=O)CC2(N(C)C)CC2)=O)CCCO1 8731,CC(C)(C)C(O)CCNC(=O)C(C)(O)Cn1cc(Br)cn1 8732,C(=O)(C1Cc2ccccc21)NC1CCCN(C(c2nnc(CC)o2)C)CC1 8733,C1(N(C)C(C2CC(C)(F)C2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 8734,CN1CCCCC1CC(N1CC(CO)(NC(=O)CCc2ccccc2)C1)=O 8735,C1(NC(NCc2cc(C)on2)=NCc2ccccc2C2CC2)CC(C)OC(C)C1 8736,c1(C(N(CCC)CCNC(C2(C)CCN(C)C2=O)=O)=O)c(Cl)ccc(O)c1N 8737,Cc1cc(F)cc2c1N(C(=O)N(CCC#CCO)CCC(C)(C)C#N)CC2 8738,Cc1ccn(C(C)(C)C(=O)NC(C)CCNC(C2CC(OC(F)(F)F)C2)=O)n1 8739,c1(C(=O)NCCN(CCOC)C(C2(C)CCCCO2)=O)nc(C)ccc1OC 8740,c1(C(=O)NC(C2C(C(N(C3C(C)C3)C)=O)OCC2)=O)cccc(F)c1O 8741,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8742,C(CC(C)CCNC(C1CNC(=O)N1)=O)NC(C=CSC)=O 8743,c1(CC(=O)NC2(CNC(C(C)NC=O)=O)CCOC2)cn2ccccc2n1 8744,C1(C(N(C2CCCN(C(=O)CN(C3CCC3)C)C2)C)=O)CCC2(CCC2)C1 8745,C(=O)(C1SCCc2ccccc21)N1CC(CNC(C(C)(C)F)=O)CC1(C)C 8746,C1(N(C(=O)CCCc2ccsc2)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8747,C(=O)(C(C)(CNC(=O)NC(c1nc(CO)cs1)(C)C)c1ccc(Cl)cc1)OC 8748,c1(C(=O)NC(C)CNC(C2COC(=O)N2C)=O)cc2c(cc1O)CCCC2 8749,CC(C)C(O)C(C)C(=O)NC(C)(C)CC(=O)NC12CCC(C1)OC2C 8750,CN1CCNNS(=O)(=O)c2cc(OC(F)F)ccc2CC1 8751,c1(C(N(CC(=O)NC(C(N)=O)C2CC2)CCC)=O)ccc(N)cn1 8752,C12(CCCOC1)C(=O)N2.Cn1nnnc1C(=O)NC1CCCC1C(=O)OC(C)(C)C 8753,N1(C(CC)C(=O)OC(C)(C)C)CCN(C(=O)NCC2(C)CCCC2O)CC1 8754,c1(C(=O)NC(C2OCCN(C(C(C=C)CC)=O)C2)C)cc(N)cc(F)c1 8755,Cc1ncc(NC(=O)CCC2CCCCN(C(=O)CSC(C)(C)C)C2)c(C)c1C 8756,c1(C(=O)NC2C(C)CN(C(=O)C3=CCSC3)C2)cccc2cnccc12 8757,c1(C(=O)NCCOCCOCCNC(C2(O)CCOC2)=O)ccc2c(c1)CCO2 8758,C1(CNC(c2n(CC)c(O)nc2)=O)CN(C(C2CCCCC2)=O)CC2(CCC2)O1 8759,c1(C(=O)NC2(CCNC(CN(C(C)=O)C)=O)CC2)cccc2ccn(C)c12 8760,N1(C(C=CCC)=O)CCCCC(COCC)C1.c12csc(n1)CNC2=O 8761,c1(NC(c2c(C(=O)Nc3c(C)cnc(Cl)c3)cccn2)=O)ccc2ncccc2c1 8762,C(=O)(C#CC1CCCOC1)NC1CCC(CN=c2nc(C)[nH]s2)C1 8763,C1(N2C(=O)CC3(CC3)N(C3CCCCC3)C2=O)CCC2CC12.c1(S)cccs1 8764,c1(NC(C2N(C(c3ccc(CC)s3)=O)C3C(C2)C3)=O)nc2cncnc2s1 8765,Cc1nc(C2CCN(CCSc3ccccc3)CC2)nc2c1CCCC2 8766,C1(C(=O)NCc2n(CC#C)cnn2)CCCN(C(=O)CCNC(C)=O)C1 8767,Cc1onc(CN2CC(C)C2)c1C(=O)NCC1CCN1C(C1CC(C)(C(C)C)C1)=O 8768,C1(CC(=O)N(CC(C)O)CCNC(c2c(C)cn(C)c2)=O)CCC2(CCC2)O1 8769,C1(C(C)(C)C)CCCC(CNC(=O)Nc2cc(C3CCOCC3)nn2C)C1 8770,C(=O)(C1Cc2c(Cl)cccc21)NCCN(C)C(c1cnc(CCC(F)(F)F)s1)=O 8771,c1(C(N2CC(CNC(=O)CSCC(F)F)C(O)C2)=O)ccnc2ccsc12 8772,c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)nc(C)c(C)nc1C 8773,N1(C(CCC(C)SC)=O)CCC(CNC(=O)CC2COC(=O)C2)CC1C 8774,CC(C)CC(C)(CO)NC(=O)C(C)CNC(c1occc1C(C)C)=O 8775,N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2(F)CCCC2)=O)CC1C1CCC1 8776,N1(C(c2n(CC)nnc2)=O)CCC(C)C1CNC(=O)CS(=O)(=O)N(C)C 8777,c1(C(=O)NCCCCOCC)ccc2[nH]nc(Cl)c2c1 8778,N1(C(C(COC)C)=O)CCC(CC(=O)NC2CCCN(CCO)C2)CC1 8779,c12cc(cc(Br)c1)OC2.C1(C(=O)NCC(O)Cc2ccccc2)CC(O)CN1 8780,c1(C(C(=O)NC(C)(C)CC)N(CCC#C)C2CC2)cnc(C)nc1 8781,C12(C(=O)NCCC)CCCC1(C(=O)N(C(C)CN(C(=O)CC1(O)CCC1)C)C)C2 8782,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8783,c1(C(N(C(CC(=O)NC(c2cncn2C)CC)C)C)=O)cccc(C)c1F 8784,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2)=O)cc2c(Cl)cccc2[nH]1 8785,C1(C(N2CCC(NC(CC(C)C3CCCCC3)=O)CC2)=O)CC2CCC(C1)C2F 8786,C(C(=O)NOC1CCCCC1)C1CC(CN(C(C(C)SC)=O)C)C1 8787,C(C1C(C(=O)N(C)CC2CCCN2C(=O)C(C2(O)CCCC2)F)C1(C)C)=C(C)C 8788,C(=O)(CC(C)CC(=O)OCC)N(CCCNC(=O)C#CC(C)(C)C1CC1)CC 8789,n1(CC)ccnc1C(F)(F)C(=O)NC1CC1CNC(=O)C(F)CSc1ccccc1 8790,c1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)cc(O)nc(Cl)c1 8791,C(C(=O)N1OC2CCC1CC2)(c1c(OC)c[nH]n1)NC(=O)C(C)C1CCOC1 8792,Cc1cccc(F)c1C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C.C12CC1C2 8793,C1(O)(C(C(=O)OCC)(F)F)CCN(CC(F)(F)CC)CC1 8794,c1(N(C)C(=O)Nc2csc(NC(=O)OC(C)(C)C)c2)ccc(C(F)(F)F)cc1 8795,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NCC(C=C)(C)C 8796,C1(C(N2CCN(C(CCC)=O)CC2CC(F)(F)F)=O)CCc2cnc(C)n2C1 8797,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8798,N1(C(CC(C(=C)C)O)=O)CCC2(CCC2)C(CNC(c2cc3c[nH]nc3s2)=O)C1 8799,c1(C(N2CCC(CNC(Cn3ncc(C)c3)=O)C(C)C2)=O)[nH]c2c(c1C)CCC2 8800,C=CC(C)(C)CC(=O)N1CCN(C(=O)Cc2ccc(Br)nc2)C2CC12 8801,c1(C(=O)NCCCN)cscc1C1CC1.C(=O)(CO)OC.C1C(=O)N1C(C)C 8802,C1(CN(C)C(c2cnn(CC(F)F)n2)=O)COCCN1C(=O)CC(Cl)Cl 8803,Cc1cc(C(=O)NCCN(C)C(c2cc(C(=O)C(C)C)c[nH]2)=O)nn1C(F)F 8804,c1(N(CCN(C(C)C)C(c2ccncc2Cl)=O)C)ncc2c(Br)cccc2n1 8805,Nc1nc(C(N2CCC(CNC(c3cc[nH]n3)=O)C(F)(F)C2)=O)ccc1[N+](=O)[O-] 8806,C(=O)(C(CC(C)C)NC(C)=O)NCC1C(C(=O)NCC(C(=O)OC)(F)F)OCC1 8807,c1(C(N2C(C(=O)NCCC34CC(CCO3)C4)CC2)=O)coc2ccccc12 8808,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8809,Cc1cc(C(N2CCCCC2CNC(c2cnoc2C)=O)=O)cc([N+](=O)[O-])c1Cl 8810,c1(OC)ccc2cc(C(=O)Nc3cccc(C(N4CCC4)=O)c3)c(O)nc2c1 8811,C1(C(C)(C)NC(C23CC(C2)C3)=O)CCN(C(=O)Cc2coc(C3CCCC3)n2)C1 8812,C(=O)(C1CSc2ccccc21)NCC1CCC(NC(C(C2CC2)OCC)=O)CC1 8813,c1(C(CNC(c2cnc(CC)s2)=O)NC(C2CCNC2=O)=O)ccc(F)cc1F 8814,n1(CC)ccc(CN(C)C)n1.N12CCC1C(=O)NC1(CC1)CC2=O 8815,Nc1cccn(CC(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)c1=O 8816,N1(C(c2c(COC)c[nH]c2)=O)CCN(C(c2n[nH]c3c2COC3)=O)CC1C 8817,C1(C(N(CCC(=O)N(CC(C)SC)C)CC#C)=O)CNC(=O)CC1C 8818,n1(CC)nnc(C(N2CCCCC2CNC(c2nc(C3CC3)cs2)=O)=O)c1C 8819,c1(CNc2c(OC)ccc(COCC)c2)c(C)cccc1C#N 8820,C(=O)(C(CC)C(C)O)N1CC(OC)(CNC(=O)Cc2ccccc2CC#N)C1 8821,CC1CN(C(c2ccc3snnc3c2)=O)CC(C)N(C(=O)Cc2cccn2C)C1 8822,C1(O)(CC(N2CC(C)(NC(CC3C(C)C3)=O)C2)=O)CCCN(C)C1 8823,CN1CCN(C(C2C=CC=CC=C2)=O)CC1C(N1CCC2CC12)=O 8824,C(=O)(CCCCC(N)=O)NC(CC(=O)NCc1c(C)ccnc1)CC1CC1 8825,C1(NC(C(CC)(C)OC)=O)(CNC(C2CCC2)=O)CCC(F)(F)CC1 8826,c1(C(N2CCN(C(c3[nH]cc(C#N)c3)=O)CC2CCO)=O)nccc2nn[nH]c12 8827,c1(C(N2C3C(C(=O)Nc4c(C)c(O)ccc4)C(C3)C2)=O)ccc(F)c(F)c1Cl 8828,C1(N(C(=O)C=Cc2ncc[nH]2)C)CCCN(C(C2CC3(CSC3)C2)=O)C1 8829,C1(NC(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(c3ccsc3)=O)C2C1 8830,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CCC(=O)OCC)C2COCC2O1 8831,C1(NC2CC(OCC)C2SC)CCCCCC1C 8832,c1(CN2CCC(C)(C(=O)NC(c3cnn(C4COC4)c3)C)C2)ccc(F)c(CO)c1 8833,c1(C(N2CC(NC(C=C(C)C(=O)O)=O)C(F)C2)=O)ccc2sccc2c1O 8834,C1(c2cn(CC3(CNC(C(C4CC4)OC)=O)CC3)nn2)COC(C)(C)C1 8835,C1(CNC(C(C)NC(=O)OC)=O)N(C(=O)CCCC(C)(F)F)CCCC1(C)C 8836,C1(N(CC(=O)N(C2(N(C(CSC3CC3)=O)C3CC3)CC2)C)C)CCCC1 8837,C1(C(=O)NC(CCCCCC)C)CCN(C(=O)CCC2CCC2)C(C)(C)C1 8838,c1(SCC(=O)NC2(CCO)CN(C(=O)CC3CCOCC3)C2)c[nH]nc1[N+](=O)[O-] 8839,c1(N)nc(=NCc2ccncc2)[nH]c2ccsc12.CCS(=O)(=O)c1ccccc1 8840,N1(C(C=CCOC)=O)CC(NC(=O)CC2(C)CCOCC2)C(c2ccccc2)C1 8841,C1(C(=O)OC)CCCC12CCCN(C(=O)CC1CCC(F)(F)CO1)C2 8842,C(C(C)(C)C#CC(=O)Nc1ccc(SCCF)cc1)NC(CCSC(C)(C)C)=O 8843,O=C1OC(C(=O)OCC2CCc3ccc(F)cc3O2)Cc2ccc(Cl)cc21 8844,Cc1ccc(C)c(CC(=O)NC(CNC(c2cncc(C)c2C)=O)C2CC2)c1 8845,c1(OC)c(C(N)=O)oc2ccccc12.N12C3CCC1C(C3)C(=O)N1CC(C1)C2=O 8846,N1(C(COCC(C)C)=O)CC(S(=O)(=O)N2CCN(C(C3CCCSC3)=O)CC2)C1 8847,C1(CCC(=O)NCC(CNC(c2n(C)ccn2)=O)O)CCCC(=O)N1 8848,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1C(C)=O)NCCC(C)(C(=O)OC)OC 8849,C(C(C(C)(C)C)NC(c1c[nH]nc1C1CCCO1)=O)NC(C=CCOC)=O 8850,c1(CCC(=O)NCCN(C)C(C2CC2(Br)Br)=O)cncnc1 8851,c1(C(N2C(C(N3CCCC(Br)C3)=O)CNCC2)=O)ccc(Br)c(O)c1 8852,C(=O)(C(CO)C(C)(C)C)N(CC(=O)NC1CC2(CCOC2)C1)C1CCC1 8853,N1(C(C(C)O)=O)CCC(C(=O)NCC)C1C(=O)NCCCCOCC#C 8854,CCCC(C(=O)NCCn1cc(C(N2CCC(N(C)C)CC2)=O)cn1)NC(N)=O 8855,N1(C(c2c(CC)cccc2)=O)CCC2(CCCCN(C(=O)C3CCCS3)C2)C1 8856,N1(C(c2cc(CC)nc(O)c2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2C1 8857,C1(CC(=O)N(C)CCNC(=O)CC2(C)CCC2)COCC1(C)C 8858,C1(C(=O)OC)CCN(C(=O)C2C3CC4C(C3NC(c3csnc3Cl)=O)C24)O1 8859,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8860,CC(C)(CCC(=O)N1CC(NC(c2ccc(Cl)c(Cl)c2O)=O)C1)[N+](=O)[O-] 8861,C=CCCCC(=O)NC1CC1CNC(=O)C(c1ccc(Br)cc1)SC 8862,C1(O)(CC(=O)NC(CNC(C(CCNC(C)=O)OC)=O)CCOC)CCCN(C)C1 8863,C(c1c(F)ccc(Cl)c1Cl)=CC(=O)N(C1CC1)CC1N(C(C(C)C#N)=O)CCC1 8864,c1(C(=O)NC(CNC(C=CC(CC)C)=O)(C)CO)cc(S(N)(=O)=O)c(C)cn1 8865,N1(C(CC(CC)OC)=O)CCOC2(CCN(C(=O)CS(=O)(=O)NC(C)C)CC2)C1 8866,C(=O)(CC(=O)NCc1nc(C(=O)N(C)Cc2cn(C)nn2)co1)NCC#C 8867,Cc1cncc(NC(=O)CNC(=O)CNC(=O)C(C)(C)N2CCCC2)n1 8868,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)c2Br)=O)C(CC)C1 8869,C(=O)(C1CCCn2ncnc21)N1C(C(=O)NC2CN(C(C)=O)C2)CC2COCC21 8870,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8871,C1(C(=O)NCC2(CCNC(C3CC4CC4C3)=O)CC2)CCC(F)(F)CO1 8872,C1(CC(C)C)CCN(C(c2cscc2Cl)C(=O)NC2CC2)CC1 8873,c1(CC(=O)N(CC(C)CNC(=O)CC2CCCN2C)C)cnccc1Cl 8874,C1(O)(CC=CC(=O)NCC(=C)CCNC(=O)C=Cc2cnc[nH]2)CCCOC1 8875,C1(F)(CNC(CC2CC(OCC)C2)=O)CCN(C(c2sc(C)nc2CC)=O)C1 8876,C(C1CN(C(=O)C(c2ccccc2)F)CC1C(=O)NCC1CNC(=O)C1)=CC 8877,C1(C)(C(=O)NCC2CN(C(c3c(C(C)C)ocn3)=O)CC2O)CCCCC1(F)F 8878,C1(C(=O)OC)C(CC(=O)NCC(O)CN(C(=O)Cn2cc(Cl)cn2)C(C)C)C1(C)C 8879,CC(C)(C)C(C)(C)C(=O)N1CCC(CF)(NC(=O)CC2CCC=CCC2)C1 8880,CC(C)CC(CNC(=O)CC1CNC(=O)C1)NC(C1(C)CCOCC1)=O 8881,c1(O)cccc(I)c1F.N1(C)CCC(NC(c2ccc(CCC(=O)OCC)[nH]2)=O)CC1 8882,N1(C(C(n2c(C)ccn2)C)=O)CC2C(C(=O)N(C3CCSCC3)C)C2C1 8883,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8884,N1(C(c2nc(CC(C)C)sc2)=O)CC2CCC1C(CNC(=O)C(CO)N(C)C)C2 8885,C1(O)(CNC(=O)COc2ccccc2Cl)CCN(C(c2cccc(O)n2)=O)CC1 8886,C1(C(=O)NC(C(NOCCC(C)C)=O)c2cccnc2)C2CCC(C2)C1C 8887,c1(C(=O)NC(C2CCOC2)C(=O)NCC2C(C)(C)CCCO2)cc2cccn2cn1 8888,C12CN(CC1C)C(=O)CCOCCCN(C)CCCCCNC2=O.CC.OC 8889,N1(C(C2(C(F)F)CC(=O)C2)=O)CCn2cccc2C1CC 8890,N1(C(C(C)n2cnnn2)=O)CCC(CNC(C2(Cn3cc(Cl)cn3)CC2)=O)C1 8891,c1(C(N2C(C3CCN(C(CCc4cnc(C)s4)=O)C3)CCC2)=O)ccccc1F 8892,C1(C(=O)NC(CNC(C[SH](c2ccccc2)CC#C)=O)C2CC2)CCC(C2CC2)CC1 8893,N1(C(=O)CSc2ccc(F)cc2)CCCC(N(CCO)C(c2cnco2)=O)C1 8894,c1(C(N(CCNC(C(c2c(Cl)cccc2Cl)C)=O)C)=O)coc2c1C(O)CCC2 8895,c1(C(=O)NC2CC3(CN(C(c4c(C)nc(C)o4)=O)C3)C2)cc(Cl)cc2c1CCC2 8896,c1(CCC(=O)NC(C)CN(C(=O)CCCOC(C)(C)C)C)c(Cl)cnn1C 8897,CCC(CC(F)F)C(=O)N(C1CCN(Cc2ccnc(-c3ccccc3)n2)C1)C 8898,c1(C(=O)NCc2csc(C(=O)NC(C(F)(F)F)C3CC3)c2)cnncc1O 8899,N1(C(C2(C)C(C)C2)=O)CCC2(CC1)CN(C(=O)CNC(C1CCCC1)=O)C2 8900,C(CC)(C(C)(F)F)N(C(CC(C)OC)=O)C.C1=CCNC1=O 8901,C(CC(O)C(F)(F)F)CN(C(C(CCN(C)C)NC(C(Br)=C(C)C)=O)=O)C 8902,c1(CC(N2CC(C)CC(NC(C=CC(C)C)=O)C2)=O)ccc([N+](=O)[O-])cc1 8903,C1(C(=O)NCCC2(CNC(C(C)C3CCC3)=O)CC2)CC(=O)c2ccccc2O1 8904,C1(C(=O)NC(c2n[nH]c(=N)s2)C2N(C(CC)=O)CC2)CC12CC(C)(C)C2 8905,c1(CN2CC3(C(C(=O)NC(C)CO)C3)C2)cc(Br)ccc1O 8906,C1(C(N2CC(N(C(c3c(OC)c[nH]n3)=O)C)C3(C2)CC3)=O)CC=C(C(C)C)CC1 8907,N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(=O)C(O)C2CC2)CC1CO 8908,c1(C(=O)NCCCN(C(=O)CN(C)C(N)=O)CCC)c(C)c(C)cc(C)c1C 8909,N1(C(CSCC#C)=O)CCC(CC(=O)NCC2CCCCO2)C1 8910,N1(C(C2=CCN(C(CC3(OCC)CCC3)=O)C2)=O)CC2CCCC2(CO)C1 8911,N1(C(C(COC)O)=O)CC2CCC(C1)N2C(=O)C(C1CCCN(C)C1)(C)C 8912,Cc1cc(=O)ccn1CC(=O)NCC1C2CN(C(c3cc(=O)n(C)cn3)=O)CC12 8913,C(C)(CCCCCO)NC(C1C(NC(CC2ON=C(CC)C2)=O)C1)=O 8914,C12(C(=O)NC3C(NC(C=C(C)c4cccs4)=O)CCC3)CCN(CC1)S(=O)(=O)C2 8915,N1(C(C(c2cncc(OC)c2)(F)F)=O)CC2CC(NC(c3cnnn3C)=O)CC1C2 8916,C(=O)(CCCC(F)(F)F)NCC(C)(C)NC(c1ccc(N)c(F)c1F)=O 8917,CCC(C)C(C(=O)NC1CCOCC1NC(=O)CC1CC(OC)C1)N(C)C 8918,Cc1[nH]nc2ncc(C(=O)NCC3(F)CCC(NC(c4nncs4)=O)C3)cc12 8919,N1(C(C(C)NS(CCC)(=O)=O)=O)CCC2CCC12CNC(=O)CNC(=O)C1CC1 8920,CC1(C)CC(CNC(C2CCN(C3CCC3)CC2)=O)CN1C(=O)CCS(N)(=O)=O 8921,c1(C(c2n(CC=C)nnn2)NC(c2csnn2)C)cccc(S(N)(=O)=O)c1 8922,C1(NC(c2ncn(CC)n2)=O)COCCC1C(=O)N(C)CCOC 8923,c1(C(=O)NCC2(F)CC(NC(c3c[nH]nc3F)=O)C2)ccc([N+](=O)[O-])cn1 8924,c1(C(=O)NC2CN(C(C=CCC)=O)C(CC)(CC)C2)cc(Cl)cc(Cl)c1OC 8925,CC1CCN(C(C2CC23CCCC3)=O)C1CNC(=O)CSc1cccc(F)c1 8926,CC(F)(F)CC(=O)NCC1CC1CNC(c1cnc(Cl)[nH]1)=O 8927,C1(C(=O)NCc2ccc(CC)nc2)CC(O)CCN1Cc1ccnc(F)c1 8928,CC(CO)CCCNC(c1cc(CCNC(C2(n3ccnn3)CC2)=O)on1)=O 8929,c1(OC)cccc(C(N2CCC(c3ccc(OCC(N)=O)cc3)C2)=O)c1Br 8930,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8931,C1(CC(N2CCC(NC(c3cc4occc4s3)=O)(CO)C2)=O)CCS(=O)(=O)CC1 8932,C1(NC(=O)NC(CC(=C)Cl)CO)CCOC2(CCCC2)C1 8933,c1(C(C)(C)C)ccc(COC(c2cnc(-c3ccccc3)[nH]2)=O)cc1F 8934,c1(CCC(=O)OCC(CC(=O)OC(C)(C)C)(C)CO)ccc(F)cc1C(F)(F)F 8935,CC1(c2ccccc2)CCCN1C(=O)Cc1cccc(OCC(F)(F)F)c1 8936,C1(N(C(C(n2ccc(C)n2)C)=O)C)CN(C(C2CC(N3CCCC3)C2)=O)CC1(C)C 8937,C1(NC(C(C)NS(C)(=O)=O)=O)CN(C(=O)COCC2CC2)CCN1C(C)=O 8938,C=CC(C)(CC)C(=O)NCc1cnn(C)c1C(=O)NCc1cc(O)cc(F)c1 8939,C(=O)(C(C)C(O)C(C)CC)NC1(C)CCN(C(C2(C#C)CCCCC2)=O)C1 8940,c1(CC)ccc(OC)cc1C(=O)NC1CN(C(=O)C2CC2)CC1O.C(=O)(CC#N)N 8941,C(=O)(CC1OCc2ncccc21)N(C)CC1C2CN(C(=O)COC(F)(F)F)CC12 8942,C1(NC(C2CC2Br)=O)(CO)CCCN(C(c2ccc(Cl)cc2)=O)C1 8943,Cc1ncc(Cl)cc1C(N1CCCC(CCC(=O)NC(c2cn[nH]c2)C)C1)=O 8944,C1(C)(NCC2C(CC(=O)C=O)C2)CCN(C(=O)CC(C)(C)C2CC2)C1.CCO 8945,c1(CC(CC)O)nc(SC)nn1Cc1ccc(Cl)cc1 8946,C1(NC(CCN(CCC)C)=O)COC2(CNC(c3ccns3)=O)CC1C2 8947,Cn1nccc1C=CC(=O)NCC1CCC(C(=O)NC(C)(CO)CO)O1 8948,C1(C(=O)NCC(C)NC(C2CC(CCC)C2)=O)(NCC)CCOC1 8949,CC(=O)CCCC(C)C(=O)N1CCC(C(N2CC3C(C(N)=O)C3C2)=O)C(O)C1 8950,C1(c2onc(-c3occ(C)c3)n2)CCN(CC(F)(F)F)C2(CC2)C1 8951,C1(COC)CN(C(=O)CNC(=O)CC2CCCC(=O)C2)CCN1C(=O)C(C)(C)C 8952,CCC(CC(=O)NCC(CNC(c1nc(C)sc1N)=O)OC)c1ccccc1 8953,C(=O)(CCS(=O)(=O)C1CCCC1)NCCOCCOCCOCCC#C 8954,C1(CNC(CSCC)=O)CCN(C(=O)CCn2cc(Br)c(C)n2)C12CC2 8955,Cc1nc2ncccc2cc1C(=O)NCC(O)CN(C)C(c1nsnc1O)=O 8956,c1(OC)ccc2[nH]c(C(N3CCC(CCNC(C4C=CCCC4)=O)C3)=O)cc2c1 8957,Cc1coc(C(=O)NC2C=CC(CC(=O)N(C(C)CC3CC3)C)C2)c1 8958,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 8959,c1(CN(C)C(C2(CO)CC2)=O)c(Cl)nn(C)c1Cl 8960,C1(NC(c2ccc(OC)s2)=O)CC2CCCC(C1)N2C(C1(C)COC1)=O 8961,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 8962,C#CCCCCCCC(=O)NC1CC1CNC(=O)CCc1c(Cl)cccc1Cl 8963,C1(C(=O)OCc2ccc(C)cn2)CC2CCCN2C(=O)N1 8964,N1(C(C(C)(C)OC)=O)CCC2CCC(NC(C3CCC4(CC4)C3)=O)C2C1 8965,c1(C(N(CC(CNC(c2ncc(C)cc2C)=O)O)C)=O)ccnc2ncccc12 8966,C1(CC(=O)NCCC(C(C)C)NC(=O)CCC2CCCCC2)NC(=O)CNC1=O 8967,C(C)(CN=C(NCC1C2CCCCC12)Nc1ccccc1)OCCOC 8968,c1(C(N2CC(CN(C(CCNC(C)=O)=O)C)C2)=O)cnc2cc(Br)ccn12 8969,c1(C(=O)NC2CN(C(Cc3ccc(OCC)nc3)=O)C2)oc(S(N)(=O)=O)cc1C 8970,C1(C(=O)NC2C(C)(C)C(=O)NC2)CCN(C(=O)C(C)(C)C2CCCC2)O1 8971,Cc1nc2cc(C(=O)NC3CC(NC(c4ccc(Cn5cccn5)o4)=O)C3)sc2s1 8972,c1(OCC=C)ccc(Cl)c(C(=O)N(C(C)CNC(C2(O)CC=CC2)=O)C)n1 8973,c1(NC2CC(O)(CNC(CN(C(COC)=O)C)=O)C2)nc(C)ccc1O 8974,C1(C(=O)NC(C(=O)NC(CN(C(C)C)C)C)Cn2cncn2)CCCSC1C 8975,c12ccc(cc1)OCC(=O)N1CC(F)(C1)CNC2C.C1(C(=O)NC)CS(=O)(=O)C1 8976,C(CC(O)CNC(C1CC(NC(=O)OC)C1)=O)NC(C1(C=C)CC1)=O 8977,C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(=O)Cc2cnccn2)CCC1C 8978,N1(C(CC2C(C)CC2)=O)CC(NC(=O)COCC2CCCC2)C(F)C1 8979,c1(C(N2CCC(C3N(C(COC)=O)CC3(C)C)CC2)=O)cc(F)cnc1O 8980,c1(COCC)nc(C)c(C(=O)NCC(C)(C2CC2)NC(=O)CCCC2(C)N=N2)s1 8981,Cc1ccc(CCC(=O)NCC2CC2CCC(N)=O)s1 8982,C12(C(=O)NCC(C#C)CC)CC(CN(C(=O)CNC(=O)C3CC3)C1)C2.OC 8983,C(CCC(=O)N1CCC(N(C(=O)CCC=C)CCO)C1)=CCC=C 8984,N(C(=NCC)N1CCN(C(C)=O)C(C)(C)C1)C(C#C)(CC)CC 8985,N(C(=NCCCNc1ccc(Cl)cc1)NC1CCCCC1C)C1C(CC(C)C)C1 8986,C(=O)(C(C)OC)N.C(=O)(C(C)OCC(F)(F)F)N(CCN(CC=C)C)C1CC1 8987,c1(C(=O)NC(CC(C)NC(=O)C(C2CCCCCC2)C)C)cc(N)ccn1 8988,Cc1cccc2[nH]cc(C(=O)N(C)CCNC(=O)C(N3CCCC(O)C3)C)c12 8989,c1(CNC(N(CC(O)Cc2ccccc2F)C)=O)cncc(C(C)(C)C)c1 8990,Cc1nc2cc(C(N3CC4CC(NC(c5cccc(Cl)c5F)=O)C4C3)=O)[nH]c2s1 8991,S(=O)(=O)(c1ccc(N2CCN(C)C(CCO)C2)c(Br)c1)NC(CC)CCC 8992,C(c1c(C)nn(C)c1Cl)=CC(N1CCCC(NC(CS(CC)=O)=O)(CO)C1)=O 8993,C(N=c1[nH]c(Cl)ncc1C)C1CN(C(C2C(OCC)C2)=O)CC1(C)C 8994,c1(C(N(CC)CC2CCCN2C(=O)C(C)(O)C(C)C)=O)cc2cccnn2n1 8995,C1(O)(C(=O)OC)CCN(CCC(N2CCN(C3CCNCC3)CC2)C)CC1 8996,c1(C(N(C(CCNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)ncc(Cl)c(N)c1Cl 8997,c1(C(C)C)ccc(SNCc2cnn(C)c2)cc1OCC(F)F 8998,N1(C(C(c2ccnn2C)C)=O)CC2CC(NC(C3C4CN(C)CC34)=O)CC1C2 8999,C1(C(N2CC(CCNC(c3ccn(C)n3)=O)C2)=O)C2CCN1CC2 9000,C1(NC(C2(CC)CC2)=O)CS(=O)(=O)CC1NC(=O)Cc1c(O)ncnc1O 9001,c1(CC)ccc(OC)c(C(=O)NC2CCC2NC(=O)CCCCSC)c1 9002,Cc1cc(NC(=O)CN2C(=O)CNC2=O)ccc1NC(=O)C(C)C1CCC1 9003,CC1CN(C(c2ccc(CNC(=O)CC(C)(C)O)nc2)=O)Cc2nncn21 9004,C1(CC)CCN(C(c2ccc(O)nc2)=O)C1C(=O)NCc1cc(=O)cc[nH]1 9005,C1(CNC(C2CCN(C3CCCCC3)C2)=O)CC2CC2N1C(=O)Cc1ccccc1 9006,c1(N2CC(CC)(CC)OCC2)nc(=NCc2cc(C)cc(F)c2)[nH]c2cc[nH]c12 9007,c1(C(=O)NC2C(CNC(=O)C=Cc3ccncc3)CCC2)ncc(Cl)cc1Cl 9008,C#Cc1ccc(NC(C2CCN(CCNC(=O)C(c3ccccc3)O)CC2)=O)cc1 9009,n1(C(C)C(N2CCCC2CNC(C2CC2CN(C)C)=O)=O)cc2ccccc2n1 9010,C(C(C)S(C)(=O)=O)NC(=O)C#CC(=O)N(C)C.C1C(C)C(=O)N1C.CO 9011,C1(NC(c2cnno2)=O)CCCC1NC(=O)C1CC1 9012,c1(C(=O)OCS(C(C)C)(=O)=O)ccnc(C(=O)N(CCO)CC2CCOCC2)c1 9013,C1(C(N2CCN(C(c3scc(COC)c3)=O)CC2)=O)CC2C=CC1CC2 9014,C1(NC(c2c(CC)scn2)=O)C2CC3CN(C(c4c[nH]c(=N)s4)=O)C1C3C2 9015,N1(C(c2cc(C)no2)C(=O)NCC2CCCO2)CCCC(c2ccc(F)cc2)C1 9016,CN1C(=O)CCCC1C(N1CC(C2CC2C(N2CC(NC(=O)C3CC3)C2)=O)C1)=O 9017,C1(OCC)CC2(C1)CC(C(=O)NCC(C)(CO)NC(c1cc(C(C)C)no1)=O)C2 9018,C(C#CC(=O)NCC1CC1)N(C(C=CCOCCOC)=O)CCC1CCCC1 9019,CC1(CNC(=O)CCCCO)CN(C(C2NC(=O)CC2C(F)(F)F)=O)CCO1 9020,c1(OC)c(C(=O)Nc2nc(OC)c(C3CC3)c(Cl)n2)[nH]c2ccccc12 9021,N1(C(CC=C=C)=O)Cc2cnn(C3CCN(C(c4cocc4C)=O)CC3)c2C1 9022,C(C(C(=O)NC1CC(F)(NC(=O)CSCCC(C)C)C1)OC)OC 9023,C(=O)(CC(C)C(=O)c1ccccc1)NC(CN(CC(C)(C1CCC1)OC)C1CC1)=O 9024,N1(N(C2CCCC2)CCOC)CCC(C(=O)OC2(C=O)CC2)CC1.C(N)(=O)N 9025,c1(C(=O)NCC2(C(C)NC(C(C)=C3CCC3)=O)CC2)nc2cccnc2s1 9026,C1(C(N(C(C)C)CC2CCC2)=O)CN(C(C2CC(O)C2)=O)CC1CC(C)(C)C 9027,c1(OC)ccc(CCCC(=O)OC(C)C(=O)NC2(C(=O)O)CCCCC2)cc1 9028,c1(C(N2CC(N(C(CC=CC)=O)C)C(C)(C)C2)=O)c(C)oc2ccccc12 9029,C(C(=O)N1CC(O)CCO1)(C(C)(C)O)COC(CC(=O)OC(C)(C)C)=O 9030,C=CCCC(C(=O)N1CCCC(CCF)C1)NC(=O)CN1CCCNC1=O 9031,CCC(C)(CO)C(=O)NC(C)(CNC(C1(C)CCCCC1)=O)C1CC1 9032,c1(C(CC)NC(=O)Cc2csnc2C)ccc(CNC(C2CCCCS2)=O)cc1 9033,N1(C(Cc2c(C)ncs2)=O)CC2COCC(C1)C2NC(=O)CN1CCCC1=O 9034,N1(C(CC)=O)CCC=C(CNC(C2CC(=O)N(CCOC)C2)=O)C1 9035,Cc1ccc(Cl)c(OC(C)C(=O)NC(C)(C)CCNC(=O)C(O)CC)c1 9036,c1(CCC(=O)N(C(CNC(c2cnn(C)c2)=O)C2CC2)C)ccccn1 9037,O=S(=O)(Oc1cc(Br)ccc1Cl)c1c[nH]ccc1=Nc1cccc(OC(F)(F)F)c1 9038,N1(C(c2c(CC)onc2)=O)CC=C(CNC(=O)C(c2ccccc2)OC)CC1 9039,c1(C(C)=O)cccc(C(=O)NCC(CO)NC(c2cnc(Cl)[nH]2)=O)c1 9040,C1(NC(C(CC)=CC)=O)CC2CN(C(=O)CCOc3ccc(CSC)cc3)CC12 9041,CC1(C)C(NC(C2CC(=O)C2)=O)CCN1C(=O)Cc1cc(-c2ccccc2)on1 9042,C=CCN=c1[nH]cc(C(N2CCN(C(=O)CN(CC(=O)NCC)C)CC2)=O)s1 9043,C1(C(=O)NC(C(C)C)CCNC(=O)CCc2cccnc2)CCC2CCCCN12 9044,C1(OC)CC(C)CN(C(N2CCN(c3ccccc3)CC2)=O)C1 9045,C(c1ccco1)=CC(=O)NC(C(=O)NCCOCC#C)C1CCOC1 9046,CN1CCN(C(c2cc(C3CC3)ccn2)=O)c2ccc(O)cc21 9047,Cc1cc[nH]c(=N)c1C(=O)NCC1CCCCN1C(c1cn(CC2CC2)nn1)=O 9048,N1(C(COC2CN(C(C)=O)C2)=O)CCC(CCNC(c2cnc(Cl)s2)=O)CC1 9049,c1(C(=O)NC(c2nnc(C)s2)C)ccc(CNC(=O)CCc2nccs2)cn1 9050,Cc1sc(O)nc1C(N1CCCCC1CNC(C12CC(O)C1C2)=O)=O 9051,C(=O)(C(CC(F)F)N(C(=O)COc1cccnc1)C)Nc1ccc(CC)cn1 9052,c1(CNC(C2N(Cc3nc(C)sc3C)CC2)=O)cc(Cl)ccc1C 9053,CC(C)(CC(F)F)C(=O)N1CCCC(CNC(=O)Cn2cc(Br)c(=N)[nH]2)C1 9054,O=C1CCN(C2CC2)C(=O)N1c1ccc(Cc2cscc2Br)cc1 9055,C1(NC(C(CC)(CC)CC)=O)C2CC3CN(C(c4cnc(C5CC5)[nH]4)=O)C1C3C2 9056,C(CC(C(=O)NCc1nc(C)no1)NC(=O)C(C)CC1CC1)OCC 9057,C(=O)(CC(C)CNC(=O)C(O)CCNC(=O)CCc1nc(C)no1)OC 9058,n1(CCC(=O)NCC2CC2CNC(c2ccon2)=O)nnc2ccccc2c1=O 9059,C1(C(C)NC(C2(CC=C)COC2)=O)CCCN(C(C2(F)CC2)=O)C1 9060,C1(CC(=O)NCCc2cc(C(N(CC(C)(C)O)CC)=O)no2)NC(=O)NC1=O 9061,c1(C(N(CC(=O)N(C(CO)CO)CC)CC2CC2)=O)csc(O)n1 9062,Cc1c(C(=O)NC(C)CN(C(C2COCCN2C)=O)C2CC2)c[nH]c1C#N 9063,C(=O)(CC(O)CC(C)C)N1C(C(N2CCC(C(C)(C)OC)C2)=O)CC(OC)C1 9064,C1(CCNC(CN(CC)CC)=O)C(C)CCCN1C(c1cnn(C(C)C)c1)=O 9065,C1(C#N)(C(N2CC(C)C(NC(C3(C4CCCO4)CCC3)=O)C2)=O)CC2C=CC1C2 9066,C1(NC(C(c2ccnn2C)NC(c2c(C)oc(C#N)c2)=O)=O)CC2(C1)CC21CCC1 9067,C(=O)(CCCCN=[N+]=[N-])N(CC(=O)NCC(C#C)CC)CCOC 9068,CCCN=C(NCCCn1ccnn1)N1CCCC(c2ccon2)C1 9069,c1(C(=O)NCCN(C(=O)CC(C)c2ccco2)C(C)C)ccnc(N(C)C)n1 9070,N1(c2nc(C)nc(O)c2C)CCC2(CCOC2)C(CNC(=O)COC(F)F)C1 9071,C1(C(N2CC(C(C)NC(c3cncn3C)=O)C2)=O)(COC)CCCO1 9072,C1(C(N(CCCNC(C(C)n2ccnc2)=O)C)=O)Cc2nccnc2C1 9073,N1(C(C(C)SCCCC)=O)CCC(C)(C)C1C(N1CCC(C)(N(C)C)CC1)=O 9074,N(S(=O)(=O)NCC1CC(Br)(Br)C1)CCCOC 9075,C(N=c1[nH]c(=NCCS(N)(=O)=O)[nH]c2c1CSC2)C1C(C)(C)C1 9076,Cc1ccc(C(N2CCN(C(=O)CC3(C4CC4)CC3)C(CO)C2)=O)nc1C 9077,Cn1ccc2ccc(C(=O)NCC3(O)CC(NC(C4CC(C(F)(F)F)C4)=O)C3)cc12 9078,CC1(C)CN(C(=O)C(F)C(F)(F)F)CC1CNC(=O)C1=COCC1 9079,C1(NC(N(CCCN(C(C)=O)C)C)=O)CCC(N2CCCC2=O)CC1 9080,CCC(CNC(C1CC2CC2C1)=O)N=c1nc(O)c(Cl)c[nH]1 9081,CC1(C(=O)NCC2CCCCN(C(c3cncc(Cl)c3)=O)C2)CCCCNC1=O 9082,C1(S(C)(=O)=O)(CNC(=NCCC(CF)C(F)(F)F)NCC2CC23CCC3)CCC1 9083,Cc1ccnc(C(=O)NCCOC(C23CC(OC(C)(C)C)C2C3)=O)c1 9084,c1(C(=O)OC)cnoc1NC(N1CC(C)(c2ncc(C(F)(F)F)[nH]2)C1)=O 9085,C1(NC(C2CC3(CC(=C)C3)C2)=O)CCC2CC1CN2C(=O)Cc1conc1C 9086,c1(CSC)cc(C(=O)NCC2(CNC(C3CCN(C)CC3)=O)CCC2)ccc1F 9087,C(CNC(C1CC(CF)C1)=O)(CC(=O)NC(CO)C1CCC1)OC 9088,CC(C(C)CO)NC(=O)C(Cc1cc[nH]n1)NC(=O)Cc1csnn1 9089,N1(C(c2cncc(C=C)c2)=O)CCN(C(c2nc[nH]n2)=O)CCC1C 9090,C1(NC(C23CC(C(=O)OC)(C2)C3)=O)CC(F)CN(C(=O)Cc2ccc(O)cc2)C1 9091,c1(C(N2C3(C(=O)OC)CCC3CC2)=O)ccc2c(c1)nc(O)n2CC(C)C 9092,Cn1ccc(C(=O)NCCC2CCN(C(c3ccnn3C(F)F)=O)C2)c1 9093,c1(SC(C)(C)C2(NCC3(O)C(C)C3)CC2)cc(F)c2ncccc2c1 9094,CC(C)(O)C(F)C(=O)NCC1(CCNC(=O)CC2COC(=O)C2)CC1 9095,C1(CC(=O)NC(C2CCN(C(c3cnn(C)c3Br)=O)CC2)C)CC2CCC1C2 9096,Cc1nc(C(=O)NC(C)CCCCNC(c2occc2Br)=O)[nH]c1C 9097,C1(OC)CN(C(C2CCN(C)C2C(=O)NOC(C2(C)CCC2)=O)=O)CC1OC 9098,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(CNC(=O)CN(C)C2CC2)C(C)(C)C1 9099,N(C1CCc2c(Cl)cc(Cl)cc21)S(=O)(=O)CC1CC2(CCCO2)CO1 9100,N1(C(C2C(C3C(C)C3)C2)=O)CCC2(CCCC2NC(c2cccn2C2CC2)=O)CC1 9101,CC(CNC(=O)Cc1ccnn1C1CCCCC1)(CO)NC(=O)C(O)C1CCC1 9102,N1(C(C(C(C)C)CO)=O)CCC2CCC(C1)N2C(c1csc(C2CC2)n1)=O 9103,c1(C(=O)NCC(CC)(C)NC(C2CS(=O)C2)=O)nc(Cl)c(Cl)s1 9104,C=C(C)CC(C(=O)NCC=CCCC)NC(C1CCOC(=O)CC1)=O 9105,c1(NC(c2csnn2)C)ncccc1S(=O)(=O)N1CC2CC3CCCN3C2C1 9106,c1(C(=O)NC(CC(C)NC(C2CC2C2CCC2)=O)C)ccnn(C)c1=O 9107,N1(C(C2=NOC(CNC(C=CC3N(C)CCC3)=O)C2)=O)CC(O)CC(O)C1 9108,N1(C(c2ccccc2CCC)=O)CCN(C(c2ncn(CC(=C)C)n2)=O)C(C)C1 9109,c1(C(=O)NC(CC(C)NC(Cc2c(C)ncc(Cl)c2)=O)C)cc2n(n1)CCCO2 9110,C1(CNC(C(c2ccnn2C)C)=O)CC(F)(F)CN1C(c1cc(Cl)c(Cl)n1C)=O 9111,C12(NC(CCCC3CCCC(=O)N3)=O)CCCC1N(C(C1CCCC1)=O)CCC2 9112,C(=O)(CN=c1cc[nH]cc1)NC(c1cccnc1)C(=O)NCc1c(C)cnn1C 9113,C12(CNC(CN(C)C(=O)C3CC3)=O)CCC(CC1)CN2C(C1CC12CC(O)C2)=O 9114,c1(N(C)CC2COC(=O)O2)nc2cccc(F)c2c(=NCC2(N(C)C)CC2)[nH]1 9115,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9116,c1(N(C)C)ccccc1C(c1nnnn1C1CC1)NC1C2COCC12 9117,Cn1cnnc1CC(=O)N(C1CCN(C(=O)COc2cccnc2)C1)CC1CC1 9118,c1(CNCC(C2CCCC2)NC(C(F)(F)Sc2cn(C)nc2)=O)[nH]ncc1C#N 9119,c1(CNC(c2c(NC(C3C(NCC)CCC3)=O)cccc2)=O)ccc(C)cc1O 9120,C1(C(=O)NC(C)Cc2ccccn2)(OC)CCCCC1.N12CCCC1C2=O 9121,N1(C(C)=O)CCC(O)(CCNC(=O)C(C)(C)CO)CC1.N12CCCC(C1)C2=O 9122,c1(CNC2C(C(N3CC(CCC)OCC3)=O)C2)cnc(OC)c(Br)c1 9123,c1(C(N2C(CCNC(CCCCSC)=O)CC(OC)C2)=O)nsc2ccccc12 9124,c1(C(=O)NC(C(=O)NC(C2CCCC2(C)C)C)Cc2ccoc2)ncc(F)cn1 9125,Cc1cc(C(=O)NCC2CC(C)CN(C(C3(C)SCCCS3)=O)C2)c(O)nn1 9126,c1(C(N2CCC(C)(CNC(C3N(C)CCCC3)=O)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] 9127,N1(C(C2(C)N(C(C(CC)SC)=O)CCC2)=O)CC2CC1CN2CC 9128,c1(C(N2CCC(NC(c3nc(C)oc3C)=O)C2C)=O)ccc(F)c2cccnc12 9129,c1(C(N(CCC(C)NC(c2cc(C)ns2)=O)C)=O)cc(OC)nn1C 9130,c1(C(CN(C(C)C)Cc2cc(F)ccc2F)=O)ccc(C(F)(F)F)c(Cl)c1 9131,c1(CNC(=O)CN2CCN(CC3CCCCS3(=O)=O)CC2)c(F)ccnc1F 9132,N1(C(CC(=O)NCC)=O)CCC2(CCCC2NC(=O)C(C)(O)COC)CC1 9133,c1(OC)cccc(C(=O)NC2CN(C(c3csc(Cl)c3)=O)CC2C)c1 9134,Cc1ccn(C)c1C(=O)N(CC(C)(C)CNC(c1nn(C(F)F)cc1Cl)=O)C 9135,C(=O)(CCC(=O)NC)NC1(COCCOC)CCN(C(=O)Cc2ncc(Cl)s2)C1 9136,C1(C(N2CC(CC(=O)OCC)CC23CCC3)=O)CC(=O)c2cc(Cl)ccc2O1 9137,C1(CC(=O)NC2C(NC(C(C)NC=O)=O)CCC2)COCC1(C)C 9138,C(CC(CC)C(=O)N1CCC(NC(=O)CCc2ccccc2C#N)C1)=CC 9139,c1(C(N(C)CC2(NC(COCCCCC)=O)CC2)=O)ccnn1C(C)CC 9140,c1(C(N2C(CNC(C(CC)N(C)C)=O)C(C)CC2)=O)nnn2ccccc12 9141,c1(C(N(C2CCN(C(=O)CC3CCC3=O)CC2)CC)=O)cccc2ccccc12 9142,C1(NC(C2CCSC2)=O)CC2CN(C(=O)Cc3cc[nH]c3)CCN2C1=O 9143,CC(C)CC(C(=O)N1CCC(CNC(c2ccsc2)=O)C(O)C1)C(C)C 9144,N1(c2cc(Nc3ccc(Br)cc3F)nc(COC)n2)CCc2c(cc(C#N)n2C)C1 9145,c1(C(N2CCC(NC(CN3C(C)CCCC3)=O)(CF)C2)=O)ccn2nnnc2c1 9146,CC(F)(F)CCC(=O)N(CC(=O)NC1CCC12CCCC2)C1CCC1 9147,C1(C(=O)OC)C2CC1N(CCC1(n3cc(CCC4CCCO4)nn3)CCOCC1)C2 9148,C1(CCC)CN(C(=O)C(C)C(=O)OC)CC1NC(=O)CSCC(=O)OC(C)(C)C 9149,c1(CC)nn(C)c(Cl)c1C(N1CC(CC(C)NC(=O)CN2C(=O)CCC2=O)C1)=O 9150,c1(C(=O)NC(CC)CN(C)C(c2cn(CCCF)nn2)=O)nn(C)c(N)c1C 9151,Cc1cc(C(N2CCC(O)(CNC(C3(O)CCOCC3)=O)CC2)=O)cc(C)n1 9152,C1(F)(CNC(Cc2ccc(CCCC)cc2)=O)COCCN(C(=O)CCC#N)C1 9153,C1(C(=O)NC(CNC(C2(OC)CCSCC2)=O)C(C)C)CC2(C)CC1CO2 9154,C1(CNC(=O)C(F)n2cccn2)CN(C(C2(Br)CC2)=O)CC1O 9155,c1(OC)cc(N)c(C(=O)NC2CCCC(N)CC2)cc1Cl 9156,C1(C(=O)NCCC2N(C(C(C)(C)n3ccnc3)=O)CCC2)CC1C1CCCC1 9157,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CC1CN2C(C1CCCCO1)=O 9158,c1(-c2cc(C(=O)NCC(CC=C)NC(C3CCCO3)=O)n[nH]2)ccccc1C#N 9159,Cn1ncc2c(CNC3CN(C(c4scc5c4OCCO5)=O)CCCOC3)cccc12 9160,CC1CN(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCN(C(C3CCCS3)=O)C2)O1 9161,N12CCC3(CC1)CCN3CC2=O.N1(C(C)=O)CCN(S(=O)(=O)CCCCl)CC1 9162,C1(CC(N2CC(OC)C(NC(C34CC(C)(CO3)C4)=O)C2)=O)CCC(=O)NC1=O 9163,N1(C(C(C)(C)n2cc(Br)cn2)=O)CC(NC(C2CC3C=CC2C3)=O)CC(F)C1 9164,CN1C(=O)CN(CC(N2CCCC2COC=O)=O)C1=O.c1(C(C=O)=O)ccccc1 9165,c1(C(=O)NCC(C)CNC(C2CCCO2)=O)[nH]cc2c1CCS2(=O)=O 9166,C1(NC(=O)OC(C)C)CCN(C(=NCCCF)NCCC2CCCC2(F)F)CC1 9167,c1(C(N)=O)cc2cc(C(N3CCC(OC4CCNC4)CC3)=O)ccc2[nH]1 9168,c1(OC)c(CNN(C)C(C)=O)cccc1C.C12=CC=C(C=C1)C2 9169,CCCCCCN(C(c1cnc(C)[nH]1)=O)CC.C(C)(C)(C)O 9170,Cc1ccc(CC(N2CC3C(C(=O)NCc4ccnnc4)C3C2)C)cc1C 9171,C1(COC)CCCN(C(c2nccn2C)CC(=O)Nc2ncc(C(F)(F)F)[nH]2)C1 9172,C1(O)(CNC(COCC(=O)OC)=O)CCN(C(=O)CCC2CCCCC(=O)N2)CC1 9173,C(=O)(CC(C)(F)F)NC1CCC(N(C(c2c(C(C)C)occ2)=O)C)C1 9174,C1(C(=O)NCC2(CCNC(C(C)NC(N)=O)=O)CC2)CCCCN1C1CCCC1 9175,CC1(C)C2CN3C(C12)C3=O.C1(NC(=O)CCCN2CCCC2)C2C3CCC(C3)C12 9176,N1(CCC(=C)C)CCOC(CNC(c2ccc(C#N)o2)=O)C1 9177,C1(C(C)C)(C(=O)N(C(C)CCO)C)CCN(C(C2CCC2C)=O)C1 9178,C1(CCC)(NC(c2n[nH]c(CC)n2)=O)CCN(C(c2ccc(F)s2)=O)CC1 9179,N1(C(=O)Cc2cc[nH]n2)CCCC(C2CCCCN2C(c2ccc(F)cc2)=O)C1 9180,c1(NC)nc(N2CC3(CC4CC4)CCC2C3)nc2ccccc12.c12cn(nn1)C2 9181,c1(C(N2CCCC2c2cn(CCOc3ncccn3)nn2)=O)sccc1CC(=O)O 9182,N1(CC2CC(C)(C)N(C(=O)CNC)C2)CC2CC3CC2C1C3.C1(C=O)CCC1 9183,C(C)(C(=O)NCC(C)(C1CCC1)NC(=O)CSCC(N)=O)OCC#C 9184,C1(CC(=O)NC)CN(C(=O)CCC2CCC(NC(c3ccoc3Cl)=O)C2)CCO1 9185,c1(C(N2CCC3(C(C(=O)Nc4ccnc(CO)c4)C3)C2)=O)ccc2occc2c1 9186,N1(CC(=O)NCCCOCCNC(C2C(C)C2C)=O)CCC(C(N)=O)CC1 9187,Cc1cc(C(=O)NCCN(C(=O)CC2C=CCC2)CC(C)O)nn1C(F)F 9188,C(C(=O)NCC1(C)CCCN1C(=O)CNC(=O)C1CC1)(C(C)C)NC(C)=O 9189,N1(C(C)C(=O)NCc2cccs2)CCC2(CC1)SCCS2 9190,Cc1nccc(C(=O)NCC2COC(CNC(=O)CCSc3n[nH]c(C)n3)C2)n1 9191,N1(C(C)=O)CC23CCCC2(C1)CN(C(=O)Cc1c(C)cc(C#N)cc1C)C3 9192,C1(NC(C(C2CCCN2Cc2cccc(CO)n2)C)=O)CN(C)CC1O 9193,C1(CNC(C2(C(C)O)CC2)=O)CN(C)CCO1.c1(CC(=O)NCC)ccc(F)nc1 9194,c1(C(N(CC(N2C(C#C)CCC2)=O)CC(C)C)=O)cc(C#C)ccn1 9195,c1(C(=O)NC(C2(CNC(C(C=C)(C)C)=O)CC2)C)ccnc(C)c1O 9196,C#CCC(C)(C(=O)N1CC(=O)NC(CC)C1)NC(=O)CCOC1CC1 9197,c1(C(N2CCN(C)CC2CNC(C2CC(C)(F)C2)=O)=O)ccc2[nH]ccc2c1 9198,n12c(nnc1C)N(CC)C(CC)C2.c1(C(CC)OCC)ccccc1Cl 9199,c1(COC)cc(C(=O)NCCOCCNC(=O)CCc2cc(Cl)cs2)on1 9200,c1(C(=O)NC2(CC)CCN(C(c3c[nH]nc3F)=O)CC2)cn2cccnc2n1 9201,c1(C(N2CCC(O)(CNC(c3ncc(C)nc3)=O)C2)=O)cccc(Br)c1C 9202,N1(C(Cc2ccn(CC)n2)=O)CCC(NC(c2cnn(C3CCC3)c2)=O)C(O)C1 9203,c1(C(C(=O)NC2CC(F)(CNC(CCC(C)C)=O)C2)(F)F)cc(Cl)ccc1Cl 9204,N1(C(c2n(CC)ncc2)=O)CC(CC(=O)NC(c2cnsc2)C)C(C)C1 9205,C(=O)(C(C)C)NC(C1C(CNC(COCC(N2CCCC2)C)=O)C1)=O 9206,C(C)(CN=c1ccc(C(F)(F)F)c[nH]1)N.C(=O)(C[SH](=O)=O)N(C(C)(C)C)C(C)=O 9207,C1(C#N)(OC)CC(NC(=O)OC(C)(C)C)C1.C1C(C)C(=O)O1 9208,c1(-c2nc(CCOC)nn2CCF)ccncc1C=CC(N1CCCC(C)C1)=O 9209,Cc1nn(C)c2c1CCN2C(=O)NC1CCN(CCF)C1=O 9210,C=CCC(F)(F)C(=O)N1CCC(CC(=O)NCC2(O)CC3C=CC2C3)C1 9211,Cc1ccc(CS(N2CC(NC(c3oc(C)nc3C)=O)C(F)C2)(=O)=O)cc1 9212,C1(C)(CC(=O)OC)CC(CN)CN1C(=O)Cc1cnn(-c2ccccc2)c1 9213,CS(=O)(=O)c1ccc(C(N2CCN(C(C3(O)CCSC3)=O)CC2C2CCC2)=O)s1 9214,CCC(CC)C(=O)NCC(=O)NCCC(C)N(C)C(c1cc(C)sc1C)=O 9215,C1(c2n(C)nnn2)(NCCc2cccn2Cc2ccccc2)CC1C1CC1 9216,C=CCCCC(=O)NC(C1CCCN(C(=O)C(C)CSC)C1)(C)C 9217,c1(C(N2CCC(NC(CCCC(=C)C)=O)CC2C)=O)cnc2[nH]nnc2c1 9218,c1(OCC(=O)NC(CC)(C)CNC(=O)CN2CCCC2C)cc(F)ccc1F 9219,c1(C(N2CC(CCOC)N(C(=O)CSC)CC2)=O)cccc2c1COC2 9220,C1(F)(CNC(C2CC23CC3)=O)CC(CNC(c2cnn(CCN(C)C)c2)=O)C1 9221,N1(C(C2(OC)CCCCC2)=O)CCCC(O)(CNC(=O)CCn2ccnn2)CC1 9222,c1(C(C(=O)NC(C2CC(F)(F)C2)CNC(C(N)=O)=O)N2CCCC2)ccccc1 9223,N1(C(C2CC(c3cccc(O)c3)C2)=O)CCC2(CC1)CN(C(c1ccns1)=O)C2 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9278,C1(C(=O)NCCCCN(C(=O)COC2CCCCC2)C)CCc2nnnn2C1 9279,N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCOC2)C(CNC(C2(F)CC2)=O)C1 9280,c1(-n2c(-c3cc(Cl)n(C4CCC4)n3)nc(CSC)n2)ccc(F)c(C)c1 9281,Cc1ccc(C(=O)NCCC2CN(C(=O)C=CC=C(Cl)Cl)CC(C)O2)c(F)c1Cl 9282,c1(OC)ccc(C(N2CCC(CO)C(NC(c3sccc3C)=O)C2)=O)cc1N 9283,CC1CC(C(=O)NC(C)(C)CF)=NO1.c12nc(co1)C(=O)N1CC(C1)C2 9284,N1(C(c2[nH]cc(C)c2)=O)CCCC12CCN(C(C1(C)CCCO1)=O)CC2 9285,N1(C(CC=CC=C)=O)CC2(C1)CN(C(c1cc(C#N)c(C)cn1)=O)CC2CO 9286,c1(N2CCC(OCC(COc3c(C)cc(Cl)cc3)O)C2)cc(N=[N+]=[N-])ccn1 9287,c1(CC)ccc(-c2ccc(F)c(C(=O)N=c3nc[nH]s3)c2)cc1F 9288,CC(CCCCCO)NC(=O)C(C1(C)CC1)NC(=O)C=CC1CCCC1 9289,N1(C(c2ccn(CC)n2)=O)CCC(C2CC2)C1CNC(=O)C=Cc1nc(C)co1 9290,C(=O)(CCC(=O)NC1CCCC1)NCC1N(C(C2(C=C)CCC2)=O)CC1 9291,C1(OC)CC(NC(C2CN(C(N)=O)C2)=O)CN(C(c2snc(O)c2Cl)=O)C1 9292,c1(NC(=O)C(=O)NC2(N3CCOCC3)CCC2)ccc2nccn2c1 9293,c1(C2C(C)C2)cc(C(=O)N(C2CN(C(c3cc(Cl)no3)=O)C2)C)on1 9294,c1(C(=O)NC(C)C(CO)NC(c2cc(C(N)=O)no2)=O)cc2sccc2[nH]1 9295,C(CCC(C)C(=O)NOC(CC(C)C)C(=O)NCC1CC2(CCC2)CO1)OC 9296,c1(C(=O)NC(C2CCCN2C(c2ccnnc2Cl)=O)C)cc2scc(Cl)c2[nH]1 9297,Brc1cc(C(c2ccccc2)NC(C2CCCCC2)C2CCC2)ccn1 9298,c1(COC)cccnc1C(=O)N(C1CCN(C(=O)C=Cc2cc[nH]n2)C1)C 9299,C1(CC(=O)NC(CNC(C=CC(CC)C)=O)C2CC2)CCOC2(CCOCC2)C1 9300,C12(NC(=O)COc3ccccn3)CCN(C(C3CCOCC3)=O)CC1C2 9301,S(=O)(=O)(c1cccnc1NCCn1ccnc1)NCc1scc(CC)n1 9302,c1(C(=O)NC(CC)CNC(=O)COc2cccc(O)c2)cnc(C)nc1C 9303,c1(C(C(=O)OC)=O)ccc(C(=O)NCC2CCN2C(=O)C(O)CC2CCCO2)nc1 9304,Cc1nn(C2CCC2)cc1C(C(=O)NC1CCCCC1)N(C1CC(O)C1)C 9305,C1CCC(=O)N1.C1(NC(=O)CC2CCOC2)CC(F)(CO)C1 9306,c1(CN(C)C(=O)NCCc2ccc3ccccc3c2)cccc2ccc(F)cc12 9307,c1(OC(C)C(=O)NC2C=CC(NC(=O)C3=CCC3)C2)ccc(F)cc1 9308,C12(CNC(=O)CN3CCC(NC(C4CCC4)=O)CC3)CC=CC(C1)OC2 9309,N1(C(c2ccn(CC)c(=O)c2)=O)CCN(C(=O)C2=C(C)OCC2)C2CCCCC12 9310,C(=O)(C(=O)C(F)(F)F)N1C(C(C)NC(C(CC)OCC)=O)CCC1 9311,c1(C(N2CCC(C)(C(N3CC(F)(F)C3)=O)C2)=O)cc2cccc(O)c2[nH]1 9312,c1(C(=O)NC2C3(CC(NC(C#CC(C)(C)C)=O)C3)C2)nc(=N)[nH]c2ccccc12 9313,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CC(C)N(C(=O)C2=COCC2)CC1C 9314,C1(c2n(C)ncc2)CCCC(c2nnnn2C2CC2)(NCCCn2nccn2)C1 9315,c1(-c2cc(CC(=O)Nc3c(C(C)O)cccc3)ncc2)cccc2c[nH]nc12 9316,N1(C(C(c2ccccc2)C)=O)CC=C(CNC(C2CC2Cl)=O)CC1 9317,c1(N2CCCC(C)(C(=O)NCC)C2)nccc(=NC2CC3CSCC3C2)[nH]1 9318,N1(C(CCN2CC(C)C2)=O)CCCC1C1(O)CN(C(=O)C=CC2CCC2)C1 9319,N1(C(C(CO)C)=O)CCC(CSC)(CNC(=O)C(C)OCC2CCCO2)C1.CO 9320,n1(CC)nnc(C(=O)NC(C)C(C)NC(c2ccc(-c3cccs3)[nH]2)=O)c1C 9321,N1(C(C2C3N(C(C(COC)(C)OC)=O)C(CC3)C2)=O)CC2CCCC(O)C2C1 9322,c1(OC)ccc(I)c(NC(=O)COC(C2CCCCC2SC)=O)c1 9323,Cc1ccc(NC(C2(CNC(=O)CNc3ccccn3)CCCO2)=O)c(O)n1 9324,S(=O)(=O)(c1cccnc1NCC1CCCC1O)NC(c1c(C(F)(F)F)cccc1F)C 9325,c1(C(=O)NCCCNC(C(C)CC2CCCCC2)=O)c[nH]c2ccc(C#N)cc12 9326,c1(OCCN(C(=O)NC(CCCCC)c2ccccc2F)CC)cc(Cl)ccc1C 9327,N1(C(=O)CCc2cccc(O)n2)CC2C3CCC(C2C1)N(C(=O)CSC1CC1)C3 9328,C1(N(C)C)CCC(C(=O)NCC=CCNC(=O)Cn2ccnn2)C1 9329,c1(C(=O)NCCC2CN(C(C3CC(O)C3)=O)CC(C)O2)cc(O)cc(F)c1F 9330,c1(CNC(C2CN(C(c3ccon3)=O)C2)=O)ccc(SC(F)F)cc1 9331,C1(N(C(c2ccn(CC)n2)=O)C2CC2)CCCCC1n1cc(-c2ccc(F)cc2)nn1 9332,C(=O)(CCC(C)(C)F)N1CCC(C(=O)NCCC(C)(C)C)(CO)C1 9333,Cc1ccc(C(=O)OCCCCC2CCOCC2)cc1 9334,C#CCCCC(=O)Nc1ccc(N2CCN(C(C)=O)CC2)cn1 9335,c1(OC(C)C)cnc(C(=O)Nc2cccnc2-c2cncc(CN(C)C)c2)cn1 9336,C(=O)(C1CCCc2n[nH]cc21)N(CCCNC(=O)COCCSC)CC 9337,C(=O)(C(C)(O)C(C)(O)C(=O)OCC(=O)N(CC(C)C)C1CC1)OC 9338,CC.N1(CCSCCN(C(=O)CN)CC)CCC1 9339,C1(CNC(COCC#C)=O)C(C)CCN1C(=O)CSc1cccc(Cl)c1 9340,c1(C(=O)NC(CC)(C)CNC(c2ccc(C)n2C)=O)cc(C(F)F)nc(SC)n1 9341,N1(C(CC(CC)c2ccccc2)=O)CC2CC1CCC2NC(=O)Cc1cnns1 9342,C1(C)(CNC(C2OCCN(C(c3ccc(CC)[nH]3)=O)C2)=O)CC2CCC1C2 9343,C(c1cccc(F)c1)=CC(=O)NCC1(NC(C2CCCNS2(=O)=O)=O)CCC1 9344,C(=O)(CS(=O)(=O)C1CCCC1)N(C1CCC(NC(c2csc(C#N)c2)=O)C1)C 9345,N1(C(c2n(C)ncc2)=O)CCC2(CC1)CC2C(=O)NC(c1ccc(F)cn1)Cl 9346,c1(C(=O)NCC(C)CN(C(=O)Cc2cnn(C)n2)C)ccc2oncc2c1 9347,C12(NC(C(CCOC)NC(c3[nH]nnc3C)=O)=O)CCC(C1)OC2C 9348,Cc1cn2nc(C(=O)NC(C)CN(C)C(C3CC4(CC4)CO3)=O)cc2c(=O)[nH]1 9349,Cc1cc(C(N2CC(NC(c3ncccc3C)=O)C3CC23)=O)sc1C 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9529,C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(C2CN(C(=O)NC)C2)=O)C(O)C1 9530,n1(CC)cnc2c(NC(C)C(C(C)C)NC(=O)CN(C)CCO)nc(Cl)nc12 9531,c1(NC(N2CCC(NS(NC)(=O)=O)CC2)=O)cn2c(F)cccc2n1 9532,N1(C(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CO)C(c2ccccc2)C1 9533,Cc1cncc(NC(=O)C(N2CCN(CC3CC(N)C3)CC2)=O)c1C 9534,C(=O)(N1CC(O)C(O)CO1)C1OCCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 9535,C1(CNC(C(c2ccc(SC)cc2)C)=O)CCCCN(C(=O)CCCC(C)C)C1 9536,c1(C(=O)NCC(C)(O)CNC(c2cccc(CC3CCC3)c2)=O)cccnc1S 9537,Cc1ccn2cc(COC(C3(C)CCCN3C)=O)nc2n1 9538,C1(N2CCC(N(C(=O)CC=C(Cl)Cl)C)C2)CCN(C(=O)COC2CC(F)(F)C2)CC1 9539,N1(C(C(c2ccccc2)C)=O)CC2CC1CN2C(C1(COC)CCCO1)=O 9540,C1(CC(=O)N(CCCOC)CCO)CN(C(c2cnc(C)cn2)=O)CCC1C 9541,Cc1ccccc1SCC(N1CCC(C(C)Nc2ncccn2)C1)=O 9542,C=CCCCCCC(=O)NC(C1CCCN(C(c2ccc(N(C)C)o2)=O)C1)C 9543,Cc1ccc(NC(C2CCCN2Cc2nn(C)cc2[N+](=O)[O-])=O)c2cccnc12 9544,C1(C(=O)NCC2(CNC(C(c3ccc(Cl)cc3)CC)=O)CC2)CC2(CC2)CO1 9545,c1(N(CC(CN(C(C2CN(C)C(=O)CC2)=O)C)O)C)c(C#N)c(=O)n(C)c(=O)n1C 9546,c1(N(CCNC2CC(C)N(C(c3cncc(N(C)C)c3)=O)C2)C)ncnc(Cl)c1F 9547,CC(C)(C)CC(O)CC(=O)NCC1CC(C)(C)CN1C(c1cnn(CCF)c1)=O 9548,c1(C(N2CC(NC(C=CC)=O)C(c3ccccc3)CC2)=O)cc(F)c(F)cc1Cl 9549,CC(C)CC(F)C(=O)NCCC(C)NC(=O)CCC(=O)c1cccc(Cl)c1 9550,c1(CNC(c2nncn2C)C)cc(F)c(C(F)(F)F)cc1F 9551,c1(C(N2CC(O)(CNC(C3C(CC)OCC3)=O)C2)=O)ncnc(C(C)(C)C)n1 9552,Cc1ccccc1C(C)NC(c1oc(CNC(c2ncncc2N)=O)cc1C)=O 9553,Cc1ccc(CN(C)C(C2CC(C)N(C(C3(NC(N)=O)CC3)=O)C2)=O)cn1 9554,C(=O)(C(C)(C)C(C)(C)C)N(C)CC1(NC(CCCC=C)=O)CC1 9555,N1(C(c2cncc(Cl)c2)=O)CC2(CCC(C(N3CC(OC(F)(F)F)C3)=O)O2)C1.CCS 9556,C1(O)(CC(=O)NCCNC(=O)Cc2ccc(-c3csnn3)cc2)CCCOC1 9557,c1(N(C)C)ccc(C(=O)NC(c2ccccc2)CNC(=O)C2CC2)cn1 9558,N1(C(C(CC#C)C)=O)CCC2(CCC(CNC(C3(C(F)(F)F)CCC3)=O)O2)CC1 9559,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1CCC(=O)NC1CC(C(F)F)C1 9560,C1(C)(NC(C2C3C(NC(c4n(CC)ccn4)=O)C4C(C3)C42)=O)CCC(C)(C)CC1 9561,C(=O)(C(CN(C)C)N(C)C)NC(C)C(=O)N(C1CC(C)(C)C1)C 9562,N1(C(C(CCC=C)(C)C)=O)CCC2CN(C(c3cc(C(N)=O)[nH]n3)=O)CC2C1 9563,c1(NCC(CC)CO)ccc(S(=O)(=O)N2CCC(C3CCCCC3)C2)cc1Br 9564,C1(C(N(CC(N2CCOCC2)(C)C)C)=O)CCN(C(=O)C2CC3CCC(C2)O3)O1 9565,N1(CC2C(N)COCC2)CCC(C2CCC3(CC2)OCCO3)CC1 9566,N1(C(c2ccc(CSC)cc2)=O)C2CCC1CC(NC(=O)C(O)C(F)(F)F)C2 9567,c1(C(N2C(CC(=O)NCC(F)(F)F)CCCC2)=O)cc(F)ccc1F 9568,c1(NCCO)ccc2cc(OC)c(F)cc2n1.N1(CC)CC2C(C1)C(F)(F)C2(F)F 9569,Cc1cc(C(=O)NC2CCOC(CNC(C3(C)CC3)=O)C2)c2sc(=N)[nH]c2n1 9570,c1(OC)cccc(CNC2CN(C)CCN2C(C)=O)c1OC12CC(F)(C1)C2 9571,CC(C)C(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)C(C)C1 9572,C1(CC)(NC(=O)C(C)CC2CC2)CCCN(C(c2ccc(C)c(C)n2)=O)C1 9573,C=C(Cl)CCC(=O)N1CCCC(C(C)NC(c2cccnc2CC)=O)C1 9574,N#Cc1cc(CNC(C2(F)CCCN(C(=O)CC3CCSC3)C2)=O)ccn1 9575,C1(C(C)NC(=O)CCC2CC(NC(c3ncnn3C)=O)C2)CN(C)CCO1 9576,C(=O)(CCN=[N+]=[N-])N1CCC(N(CC#C)C(C2CCCS2)=O)C1 9577,CCC(C(=O)N1C2CCC(C2)C1C(=O)N(CCCN(C)C(C)=O)C)C(C)C 9578,C=CCCC(CC(C)C)C(=O)NCCOC1CN(C(=O)CC(C)(C)CC(F)(F)F)C1 9579,C1(NC(C2(F)CCCOC2)c2n(CCSC)nnn2)CCCC2(C1)CC(O)C2 9580,C1(c2ccccc2)(C(=O)NCCSC(C)C)CCN(C(c2nncn2C)C)C1 9581,C1(NC(c2cc(CC)ncn2)=O)CCC(C)N(C(=O)CNC(=O)C(F)(F)F)C1 9582,Cc1ncc(Cl)cc1CC(=O)NC1CC(F)(F)CC1NC(c1ccon1)=O 9583,C=C1CCN(C(=O)CN2CCOC2=O)C(C(=O)NC2CCCNC2=O)C1 9584,N1(C(C(n2ncc(C)c2)C)=O)CCC(N(C(=O)C=Cc2cn(C)nn2)C)CC1 9585,C1(CC(=O)NCC2(COC)CCCO2)COCCN1C(C1CN(C2CC2)C1)=O 9586,c1(C(N(CCNC(C2C3COCC23)=O)CC)=O)cc2c(s1)CCCC2 9587,c1(CC)nnc2cc(N3CCN(C(c4ccn(CC#N)n4)=O)CC3C)ncn12 9588,C(=O)(C(CC(C)CC)NC(C1CCC(=O)CC1C)=O)NCC(=O)OCC=C 9589,C1(N(C)C)COC2(C1)CN(C(=O)CCC(=O)Nc1ccncc1Br)C2 9590,c1(N(CCCCN(C(CCCN(C)C)=O)C)C)cc2nncn2cn1 9591,CC(C)CC(O)C(C)C(=O)NC1CC(CC(N2CCC2C(C)C)=O)C1 9592,O=C(NN1C=NC=NOC1=O)C1CCCCN1C(C1CCCC1O)=O 9593,C1(NC(CN(C)CCNC(=O)CSC(F)F)=O)C2CCCCC12 9594,c1(C(N(C(C)CN(C(=O)COC2CCOC2)C)C)=O)[nH]cc2c1CCCC2 9595,CN=c1[nH]cc(C(=O)OCc2cnccc2C2CC2)s1 9596,c1(C(=O)NCC(C)CNC(C2COC(=O)N2)=O)nc2ncccn2n1 9597,c1(C(=O)NC2(C)CN(C(Cc3cc(C(C)C)no3)=O)C2)ccc2[nH]ccc2n1 9598,N1(C(c2cc(OCC)no2)=O)CC(C)CC1C(=O)NC1CN(C2CCC2)C1 9599,c1(C(N(CCCCN(C)C(c2c[nH]c(=N)s2)=O)C)=O)cc(=O)cc(Cl)[nH]1 9600,Cc1cc(NC(=O)C(N2CCC(NC(C3CN(C)C3)=O)C2)C)ccc1F 9601,c1(OC(C)C)cccc(CC(=O)NCC(C)NC(=O)C=C(Cl)Cl)c1Cl 9602,c1(C(=O)NC(C(C)C)CNC(=O)CCc2ncccn2)ccc(N)c([N+](=O)[O-])c1 9603,CC1(CC(=O)N(CCN=[N+]=[N-])CC(C2CC2)NC(C)=O)CCS(=O)(=O)N1 9604,C(=O)(C(C)(F)C(F)(F)F)N(CCCCCCNC(C(N1CCCCCC1)C)=O)C 9605,N1(C(C2CC(C)(C)C2)=O)CCC(C(N2C3CCC2CC(CO)C3)=O)CC1(C)C 9606,Cc1ccc(NC(=O)NCc2ccc(Cl)s2)cc1N(C)C 9607,Cc1ccc(=O)n(CC(N2CCN(C(C3(Cl)CC3)=O)CC2CC2CC2)=O)c1 9608,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)OCCC2)=O)c(C)nc2ccccn12 9609,C(C(O)C(=O)NC1(CC=CC(=O)NCC2CC23CCC3)CCC1)SC 9610,Cc1cc(C(=O)NC2(CCC(=O)NC3CCCN(C)C3C)CCC2)nc(C)n1 9611,c1(C(C)=O)cc(NC2CC(F)(CNC(=O)C(F)C3CCOC3)C2)ncc1[N+](=O)[O-] 9612,N1(C(C(CC#C)C)=O)CC2CCCC2(NC(=O)CSc2ccc(C)cc2)C1 9613,c1(C(C(=O)NCC(C)C)N(C(C#C)C)C)cc(C)nnc1C.C1CC1 9614,C1(C(=O)NCC2CCN(C(c3nnn(C)n3)=O)CC2)CCC2(CCCC2)CC1 9615,n1(CCC(C)C)nc(C2OCCc3ccccc32)nc1-c1coc2c(F)cccc12 9616,CC(=O)CCC(=O)N1CCCCC1C(=O)NCC(C)(O)C1CCCC1 9617,N1(C(C2CN(C(C)=O)C2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)CCC1C 9618,N1(C(c2c(C)cc(O)nc2)=O)CC(N=c2ccnc(Cl)[nH]2)C2(CCC2)C1 9619,O=C(C1CCCc2ncnn21)NCCC(F)Cn1cc(CC2(O)COC2)nn1 9620,c1(C(=O)NCC2(C)CCC(NC(C3(CF)CCC3)=O)C2)cc(F)c(F)c(O)c1F 9621,C1(CN(C(C2CCC(OC)C2)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1 9622,c1(OC)cccc(C(=O)Oc2nccs2)n1.C12(CCC1)C(=O)CO2.C1(=O)CN1.CO 9623,C(=O)(C(CC=C)C(C)C)N1CCC(CCC(N2C(C#C)CCCC2)=O)C1 9624,C1(CNC(c2cc(SC)oc2C)=O)CCN(C(c2cc(N)cc(F)c2)=O)C(C)C1 9625,N1(C(=O)CC2CCN(C(c3n[nH]cc3Br)=O)CC2)CCC(F)(F)CC1 9626,c1(C(C)NC(=O)NC2(c3cccs3)CCCCC2)cc(Cl)ccc1Cl 9627,CC1(CCNC(C2(O)CC(CN(C)C)C2)=O)CCN(C(=O)CSc2nc[nH]n2)C1 9628,n1(CC(=O)N(C2CN(C(C3CCOC(=O)CC3)=O)C2)C)[nH]cc2c(=O)ncnc1-2 9629,CC1CC(C(N2C(C(=O)Nc3ccccc3)CC2C)=O)CCC1=O 9630,c1(Cc2scc(C(=O)NC3CC(C)(NC(C(C)CO)=O)C3)n2)cccc(Cl)c1 9631,N#Cc1ccc(C(=O)NC2CCCN(C(c3csnn3)=O)C2)c(F)c1 9632,N1(C(C=CC(=O)OCC)=O)CC(CNC(=O)C2=C(C)OCC2)CC1(C)C 9633,Cc1oc(C)c(C(=O)NCC2CN(C(=O)CC34COC(C)(C3)C4)CCN2C)c1C 9634,C12(NC(c3c(F)ccc(OC)c3)=O)CCOCC1CNC2 9635,C12(NC(C3(NC(=O)OC(C)(C)C)CC4CCC3C4)=O)CC3CC(C1)C(O)C(C3)C2 9636,c1(C2(N(C(=O)CCn3cc(-c4ccccc4N)nn3)C)CC2)ccc(F)cc1F 9637,N1(C(C2(Cl)C(C(C)=O)C2)=O)CC2CC2(CNC(C2CC2c2c(C)coc2C)=O)C1 9638,C1(C(=O)NC(c2cn(C)nn2)C(=O)NC(C(C)SC)C)CC12CCCC2 9639,C1(C(N(CC)CC2CCCC2O)=O)CCC(CNC(c2cnnc(O)c2)=O)CC1 9640,C1(NC(c2c(CC)ocn2)=O)CCC(C(=O)NCC(=O)N2CCC2)CC1 9641,C(=O)(C1=NNC(=O)C1)N.C(CCC(=O)C(N1C(C)C1=O)CC)OCCC 9642,C=CCC(CC(=O)NCCC(O)C(C)CC)NC(=O)CNC(=O)CC 9643,C#CCCC(C(=O)N1CC(C)(OCC)C1)NC(=O)C(COC)CSC 9644,C1(C)(CNC(c2ccc(C)c(Cl)c2)c2n(C(CCCCC)C)nnn2)CCCN(C)C1 9645,c1(C(=O)NCC(C)N(C(C(CCCC)C)=O)C)cc(=O)c2cc(Cl)ccc2o1 9646,C=CCN=C(NCC(C)(C)COC)N(C)CC12CC(C)(CO1)C2 9647,c1(C(C)(C)OC)ccc(C(=O)NCCC(C)NC(c2nocc2Cl)=O)cc1 9648,C12(C(=O)NCC3N(CC)CCC3)COCC1CN(C(=O)Cc1ccn(C)c1)C2 9649,c1(OC)cc(F)c(C(c2nnnn2C2CCOC2)NC2(C)CCSCC2)c(F)c1 9650,C1(C(=O)NC(CC)(C)CC)CN(C(=O)C(O)C(C)C)CC1(F)F 9651,C1(NC(CN(C(=O)OC)C)=O)CC2CCC(C1)N2C(=O)Cc1sccc1Cl 9652,C(=O)(C(CCOC)OC)N1CC(CC=C)(NC(c2sccc2CO)=O)C1 9653,N1(C(CC(C(F)F)NC(C2(C)C(C)(C)C2(C)C)=O)=O)CCC(O)(C2CC2)CC1 9654,C(C(C)(C)C(=O)NCC1(CNC(C2COCCN2C(C)C)=O)CC12CCC2)OC 9655,c1(NCCC2(C=C)CCC2)ccc2c(c1)C(=O)N(CC1(S(C)=O)CC(C)C1)C2=O 9656,C1(N(C(CCOCCC)=O)C)CCCN(C(c2cccc(C)c2Br)=O)CC1 9657,CC(C)(C)C(=O)N(CC(=O)NCC(O)CNC(=O)CCN1CCCC1)C1CC1 9658,CCCCCCOCC(=O)NCC(C)(C)CNC(=O)CCc1ccn(C)c1 9659,c1(-c2ccc(COC)s2)csc(=Nc2ccc(C#N)cc2)n1C1COCC1C 9660,C=CCC(C)C(=O)N(C(C)CCNC(=O)CNC(c1ccco1)=O)C 9661,N1(C(c2c(C(C)C)cco2)=O)CC2CC3CC2C1C3NC(=O)C=C1CC1 9662,C1(C(=O)NC2CCC(CNC(c3cn(SCC)nc3)=O)CC2)CC2CC1CC2O 9663,C1(CN=c2[nH]cnc(Cl)c2C(C)=O)(OCCC)CC2(CCOCC2)C1.C1C(=O)N1 9664,C1(CCOC)(C(=O)NC(C)CF)CCN(C(=O)CC2CCC(=O)C2)CC1 9665,C1(NC(CC2(OC)CCC2)=O)CN(C(C2CCCO2)=O)CC1O 9666,c1(C(=O)NC(CN(C(c2cccc(C)n2)=O)C)C)cn2c(n1)C(C)CCC2 9667,N1(C(CCC(CC)OC)=O)CCC(C)(C)C(NC(c2ccc3scnc3c2)=O)C1 9668,c1(C(N2CCC(N(C(=O)C(F)C(F)(F)F)CCCC)CC2)=O)c(C)cc(C)nc1C 9669,CC(C)(C)CC(O)CC(=O)NC1CCN(C(c2ccc(F)c(N)c2)=O)CC1O 9670,C1(OCC(=O)N(CCCNC(C(CCSC)O)=O)CCO)CCC(F)(F)CC1 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9741,c1(OC)cn(C)c(C(N2CCC(C(F)CNC(C3CC3Cl)=O)CC2)=O)cc1=O 9742,c1(OC)cc(C(=O)Nc2cscc2-c2cn(CCCCF)nn2)ccc1C 9743,c1(NC(=O)C2CC2)ccccc1Sc1ccsn1 9744,CC1CN(C(=O)CC2CCCN2C(C2CC(=O)OC2(C)C)=O)C(C)C1C 9745,C1(CCNC(C2CN(C3CC3)C2)=O)CCN(C(=O)CNC2CCSC2)CC1(F)F 9746,N1(C(C2=CCCC2C)=O)CCC2CC2(C(=O)NCCOC2CC2(F)F)CC1 9747,c1(SCC(=O)NC2C3CN(C(C(CC)(C)OC)=O)C2C3)nc2ccccc2s1 9748,c1(C(=O)NC(C(=O)NC(CNC(=O)OC)C)C)ccc(C)cc1 9749,NC(CCc1ccoc1)C(=O)NC(c1ccccc1F)C1CC2CCC1C2 9750,N1(C(CC2C(C)(C)OCC2)=O)CCC2CCCC12OCC(=O)NOCC(F)F 9751,C(=O)(C(C(C)(C)C)NC(=O)CC(O)CN(C)C)N(C1CC(O)C1)C 9752,C1(NCC)CCC(C(=O)NCC(O)CN(C)C(C2CC(OC(C)=O)C2)=O)CC1 9753,N(C(=NCCCCl)NCc1nc2c(s1)COCC2)CC1CCN(C(C)=O)CC1 9754,C(=O)(C1=NOC(C)C1C)NCC1OCCCN(C(c2c(OC)cncc2)=O)C1 9755,C1(CNC(C2(CC=C)CN(C(c3n[nH]c4c3COC4)=O)C2)=O)CC2OC1C1CC21 9756,c1(C(N(CC(N)=O)C)=O)cnn2c(-c3ccc(Cl)cc3)ccnc12 9757,CC1=C(C(=O)NC2(C)CN(C(=O)CC3=CCOCC3)C2)COCC1 9758,c1(N(C)CC2CCOC2)nnc(C(F)(F)C2CC2)n1CC1(F)CCCC1 9759,CC1CC(CNC(=O)C(C)NC(N)=O)CCN1C(c1cncn1C)=O 9760,C1(O)(C(=O)NC(CC=C)CNC(c2csnn2)=O)CCCC(C)(C)C1 9761,c1(C(=O)NC(c2cncn2C)C(=O)NC(c2cccs2)CC)ccc(O)c(F)c1 9762,c1(SC)ccc(C)c(C(=O)N(CCCCN(C(=O)CCCCCF)C)C)c1 9763,C1(CC(=O)NCC(C(C)C)NC(C=CC)=O)CCN(C2CCSC2)CC1 9764,C=C(Cl)CC(C(=O)N1CC(O)(C2CC2)C1)NC(c1ccc[nH]1)=O 9765,N1(C(CCN(C)C(C2COCCO2)=O)=O)CCC([N+](=O)[O-])CC1 9766,N1(C(C)C(=O)NCC2(C)CCC(C)C2)CC2CCCC(NC(c3ccco3)=O)C2C1 9767,N1(C(C(C)C)=O)CCCC(NC(=O)C(C)(c2ccccc2)C2CC2)CC1 9768,c1(C(N2CCCC(N(C(=O)Cc3cc[nH]n3)CC)C2)=O)ccc(C)c(Cl)c1 9769,C(=O)(C(C)C(C)NC(c1occ(CC)c1C)=O)NCc1c(CC)c[nH]n1 9770,C(=O)(C#CC1CCCOC1)NC1(C)CN(C(c2c(C)ncn2C)=O)C1 9771,C1(CC)(CO)CCN(C(C2C3CCN(C(=O)C(F)=C(C)C)CC23)=O)CC1 9772,c1(C(=O)NCC(CC)N(C)C(c2coc(O)n2)=O)ccc2occc2c1 9773,N12CCN(CC1CC(F)F)C(=O)N(CC=C)CC2=O.C1(=O)CN1C.OC 9774,c1(C(=O)NC23CC(NC(CCc4cc(C)[nH]n4)=O)(C2)C3)ccc2c(n1)CCCC2 9775,CC1CC(CNC(=O)CCn2cccc2)CN1C(=O)CCc1ccnc(Cl)c1 9776,C1(OC)CCC2(CC1)CC2ONC(N1CC(CC#N)C1)=O.N12CCC(CC1)C2 9777,C1(C(N2C(CCNC(C(C)OCC#C)=O)CCC2)=O)CCc2nnnn2CC1 9778,C1(CC(=O)NCC2(OC)CCOC2)CN(C(c2sncc2C)=O)CCC1C 9779,c1(C(=O)N)ccc(OC)cc1.C(C)(C(=O)NCC1(n2cnnn2)CCC1)OCC=C 9780,CCCCS(=O)(=O)N1CCC(C(=O)NC2CC2NC(=O)CNC=O)CC1 9781,C1(F)(C(=O)NC(C=C)CC)CCCN(C(c2cnsn2)=O)C1 9782,C1(C(=O)NC(CC)(C)CC)CN(C(=O)CNc2ccccn2)CCC1O 9783,c1(C(=O)NC2(CF)CCN(C(C3C(C)CCC3)=O)C2)ccc(Cl)c(F)c1N 9784,c1(NCc2cncc(OC)c2)ncc(C)cc1S(=O)(=O)N1CC(C#N)(CCF)C1 9785,C(=O)(C(CCC(C)C)NC(=O)Cc1cc[nH]c1)N1CCC(C)(OC)C1 9786,C1(CNC(Cc2ccc(C)nc2)=O)CN(C(=O)CC2CC2C)CC(C)(C)O1 9787,c1(C(N2CCC(NC(c3ccc(C(N)=O)cc3)=O)C2)=O)ccc(O)c(F)c1 9788,C1(C(=O)NC(c2ncc[nH]2)CO)(CC)CCN(C(c2cc(Cl)no2)=O)C1 9789,C1(CNC(c2ccc(C)s2)=O)CCc2nc(NC(=O)C(CO)NC(N)=O)sc2C1 9790,C#CC1CC2(C1)NC(=O)N(c1ccc(OCC(F)(F)F)s1)C2=O 9791,N1(C(CC(=C=C)C)=O)CCN(C)C(CNC(=O)C=CC(N2CCOCC2)=O)C1 9792,C(C)(CCC(=O)NC1CN(C(c2ccncc2C(F)(F)F)=O)C1)OC 9793,Cc1nc(N)cc(C(N2CCN(C(=O)C(O)CN(C)C)CC2CO)=O)c1C 9794,C1(C(=O)NCC2N(C(CCC(C)C#N)=O)CC(F)(F)C2)CCS(=O)(=O)C12CCC2 9795,CCN=C(NCc1n(C2CCC(C)(C)CC2)c(O)nn1)N1CCCC2(CCSC2)C1 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9884,C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(=O)Cc1n[nH]c(C)n1 9885,N1(C(CS(=O)(=O)NC)=O)CC2C3CCC(C2C1)N(C(c1ccc(C)nc1N)=O)C3 9886,S(=O)(=O)(c1ccc(Br)c(OC)c1)NC1C(NC(c2cc(OC)c(F)cc2F)=O)C1 9887,C1(NC(C2CC3CCC(C2)C3O)=O)CC2CN(C(C3CC(O)C3)=O)CC2C1 9888,CC1CCC(C(N2CC(O)(C(F)(F)F)C2)=O)CN1C(c1cncnc1)=O 9889,N1(C(C(CC=CCC)C)=O)CCC(C(N2C3CCC2CC(OC)C3)=O)CC1(C)C 9890,N1(C(c2cc(CC)no2)=O)CCC(C2CCN(C(=O)CCCC(F)F)CC2)CC1 9891,C1(C(=O)NC(CC)CNC(=O)C(C)(C)COC(C)C)CCc2n[nH]cc2C1C 9892,c1(C(=O)NCC2(F)CC(NC(CC3CC(=O)NC3)=O)C2)csc2nnsc12 9893,C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1c[nH]ccc1=O)=O 9894,C1(CC(=O)NCC#CCOC)CCC(C)(C)OC1.C1(=O)CCCN1 9895,C1(CC)CN(C(=O)Cc2ccc(O)cc2)CCC1NC(c1ncc(C)cn1)=O 9896,N1(CC(C)NC(COCC)=O)C2CCC1CN(C(c1ccccc1OC)=O)CC2 9897,C12(CNC(=O)Cc3cnn[nH]3)CCCC1N(C(=O)CN1CCCCC1=O)CCC2 9898,C=C1CC2(C1)C(=O)NC2.C1(CC(C)SC2CCC2)CN(C(=O)COCC)C1 9899,CCC(C)CC(CO)NC(=O)Nc1ccc(-n2cncn2)cc1C 9900,C(C)(C(C)(C)CO)NC(C1C(CNC(C2(CC)CCCC2)=O)CCC1)=O 9901,Cc1nn(CC(N2CCC(NC(=O)COCC3CCOC3)C2C)=O)cc1[N+](=O)[O-] 9902,C1(NC(c2cnsc2)=O)CC2CCC1N2C(=O)COc1ccc(F)nc1 9903,c1(C(=O)NCc2c(CC)noc2)cccc(CNC(C2CCC3(CC3)C2)=O)n1 9904,N1(C(c2c(C)cc(Cl)cc2C)=O)CC2CC3CC2C1C3NC(=O)COC(F)(F)F 9905,N1(C(CCCOCCC)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)CC 9906,N1(C(C(C)C#N)=O)CC(F)(F)CC1CCNC(c1ccc(C(C)(C)C)cn1)=O 9907,C(CCCC(CO)NC(=O)Cc1cnn(C)c1)NC(C1(N(C)C)CC1)=O 9908,N1(C(COC)CNC(=O)CCn2ccnc2C(C)C)CC2CCC1C(C(=O)O)C2 9909,C=CCN=C(NCCN1CCOCC1)NCC1(COC)CC1c1nccn1C 9910,Cc1cc(C)n(C(C)CC(=O)NCCC(C)NC(=O)CSCc2ccccc2)n1 9911,C(=O)(CC(=O)NCC1C(C(=O)NC2CCC2(C)C)C1(C)C)N(C)C 9912,N1(C(c2c(CC)oc(C)c2)=O)CCCC(NC(c2cc(C)[nH]c2C)=O)C1CC 9913,C(=O)(C1=CC2(CCOC2)C1)NCC1C(C)(C)CCN1C(=O)CCC(CF)CF 9914,c1(C(N2CC(NC(CCC=CC)=O)C(O)C2)=O)ccc2snnc2c1 9915,CCC(CC(=O)OC)NC(=O)C(CC1CCCCC1)OC 9916,C(=O)(C1=CC2CCCCCC12)N(C)CC1(CNC(c2ccc(C)o2)=O)CC1 9917,c1(C(=O)NC(c2cc3ccccc3[nH]2)C)nccc2c1CCOC2 9918,Cc1cc(C(=O)NCCC(C)NC(=O)C(C)C#N)n[nH]1 9919,N1(C(C(C)OC2CCCCC2)=O)CC(F)(F)CC1(C)CNC(c1csc(Cl)n1)=O 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9938,C1(C(N2CC(C(C)NC(C3(O)CCOCC3)=O)OCC2)=O)CC(F)(F)C1(C)C 9939,c1(NC(C2CCCCO2)CC)cccc(C(=O)O)c1OCC 9940,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(c2sc(F)cc2Cl)=O)CC1 9941,c1(C(N2CCOCC(NC(c3c(COC)cco3)=O)C2)=O)ccc2c(c1)CCC2 9942,N1(C(C(CCCNC(=O)NCc2nc(C(C)(C)C)sc2)O)=O)CCc2ccccc21 9943,C1(NC(=O)CNc2ncccn2)CC(O)CN(C(C23CCCC(CO2)C3)=O)C1 9944,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCCC1CCNC(C1CC12CC2)=O 9945,c1(CNC(CN(C(C2C(CCC)CCCC2)=O)C(C)C)=O)cc2n(n1)CCO2 9946,N1(C(C2C(C)C2)=O)CCCC1(CNC(c1cccs1)=O)CNC(N)=O.C12CN(C1)C2 9947,C1(C)(C(=O)NCC(CC)NC(c2cccc(C(C)(F)F)n2)=O)CCC(=O)NC1 9948,Cc1cnccc1C(=O)NCCSCC(=O)NCCC1CCOC(C)C1 9949,c1(C(N(C)C)=O)ccc(C2C(=O)N2)cc1.C12(C(=O)NC(C)(C)C)CC(C1)NC2=O 9950,C(CCCCCC(=O)N1CCCC(CF)C1)NC(c1c(=N)[nH][nH]c1)=O 9951,c1(C(C)NC(=O)CN(C)C2CC2)ccc(NC(=O)C2=COCC2)cc1 9952,C(=O)(C1=NOC(CNC(=O)C2=C(C)CC2)C1)NCc1cc(OC)nn1C 9953,C(CCC1(C)CC1)(C(=O)NCCC1CC1)N(C(COCC)C)C 9954,C(=O)(CC(C)(C)C(=O)NC1COCCC1C(=O)NCCCS(C)=O)OC 9955,c1(C(N2CCC(CCCC)CC2)C(=O)NC2CCOC2)ccc(Cl)c(OC)c1 9956,N1(C(C(C=CC)O)=O)CCC(c2ccc(CNC(=O)C(=O)NCC)nc2)CC1 9957,N1(C(CCC2CCN(C(C3(OC)CCOC3)=O)CC2)=O)CC2C(C1)C2(F)F 9958,C1(CNC(c2c[nH]cc2Br)=O)C2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 9959,C1(NC(C2(NC(C)C)CC2)=O)CN(C(c2cncc(Cl)n2)=O)Cc2nccn2C1 9960,c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)nnc2n1CCCCC2 9961,n1(CC(=O)NCCC2CCC(NC(=O)COC3CCCCC3)C2)cccnc1=O 9962,CCC(CC1CC1)C(=O)N(C)CCOCCNC(=O)C(=O)Nc1ccc(Cl)cc1 9963,CS(=O)(=O)CCCC(=O)N1CCN(C(c2cnc3n2CCC3)=O)C(C2CC2)C1 9964,n1(CC)nnc(C(=O)OCCSC2CCC(=O)N2C(=O)CCC=CBr)c1C 9965,C1(CC(=O)NCCc2cc(C(=O)NC(C3CSC3)C)no2)CCCCC1C 9966,N1(C(CCc2c(C)ccs2)=O)CCOC(CC(N2CCC(C(F)F)CC2)=O)C1 9967,N1(C(C23CCOCC4C2C3C4(c2c(C)nn(C)c2Cl)OC)=O)CCN(C(C)=O)CC1C 9968,C1(C(=O)N(CC(C)O)C)(CNC(C2C(C(=O)OC)C2)=O)CCCC1 9969,N1(C(C2(C)CCC2)=O)CCC2(CCCN2C(=O)CS(=O)C(F)(F)F)C1 9970,c1(C2C(=O)NCCN2CC2CC2)nc(C(C)(C)C)cs1.c1ccccc1.CC(C)C 9971,c1(CC)cccc(CC)c1CC(=O)N(C)CC1CCCN1C(C1CCOC1C)=O 9972,N1(C(c2c(CC)nco2)=O)CC2OCCN(C(=O)C(C)C(O)C(C)C)C2C1 9973,CC1(c2cn(CCCF)nn2)CCN(CCO)CC1.C1(NCCC#N)CCCCC1O 9974,Cc1cc(NC(c2nccnc2Br)=O)n(C2CCOC2)n1 9975,N12CCCC(C1)N(C(=O)C(C)C)C1(CC1)C2=O.C(C(C)C)NC(C)=O 9976,CC1N(C(C(c2cccc(Cl)c2)CCc2ccc(Cl)cc2)=O)CC(C)OC1(C)C 9977,C1(C(N2CCC(NC(C3CN(S(CC)(=O)=O)C3)=O)C2C)=O)CCc2c[nH]nc2C1 9978,C12CCCCN1C(=O)C21CC1.c1(C(N2CCC(N)C2)=O)sccc1CC#N.CCC 9979,c1(C(=O)NCC2C(CNC(Cc3ccc(CCC)cc3)=O)C2)ccc(F)cc1O 9980,C1(NC(N(C(C)C)CCc2ccsc2C)=O)CC=CCN1C(=O)OC(C)(C)C 9981,C(=O)(CCCCCCC)NCCc1cc(C(=O)NCC(CCOC)(C)O)no1 9982,c1(-c2cc(C(N(CCN(C(C3C(C)C3)=O)C)C)=O)sc2)cccc(F)c1 9983,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 9984,O=C1CCC(C(=O)NC2CC3CCC2N3C(C2CC2F)=O)=NN1 9985,N1(C(=O)C(F)(F)c2ccncc2)CCC2(CC1)CCN(c1ncc3ccnc-3[nH]1)C2 9986,C(C1=CCN(CCC(=O)OC(C)(C)C)CC1)NC(CCCCOC)=O 9987,C(=O)(C(C)CC(C)(F)F)N1CCC(O)(CNC(c2c(C)n[nH]c2C)=O)C1 9988,C1(N(c2ccc(Cl)cc2F)CC)CCCN(Cc2cn(C(C)CO)nn2)CC1 9989,C(CO)(CCCCNC(c1ocnc1C1CC1)=O)NC(C1(CC)CC=CCC1)=O 9990,C(C(C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCSC2CCCC2)C1)OCC 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10009,c1(C(N2CC3C(NC(C4CCC(C)O4)=O)(C3)C2)=O)cc2c(Cl)nccc2s1 10010,CS(=O)(=O)c1cccc(C(=O)NCC(O)CNC(c2ccccc2)=O)c1F 10011,C1(C(N(C)C2CC2)=O)CNC(=O)C12CCN(C(=O)C(C)(O)C(F)(F)F)CC2 10012,CCCC(O)CC(=O)NC(CNC(c1nc(C)ccc1F)=O)CC 10013,C1(CCOC)(NC(=O)CN(C)C)CCN(C(C2CCNC(=O)C2)=O)C1 10014,c1(NC(C23CC(NC(C4COCCO4)=O)C(OC2)C3)=O)cn2ccccc2n1 10015,CC(CCC(C)(C)C)C(=O)NCC(C(=O)N1CC(CO)C(O)C1)C(C)(C)C 10016,C1(C(N2CC(Cn3cc(CCNC(N)=O)nn3)OCC2)=O)CC2(C1)CC2(F)F 10017,N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(=O)C(C)=CC1CC1 10018,c1(C(N(CCNC(C=C(C)C2CC2)=O)CC2CC2)=O)nc2nc(C)ccn2n1 10019,C#CCC(CC(=O)NCCC(O)CC(=O)OC)NC(=O)CC=C(C)C 10020,C(C(C)(C)C(=O)NCC1(CCNC(=O)C(C2CCCCC2)=O)CCCC1)SC 10021,c1(C(=O)NC2CCCN(C(=O)C(O)C(F)(F)F)C2)ccc(F)c(C(F)(F)F)c1Cl 10022,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)C(NC(C2CCCS2)=O)C1C 10023,N1(C(CCC(=O)NC)=O)CCN(C(=O)C(C(C)C)OC)CC(C)(F)C1 10024,N1(C(C(C)=C2CCCC2)=O)CCCC(CNC(c2c(C)noc2C2CC2)=O)C1 10025,c1(C(C)=O)cccc(SCC2(F)CN(C(C3CC(CCF)C3)=O)C2)c1.C1C(=O)N1 10026,C1(C(=O)NC(CC)CNC(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10027,c1(C(N2CCN2C(=O)NCc2c(C)ccs2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1C 10028,Cc1ccc2nnc(CCNC(=O)NCC3CC4CCCC4C3)n2c1 10029,N1(CC(N2C(C(C)NC(c3ccccc3)=O)CCC2)=O)CCCN(CCOC)CC1 10030,C1(C#N)(CC(=O)N(CCCNC(=O)C(C)CC2CC2)CC)CCOCC1 10031,C(=O)(C(CC(C)C)Sc1ccccc1)N(CCN(C(=O)C(O)C1CC1)CC)CC 10032,C1(F)(C(c2nnnn2CCC2(C)CC2)N(CCCCOc2cccs2)C)CCCC1 10033,c1(CC(=O)NCC(c2ccccc2)NC(C2N(CC)CCC2)=O)ccnc(O)c1 10034,N#CC1CN(C(c2ccc(CCF)cc2)=O)CCN1C(C1(CC#N)COC1)=O 10035,CCCCC(O)CC(=O)NCC1CCC(C(=O)NCC2CC2CC)O1 10036,C12C3CCC1CN(C3)C2=O.C1(NCC2(CS(C)(=O)=O)CC2)CCC(=O)N1 10037,C(C(F)(F)C(=O)NCC1(NC(C2(CO)CC2)=O)CCOC1)OC 10038,N1(C(Cc2nc(C)[nH]n2)=O)CCN(CCNC(c2cc(C#N)no2)=O)CC1 10039,N1(C(C=COCC)=O)CCCC(N(C(=O)CCOCC2CCC2)C)C1 10040,N1(C(c2nccc(C(C)C)c2)=O)CC2(C1)CN(C(=O)CCS(C)=O)CC2CO 10041,c1(OC)ccc(-c2nc(C)c(CNC3(CO)CC(c4ccccc4)C3)[nH]2)cc1 10042,c1(OC)cc(C)cnc1COC(C1(C(F)(F)F)CCCCCC1)=O 10043,N#Cc1c(F)cc(C(=O)NC2CCC(NC(=O)C3=CSCS3)C2)cc1F 10044,Cc1ccc(F)c(-c2ccc(C3CCN(C(=O)NC(C)CC(=O)O)CC3)cc2)n1 10045,C(C(C)(C)CCCc1nc(-c2ccco2)nn1CCC(F)(F)F)OCC 10046,Cc1ccc(C(c2ccnc(OCO)c2)NC(C2(CO)CC2)=O)cc1 10047,N1(C(CC(CC)SC)=O)CCC2(CC(NC(c3csc(O)n3)=O)C2)C1 10048,C(=O)(C1=C(CCl)N(c2cccc(Cl)c2)C(=S)NC1c1ccc(=O)n(C)c1)OCC 10049,C(=O)(C#CC1CCOC1)NCC1C(C(=O)NC2C(C)(C)C2(C)C)CC1 10050,C(=O)(NNC(=O)CCC(=O)NNc1cccc(C)c1)c1c(OC)cccc1 10051,C(=O)(C(CN=[N+]=[N-])NC(=O)CN1CCN(C)CC1)N(CC=C)C 10052,CCCC(C(=O)NCC1CCN1Cc1csc(CC)n1)OCC 10053,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10054,Cc1cc(CN2CCCC3(CCC3O)C2)n2ncnc2n1 10055,N1(C(C2CCC(C#N)C2)=O)CCC2(C1)CN(C(=O)CCc1cc(Cl)cs1)CCO2 10056,N1(C(CNC=O)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10057,C1(NC(CCC#CC)=O)CC2(NC(c3sc(C(C)OC)nc3C)=O)COC1C2 10058,C1(C)(CCNC(C(C)O)=O)CCN(C(c2ccc(-c3cccnc3)cc2)=O)C1 10059,c1(C(=O)O)cccc(CN2CCC(C(N3CCC(Br)C3)=O)C2)c1.NCCO 10060,Cc1ccc2c(C(=O)NC3(CCCCNC(=O)CCCS(C)(=O)=O)CC3)c[nH]c2c1 10061,C1(NC(C(C)=CC)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1CO 10062,C=C(C)CCC(=O)N(C1CC(NC(=O)C(CCC)c2cccc(Cl)c2)C1)C 10063,N1(C(Cc2ccc(C)nc2)=O)CCN(C)C(C(C)C)C1.C1CCCC(=O)N1 10064,N1(C(c2c(C)cccc2C)=O)CC2(C1)CN(C(C1CCSCC1)=O)CC2CO 10065,C1(C(N2CC(C)(O)C2)=O)(CF)CCN(C(=O)CCC2CCC2)C1 10066,CC(C(O)C(F)F)NC(C1CC2CC2N1C(c1cccc(CC#N)c1)=O)=O 10067,c1(C(N2CCCCC2c2ccc(C)o2)C(=O)NC(CC)C)cc(Br)ccc1F 10068,CC1(C)C(c2cn(C(C)(C)C(=O)O)nn2)CCN1C(=O)C(CO)N1CCOCC1 10069,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10070,CN1CCCC1(C)C(=O)NCCOC1CN(C(=O)CC2CCCS2(=O)=O)C1 10071,C(=O)(C#CC1CCCO1)NCCCOCCOC1(F)CC1.O=C1CN1 10072,C1(C(=O)NCCCCNC(C(C)CN2CCOCC2)=O)Cc2ccc(F)cc2O1 10073,C1(c2ccccc2)(NC(C(C)C2CCC2)=O)CCN(C(=O)COC2CC2)C1 10074,c1(C(N2CCC(N(C)C(c3cocn3)=O)C2)=O)ccc2[nH]c(=N)ccc2c1 10075,c1(C(N2CC(NC(C3(O)CCOC3)=O)CC(C)(C)C2)=O)cnnc2ccccc12 10076,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CCc2cnccn2)C1C 10077,c1(C(=O)OCC)csc(Cl)c1NC(=O)CC1CCC(C(N)=O)O1 10078,c1(OC)ccc(O)cc1C(=O)NC1(C2CCCN2C(C2CCC2OC)=O)CC1 10079,c1(C(N2CC(NC(c3c(C)nccc3)=O)C(O)C2)=O)cc(C2CC2)nnc1O 10080,c1(C(=O)NCC2CCN(C(c3c(CN(C)C)cco3)=O)C2)cncnc1O 10081,n1(CC(CC)CC)nc(CS(C)(=O)=O)nc1-c1ccc(OC(C2CCC2)C)cc1 10082,CC(CCN(C(=O)CCC1OCCO1)C)NC(=O)Cc1nc[nH]n1 10083,Cc1cccc(N2CCC(NC(=O)CC3(C)CCOC3)C2=O)c1 10084,N1(C(c2cn(CCCl)nn2)=O)CCC2CN(C(C3CC(C4CCC4)C3)=O)C2C1 10085,C1(CC(NOCC=C)=O)(OC)CCN(C(=O)C(C)n2cccc2)CC1 10086,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10087,C1(C(=O)NC(C)CCNC(C2(O)COC2)=O)COCOC1 10088,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10089,CC(=O)CCCC(=O)N(CC(=O)NCC1CC(O)C1(C)C)C(C)C 10090,C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccc(O)nn2)=O)CCC1CO 10091,N1(C(c2ncn(C)n2)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)CC12CCCCC2 10092,CCC(C(=O)NCC1(C(C)NC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10093,N1(C(CC=C)=O)CC2CC1C2C(N1C(C)CCC1C)=O 10094,C1(C2CN(C(=O)CSc3ccc(C#N)cc3)C2)(NC(CC(C)CN(C)C)=O)CC1 10095,c1(C(=O)NCc2cccc3cc[nH]c23)cnn2cc(C(F)F)cnc12 10096,c1(C(=O)NC(C(=O)NCc2c(C)scc2)C2CCCC2)cc([N+](=O)[O-])n[nH]1 10097,CC1CC(C2CN(C(=O)CN(C(C3OCCCC3(C)C)=O)C3CC3)C2)=NO1 10098,c1(C(N(CCC(=O)N(CC(=O)NCCC)C)CC2CC2)=O)cc(C)c[nH]1 10099,c1(C(=O)NCC(CNC(CCCOCC=C)=O)O)ccc(S(=O)(=O)C(F)F)cc1 10100,Cc1cccc2c(C(N3CCCC3CCNC(C34CCC(CO3)C4)=O)=O)n[nH]c12 10101,c1(C(N2CC(C)CC(NC(Cc3nnc(C)o3)=O)C2)=O)cc2cn[nH]c2cn1 10102,c1(SCC(=O)NC2CC(NC(CC3C(C)(C)C(O)C3)=O)C2)ccccc1[N+](=O)[O-] 10103,CC1C(=O)CC2CCC1N2C(=O)CC(C(C)(C)C)N(C)C 10104,Cn1cc(C2CC2C(=O)NC2(CNC(=O)C(c3cccs3)SC)CCOC2)cn1 10105,c1(C(=O)NCC2CC(COC)CN2C(=O)C(F)F)cccc(Br)c1C 10106,c1(C(N2C(CNC(C(C(C)C)C)=O)CC(O)C2)=O)cc(=O)n(C)cc1Br 10107,c1(OC)ncnc(-c2nn[nH]n2)c1F.N12CCCC1C1(O)CN(C1)CC2=O 10108,C(=O)(C(O)C1=CCCCC1)NC1CCN(C(CC(=O)NCC#C)=O)C1 10109,CCC(C)(CS(C)(=O)=O)C(=O)N(CC(O)CN(C(=O)C(C)OCCN(C)C)C)C 10110,c1(C(=O)NCC2(O)CC(NC(C(CC)N(C)C)=O)C2)cc2c(C#N)cccc2[nH]1 10111,N1(C(COCC#C)=O)CC(C2CCCN(C(C3(CC)CCCO3)=O)C2)C1 10112,N1(C(Cc2c(C)nc[nH]2)=O)CCC(C(F)(F)F)C(NC(C2(C(C)C)CCC2)=O)C1 10113,CN1CCCC(F)(C(=O)NCC2CCN(C(=O)CCc3ccn(C)n3)C2(C)C)C1 10114,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10115,CC(C1OCCc2ccccc21)NCCc1ccccc1F 10116,O=C(C(O)CSc1cccnc1)N1CC(NC(C2C=CCS2)=O)C1 10117,N1(C(Cc2c(C)scc2)=O)CCC(CC(=O)NCCCCCCO)C1(C)C 10118,C1(NC(C2(CCC)CCC2)=O)COCCN(C(=O)C(C)Oc2cccnc2)C1 10119,N12CC=CCC1C(=O)NCC2=O.C(CC(=O)NC(=O)NC)N(CC=C)C 10120,C1(NCc2ccc(OCCCC)nc2)CC2(CCC(NC(C)=O)CC2)C1 10121,n1(CC)nccc1S(=O)(=O)NC1CCC(NC(c2nc(C(=O)OC)n(C)n2)=O)C1 10122,N(C)(S(=O)(=O)N(C)CC1CC1)CC#C 10123,c1(C(CN(C)C)NC(=O)NC(Cc2cncs2)CO)cnn(C)c1 10124,C1(C(=O)NCc2cc(CC)[nH]n2)CCN(C(=O)CC2CCOC2)O1 10125,N1(C(c2c(CC)nc(C)nc2)=O)CCOC2CCN(C(c3ccc(Cl)[nH]3)=O)CC12 10126,C1(CNC(CSCCOC)=O)CN(Cc2scc(C(=O)OC)n2)C2CC12 10127,C(N=c1[nH]c(N(CCC#CBr)C)nc2c1CCCCC2)c1ccc(COC(F)F)cc1 10128,C(=O)(CS(=O)(=O)CCO)N1CCC(NC(CNC(C(CC)C)=O)=O)(CO)C1 10129,N1(C(C(CC)F)=O)CC(C)OC2(CCN(CCOCCOC)CC2)C1 10130,C1(C(=O)NC2CC(CNC(c3c(CC)noc3)=O)C2)CCCCC12OCCO2 10131,c1(OC)ccc(Cc2nc(C3(C)COC3)no2)cc1C#N 10132,c1(NC(C(=O)NC2CCC(C)(CC)C2)(C)C)ncnc2ccc(NC)cc12 10133,C(CCCCC(=O)NC1(CC(C)(C)C)CC1)N(C(=O)CC1CC2(CC2)C1)C 10134,Cc1nsc(NC(C2CC2)=O)c1C(=O)NCC1CC(C)CN1C(=O)CC(C)C 10135,C(CC(C)C(F)(F)F)NC(CC1(O)CCN(C(Cc2cccc(C)c2)=O)C1)=O 10136,C1(CNC(C(CC=C)NC(C)=O)=O)CC(C(=O)NCC2(N(C)C)CCC2)=NO1 10137,N1(C(C(C2CC2)SC)=O)CC(NC(=O)CC2CN(C)C2)C(C)(C)C1 10138,C1(NC(C2CCCOC2c2cn[nH]c2)=O)CC2(CCN(C(=O)CC3CCC3)C2)C1 10139,C1(NC2CCC(CC(=O)NC)C2)CCN(Cc2cccc(OC)c2C)CC1(C)C 10140,c1(C(N2C(C(=O)NCC3CCN(CC)C3)CC=CC2)=O)ccc([N+](=O)[O-])o1 10141,C(=O)(CCCCC(F)(F)F)NC1CC(CNC(=O)CSc2ccoc2)C12CCC2 10142,C(C(C)(C)CC(=O)NCC1(C)CCCO1)OC.C1C(=O)NCCS1 10143,C1(NC(C(C)OC)=O)CCN(C(c2ccc(NC(C)=O)s2)=O)CC1(C)C 10144,CC(C)C(C(=O)NC(CN(C)C(c1cnn(C)c1C1CC1)=O)(CO)CO)NC=O 10145,C(=O)(C1COc2ccccc21)NCCCCN(C(=O)C1Cc2ccc(Cl)cc21)C 10146,N1(C(=O)OCCCn2cc(CC(O)CO)nn2)CCCC(C)(CO)C1.CC(C)C 10147,N1(C(CCc2ncc(CC)o2)=O)CCCCC1CNC(=O)Cn1cnnc1 10148,c1(CCC(=O)Oc2c(OC)ncnc2NC(C)(C)C2CC2)cccc([N+](=O)[O-])c1 10149,N1(C(CCCN(C(=O)OC)C)=O)CCC(COCC)CC1.C12CN(C1)N2.C1CC1 10150,CC(C(=O)NC1(C)CN(C(=O)CN2CCCC2CO)C1)F 10151,Cc1ncc(CNC(c2ccc(-c3ccnn3CCC(C)C)nc2)=O)cc1Br 10152,C(=O)(C1CCc2ccccc21)N1CC2(C1)C(=O)N2.c1(CSC)cc(C)sc1C 10153,C1(COC)(NC(c2cnn(C(C)(C)C)c2)=O)CCCN(C(=O)Cc2ccns2)C1 10154,C#CCCCCCC(=O)N1CC(C2CN(C(C3CCCOCC3)=O)C2)C1 10155,Cc1cc(C(=O)NC2(C(=O)N(CC(C)(C)C)C(C)C)CCCC2C)ncc1N 10156,c1(C(=O)OCC)ccc(S(=O)(=O)N2CCCOC(CO)C2)nc1 10157,c1(C(N2CCN(C(c3c(F)cccc3F)C)C(CO)C2)=O)nccc2nc[nH]c12 10158,c1(C(=O)NCC(C)(c2nc[nH]n2)NC(C2CCC2(F)F)=O)cncc(C(=O)OC)c1 10159,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10160,c1(C(N2CCC(N(C)C)CC2)C(=O)NCC(=C)C)sc(C)c(Br)c1C 10161,C1(C#N)(N)CCN(C(=O)Cn2ccccc2=O)C1.c1(C(=O)OCC)ccc(SC)nc1 10162,C(=O)(CC(C)C(=O)NC(CNC(=O)CN(C)Cc1cccc(F)c1)C(C)C)OC 10163,c1(C(N(CCc2cn(-c3cccc(OCC)n3)nn2)C)=O)ccc2snnc2c1 10164,c1(C(N2C(CNC(CNS(N)(=O)=O)=O)CC(O)C2)=O)cnn2c1CCC2 10165,O=C1CC2(CCC(NC(=O)C(=O)N(CCO)CCO)C2)CN1 10166,CC(CSCc1ccccc1)C(=O)NC(C)CC(=O)N1CCCC1CO 10167,C(=O)(C(CNC(C1(C)CCCC1O)=O)C(C)C)N1CC(Sc2ccc(C)cc2)C1 10168,C1(CNC(C(C)NC(=O)C2CC2)=O)CN(C(=O)CC2(C#N)CC2)CC1C 10169,CCCC(CCC)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1OC 10170,C(C1c2ccccc2C(=O)N1C)OC(COCC(C)C)=O 10171,c1(N(C2CCN(C(c3cnc(SC)s3)=O)C2)C)ncnc2sc(C(F)(F)F)nc12 10172,S(=O)(=O)(C1CCOCC1)N1CC(NC(C)C)(CO)C1.Cc1ccc(O)c(C(=O)O)c1 10173,N1(C(=O)OC(C)(C)C)CC2(CNC(=O)NCCc3cncn3C)OC2C1 10174,n1(CC(=O)NC(C2(O)CCCCC2)C(=O)NC(CCC)CO)ncccc1=O 10175,c1(C(N2CCC(NCCCCOCC)CC2)=O)cnn2cc(OC)ccc12 10176,N1(C(C2(OCC)CCOC2)=O)CCN(CCNC(=O)CC2CCC(C)(C)O2)CC1 10177,C1(N(C(N(c2ccccc2)C)=O)Cc2nccn2C)CC2CC1CN2 10178,c1(COCC)ccccc1NC(=O)NCCN(C(=O)CCc1ccn(C)c1)C 10179,CC(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)CC1)=O)CC(F)(F)F 10180,C1(C(=O)NCC(CNC(Cc2c(C)n[nH]c2)=O)C)CCCN(C(C)C)C1 10181,c1(N2CCOCC(CNC(c3nc(CC)[nH]n3)=O)C2)nnc(C)c(C)c1C#N 10182,c1(SCc2[nH]cc([N+](=O)[O-])c2)ccc(Br)c(Br)n1 10183,CN1CCCC1C=CC(=O)NC1CCC(NC(c2csc(Br)n2)=O)CC1 10184,C12(CNC(c3ccccc3)=O)CCC1CN(C(c1ccc(=O)n(CCO)c1)=O)C2 10185,C1(NC(c2cn(CCOC)nc2)=O)(CO)CCN(C(c2ccnc(S)c2)=O)CC1 10186,N1(C(Cc2cn(CC)nc2)=O)CC(N(C)C)C(CNC(=O)CC2CC=CC2)C1 10187,C1(CCC(=O)Nc2cccc(C)c2C(=O)OC(C)C)CCc2ccccc2C1=O 10188,c1(OC)nsc(NC(=S)NC(n2cc(F)cn2)C)c1C(=O)NC1CCCC1 10189,C1(O)(C(C#C)C)CCN(C(=O)CC2(CC=C)CCOC2)CC1 10190,C12(C(N)=O)CCCN(C(=O)NC3CCC3)CC1C2.n12nccc1SCC2 10191,C1(C(C)C)CCOC1C(=O)NC1CC(N(C(=O)Cc2nncs2)C)C1 10192,C(CCCC(=O)N1CC2C(C)C2C1)NC(COCC)=O 10193,CCS(=O)(=O)CCN(C(=O)CC=CCNC(=O)C(C)CN(C)C)C 10194,c1(C(N2CCCC(CNC(C(C)(C)OCC)=O)C2)=O)cc(Cl)c(OC)cc1C 10195,C(=O)(C(C)N(C(=O)C(C)OCC)CC=C)N(CCCF)CC#C 10196,C(=O)(CC(C)c1cnn(C)c1)NCC(CC)NC(=O)CCCSC(C)(C)C 10197,C(=O)(CC(C(C)C)NC(C1CN(C)CCO1)=O)N(C(CC)CC)C 10198,c1(CNC(N(CC(C)O)C2CCC2)=O)cnc(Cl)s1 10199,N1(C(C2CN(C(C)=O)C2)=O)CCC(CCNC(C2(C)CCCCC2)=O)CC1C 10200,c1(C(N2CC(C)CCC(=O)N3CCC2CC3)=O)cc(N(C)C)ccc1F.CN 10201,N1(C(c2cncc(CC)c2)=O)CCOC2(CCN(C(C3(CSC)CC3)=O)CC2)C1 10202,c1(CN2C(C(=O)NCc3ncccc3F)CSCC2)cc(Cl)ccc1Cl 10203,N1(C(CCC2C(C)C2)=O)C2CCC1CN(C(c1ccns1)=O)C2 10204,Cc1cc(C(=O)NCC(O)CNC(c2cccc(Cl)n2)=O)c2c(C)nn(C)c2n1 10205,c1(NC(C(CC2CCC2)NC(CC(CC)C2CCC2)=O)=O)cnc2ccnn2c1 10206,N1(C(CCOCCCNC(c2nsnc2O)=O)=O)CC23CCC2(COC3)C1 10207,c1(NC(CC2(C)CCN(C(=O)Cc3ccc(CO)cc3)C2)=O)ccc(F)c(O)c1 10208,Cc1nn2c(C(N3CC4CC4(NC(=O)CN(C(=O)C(C)C)C)C3)=O)c(C)nc2s1 10209,CCC(Cc1cccc(C)c1)C(=O)NCC(C(C)C)NC(=O)CC1CC(F)(F)C1 10210,C(=O)(C(C(C)C)c1cccc(OC)c1)NCCN(C(=O)COC)CC 10211,C(=O)(CC(C)C(F)(F)F)NC1CN(C(C(C2CC2)OCC)=O)C(CO)C1 10212,C1(CCNC(CCC#CC)=O)CN(C(C2CC3CCC3C2)=O)CCS1(=O)=O 10213,C1(C(=O)NC2(CC)CC2)C(C2CC2)CCN1C(=O)COC(C)C 10214,C12CCCN(C1=O)C(=O)c1ccc(cc1)CS(=O)(=O)N2C.CN.OC 10215,N1(C(CC2(C(=C)F)CCC2)=O)CCC(C(=O)NCC(Cl)C(C)(F)F)C(C)C1 10216,N1(C(C)C(=O)NC(N2CC(C(=O)NC3CCCC3)C(F)C2)=O)CCC(N(C)C)CC1 10217,C(=O)(CCC(=O)NCCCCCCNC(C1CC1(Br)Br)=O)NCC 10218,C1(NC(C2(C(=O)NC)CCC2)=O)CN(C(c2cc(Cl)ccn2)=O)C2(CCOC2)C1 10219,c1(C(N2C(C)C(NC(=O)CCc3ccccn3)CC2)=O)cc2ncccc2s1 10220,C1(NC(C(CN(C)C)NC(c2cc(CC)sn2)=O)=O)CNC(=O)C12CC2 10221,C#Cc1ccc(C(N2CCCC2CCC(N2CCOC(C(N)=O)C2)=O)=O)cc1 10222,c1(CCC(N2CCC(Cc3cn(CCCCO)nn3)C2)=O)ccc2c(c1)CCO2 10223,C(=O)(C(CC(C)C)C(C)C)NCCN1CCN(C(c2c(N)ccc(C)c2)=O)CC1 10224,Cc1c(CN2CC3(CCN3C(c3cc(Cl)cc(Cl)n3)=O)C2)[nH]c2ccccc12 10225,N1(Cc2cn(C)nc2)CCCCC1C(=O)NCC1CCCS1(=O)=O 10226,C1(C(=O)OC)CN(C(C)=O)CCN1Cc1nc(-c2cccc(Cl)c2)no1 10227,Cc1ccc(C(C)C(=O)NCCC2(CNC(=O)C=CSc3ccccc3)CC2)s1 10228,N1(C(c2cnc(C)[nH]2)=O)CCCC12CCN(C(=O)C(C)CC(C)(F)F)C2 10229,CC(N=[N+]=[N-])C(=O)N1CC(C(=O)NCC2COCC2O)C(C)C1 10230,c1(OCC(N2C(Cn3cc(CN)nn3)CCC2)=O)csc2ccc(F)cc12 10231,c1(C(=O)NC2CC(NC(C3=CCC(C)(C)CC3)=O)C2)cc(Cl)cc2c1NCCC2 10232,N1(C(COCC)=O)CC2(CCN(C(c3cc(OCC)ccc3F)=O)C2)C1 10233,C1(CNC(C2(OC)CC2)=O)C(C)CCCN1C(=O)CCC(=O)c1cccnc1 10234,c1(N2CC3C(CCC)(C(=O)OC)C3C2)cnn2ccnc(N)c12 10235,C1(NC(C=CC(CC)=CC)=O)CC2C(NC(=O)CN(C)C(=O)OC)C2C1 10236,C1(C(=O)NCC(CCC)OC)CCC2CCC1N2C(=O)CNc1ccccn1 10237,N1(C(c2c(C)oc(C3CCOCC3)n2)=O)CCc2nncn2CC1 10238,CC(C)C(C(=O)NC(C)CNC(=O)C#CC(C)C)c1cccc(C2CC2CO)c1 10239,c1(C(=O)NCC(C2(O)CCN(C(c3cccc(C)c3)=O)C2)C)nc(C)n(C)c1C 10240,c1(CC)cc(C(N2CC(NC(=O)CS(=O)CC)C(C)C2)=O)nn1C(C)(C)C 10241,c1(OC)ccc(CNCC(N)C(C)C)cc1Cl 10242,C12(CNC(c3cncc(SC)c3)=O)CCC(CC1)CN2C(C1CC1C(F)(F)F)=O 10243,c1(COC)ccoc1C(=O)N(C)CCN(C)C(c1ccc(C(C)C)o1)=O 10244,c1(NC(c2ccc(CCC)nc2)C)ncnc(NCC2CC(C)(C)CCO2)c1C 10245,N1(C(C(C2CC2)SC)=O)CCC(CNC(=O)CCOCC2CC2)CC1 10246,N1(c2nncc(C(=O)OC)c2)CCC(C)(O)C(C)(O)C1 10247,N1(C(CC2(CC)CCC2)=O)CCC2(CCC2)C(NC(=O)C(F)C2CCOC2)C1 10248,C1(N(C(C2(COC)CCC2)=O)C)CCC(n2cc(CC(C)(C)O)nn2)CC1 10249,S(=O)(=O)(c1ccc(NCC(O)C(C)(C)C)cc1Br)NCC(C1CCCCC1)SC 10250,N1(C(CCCCCOC)=O)CC(CNC(C2(CF)CC2)=O)CC12CCC2 10251,N1(C(c2cccc(CC)c2C)=O)CC2=C(C1)CN(C(C13C4C5C1C1C3C4C51C)=O)C2 10252,c1(C(N2CC(COCC)C2)=O)cc(CNC(=O)C(c2cnn(C)c2)C)ccn1 10253,C(=O)(C(C)(C)C(C)(F)F)NCC(C)CNC(=O)C(CC(F)F)N(C)C 10254,Cn1c(C(=O)NCC2CCN2C(c2cc(CO)on2)=O)cc2cc(Cl)ccc12 10255,C(=O)(CCCC(=O)N1CCC(C2OCCO2)C(N)C1)C(=O)C=CC(F)(F)F 10256,C1(NC(c2c(CC)nc(C)nc2)=O)CN(C(=O)Cc2ccnn2C)CC12CCC2 10257,N1(C(C(=O)NCCSC)=O)CCN(C)c2ccc(COC(C)(C)C)cc21 10258,C(=O)(CCCCN(C)C)NCC(=O)N(C)Cc1c(C)nco1 10259,C(=O)(N=c1[nH]c(Cl)c([N+](=O)[O-])cc1C)c1c(C)n(C)cn1 10260,C1(CC=C)(NC(c2ncn(C(C)(C)C)n2)=O)CN(C(=O)C(F)CC2CC2)C1 10261,N1(CC=C)CCN(C(c2cn(C)nn2)(C)C)CC1.c1(OC)ccn(C)n1.C1(=O)CO1 10262,Cc1ccc(C(N2CCC(NC(=O)CN(C)C)C(c3ccccc3)C2)=O)c(F)c1 10263,C1(COC)(NC(=O)CCN2CC(F)C2)CCN(C(C2CC2(C)Br)=O)C1 10264,C12(CNC(C(c3ccc(F)c(Cl)c3)C)=O)CC(CO1)N(c1nccc(CO)n1)C2 10265,c1(CC(=O)NC2C(OC)CN(C(=O)CSCC(N)=O)C2)cccc(F)c1F 10266,c1(C(C(=O)NC(C)CN(C(=O)Cn2cc(C(F)(F)F)cn2)C)C)cccc(Cl)c1 10267,C(=O)(CCCCCNC(N)=O)NC(C1CN(C(c2cc(OC)cc(Cl)c2)=O)C1)C 10268,N1(C(C2C(NC(C34CC(CO)(C3)C4)=O)CCC2)=O)CCC([N+](=O)[O-])CC1 10269,C(=O)(CCCCCC#N)NCC=CC(=O)NCC(C(=O)OCC)O 10270,C1(CNC(CS(CC)=O)=O)COCCN(C(C2CC(N3CCCC3)C2)=O)C1 10271,C(C(CC(=O)N(C1CCSC1)C)NC(=O)C=Cc1cc(C)no1)OC 10272,C1(NC(C(C2CCC2)OC)=O)COC2C(NC(c3cc([N+](=O)[O-])n[nH]3)=O)COC12 10273,C(=O)(CCC(C)(C)C)N1CC(C)C(CCC(=O)NCc2cn(CCF)nn2)C1 10274,c1(C(N2CCC(CNC(Cn3nc(C)c(C)c3C)=O)C2)=O)cnc2cc[nH]c2c1 10275,N12CC3CCC3(C1)C2=O.Cc1cc(C(=O)Nc2ncc(CCO)s2)nn1C 10276,c1(C(=O)NC(CC=C)CNC(=O)C=Cc2scnc2C)cccc(S(C)=O)c1 10277,N1(C(C(CSC)C)=O)CCC(O)(CNC(c2c(C)coc2C)=O)C1 10278,c1(NC(c2c(-c3c(OC)ncc(C)c3)cccn2)=O)nnc(C)c(C)c1C#N 10279,Cn1nnc(C(=O)NCCOCCCNC(=O)CCCC2CC2)n1 10280,C12(NC(c3c(CCCC)ocn3)=O)CCN(C(c3cnc(CC)o3)=O)CCC1C2 10281,N1(C(CSCCC)=O)CCCC2(NC(c3cncc4sccc34)=O)CC2C1 10282,c1(N(C(CC(C)NC(c2ccc(OCC)cc2)=O)C)C)ccc2nnnn2n1 10283,N1(C(C(CC)NC(C23CCC(CO)(CC2)C3)=O)=O)Cc2c[nH]nc2C(C)C1 10284,C12CCN(C13CC3)C(=O)OCCNCC2.c1(CC)[nH]cnc1COC 10285,c1(C(N2CCC(C)(NC(C3C4COCC34)=O)C2)=O)cccc2c1OCCN2 10286,c1(C(=O)NCC2CC(NC(CN3CC(C)C3)=O)C2)cnc2[nH]cnc2c1 10287,c1(NC(CN(C(C)(C)C=CCC2CCC2)C(C)=O)=O)cc(C)cc(C)c1C 10288,N1(C(=O)NCC2C(C)C3CCC2C3)CC(=O)N2CCCCC2C1 10289,c1(C2CCN(C(C3(C)CC(OC)C3)=O)C2)ccc(C2CC2)c(C)n1 10290,C1(CNC(c2cnc(C(C)OCC)s2)=O)CN(C(=O)C=CCO)CCN1C 10291,C(CSC)(CC(=O)NC1CC(C(N)=O)C1)NC(C=CCCC)=O 10292,N(C1CCc2cccnc21)C(C1N(C(=O)CCc2cnco2)CCN(C)C1)=O 10293,C(=O)(NN=Cc1cccnc1)n1c(C)cc2ccccc21 10294,N1(C(c2c(C)ncs2)=O)CCC2(CC1)COC(CNC(=O)CC(C)CF)C2 10295,C(=O)(N1CCCc2nccn21)c1ccc(CN(C(=O)CC2CCC2)C2CC2)cn1 10296,c1(CC(=O)NCCN(CCC)C(C2CC(=C3CCC3)C2)=O)cc(CC)no1 10297,N1(C(c2cncc(C=C)c2)=O)CC2(C(=O)NCC3CCOC3)CCC1CC2 10298,c1(OC)cc(OC)cc(C(=O)NC2CCCC2NC(=O)CCOCC(=O)C2CC2)c1 10299,C1(NC(CCCOC)=O)CCC(C)N(C(c2nocc2-c2ccccc2)=O)C1 10300,CC#CCC(C(=O)NCCC(=O)NCCC)NC(c1cc(CO)n(C)n1)=O 10301,Nc1cc(C(=O)NCC2(NC(=O)Cn3cnnc3O)CCOC2)cc(F)c1 10302,c1(OC)cccc(C(c2nnnn2C2(C)CC2)NC2CCC2C(N)=O)c1 10303,CC1(NCCn2cnnc2)CC(NC(=O)C(F)CC2CC2)C1 10304,c1(CC)cc(N)ccc1C(=O)NCCC(O)CNC(=O)CCC1CCCOC1 10305,N1(C(CONC(C2CC(=C)C2)=O)=O)CCN(CC(C)O)CC1 10306,C(CC(=O)NCCCC1CC1C)(C(F)F)NC(C1(CC#C)CCCO1)=O 10307,c1(OC)ccnc(O)c1C(=O)N(C1CCCCN(C(C2C3CC(=O)CC23)=O)C1)C 10308,N1(CCC)CC(C)N(C(c2ccc(C)c(CC)c2)C(=O)NC(C)(C)CC)C(C)C1 10309,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 10310,CC(CC1CCC1)C(=O)NCC1(NC(c2cnnn2C)=O)CCCC1 10311,C1(C(C(C)C)NC(Cc2nnc(C)o2)=O)CCN(C(C2(O)COC2)=O)CC1 10312,C(=O)(C1=CC2CCC1C2)NCCC12CN(C(CCn3ccc(C)n3)=O)C(CC1)C2 10313,S(=O)(=O)(c1ccc(OC)cc1)NCCCc1cccc(OC)c1 10314,c1(N2CCC(N(C(C(COC(C)C)(C)C)=O)C)C2)nc(O)c2ccc(Cl)cc2n1 10315,c1(C(C2(O)CCC2)CN(C(=O)NCCCOC(C)=O)C)ccccc1 10316,C1(Nc2scc(C(=O)OCC)n2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC12 10317,N1(CCNC(=O)CN2CCC(C(=O)NC3CC3)C2)CCC(C(=O)O)CC1 10318,c1(N(CC(CN(C(c2c(C)occ2)=O)CCO)C)C)ncnc(Cl)c1C 10319,C1(CNC(C=CS(C)(=O)=O)=O)CN(c2nc3ccc(F)cc3o2)CC2(CCC2)O1 10320,N1(C(C(=O)NCC(CC)NC(c2ccnn2C(C)C)=O)C)C(=O)CCC1=O 10321,c1(C(N2CCN(Cc3cnc(OC)c(Cl)c3)C3C2C3)=O)ccc2c[nH]nc2c1 10322,C(=O)(CCNC(=O)C(F)C1CC(NC(=O)C(F)F)C1)N(C)CC1CC1 10323,Cn1cnc2nc(N3CC=CC(N(C(=O)Cc4ccon4)CCO)C3)ncc12 10324,CC(C)(C)C(O)C(=O)NCC1(NC(C2CC3(CC(=O)N3)C2)=O)CCCCCC1 10325,c1(CC(=O)OC)ccccc1NC(C1CN(C(c2[nH]nnc2C2CC2)=O)C1)=O 10326,Cn1ccc2nc(N3CCCC(S(=O)(=O)N(C)C)C3)ncc12 10327,c1(CN(C(CC2CCCCCC2)CO)C)ccc2c(c1)CCCN2 10328,c1(CC(N2CC3CC(C2)CN(C(C2(CF)CC2)=O)C3)=O)ccc2nsnc2c1 10329,CCC(C)(C(=O)NCC1CN(C(=O)Cc2cc(C)[nH]n2)C(C)(C)C1)C(N)=O 10330,C#CCC(C(=O)N(C1CCN(C(=O)CC2CCCC2O)CC1)C)OC 10331,c1(CNC(C2(C(=O)OC)CC2)=O)cnc2c(c1)N2.C1(C(=O)CO)CC(F)(CO)C1 10332,C(C#Cc1cnn(C)c1)N(C(C)C)Cc1sccc1Cl 10333,C1(CC)CN(C(C2(CC)CCC2)=O)CCC1NC(C1CC(C)(C(C)(C)C)C1)=O 10334,c1(C(=O)NCC(C)(C(C)C)NC(CCC(C)OCC)=O)cccc2c1OCCO2 10335,CC(C)CC(=O)C(=O)NCCCCC(=O)NC(C)C(F)F 10336,N1(C(CCOC(C)=O)=O)CCC2(CC1)OCCCC2NC(=O)C(C)SC(F)(F)F 10337,C1(CC(=O)NCc2cc(C)on2)C2CN(C(=O)CCc3nccs3)CC12 10338,C1(OCC)CCC1C(=O)N(CC(=O)N(C1(C)CCC1)C)CC 10339,C(CCF)(C(=O)N(CC)Cc1cccs1)NC(CCSCC)=O 10340,C#CCCCCCCC(=O)NC(C(=O)NC1CCC(=O)NC1(C)C)C(C)C(C)OC 10341,C(=O)(CC(O)CC(C)C)NCCCC(C)NC(c1onc(CC)c1C)=O 10342,N1(C(C(Cc2ccc(O)cc2)N(C)C(=O)NC(C)(C)C)=O)CC(CC2CC2)C(O)C1 10343,N1(C(=O)NCc2cn(CC(CC)O)nn2)CCOC(C2(C)N=N2)C1 10344,C1(C2(O)CN(C(C(CC)F)=O)C2)CCNC(=O)C1 10345,C(c1ccc(CN(C2CC2)Cc2cc(Br)ccn2)cc1)=CC(=O)O 10346,CC(C(=O)NCCOCCOCCNC(=O)C=Cc1ncc[nH]1)C(C)O 10347,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10348,c1(CN2CCC(C#N)(C(C)(C)O)C2)cc(Br)cc(F)c1O 10349,S(=O)(=O)(c1ccc2[nH]c(=NCCc3ncccn3)sc2c1)NC(CCC)C(C)C 10350,CC1CCCC(CC(=O)NCCC(C)(C)NC(c2nn(C)nc2Br)=O)C1 10351,N1(Cc2cc(OC)cc(Br)c2)CCC2(CC1)CC2NC(c1ccn(C(C)C)n1)=O 10352,C1(NC(C(CC)OCC)=O)CC2CN(C(=O)CC3CC3C)CC2C1 10353,C1(C(=O)NCC2(NC(c3nn(C)c(F)c3)=O)CCCCC2)CC(C2CC2)=NO1 10354,C1(O)(CCNC(c2cc(N(C)C)ncc2)=O)CCN(C(=O)C(C)(C)F)CC1 10355,c1(C(=O)NCC(C)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10356,c1(NC(C23CC(OC)C2C3)=O)ccc2c(c1)CN(C(=O)C(CN(C)C)N(C)C)C2 10357,C(=O)(C1CCCc2nncn21)N1CCCC(N(CCCCCC(=O)NC)C)C1 10358,C(=O)(C(CC(C)C)OC)NCC1N(C(CCCC=C)=O)CC1 10359,C1(C(Cc2nnnn2C)NC(c2ncnn2C)CC)CCC(F)(F)CC1 10360,CCN=c1cc[nH]cc1C(F)(F)F.CC(CNC=O)NC(=O)COCCOCCO 10361,C12(NC(CNC(N)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10362,c1(Cc2cc(-c3cn(C4C(SC)CNC4)nn3)on2)ccc(Cl)cc1 10363,N1(C(=O)NCCc2c(C)non2)CCN(c2ccc(F)cc2F)C(=O)C1 10364,C1(C2(O)CCN(C(=O)C(C)C(C)(C)C)CC2)(NC(CCc2scc(C)n2)=O)CC1 10365,N1(C(C2(F)CCN(C(C(COC)COC)=O)C2)=O)CCSC2(CCC2)C1 10366,C(=O)(C(C(=O)O)C(C)C)N1CC(NC(=O)OC(c2cccc(C)c2)C)C1 10367,CC1COC(C)CN1C(c1ccc(Cl)s1)C(=O)NCC1CC1 10368,C=C(Cl)CN=c1[nH]c(NCc2ccc3c(c2)CN(C)CCC3)nc2c1CC(C)CC2 10369,C1(NC(C(=O)NC(C)C)=O)CCCC1CNC(c1c[nH]nc1C(F)(F)F)=O 10370,C#CCC(CC(=O)Nc1cncnc1C)NC(C1OCCC1C(C)C)=O 10371,c1(OC)cc(C(N2CCC(NC(=O)C=C3CCSCC3)C(C)C2)=O)ccc1C 10372,c1(C(N(C2CCN(C(C3CC4COCC4C3)=O)C2)C)=O)ccc([N+](=O)[O-])cc1Cl 10373,C1(C(N(C(CNC(c2cc(C)n(C)c2)=O)C)C)=O)CNC(=O)CC1C 10374,Cc1cc(C(N2CC3CCN(C(C4CCCN4C(C)C)=O)C3C2)=O)c2cc[nH]c2c1 10375,N1(CC)C(=O)CCC1CC(=O)NC1CC(N(C(=O)Cn2nnc(C3CC3)n2)C)C1 10376,c1(CCC(=O)N(CCN(C(c2c(C)cco2)=O)C)C)cc(Cl)sc1Cl 10377,C(C(=O)NCCC1(C(=O)NCCC(C)(C)C)CCCC1)(C(C)C)SC 10378,N1(CCCNC(c2cccc(OC)c2)=O)CCC(O)C(NC(c2cccnc2)=O)C1 10379,c1(C(=O)NC(C)CC(C)NC(=O)CCCc2ccc(Cl)cc2)ccc2ncsc2c1 10380,c1(CC)cnn2ccc(C(N3CCN(C(=O)Cc4csc(C)n4)C(C)C3)=O)nc12 10381,c1(C(N2CC(c3cn(CCOC)nn3)SCC2)=O)cnc2sccn12 10382,N1(C(c2c(Cl)ncc(OC)c2)=O)CC2CN(Cc3ccc(Cl)cc3O)CC(C1)O2 10383,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10384,C#Cc1ccc(CN=c2[nH]c(C(N3CCC(C(N)=O)C3)=O)cs2)cc1 10385,c1(CN2C(C(=O)NCCCCC=C)CNCC2)ccc([N+](=O)[O-])c(F)c1 10386,N1(C(c2nnn(CC)c2C)=O)CCCCC(N(C)C(C2CCCSC2)=O)C1 10387,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(=O)C=Cc1cc[nH]c1)CCO2 10388,CC1(CNC(=O)NC2CC(N3CCCC3)C2)CCC(CO)CC1 10389,C(CCCCCNC(C1CCC(OC)C1)=O)n1cc(CC(=O)OC)nn1 10390,C(CN=c1nc(N2CCN(Cc3nccs3)CC2)cc[nH]1)C1CC(C)(C)OCC1 10391,Cc1nc(C(N2CC3CC2C3NC(=O)CC2(C)CCCO2)=O)cn1C(F)F 10392,N1(CC)CCN(C(=O)CCC(C)(C)NC(=O)CC(C)COC)C(C)C1 10393,c1(C(N(C(C)CNC(=O)CC2COCC2O)CC)=O)csc(-c2ccccc2)n1 10394,C(=O)(CCC(C)(C)F)NC(CC)CN(C(=O)CN1CCC(C)C1)CC 10395,C(=O)(C#CC1(C)CC1)NC1C(NC(C2(OC)CCOC2)=O)CCC1 10396,C1(OC)CCN(C(=NCCCCC(F)(F)F)NCC(c2ccccn2)O)C1 10397,C1(C(=O)NCC(C(=O)NC(COC)(C)C)C)C2CC(=O)CC12 10398,C(=O)(C(CC(C)C)C(N)=O)NC(CC)CNC(c1sc(F)cc1Cl)=O 10399,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10400,C1(=O)CC(C)CN1.C(CO)(CCF)SC.C1CC(=O)N1CCOC 10401,C1(C(NOCCCN(C)C)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1(C)C 10402,C1(CNC(C=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10403,Cc1cccc(Cl)c1C(=O)NCC(N1CCCC1CC(N1CCCC1C#N)=O)=O 10404,c1(C(c2n(C(CC)C)nnn2)NC2COC(C)(C)C2)cc(OC)c(OC)cc1F 10405,Cc1ncc(CNC(=O)C(C2CCN(C(c3csc(C)n3)=O)C2)C)s1 10406,c1(OC(C)C(=O)NCC2(O)CN(C(c3ccc(F)cc3)=O)C2)cncc(Cl)n1 10407,N1(C(CC(C)c2cccnc2)=O)C2CC1CN(C(=O)Nc1ccccc1F)C2 10408,c1(CC(N2CC(CCNC(C(C(C)C)O)=O)OCC2)=O)cccc2ccncc12 10409,N1(C(=O)NC2(CC(C)C)COC2)CCC(N=c2nc(C3CCCC3)[nH]s2)CC1 10410,C1(CNC(C=Cc2n(CC)ccn2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10411,C(c1ccncn1)=CC(N1CC(NC(=NC)NCC=C)C1)=O.C(C)(C)(C)C(=O)O 10412,c1(CNC)cn(CC)nn1.N1(C(CC2(COC)CC2)=O)CC(CC(=O)OC)C1 10413,C(=O)(C1(C)CCn2ccnc21)N(C(C)C1CC1)CCc1csc(S)n1 10414,C1(C(=O)Nc2cncc(C(N)=O)c2)CCOCCN1C(=O)Cc1ccoc1 10415,C(=O)(CCCS(C)(=O)=O)N1CCC(c2noc(C3CCOCC3)n2)(C(=O)OCC)C1 10416,C=CC1(O)CCN(C(=O)CCN(CCC)C(c2cc(O)n(CC)n2)=O)C1 10417,c1(C(=O)NCC2CCN(C(c3c(C)onc3)=O)C23CC3)c2c(nn1C)CCSC2 10418,c1(C(=O)NC2CN(C(C(CC#C)C)=O)CC2C(F)F)ccc([N+](=O)[O-])o1 10419,Cc1cc(C(=O)NC2CC(O)CN(C(C3CC(=O)OC3(C)C)=O)C2)cc(Cl)c1 10420,C1(C(=O)NCC2(C(=O)NCC(CN(C)C)CO)CC2)CCC(C)(C)C1 10421,C1(C(N2CC(C)C(NC(COCCOC)=O)C(C)C2)=O)CCc2nnnn2CC1 10422,Cc1cc(=NCC(C)CNC(=O)C=C2CCSCC2)[nH]c(CO)n1 10423,C(=O)(C(C)S(=O)(=O)CCC)N1CC(CN(C(c2c(CC)scc2)=O)C)OCC1 10424,N1(C(C)=O)CC=CC(N(C2CCCN2S(C)(=O)=O)C(=O)Cc2cccs2)C1 10425,C1(C(=O)NCCCN(C(c2ccncn2)=O)C2CC2)CCC(C(F)(F)F)C1 10426,Cc1nc(C2CC2)ncc1C(N1CCC(CNC(=O)CC2CCCO2)C1(C)C)=O 10427,C#Cc1cnc(C(N2CCOCCC2C(=O)NCCN2CCCCC2)=O)c(C)c1 10428,C1(CC(=O)NC(c2ccccc2)C(=O)NC(C2CC=CCC2)C)COC(=O)C1 10429,C(c1ccco1)=C(C(=O)N(CCC(=O)OC)CC#C)C.C1(CC(=O)N)CCOC1 10430,C(=O)(C1=CCC(C)CC1)N1CCC(C(C)NC(=O)Cn2cnnc2O)C1 10431,c1(C(N2CC3C(NC(c4cc(C)nc(C)c4)=O)(CC3)C2)=O)nc2cccnc2s1 10432,c1(C(=O)NC(CNC(C(COCC)F)=O)CC2CC2)cncc(C(=O)N)c1 10433,C(=O)(CC(O)CN(C)C)NCC(C(=O)NCCCC1CCC1)C(C)N(C)C 10434,c1(CC)cccc(F)c1C(N1CCN(C(c2ccc(OC)cc2O)=O)CC1C)=O 10435,c1(C(=O)NC2CCN(C(CN(S(CC)(=O)=O)C)=O)C2)c(N)ccc(F)c1C 10436,C(CCC(C)(C)C(=O)Nc1ccc2[nH]ccc2c1)SC 10437,Cc1ccc(C#N)c(C(N2CC(n3cc(C4CCOCC4)nn3)C(O)C2)=O)c1 10438,N1(C(C(C)CN(C)C)=O)CC2(CC2)CC1CNC(=O)C(C)OCCN(C)C 10439,Cc1cc(C(=O)NCCCCNC(c2sc(C)cc2Br)=O)ncc1F 10440,C1(NC(CC(C)(C)NC(CCN(C)CC)=O)=O)CCCCC1(C)O 10441,N1(C(C2(F)CCN(C(c3ncc(Br)cc3Cl)=O)C2)=O)CCc2nc(Cl)ccc2C1 10442,c1(C(=O)NC2C=CC(CNC(CN(CCC)C)=O)C2)cc(C)nc(C)n1 10443,N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC(NC(C3CCS(=O)(=O)N3)=O)C1C2 10444,CCCCC(C(=O)N1CCC(CCO)CC1)NC(c1cn(C)nc1OC)=O 10445,C1(C(N2CC3C(NC(c4ccc[n+]([O-])c4)=O)C3C2)=O)COc2ccc(O)cc2O1 10446,Cn1cnc2ccc(C(=O)NC3CC4(C3)CC(NC(=O)C(F)C(C)(C)O)C4)nc12 10447,C(=O)(CCC(O)C(C)(C)C)N1CCC(CCNC(CNC(CN(C)C)=O)=O)CC1 10448,N1(C(C2CC(SC)C2)=O)CC2CCC(CNC(c3c(SC)ccs3)=O)(C2)C1 10449,c1(OCC)ccc(C(O)CNC(=O)NC2(c3ccccc3)CC(C)C2)cc1 10450,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(CC)nc2)=O)ccc(Cl)c(F)c1 10451,Cn1cc(C(C(=O)NCc2ccco2)N(C2CC(=O)NC2=O)CCOC)c(I)n1 10452,CCCC(CN=c1cccc(S(=O)(=O)NC2CCc3ncsc3C2)[nH]1)OC 10453,C1(CC(=O)N(CCOCCNC(c2c(C)csc2)=O)C)CCCC(=O)N1 10454,CCC(CC(F)(F)F)N=c1[nH]c(=NCC2(C)CC3(CC3)C2)[nH]c2cc[nH]c12 10455,C1(C(=O)NCCOCCN(C(C(C)C2=CCCC2)=O)C)CCC2(CC1)CC2(F)F 10456,C1(C(=O)OCc2ccc(N3CCCC3)nc2)CCCC12CCOCC2 10457,CC(C)CN=C(NCc1cnc(OC(F)F)nc1)NCC1(CO)CC1C(F)(F)F 10458,CC(CO)C(=O)NCCOCCCN(C)C(c1cnn(C)c1)=O 10459,C=Cc1ccc(C(=O)NCC(C)(O)CNC(=O)C(c2ccccc2)OCC)cc1 10460,C(CCCC(=O)N(CC(O)CN(C(=O)COCCOC)C)C)OC 10461,n1(CCC(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)c(=O)nc(O)c2ccccc12 10462,c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cc(Cl)nn1C 10463,c1(CC)nocc1CN(C(=O)C(c1cn(C)nn1)NC(=O)C=C(C)C1CC1)C 10464,c1(C(=O)NC)ccc(CNC(c2ccc(C(F)(F)F)cc2)C)cc1 10465,C(=O)(CS(=O)(=O)CCCC)N1C(CNC(C(CC)=CC)=O)COCC1 10466,CN(N=Cc1ccccc1)c1ccc(S(=O)(=O)N2CCCOC2C(=O)O)cn1 10467,C1(NC(CSCC#C)=O)CN(C(=O)C(C)ONC(=O)OC(C)(C)C)CC1(C)C 10468,Cc1ccccc1C(=O)NC(CCN(C)C)C(=O)N1CC(C)C(C)C1 10469,c1(C(N2CCCCC2)CNC(NC2C(C)C2)=NCCF)nnc2c(=O)[nH]ccn12 10470,c1(CC(=O)N(CC(CC)NC(C2(C)CCCCCC2)=O)C)ccc(C)c(OC)c1 10471,CC1CC=C(C(=O)NCC(C)(C(C)C)NC(=O)CCCN2C(=O)CNC2=O)CC1 10472,c1(C(O)Cc2ccncc2)nc(-c2ccccc2Cl)nn1-c1ccnc(F)c1 10473,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC2(NC(C2CCO2)=O)C1 10474,N12CC(C)C(C)(C1)OCC2=O.C(C(=O)NCC(=O)NC)(C(C)C)OCC 10475,c1(OC)ncc(NC(C2(F)CCN(C(=O)Cc3ccccc3O)C2)=O)cc1F 10476,C12(CCCCC1)CC(=O)N2.Cc1ncc(CCNC(c2coc(N(C)C)n2)=O)s1 10477,CC(=NO)C1CC(C(=O)NC(C2CCN(C(=O)COC(F)(F)F)C2)C)C1(C)C 10478,c1(C(N2C(CNC(c3n(C=C)nnc3)=O)CCCC2)=O)ccc(Br)c(O)c1 10479,N1(C(c2c(C)n[nH]c2C)=O)CCC2(CC1)CC2CNC(C1CCCC(=O)O1)=O 10480,c1(C(N2CC(NC(=O)CCc3ccsc3)CC(C)C2)=O)cncc(P(C)(C)=O)c1 10481,N1(C(=O)CC2CCCCN2C(=O)CC2(O)CCOC2)CCOC2(CCC2)C1 10482,N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cc(Cl)cnn2)=O)C1C 10483,C(C)(CN=c1[nH]cncc1C)NC(C(c1ccc(C)cc1)C)=O 10484,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10485,C(=O)(C(O)CCS(C)=O)N(CCC)CCNC(c1ncc(F)cc1F)=O 10486,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10487,C#CCC(O)C(=O)N1CC(C(=O)NCCCCC2CC2)C(F)C1 10488,N1(S(CCCC)(=O)=O)CCC(C(=O)NCCc2nccs2)(CO)CC1 10489,c1(CC)nccnc1C(N1CC(C)C1C(=O)NC1CCC2(C(C)C)CC12)=O 10490,C1(C(=O)NC2CCCC(CNC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 10491,C1(C(=O)OC)CC(C(=O)N(C(C)CCNC(=O)CC23COCC(C2)C3)C)C1(C)C 10492,C12(CCCCO1)C(=O)NC2.C(=O)(C(C)C(=O)N(C)C)NCCC1(CSC)CC1 10493,C#Cc1ccc(OCC(CC(=O)OCC)NC2(C)CNC(=O)C2)cc1 10494,c1(OCCC(=O)NCC2(NC(c3c(C)nc(C)o3)=O)CCC2)ccc(C)c(C)c1 10495,N1(C(COc2cccc(C)c2)=O)CCN(C(c2cc(F)ccc2F)=O)C2CC12 10496,N1(C(c2ccc(C(C)(C)C)o2)=O)CCC(O)(CCNC(=O)Cc2ccsc2)CC1 10497,C1(NC(C2(CC(=O)OC)CC2)=O)COCCC1NC(C1CC1C(=O)OC)=O 10498,Cn1cc2cccc(CN3CCN(CC(=O)Nc4cccc(Br)c4O)CC3)c2n1 10499,CN1CCN(Cc2cn(CCCC(=O)NCC(C3CCCC3)=O)nn2)CC1 10500,CC(C)CC(CC(=O)NCc1ncoc1C1CC1)NC(=O)CC1CC2CC2C1 10501,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2nocc2C)C(C2CC2)C1 10502,C1(NC(c2cnsc2)C)CC2CC1CC2(F)F 10503,c1(OC)ccc(F)cc1C(=O)Nc1ncc(CCSC)s1 10504,N1(CC(=O)NCCC2CCC(NC(Cc3nc(C)sc3)=O)C2)CCCNC1=O 10505,N1(C(Cc2ccc(OC)cc2Cl)=O)CC(=O)N2CCCC2C1 10506,N1(C(Cc2cc(CC)no2)=O)CCCC(CO)(Nc2nc(CC)ncc2Br)C1 10507,C1(NC(C2C=CCN(C(c3n(C)c(=O)ccc3)=O)C2)=O)CC2(CCCCC2)C1 10508,c1(C(N2CCN(Cc3ccc(F)cn3)C3CC23)=O)cc(Cl)c(Cl)cc1Cl 10509,CCC(CC)C(C)C(=O)N1CC(C)(CNC(c2c(C)cccc2C)=O)CC1(C)C 10510,N12CC3(CCCN3C(=O)c3ccc([nH]3)C1=O)C2.c1(OCCCC)ccc(C)o1 10511,c1(CNC2CCN(C(=O)CCCC3CCOCC3)CC2O)c(Cl)cc(F)cc1Cl 10512,N1(C(C=Cc2ccc(OC)cc2)=O)C2CCC1CN(C(c1cnns1)=O)C2 10513,N1(C(c2n(CC)ccc2)=O)CCCC2C(NC(C3C4CC5C(C4)C35)=O)C(C)(C)C12 10514,C=CCCCC(C(=O)N1CC(F)C(F)C1)NC(C1CC2CCC2C1)=O 10515,N1(C(c2n(C)ccc2)=O)CCCC2(CCC(NC(C3(C#N)CC4(CC4)C3)=O)C2)C1 10516,N1(c2c(Br)cnc(C)n2)CCC(O)(C2(NC(=O)CCSC(F)(F)F)CC2)CC1 10517,Nc1cc(C(=O)NC2CCCCN(C(c3csc4nccn34)=O)C2)cc(F)c1O 10518,C1(C(=O)NCC(CNC(c2onc(COC)n2)=O)O)CCSC(C)C1 10519,c1(C(N2C(CCNC(C3(N(C)C)CC3)=O)CSCC2)=O)cccc2cnccc12 10520,c1(C(=O)NC2CN(C(C3C(C)(Br)C3)=O)CC2O)cc(F)cnc1Cl 10521,Cc1cc(S(C)(=O)=O)cc(C(=O)NC(C)CNC(=O)CC(O)C(C)C)c1C 10522,C(=O)(CC(C)COC)N(CC=CC(=O)N(CC#C)CC)CC1CCCO1 10523,C1(C(N2C(C(C)(C)C)CN(C(c3ns[nH]c3=O)=O)CC2)=O)CCCCCC1(F)F 10524,N1(C(CC)=O)CCOCC(NC(C2C(C)CCN2C(=O)OC(C)(C)C)=O)C1 10525,C(C(CNC(C1(c2ccncc2)CC1)=O)C(F)(F)F)NC(=O)CC1COCC1O 10526,C1(NC(c2cnc(C)nc2)=O)CC12CCN(C(=O)CC(C)CF)CC2 10527,c1(C(=O)NC(C(=O)N2C(C)(C(C)C)CC2)CCN(C)C)cncc2[nH]ccc12 10528,CCCCCC(C)CC(=O)NC1(C(=O)NC2CN(C)C(C)(C)C2)CC1(C)C 10529,CC1CCCC(CC(=O)NCCN(C)C)C1.C12(C)CN(C1)C(=O)CCOC2=O 10530,c1(C(=O)NC2(CNC(c3nc(CC)sc3)=O)CC2)c(Br)nnn1C 10531,N1(C(CCCc2scc(C)n2)=O)CC2(CCN(C(c3cccc4sccc34)=O)C2)C1 10532,c1(C(N(C(CNC(C(CCOC)NC(C)=O)=O)C)C)=O)ncc(N)nc1C 10533,C1(C(=O)NCCCCCCN(C(CCCCC=C)=O)C)Cc2ccc(F)cc2C1 10534,C#CC1(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CS(=O)(=O)CC)CC1 10535,c1(C(=O)NC2(CCNC(c3coc(C(F)(F)F)n3)=O)CC2)ccc2nnnn2c1 10536,CC1C(C)N(C(=O)CCCN(C)C(c2cccn(C)c2=O)=O)CCN1C 10537,N#Cc1ccccc1OCC(N1CCC(CCNC(c2csnc2Cl)=O)CC1)=O 10538,c1(C(N2CCCC2CSc2c(F)cccc2F)=O)c(O)nnc2c1CCC2 10539,CC(C)CC(CNC(C12CC(F)(C1)C2)=O)C(=O)NC(C)CS(C)(=O)=O 10540,Cc1cc(SCCOCC(=O)NC2CN(C(C3CCC(C)C3)=O)C2)on1 10541,CC1CN(C(=O)CSc2nncs2)CC(C)N(C(C2(O)CCOCC2)=O)C1 10542,N1(C(C2CN(C(C)=O)C2)=O)CC(NC(=O)CCCc2cncs2)CC1CO 10543,N1(C(C(CSC)C)=O)CCCCC(C(=O)NCc2nc(=O)o[nH]2)C1 10544,n1(CC(=O)NCC2OCCN(c3ccnc(C(=O)OC)n3)C2)nc(C)c(Cl)c1C 10545,c1(OC)cc(CCNC(=O)C(C)Oc2ccc(F)cc2)cc(OC)c1O 10546,C1(C(=O)NCC=C2CCN(c3ncc(I)cn3)CC2)CC12CCCCC2 10547,Cc1ccc(S(=O)(=O)N(C(CCN(C2CCCC(O)C2)C)=O)C)cc1 10548,c1(C(=O)NC2CN(C(C(C)SC)=O)C(C)(C)C2)cc2ncccn2n1 10549,Cc1cc(C)c(C(=O)NC2CCC2CNC(c2nc(-c3ccncc3)cs2)=O)o1 10550,c1(NC(C)C)nnccc1C(N1CCC(CN(C(=O)CN2CCC(C)C2)C)C1)=O 10551,c1(C(=O)NCCC(CNC(c2nsnc2O)=O)OC)cc2ccncc2[nH]1 10552,C1(C(=O)NCC2(O)CCN(C(=O)CN3CCOCC3)C2)CC12CC(F)(F)C2 10553,N1(C(CC(C)OC)=O)CC(NC(c2cccc(-c3cn[nH]c3)c2)=O)C(C)C1 10554,CC(C)(C)C#CC(=O)N1CCN(C(=O)C=C2CCCCC2)C(c2ncc[nH]2)C1 10555,C1(C(N2C(CC(=O)NCC3CC4C=CC3O4)CCC2)=O)NC(=O)C2CC12 10556,Cc1nc(C2CC2)[nH]c1C(N1CCC(NC(C2SCCC2C)=O)CC1)=O 10557,C1(CC(=O)NCCCCCNC(c2ccc(CSC)cc2)=O)CCC(=O)NC1=O 10558,CCCCC(CNC(=O)CC1COCC1O)NC(C1CC(=O)N(C)C1)=O 10559,CC1(C)CCC(C(=O)NCCC2(C)CC2(F)F)CN1C(C1CCC(=O)N1)=O 10560,C1(NC(=O)COc2cccc(F)c2)CN(C(C2(C(F)F)CCC2)=O)CCC1F 10561,Cc1ccc(CNC(=O)C(C2CC2)N(C(=O)C(C)CCN(C)C)C)cn1 10562,c1(OCC)c[nH]nc1C1CCN(C(=O)CC(C)C2CCCCC2)C1 10563,N1(C(c2n(CCC(=O)Nc3coc(Br)n3)nnn2)CC)CC(C(N)=O)C(C(N)=O)C1 10564,C1(NC(CCN(C)CCO)=O)CCC(N(C)C(c2conc2C2(C)COC2)=O)C1 10565,C(=O)(CCCCC(N)=O)N1CCC(NC(c2n(C)nnc2)=O)CC1C1CC1 10566,c1(C(C(=O)NC(CC(C)NC(CC=CC)=O)C)C)cccc(C)c1 10567,C1(C2CCN(C(c3cc(C4(C)CC4)on3)=O)C2)(NC(Cc2cn(C)nc2)=O)CC1 10568,c1(NC(c2ccccc2)=O)cc(N2CCOC(C(F)(F)F)C2)c(Br)cn1 10569,c1(C(=O)NCC(CNC(C(C(C)O)N(C)C)=O)O)cc2nccn2c(O)n1 10570,c1(C(=O)NC2(CNC(C34CCCC3C4)=O)CCCC2)ccc(Cl)cc1O 10571,C1(C2CN(C(C34CCCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10572,C(=O)(C(CC)CC(C)C)NCc1cncc(C(=O)NC(CCC(=C)C)C)c1 10573,c12nn3ccccc3c1CNC2=O.CN1CCC(CN2CCOCC2)C1 10574,C(=O)(CCN(C(c1cocn1)=O)CC)N(CC#C)CCF 10575,C1(NC(CC=CCC)=O)COC2CN(C(C3CCCCC3)=O)CC12 10576,CCCCC(C)C(=O)N1CC(CNC(=O)C(c2cnn(C)c2)O)C1 10577,Cc1ncnc(C(=O)NC(Cn2ccnn2)C(N2CCOC(CCF)C2)=O)c1C 10578,c1(-c2cc(C(=O)NC)c(O)cc2)cnn2c1CN(C(C1CCCCC1C)=O)CC2 10579,C1(C(=O)NCC=CCNC(C)=O)CC=CCN1C(C1CCC1OC(C)C)=O 10580,c1(C(=O)NCC(CC)NC(C2CCC2)=O)oc(-c2cnn(C)c2)nc1C 10581,Cc1nc(C)c(CC(=O)NCC2CCCCN2C(=O)COc2cn[nH]c2)c(O)n1 10582,C(=O)(CCC1=NNC(=O)CC1)NC(C)CNC(=O)CC(C(F)F)n1cccn1 10583,N(C(=NCCN1CCCC1)NCC1=CCOCC1)CC(c1ccc(C)cc1)(C)C 10584,c1(C(C(=O)NCCC(=C)CNC(c2oncc2C)=O)C)ccc(Cl)c(Cl)c1 10585,Cc1ccc(O)c(CNC(=O)CC2CCCN(C(=O)CC#N)C2)c1 10586,c1(C(=O)NCc2c(C(NOCCCC=C)=O)n(C)nc2)cc(C#N)ccc1C 10587,C1(C(N(CCN(C(c2cnc(C(C)C)n2C)=O)C)C(C)C)=O)CCCCN1N=O 10588,c1(CC2(C(C)NC(=O)Nc3snc(C)n3)CC2)c(Cl)cccc1Cl 10589,CC1CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1cnc(C2CCCC2)[nH]c1=N 10590,C1(C(N2CCCC(CCC#C)C2)=O)CC2(CC(NC(=O)C(C)(C)C=C)C2)C1 10591,S(=O)(=O)(c1ccc(NCC(C)NC2CC2)cc1Br)N(C(CC)C)C 10592,N1(C(c2cc(CCC)n(C)n2)=O)C2CCC1CN(C(=O)C(O)CCC(C)C)CC2 10593,n1(CC(=O)NC2(N(CC)Cc3ccc(C)cc3)CC2)cnc2ccccc12 10594,c1(C(N2CC(NC(c3ccc(C)cc3F)=O)C(C)C2)=O)ccc(Br)c2cc[nH]c12 10595,S(=O)(=O)(c1ccc(F)c(F)c1)N1CC(C(=O)Nc2cnns2)C(F)(F)CC1 10596,C(=O)(C(C)S(N)(=O)=O)NCC(CNC(C(c1ccccc1)OCC)=O)C 10597,c1(Cn2cc(C3CCN(C(C4C(C(C)C)C4)=O)C3)nn2)ccc2ccccc2c1 10598,C1(n2c(C34CC5CC(CC3C5)C4)nc(CCCN(C)C)n2)CCOC2(CCC2)C1 10599,c12nnn3c1CCCC3C=CC=C1N(C(=O)COCCF)CCN(C1CC)C2=O 10600,c1(NC(C2C(C(=O)OC)CCC2)=O)ccc2c(c1)COC2.N12CC3CC3(C1)C2=O 10601,c1(C(N(C2CCCC(NC(=O)C(=O)C(C)(C)C)C2)C)=O)cc(F)cc2ccoc12 10602,N1(C(c2n(CC)ccn2)=O)C(C(=O)NCc2cnn(C(C)C)c2F)CCC1C(C)C 10603,c1(C(N)=O)c(NC(C2CCCCCC23CCC3)=O)cnc2ccccc12 10604,c1(CNC(c2cccnc2S)=O)ccc(C(N2CCCC2CCCO)=O)nc1 10605,C(=O)(CCCCC(=O)NC(C1CCN(C(C2CCOC2(C)C)=O)CC1)CO)NC 10606,c12cccc(c1)CC(=O)N2.C1(OCC(C2(OCC)CC2)=O)CCCC1.C(C)C 10607,C1(C(=O)NC(CCC)C2CCC2)CCC(C)(C)N(C(=O)C(F)C2CCC2)C1 10608,CCCC(C(=O)NC1CCC(N(C)C(c2cn(CC)nc2C)=O)CC1)NC(N)=O 10609,c1(C(N2CCC(Cc3ccccc3Br)C2)=O)ccnc2ncnn12 10610,C=CCC(C)(C)C(=O)N1CCN(C(=O)COCCC)C(C2CC2)C1 10611,N1(C(COCCCCC)=O)CCC(C)(C)C1CC(N1CCC1C1CC1)=O 10612,CCC(C)(C#N)C(=O)NC(CNC(=O)COCc1scnc1C)CC(F)(F)F 10613,c1(OCCC(=O)NCC(CC)NC(c2ncc(CC)s2)=O)cccc(CSC)c1 10614,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN(C)C)C3)cc1S(C)(=O)=O 10615,N1(C(C(c2cccnc2)C)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)C2 10616,C1(CCn2cc(C3(N(C)C)CCCC3)nn2)CCCN1C(=O)C(F)C1CCC1 10617,N12CCCC3CN(CCC13)C(=O)CC=CC2=O.C(c1ccccc1)=CC 10618,C12(C(=O)NC(C)CCNC(c3nnc(O)cc3O)=O)CCCC(C1)C(=O)N2 10619,c1(C(=O)NCC2(CNC(C3CN(CCCC)C(=O)C3)=O)CC2)cc(C#N)ccc1O 10620,c1(CNC(C2CCCCS2)=O)ccccc1-n1cc(CN2CCCC2=O)nn1 10621,C1(C(=O)NC(c2ccccc2)C)CON(C(=O)C(C)C(F)F)C1 10622,C1(NC(C(C)NC(=O)C(C)(C)C)=O)CCN(C(=O)Oc2ccc(Cl)cc2)CC1O 10623,c1(C(N(C2CCN(Cc3scnc3Cl)C2)CC)=O)cc(-c2cccnc2)no1 10624,Cc1oc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10625,N1(C(=O)C2=C(Cl)CCCC2)C2CCC1C(F)C(C(=O)NC1(CO)CC1)C2 10626,N1(CC)CCN(C(c2ccc(NC(c3n[nH]c(C)c3Br)=O)cn2)=O)CC1=O 10627,C(=O)(N=c1[nH]c(Cl)ncc1O)C1N(C(c2ccc(C(F)(F)F)o2)=O)CC2(CC2)C1 10628,C(=O)(C(O)C(F)F)NCC(C)NC(c1ccc(N(CCO)C)cc1)=O.CCO 10629,c1(OCC)cnc(C(=O)NC(C2CCN(C(=O)C(F)C3CCCC3)C2)C)cn1 10630,C(=O)(NN(C(=O)C1CCc2ccc(F)cc21)C(=O)O)c1ccccc1.CS 10631,CCCCCC(O)C(=O)NCC=CCNC(C1CCCN(c2cnn(C)c2)C1=O)=O 10632,C=CCCC(C(=O)N1CC(C)(C)C1C(N)=O)NC(C1(C)CCC2CC2C1)=O 10633,c1(C(=O)NC2(C)CCN(C(C(CC#C)CC#C)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 10634,C1(NC(c2cc(CO)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10635,c1(N)nc(OC)c(OC)c(Cl)n1.c1(C(=O)NC(CNC(=O)OC)C)ccncc1 10636,N1(C(c2c(C)cco2)=O)CCC2CC(CNC(C3(C(F)F)CCC3)=O)CCC2C1 10637,Cc1onc(C(=O)NCC2CCCC(NC(C3CC(=O)C3(C)C)=O)C2)c1[N+](=O)[O-] 10638,Cc1ccc(C)c(C(N2CC(CNC(C3C(F)(F)C34CCC4)=O)C2)=O)c1O 10639,CN1CCCC(C)(C(=O)NCC2(O)CCN(C(C3(CO)CCCCC3)=O)C2)C1 10640,C(=O)(CCN=C(NCCN1CCC(N(C)C)C1)NC1CCCS(=O)(=O)C1)N(C)C 10641,OCC(CC1CCCC1)CN=c1[nH]c2c(c(=NCCCC(F)(F)F)[nH]1)SCC2 10642,c1(C(N2CCN(C(c3noc(COC)c3C)=O)C(C)C2)=O)nccn2ccnc12 10643,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10644,N(C(=NCCCCl)NCC1CCOC1)CC(F)(F)Cl 10645,c1(NC(=O)C=Cc2ccc(Cl)cc2F)cc([N+](=O)[O-])ccc1-c1nn[nH]n1 10646,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)Cc2cnc[nH]2)C)COCC1 10647,C1(OC)(CNC(=O)CC2CCC2)CCN(C(=O)CC(N2CCCS2(=O)=O)C)C1 10648,CS(=O)c1ccc(-c2cnc(NC(c3cccc(C(F)(F)F)c3)=O)c(O)c2)cc1 10649,c1(OCCC(C)C)ncccc1NCc1cc(OC)ccn1 10650,C1(NCC(=O)N(C)Cc2ccncc2)CCN2CCCCC12 10651,c1(C(N2CCC(NC(c3cncnc3)=O)CC2C2CC2)=O)cc([N+](=O)[O-])ccn1 10652,C=C1CC2(C1)CC(C(=O)N(C1CCCN(C(=O)C(n3cc(Cl)cn3)C)CC1)C)C2 10653,C(=O)(C(C)(C)C1CCN(C(=O)C(=O)Nc2cnn(CC3CC3)c2)C1)OC 10654,C1(OC)CCN(c2cc(C)nc(NC=O)n2)C(C)C1.c1(C)cc(Cl)ccc1Cl 10655,C1(CNC(CCc2c(SC)cccc2)=O)CN(C)CCN1C(C1CC1C(C)O)=O 10656,C1(O)(C(C)NC(C2C(OC)C2)=O)CCN(C(c2cnccc2Br)=O)C1 10657,N1(C(C2CCS2(=O)=O)=O)CCC(CCNC(C2(F)CCCC2)=O)CC1 10658,c1(C(C(=O)N(CCNC(=O)C(F)(F)Cc2ccccc2)C2CC2)=O)ccc(F)cc1 10659,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10660,Cc1nnc(CCC(N2CCCC(CN(C)C(C3CCCN3C(C)C)=O)C2)=O)n1C 10661,C(=O)(C1=C(F)CN(C(C2CCCC(=O)C2)=O)CC1)N(C)Cc1cscn1 10662,C1(NC(CCN(CCC)C)=O)CC2CC1CN(C(c1ccnn1CC1CC1)=O)C2 10663,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(=O)C(=Cc1ccco1)C 10664,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CC(C)(C)C2)=O)C1 10665,CC1(F)CC(C(=O)NC2CCCC2CNC(=O)Cc2cc(SC3CC3)no2)C1 10666,C#CCCCCC(=O)NC1(CNC(c2ccn(C)c(=O)c2)=O)CC1 10667,c1(CNC(c2n(CC(=C)C)nnn2)c2nnc(C3CC3)s2)cc(F)c(F)cc1F 10668,N1(C(C2C(CCC)C2)=O)CCCC2(C1)CN(C(c1ccc(N)cc1F)=O)C2 10669,c1(NC(C2CC(NC(CNC(c3cn(C)nc3)=O)=O)C2)=O)ccnc(Cl)n1 10670,Cc1cnn(CCCNC(=O)CCN(C(=O)CCCn2cccn2)C2CC2)c1 10671,CCC(C)CC(=O)NC1CCCC1C(=O)Nc1ccc(NCCO)cc1 10672,C(=O)(C(O)CCC(F)(F)F)N1CCCC(NC(C(CSC)O)=O)(CO)C1 10673,CCC(CC)(C(=O)OC(C)(C)C)C(=O)NCCCN(C)C(C1C(OC)C1C)=O 10674,C1(C)(COC)CC(NC(=O)CC2CC2)CN1C(=O)Cn1cnc([N+](=O)[O-])n1 10675,CC1OCCC1(C)C(=O)NC1CCOC(C(=O)N(C)CCc2nccs2)C1 10676,C(CCN=c1[nH]c(=NC2CCC(O)CC2)[nH]c2c1CCCCCC2)N(C(C)=O)C 10677,CCCC(CC)C(=O)N1CC(NC(=O)Cn2nc(Cl)ccc2=O)CC(F)C1 10678,c1(C(=O)OCc2cn(C)c(=O)cc2)ccc2ccnc(Cl)c2n1 10679,c1(C(=O)NC2COCC2n2cc(-c3cc(C(N)=O)no3)nn2)n[nH]c2c1COC2 10680,N1(C(C(C(C)C)F)=O)CCCN(C(=O)CN2CCCCC2C)CCC1 10681,C(CC(C)C)(C(=O)N1CC2(C1)CN(C(c1cscc1C(F)(F)F)=O)C2)OC 10682,CCC(O)C(C)C(=O)NCCOC1CCN(C(=O)CN2CCCC(N(C)C)C2)C1 10683,C(=O)(C1=COCCO1)NCCCN(C)C(c1c(Cl)cnn1C1CCCC1)=O 10684,C1(NC(CCCc2onc(C)n2)=O)CC2(CCCN(C(=O)C3=NOC(C)C3)C2)C1 10685,N1(C(Cn2c(C)cc(C)n2)=O)C2CCC1C(NC(=O)Cc1ccsn1)C2 10686,N1(C(c2c(C)ccc(-n3cccc3)c2)=O)CC2CC(=O)CC1C2 10687,C12(C(=O)NCCC3OCCN(C(C(CCSC)O)=O)C3)CCC(CC1)C2(C)C 10688,Cc1nc2c3ccn2c3n1.N1CCC2CCC(C1)N2C(=O)C(C)n1ccnc1 10689,C1(CC(=O)OC(C)(C)C)(NC2CC3CC3C2)CCOCC1 10690,N1(C(CCNC(C)=O)=O)CC2COCC(C1)C2NC(=O)CCCc1ccc(F)cc1 10691,C(CC(=O)N(C(C)(C)CO)C)(C(F)F)N(C(C=C(CC)C)=O)C 10692,c1(CC(N2CC3C(NC(C4CC(C5CCC5)C4)=O)C3C2)=O)nc2ncccn2n1 10693,C1(NC(C(COC)COCC2CN(C(=O)C(C)(C)C)C2)=O)CCc2nn[nH]c2C1 10694,C1(NS(CCN(C(C)C)C(C2CCCO2)=O)(=O)=O)CCCC1C1CCCC1 10695,c1(C(N2CC(Cc3cn(C)nc3)OCC2)=O)nnc2ccsc2c1N 10696,C1(NC(C=C(CC)C)=O)CC2CCC1C1CN(C(=O)C(=CC3CCCC3)C)CC21 10697,N1(C(c2ccc(C)nc2C)C(=O)NCCC)CCCC(O)(C2CC2)C1 10698,C(c1ccc(C)cc1C)=C(C(=O)Nc1c(C(=O)OC)cccc1)C 10699,N1(C(CC(=C)I)=O)CCCN(C(=O)C(C)COC)CC1 10700,c1(C(N2CCC(C)C2CNC(c2nnsc2CO)=O)=O)ccc(N(C)C)cc1F 10701,C#Cc1ccc(C(N2CCN(C(=O)OC)C(C(=O)OC(C)(C)C)C2)=O)cn1 10702,Cc1cc(=O)c(C(=O)NC(C2CN(c3ncc([N+](=O)[O-])cn3)C2)C)cn1C1CC1 10703,C1(NC(C2CC(CCC)C2)=O)CC(O)CN(C(c2ccc(SC)cc2)=O)C1 10704,N1(C(CSCCC)=O)C2CC=C(C(=O)Nc3cc(C)nnc3O)C1CC2 10705,c1(C(N(CCN2CCN(C(CCC#C)=O)CC2)C)=O)c(F)cccc1Cl 10706,C(C(CC(C)C)C(=O)NCC1COCC1NC(c1occc1C(=O)OC)=O)OC 10707,S(=O)(=O)(c1ccc(N2CCCC(C)(C(C)(C)C)C2)c(Cl)c1)N(C)CC1CC1(C)C 10708,S(=O)(=O)(c1cc(C)ccc1F)NC1(C(=O)OC)C(CC)CC1 10709,C1(C(C)C)COCCN(C(=O)C(=O)N(CCCO)CCn2cc(CN)nn2)C1 10710,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10711,C(CCN=c1[nH]c2c(c(=NCCN3CCOC3=O)[nH]1)COC2)OCC(C)C 10712,c1(CC)noc(C)c1C(N1CCC(C2CCCCN2C(C2(CC)COC2)=O)C1)=O 10713,Cc1nc(NC(CNC(C2CCC3CC(C)CN3C2)=O)C(C)C)c2ccsc2n1 10714,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10715,C1(NC(=O)CCc2cccc(Cl)n2)CN(C(=O)CC(F)(F)Cl)CC12CC2 10716,N1(C(C2C(C)=CCC=C2)=O)CCCC(C)(C(=O)NCc2cc(O)ccc2C)C1 10717,c1(C(=O)NCC(C)CNC(C23CC(C(F)F)(CO2)C3)=O)ncc2ccccn12 10718,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCC1NC(=O)CCCSn1cccn1 10719,CCCCC(O)C(=O)NCC1CCN(Cc2cn(CCOC)nn2)CC1 10720,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(N(C(=O)C(O)CN(C)C)C)CC1 10721,c1(SC)c(C(=O)NC2(C)CN(C(c3ccc(C)nn3)=O)C2)cccc1F 10722,c1(CC)nc[nH]c1C(=O)N(C1CC(NC(=O)CCc2cc[nH]n2)C1)C 10723,S1(=O)(=O)c2ccc(cc2)C(=O)NCC(C)N1C.C1(NC)CCCC1C(=O)NC 10724,Cc1cnc(C(N2CCC(NC(C3CCC(C)O3)=O)C23CC3)=O)c(C)c1 10725,CC1CCN(C(=O)N(C2CC2)C(c2ccccc2Br)C)CCC1c1ccccc1 10726,c1(-c2nc(COc3cccc(NC(C)=O)c3)on2)cccc2c(C)cccc12 10727,C(C1CN(C(CC(C)(O)CCC)=O)CC1C(=O)NC1(CCCF)CC1)=CC 10728,c1(OC)ncccc1C(=O)NCC1CCN1C(C1CC2(CCC2)C1)=O 10729,c1(CC)noc(CCCNC(=O)NC(C)(C)CNC(=O)OC(C)(C)C)n1 10730,C=CC1(C(=O)NCC2CCC=CCCC2)CCN(C(C2CCCCS2)=O)C1 10731,C=CC(C)(C)CC(=O)NC1(CCNC(=O)CCS(C)(=O)=O)CCC1 10732,C1(C(N(CCNC(=O)C(C2CC2)OC)CC)=O)CCS(=O)(=O)C1(C)C 10733,c1(C(=O)NC(CCN(C(CN2C(C)CC2)=O)C)C)nn(C)cc1N 10734,C1(CC)CCN(C(=O)CC(C)(C)O)C1CNC(c1cc(C)ncn1)=O 10735,C1(C(N2C3(C(N(C)Cc4cccs4)=O)CC3CC2)=O)CCCCC(=O)N1 10736,c1(C(N2CC3C(CNC(c4c(OC)scc4)=O)(C3)C2)=O)cc2cccnc2cn1 10737,C1(OC)CN(C(=NCc2n[nH]cc2C2CC2)NCC2CCCCO2)CC1C 10738,Cc1c(C(F)(F)F)n[nH]c1C(N1CC(CNC(c2cccc(N)n2)=O)CC1C)=O 10739,c1(CC)nc(Cl)nc(N2C3CCC2C(CNC(=O)CCC2CCC2)C3)c1C#N 10740,FC(F)C(F)(F)CCN=c1[nH]c(N2CC=C(Br)CC2)nc(Cl)c1F 10741,c1(OCC(N2CC(CNC(C(C)(C)OC)=O)C3C2C3)=O)ccc(Cl)cc1C 10742,C1(CNC(Cn2c(C)ccn2)=O)CC2(CC2)CN1C(c1cnn(CCO)c1N)=O 10743,C1(C(C)C)C(C(N)=O)CCN1C(c1cnn[nH]1)=O.c12cnn(C)c1NC2=O 10744,C(=O)(C1=CCCC1C)N1C(CO)CC(NC(c2n(CC)c(O)nc2)=O)C1 10745,C1(C(N(CC(CNC(c2n(CC)nc(C(C)C)c2)=O)C)C)=O)Cc2nccn2C1 10746,c1(NC(N(C(C(CC)C)C)C2CC2)=O)c(F)cncc1F 10747,c1(C(=O)OCc2c(C)ccc(I)c2)nnc2c(C)cc(Br)cn12 10748,S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC(C)CCNC(=O)C(C)OC(C)(C)C 10749,C(=O)(CCN(OC)C(=O)c1coc2c1CN(C(C1OC3CCC1C3)=O)C2)OC 10750,c1(C(C)C)nc(C(N2CCOC(C3CCOC3)C2)=O)nn1-c1ccccc1 10751,c1(COC)csc(COC(C2(CC(=O)OC)CNC2)C)n1 10752,C1(C(=O)OC)CC(NC(=O)NCc2cn(C)nc2O)CCO1 10753,c1(CNC(C(C2CCCN(C(=O)CCc3ccncn3)C2)C)=O)cccc(Cl)c1 10754,CCCC(C(=O)OCC(c1ccccc1)C(=O)OC1CCCOC1)n1cccc1 10755,c1(CNC(c2ccc(SC)cc2)c2ccccc2)c(Cl)cc(C(N)=O)cc1Cl 10756,c1(C(=O)NCC(C)CNC(c2cnoc2C2CCC2)=O)cc(F)cc2nn[nH]c12 10757,c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2csc(Cl)c2)cn(C)nc1Cl 10758,Cc1c(C(=O)NCC2(O)CN(C(=O)C(F)C3CCC3)C2)cnn1C1CCCCC1 10759,C1(C)(C(=O)NC(c2ccccc2F)CNC(CC2(C)CC2(Cl)Cl)=O)COC(=O)OC1 10760,CC(C)(C)C(=O)NCC1CCCC1NC(=O)C(c1ccccc1)SC(F)(F)F 10761,C(CC(C(=O)NC(c1ncc(F)cn1)C)NC(C1CC(F)C1)=O)=CC 10762,N1(C(=O)NCC2(CC(F)(F)F)CCCOC2)CCC(C2(O)COC2)CC1 10763,C12CN(CCO1)CCS2.C1(C(=O)NNC(c2cc(C3CC3)on2)=O)(CO)CCCO1 10764,C1(CNC(CC=C)=O)CC(C)(C)CN1C(=O)COCC1(O)CCCOC1 10765,C1(CCC)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)NCC1CCCS1 10766,N1(C(c2scc(C)c2)=O)CCC(NC(c2cnc(C3CC3)s2)=O)CC1C1CC1 10767,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10768,N1(C(C2C(CC)CCC2)=O)CCCC2(C1)CN(C(c1cccc3ncnn13)=O)C2 10769,c1ccc(NC(C2(C(=O)NC3CCC(OC)(CO)CC3)CC2)=O)c(O)c1.COC 10770,CCCCC(C)CCC(=O)NCC1CC(F)(F)CN1C(c1coc(C#N)c1)=O 10771,c1(C(N2C(CNC(=O)Cc3ccc(Cl)cc3)CCC2)=O)cc([N+](=O)[O-])sn1 10772,CC1CC2(CC(C(=O)NCCOC3CCN(C(=O)CC(=O)N(C)C)C3)C2)C1 10773,CC1CCN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC1OCCCC1(C)C 10774,C1(CNC(CC2(OCC)CCC2)=O)CN(C)CCN1c1ncnc(Cl)c1CC 10775,C(=O)(CCC(CC)NC(=O)C(C)(C)C(C)O)NCCn1ncc(CC)c1 10776,Cc1ccc(C(O)C(=O)NCC2(NC(C34CCC3C4)=O)CCCC2)cc1 10777,N#Cc1ccc(C(CO)NC(CN(C(N)=O)Cc2ncc[nH]2)=O)cc1 10778,C1(NC(CS(CC)(=O)=O)=O)CCC2CCN(C(c3ccco3)=O)C1C2 10779,C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 10780,C1(C(=O)OC)CC(C)(C)CCN1C(c1cccc(C)n1)C(=O)NC1CCOC1 10781,Nc1c(C(=O)NC2CC(CCNC(=O)CN3CCCC3CO)C2)cc(F)cc1Cl 10782,c1(CC(C(=O)C(C(N2CCSCC2)C)=O)O)ccc(F)cc1.C1(C(NC)=O)CC1 10783,c1(NC(=O)Cc2cc(F)cc(Br)c2)ccc(OCCF)cc1F 10784,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2CC)=O)c1N 10785,C(=O)(CN=S(C)(C)=O)N1CCC(NC(c2nc(COC)oc2)=O)C1 10786,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10787,Cc1cc(C(=O)NCC2(CNC(=O)CC3COC(=O)C3)CCC2)n(CC(F)F)n1 10788,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10789,C1(C(=O)Nc2cn(CCOC)nc2)CC(C)(C)CN1C(c1coc(N(C)C)n1)=O 10790,C1(NC(C2(C(=O)OC)CC2)=O)CCCCC1NC(=O)C=CC1CC1 10791,C(=O)(C(=O)CCCC)N1CCC(N(C(CC=C(C)C)=O)CC2CCCO2)CC1 10792,C1(NC(c2n(CC)nnc2)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10793,c1(C(N(C2CCN(C(=O)Cc3cscc3F)C2)C)=O)nncc2c1CCCC2 10794,C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC1CN(C(c1sncc1C)=O)C2 10795,C1(C(=O)OC)CCC2(CCC2)N(C(C2(O)CC(CN)C2)=O)C1 10796,C1(NC(C2CC3C=CC2C3)=O)CCC2(CCN(C(=O)COC3CC3)C2)C1 10797,C1(NC(C2CC(NC(C(C(C)C)O)=O)C2)=O)CC(C)CCC1O 10798,c1(CC)nc(N2CCC(C)C(NC(c3cnnn3CC)=O)C2)c2ccsc2n1 10799,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10800,Cc1cc(OCC(=O)NC2CC(NC(C3CCOCOC3)=O)C2)ccc1Cl 10801,C(=O)(CCC[N+](=O)[O-])N1C(C(C)NC(CC(c2c(C)noc2C)C)=O)CCCC1 10802,C1(C(=O)NC(C(=O)NCC(C2CCCC2)C)C2CCC2)CC2C=CC1C2 10803,Cc1nn(C)c2c(N3CCC(C(N)=O)C3)nc(=NCC3(C)NC(=O)NC3=O)[nH]c12 10804,C(N=c1[nH]c(NC2CC23CC3)nc2ccccc12)N(CC(=O)NCC(C)C)C 10805,c1(OC)ccc2ccc(CN3CC4CC(C3)N4C(C3(C)COC3)=O)cc2c1 10806,C1(C(=O)NCCOCCNC(C2(COC)CCC2)=O)C=CCCC1 10807,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10808,C1(CNC(c2cc(OCC)no2)=O)CN(C(c2c(C(C)C)n[nH]c2C)=O)CC1C 10809,c1(C(=O)NCC(CC)(C)NC(c2ccnnc2)=O)cccc2c1ncn2C 10810,N1(C(CN(C(C)=O)C)=O)CCC(C2N(C(=O)CC3CC3(C)C)CC2(C)C)CC1 10811,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10812,C1(C(N2CC(CNC(=O)CSC)C(C(F)(F)F)C2)=O)(COC)CC=CCC1 10813,c1(OC)cc(CCC(=O)NC(C)C(CO)NC(c2cnsc2C)=O)on1 10814,Cc1ccsc1C=CC(N1CCC(OCCNC(=O)CCC2CCCN2C)C1)=O 10815,C12(C(N3CCC(C)(CNC(c4ccccc4CO)=O)C3)=O)CC(C)(CCO1)C2 10816,CCC(C)CCC(O)CC(=O)NCCNC(=O)Cc1ccc(C)nc1 10817,C12(C)CCC(C1)NC(=O)C(=O)NCC2.c1(CN(S(C)(=O)=O)C(C)=O)ccccc1 10818,c1(CC(N2CC(NC(c3cncc(C#C)c3)=O)C2)=O)cn2cc(C)sc2n1 10819,C1(CN(C(C(C)NC(CC)=O)=O)C(C)C)CCN(C(=O)COCCF)C1 10820,Cc1cccc(C(=O)NCCC(C)NC(c2ccc(C3CCCCC3)cc2)=O)c1 10821,C(CCCCC(=O)NCCc1cnc(C)s1)NC(C1(OC)CCC1)=O 10822,N1(C(C(C(C)C)F)=O)CC2CCCC(Nc3ncccc3C(F)(F)F)C2C1 10823,CC(C)CC(C)OCCC(=O)N(CC(C)(C)NC(=O)CN1CC=CC1)C(C)C 10824,c1(CCNC(=O)CN2CCN(C(=O)Nc3ccccc3)CC2)cnc(Cl)c(Cl)c1 10825,CCC(F)(F)CC(=O)N1C2CCC(C2)C1CNC(=O)C(C)Oc1ccccc1 10826,C1(C(=O)NC2CC(NC(CCCC#CC)=O)CC2O)CCc2nn[nH]c2C1 10827,c1(SC(C)C(=O)NCCCN(C(c2cn(C(C)C)nn2)=O)C2CC2)ccccn1 10828,C1(O)(C(N2CCCCC2CC(=O)NC2CC(CF)C2)=O)CCOCC1 10829,c1(OC(C)C)ncccc1C(=O)NCC1CC(NC(=O)CC2CC23CC3)CCO1 10830,Cc1ccc(-c2cn(-c3nccnc3C(=O)NCC3COC(C)C3)nn2)c(Cl)c1 10831,c1(NC(C(CN(C(=O)CC2CCCS2(=O)=O)CC)SC)=O)ccc2nn[nH]c2n1 10832,N1(C(C(c2cnccn2)C)=O)CCC(C)(C)CC1C(=O)N(C(C)CO)C 10833,C(c1ccccc1Cl)=C(C)C(=O)NCC1CCN1C(C1CC(C)(O)C1)=O 10834,c1(CNC(C2C=CC(NC(C3(C(C)(F)F)CC3)=O)C2)=O)cc(F)cc(Cl)c1 10835,S(=O)(=O)(c1cccc(N2CCC3(CC2)CC3)n1)NCC1CCC(C)C1 10836,C1(C)(CC)CC(OCC2(CC)CCOCN2C(=O)OC(C)(C)C)CCO1 10837,C1(NC(C2CC2NC(=O)C(=O)NCCCOC)=O)CCN(C(C)(C)C)CC1 10838,c1(COC)cnc(N2CCCC2NC(c2cc(OC)ccc2OC)=O)c(Cl)c1 10839,CCC(C)C(CC(=O)NC1CCC1CO)NC(=O)C(C)(C)C1CCOC1 10840,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10841,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CC)c(C)coc1CC 10842,c1(CN(CC(=O)NCCc2cncs2)CC2CC2)ccc(F)cc1Br 10843,CC(C)C(C(=O)N(CCC(C)NC(C1CCC(=O)C1)=O)C)N(C)C 10844,N(C1COc2ccc(Cl)cc21)CC(=O)NCC1COc2ccccc2C1 10845,c1(NC(C2CN(C(c3cnc(COC)s3)=O)C2)C)nc(C)nc2sccc12 10846,c1(C(=O)NC(C2CCCN2C(=O)CC2(O)CCC2)C)cccc2ccncc12 10847,c1(C(=O)NCC2N(C(c3nc(C(C)=O)sc3)=O)CC2)cccc(I)c1C 10848,C1(NC(=O)NCCn2cc(CN3CCC(=O)NC3=O)nn2)CNC(=O)CC12CCC2 10849,N1(C(c2cnn(C)n2)C(=O)NCC2CCOCC2)CCCC(c2ccnn2C)CC1 10850,c1(OC)ccc(CO)cc1CN1CCC(O)C(C(=O)Nc2nc(C)ccc2F)C1 10851,C12(CNC(c3n(CC(C)C)ncc3)=O)CC1CN(C(C1CC(C)(F)C1)=O)C2 10852,c1(NC(C2(C)CN(Cc3c(N(C)C)cc(F)cc3)C2)=O)cc(Br)cc2[nH]ccc12 10853,Cc1cn(C(C)C)cc1C(=O)NC1CC(CCNC(=O)CC=CC(C)(C)C)C1 10854,CCC(C)(CNC(=O)CCC1CCCN1C)C(=O)NC1CC1CCOC 10855,N1(C(c2cncc(OC(C)C)c2)=O)CCC(NC(C2(C)CCC2)=O)C(C(C)C)C1 10856,C1(CC#C)(C(=O)NC(c2noc(C)n2)C)CCN(C(c2nnsc2C)=O)C1 10857,c1(C(C)(C)C)ncc(C(=O)NCCC2CCN(C(c3cn(C4CC4)cn3)=O)C2)o1 10858,N1(C(Cn2c(C)nnn2)=O)CCCC(NC(c2ncoc2C2CC2)=O)C(F)C1 10859,N1(C(C(C)C2CCOC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10860,c1(C2C(=O)NCCCS2)cc(F)cc(F)c1.C(CC1CC1)SCC 10861,N1(C(CNC(CC)=O)=O)CCC(C(=O)NCCCC(C)(C)C)C12CCC2 10862,N1(C(c2cnc(-c3ccccc3)[nH]2)C(=O)NCC)CCC(NC(N)=O)C1 10863,N1(C(Cc2cc(OC)c(O)cc2)=O)CCC2(CNC(=O)CC3CC3)CCCCC12 10864,c1(OCOC)ccc(C(=O)NC(C)C(C)NC(c2ocnc2C)=O)cc1 10865,c12ccc(cc1)OCC(=O)C2N.CCCCN(C)C 10866,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(C(CC)CC)C1)=O 10867,c1(C(=O)NC2CC3(C2)CC(NCc2ncc(Cl)cn2)C3)noc2ccc(Br)cc12 10868,c1(CCC2CC2C(=O)NN(CCCN(CCCOC)C)C)ccnn1CCF 10869,Cc1cc(C(=O)NC2CC3CC2CN3C(=O)CC2(CO)CC2)cc2nn[nH]c12 10870,CCCC(C(=O)N(C(C)CC(=O)Nc1nnn(C)c1C)C1CC1)NC(N)=O 10871,CN(C)S(=O)(=O)N(C)CC(=O)OCc1nnc(C(C)(C)C)s1 10872,C(=O)(C(O)C1=CCCCC1)N1C(CNC(c2c(C)cnn2C(C)C)=O)CCC1 10873,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10874,c1(C(N2CCC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 10875,c1(C(=O)NCC(C(C(C)C)C)NC(=O)CC2(C)CC2)cc2ccc(O)cc2[nH]1 10876,C1(CCNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10877,c1(C(N(C(C)C(N2CCC(CC(N)=O)C2)=O)CC)=O)cccc(=O)n1C 10878,n1(CCC)c(C(N2CCC(NC(=O)C(O)C(F)F)C23CC3)=O)cc2ccccc12 10879,C(=O)(CCCc1nncs1)NCC(C)(C1CC1)NC(=O)CCOCC1CCC1 10880,C1(OCC=O)CCN(C(=O)C(O)Cc2ccc(Cl)cc2)CC1.C(COCCN)OC 10881,C(=O)(CC=CC(C)(C)C)NCC=CCNC(CC1(C)CC1)=O 10882,c1(C(=O)NC2CCN(C(c3c(OC)nccc3)=O)C2(C)C)ccc(S(C)=O)cc1 10883,C(N=c1[nH]c(=NCc2cn(C)nc2Br)[nH]c2c1CC(C)CC2)C1CN(C)C(=O)C1 10884,C1(N(C(C2(CNC(CC3CC(=C)C3)=O)CC2)=O)C)CCCC(C)C1C 10885,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10886,S1(=O)(=O)c2ccc(cc2Cl)NCCN1C.c1(C(=O)NCCSC)cccc(Cl)c1 10887,C(=O)(CCCCC(N)=O)N1CCC(C(=O)Nc2ccc(OC)cc2F)C(O)C1 10888,C(=O)(CCCC(C)(F)F)N1CC(NC(C(C#N)=CC(C)C)=O)C(C)(C)C1 10889,c1(C(=O)NC(C)CCNC(=O)C=CC2CC2)c[nH]c2cccc(Br)c12 10890,c1(C(N2CCN(C(Cc3cc(C)no3)=O)C(CO)C2)=O)c(F)c(F)cc(F)c1F 10891,C(=O)(CP(C)(C)=O)NC1(C(=O)NC(c2n(C)ncc2)CO)CCCC1 10892,c1(NC(C2N(Cc3ccc(C(=O)OC)cc3)CCC2)=O)nnc(Cl)cc1Br 10893,c1(N2CCC(CNC(C3=C(C)CCOC3)=O)C(O)(C)C2)cc2nnc(C)n2cn1 10894,N1(C(C2(C(C)OC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10895,c1(C(=O)OCC)c(N(C)CC(c2ccccc2C)NC2CC=CCC2)ncnc1Cl 10896,C1(C(N2CCC(N(C(CC3(OC)CC3)=O)C)C2)=O)Cc2ccccc2O1 10897,C1(O)(CN(C(C(C)=C2CCCC2)=O)C)CCCN(C(C2CN(C(C)C)C2)=O)C1 10898,C1(C)(C(=O)NCC(C(C)C)NC(=O)C(C)S(N)(=O)=O)CC2(CCC2)C1 10899,N1(C(CSCC(N)=O)=O)CCC2(CC1)COC(CNC(C1CCCCO1)=O)C2 10900,c1(CCNC(=O)NC(CO)CF)nc(-c2cccnc2)no1 10901,N1(C(c2nn(C)c(F)c2)=O)CCC(NC(C2(C3CC3)CCCO2)=O)C(O)C1 10902,c1(C(=O)NC(C)CN(C)C(c2cccc(CS(C)=O)c2)=O)cccc2nsnc12 10903,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)NC1(C)CC(N(C)C)C1 10904,C(CO)(CCCCNC(N1CCC(SC)C1)=O)NC(CCC(=O)NCC)=O 10905,N1(C(C)C(=O)NCC2(CCNC(=O)CCCN(C)C)CC2)CCc2sccc2C1 10906,c1(COC)nc(C)c(C(=O)NCCC(C(C)C)NC(c2n[nH]cc2C(C)C)=O)s1 10907,C1(NC(c2c(OC)n[nH]c2)=O)C2CCC1N(C(=O)Cn1ccc(Br)cc1=O)C2 10908,c1(CC)c(F)cc(-n2cc(C3CN(C(C4CCCN4C)=O)CCO3)nn2)cc1F 10909,n1(CC)cc(CN(C)C(C2CCC(NC(=O)CC(C)N(C)C)C2)=O)cn1 10910,C1(CN2CC(CCCCNC(CC3CCCC(C)(C)O3)=O)C2)CCC2(CCC2)OC1 10911,c1(C(N(CCC)CCNC(c2cccc(CSC)c2)=O)=O)nccc(OC)c1O 10912,S(=O)(=O)(c1ccc(C(=O)N(CC(C)O)CCF)c(OC(=O)CCNC(C)C)c1)NC 10913,N1(C(C(C)(C)NC(=O)NCCC)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(C)C1 10914,c1(C2(C(N3C(CN4CC(C(=O)NC)C4)CCC3)=O)CC2)ccc(F)nc1 10915,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10916,Cc1noc(C)c1S(=O)(=O)N1CCOCC1C(=O)N(CCO)CC1(O)COC1 10917,c12cc3cc(cnc3o1)NC2.c1(C2C(C)CCS2)ccccc1Cl 10918,c1(NC(CC2(N(C(COC(CC)CC)=O)C)CC2)=O)c[nH]nc1SC 10919,c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)c(F)ccc(Cl)c1F 10920,C#CC1CN(C(=O)C(CNC(=O)CC2CCC(C)(C)C2)CC(C)C)CCN1C 10921,C(c1ccccc1Cl)=C(C)C(=O)NCC1CCC1NC(=O)CCCCC1CC1 10922,c1(CC(N2CC(N(C(=O)CCN(C)CC)CC)OCC2)=O)ccc(C)c(OC)c1 10923,c1(C(C(=O)NCCOCCCNC(C(C)Cc2cnc[nH]2)=O)F)ccccc1F 10924,c1(CC(N2C3C(NC(c4occc4F)=O)CC(C3)C2)=O)cccc2occc12 10925,C(=O)(CC(F)(F)C(F)(F)F)NCC1C(NC(c2c(C)n(C(C)(C)C)nc2)=O)C1 10926,C1(CNC(=O)CC2CC(NC(=O)Cn3ccnn3)C2)CNC(=O)CO1 10927,c1(OCC(=O)NC2C(C)CN(C(C34CC(F)(C3)C4)=O)C2)ccc(Cl)c(Br)c1 10928,C1(CNC(c2c(COC)noc2)=O)C(C2CC2)CCN1C1CC(C(=O)NCF)C1 10929,c1(C(=O)NC(C(C)NC(C=CCC)=O)C(C)C)c(C)nc(C(C)(C)C)nc1S 10930,N1(C(CC=CCCCCC)=O)CCC2CCC(C1)N2C(C1(SC)CC1)=O 10931,C1(O)(CCC)CCN(C(C2CCCN(C(C3OCCCC3(C)C)=O)CC2)=O)CC1 10932,Cc1nccnc1CNC(c1csc(-c2ccn(C)n2)n1)=O 10933,Cc1nnc2n1CC(C(=O)NCCN(CCCN(C)C)C(c1cocn1)=O)C2 10934,N1(C(c2ccc(CC)[nH]2)=O)CC(COC)CC1CNC(=O)CSC 10935,C(=O)(C#CC1CCOCC1)NCC(CCNC(c1c(CC)nc(C)o1)=O)(C)C 10936,N1(C(c2ccc(SC)cc2)=O)CCC2(CC1)CC2NC(=O)C(C)N(C)C 10937,c1(C(=O)NCC2CC2CNC(c2cnc[nH]2)=O)cccc(Cl)c1 10938,C(C)(CNC(=O)Cn1cc(C(=O)OC)cn1)(C(C)C)NC(CC(=O)NCC)=O 10939,c1(C(N(CCCCCNC(=O)C2=COCC2)C)=O)cnn2c1N(C)CC2 10940,c1(CN2CCC(CC(=O)NC(C(=O)OCCC)C)CC2)c(C)cccc1Br 10941,C1(NC(C(CN(CCC)CC)F)=O)CC12CC(NC(C1(C)C=CCCC1)=O)C2 10942,c1(CCC)n[nH]c(C)c1Cl.CCCCCCN(C(=O)CNCC)C 10943,N1(C(CSCC#C)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CCC2 10944,C=CC(C)(C)CC(=O)NC(CCOC)C(=O)N1CCC(COC)C1.C1(C)CC1 10945,c1(C(N2CCC(NC(c3cn(C)c(=O)n3C)=O)C(F)C2)=O)cc2ccccn2n1 10946,N1(C(c2nc(OC)sc2)=O)CCC(C2CCN(C(=O)C(=O)NC(C)C)C2)CC1 10947,c1(CCC(N2C(C)CCC(NC(C=C(C)Cl)=O)C2)=O)ccc2ocnc2c1 10948,c1(CC)ccc(C(=O)NC2CC23CC(NC(C2CC2C(N)=O)=O)C3)cc1C(F)(F)F 10949,N#Cc1cc2c(cc1NC(N1CCC3NCC13)=O)CCCC2 10950,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 10951,N1(C(CCCNC(=O)OC)=O)CCN(C(c2ccc(C)c(C)c2)=O)C2CCC12 10952,C1(n2cc(-c3cn(CCC=C)nc3)nn2)CCCN(C(C2CCC(=O)CC2)=O)C1 10953,c1(NC(C2N(Cc3c(C)noc3)CCC2)=O)cc(Br)ncc1F 10954,C1(c2cn(CC(F)(F)F)nn2)(OC)CCN(C(C)C)CC1.C1(C=O)CCCC(C)O1 10955,c1(C(=O)OC)ccc(CNCC2(NC(=O)CC3C=CCC3)CC2)nc1O 10956,C1(C(=O)NC2C(NC(c3cccc(C(F)F)c3)=O)COC2)CS(=O)(=O)CC12CC2 10957,C1(CC)CC2(CCN1C(CCNC(C1CC1CC(=O)OCCC1CC1)=O)=O)CC2 10958,Cc1c[nH]cc(C(N2CC(NC(=O)CSc3cn[nH]c3)CC(O)C2)=O)c1=O 10959,C1(NC(c2ccc(C)c(O)n2)=O)CCC2(CC1)CCN(C(=O)C(F)F)C2 10960,CC1(NC(=O)CCc2nccs2)CCN(C(=O)C(F)CC2CC2)C1 10961,C#CC1(NC(=O)C(CCC=C)NC(c2cnn3c2OCC3)=O)CCCCCC1 10962,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 10963,c1(C(N(CCNC(c2csc(CCC(F)(F)F)n2)=O)C2CC2)=O)ccc(F)cc1 10964,CC1(O)CCC(C(N2CCCOC(CNC(=O)COCC3CCOC3)C2)=O)CC1 10965,c1(OC)cccc(S(=O)(=O)N2CC3CCC2CN3C(=O)C(C)Cn2cccn2)c1 10966,N(C1CCc2c(C(=O)O)ccnc21)C(COc1nc2ccc(C)cc2s1)=O 10967,c1(CCC)cc(C(=O)NC2CCC(CNC(=O)C(O)C3CC3)CC2)ccn1 10968,C(CCCC(=O)N1CCCC1C1(C(N2CCCN(C(C)C3CC3)C2)=O)CC1)OC 10969,C1(C(=O)Nc2cccc(OC(C)C)n2)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 10970,C1(C(=O)NCC2CC3CCC(C2)N3)C2CCCCCCC12 10971,Cc1cccc(Cl)c1C(=O)NC1CC(NC(=O)CCC2CCCCC2)C(O)C1 10972,C1(C(N2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)CSCC(F)F 10973,c1(C(=O)NC2CCCN(C(C(CCC)(C)C)=O)C2CC)nccc2ncncc12 10974,C1(N(C(c2cccn2CC)=O)CC)CCCN(C(C2CCC2(F)F)=O)CC1 10975,C1(C(N2CCC(C)(NC(C3CC(O)C3)=O)C2)=O)CCC(C2CC2)CC1 10976,c1(-c2cn(CCCC=O)nn2)ccc(Cl)c(Cl)c1.n1(CC(=O)O)cccn1 10977,CN1CC=C(CCOC)CC1.C1(CNC(C2(N)CC(O)C2)=O)CC2CCC(C1)C2 10978,C12(C(=O)Nc3cccc(O)c3)CCC(CC1)N2Cc1ccccc1 10979,c1(C(=O)NC2CN(C(C3CC(n4cccn4)C3)=O)C2)cnc(C(F)(F)F)cn1 10980,c1(NCC2(F)CCCN(c3ccnc(SC)n3)C2)cnc2[nH]c(C)nc2c1 10981,C12COCCN(C1)C2=O.C(C(=O)C1C(CNC(=O)OC(C)(C)C)C1)=CC=CC 10982,c1(C(N2C(Cc3n(CC)cnn3)CCCC2)=O)ccc2c(c1)C(=O)OC2(C)C 10983,O=C1CCCC2CN(C(=O)C(N)Cc3nc4cc(Br)ccc4o3)CC2N1 10984,c1(NC(=O)NC)nc2ccccc2nc1N1CCCC(F)(COC)C1 10985,c1(CN(C)C(N2CC(CC3CCSC3)C2)=O)ncccc1OC1CCC1 10986,C1(OCC)CC(Cn2cc(C(=O)NC(C3COC3=O)C)nn2)C1(C)C 10987,C12(NC(c3coc(Br)c3)=O)CCC(CN(C(=O)Cc3sccc3Cl)C1)C2 10988,c1(CC)nc(C)n(C)c1C(=O)NC1CCCCCCN1 10989,Cc1cc(C(=O)Nc2ncoc2C2CN(Cc3[nH]c(C)nc3C)C2)c(O)nn1 10990,CC(C)C(C)(CNC(C1CCCC(C)O1)=O)NC(=O)CO 10991,C1(C)(CNC(c2[nH]cc(C(C)=O)c2)=O)CCCN1C(=O)C(O)Cc1cccc(Cl)c1 10992,C1(CNC(C(CC=CC)C)=O)CC2CCCCC2N1C(=O)CCC(=O)c1ccc[nH]1 10993,C1(CCC(N2CCC(CNC(C3CC(C)(C(=O)OC)C3)=O)C2)=O)CC(C)(C)CO1 10994,c1(C(=O)NC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 10995,C(CCC(=O)NCC1(C(N2CCC(CCCO)C2)=O)CCCO1)N(C)C 10996,C(c1ccc(Cl)cc1)=CC(=O)NCCC1CC(OC)CN1C(=O)CCC1CCC1 10997,Cc1nc(C(N2CCC(C(C)(C)C(=O)NCCOC3CC3(F)F)C2)=O)cs1 10998,C(=O)(C(C)CF)N(c1ccccc1)CCNC(C1C(OC)C1)=O 10999,c1(N2CCC(CCC)C2)cc(NC(C)COc2ccccc2)nc(Cl)n1 11000,N1(C(C=C(CCC)C)=O)CC=CC1C(=O)NC.CC(C(F)F)=C 11001,c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C)NC=O)C2)cnc1O 11002,c1(C(=O)CNC(c2cccs2)=O)cc(Cl)ccc1OCC1CCCO1 11003,C1(C)(NC(C(CCN(C)C)NC(c2coc(CO)c2)=O)=O)CC2CCC1C2 11004,c1(NC(c2[nH]cc(C(N3CCC(CC(=O)N(C)C)CC3)C)c2)=O)ncc(C)c(C)n1 11005,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(c1cnn(-c2nccs2)c1)=O 11006,N1(C(C(CC)=CC)=O)CCC(N=[N+]=[N-])(C(N2CC(n3cccn3)C2)=O)C1 11007,N(C1CCOc2cc(CNC3CC3)ccc21)C(=O)C(N1CCCC12CCNC2=O)=O 11008,N1(C(c2c(C)[nH]nc2I)=O)CCOC2(CCN(C(=O)C(N)=O)C2)C1 11009,N1(C(CCCC#N)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1CC1CC1 11010,C#CCC(C)(C(=O)Nc1ccc(CC)nc1C)NC(=O)CCCCCF 11011,C1(C(N(C2CCOCC2)C)=O)CC2C=CC1N(C(=O)CC(=O)OC(C)(C)C)C2 11012,CC1(C)C(NC(=O)CN2CCCC2)CC1CNC(C1CN(C2CCOCC2)C1)=O 11013,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11014,C1(C)(NC(C(F)=CCC)=O)CCN(C(=O)CCc2ccn(C)n2)CC1 11015,CCC(C(=O)NCC1(C(C)(C)O)CN(C(=O)CNS(N)(=O)=O)C1)NC1CC1 11016,N1(C(COCCC#C)=O)CCC(CN(C(=O)CCC2CCC(C)O2)C)CC1 11017,n1(CC)nc(C(=O)OC2CCN(c3cccc(C)c3)C2=O)c(C)n1 11018,C(=O)(C1=CCCSC1)Nc1ccc(C2CCC(CNC(COCC)=O)CC2)cc1 11019,C(=O)(CCC(=O)NC1CC(NC(C2(c3ccccc3)CC3(CC3)C2)=O)C1)NC(C)C 11020,N1(C(CC(CNC(=O)CN(CCCN=[N+]=[N-])C)OC)=O)CCN(C)CC1C 11021,C(=O)(C#CC(C)(C)O)N1CCCC(NC(C(CC)(C)C)=O)C1 11022,N1(C(CN(C(c2cc(CC)on2)=O)C)=O)CCN(C(=O)C(O)C(C)SC)CC1 11023,C(C(=O)NCc1cc[nH]c1C(=O)Nc1cn(C)nc1C1CCC1)(C(C)(C)C)OC 11024,c1(C(=O)NCC(CCOC)NC(=O)C=C(C2CC2)C2CC2)ccc2snnc2c1 11025,N1(C(CCCSC)=O)C2CCC1C(CNC(c1cc(Br)c[nH]1)=O)C2 11026,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(=O)Cc2n[nH]c(=N)s2)CC1 11027,C1(C(=O)NCCCOCCCO)C2CC3C(C2NC(C2(CC)CNC(=O)C2)=O)C13 11028,C1(NC(C2CC2CF)=O)CCN(C(=O)COc2ccccc2)C1C1CC1 11029,N1(Cc2cn(CCN3CCN(C)CC3)nn2)CCC(C(C2COC(=O)N2)C)CC1 11030,C(=O)(CN=S(C)(C)=O)N1C(CN(C(=O)CSc2ccncc2)C)COCC1 11031,N1(C(c2cnc(COC)s2)=O)CC=CC(NC(=O)CC2CCCO2)C1 11032,CCC(CO)CCNC(C1C=CCCN1C(=O)Cc1cn[nH]c1)=O 11033,N1(C(C(C(C)NC(=O)CC2CCCCC2)C)=O)CCCC(C)(C)C1 11034,C1(CNC(c2c(C)cco2)=O)C(C2CC2)CCN1C(c1ncc[nH]c1=O)=O 11035,c1(CC)nnc(CN2C(C3COC3)C2=O)s1.OC.OC 11036,C=CCCCC(C(=O)NC(C)(C)C)NC=O.C(C=C)(C(F)(F)F)N 11037,c1(C(N2CCC23CN(C(=O)Cc2ccncc2)C3)=O)cccc(OC(F)F)c1F 11038,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11039,c1(C(N2C3C(NC(C(C)CN(C)C)=O)CC(CC3)C2)=O)nccc2cccnc12 11040,C1(NC(C(CC)CC)=O)CCN(C(c2ccoc2)=O)C(c2ccccc2)C1 11041,CC(C)(CNC(c1nn[nH]c1C(F)(F)F)=O)CNC(=O)CCc1cncnc1 11042,Cc1cc(CCC(N2CCCCC2CNC(C2C=CC=CC=C2)=O)=O)cc(C)n1 11043,C1(NC(N(CC)CC2CCSC2)=O)CCCCC12CCCC2 11044,c1(C(=O)NC2C(C)N(C(=O)Cc3cncnc3)CCC2)cn2ccccc2n1 11045,c1(C(N(C(C)CNC(C2CN(C(N)=O)C2)=O)C)=O)nc2c(s1)COCC2 11046,N1(C(CC2CC(NC(c3c(=N)[nH]cnc3)=O)C2)=O)CC2(CC=CC2)C1 11047,c1(C(CNC(C2CCCCC2)=O)Nc2c(C(=O)OC)ccnc2)ccc(F)cc1 11048,N#CC1CCN(C(=O)NC2CCOCC2C(=O)NC2CCCCC2)CC1 11049,c1(CNC(C2C=CCN(C(c3c(CC)nccn3)=O)C2)=O)cnc(F)cc1C 11050,N1(C(C(CC=C)C)=O)CC(NC(c2ccnnc2O)=O)CC(C)C1 11051,CC(CN(C)C)CCC(=O)N1CCN(CC(N2CCOC(CF)C2)=O)CC1 11052,C(=O)(CCC(=O)NN(C)C)N1CCN(C(C2C(C)OCCO2)=O)CC1CO 11053,c1(CN(C(C2CCCO2)=O)C)nc2c(s1)CN(C)CC2.C12CCCCN(C1)C2=O 11054,C1(CNC(Cc2c(C)cccc2)=O)CC2(CO1)CN(C(c1c(C)n[nH]c1C)=O)C2 11055,C1(O)(CC(=O)NCC(C)OC(C)(C)C)CCN(C(=O)CCc2nc[nH]n2)CC1 11056,c1(C(CNC(C)=O)OC)cn(CC(F)CCNC(=O)C(F)F)nn1 11057,C12CCCCC1CNC2=O.CC1(C(N2CCCC2Cc2ccccc2)=O)CCOC1 11058,c1(CN2CC(O)(CCNC(c3cnn(-c4ccccc4)c3)=O)C2)cccc(Br)c1 11059,N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C(F)OC(F)(F)F)C(C)C1 11060,c1(OC)ccc(Br)cc1CC(N1C(C(N2CC(CC(C)C)C2)=O)CC2CC12)=O 11061,N1(C(C(=O)NC(CC)C)CCCC(C)C)CC2(C1)NC(=O)NC2=O 11062,c1(CCN(C(=O)COC(c2ccccn2)=O)C)cccc(F)c1 11063,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11064,c1(C(COC(CSCCSCC#C)=O)=O)ccc(Br)c(Cl)c1.C1CO1 11065,CCC(C)CC(=O)N(CCCNC(C1(c2ccc(Cl)s2)CC1)=O)C(C)C 11066,c1(CC)ncccc1C(N1CCC(CCC(=O)OC)CC1)C(=O)NC1CCOC1 11067,N1(C(c2c(C)coc2)=O)CCN(C(=O)CC23COCC(C2)C3)C(C)C1C 11068,c1(C(=O)NC(CSC)C(=O)NC2CCC(F)(F)C2)cc(C#N)ccc1F 11069,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11070,c1(CC)occ(C)c1C(=O)NCC(C)C(=O)N1CCCC1C(=O)N.NC 11071,C(=O)(CN=c1cc[nH]cc1)N1C2CN(C(c3c(N)ccc(Cl)c3)=O)C(CC2)C1 11072,Cc1ccc(C(=O)O)c(-n2cc(-c3ccns3)nn2)c1.C12CCCN(C1)C2 11073,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11074,c1(OC)c(NC(=O)NCC(C)(O)CCO)cnn1C 11075,C(CC(C)C(=O)NCC1(F)CCC(NC(=O)CCc2cncc(OC)c2)C1)OC 11076,C1(O)(C2C(=O)NOC2)CCCCC1.C=CCN(C)CCNC(C)=O 11077,Cn1oc(C(=O)NC2CCCC2CNC(C23CC(C(F)F)(CO2)C3)=O)cc1=O 11078,c1(C(=O)NCC)cc(Cl)ccc1Cl.C1(N)CCOCC1.c12cn(nn1)C2 11079,c1(C(NNC(C(=O)N(C(C)C2CC2)CC)=O)=O)cn2c(n1)C(C)CCC2 11080,N1(C(C2C(=C)C2)=O)CCCCCC(NC(=O)C(C)SC)C1 11081,Cc1ccc(C(C(=O)N(CCCCCNC(C2(F)CC2(F)F)=O)C)C2CC2)cc1 11082,C1(CNC(CC(=C)C)=O)CN(C(c2ccc(C(C)C)nc2O)=O)CCCO1 11083,CN1CCCCC1CC(=O)NC1CCCC1(C)CNC(c1csc(C(F)F)n1)=O 11084,c1(C(=O)NC(CC)CN(C(=O)C(C)CSC)C)cc(OC)c2c(c1)OCO2 11085,C1(CC(=O)NC2C(NC(c3cnc(C(C)C)s3)=O)C2)CC(=O)NC1=O 11086,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11087,c1(OC)ccc(C)c(C(=O)NCC2(CCCNC(=O)C=C(C)C)CCCC2)n1 11088,O=S(=O)(c1cccc(F)c1F)Nc1ccc(-c2cccc3c2OCC3)s1 11089,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cc(Br)n(C)n2)=O)ccc1C 11090,c1(C(N2CCC(N(C(=O)CC3CCC(=O)N3C)C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 11091,c1(C(N2CCC(CC)C2C(=O)NCC2CC(C(C)C)C2)=O)ccc2n[nH]cc2c1 11092,c1(OCC(=O)NCC2C(CNC(C(C)C3CCC3)=O)C2)cccc(Cl)c1Cl 11093,c1(N2CC3CCN(C)C3C2)nc(=NCc2nnc(C(C)(C)C)s2)[nH]c2ccsc12 11094,c1(C(N(C2C(O)CCN(C(c3nc(C)oc3C)=O)C2)C)=O)cccc2c1OCC2 11095,C(=O)(C(CC(N)=O)NC(C1CC2(C1)CC21CC1)=O)NC1(C(C)C)CCC1 11096,Cn1cnn(CC(N2CC(CNC(=O)CCc3ccc(Cl)cc3)C2)=O)c1=O 11097,C1(n2c(C)ncn2)COCCN1N1CCC(CO)CC1.C(C)C 11098,c1(CC(N2C(C(=O)NC34CCN(CC3)C4)(CC)CCC2)=O)coc2ccccc12 11099,c1(C(N2CC(CC)N(C(c3cscc3C)=O)CC2)=O)cnn2ccc(OC)cc12 11100,c1(CCC)cc(NCC2CN(C(=O)C(C(C)C)NC(C)=O)CCO2)nc(Cl)n1 11101,C1(C(=O)NC(C)CN2CCCC2)C2CCCC2CN1C(=O)Cn1ccc(Cl)n1 11102,N1(CC)CC(NC(=O)Nc2ncn(C(C)C)n2)CC1=O.C12CN(C1)C2=O 11103,n1(CC(=O)NC2CCCN(C(C3OCCCO3)=O)C2)nc(O)ccc1=O 11104,CCC(CNC(=O)C(=O)NC1CC(=O)N(C(C)C)C1)(CC)c1ccccc1 11105,Cc1c(C(=O)N(CCC(=O)NC(CO)CCF)C2CC2)ccn1C 11106,c1(-c2cn(CC3CCN(C(CN(C)C)=O)C3)nn2)cc(CO)ccn1 11107,CCC(C(=O)NC1(C(=O)NCC(F)Cl)CC1)C(C)C 11108,c1(C(=O)NCC2C(CNC(c3cccc(OC(F)F)n3)=O)C2)ccc(F)c(Cl)c1F 11109,CC1(C)C(C)(C)C1(F)C(=O)NCC1CCCN(C(c2nnc(O)nc2O)=O)CC1 11110,c1(C(=O)NCCN(C2CCCC2)C(C2CC3CCC2O3)=O)nc2ccccc2s1 11111,C(CCNC(N)=O)(C(=O)OCCOCCCC1CCOC1)N(c1ccccc1)C 11112,CN1CCCCC(C(=O)NCC(C)(C)CNC(C2(C)CCC(=O)C2)=O)C1=O 11113,c1(CCC)noc(CCC(=O)NC2CCN(C(=O)C=C(C)C(F)F)C2)n1 11114,C1(CNC(c2occ(C)c2)=O)CC(C)N(C(c2cn(C(C)(C)C)cn2)=O)C1 11115,C(C)(CCC(C)(C)C)NC(Cn1c(SCCC)nnn1)=O 11116,CC(C)P(=O)(CC(=O)NCC(C)CN(C(=O)C=CC(=O)N(C)C)C)C(C)C 11117,C1(O)(CSC)CCCC1C.C12(CCCC1)C(=O)NCCC1(CC1)C(=O)N2 11118,CCCCC(CNC(=O)CCOc1cccc(F)c1)NC(C1(OC(C)=O)CC1)=O 11119,CC(=O)C(C)CC(C)C(=O)N(C)CCN(C)C(c1n[nH]c2c1CCC2)=O 11120,c1(C(=O)OCC(=O)NC(Cc2ccncc2F)C(=O)O)cccc(F)c1C1CC1 11121,c1(C(C)N(C)C(=O)N(C)CC2CCCO2)cnn(C)c1 11122,Cn1nnc2ccc(C(N3CC(NCc4ccc(I)cc4)C4(CC4)C3)=O)cc12 11123,N1(C(c2ccc(CC)s2)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(CO)C1 11124,c1(C(=O)NC2C(CNC(CC(=O)NC3CC3)=O)C2)nnc2ccccc2n1 11125,c1(NC(C(C)NC(c2ccoc2)=O)=O)cccc(CNC(C2(C)CCOC2C)=O)c1 11126,c1(CC(C)C(=O)NCC(O)CN(C(=O)CN2CSCC2=O)C)ccc(Cl)c(Cl)c1 11127,N1(C(C(C)=CC)=O)CC2CCN(C(c3nc4ncc(C)cn4n3)=O)C(C2)C1 11128,N1(C(CCC2(NC(COCCOC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 11129,C(CC(C)(C)C(=O)NC(C1CCOC1)CNC(c1cnc(OC)cn1)=O)OC 11130,C(C(CCC(=O)O)C(F)(F)F)NC(NNC(=O)c1c(Cl)cccc1Cl)=S 11131,N1(C(C(CN(C)C)O)=O)CCCC(C)(NC(=O)Cc2ccsc2Br)C1 11132,N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C)N(C(c3ccsc3Cl)=O)C2C1 11133,c1(CCC)cc(C(=O)NCCC(C)NC(C2(C(F)F)CC(O)C2)=O)c(C)o1 11134,CCCC(O)C(CO)NC(C1CC=CC(NC(=O)Cn2cnnc2O)C1)=O 11135,CCCCC(O)C(=O)NC(CCC(=O)N(CCO)CCN(C)C)C(C)C 11136,C(=O)(CCS(=O)(=O)C(F)(F)F)Nc1n(C)ncc1C1CC1.C12COCC1C(=O)N2 11137,CC1COCCC1N(C(=O)CCC1CC(NC(=O)CCn2cccn2)C1)C 11138,C1(NC(c2ocnc2C2CC2)=O)CN(C(=O)COC2CCCC2)CCC1CO 11139,CC(C)CC(C(=O)N1CC(C(=O)NCc2ncoc2C2CC2)CC(C)C1)C(N)=O 11140,CC(C)(C)C(CNC(=O)C(O)Cn1cncn1)NC(=O)C(O)C1CCC1 11141,C(=O)(C(O)CCCNC(=O)CC1CCSCC1)NCC(C)(CO)OC 11142,N1(C(c2cnc3n2CCCC3)C(=O)NCC(C)C)CCC2(CCN(C)CC2)C1 11143,N1(C(C(CC)OC)=O)CCC(C(F)F)(CNC(=O)CCn2cccnc2=O)C1 11144,c1(CC(N2CCC3CN(c4ncc(F)cn4)CC23)=O)cc(F)c([N+](=O)[O-])cc1F 11145,c1(C(=O)NCC(CC)NC(C2(O)CCOC2)=O)ccsc1C(F)F 11146,c1(C(=O)NC(C2N(C(CC(C)O)=O)CCCC2)C)ccc(S(=O)(=O)CCO)cc1 11147,N1(C(CSCC#C)=O)CC2CCC1CN2C(=O)CC1CCC1C1CC1 11148,C1(CNC(C2CCC(CC)O2)=O)CC2CCC1N2C(C1(C)CCC(=O)C1)=O 11149,C(=O)(C1CCC(=O)c2ccccc21)NCC(CNC(c1c(C)nn(C)c1F)=O)O 11150,c1(CN(c2nccc(N3CCCCC3CC(N)=O)n2)C)ccc(Br)cc1F 11151,CC1(NC(c2c[nH]c(C(F)(F)F)c2)=O)CC(NC(C2CCCS2)=O)C1 11152,C(N=c1cc[nH]cc1S(=O)(=O)N(CCCF)C)c1cnc(CC)s1 11153,N1(C(C(C2CCCC2)NC(C2NC(=O)CC(C)C2)=O)=O)CCC2CCC(C1)N2C 11154,C1(C(=O)NC(CC(C)NC(C(C)(C)OC(C)C)=O)C)CC12CCOC2 11155,CC(CN(C)C)CCC(=O)NCC1(C(N)=O)CN(c2ncc(O)cn2)C1 11156,N1(C(C(C)N(C(=O)CC2CCCC(C)O2)CC)=O)CC2(COC(=O)C2)C1 11157,c1(C(=O)NC23CC(NC(C=CC=CCC)=O)(C2)C3)ccc(CO)c(C)c1 11158,C(=O)(CCCCCNC(C1CCOCC1)=O)N1CC(CN(C)C)C1 11159,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11160,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11161,c1(C(N2CCC(N(C(C=CSC)=O)C)C(C)C2)=O)ccc2snnc2c1 11162,C(=O)(CC(O)c1ccccc1)NCCC(C)NC(c1nc(Cl)cs1)=O 11163,Cc1nc(NC(C2CCC2)C)cc(=NC(C)c2nc3c(s2)CCC3)[nH]1 11164,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2CCCO)=O)C(F)C1 11165,C(=O)(CC1OCc2ccccc21)N1CCN(CCNC(C(CCOC)C)=O)CC1 11166,Cn1ncc(C2CCC2)c1C(=O)NC1CC1CNC(C1(O)CC1)=O 11167,C1(CCC(=O)N(CCOCC)CC)CCCN1C(C1CC2(CC2)C1)=O 11168,c1(-c2n3nc(n2)C3)cnc2cccnc2c1.Cc1c(Cl)sc(Cl)c1Cl 11169,c1(C(N2CCC(CC)C2CNC(=O)CC2CCCC(C)C2)=O)ccn2ccccc12 11170,C1(NC(C(C)NC(C)=O)=O)CC2CN(C(c3ccc(C)n3C)=O)CC12 11171,N1(C(C(Cc2cn[nH]c2)NC(c2cc(OC)no2)=O)=O)CCOCC1CC(C)C 11172,CC1CC(C(N2CC3(CSC3)C2)=O)CCN1C(C1CC=CCC1C)=O 11173,N1(C(c2ccc(CC)o2)=O)CC2CN(C(c3cnn(CC)c3)=O)CCC12 11174,C1(N=[N+]=[N-])(C(=O)NCC(CCC)OC)CCN(C(=O)CCCC(C)(C)C)C1 11175,N1(C(c2nc(C)ncc2)=O)CC2CCN(C(c3ccn(CCN(C)C)n3)=O)CC12 11176,c1(C(N2CCCCC3(CC3)C2)C(=O)NC2(C)CC2)cccc(C#N)n1 11177,C1(NC(C(C2CCCCC2)N(C)C)=O)CCN(C(=O)CC#N)CC1O 11178,c12nccn1CC2.C(=O)(C(C)(F)F)N(CC(N1CC(C(N(C)C)=O)C1)=O)C 11179,N1(C(=O)CC2=CCCCC2)CCCC2C1CCCN2C(=O)Cc1cnoc1 11180,C(CC(F)(F)Cn1cc(-c2cccnc2)nn1)NCC(=O)Nc1cnoc1 11181,N1(C(C2CC(CC)N(C(c3ccccc3C)=O)CC2)=O)CCC2(CC=CCO2)C1 11182,N1(C(=O)C2CC2)CCC2CN(C(=O)CNc3[nH]c4ccc(C)cc4c3)CC2C1 11183,C1(C(=O)NCCCN(C(=O)CC2CCCCO2)CC)(CF)CCOCC1 11184,c1(CCC(=O)NC(C2CCN(C(C3CC=CCO3)=O)CC2)C)ccccc1C 11185,S(=O)(=O)(c1cccs1)N(CC(=O)NCCN(C(Cc1c(C)nsc1)=O)C1CC1)C 11186,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11187,c1(C(=O)NCC2N(C(CC=C)=O)CCC2)ccc(Br)c2cn[nH]c12 11188,c1(C(N(C2CCCN(C(=O)CC3CCC(C)CC3)C2)CC)=O)c[nH]nc1[N+](=O)[O-] 11189,N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(C)cnc2Cl)=O)CC1C 11190,C1(CC(N2CCC(OCCN(C(C3C(OCC)C3)=O)C)C2)=O)CCCS(=O)(=O)C1 11191,c1(N(CCC(C)(C)C)C)ccc(S(=O)(=O)NCC2CC(CO)C2)c(Br)c1 11192,Cc1cc(C)cc(C=CC(=O)NC2(CCCCNC(=O)CCC(C)(C)F)CC2)c1 11193,CC(C)(CF)C(=O)NC1CCC1CNC(C1CC12CC2)=O 11194,N1(C(c2c(CNC(c3c(C)cno3)=O)occ2)=O)CCN2CCCCC1C2 11195,N1(C(C(Br)=C(C)C)=O)CC(CNC(=O)COC2CCCCC2)CCC1C 11196,N1(C(c2cc(C)oc2)=O)CC(NC(c2cccc(C(F)(F)F)c2C)=O)CCC1C 11197,C(=O)(CCS(C)(=O)=O)N1CCC(CC)C1CNC(=O)C(=Cc1cccnc1)C 11198,C1(C(=O)NC(C)CCF)CN(C(=O)Cn2ccnn2)C2(CCC2)C1 11199,c1(OC)ncc(C=CC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)cn1 11200,C=CC1(CC(=O)NCC(c2ccnn2C)O)CN(C(=O)CCn2ccnn2)C1 11201,Cc1onc(C2CC2)c1C(=O)NC1CCN(C(c2ccc(N)cn2)=O)C1 11202,C1(C(N(C2CCN(C(C(F)(F)C3(OC)CCC3)=O)C2)C)=O)CCCCC1C(N)=O 11203,N1(C(c2c(Cl)cn(C)n2)C(=O)NC2CCOC2)CCCC2(CCCNC2=O)C1 11204,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)CC1 11205,C1(C(N2C(C(C)NC(c3c(Cl)ccc(C)c3)=O)CCC2)=O)CCCC2CCCN12 11206,Cc1cc(-n2cccn2)nc(=NC(C)C2CCCCN2C(=O)CC2CCC2)[nH]1 11207,C1(CN(C(C(C)O)=O)C)CCCN(C(=O)C=CCN2CCC2)C1 11208,c1(C(=O)NC2CCN(CCOC3CCOCC3)C2)ccc(O)c(Br)c1 11209,c1(NC(C(CNC(=O)CCNC(N)=O)OC)=O)cccc(C(C)F)c1 11210,c1(N2C3CN(C(c4c(OC)cccc4F)=O)C(C3)C2)ncnc2c(C)cccc12 11211,CC1=C(C(=O)N2CCCCC2CCNC(C2CCCS2)=O)CCC1 11212,N1(C(c2cnc(C(=O)OC)s2)=O)CC2CN(C(c3c[nH]cc3Br)=O)CC2C1 11213,c1(C(C)C)cc(C(N2CCCC2CN(C)C(C2CCOC2)=O)=O)nc2ncnn12 11214,Cc1cc(O)ccc1CNC(C1CC(NC(=O)CCCn2cccc2)CCO1)=O 11215,c1(C(=O)NCC23C(CN(C(C(CC)COC)=O)C2)CC3)cnc2[nH]cnc2c1 11216,C1(OC)CC(OC)CN(C(=O)NC2CC(CC(Cl)(Cl)Cl)C2)C1 11217,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(C3CC3)C2)CC12CCC2 11218,N1(C(C(COCC)(C)C)=O)CC(NC(=O)C(C)Oc2ccc(F)c(F)c2)C(C)(C)C1 11219,C1(C)(CNC(C2CN(CC)C(=O)C2)=O)CCCN(C(=O)CN2CCCCC2=O)C1 11220,C#CCC(C)(CNC(C1(CNC(c2ccc(OC)s2)=O)CC1)=O)CO 11221,CC(CC(C)(C)C)C(=O)NCC12CC(CO1)N(C(=O)COC1(C)CCCC1)C2 11222,N1(C(CC(C)F)=O)CCCC(CN2CCN(C(c3ccc(C(N)=O)s3)=O)CC2)C1 11223,N1(C(Cc2nc(C)oc2)=O)CC2ON=C(CNC(c3nsnc3O)=O)C2C1 11224,C1(C(N(CC(C)NC(CCCc2ccc(C)cc2)=O)C)=O)CC2CCC(C1)S2 11225,C(=O)(C(C(C)(C)C)OCC)N(CCC)CCNC(C12CCCC1CC2)=O 11226,N1(CC(N2CCC(C3CCCN3C(C34CC(F)(C3)C4)=O)C2)=O)CCC(F)CC1 11227,c1(N2CC(C(C)C)OCC2)nc(NC2CC2C(F)(F)F)c2cnn(C)c2n1 11228,c1(C(C)=O)ccc(CC(=O)NC2CCCN(C(C3(C)CC3)=O)C2)cc1O 11229,C1(OC)(CNC(=O)CCSC)CCN(C(c2nc(Cl)sc2Cl)=O)CC1 11230,Cc1[nH]c(C(=O)NC(C2CCN(C(=O)CC(C)(F)F)C2)C)c(C)c1C 11231,CC1OC(C)C(NC(c2ccc(CNC(c3ccc4c(c3)CC4)=O)cc2)=O)C1C 11232,c1(C(N2CCCC(N(C)C(C3CCCC3)=O)CC2)=O)cc(N)cc(O)c1F 11233,N1(C(C2C(COC)C2)=O)CCCC(CNC(C2CC(C)(C(=O)OC)C2)=O)C1 11234,CC(C)C(CNC(c1ccsc1)=O)C(=O)N(CC(F)F)C1CC1 11235,N1(C(=O)OC(C)(C)C)CC(C)(C2(C(N3CCn4nncc4C3)=O)CC2)CC1(C)C 11236,O=C(C#CC1CCCCO1)NC1C2CC1N(C(=O)CN1CC3CC3C1)C2 11237,Cc1cn2c(n1)CCC(C(=O)NCCN(C(c1ccc(C)n1C)=O)CC1CC1)C2 11238,C1(N(c2cc(OC)ccn2)C(C(=O)NCC(CC)OC(F)F)=O)CCCCCC1 11239,N12CCC(CC1)NCN(C)CCCC2=O.C1(C2CC2)CCCO1 11240,Cc1ccnc(CNC(C2COCCN(C(c3ccncc3)=O)C2)=O)c1F 11241,C1(NC(c2n(CCC)nnn2)(CCOC)c2ccccn2)CC2CCC(C1)C2 11242,c1(C(N(C)CCNC(c2ccsc2Br)=O)=O)ccc2sc(=N)[nH]c2c1 11243,N1(CCNC(=O)NC(C2CCCCC2)c2sccc2Cl)CCS(=O)(=O)CC1 11244,Cn1nc(SCCn2cc(C(C)(C)C(=O)O)nn2)nc1-c1ccon1 11245,C#CC1(C(=O)NCC2CCCN2CC)CCN(C(=O)C(n2ccnc2C)C)CC1 11246,CC1(C)CCCN(C(C2CC(F)(F)C2)=O)C1CNC(C1CCC(=C(F)F)CC1)=O 11247,C(=O)(CCCCCCC(=O)N1CCC(C)C(NC(c2ccc(SC)o2)=O)C1)OC 11248,C12(C(=O)NC(COC)CCO)CCCC1N(C(c1cccc3occc13)=O)CC2 11249,n1(CCC(=O)NCC(C)(CO)NC(c2n(C)ncc2)=O)cnc2ccccc12 11250,c1(C(=O)Nc2cn(C)nc2C(=O)NC(c2n(C)ccn2)CO)ncc(Cl)cc1Br 11251,Cc1cc(CCC(=O)N(CC(C)NC(=O)C(F)F)C)c(C)n1C1CCC1 11252,C=C(Cl)C(C)(C)C(=O)NCC1CC(CCNC(C2CC2c2cccnc2)=O)C1 11253,C(=O)(C1CCc2nccn21)N1C(CNC(C2CCC3(CCC3)O2)=O)CCCCC1 11254,C(=O)(C(CNC(c1cc(O)cc(=O)o1)=O)C(C)(C)C)NCC1CC(CC)C1 11255,C1(NC(C23CC(C)(C2)C3)=O)CCC2CC1CN2C(=O)Cc1ncncc1Cl 11256,C(C)(C)(CC(=O)NCC1CCCCN1C(=O)CC12COCC(C1)C2)OC 11257,c1(C(=O)NCCN(C(C)C)C(c2cc(Cl)cn2C)=O)nc2n(c1Cl)CCCC2 11258,N1(C(CN2CCCC(CC)C2)=O)CCC(NC(=O)Cc2ccsc2C)C12CC2 11259,N1(c2cc(N(C)CC3(CO)CCC3)nc(C(C)C)n2)CCOC2(CCCSC2)C1 11260,c1(C(N2C(CN(C)C(C3CCCCO3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 11261,CC(C)CC(C(=O)N(C)C)NC(=O)CCCCCNC(=O)C(C)C#N 11262,C1(CN(C)C(C2C3CN(C(=O)CC(O)c4ccccc4)CC23)=O)CCCCCC1 11263,CCC(CNC(c1c[nH]cc1C)=O)(CC)NC(c1ccc(C(=O)NC)cc1)=O 11264,N1(C(c2noc(CC)c2C)=O)CCC2(COC(CNC(=O)CCS(C)(=O)=O)C2)C1 11265,Cc1ccc(C(=O)NC2CN(C(=O)CSC3CCCO3)CC2C)n1CC(F)(F)F 11266,CCCC(C(=O)Nc1nc(C)sc1C)NC(=O)COC1CCCC1 11267,N1(C(CCC=CC(C)C)=O)CC2(CCCC2)C1 11268,CCC(CN(C)C)C(=O)NCCCN(C(c1cc(C(C)(C)O)ccn1)=O)C1CC1 11269,C1(CCNC(c2cc(C)on2)=O)CCCCN1C(=O)CCc1cncc(O)c1 11270,C(CCS(=O)(=O)NCC(N1CCC(c2cn(C(C)OC)nn2)C1)=O)OC 11271,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11272,CC1CC(C(N2CCC(n3cncn3)C2)=O)CCN1C(=O)CCF 11273,n1(CC(=O)NC(CCOC)CNC(=O)Cn2ccc(C3CC3)n2)c(C)ccc1C 11274,Cc1ncc(F)c(N2CCC(C)(NC(c3cccs3)=O)C2)n1 11275,C1(NC(c2n[nH]cc2-c2ccncc2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11276,c1(C(N(C2CN(C(=O)C(F)n3cccn3)CCC2O)C)=O)cccc2nccn12 11277,N1(C(CSC)=O)CCCCC1CN(C(=O)C(C)(C)c1ccnn1C)C 11278,c1(CC(=O)NCC(N(C(C(CCC)OC)=O)C)C2CC2)ccc2ocnc2c1 11279,CCC1c2ccsc2CCN1C(c1cccnn1)C(=O)NC1CCCCC1 11280,C(C(C)(C)C(=O)NCCCN(C(=O)C(O)CCSC)CCO)OCC 11281,Cc1cc(OC(F)F)cc(NC(=S)NC2CCCC(C)C2)n1 11282,Cc1cnccc1C(C)C(=O)NCC1(F)CN(C(C2CC2F)=O)C1 11283,CN1CCCC1C=CC(=O)NCC1(NC(=O)C=Cc2ccoc2)CCC1 11284,c1(CCC(=O)NCC(CC)NC(=O)C(C)=CC(C)(C)C)ccc(OC)c(OC)c1 11285,C1(C(=O)NC(CCCNC(c2cccc(CC)c2)=O)C)C(C)OC(C)C1C 11286,C(CO)(C(=O)N1CC(O)(CNC(C2CC2Br)=O)C1)NC(N)=O 11287,c1(C(N(CC(=O)NCC(=C)Br)C)=O)n[nH]c(C)c1O 11288,Cc1cc(Cl)cnc1C(N1CC(O)(CCc2cn(C3CCCCC3)nn2)C1)=O 11289,Cc1cc(F)c(C(N2CCN(CCN3CCCCC3=O)C(=O)C2)=O)cc1F 11290,c1(NC2CCC(C(=O)OC)O2)cc(F)ccc1C(=O)N(C)C 11291,CCC(CC(=O)NCc1cnsc1)NC(=O)CC1CC(C)C1 11292,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CCC(=O)C1)=O 11293,C(C(C(C)C(C)C)NC(c1cnn(C)c1)=O)NC(c1c(CC(=O)OC)cnn1C)=O 11294,C=CC1OCCC1C(=O)NCCOC1CN(C(=O)CC(O)CN(C)C)C1 11295,C=CC(C)C(=O)NCC(CO)NC(=O)CC(C1CC1)NC(=O)NC(C)(C)C 11296,c1(NC(=O)NC(c2ccnn2C)C)cc(C(N)=O)c2n1CCOC2 11297,NS(=O)(=O)CC(=O)NCC1CN(C(=O)Cc2sccc2Cl)C1 11298,Cc1ccc(C(=O)NCCN(CC(C)O)C(c2coc(Br)c2)=O)o1 11299,c1(C(N2C(CNC(C(C)(C)n3cccn3)=O)CCC2)=O)cccc(Cl)c1N 11300,C1(CNC(c2ccc(C)nc2O)=O)COC(C)(C)CN1C(=O)Cc1coc(C)n1 11301,c1(OC)cc2[nH]ncc2cc1NC(C1CCN(C(c2cnccn2)=O)C1(C)C)=O 11302,c1(OCCC2CCCC2C(=O)OC(=O)OCC)ccc2c(c1)OCCO2 11303,Cc1cnccc1C(=O)NC1(C2CCCCN2C(c2nn(C(C)C)nc2C)=O)CC1 11304,c1(C(N2CC(O)(CNC(C3CC(O)C3)=O)C2)=O)ccc(-n2cncn2)nc1 11305,N1(C(C(C=C)O)=O)CC(C)(C)CC1CC(=O)N(C)CC1CCCC1 11306,C1(C(N2C(CNC(Cc3cccc(OC)n3)=O)C(C)CC2)=O)CC(=O)CC(=O)C1 11307,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)OCC=C)CC2C1 11308,c1(C(N2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)CC(C)C2)=O)cc2c(cn1)OCCO2 11309,c1(C(=O)NCC(CC)NC(=O)Cc2cnc(C)o2)nc(C)n(C)n1 11310,C(C#CC(F)(F)F)C(N1C(C2CCN(C(=O)CCF)C2)CCC1)=O 11311,c1(N2CCCC(CC)CC2)ccc(S(=O)(=O)NC2CC(C(N)=O)C2)cc1Cl 11312,c1(C(=O)NC(CN(C(c2c(C)sc(Cl)n2)=O)C)C)ccc2c(c1)C=CCC2 11313,c1(C(C(=O)NCC23CC(NC(CCCNC(C)=O)=O)(C2)C3)OC)cccc(C)c1 11314,Cn1c(C(N2CCOC(C3CN(C(=O)C(F)=CCCF)C3)C2)=O)cnc1O 11315,C(N=c1cc(C)nc[nH]1)C1CN(C(C(C)NC(COC)=O)=O)CC1(C)C 11316,C(CCO)(C(C)(C)O)NC(C(Cc1cc[nH]n1)NC(COCCSC)=O)=O 11317,c12ccc(c(F)c1)C(=O)N1C(CC(C)C1)C(=O)N2.c1(CO)cncc(O)c1 11318,C1(C(N(C(CC(=O)N2C(CC)COCC2)CC)C)=O)CC2COCC(C1)C2 11319,c1(C(=O)NCC(CO)NC(c2ccc(COC)cc2)=O)cccc([N+](=O)[O-])c1 11320,Cc1nnsc1.C(CN(C)C)(C(=O)N1CCC(c2cc[nH]n2)C1)N 11321,c1(CN=c2cc(NCc3ccc(Cl)o3)nc(COC)[nH]2)nc(O)c2ccccc2n1 11322,n1(CCNC(C(C2CCOCC2)C)=O)cc(C(c2ccccn2)O)nn1.C12CC1C2 11323,Cn1nccc1CCNC(N1CCC(c2nncs2)C1)=O 11324,N1(CN2CCC(c3n(C)c(=O)on3)C2)CCN2C(=O)COCC2C1 11325,C(N=c1cc(C)c(O)n[nH]1)C1(F)CCN(C(c2c(OC)cccc2OC)=O)CC1 11326,N1(C(CNC(C(CC)C)C#N)=O)C2CCC1C(NC(=O)C(F)(F)F)C2 11327,c1(C(NOCC(=O)N(C2CCN(C)CC2)C2CC2)=O)cccc2[nH]ncc12 11328,C12(C(N3CCCC(N(C(C4CCN(C)C4=O)=O)C)C3)=O)CCC(CC1)CO2 11329,C1(NC(C(C)SCCCC)=O)CN(C(c2cc(COC)on2)=O)CC1C 11330,Cc1cc(C)c(C(N2CC3CCC2C(NC(c2cccs2)=O)C3)=O)c(C)c1 11331,C1(NC(CCSCCC)=O)C(C)CCN(C(=O)C(c2ccn(C)n2)C)C1C 11332,N1(C(CC2(OC)CCCC2)=O)CCCC2CN(C(c3csnc3Cl)=O)CCC12 11333,Cc1ccc(C(=O)NCC=CCNC(=O)C(=Cc2c[nH]cn2)F)cc1F 11334,C(C(C)(C)C(=O)NCC1CCC(C(C)N)C1)NC(=O)C1CC1 11335,C(C(C)(COC)C(=O)N1CCC(NC(c2ccc(CO)nc2)=O)C(CO)C1)OC 11336,N1(C(C(C)C2CC2)=O)CCC(CO)CC1C(=O)NOCC(O)CO 11337,Cn1cnc(C(=O)NCCC2CCC(NC(=O)COC3CCOC3)C2)n1 11338,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11339,c1(C(N2CCCC(CC)(NC(=O)C3=CCCC3(C)C)C2)=O)ccc(Cl)c(C)c1N 11340,C(=O)(CCCSc1ccccc1)N(C)CC1CC1NC(c1cncn1C1CC1)=O 11341,S(=O)(=O)(c1cccc(F)c1C)N1CCC(O)(C(C)NC(C2(CC)CCC2)=O)C1 11342,C(CCCCCC(=O)N(c1csnc1C)C)NC(C(OC)OCC)=O 11343,C1(CC(=O)N(C2CCCN(C3CCOCC3)C2)CC2CC2)CCNC2(CC2)C1 11344,CN1CCCC1C(N1CCC(c2cc(C(C)(C)C)cs2)C1)=O 11345,c1(C2(C(N(C3CN(C(c4cn(C)cn4)=O)C3)C)=O)CCC2)ncccc1F 11346,C1(C(C)C(=O)N(CCC(=O)NC(C)C(=O)NC2CC2)CCO)CCC(=O)N1 11347,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11348,C#Cc1cccc(CC(=O)NC2CCN(C(=O)CC=C=C)C(C)C2)c1 11349,N1(C(C(CC)=CC)=O)CCN(C(=O)C=C(C)c2cccs2)CC(CO)C1 11350,C#Cc1ccc(NC=O)nc1.C(C)(C=C)(C1CC1)N 11351,c1(C(N2CC3CC3C2)=O)ccsc1SCc1cc(O)no1 11352,c1(C(CNC(c2ccc(C)n2C)(C)C)=O)cc(Cl)ccc1C 11353,C=C(C)C1OCCC1C(N1CCC2(CC2NC(C2CCCN2C=O)=O)C1)=O 11354,N1(C(c2cc(OC)no2)=O)CCC(C2CC2)(NC(C23CC(OC)C2C3)=O)C1 11355,c1(OC)ccccc1NC(=O)C(N1CCC(C)(CNC(C2CC(OC)C2)=O)C1)=O 11356,N1(C(c2ccccc2)C)CC2(CCCC2)c2cc(Br)ccc21 11357,c1(NCC2CC(=C)C2)ccc(S(=O)(=O)N2CC(CO)C3(CCOCC3)C2)c(Cl)c1 11358,C(=O)(C(CC)C(=O)OC(C)(C)C)NC(CNC(c1nccc(CC)c1)=O)C 11359,CC1=C(C(=O)NCC2CCC2NC(=O)CN2CCCC2=O)Cc2ccccc2O1 11360,C1(C)(NC(=O)C(=O)NC(C(C)(C2CC2)OC)C)CN(C(c2cnc(CN)o2)=O)C1 11361,N1(C(Cc2nc(C)[nH]n2)=O)CC2(NC(=O)CC(C)OC(C)(C)C)CC1C2 11362,c1(C2(N(CCc3cc(CO)ccn3)C(c3ccccc3)C)CC2)ccccc1F 11363,c1(CNC2CC(CC(=O)NCc3cccc(C(=O)OC)c3)C2)c(I)ccnc1Cl 11364,C1(C(N(C(C)C)C2CC2)=O)CN(C(=O)C(O)CN(C)C)CCC1(C)C 11365,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11366,C12(C(=O)NCC(CC(=O)OC)C)CCC(CN(C(=O)CCCNC(C)=O)C1)C2 11367,N1(C(CSCC(C)=O)=O)CCOC(CNC(=O)C(C)(C)c2csc(C)c2)C1 11368,n1(CC=C)cc(C(=O)NCCN(C(c2cn(CC)nn2)=O)CC)nn1 11369,CCC(C(C)(C)C(=O)OC)OC(c1c([N+](=O)[O-])cnn1C)=O 11370,c1(SCC(=O)NCC(Cn2cc(-c3cnn(C)c3)nn2)OC)ccc(CO)cc1 11371,CCC(C)CC(C(=O)Nc1cc(CO)ccc1C)NC(c1coc(C)n1)=O 11372,N1(C(C2(C(=O)OC)CC(=C)C2)=O)CCC(C)CC1.c1(C(=O)NC(C)(C)C)cnccn1 11373,N1(C(C2CC2F)=O)CCCC2(C1)CN(C(c1ccnc(OCC3CC3)c1)=O)C2 11374,C(C)(C)(CCCC(=O)N1CC(CC(C)C)C1)NC(c1cc(COC)on1)=O 11375,CCC(C(F)(F)F)CC(=O)NC1(CC2CC2)CC1 11376,N#CC1CCCCC(C(=O)NCCN(CCOCCO)C(c2ccc[nH]2)=O)C1 11377,c1(OC)ccc2ccc(C(=O)NC3NCCC3(C)C)nc2c1Br 11378,CC1CN(C(c2cc(Cl)ccn2)=O)CCCN1C(=O)CCCN1CCCCC1 11379,C1(CN(C(=O)C=CCNC(C2(C#N)CC2)=O)C)CCC(F)C1 11380,C(=O)(C(C)(CC)C(=O)NCC1CCN1C(c1c(SC)cccc1F)=O)OCC 11381,C1(C2(O)CCC2)(C(=O)NCC(c2ccccc2)NC(c2ccc(C#C)o2)=O)CC1 11382,Cc1cc(C(=O)NC2CCCC(NC(c3ccsn3)=O)C2)ncc1S(N)(=O)=O 11383,C1(C(=O)OC)CC(C)CN1C(c1c(Br)cnn1C)C(=O)NC(c1ccccc1)C 11384,N1(C(c2ccc(N(C)C)nn2)=O)CCN(C(c2ccc(N)cc2Cl)=O)CC(O)C1 11385,CC1(C)CCc2c1n[nH]c2C(=O)NC1CCSC12CN(C(=O)C1CC1)C2 11386,N1(C(Cn2cc(C(N(C)C)=O)nn2)=O)C2CCCC1CC(NC(=O)CCCF)C2 11387,N12CC3CCC1C(C3)CNc1ccc(cn1)C(=O)C2=O.CC1CCC(C(=O)OC)C1 11388,c1(C(=O)NCC(C)(C)NC(CCC#CC)=O)cc2c(C)sc(C)c2s1 11389,Cc1nc(C(F)(F)F)c(C(=O)NC2CC(NC(=O)C(C)(C)C(C)C)C23CCC3)n1O 11390,N1(C(C(CO)NC(N)=O)=O)CCC(F)(C(=O)NCc2ccccc2F)C1 11391,N1(C(C(CC2(n3cc(SC)nn3)CC2)Cc2ccccc2)=O)CCCCCC1C 11392,C1(NC(c2csc(C(F)F)c2)=O)CC(NC(c2ccc[nH]2)=O)C12CCC2 11393,c1(CC)cc(C(=O)NCCCC(=O)NCCC2CCC(=O)N2)c(C)o1 11394,CCC(CC)(CCO)N(C(=O)CN1CCN(S(C)(=O)=O)CC1)CC 11395,N1(C(c2cc(CC)no2)=O)CCC(C(=O)NC(C)C(C)C(=O)OC)=C(F)C1 11396,c1(-c2ccc(CN3C(=O)CNCC3)cc2)cc(Br)c2[nH]c(=N)sc2c1 11397,N1(C(C(C(C)C)OCC)=O)CCC(O)(CNC(=O)CCOCC(F)F)CC1 11398,C1(C(=O)NCC2(NC(CCN(C)CCO)=O)CCC2)CC(=O)N(O)C1 11399,C1(C(C)CNC(=O)NC(CCC)CO)(CO)CCOCC1 11400,C(=O)(C1Cc2ccccc21)NCC1N(C(CC=C=C)=O)CC1 11401,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11402,N1(C(C2N(C(CCC3CC(C)C3)=O)C3(CC2)CC3)=O)CCC2CN(C)CC12 11403,C1(OC)CN(C(=O)C=CC2CCCC2)CC1NC(C1CCN1S(C)(=O)=O)=O 11404,c1(Cc2ccsc2)cccnc1.C1(=O)CCCC2(CC2)C(=O)NC2CC(C2)N1C 11405,c1(C(N2C3(CNC(C=CCC)=O)CCC2CC3)=O)ccc(Br)c(F)c1C 11406,C#Cc1ccc(CN(C(=O)C(=O)NC2(NC(=O)CC(CC)CC)CC2)C)cc1 11407,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11408,C#Cc1ccc(C2CC2C(N2CCN(C(=O)C(C)CC(C)C)C(CF)C2)=O)cc1 11409,n1(CC2C(C)C2)nc(-c2ccc(Cl)cc2)nc1C1CC(C(F)F)C1 11410,C(=O)(C(F)C(C)(C)O)N(CCNC(=O)CSCCC#N)CC 11411,C12(C(N(C(C3CCCC3)C)C)=O)CC(CO)(CN1C(c1sccc1C#N)=O)C2 11412,c1(C(=O)OC)sc(C(N2CC=CC(NC(=O)CC3(OC)CCCC3)C2)=O)cc1N 11413,Cc1cc(Br)cc(C)c1NNC(=O)NC1CCCCCC2CC12 11414,c1(NC(C(C2CCCN(C(CCCOCCC)=O)C2)C)=O)cncc(C)c1O 11415,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11416,N1(C(CC(C)C)=O)CCC(NC(=O)CCNC(=O)C(C)(C)C)C(F)C1 11417,C1(C(N(CCOC)CCNC(c2coc(C3CC3)n2)=O)=O)CC2OC(=O)OC2C1 11418,C1(CCNC(=O)NC(Cc2ccc(Cl)nc2)CO)CCC2(CC1)OCCO2 11419,c1(CC)cc(C(=O)N(CCCNC(=O)CC2CCC(C)C2)C)no1 11420,S1(=O)(=O)c2ccc(cc2Br)CN1.CC(CN(C)N1CCC=CC1)N1CCCC1 11421,C1(C(=O)N(C)Cc2ccns2)(NC(C2N(C)CCC2)=O)CCCC1 11422,C12CCCC(C1)NC2=O.C(=O)(CS(N)(=O)=O)N(CC(C)(C)NC(CC)=O)C 11423,c1(C(N(CCC(=O)NCc2nc(C)c(C)o2)CC)=O)cccc(F)c1C 11424,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11425,c1(C(=O)NC2COCCN(C(c3cc(Br)ncc3Cl)=O)C2)cc(O)c(Br)c(O)c1 11426,CCCCC(CNC(c1n[nH]c(C)c1F)=O)NC(=O)Cc1cncc(Br)c1 11427,c1(C(N2C(CNC(CCC=C)=O)CN(C)CC2)=O)c(F)cc(OC(C)C)cc1F 11428,C1(N2CCN(CC(=O)OC)CC2)COC2(CCN(C(=O)CNC(=O)C(=O)O)CC2)C1 11429,N1(C(C2(C(C)C)CC(=C)C2)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11430,C1(N=[N+]=[N-])(C(=O)NCCC(C)(C)SC)CCN(C(c2oc(C)nc2C)=O)C1 11431,C1(NC(CC(CNC(c2ccnn2CCF)=O)O)=O)CCCCCCC1O 11432,N1(C(C2(CNC(=O)CCc3ccncc3)CC(=C)C2)=O)CCCC(N=[N+]=[N-])CC1 11433,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOC2(C)C)C(C)(C)C)CCO1 11434,Cc1ncc(C(N2CC(CNC(=O)C(C)(C)n3cc(Cl)cn3)CC2C)=O)cc1Cl 11435,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(=O)CCCF 11436,CCCC(CCC)C(C)NC(c1ccc(F)cc1Cl)C 11437,N1(C(CC=C)=O)CCCC(O)(CCNC(c2cc(CN(C)CC)c[nH]2)=O)C1 11438,c12occc1CNC2=O.C(CCCF)N(C(=O)C=CC(C)(C)SC)C 11439,C1(C)(C(=O)NC2C(C(=O)NCCCCOCC)CCOC2)CCC(=O)CC1 11440,N1(NCCCC(O)CO)CC(C(c2c(CNC(C(=O)OC)=O)ccs2)=O)CC1=O 11441,CC1CN(C(C23CC(CO)(C2)C3)=O)CC1NC(C1CCC(N2CCCC2=O)CC1)=O 11442,C(=O)(CC1=CCOCC1)NC1(CO)CCN(C(C(C)Cc2cccnc2)=O)C1 11443,C(C)(CCCCNC(c1ccnn1C)=O)NC(CN(C)C(C1CCCC1(F)F)=O)=O 11444,N1(C(C2(CC)COC2)=O)CC(Nc2ncc(C(=O)OC)cc2C)CC(F)C1 11445,CN1CCN(C(=O)C=CCCC=C(C)C)CC1CNC(=O)CSc1nnc(S)s1 11446,N1(C(c2cc(COC)on2)=O)CCCC(F)(C(=O)NCC(C)(C)OCCO)C1 11447,CC(C(C)(C)NC(c1ccnn1CCF)=O)NC(c1cnn(C(F)(F)F)c1)=O 11448,C(CC1=CCN(C(=O)C#CC2CC2)CC1)NC(C(N1CCCCCC1)C)=O 11449,C1(CNC(CC2CCC(=O)NC2)=O)(NC(c2csnn2)=O)CC2CCC1CC2 11450,c1(C(N(C2CN(C(CN3C(=O)C(C)C(C)C3=O)=O)C2)C)=O)c[nH]c2cnccc12 11451,N1(C(C=CC=CC)=O)CC2CC2(NC(=O)Cc2cc[nH]n2)C1 11452,C1(CNC(c2nc(CC)[nH]n2)=O)CCC(CNC(=O)CC2CCC2(C)C)CC1 11453,C12(C(N3CC(NC(C)=O)C(O)C3)=O)CCCC(C)(C1)OC2 11454,C1(O)(NC(C2CCN(c3nccc(C(=O)OCC)n3)C2)=O)CCCC(C)(C)CC1 11455,O(NC(=O)C(F)(F)c1cncc(Nc2ccsc2)c1)C(=O)OC(C)(C)C 11456,Cc1cncn1CC(=O)NCC(C1CCCCC1)NC(c1csnn1)=O 11457,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(=O)C(C(C)C)NC(C)C)C1CC 11458,c1(C(=O)NCC(C)(CC)NC(C(C=C)CC)=O)cnc2ncnn2c1O 11459,Cc1ccc2ccccc2c1NCC1CC(O)(CO)C1 11460,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(C)CC2(C)C)=O)CC1c1ccnn1C 11461,c1(OC)cccc(C(=O)NC2CC(CNC(=O)CC3CCSCC3)C2)c1F 11462,c1(C(=O)Nc2cc(C#N)nc(C)n2)n[nH]c2cc(-c3cc4sccc4s3)ccc12 11463,Cc1ccnc(C)c1CNC(c1coc(CNC(C2CCC(C)C2)=O)c1)=O 11464,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11465,c1(C(=O)NCCC23CCCC2C3)cccc(N2CCCCC2)n1 11466,N1(C(C2CC2[N+](=O)[O-])=O)CCC(CN2CCCCC2)CC1.c12c[nH]nc1CONC2=O 11467,c1(C(=O)NCC(CCCC)NC(=O)C(F)C2CCC2)cnc2c(C)cccc2c1 11468,N1(C(C(c2nc(C)[nH]n2)NC(c2cccn2C)=O)=O)CCC2CCCC12CO 11469,N1(C(c2cc[nH]c(=N)c2Cl)=O)C2CCC1c1ccccc12 11470,C1(F)(C(N(CCO)CC)=O)CCN(C(=O)C(C2(O)CCCC2)F)C1 11471,C(=O)(NN(C)C(=O)N(C)C)Nc1ccc(Cl)cc1.c12nc(cs1)NC(=O)C2C 11472,C1(NC(c2nnn(C)c2N)=O)CC2(C1)CC(NC(c1cc(Cl)c(Cl)n1C)=O)C2 11473,N1(C(Cc2cc(C)c(O)c(C)c2)=O)CC2(C)CN(C)CC2(C)C1 11474,C1(CNC(CSC)=O)(NC(c2cnc(C(F)F)cn2)=O)CC(F)(F)C1 11475,C1(NC(c2cccc(OC(F)F)c2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11476,C1(C(=O)NCCOCCC(=O)OC)COCCC1NC(=O)Cc1ccccc1C 11477,N1CCC2CCCC12.c1(CC(=O)NCC)ccc(CNC(=O)C=NOC)cc1 11478,C#Cc1cc(F)c(C(=O)NC(CNC(C2CC2C)=O)C(C)(C)C)cc1F 11479,C(=O)(C1CCCc2ncccc21)OCCCCCOC 11480,Cc1cncc(CC(N2CC=CC2C(=O)NC2C(C)CCC2C)=O)c1 11481,C(C(C(=O)NC(C)Cn1ccnc1)NC(=O)C(N1CCCC1C)C)OCC 11482,C(CCCS(C)(=O)=O)NC(c1cc(C#N)cn1C)c1n(CCCOC)nnn1 11483,C1(NC(CCCC(=C)C)=O)(CNC(=O)C(C)P(C)(C)=O)CC2CCC1CC2 11484,c1(OC)cc(C(C(=O)NCCC2(C)CC2)N(CC(C)(F)F)C)c(F)cn1 11485,N1(CC)CCCC(NC(=O)CC(C)OC(c2nnc(CC)o2)C)C1C 11486,C(C)(C(CC(=O)NCC1CC(SC)C1)NC(=O)C(C)c1cc[nH]n1)OC 11487,C12(CNC(C3C(CCC)C3)=O)CCCC1N(C(c1nonc1CC)=O)CC2 11488,c1(NCC(c2cccc(F)c2)OCC)nc(Cl)c(C#N)n1C 11489,CC1(C2(C)CC2C(N2CCCC(n3cc(CCS(N)(=O)=O)nn3)C2)=O)CC1 11490,C12(C(=O)O)CC(c3ccccc3C(N3CC4CC3C4)=O)(C1)C2F 11491,CC(C(=O)NCc1cnn(C2CCNCC2)c1)(C(F)(F)F)c1ccccc1 11492,c1(C(N2C(C(C)NC(c3cnc[nH]3)=O)CCCC2)=O)cc2ccc(Cl)cc2c(=O)o1 11493,C1(CNC(C(C)NC2CCCCC2)=O)CC2(CCC2)CN1C(=O)C1=COCCC1 11494,C(=O)(CCCCCNC(=O)CCCN(C)C)N1C(CC(=O)OC)CCC1 11495,c1(NCC(c2n(C)ncc2)O)[nH]c(=NCC(Cl)(Cl)Cl)nc2c1cnn2C 11496,Cc1nn(C)c(CNC(=O)NCC2(Cc3cccc(F)c3)CC2)c1Cl 11497,N1(C(C(COCC)NC(=O)C(C)(C)OCc2ccccc2)=O)CCC(CO)CC1 11498,c1(OC)cnc(C(=O)NCCCC(C)NC(C2CN(C)CCO2)=O)c(OC)c1 11499,c1(C(N2CC(NC(COCCCC#C)=O)C(CCOC)C2)=O)cc(=O)cc(Cl)[nH]1 11500,c1(NC(n2cccn2)C)nccc(N2CCCC(C)C2)n1.n1(C)ccnc1 11501,CC(C)CC(C(=O)N(c1ccccc1)CCCN(C)C)ONC(=O)CC1CCOC1 11502,c1(C(=O)OCC)c(C(=O)NCC2CCC(NC(=O)CCF)C2)cnn1C1CCCC1 11503,N1(C(COCCC#C)=O)CCC2CN(C(c3cnc(C)nc3CC)=O)CCC2C1 11504,Cn1nc(Cl)cc1C(=O)NCC1CCCN(C(=O)CC2(n3cccn3)CC2)C1 11505,C1(C)(C(=O)OC)CCCN(N2CCCC(O)CC2)C1 11506,c1(C(=O)NCCC(C)(C)NC(C2CCCC(=O)N2)=O)c[nH]cc(Cl)c1=O 11507,Cc1ccc(C(C)C(=O)N(CCn2cc(-c3ccc(C)o3)nn2)C2CC2)cc1 11508,CC1(C)CC(=O)OC1C1CN(C(C2C=CCCN2C(C2OC3CCC2C3)=O)=O)C1 11509,C(CC(O)CCO)NCC1CC(CCC(=O)NC(=O)CCCn2cccc2)C1 11510,C1(=O)C(CCCOC)N1.C(=O)(CC(CN(C)C)CC)N(C)Cc1ccn(CC)n1 11511,C1(C(=O)NC2C(CO)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11512,CCC1C(=O)NC2(CCCC2)C(=O)N1C.c1(C)cnco1.OC 11513,Cc1[nH]c(C(=O)NCC2CCCO2)c(C)c1C(=O)NC(c1ccc(F)cc1F)C 11514,N1(C(CC2CC(C)C2)=O)CC(C)(C)OCC1NC(c1sccc1NC(=O)C1CC1)=O 11515,N1(C(C2C(CC)C2)=O)CCC2CN(C=O)CC2C1.C1(C2CCCO2)CCC1 11516,c1(CC)ncc(C(=O)NC2CC(CNC(c3cccc(C)n3)=O)C(O)C2)c(O)n1 11517,N1(C(CC2(C=C)CN(C(C3CCC(C)=C(C)C3)=O)C2)=O)CCCC2CCCCC12 11518,N1(S(c2ccc(NC(C)C)cc2)(=O)=O)CCC2(C1)NC(=O)N(C)C2=O 11519,c1(C(CC)(C)C)ccc(C(=O)N(C2CCN(C(=O)COC3CCOC3)C2)C)cc1 11520,C1(CC(=O)NCC(N(C(c2c(CC)oc(C)c2)=O)C)C2CC2)CCCNC(=O)C1 11521,Nc1cc(Cl)nc(Cl)c1C(N1CC2(COC(CNC(=O)Cc3cnoc3)C2)C1)=O 11522,Cc1ccc(C=CC(=O)NCC2(O)CN(C(C3(Br)CC3(C)C)=O)C2)cc1Cl 11523,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 11524,C(=O)(C1CCc2ccccc21)N1CC(F)CC(CNC(c2ccc(O)cc2)=O)C1 11525,C(=O)(CCCCc1cnc[nH]1)NCC1C(NC(C(CC)O)=O)C1 11526,c1(C(c2nnnn2C)SNC2(CCC)CC2)cc(Cl)nc(Cl)c1 11527,C1(Nc2ncnc(N3CCC(SC)CC3)c2C)CCc2nncn2C1 11528,C1(CNC(CCCC)=O)(OC(C)CCC(=O)OC)CCN(C(C)=O)C1 11529,C1(C(=O)OCC)CCc2nc(C(N3CCCC3C(=O)NCC)=O)sc2C1 11530,N1(C(c2cnc(CC)o2)=O)CCC2CC12C(=O)NCC(CC)CC 11531,CCC(CC)C(=O)N(CC(C)NC(c1cnn(C(C)(C)C)c1C(F)F)=O)C 11532,C(=O)(C1=C(Cl)CCCC1)NC(C)C(N1CC(S(C)=O)C1)=O 11533,c1(C(N(CCNC(c2c[nH]c(=NC)s2)=O)CC)=O)cccc(S(=O)(=O)C(F)F)c1 11534,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11535,O=C(CCC=CBr)NC1(c2ccccc2)CCN(C(C2CC=CCC2)=O)C1 11536,c1(NC(C2C(NC(CCSC(c3nncn3C)C)=O)CC2)=O)ccc(F)cc1 11537,C(CCCCCCC(=O)NCC1(c2nn[nH]n2)CCC1)N(C)C 11538,C=CC1CN(c2cc(N3CCC(CC(=O)NC)CC3)ncn2)CCC1CC 11539,c1(C(=O)NCCC2(NC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11540,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11541,N#CC1(C(N2CCCCCC2C(=O)NC2CCC(C(N)=O)C2)=O)CCOCC1 11542,CC1(C)CN(C(c2ccc(C3CC3)o2)=O)CC(CNC(C2(C)CC2(F)Cl)=O)O1 11543,C(CN(C)N1CCC(C(=O)OC(C)(C)C)CC1)N(C)C(c1ccco1)=O 11544,c1(CN2CCC(C)(C(N3CCC(c4ccncc4)C3)=O)C2)ccc(Br)cc1S(C)(=O)=O 11545,N1(C(c2c(CCC)occ2)=O)C2CCC1CN(C(C1CC3CC3C1)=O)CC2 11546,c1(C(=O)NCC(C)CN(C(=O)CN(C)CCO)C)ccc(Cl)cc1Cl 11547,c1(CSCC(=O)N(C(C)CNC(C2CCO2)=O)C)ccc(Cl)s1 11548,O=C1Nc2ccccc2CC1CC(N1CC2CCCC2C12CC2)=O 11549,C(=O)(C(F)C1=CCCCC1)N1CC(C)N(C(=O)C=Cc2cncnc2O)CCC1 11550,CC(CC(=O)N1C2CCC1(CNC(c1cc(C(C)(C)C)on1)=O)CC2)C(C)(C)C 11551,C(=O)(CCCCCNC(=O)C(C)(C)C(=O)OC)NC1C(COC)CCCC1 11552,c1(C(=O)NCC2CN(C(c3n(CC)ccc3)=O)C2)cc(Cl)ccc1OC(F)(F)F 11553,C(=O)(CC1=CCOCC1)NCc1c(CNC(c2ncc(OC)cn2)=O)cccc1 11554,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11555,c1(C(=O)NC23CCN(C(c4c(OC)n[nH]c4)=O)CC2C3)cnc2cc(C)nn2c1 11556,c1(C(N(CC(C)NC(C2CC23CCOCC3)=O)C)=O)cnc(O)c2c1NCCC2 11557,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11558,CCC(O)C(F)(F)C(=O)NCCN(c1ncnc2[nH]ccc12)C1CC1 11559,C(=O)(C1CCc2c(Cl)cccc21)NCC1CC(NC(c2cc(C#N)sc2)=O)C1 11560,c1(C(=O)NCC2(CNC(Cc3c(C)cc(C)s3)=O)CC2)cc2[nH]nc(C)c2cn1 11561,CCC(C(=O)NC1(C(=O)NON2CCC(C)C3(CCC3)C2)CCCC1)C(C)(C)CC 11562,c1(NC(C2C(C=C)C2)=O)cccc(F)c1SCC1CCCN1C(=O)CCCCC 11563,N1(CCN2C(=O)COCC2)CCC(C2CCC3(CC2)OCCO3)CC1 11564,C1(C(=O)NC(C(=O)OCC)CC2CC2)CCC(C)N1C(=O)C(C)OC1CCOC1 11565,C=C1CCC(C(=O)NCC23CC(NC(c4cnn(C(C)C)c4C)=O)(C2)C3)CC1 11566,N1(C(c2cccc(-n3cc(CC(C)O)nn3)c2)=O)CCC2(CCCN(C)C2=O)C1 11567,C(=O)(CC(C)C(F)(F)F)N1CCC(NC(C(COC)(C)C)=O)C(O)C1 11568,c1(C(=O)NC2CN(C(C(C)C)=O)CC2C)cc2ccoc2cc1F 11569,C(N=c1cc[nH]c(=NCCCc2cccc3ccccc23)[nH]1)c1c(=N)[nH]cnc1 11570,c1(OC)cc(C)cc(C(=O)N(C)CC2(NC(C3CC34CCSCC4)=O)CC2)c1C 11571,C(=O)(C1=C(Cl)CCCC1)NCC(C)CC(=O)N(C)CC1CCOCC1 11572,Cc1nc(C)c(C(=O)NC2CN(C(c3ccnc(Cl)c3)=O)C2)[nH]1 11573,C1(NC(=O)CC2CCOCC2)CCOC(CNC(c2ccc(CC3CC3)s2)=O)C1 11574,C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(c1cncs1)=O 11575,N1(C(CC2CC(C)(C)OC2)=O)CC2(CCN(C(c3cc(S(N)(=O)=O)c[nH]3)=O)C2)C1 11576,N1(C(C2CCN(C(c3ccc(C=C)cc3)=O)C2(C)C)=O)C2CCC1CC(=O)NC2 11577,N1(Cc2cnc(C)nc2)CCN(C(c2cccc(=O)o2)=O)CC1C 11578,Cc1nn(CC(=O)NC2CN(C(C3CCCS3)=O)C2)cc1OC(C)(C)C 11579,CCC(C)(C(=O)N1CCC(CCNC=O)C1)OC.C1(=O)C(CCOCCO)N1 11580,N(C1CCNc2ccccc21)C(=O)CC1CCc2ccccc2C1 11581,c1(CC(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)cccc(Cl)c1F 11582,Cc1ccc(=N)[nH]c1C(=O)NCC(CO)NC(=O)CCn1cncn1 11583,C(CC(=O)NCC(=O)OC(C)C)(CC(C)C)NC(C1ON=C(CC)C1)=O 11584,C(=O)(CC(F)(F)C(C)C)N(CC(C)N(C(C(COCC)C)=O)C)C 11585,CP(C)(=O)c1cncc(C(N2CCCN(C(C3C4COCC34)=O)C(CO)C2)=O)c1 11586,c1(C(=O)NCCCN(C(=O)CC2(COC)CCCC2)CC)ccc(C)n(C)c1=O 11587,C(CCN=C(NCc1ccc(C(F)(F)F)c(C)c1)N1CCC(C(F)F)C1)OC 11588,C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(NC(c2cccc(C)n2)=O)CC1 11589,CC(C)C(C(=O)N(CC(O)CN(C(=O)C(O)Cc1ccccc1)C)C)NC(N)=O 11590,C1(C(=O)NCC=CCNC(c2cc(O)nc(O)n2)=O)CCc2nnc(O)n2C1 11591,c1(C(C(C)NC(=O)N(n2cnnc2)C)O)ccc(Br)cc1 11592,C1(C(N2CCCC(COC)C2)=O)CC2(CC(NC(=O)Cc3ccc(F)cc3)C2)C1 11593,N1(C(C(c2ccc(C)cc2)C)=O)CC2CC(NC(c3cnc(O)s3)=O)CC(C2)C1 11594,c1(NC(=O)OCC)cccc(NC(c2cc(Br)ncc2F)=O)c1C 11595,c1(C(=O)NC2CN(C(C3(C)CCOC3)=O)CC2F)ccc(F)c(O)c1 11596,N1(CCNC(C(COC(C)C)(C)C)=O)CCCN(C(C2COCCN2C)=O)CC1 11597,c1(NC2CC2)ccc(OC(c2ccc(C(CC)=O)cc2)(C)CO)c(F)c1 11598,C1(C(C(=O)C=C2CCN(C(C3(C(=O)N)CCC3)=O)C2)NC2CC2)CC12CCOCC2 11599,c1(C(N(c2nnc(Cc3ccccc3)n2CC)CC)=O)ncc(F)cn1 11600,N#Cc1ccc(F)c(CNC(=NCCCF)NCc2cnccn2)c1 11601,CCC(C(=O)NC1(CO)CN(C(C2CC2c2ccncc2)=O)C1)C(C)O 11602,c1(OC)ccc2c(c1C(=O)NC1CN(C(=O)CCS(C)=O)CC(F)(F)C1)CCC2 11603,C(=O)(C(O)CCCNC(C1(F)CCC1)=O)N1CC(OC)(CO)C1 11604,C(C(C(=O)N1CC(N2CCCC2)C1)OCCF)OC(C)C 11605,C1(CC(=O)N(C2CC(=O)NC2)CCO)COCCN1Cc1cccc(OC(F)F)c1 11606,C(CC(C)P(C)(C)=O)N(C(C(n1cc(-c2ccc(C)nc2)nn1)C)=O)C(C)C 11607,C=CCC(C(=C)C)C(=O)N1CC(NC(c2cc(C)nc(C)c2)=O)C(O)C1 11608,C(C(C)CC(=O)N1CCCC1CNC(=O)C(c1ccccc1)N(C)C)NC(C)=O 11609,C#CCC(C)(C(=O)NC1CCCCC1C(N)=O)NC(=O)CCOC1COC1 11610,c1(C(=O)NC(C(C)NC(c2cc(CCC)[nH]n2)=O)C)c[nH]c2cc(F)ccc12 11611,C(=O)(CCCCC)N(C(C)C(=O)NCC1CC1C(C)C)CC 11612,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCc2noc(C(C)C)n2)CCC1(C)C 11613,C=CCCC(CO)NC(=O)CCCNC(=O)CN 11614,c1(CC)ccc(C(=O)NC2(C(=O)NC(CO)CCOC)CCN(C)C2)cc1 11615,c1(C(=O)NCC(CCCC)NC(C2(C(F)F)CCCO2)=O)nsc2ccccc12 11616,Cc1ccccc1C(C)CC(=O)NCC1(C)CCCN1C(=O)C(N)=O 11617,C1(O)(C(N(CC(C)NC(CC2CC(=C)C2)=O)CC)=O)CCCC(C)(C)CC1 11618,N1(C(c2c(CC)noc2)=O)CC2(CCCC2NC(=O)C(c2ccccc2)C)C1 11619,CCCC(O)(CNC(=S)Nc1cccc(F)n1)c1ccccc1 11620,c1(C(N2CCN(C(C(CC)SC)=O)CC2CF)=O)coc2c(F)cccc12 11621,C=CCCC(C(=O)NC1(C)CC2CCC1C2)NC(=O)C(F)C1CCC1 11622,Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3ccn(C4CC4)n3)=O)C2C1)=O 11623,Cc1cc(F)ccc1CNC1(C)CCOC1C 11624,CN=c1nc(N2CCC(C(=O)N(C)C)C2)[nH]c(=NCCN2CCC3(CC2)CC3)[nH]1 11625,N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC1)CCN(Cc1cc(Cl)ncc1Cl)C2 11626,C1(C(C)C)C(=O)N1.c1(C(N(CCOCC)CC)=O)cccc(C(O)C(F)(F)F)c1 11627,N1(C(CN(CCOC)C)=O)CC(CN(C)C(C2(OCC)CCC2)=O)C(O)C1 11628,C=CCC(CNC(c1cnc[nH]1)=O)NC(=O)CC1COCC1O 11629,N1(C(c2ccc(C)cc2C)=O)CC2CC(C)N(C(=O)C(F)CC3CCOC3)C2C1 11630,C1(C(N2C(CC(=O)NCCC(C)OC)CCCC2)=O)CC(C)(C)CN1C 11631,C1(C(N2CCN(C3CCC(NC(CSC)=O)CC3)CC2)=O)Cc2nncn2C1 11632,C1(C(=O)NC(C)CC2CCCCC2)CCN(C(=O)CCC2CC2(C)C)C1 11633,Cc1ccc(OCCC(=O)NCCCCN(C)C(C2CCCS2(=O)=O)=O)cc1C 11634,CN1CCOC2CN(C(C3CC(C)(NC(=O)CC4CCCOCC4)C3)=O)CC12 11635,c1(C(=O)NC(CNC(C(CC)n2cncn2)=O)(C)C2CC2)cccnc1C 11636,CCC(C(F)(F)F)S(=O)(=O)C(C1COCCN1Cc1ccc(F)cc1)=O 11637,CC(CC(=O)NC1(CF)CCN(C(=O)C=CS(C)(=O)=O)C1)C(F)(F)F 11638,c1(C(C)F)ccc(C(=O)NCCC(C)NC(C2CC2(c2ccccc2)C)=O)cc1 11639,C1(F)(CNC(C2C=CCC2)=O)CCCN(C(c2cc(F)n[nH]2)=O)C1 11640,c1(CC)nn(C)c(C(=O)NC2(CC)CCCN(C(c3cnc(O)n3C)=O)C2)c1Cl 11641,C(=O)(C1CNC(=O)c2ccnn21)N(C1CCN(c2ncns2)C1)C 11642,N1(C(C(C(C)(C)C)C2CCC2)=O)CCCC(NC(=O)CC(F)(F)F)CCC1 11643,N1(CC(=O)Nc2cccc(CC(N)=O)c2)CCC2(CCc3cccnc32)C1 11644,CCS(=O)c1ccccc1CC(=O)NCCOC(C)C 11645,C1(C2N(C(Cc3c(C)cc[nH]3)=O)CCC2)CCN(C(C2CC(F)(CO)C2)=O)CC1 11646,C1(COC)(CNC(C2CC23CC3)=O)CN(C=O)C1.c1(CC(C)N)ccccc1 11647,c1(OC)ccccc1C1C(C(c2c(C(=O)Oc3ccccc3)cnn2C)OC)C1 11648,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11649,N1(C(C2CCN(C(CC3C(OCC)CCCC3)=O)O2)=O)CCCC2OCCC2C1 11650,c1(CC(=O)NCc2scc(CNC(CC(C(C)O)C)=O)n2)ccc2[nH]ccc2c1 11651,N1(C(CCC=C=C)=O)CCOC2CN(C(c3ccc(O)cn3)=O)CC12 11652,c1(SC)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2C)=O)cnn1C 11653,c1(CC(=O)NCC(N(C)C(c2ccc(C(N)=O)s2)=O)C2CC2)ccc(O)nc1 11654,CC1CC(O)CCN(C(=O)NCc2ccccc2CN2CCCCC2)C1 11655,C12(C(=O)NCC3CN(C(C4C(C(=O)OC)C4)=O)CC3O)C3CCC(CC13)C2(F)F 11656,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(=O)N)C2C.c1(C2C(CC)C2)ccccc1 11657,C1(C(N(CC(C)(C)Nc2cc(=O)n(C)cn2)C)=O)CC2(C1)CC1(CC1)C2 11658,C1(C(N(C2(C(=O)NCc3nc(CC)on3)CC2)C)=O)CCC(C2CC2)C1 11659,c1(NC(c2n(CCC)nnn2)(C23CCCC2C3)C)ccc(OCCO)cc1 11660,CC1(C)CC(NC(c2cccnc2O)=O)CN1C(=O)CSc1ccncc1 11661,C(=O)(C(C)CC(C)(F)F)NCCC1(NC(C(C)OCCC(C)C)=O)CCC1 11662,CC1CCOC1CC(=O)N(C)CC1CN(C(c2sccc2CO)=O)C1 11663,c1(C(=O)NC23CCC(NC(c4nc(CC)oc4)=O)(CC2)C3)ccc2sccc2c1 11664,C(=O)(CCCCCO)NCC1C2CN(C(c3n(C)cnc3)=O)C1C2 11665,c1(C(N(C2CCN(C(c3cccnc3O)=O)C2)C)=O)ccc2nn[nH]c2c1O 11666,C1(C(=O)Nc2c(C(=O)OC)scc2)CCCC(NC(=O)NC(C)(C)C)C1 11667,c1(C(=O)OC)cc(COC(=O)CC(O)CN(C)C)c(F)cc1F 11668,c1(C(=O)NCC=C2CCN(C(C3CN(CC)C(=O)C3)=O)C2)ccc(N)c(Cl)c1O 11669,C(CS(=O)(=O)CC(=O)N1CCC(C)N(C(c2n[nH]c(C)c2C)=O)CC1)OC 11670,c1(CNC(COC(C)(C)C)=O)cc(NC(=O)C(=O)CCCOC2CC2)co1 11671,C1(C2CCC2)(C(N(CC(O)CNC(c2ccn(C3CCC3)n2)=O)C)=O)CCC1 11672,C(=O)(CCCCN(C)C)NC(C)C(CO)NC(c1cnc(C(F)(F)F)s1)=O 11673,N1(C(C(CC)c2ccccc2)=O)CC2C(CNC(=O)CSc3ccc(F)cc3)C2C1 11674,N1(C(CCCC)=O)CCCCC1C(=O)NC1(CNC(=O)C(C)SC)CCOCC1 11675,C(=O)(C(C(C)C)N(c1c(C)ocn1)C)OCCc1ccccc1 11676,C=C=CC(C)C(=O)N1CCC(C)(NC(=O)C=CC(N2CCOCC2)=O)C1 11677,c1(C(N2C(CNC(C(CCN(C)C)O)=O)CCC2)=O)c[nH]c2cccnc2c1=O 11678,N1(C(C(CCCC)F)=O)CCc2c(ncn2-c2cn[nH]c2)C1.c1(N)cccc(O)c1 11679,Cc1ccc2cc(C(=O)NC(C)Cc3cc(Br)ccc3F)cnc2c1 11680,CC(C)(C)COC(CNC(=O)CC1CC=CC1)C1CC1.C12(CC1)CC(=O)OC2=O 11681,C(=O)(CCCCC(=O)NCCC(O)CNC(c1cncn1-c1cnn(C)c1)=O)NC 11682,N1(C(CCOCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11683,c1(C(=O)NCC2CC(C(N(C3CC(O)C3(C)C)C)=O)C2)nc(=N)cc[nH]1 11684,N1(C(c2c(CC)cncc2)=O)CCCC(C)(NC(=O)CC2COC(C)(C)C2)C1 11685,c1(CC(N2CC(NC(C3C(C(C)C)CCO3)=O)C2)=O)cc2ccccc2cc1O 11686,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11687,N1(C(C(CCC)OCC)=O)CCC(NC(C23CCC(CC2)CC3)=O)C(F)C1 11688,C1(CC(=O)NC(c2c(C)ncs2)CO)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11689,C(c1ccncc1)=CC(=O)NC1C(NC(C=CCOC)=O)CC1 11690,c1(CC)cccc(S(=O)(=O)N2CCN(C(c3cc(C)cc(Br)c3)=O)C(CC)C2)c1 11691,c1(C(=O)NCC2=CCN(C(C3CC3F)=O)CC2)cc(F)cc2nc[nH]c12 11692,c1(C(=O)NCC(CC)N(C(=O)C(C)C(C)C)C)ncnc(C)c1C 11693,C12(C(=O)NC3COCCN(C(=O)Cc4ccccc4Cl)C3)CC=CCN1CCC2 11694,C1(C(C)C(=O)OC(C)(C)C)CCN(C(c2onc(NC(N(C)C)=O)c2Br)=O)CC1 11695,c1(C(=O)NCC=CCNC(=O)C=CC=C(Cl)Cl)cccc(CF)c1 11696,C1(C(=O)NCC2(CCNC(c3ccc[n+]([O-])c3)=O)CC2)(OC)CCC(C)C1 11697,C1(C(N2C(C(=O)NCCCN(CC)CC)CC(O)CC2)=O)CC12CCS(=O)(=O)CC2 11698,CC(C)CC(CO)NC(C1COCC1NC(=O)CC1(O)CCCC1)=O 11699,O(NC(=O)C(COCC)NC(=O)CCC1CCOCC1)C(CC)CC 11700,c1(C(N(CCNC(C2(SC)COC2)=O)C)=O)ccc(=O)n2c1CCCC2 11701,N1(C(CCN(C)C)=O)CC(C(=O)N(C2CCSC2)C)C(F)(F)C1 11702,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11703,C(CC(=O)N1CCC(N(C)C(c2nc(Cl)c(Cl)s2)=O)C1)(C(F)(F)F)OC 11704,CC(C(O)C(F)F)NC(C1(NC(=O)CC(=O)NCC2CC2)CCCC1)=O 11705,c1(CS(N2CCC(NC)C2)(=O)=O)ccc(SC)c(F)c1 11706,N1(C(C2C(CC)CCN2C(=O)C(O)CN(C)C)=O)CCN(C)C2(CC2)C1 11707,C1(NC(C=CCC)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11708,N1(C(c2c(C)ccc(C)c2)=O)CC2(CCC2)CC1C(=O)NCCc1ccnn1C 11709,N1(C(C(CC)C(=O)OC)=O)CC2(CCC(NC(C3CCCOCC3)=O)CC2)C1 11710,C1(NC(C(CO)N(C)C(C2CC23CC3)=O)=O)CCCN(CCO)C1 11711,CC1CN(C(=O)CCCCc2cnc[nH]2)CCC1NC(=O)CCC#N 11712,c1(C(N2CCCC(c3c(C(=O)OC)c[nH]n3)C2)=O)cnc(O)c(-c2nn[nH]n2)c1 11713,C1(c2cc(NC(N(C3CCN(CC)C3)C)=O)on2)CCN(c2ncccn2)CC1 11714,C(=O)(C1=CCN(C(c2cc[nH]n2)=O)C1)NC(c1ncc[nH]1)C 11715,C(=O)(CC(C)(C)N(C)C(c1cccnc1)=O)N(C(C)C)CC1CCCO1 11716,Nc1cc(C(=O)NC(CC2CC2)C(=O)N2CCSCC2)on1 11717,c1(C(C)OC(C=Cc2ccc(C(=O)OCC)o2)=O)cc2cnccc2o1 11718,c1(SC)nn(C)c(CN2CCSCC2C(=O)Nc2ncccc2Br)c1Cl 11719,C1(=O)CCCCCCN1CC.C=CC1COCC1NC(C1C(C#N)C1(C)C)=O 11720,C(=O)(C1=CCN(C(C2(F)CCCC2)=O)CC1)N(c1cnc(F)nc1)C 11721,N1(c2n(CC=C)c(-c3ccc4c(c3)OCCO4)nn2)CCCC2CN(C)CCC12 11722,CC(C)(C)S(=O)(=O)CCNC(c1cnc(C(C)(C)C)nc1)c1nnnn1C(C)(C)C 11723,Cc1cc(C(N2CC(N(C(=O)C(F)F)C)C(F)C2)=O)c(C)n1-c1ccc(Cl)cc1 11724,C1(CC(=O)NC(CNC(C(C=C)O)=O)C2CCC2)CCC(C(C)(C)C)CC1 11725,C(CCCn1cc(-c2ncoc2NC(C)=O)nn1)(c1cccnc1)OC 11726,CCC(O)CC(=O)NC(C)(C(=O)N(C)CC1CCCC2CC12)C1CCC1 11727,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)C)C1 11728,c1(C(N2CC(CC(=O)N(CCCCCC)CCO)(OC)C2)=O)ncn2c1CCC2 11729,CC1CSCCN(C(C2(CNC(c3cc[nH]n3)=O)CC2)=O)C1 11730,CCC(CC(=O)NCCC1CCCCC1O)N(C(=O)C(C)N1CC(C)C1)C 11731,C1(N(C)C(C2CC2C2CC2)=O)CCN(C(c2cnc(O)s2)=O)C1C(C)(C)C 11732,c1(O)cnccc1CNC(=O)C(C1CCN(C(C2C3CCOCC23)=O)C1)F 11733,c1(CC)cnc(C)nc1N1CCC(CF)(NC(c2nn(C)cc2Cl)=O)C1 11734,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11735,c1(C(N2C(C)CC(NC(c3c(C)cc(C)nc3)=O)C2)=O)ccc2nc(S)[nH]c2c1 11736,c1(C(N2CCC(C)C2)=O)cccc(C(N2CCN(C3CC3)CC2)=O)c1 11737,c1(CC)cc(F)ccc1C(=O)NC(C)C(C)NC(C1(C2CC2)CC1)=O 11738,c1(C(=O)NCCC(=C)CNC(C2(C)CCC(F)(F)C2)=O)cnc(C2CC2)nc1C 11739,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11740,N1(C(c2c(C)nc(Cl)s2)=O)CCc2sc(C(=O)NCc3cccnn3)cc2C1 11741,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11742,C(CN=C(NC(c1cccs1)C1CC1)NC1CC2(CC2)C1)N(C)CC1CCCO1 11743,N1(C(C(CC=C)NC(C)=O)=O)CCCC(NC(=O)CCCSC)CC1 11744,N12CCC3C(CCCN3C(=O)Cn3ncc(c3C)C1=O)C2.C1(C2(C)CC2)CC(=O)C1 11745,C(CNC(=O)C(n1ccc(Br)n1)C)(C(C)C)NC(C1(CCC)CC1)=O 11746,c1(C(=O)NCCCNC(C2CCC3CC23)=O)nc2c(s1)COCC2 11747,C1(C(=O)NCC2(O)CCC2)(CC)CCN(C(=O)C(C)(O)C2CC2)CC1 11748,c1(C(N2CC(n3cc(C(=O)NCC(C)C)nn3)C2)=O)cc(Cl)cn1C 11749,C(C(=O)NC1CCOC1)(C(C)CC1CCC1)N(C1CCC1)CC 11750,c1(C(=O)OCCNC(=O)NOC2CCCCC2)ccc2c(O)ncnc2c1 11751,CC1CCC(NC(c2cnc(Cl)[nH]2)=O)CN1C(c1ccc(-c2cn[nH]c2)cc1)=O 11752,C#Cc1cncc(C(N2CC(C(N)=O)(CNC(=O)C=CCc3cncnc3C)C2)=O)c1 11753,Cc1cc(C(N2CCOC(CNC(=O)C(c3ncccc3F)(F)F)C2)=O)c(C)s1 11754,Cc1ncsc1C(Cn1cc(-c2ccccc2)nn1)NC(=O)CCN(C)C 11755,c1(C(=O)NC2CCCC(NC(c3cccc(C)c3Cl)=O)C2)cc(N)c(N)cc1F 11756,n1(CC(=O)OCC)nc(C)n(CC(=O)OCOc2nocc2C(C)C)c1=O 11757,C(=O)(CCCCCC(C)(C)C)NC(CCNC(c1ccc(CSC)o1)=O)C(C)C 11758,c1(CC)cnc(C(Cc2cncnc2)NC(=O)CCN(C)C)s1 11759,C1(CC(=O)NCC2(CC(C)C)CC2)CN(C(=O)CCNC(=O)CO)CCC1C 11760,C1(C(=O)NCC2(C)OCCN(C(C(=O)NC(C)C)=O)C2)Cc2ccccc2N1C 11761,c1(CN2C(C)(C(=O)Nc3cccc(C#C)c3)CC2)cc(Cl)cc(Br)c1O 11762,N1(C(C(CCN(C)C)NC(CC2(C(=C)F)CCC2)=O)=O)CCSCC(C)C1 11763,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2ncc(C)cn2)=O)OC(C)(C)C1 11764,N1(C(c2c(CC)ocn2)=O)CCCC2(C1)CN(C(c1c(C)noc1C(C)C)=O)C2 11765,Cc1nc(CNC(=O)CC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11766,N1(C(COCC=C)=O)CCOCC1CNC(C1CCCC(CF)C1)=O 11767,Cc1ccccc1C(N1CCOCC1c1noc(C(C)NC(=O)C(C)CO)n1)=O 11768,N1(C(C(CCC)CC)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccc(C)o1)C3 11769,c1(SC)cccc(C(=O)NCC(=O)NC(c2ccc(Br)cc2)C(=O)O)c1 11770,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11771,N12CC(C(C)C1)C2=O.c1(C(C(=O)NS(CC)(=O)=O)O)cccnc1 11772,Cc1c(F)cc(C(N2CC(NCc3ccc(C(C)C)s3)C(C#N)C2)=O)cc1Br 11773,N1(C(Cc2nc(C)[nH]n2)=O)CCC(C2(NC(=O)CCC(C)C)CC2)C1 11774,Cc1ccc(=O)n(CC(N2CCC(CCNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)n1 11775,N1(C(CCN(C)C(C2(C3CC3)CC(=O)C2)=O)=O)CC(C2CCCCC2)C1 11776,CCCCCCC(F)C(=O)NCC12CC1CN(C(C1(C)CCC(=O)NC1)=O)C2 11777,c1(NC(C2CN(Cc3cncnc3)CCN2)=O)ncc(Br)cc1Br 11778,N1(C(c2cc(OC)no2)=O)CCN(C(c2ccc(Cl)[nH]2)=O)CC1C1CC1 11779,C#Cc1cc(C(N2CCCC2(C)CNC(c2ccc(O)cc2)=O)=O)ccc1Cl 11780,C(=O)(C1=CC2CCCC12)NCC(C)(C)NC(c1cc(C)cc(C(=O)OC)c1C)=O 11781,CC(C)CC(=O)C(=O)NC(C(N1CC(CO)CC(C)C1)=O)c1ccco1 11782,C(CC(C(=O)NCCc1cccnc1)NC(=O)CCc1cncs1)OC 11783,Cc1c(C(=O)NCCn2cc(C(=O)NC(c3ncnn3C)C)nn2)ccn1C 11784,C1(C(N(CCN(C(CC2C(C)=NOC2=O)=O)C)C)=O)SC2C=CC1CC2 11785,n1(CC)nc(C(N2CC3CC3(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)cc1O 11786,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(CC(=O)NC2CN(C(C)=O)C2)C1 11787,C(=O)(C(CC(C)(C)C)NC(c1ccnc(O)c1)=O)NC1CCC(C)(OC)CC1 11788,C(CN=c1nc2[nH][nH]cc-2c(O)n1)c1c(OC(C)(C)C)cccc1 11789,C1(C(C)C)C(NC(C2CCNC2=O)=O)CCN1C(=O)CCCn1ccnc1 11790,N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2(CCCN(C(=O)Cc3cc[nH]n3)C2)C1 11791,C1(NC(c2cc(C)on2)=O)CC=CCC1C(=O)NC1CC(CC(C)(C)C)C1 11792,C1(C(N2CCC(N(CC#C)C(C3COCCO3)=O)C2)=O)CCCCC1(C)C 11793,c1(C(=O)NCC(NOCC(CC)CC)=N)ccc(Cl)cc1 11794,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11795,c1(C(C)(C)C)c[nH]c(C(=O)NC(CNC(=O)CCC2CCCCO2)CO)c1 11796,c1(C(=O)NCC2(CNC(=O)C(F)=C(C)C)CC2)cc(=O)n(-c2ccccc2F)[nH]1 11797,N1(C(c2c(C)ncn2C)=O)CC2OCCN(C(=O)CN3CCCC3C)C2C1 11798,Cc1cc(CN2CCC(C)(NC(=O)Cc3cc(C)n(C)n3)C2)c(C)s1 11799,N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(C)nc(C)n1O)=O)C2 11800,Cn1cc(Br)cc1C(=O)NC1CC1CNC(c1cncnc1-c1ccccc1)=O 11801,c1(C(=O)NCCCN(C(C(C)O)=O)CC2CCCC2)ncoc1-c1ccco1 11802,c1(C(N(CC(=O)Nc2cc3cccn3c(O)n2)CC)=O)cc(F)cc2nn[nH]c12 11803,c1(CN(C(=O)C(N2CCOC(CC(C)(C)O)C2)=O)C)ccc(SC(F)(F)F)cc1 11804,Cc1cc(F)cnc1C(N1CCCC1CCNC(C1(C(F)(F)F)CCC1)=O)=O 11805,N1(CC(=O)NCc2scc(CC)n2)CCCN(C(C2C=CCC2)=O)CC1 11806,N1(C(=O)C2=CCCO2)CC2CCCN(C(C3C=CCCC3)=O)C2C1 11807,N1(C(C2N(C(CC(C)OC)=O)CCC(C)C2)=O)CCCC(N=[N+]=[N-])CC1 11808,c1(OCC(N2CCCC(Cn3cccn3)C2)=O)ncc(Br)cn1 11809,C(=O)(C1=CCCC1C)NCc1cc(C(=O)NCC(C)OCC=C)on1 11810,N1(C(C2C(C=C)OCC2)=O)CCC2(CCN(C(C3CSCC(=O)N3)=O)CC2)C1 11811,c1(C(N2CCC(c3cncc(C)c3)C2)=O)cccc(Br)c1N 11812,C1(N(C(CC2(COC)CC2)=O)C)CCCN(C(c2coc(C)n2)=O)C1 11813,N1(C(CC2=NN(C)C(=O)C2)=O)CCC2CCN(C(c3ccc(Cl)nc3)=O)CC2C1 11814,CCC(C)(CNC(=O)C(C)CN(C)C)NC(=O)C1=CCC1 11815,N1(C(C(C2CC(NC(c3ccn(CC)n3)=O)C2)OC)=O)C(CO)CC2OCCC12 11816,C(=O)(C(F)(F)C(O)c1ccccc1)NCC(C)NC(=O)CSC1CC1 11817,C(=O)(C1CCCc2nccn21)N1C(c2nc(C)on2)CN(C)CC1 11818,C(=O)(C1=C(F)CN(C(C2CCC(C)(C)CC2)=O)CC1)N1CC2(CC(OC)C2)C1 11819,N1(C(C2C(C)N(C)CC2)=O)CC2(CCNC(=O)CCC(N)=O)CCC1C2 11820,CC(CS(C)=O)C(=O)N1CCN(C(C)CNC(c2ncccc2F)=O)CC1 11821,Cc1ccc(C(N2CCC3CN(C(=O)C4CC4)CC3C2)=O)c2ccccc12 11822,N1(C(C2(C#C)CC2)=O)CC(NC(c2coc(C)n2)=O)CCC(O)C1 11823,c1(-c2n(C3CCC(C(C)(C)C)CC3)nc(CCCO)n2)cccc2nc(Cl)cn12 11824,N1(C(c2c(CC)con2)=O)CC2CCCC2(NC(=O)C(C)n2cncn2)C1 11825,C1(F)(C(=O)NC(C(=O)O)C2CCC2)CN(C(=O)OC(C)(C)C)CC1C1CC1 11826,CC1COc2c(C(=O)NC3CCC3CNC(c3cnc(Cl)s3)=O)cccc21 11827,C(=O)(CC(=O)NCC(C)(CO)NC(=O)CC(C)OC)OC 11828,C12(NC(COC(CC)(C)C)=O)CCCCC1N(C(c1ccncc1NC)=O)CC2 11829,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11830,c1(C(N(C2CCN(C3CCN(C)C3=O)CC2)CCOC)=O)ccc2oc(O)nc2n1 11831,CC1(C)CC(C(=O)NCC23CC(NC(=O)CC4CCCS4(=O)=O)(C2)C3)CNC1=O 11832,Cc1ccncc1-c1cn(C2CC(C(=O)N(C)CCN3CCOCC3)C2)nn1 11833,C=CC(CC)CC(=O)N1CCN(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 11834,N(C(=NCCCF)N1CCCC(S(C)(=O)=O)C1)Cc1c(C)ncc(Cl)c1 11835,c1(C(N2CC(CCc3cn(C(CC)C)nn3)C2)=O)cc(Br)cc([N+](=O)[O-])c1N 11836,C1(CCNC(CC2(C)OCCO2)=O)CCCN(C(c2ncc(Cl)s2)=O)CC1 11837,c1(C(C(=O)NCCC2CCC(NC(c3cnns3)=O)C2)(F)F)ccc(F)cc1F 11838,C=CCC(CC)C(=O)NCC1(NC(c2ccoc2CC)=O)CCCC1 11839,Cc1cncc(C(N2CC(Oc3ccc(C4CC4)cn3)C(O)C2)=O)n1 11840,c1(C(=O)NC(CC(C)NC(C(CC)O)=O)C)cccc2nsnc12 11841,c1(C(N2CCCC(CN(C(C(CC)CO)=O)C)C2)=O)ccc2nonc2c1 11842,C1(OCC)CC(CNC(=O)C(=O)NCC(O)COC)C12CCC2 11843,c1(CNC(C2CC2F)=O)ccc(CNC(=O)Cn2cc(CO)nn2)cc1 11844,N1(C(C(C2CCCCC2)NC(C(=O)NC(C)C)=O)=O)CCS(=O)(=O)CC1 11845,C1(C(=O)NCC2CCN(C(C3CCOC3)=O)CC2(F)F)CCC2(CCCC2)CC1 11846,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CCc2nncn2C)CC1 11847,n1(CC)c(N2CCC(SCc3cccc(SC)c3)CC2)nnc1C1(C)C=CCC1 11848,C1(C(N(CC=C)C)=O)CCN(CC2CCN(Cc3ccccc3)C2)C1 11849,N1(C(COCCCC#C)=O)CCC(C2N(C(=O)C=CC)CC2(C)C)CC1 11850,C(=O)(C1=C(C)CCCC1)NCCCN1CCN(C(C(CCCC)O)=O)CC1 11851,C(=O)(C=CS(F)(F)(F)(F)F)N1CCN(C)C(CNC(=O)Cc2cc[nH]n2)C1 11852,c1(COC)occ(C)c1C(=O)NC(c1ccc(C)cc1)CNC(c1ccno1)=O 11853,N1(CCC)CCc2cc(CN(C)CC(C)CN(C)C)ccc21 11854,C1(NC(c2c(SC)cn(C)n2)=O)CCN(C(c2cc(F)ccc2F)=O)C1(C)C 11855,CCCC(C(=O)N1CCC(NC(c2ccc(O)c(F)c2F)=O)CC1C)S(N)(=O)=O 11856,CC1OC2(C)CC1(C(N1CC(=C(F)CNC(c3cc(Cl)cs3)=O)C1)=O)C2 11857,c1(OC)ccc(NC(C2CC(CNCC(c3ccccc3Cl)O)C2)=O)cn1 11858,C1(C#N)(C(=O)NC(C2CCCC2)CNC(C(C2CCOCC2)C)=O)CC=CC1 11859,C(=O)(CCCCCC(C)(C)C)N(CC(C)O)CCNC(C1C=CCCC1)=O 11860,C(CC(O)C(=O)N1CCC(CCc2cn(Cc3cccnc3)nn2)CC1)SC 11861,C1(C(=O)NC(C2CCCN2C(=O)CC2CCCC(O)C2)(C)C)CC(S(C)(=O)=O)C1 11862,C12(C(=O)NCc3nc(CNC(C4CCCC4C(F)F)=O)sc3)CCCN(CC1)C2 11863,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11864,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)Cn2cc(C3CC3)nn2)CCCO1 11865,c1(OC)ccc(C(O)CC(=O)NC2CC(=O)N(c3cccc(OC)c3)C2)cc1 11866,C1(C(N(CCCCC)CCO)=O)CCCCC1(C)NC(c1csc(Cl)n1)=O 11867,C#CC(CNC(=O)C(C)(CC)CC)CC(=O)N1CC=CCO1 11868,C1(C(N(CC(C)NC(c2c(C)snc2)=O)C)=O)CCCN(C(=O)C2CC2)C1 11869,C1(O)(CNC(COCC)=O)CCN(C(=O)C=C2CCCCC2)C1 11870,c1(OCC)cc(C(=O)NC(C)C=CC(=O)NCCCOCCO)[nH]n1 11871,c1(C2(SCC(CO)F)CCC2)ccccc1F.n1(C)cncn1 11872,c1(N2CCC(C(C)NC(C=COCC)=O)C2)ncc2cccnc2n1 11873,N1(C(C2(CC3CC3)CC2)=O)CCN2CCCCC1C2.C12CCCCCC1NC2=O 11874,C1(NC(CC2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1cccn1CC)=O 11875,c1(C(=O)NC(c2ccccc2)CNC(C2=C(C)CC2)=O)cc([N+](=O)[O-])n[nH]1 11876,N1(C(COCCC=C)=O)CCC2(CC1)CN(C(C1CCCN(C)C1)=O)CC(C)O2 11877,N1(C(c2c(CC)scn2)=O)CCCC(CO)(NC(=O)CNC(C2CCC2)=O)C1 11878,C1(CNC(C=CCCC)=O)C2CN(C(c3ccc(I)cn3)=O)CC12 11879,c1(CC)ccccc1CN(C(c1cc(CO)on1)C(=O)Nc1ccc(F)cc1)C 11880,N1(C(CCCOCC)=O)CCCC(CNC(=O)CCCCC2CC2)C1 11881,c1(-c2cn(CC(=O)N(CCC)C(C)C)nn2)ccc(C(=O)NC(C)C)nc1 11882,c1(NCc2c(-c3ccc(OCCOC)c(O)c3)c[nH]n2)c(F)cc(F)c(F)c1F 11883,c1(C(=O)NC2CCCC(N(C)C(C3CCC3(F)F)=O)C2)ccc2c(c1)NCC2 11884,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2nc(CC)sc2N)=O)C1 11885,N(C1CCc2cc(Br)ccc21)C(c1ccccc1S(=O)(=O)N1CCCCC1CO)=O 11886,Cc1ccc(C)c(C(=O)NC2CCN(Cc3cccc(N(C)C)c3)CC2F)c1C 11887,c1(C(=O)NC2C(C)CN(c3nc(C#N)ncc3Cl)CC2)ccc2ncccc2c1 11888,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11889,CCC(CC)C(=O)NCCCCC(C)NC(C)=O.c1(OC(=O)CC)ccc(Cl)cc1 11890,C1(N(C(CSC(C)C)=O)C)CC2CCC(C1)N2C(C1CCCCCO1)=O 11891,O(N1CCC(c2nc(C(N(CC)CC)=O)no2)CC1)Cc1cocn1 11892,c1(NC(C)CS(C)=O)ccc(S(=O)(=O)NCc2cnco2)cn1 11893,CC1(C)CC(CNC(=O)Cc2cc[nH]c2)(CNC(C2CCC(C)CC2)=O)C1 11894,c1(C(N2C(CNC(c3c(C(C)C)noc3)=O)C(C)CC2)=O)ncc(Cl)cc1Cl 11895,CC1Oc2c(F)cccc2C1NC(=O)C(N1CCCC(O)(C(N)=O)C1)=O 11896,CC1(C)CC(NC(=O)Cc2csc(Cl)n2)N(C(=O)CC2CCC3CC3C2)C1 11897,C(CCC(=O)NC(N)=O)=C(C)I.C12(CC1)CC(=O)NCC2 11898,C1(NC(C2CC(N(C(CN(C)C(N)=O)=O)C(C)(C)C)C2)=O)CCn2nnnc2C1 11899,CC(C)CC(F)C(=O)NC1CC(C)(CNC(c2csc3cncn23)=O)C1 11900,c1(C(N(C2CCCN(C(C(C)(C)N(C)C)=O)C2)C)=O)cc2n(n1)CCN(C)C2 11901,c1(SCC(=O)N(C2CCCCC2)C(=O)C(F)=CCNC(C)C)ccccc1 11902,CCCCC(C(=O)NCC1(O)CCN(C(=O)Cc2cnccc2Cl)CC1)C(C)C 11903,C(=O)(C(C)(C)C1=CCN(C(=O)Cn2cccc2)C1)NC(C)Cc1ccnn1C 11904,n1(CC(=O)NCC(C)(CNC(=O)CCOC2CCC2)OC)nc(C)nc1C 11905,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 11906,c1(N2CC(CC(C)(C)C)OCC2)nc(N2CCC(CCF)CC2)nc2c1SCC2 11907,O=S(=O)(c1cc(Br)cc(Br)c1)N1CCn2c(C3CC3)nnc2C1 11908,c1(C(=O)NCCC2(O)CN(C(C(CC#C)C)=O)C2)cc(NC(C)=O)cc(Cl)c1 11909,C1(C(=O)NC(C)(C)Cc2ccncc2)Cc2ccc(F)cc2C(=O)O1 11910,c1(C2(N(C)C)CC2)cn(C2CCC(C(=O)NCc3cnn(CCF)c3)C2)nn1 11911,c1(OC)cc(C(=O)NCC2(C(=O)NC3CCC(Br)C3)CC2)ccc1Cl 11912,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(C(F)F)c1 11913,CC1CCN(C(c2cnc[nH]2)=O)CC1CNC(c1cc(Cl)n[nH]1)=O 11914,S(=O)(=O)(c1ccc2c(c1)CCCO2)N(CC=C)Cc1cccc(Br)c1F 11915,C1(C(=O)NCc2noc(C3CC3)n2)(CC)CCN(C(=O)Cc2cccnc2)C1 11916,N1(C(C)C(N2CCC(C)CC2NC(c2ccc[nH]2)=O)=O)Cc2ccccc2C1 11917,Cc1cc2sc(C(=O)NCC(C)NC(=O)C(C#N)C(C)C)cc2s1 11918,CC(CNC(c1cnc(C(F)F)s1)=O)(CO)NC(c1ccc(C2CCOC2)s1)=O 11919,c1(OC)ccc(O)cc1NC(=O)CCCN(C(=O)C(C)(C)C(C)O)C 11920,CCC(O)(CC)CCNC(C1CC(NC(=O)C(C)c2cccs2)C(O)C1)=O 11921,c1(C(N2CCC(NC(C(CC=C)C)=O)(CF)C2)=O)cccn2c(CCC)nnc12 11922,C1(C(=O)OC)CCCCC1C(=O)NCCC1(O)CN(C(=O)C2=NOCC2)C1 11923,c1(C(=O)NC2C(CNC(c3nc(C)n(C)c3)=O)C2)cc(Cl)cc2c1CCC2 11924,C1(O)CCCC(C(=O)NOC2CC3CCC2C3)C1.N1(C=O)CCC(F)CC1 11925,N1(C(c2cc(OC)nn2C)=O)CCN(C(c2ccnnc2O)=O)C2CC12 11926,C1(c2n(C(CC)C)nnn2)(Nc2cnn(CC(C)C)c2C)CSC(C)(C)C1 11927,N1(C(C=CCN(C)CC)=O)CC2(CCCC2NC(=O)Cc2ccc(C)cc2Cl)C1 11928,C(=O)(C(C)(C)CCC#N)N1CCN(Cc2c(NC(C)=O)cccc2)CC1C 11929,C12(C(N3CCC(N(C(CCCC#CC)=O)CCO)CC3)=O)CCC(CC1)C2(C)C 11930,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 11931,c1(CNC(=O)Nc2ccnn2-c2ccccc2)cccc(C2CCCO2)c1 11932,C(CC(C(=O)NC1CC(NC(=O)CC2CC(CC)C2)C1)c1ccccc1)=CC 11933,c1(N(C)Cc2nccc(N3CCCC(CCC=C)C3)n2)ncnc2cccnc12 11934,N1(C(c2cccc(NC)n2)=O)CCC(C)(C)C1C(=O)NOCCC(F)F 11935,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 11936,C(=O)(C(O)CC(F)(F)F)NC1(C)CCN(C(=O)Cn2cnc(Br)n2)C1 11937,c1(C(CNC(C2CN(C)C2)=O)NC(C(C)=C2CCCC2)=O)ccccc1 11938,C(=O)(CCCCCC(C)C)N1CCC(C(C(N2C(CC)CCC(C)C2)=O)F)C1 11939,c1(OCC)nc(N2CCCC2CNC(C23CCCC(CO2)C3)=O)ncc1Cl 11940,C1(C(=O)NC2CN(C(c3c(CCC)nns3)=O)CC2C)CCC2(C1)CC2(F)F 11941,CC1(C)CN(C(=O)C(N)=O)CCC1NCc1ccc(F)cc1Cl 11942,N1(C(C(C)SC)=O)CCC(C2CCN(C(c3cn(C)nc3C(F)(F)F)=O)CC2)C1 11943,CC1(C)COCC1CC(=O)NC1CCC=CC1C(=O)NCCc1nncs1 11944,c1(CN2CC3(C(C(N4CCCC(CCO)C4)=O)C3)C2)cccn2cncc12 11945,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)CC1 11946,Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NC3CCNC3=O)co2)n1 11947,c1(C(N2CCC(C3N(C(COCC=C)=O)CCC3)C2)=O)ccc(Cl)c(Br)c1 11948,C(=O)(C(C(C)(C)C)NC(C1CC2CCC1N2C(c1ccnnc1)=O)=O)NC 11949,C1COCC(C)O1.C=CC(C)C(=O)ON(CCN(C)C)C 11950,C(=O)(C1=CSCCO1)N(CCCNC(=O)Cc1sccc1Cl)CCC 11951,C(N=c1nc2c(c[nH]1)COC2)C1C(C)CN(C(=O)C(F)(F)C2CCCC2)CC1 11952,C12(C(N(CC#C)C)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 11953,CC1C(NC(=O)C(C)(C)COCC(F)F)CC2CCC1N2C(c1cnn(C)n1)=O 11954,C(C(C(=O)NCC(=O)CC1CCC(=O)O1)NC(=O)CCC1(C)CC1)N(C)C 11955,C1(C#N)(C(N2CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)CCCC(=O)C1 11956,C1(NC(=O)CSc2cnc[nH]2)CCN(C(=O)CCc2ccccc2O)C2CC12 11957,Cc1[nH]nc(C(=O)NCC2(CCNC(=O)CN3CCCS3(=O)=O)CC2)c1Br 11958,C12CCCN(C1C)C(=O)OC(C)CNC2=O.c1(C(=O)NC(C)(C)C)cccnc1 11959,c12cc(ccc1N)OCCC(=O)NC1(CC1)CCNC2=O.C(C(C)C)OCC 11960,Cc1ccc(F)c(C(N2CC(CNC(=O)C(C3CCOCC3)C)C(O)C2)=O)c1 11961,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CC(C)C)C2)=O)C1C 11962,c1(C(=O)NCCC(C)NC(=O)CCC2CCCCN2C)cc([N+](=O)[O-])cnc1N 11963,N#Cc1ccc(-c2cn(C3CCCC3NC(C34CCC(C3)C4)=O)nn2)cc1 11964,N1(C(C(C(C)C)NCC)=O)CCCN(C(=O)C=Cc2cnn(C)c2C)C(C)C1 11965,c1(CNC(=O)NCCC2(OCC)CCC2)cccc(NC2CC2)c1C 11966,Cc1cc(C(=O)NCCn2cc(C(=O)NC(C)CS(C)=O)nn2)ccn1 11967,C1(C(=O)OC)CN(C(=O)CCc2cccnc2)CC1O.C1CS(=O)(=O)N1 11968,C(C(=O)CCC(=O)N=c1ccn(C2CCN(C(=O)CCCN(C)C)C2)[nH]1)OC 11969,C#Cc1ccc(C(N2CC3CC3(C(=O)NCCc3nnc(O)o3)C2)=O)cc1 11970,CCC(C)CCCC(=O)N(C1CCCN(C(=O)CCCNC(C)=O)C1)C 11971,c1(OCCC)ccc(CCC(=O)N(C(C)CCNC(=O)C(C)SCC)C)cc1C 11972,c1(COC)cc(C(=O)NCc2cn(CCN3CCC3c3cccnc3)nn2)no1 11973,C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CC2CCC(C1)N2C(C1(O)CC1)=O 11974,Cc1cc(=O)n(CCC(=O)NCCNC(=O)CSC2(c3n[nH]c(=N)s3)CC2)cn1 11975,N1(C(C(C)=CC2CC2)=O)CCOC(CNC(C2CC(F)C(=O)N2)=O)C1 11976,C(CN=c1cc(Cl)nc(C(F)(F)F)[nH]1)(C1CC1)NC(=O)Cn1cc(Cl)cn1 11977,c1(C(=O)NCCC2(C)CCN(C(COCC#C)=O)C2)c(NC(C)C)cccc1F 11978,C1(CCOC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1 11979,c1(OC)c(NC(C2CCCCN2C(c2coc(C)n2)=O)=O)ncnc1Cl 11980,Cn1cc(C(=O)NCC2(NC(C3(C)CCNC3=O)=O)CCC2)c(=O)n(C)c1=O 11981,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)CC 11982,C1(CNC(CCCC)=O)CC2(CCN(C(=O)C(C(C)C)OCC)CC2)C1 11983,c1(NC(CCC(=O)NC2(CC=C)CCN(C(=O)CC3CCC3)C2)=O)ccc(Cl)c(Cl)c1 11984,CCCC(O)C(=O)N(CCCNC(=O)CCCC#N)C 11985,N(C(=NCc1ccc(C)cc1)NC1CCOCC1)CC(C1CCOCC1)OC 11986,C1(OC)C(OC)CN(C(=O)CC2CC(F)(F)C2)C1CNC(c1c[nH]c(C)c1)=O 11987,C1(OCC)COCCC1CC(=O)N(C)CC1CCN(CCC2CC2)CC1 11988,C1(OC)CC2(CCC(C(=O)NC3CCCC(CNC(=O)CNC(N)=O)C3)CC2)C1 11989,Cc1cncc(CSc2cncc(NC(=O)C3CC3)c2)c1 11990,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 11991,c1(C(=O)NC(C2CN(C(CC(C)SC)=O)C2)C)ncnc(C)c1C 11992,C(=O)(C(=O)CC(C)C)N1CCC(C(C)NC(C2(OCC)CCOC2)=O)CC1 11993,C1(C(N2C(C3(NC(c4cnco4)=O)CC3)CCCC2)=O)CC12CC(F)(F)C2 11994,C12(C(CNC(CC3CC(C)C3)=O)NC(=O)CC3CCCOC3)CCC(CC1)C2 11995,N1(C(c2cc(C)c(C)o2)=O)CCC(CNC(=O)Cc2csc(S)n2)C(F)(F)C1 11996,CC(C)(C)CCC(F)C(=O)NC1COC2CN(C(C3CC(=O)C34CCC4)=O)CC12 11997,C1(CN(C(C2CCC(OC)C2)=O)C)CCCCN1C(c1cc(OC)ns1)=O 11998,c1(-n2cc(C(=O)N(C)C)nn2)ccc(OC(F)(F)F)cc1.C1(N(C)C=O)CCC(N)C1 11999,c1(C(=O)NCCN(C(C)C)C(C2(CCN(C)C)CC2)=O)cc(C(F)F)ccn1 12000,C(=O)(C#CC1CCCCC1)N1CCCCC(NC(c2c(SC)cn(C)n2)=O)C1 12001,N1(C(CSCC=C)=O)CC2(CNC(C3(C)C=CCC3)=O)CCC1CC2 12002,c1(CC(=O)NCC(CN(C(=O)Cc2cn[nH]c2)C)O)nc2ncccn2n1 12003,c1(C(N2CCC(CC=C)(NC(C3CSCCS3)=O)C2)=O)c(F)cc(F)c(O)c1F 12004,CC(CC(C)(C)C)C(F)C(=O)NCCC1CC(F)(F)CN1C(=O)CCC1CC1 12005,C1(N(N2CCN(C(=O)Cc3cncn3C)C(C)C2)C)CCC2(CCC2)CO1 12006,c1(OC)ccc(S(=O)(=O)N2CCCC(C(=O)O)CC2)cc1.C1CC(=O)O1 12007,CC(CC(=O)NCC(F)CO)C(C)(C)NC(c1ccc(F)cc1)=O 12008,C(=O)(C1CCc2nccn21)NCCN(C(c1cccc(CC)c1)=O)C 12009,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12010,c1(-c2cn(CC3CN(C(C(C4CC4)SC)=O)C3)nn2)ccc(C(F)(F)F)cc1 12011,c1(N(CC(N2CC(C)(NCC(C(=O)C(F)=CCCF)=O)C2)=O)C)ccc(F)c(Cl)c1 12012,c1(C(N2CC3(C(NC(CC4(C)CCCC4)=O)CC3)C2)=O)cnc2ncc(Cl)cn12 12013,Cc1nncc(C(=O)NC(c2ncsc2C)C)c1C 12014,N1(Cc2cn(CC(C3CC3)NC(Cc3cn(CC)nc3)=O)nn2)CCCC(C)C1 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12032,C1(NC(C(C(C)C)N(C)C)=O)C2CC3C1C3C2C(N1CC(F)(CO)C1)=O 12033,c1(OC)ccc(C(=O)NC(C)C(CO)NC(=O)C=CC2CCOCC2)cn1 12034,c1(CCC(=O)NC2CN(C(=O)CC3CC4(CC4)C3)C2)c[nH]c2ccccc2c1=O 12035,c1(OC(C(=O)NC(CCCCNC(C(C)=CC)=O)C)(C)C)cccc(CC)c1 12036,N1(N2C(C(=O)NC(c3scc(C)c3C)=O)CCC2)CCCC(Cc2nc(C)sc2)C1 12037,CC1(C)C2CC(C(=O)NC3(CNC(=O)CC4CSCCS4)CCOC3)CC12 12038,N1(C(C23CCC(NCc4ncc(Cl)cn4)(CC2)CC3)=O)CCN2CCCC2C1 12039,n1(CC)cc2ncccc2n1.n1(CC(=O)N(CCCNC)C)cc(CCC#N)nn1 12040,c1(C(CCC)NC(=O)OCC2CNCCO2)ccc(CN(C)C)cc1Cl 12041,C1(O)(C(C(=O)NCc2ccccc2)NC(C2CS(=O)C2)=O)CCCCC1 12042,C1(CC)C(NC(C2CS(=O)C2)=O)CCCN1C(c1ccc(C)c(C)c1)=O 12043,CC1CCc2c(C(N3CCOC(CC(=O)NCC(F)(F)F)C3)=O)n[nH]c21 12044,CC(C)C(C(C)NC(c1cscc1Cl)=O)NC(c1ncoc1-c1ccon1)=O 12045,CCCS(=O)(=O)C(C)C(=O)NCC1CN(C)CCN1C(=O)OC(C)(C)C 12046,c1(C(N2CCC3(NC(C(C)N(C(C)=O)C)=O)C(C2)C3)=O)n[nH]c2c1CCCC2 12047,C1(CNC(Cc2ccc(C)s2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12048,N1(C(CSCC)=O)CC(OC)CC(NCCNC(C23CCCC2CCC3)=O)C1 12049,c1(C(N2CCOCC2c2ccco2)C(=O)N(CCC#N)C)cccc([N+](=O)[O-])c1 12050,CCC(CNC(=O)CCC(C)NC(=O)CC(C)OC)CCO 12051,C1(c2cn(CCCCCCOC(C)=O)nn2)(NC(=O)C(Cl)=CCl)CCCOC1 12052,C1(C(=O)NCC(=C)C)COC2(C1)CN(C(=O)C(C)OC)C2 12053,c1(C(N2CCC(O)(CNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12054,C1(NC(c2c(C)cc(Cl)cc2)=O)CC2(CCN(C(C3(C(F)F)CCC3)=O)CC2)C1 12055,C(=O)(C1=NN(c2ccc(F)cc2)C(=O)CC1)NC(C(C)NS(=O)(=O)C(F)F)(C)C 12056,n1(CCC)cc(C(=O)NCCN(C(=O)CC2OCCC2C)C(C)C)nn1 12057,c1(CN(C2CCN(C(C(CC)OC)=O)C2)C)ccc([N+](=O)[O-])s1 12058,N1(C(CC(C)F)=O)CC23CCCC2(C1)CN(C(c1cnc2nccnc2c1)=O)C3 12059,C(=O)(C(C(C)C)C(N(CCOC)C)=O)NC1(C2(C(=O)NCCCC)CC2)CC1 12060,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12061,C1(NC(Cc2cn(C)nc2)=O)CC(OC)CN(C(=O)CCC(=O)c2ccc[nH]2)C1 12062,Cc1nc2cc(C(=O)NC(C)(C)CN(C(=O)CC3CCCC3C)C)ccc2o1 12063,C=CCC(C(=O)NCC1C=CCCC1)NC(=O)Cc1ccnn1C 12064,Cc1cc(C(F)F)ncc1C(=O)NC1CCC1NC(C1CCC2(CC2)C1)=O 12065,c1(CCC)cc(C(=O)N(C)CCNC(c2cc(N)c(F)cn2)=O)cc(O)n1 12066,C1(CNC(c2ccc(Cl)o2)=O)CC(F)CN1C(c1c[nH]nc1OCC(F)(F)F)=O 12067,C1(C(=O)NC2(CC=C)CCN(C(C3CCC(C)O3)=O)CC2)CCC(N=[N+]=[N-])CC1 12068,N#CC1(C(=O)NCC(CO)NC(C2CN3CCC2C3)=O)CCCCC1 12069,CC1CCC(C(=O)NC(CSc2cn(-c3ccccc3C(=O)O)nn2)C(=O)O)OC1 12070,C1(NC(C23N(C(COCCOC)=O)CCC2C3)=O)CN2CCC1(C)CC2 12071,C(=O)(C(C)(C)CO)NCCC(=O)NCc1nnn(C)n1 12072,N1(C(c2n(CC)ccc2)=O)CCCCC(CNC(C2CCCC(C(C)(C)C)C2)=O)C1 12073,N1(C(CCc2cnn(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12074,Cc1cc(C)c2[nH]c(=NCC(C)NC(=O)Cc3c(F)cccc3Cl)sc2c1 12075,C(CO)(CC(C)CC)OCCNC(C(COC)C)=O.C(=O)(C(C)(Cl)Cl)N.C1CO1.C1COO1 12076,c1(CCC(N2CCCC(N(C(C#CC(=O)NC)=O)C)C2)=O)c(C)ncnc1O 12077,N1(C(C(CC=C)OC)=O)CCC(C2CC(NC(=O)CC3CC(OC)C3)C2)CC1 12078,N1(C(C2CC3CCCC3C2)=O)CCN2C(CCS2(=O)=O)C1 12079,c1(C2C(C(=O)NC(c3ccc(Cl)cc3)(C)CO)C2)ccc(C#N)cc1 12080,CN1CCCC1CCC(=O)N(C1CCN(C(=O)CCCc2ccncc2)C1)C 12081,C1(CC)CCCC1NC(=O)CC1CN(C(c2cnn(C3CCC3(C)C)c2)=O)C1 12082,Cc1ccc(F)c(N)c1C(=O)NC1CC(C)(CNC(C2CCCN(C)C2)=O)C1 12083,Cc1sc(C)c(C(=O)NCC23CC(CO2)N(C(C2CNC(=O)CC2C)=O)C3)c1C 12084,c1(NCCCNC(=O)NC)nc(N2CCC(SC(C)C)C2)nc2scnc12 12085,CN=c1[nH]c(=NC(C)c2cccc(S(N)(=O)=O)c2)[nH]c(=NCC(C)N(C)C)[nH]1 12086,c1(C(=O)NCC(C2CCC2)NC(C2(C(=O)OC)CC2C)=O)ccc2nccn2c1 12087,N1(C(C2CC(C(C)(C)C)C2)=O)C2CCC1CC(NC(c1c[nH]c(C(N)=O)c1)=O)C2 12088,Cc1onc(-c2ccccc2)c1C(=O)Nc1cnccc1C(C)(F)F 12089,Cc1[nH][nH]c2ncnc(=NC(=O)C3CC(NCc4ccc([N+](=O)[O-])cc4Cl)C3)c1-2 12090,c1(C(C)C)nc(C(=O)NCC(C)(C)NC(c2cc(C(N)=O)no2)=O)cs1 12091,N1(C(CC2(OCC)CCC2)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1 12092,N1(C(C(C)(C)NC(=O)OC(C)(C)C)=O)CC=C(c2cccs2)C1 12093,C(=O)(CC1COc2ccccc21)NC1C(CNC(CC2(C=C)CCOCC2)=O)C1 12094,c1(C(=O)NC2CC(CNC(=O)CCSc3ccsc3)C2)cnc(-c2ccsc2)s1 12095,c1(NC(=O)C(=O)N(C2CCCC2O)CC2CC2(F)F)cccc2n[nH]cc12 12096,C(C(=O)N1CCC(O)CC1C)(C(C)(C)C)NC(CCc1cnc(C)o1)=O 12097,C(=O)(C(CC)n1cccn1)NCCSCC(=O)NCC1(CCC)CCC1 12098,N1(C(C(CCOC)C)=O)CCC(NC(=O)COCc2ccnn2C)CC1C 12099,c1(C(=O)NCCCOCCNC(c2ccccc2C(F)F)=O)ccc(F)cc1Cl 12100,CC1CN(c2cc(-c3ccccc3)ncn2)CCC1NC(C1CCC2CC2CC1)=O 12101,C1(C(N2CC(NC(C3CC(C)(C)C3)=O)C(C(F)F)C2)=O)CCn2c(O)nnc2C1 12102,C1(CC)CS(=O)(=O)CCN1C(=O)C(=O)NNC(=O)c1ccc(-c2ccco2)cc1 12103,c1(CNC(=O)OC(C)(C)C)ccc(NC(=O)CN2CCNC(=O)C2)c(Cl)c1 12104,C1(Nc2cccc(C(N3CCCC3)=O)c2)C2CN(C(C3CC3(F)F)=O)CC12 12105,CC1(C(=O)NCCn2cc(NC(c3ccccc3F)=O)nn2)CCC(O)CC1 12106,Cc1noc(C)c1CNC(C1CCN(C(C2CCC(O)C2)=O)CC1)=O 12107,C1(NC(C(C2CCN(C(C(n3c(C)cc(C)n3)C)=O)C2)C)=O)CC2CCCC2C1 12108,C1(CC(=O)NCC2CCN2C(C2CCC3CCC2O3)=O)CCS(=O)(=O)CC1 12109,C1(CNC(COC2(C)CCC2)=O)CCC2(CN(Cc3nc4ccccc4s3)C2)O1 12110,C(c1ccc(NC(N(C(CO)CO)C)=O)o1)=NC(=O)OC(C)(C)C 12111,N1(C(c2cn(CCOC)nc2)=O)CCN(C(c2c(C)ncn2OC)=O)CC2(CC2)C1 12112,CCC(C(=O)OC)C(=O)NC1CC(NC(c2ncccn2)=O)C12CCC2 12113,N1(C(CC(=C=C)C)=O)CCC2(C1)CN(C(c1cnc(C)c(OC)c1)=O)C2 12114,N1(C(C2(COC)CCCO2)=O)CC2CCN(C(c3cc(C)sc3C)=O)CCC2C1 12115,CC1CCCc2nc(C(=O)NCC(O)CNC(c3csc(S)n3)=O)cn21 12116,c1(CN(CCC(=O)O)Cc2cnn(-c3ccccc3)c2)ccccc1F 12117,C1(C(=O)NCc2ccc(C(=O)NCC3(O)CC=CC3)o2)(CC)CCCO1 12118,C1(CNC(C(c2nncn2C)C)=O)CC2CN(C(c3ccccc3O)=O)CC12 12119,c1(-n2c(CCCCN(C)C)nc(-c3ccccc3Br)n2)ccc(F)c(Cl)c1 12120,C=C(C)C(CC(=O)N1CC(OCCNC(=O)C(c2cnn(C)c2)O)C1)OCC 12121,N1(C(C2CCC(CC)O2)=O)CCC2(CCC(N(C)C(c3cn(C)nn3)=O)CC2)C1 12122,N1(C(C(C)NS(C)(=O)=O)=O)CC2CCC1C1CN(C(C3CC(=O)CO3)=O)CC21 12123,C(=O)(C1=CC2(CCN(C(=O)CCc3ccc[nH]3)C2)C1)N1C(C)CSCCC1 12124,c1(CS(=O)(=O)N(CC)CC2CC2CSC)cccc(OC(C=CC)C)n1 12125,N1(C(CC2N(C(c3cnc(C)s3)=O)CCC2)=O)CC(C)CC(C)(C)C1 12126,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12127,c1(C(N(C)CCN(C(=O)Cc2cnn(Cc3ccco3)c2)C)=O)cnc[nH]c1=N 12128,c1(NC(c2cc(C)cc(Cl)n2)=O)ccc(C(N)=O)cc1C#N 12129,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC(C1)N(C(=O)Cc1cc(O)nnc1O)C2 12130,c1(CC)nc(Cl)cc(=NCC(C)NC(=O)C(C2CC(F)(F)C2)O)[nH]1 12131,c1(CN(CCCNC(c2ocnc2CC)=O)C)ccc2cc(OC)ccc2c1 12132,c1(C(=O)NC(CN(C(c2ccc(SC)cc2)=O)C)C)ccc(F)c(C)c1N 12133,CS(=O)(=O)c1ccc(C(=O)NC2CN(Cc3ccc(Cl)nc3)CC2O)nc1 12134,C1(C(=O)NC(CCC)C2CCC2)CCCCN(C(=O)CC2CCCC2)C1 12135,c1(C(=O)N)nccn2nccc12.c1(C)cc(C(=O)NCCN(N(C)C)C2CC2)ccn1 12136,c1(OC)ccccc1CC(=O)NCC(C)Cc1ccoc1 12137,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12138,C1(C(=O)NC2C(C(N3CC(C(=O)OCC)C3)=O)CCOC2)C2CCC(C2)C1C 12139,C12(CNC(c3cc(C)c(F)cn3)=O)CCC(CN(C(=O)C#CC3CC3)C1)C2 12140,C1(CCNC(=O)NC2CCC(N3CCN(C)CC3)CC2)(OC)CCCCC1 12141,C1(N(C(=O)C(C2CCCC2)SC)CCOC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 12142,C1(NC(C(C)OCCC=C)=O)CCN(C2CCN(C(C3CC=CCO3)=O)C2)CC1 12143,Cc1cccc(Br)c1C(=O)Nc1ccsc1C(=O)Nc1c[nH]nc1C#N 12144,c1(N2CC(C)C(NC(C3COC(C)(C)C3)=O)CC2)ncc2c(Br)cn(C)c2n1 12145,CC(C(=O)NC1CC(CF)C1)NC(C1CC(CNC(N)=O)C1)=O 12146,C(=O)(C#CC1(C)COC1)NC(C1CCN(C(=O)CCc2csnn2)CC1)C 12147,N1(C(C(CC)OC)=O)CCC(C(N2CC(C(C)C)C2)=O)C1(C)C 12148,CC(C)(C)C#CC(=O)NCC1CCCCC1NC(=O)C(F)CC1CCCCC1 12149,c1(OC)ccc(NC(=O)NC2CCN(CC3CC3)C2C)c(C(N)=O)c1 12150,c1(C(N(C(CN(C(Cc2cncc(C)c2)=O)C)C)C)=O)cnc2c(c1)nnn2C 12151,CC1CCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)CCN1C(C1CCCOC1)=O 12152,C(C(C)C(F)F)NC(C(c1ccco1)NC(C(C)=C(C)C)=O)=O 12153,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12154,Cc1c(C(=O)NC2C=CCN(C(=O)C=CC3CCOC3)C2)[nH]c2c1CCCC2 12155,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(CC(C)C)n2)=O)CC1CO 12156,c1(C(=O)NCCCN(C(=O)COC2CCC2)CCC)cc2n(n1)CCCNC2=O 12157,CC(CF)C(=O)NC(CNC(c1ncc(C(F)F)s1)=O)C1CCC1 12158,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2c2ccsc2)C1)C 12159,CC1CC2CN(C(C3CCC(C4CC4)N3C(=O)CN3CCCCC3)=O)CCN2C1 12160,Cc1nc(=NCc2cc(NC(=O)Cc3csc(NC=O)n3)ccn2)[nH]cc1[N+](=O)[O-] 12161,c1(OCC)nc(NC(C(C)NC(c2cc(C3CC3)cs2)=O)C(C)C)ncc1Cl 12162,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(O)c3)=O)C2)CCn2ccnc2C1 12163,Cc1cnc2n1CCC(C(=O)NC1(CNC(=O)C=Cc3cccc(Cl)c3)CC1)C2 12164,CC(CC(=O)NC1(CO)CN(C(=O)C(C2CCCCC2)N(C)C)C1)P(C)(C)=O 12165,[N-]=[N+]=NC1CCN(C(c2coc(CNC(=O)C(=O)NCCF)c2)=O)CC1O 12166,c1(OCC=C)ccc(CNc2ccc(C(=O)O)c(C)c2)cc1OCC 12167,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(C(=O)CN3CCCC3=O)C2)C1 12168,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12169,C(=O)(C(F)C1=CCCCC1)Nc1cc(-c2c(N(CC)CC)ccc(F)c2F)[nH]n1 12170,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(C)N(C(=O)C(N)=O)CC1C 12171,C1(C(=O)NC(Cc2cc(C)on2)=O)CCC(NCc2ccccc2Br)CC1 12172,C1(NC(c2cccc(CNC(C34CSCC3C4)=O)n2)=O)CC2CCCC2C1 12173,C1(NC(C(C)C)=O)CCCCCC1C(=O)NCCC(=O)N(C)C 12174,C=C(Br)CC(C)(C)C(=O)NC1CCC(NC(C2CSC2)=O)C1 12175,C1(NC(C2CC(C)=NO2)=O)CCC(N(C(=O)CSC(C)C(=O)O)CC)CC1 12176,C1(C(=O)NCC2CCN(C(C3CCN(C(C(C)C)=O)CC3)=O)C2)CCC2(CC1)CC2 12177,N1(C(CCSCCCC)=O)CCCCC1C1(NC(=O)CNC(=O)OC)CC1 12178,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12179,c1(OC)nsc(OC)c1C(=O)NCCC(C)NC(c1ccc(OCF)cc1)=O 12180,c1(C(N2CC3(CCCCN3C(=O)Cc3nc[nH]n3)C2)=O)cc2cc(F)cc(F)c2[nH]1 12181,C(=O)(N=c1cc2ccccn2[nH]1)C1N(C(Cc2c(C)n[nH]c2)=O)CCSC1 12182,C(CCN=C(NCc1ccc(NC(C)=O)cc1)N1CC(C)S(=O)(=O)C(C)C1)OCC 12183,CCC(C)(C)C1C(=O)Oc2cccc1c2.C1C(=O)O1.C1(=O)CO1.C(C(C)C)OCC 12184,c1(C(=O)NCC2CN(C(Cc3nc(C)[nH]n3)=O)C2)ccc(F)c(C(F)(F)F)c1F 12185,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12186,C1(C(N2C(C)C(NC(c3cc(O)nn3C)=O)CCC2)=O)CCc2cnn(C)c2C1 12187,N1(C(C(C)N(CCOC)C)=O)CCOCC1CNC(=O)COCc1ccc(C)cc1 12188,C(CC(F)F)(C(=O)N(C)CCN1CCOC1=O)N(C(c1cc(C)[nH]c1)=O)C 12189,c1(C(N(C2CCN(C(CN3CCC(OC)C3)=O)C2)CCO)=O)ncc(N)cc1C 12190,N1(C(C2N(C(C3CC(CCC)C3)=O)CC=C2)=O)CCC(F)(C(N)=O)CC1 12191,Cc1oc(Cl)nc1CNC(=O)C(C)N(C(=O)Cc1ccccc1O)C 12192,C12(N(C3CCCCC3)C(N(C3CC(F)(F)C3)CC)=O)CCCC1C2(F)F 12193,C1(C)(NC(=O)N(C(C)CCS(C)=O)C(C)(C)C)CCC(C(=O)OC)O1 12194,C12COCCN1C2.n1(CC)c(C)ccc1-c1nc(CCCO)nn1-c1cnn(C)c1 12195,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12196,C(=O)(C1=C(C)CCCC1(C)C)N1CC(CNC(C(CCCC)(C)F)=O)OCCC1 12197,c1(C(NOC)=O)ccc(CCSc2sc(SC)nc2C)cc1 12198,C1(NC(c2c(CC)nn(C)c2)=O)C2CC3CN(C(=O)CC4CNC(=O)C4)C1C3C2 12199,c1(CC)cccc(CC)c1C(=O)NCCC(C)(C)NC(C1C2COCC12)=O 12200,N1(C(C2(C)CC=CC2)=O)CCOC(C(=O)NOCC2CCOC2)CC1 12201,C(C(=O)N(CCC(=O)N1CCCC1CC1CC1)OC)(C1CCC1)OC 12202,Cc1cc(C(=O)NC(C(N2CCCC2CF)=O)C2CC2)sc1C 12203,C1(NC(c2cc(C3CC3)cs2)=O)CCCN(C(=O)CC2CCCC(O)C2)CC1 12204,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(C(F)F)s2)CC(O)C1 12205,N1(C(c2cc(CC(C)C)on2)=O)CCCC(NC(C2(Cl)CC2)=O)C(F)C1 12206,Cc1ccc(OCCCNC(=O)Cn2nnc(C3CC3)n2)c(C)c1 12207,c1(C(CNC(C(CC)C)=O)NC(c2cn(C(C)C)nn2)=O)ccc(F)cc1F 12208,C1(C(=O)NC(CC)COC)CCOCCN1C(c1cnccc1OC)=O 12209,C1(CNC(COC)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12210,N1(C(C2(CC)CCCC2)=O)CCOC(C)(CNC(=O)CC2CC(=O)NC2=O)C1 12211,Cn1c(-c2ccccc2)nnc1C1CCCN(C(c2ccncc2Cl)=O)C1 12212,N1(C(C(=O)N(C)Cc2cccc(Cl)c2F)=O)CCC(O)C(F)(F)C1 12213,CCCCC(C(=O)NC1CC1C(C)(C)C)NC(c1cnc(C)[nH]c1=N)=O 12214,S(=O)(=O)(c1cnc(NCCCc2ccncc2)cc1C)NC1CC(CC)OCC1 12215,CCCC(CC)C(=O)NCC1(OC)CN(C(c2cc(O)ncc2Br)=O)C1 12216,c1(C(N(CCN(C)C)CCSC2CCCC2)=O)ccc(N2CCCS2(=O)=O)cc1 12217,Cc1cc(C(=O)NC(CNC(C2(CC3CC3)CC2)=O)C2CC2)n[nH]1 12218,N1(C(CN2CCC(OC)C2)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12219,CC1(CNC(c2cnccn2)=O)CCN(C(c2c(Br)cnn2C2CCC2)=O)C1 12220,S(=O)(=O)(c1ccc2[nH]c(=NCCCF)sc2c1)N1CCN(C)CC1 12221,C1(CNC(C=CCC)=O)CCC2(CN(C(=O)C(c3ccccc3)SC)C2)O1 12222,C1(NC(CC(CC)C)=O)CC12CCC(NC(c1cccnc1SC(F)F)=O)CC2 12223,c1(COC(C)(C)C)cccc2cccnc12.N12CC3C(C1)N3C(=O)C2N(C)C 12224,c1(C(N2CC(O)(C3CCC3)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 12225,c1(NC(=O)NOCC(c2cc(Br)no2)n2ccnn2)ccccc1 12226,N1(C(C2CC(C)(CC)C2)=O)CCCC(C(C)(O)CNC(c2ccc(C#N)o2)=O)C1 12227,N1(C(C=C(C)C(C)C)=O)CCN2C(=O)C(NC(c3cnccn3)=O)CC2C1 12228,c1(CC)nc(C)n(C)c1C(=O)NCCOCCNC(=O)CC1CCC2(CCC2)O1 12229,C1(COC)CN(C(=O)COC2CCCOC2)CCN1C(c1cnn(CCF)c1)=O 12230,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12231,c1(SC)nc(NC23CCC(CC2CNC(=O)CCCCCF)C3)cc(C(F)F)n1 12232,C(CCC(=O)NC(C)CN(C)C(c1cc(-c2cccnc2)[nH]n1)=O)N(C(C)C)C 12233,N1(C(C(C)COc2ccccc2)=O)CCC(C)(C)C1C(=O)NCc1ccccn1 12234,C1(CCNC(CC2(OC)CC2)=O)(NC(=O)CCCc2sccc2C)CCCC1 12235,N1(CCC(=O)NCC2(CN(C(C(CC)C)=O)C)CC2)CCCCC1C 12236,N#Cc1ccccc1NC(=O)C(=O)NC1CCCCC1NCCOC1CCOCC1 12237,C(=O)(C1SCc2cccnc21)N1C(C)CN(C(=O)CSc2n[nH]c(O)n2)CCC1 12238,N1(C(C2(SC)CCC2)=O)CCC(O)(C(C)NC(=O)COC2CC(F)(F)C2)CC1 12239,C(c1cc2ccccc2o1)=CC(=O)NCC1(CCNC(CC=CC)=O)CC1 12240,c1(-c2cn(C3(C(=O)NC(C(=O)OC(C)(C)C)F)CC3)nn2)ccc(F)c(F)c1 12241,CC1CCOCC1C(=O)NCC1(Sc2cccc(F)c2)CCCCC1 12242,c1(NC(=O)NC(C2CCC(=O)NC2)CC)cccc(NC(=O)C(=O)OC(C)=O)c1C 12243,c1(C(=O)NCCNC(c2c(C)[nH]cc2)=O)cc(N)c(Cl)cn1.C12=CC=C(C=C1)C2 12244,CCC(C(=O)N(CCNC(C1CC1c1ccccc1F)=O)C(C)C)C(C)(F)F 12245,C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(C(=O)OC)(C)CO)C1 12246,c1(C(=O)NC2CCN(C(=O)C3=COCCC3)CC2O)cnc2ccc(F)cc2c1 12247,c1(C(N(C2CCN(C(c3c(CC)nc[nH]3)=O)C2)C)=O)nc2cnccc2s1 12248,CCC(C)(C)C(O)C(=O)NCC1(O)CCOCC1.C1(C(=O)NC)CCC(C)(C)CO1 12249,CCC(C)C(O)C(=O)N1CCCC(C)(C(=O)NC2CC(O)(CO)C2)C1 12250,c1(C(=O)NCC=CCNC(C2C(F)(F)C23CC3)=O)cc2cc(F)c(F)cc2[nH]1 12251,C1(C(=O)NCC2(C#C)CCC2)CN(C(c2cncc(OC)c2)=O)CC1F 12252,CCC(CC)C(=O)N(C(c1ccccc1)CNC(=O)CCOc1cccnc1)C 12253,C(=O)(C#CC1CCOC1)NCC=C(C(N1CCC(CC#C)CC1)=O)C 12254,c1(C(=O)NCC(CCNC(c2ccc(C)c(N)n2)=O)O)cc([N+](=O)[O-])ccc1N 12255,CCC(CC(F)F)C(=O)N1CC(C(C)(C)C)CC(CNC(=O)CC(C)(C)SC)C1 12256,N1(C(C=C(C)C2CC2)=O)CC(CNC(=O)C=CCN2CCCC2)C(O)C1 12257,N1(C(CC2(NC(c3c(C)ncs3)=O)CCC2)=O)CCN2C(=O)COCC2C1 12258,c1(C(=O)NC2CCN(C(c3c(C)ccnc3C)=O)CC2O)cccc2c1COC2 12259,c1(C(=O)NC2C(CNC(C(CCC)CC)=O)CC2)cc(C)c(Br)c(C)c1 12260,C(=O)(C(F)C(F)(F)F)N.C1(NC(=O)CC2CCC(CO)CC2)(CO)CCOCC1 12261,C1(N(C(CC2(C=C)CC2)=O)C)CC2CC1N(C(c1csnc1C)=O)C2 12262,c1(CN2CC(NC(=O)CSc3ncccn3)C(F)(F)C2)ccc2nccn2c1 12263,C1(C2CCN(C(=O)C(=C3CCCCC3)F)CC2)(NC(C2CC2(Cl)Cl)=O)CCC1 12264,N#CC1(C(=O)NC2CCCC2NC(c2cc(C3CC3)ncn2)=O)CCSCC1 12265,N1(C(CC2CCC(C#N)C2)=O)CC2(CCC(NC(=O)C(F)C3CCCC3)CC2)C1 12266,c1(C(=O)NC(CC)CNC(=O)CC2(C(=O)OC)CC2)cc([N+](=O)[O-])n[nH]1 12267,N1(C(C(CCCC)O)=O)Cc2ccccc2CC1C(=O)Nc1cnc(C)c(Cl)c1 12268,N1(C(C(F)=CCC)=O)CC2(CCC2)CC1CNC(c1c(C)nn(C(C)C)c1C)=O 12269,C1(C(N(C)CC2CCCN(C(C(C)(C3CC3)OC)=O)C2)=O)CC2CCC(C1)S2 12270,C1(CN(C(C2(CC=C)CN(C(=O)CCc3cccs3)C2)=O)C)CCCCC1O 12271,C1(OC)CC2CC(NC(=O)C(CCNC(C3C4CN(C)CC34)=O)OC)CC12 12272,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CCC2CC2)C2CC2)C)CC1 12273,N1(C(C#CC(C)C)=O)CCC(C)C(NC(c2cc(C(N)=O)ccc2F)=O)C1 12274,O=C(CC(F)(F)C(F)(F)F)NC1CCCCC1NC(C1(c2ncco2)CC1)=O 12275,C#Cc1ccc(OC(C)C(N2CCN(C(C)=O)C(C(F)F)C2)=O)c(F)c1Cl 12276,C=CC1(C(=O)NC(C)CN2CCCC2)CCN(C(C2OCCC2(C)C)=O)CC1 12277,N1(C(Cc2cccc(C#C)c2)=O)CCN(C(c2ccc(C)c(C)c2)=O)C2CCCC12 12278,N1(C(COCCOC)=O)CCC2(CC1)OCCC2NC(c1cc(C)nc(C)c1)=O 12279,C1(C(N2CCC(CNC(C(c3ccnn3C)C)=O)(CO)C2)=O)CC2(CC(=O)C2)C1 12280,c1(C(=O)NC(C)CNC(C2(C#N)CCCO2)=O)cc(N)nc(Cl)c1 12281,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(C)CC2)C1 12282,C1(NC(c2ccn(CCC)n2)=O)CCC12CN(C(=O)CCOCC)C2 12283,CCCC(C(=O)NC(C)CC(C)CO)NC(=O)CC1(N(C)C)CCC1 12284,C(=O)(C1=CCCC1C)NC1C(CNC(C2CCCN(C(CC)=O)C2)=O)COC1 12285,C12(NC(c3cc(C)c(Cl)cn3)=O)CCCC1CN(C(=O)CSC1CCCCC1)C2 12286,CCC(CC)C(C)C(=O)N1CCC(NC(c2cncc(Cl)c2)=O)CC1C 12287,N1(C(C(C)=C2CCC2)=O)CCN(CC(=O)N(CC(F)F)C)CC1 12288,N1(C(C(C2CCC(=O)N2)C)=O)CC(C)(NC(C2(CC3CCC3)CC2)=O)C1 12289,N1(CC(=O)NC(c2ccn(C)n2)CC)CCN(C(=O)CC2OCCO2)CC1 12290,N1(C(C2N(C(c3cc(C)c(O)cc3)=O)CC2)=O)CCc2cc(C#N)ccc2C1 12291,c1(SC(c2cnc(C)s2)c2nccn2C)ccc(C(=O)O)cc1 12292,Cc1nc(Br)ccc1C(=O)NCc1ccc(NC(=O)C(C)C)cc1 12293,N1(C(CCC(=C)Cl)=O)CCC(C2CCN(C(c3n[nH]c4c3CCOC4)=O)C2)C1 12294,c1(NCC(N2CCC(CC3CC3)CC2)=O)cc(-n2ccnc2)ccc1[N+](=O)[O-] 12295,N1(C(CC=C(C)C)=O)CCN(C(=O)COCc2ccc(C)cc2)C(C2CC2)C1 12296,C=C(C)CN=C(NCC1CCCCCC1)NCC1CCC(C2CCC2)O1 12297,n1(CC(=O)NC2CC2CNc2nccc(C(F)(F)F)n2)ncc2ncccc12 12298,C(=O)(C(CC(C)(C)C)OC)NCCN(C(=O)CC1CC1(C)C)CCC 12299,CC1=CCC(C(=O)N(C)CC2(O)CCN(C(c3cncc(N)c3)=O)C2)CC1 12300,C1(NC(CC=C(C)C)=O)CCCCCCC1NC(c1cc(C)nn1C)=O 12301,c1(C(N(C(CC)COC)C)=O)coc2c1CN(C(=O)CCC1CCOC1)C2 12302,C(=O)(C(O)C(C(C)C)OCC)N(CCNC(C(CC)N(C)C)=O)C 12303,C(N=c1[nH]c(N2CCCC(C(N)=O)(N(C)C)C2)nc(=N)[nH]1)C1(N(C)C)CCC1 12304,C1(F)(CC2CCC(C(N3C(C)(CO)CCC3)=O)CC2)CC2CCC1C2 12305,C1(N(C(c2c(C)nccc2)=O)C)CN(C(C2CC3C=CC2C3)=O)CC1(C)C 12306,c1(N2C(C(=O)NCc3ccc(C(=O)OCC)[nH]3)CNCC2)nc(C)cc(C)n1 12307,Cc1ccsc1CC(=O)NC(CNC(=O)COC(F)F)C(C)C 12308,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12309,COn1cnc(C)c1C(=O)NC1CN(C(=O)COCC2CCOC2)CC1F 12310,c1(C(=O)NCCCC2N(C(C(C=C)(C)C)=O)CCCC2)ccc2cnccc2c1 12311,C(CCC(=O)NCC(C)N(C)C(c1cnn(C2CC2(F)F)c1)=O)OCCOCC 12312,Cc1cnn(C)c1C(=O)NCCCC1CN(C(c2ccccc2O)=O)CCO1 12313,C1(CNC(C2N(Cc3cc(C(=O)OC)nn3C)CC2)=O)CC12CCc1ccccc12 12314,N1(C(c2cc(C)c(C)s2)=O)CC(C(N2CCCCCC2)=O)CC12CCC2 12315,N1(C(N2C(C)(C(=O)Nc3cccc(C(N)=O)c3)CC2)=O)CCCC(C)(O)CC1 12316,c1(C(=O)NCC2CN(C(C=COCC)=O)C(C)(C)C2)c[nH]c2ccccc12 12317,C(=O)(C1=NNC(=O)C1)NC(CCCCNC(Cn1c(C)ncc1)=O)C 12318,O=C(C1=CCCO1)NCC1CCN1C(C1CCCC(c2ccccc2)C1)=O 12319,CC1CC(NC(=O)CCc2cccc(O)n2)CN1C(c1cscc1Cl)=O 12320,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12321,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(F)(F)F)C2)=O)C1 12322,N1(C(CN=[N+]=[N-])=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 12323,C(=O)(CCCC(=O)NCc1csc(CNC(C2CCC(C)(C)CC2)=O)n1)NCC 12324,c1(CC)ccccc1C(=O)NCCC(N1CCC(C)C1CNC(=O)CCSC)=O 12325,N1(C(C2(SC)CCC2)=O)C2CCC(C2)C1CNC(C1CN(C)CC1C)=O 12326,C1(CNC(C(CC(C)C)F)=O)CC2(CC2)S(=O)(=O)N1 12327,Cc1ccc(C=C(C#N)C(N2CCC3(NC(=O)Cc4sccc4C)CC3C2)=O)cc1 12328,C(=O)(C1CCOc2c(F)cccc21)NCn1cc(C(c2c[nH]nc2C2CC2)C)nn1 12329,C1(NC(COCCC#C)=O)CCCOC12CCN(C(C1(O)CC1(C)C)=O)CC2 12330,Cc1cccc2c1c(CNC(=O)Cc1csc(NC(=O)C(O)C(C)C)n1)cn2C 12331,N1(CCN(C(c2n(CCC)ncc2)=O)C(C)C)CCN(c2ccc(Cl)nn2)CC1 12332,c1(C(N(C2CCN(C(=O)C=CCOCc3ccccc3)C2)C)=O)c(N)cnn1C 12333,c1(C(N(CCC(C)NC(c2ccc([N+](=O)[O-])cc2)=O)C)=O)cc2c(ccn2C)[nH]1 12334,C(=O)(CCCCC(C)C)NC1C2(CN(C(C3CCC(CC)CC3)=O)C2)CC1 12335,C(N=c1nc2c(ncn2C)c(NCc2ccoc2C(F)(F)F)[nH]1)C1CC(=C)C1 12336,c1(CC(=O)NCC2N(C(CCC(N)=O)=O)CCCC2)cccc(Cl)c1F 12337,Cn1cc(C(=O)C(N2CCC(OCC(=O)NCc3cccnc3)C2)=O)cn1 12338,c1(OC)cc(C)c2cc(-c3cnccc3N3CCCC3)[nH]c2c1 12339,CC(C)C(C(C)NC(c1c[nH]nc1-c1ccncc1)=O)NC(=O)CSCC(N)=O 12340,N1(c2snc(C(C)(C)C)n2)CC2(C1)SCCC2NC(C1CC(F)CN1C)=O 12341,CC1NC(=O)C2=C1N(CCF)C(=O)NC2c1ccc2c(c1)C(N)CCC2 12342,C1(N(C)C)CCC(CNC(=NC)NCCCNC(C)=O)CC1 12343,C12(C(=O)NC3CCC(C(=O)NC)CC3)CCN(C(=O)C(C)(C)SC)CC1C2 12344,c1(CN(C(CN(C)CCc2ccccc2)=O)C(C2(O)CC2)=O)cc(F)cc(Cl)c1 12345,C=CCN=C(NCCNC(=O)N(C)C)N1CCC(C2CC2)CC1 12346,N#CC1(C(=O)NC(C2CCOC2)CNC(C2CC(F)(F)C2)=O)CC2(CCC2)C1 12347,Cc1c(C(N2CCC(C)(NC(=O)CN3CCC3C)C2)=O)[nH]c2ccccc12 12348,Cc1cnc(C=CC(=O)NCC2CCC(NC(c3sc(C)nc3C)=O)C2)[nH]1 12349,N1(C(c2ccnc(F)c2)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12350,Cn1nc(C(N2CC(C)(C)CC2C(N2CCC(N=[N+]=[N-])C2)=O)=O)ccc1=O 12351,C12CC13CCN(CC3)C2.CC1CC(C(=O)OC(C)(C)C)CCN1C(=O)OC(C)C 12352,c1(C(=O)NC2C(O)CCN(C(Cc3c(C)nccc3)=O)C2)ccc2n[nH]cc2c1 12353,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N(C)C2)=O)C3)c1[N+](=O)[O-] 12354,CP(C)(=O)c1ccnc(C(N2CCCN(C(C3CCC(=O)NC3)=O)CCC2)=O)c1 12355,c1(C(N2C(CNC(c3cnc(C)s3)=O)CC(O)C2)=O)cccc(CO)c1C 12356,C1(NC(CCOCCOCC)=O)CCCC1NC(=O)CCC1CCN(C)C1 12357,Cn1cc(C(N2CC3CC3(CNC(=O)C=C3CCC(C(F)F)CC3)C2)=O)n(C)c1=O 12358,CCC(COC)C(=O)N(C)CC=CC(=O)N(CC)Cc1ccc(O)cn1 12359,c1(C(C(=O)NCC(c2ccccc2)N(C)C(c2cnco2)=O)O)ccccc1Cl 12360,N1(C(COc2ccc(C)cc2)=O)CC2(CCC2NC2CCN2C2CCCC2)C1 12361,CC(=O)CCCC(=O)NC(C1(CNC(=O)Cc2ccnc(O)c2Br)CC1)C 12362,N1(C(=O)COC2CCCCC2)CCC(CNC(C2CC2Cl)=O)C12CCC2 12363,C12(C(=O)NCC(CNC(C3(CC(F)F)CCC3)=O)OC)CC(C(C)C)(C1)C2 12364,C1(O)(C(C)NC(=O)CCC2(O)CCC2)CCN(C(C2(CF)CC2(F)F)=O)C1 12365,c12cccc(c1)C(=O)NCC21CCC1.N1(C(C(C)C)=O)CCC(c2nc[nH]n2)C1 12366,C1(C2CCCO2)CNC(=O)O1.CC1CNC(=O)NN1C 12367,CC#CCC(CO)NC(C1CC(NC(C2CN(C)CC2C)=O)C1)=O 12368,C(=O)(C(F)C(=O)NC1CN(C(=O)Cc2nncn2C(C)C)CC1C)OCC 12369,C(=O)(N=c1[nH]onc1C#N)Nc1nc(-c2cnc(CCCC)nc2)sc1 12370,N1(C(C2CC(CSC)C2)=O)CCN(C(=O)C#CC(=O)N(C)C)C(C)C1 12371,C1(CCOC)(NC(c2cc(C(C)C)sn2)=O)CCN(C(C2CSCCS2)=O)C1 12372,C1(CC)C(NC(c2ccc(OC)s2)=O)CCCN1C(=O)C=Cc1cnccn1 12373,C=CC1(O)CN(C(=O)C(CCN(C)C)NC(c2ccc(O)nc2)=O)C1 12374,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12375,N1(C(CCNC2CC(N=[N+]=[N-])C(O)C2)=O)CCn2nncc2C1 12376,CC1OC2(CNC(c3occ4c3CCC4)=O)CC1(NC(C1CC13CCOC3)=O)C2 12377,c1(C(N2CC(C)C(CNC(C3(O)CC(F)(F)C3)=O)CC2)=O)ccc2ncccn12 12378,C1(NC(CCN(CCCN(C(=O)C(c2cccnc2)O)C)C)=O)CC1C1CC1 12379,c1(NCC2CC(=O)NC2)ncccc1S(=O)(=O)NC1CCc2ncsc2C1 12380,c1(C(=O)OC)c(OCC2CC(NC(=O)CCOCC(N)=O)C2)cccc1Cl 12381,N1(CCNC(C(CC2CCC2)OC)=O)CCN(C(C2(CC3CC3)CC2)=O)CC1 12382,C=CC1(CC(=O)NC2(CC(C)(C)C)CC2)CN(C(C2CC(C)(C)CO2)=O)C1 12383,C1(COC)CC2CC2N1N1CC(NC(=O)NC(C)(C)C)C(C)C1 12384,C1(C(=O)NCCN(CCOCCO)CC)CCO1.C(=O)(C1=CCOC1)OC 12385,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C(F)=C2CCCC2)C1 12386,c1(C(=O)NCC2N(C(C3C(C)C3)=O)CCC2)ncccc1Br 12387,CC1CCC(C)(C(=O)NCC(F)CNC(=O)C(O)Cc2ccccc2)C1 12388,c1(C(CNC(c2nnsc2C(F)F)=O)NC(c2cc(Cl)c[nH]2)=O)ccccc1F 12389,CC1COCCC1CNC(=O)COC1CC(NC(=O)CC2CCCSC2)C1 12390,c1(NCc2c(C)noc2C)cc(Br)ccc1S(=O)(=O)N1CCOCC2COCC12 12391,C1(NC(Cc2cn(CC)nc2)=O)CC2CCC(C1C)N2C(=O)C(C)S(=O)CC 12392,c1(C(N2CC3C(CNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12393,N1(c2c(Nc3cnn(C)c3C3CC3)cc(Br)cn2)CCCC(C)(C(=O)O)C1 12394,CON(C)C(=O)CN(C)N1CCOC(COOC(F)F)C1 12395,c1(OC)cccc(C(C)NC(=O)NC(C(O)CO)c2ccccc2)n1 12396,CC1CSCCN(C(=O)C(=O)NCc2cnn(C3CCCCC3)c2)C1 12397,CC1CC(CNC(C2(F)CCCOC2)=O)CN1C(=O)CN1CCOC1=O 12398,C(CC(O)C(=O)N1CCC(C)(NC(=O)CCSc2ccccc2F)C1)N(C)C 12399,c1(N2CCC(=CCC)C2)ccnc(NCC(c2ccncc2F)C)n1 12400,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12401,C1(C(N2CC(c3cn(CC(C)O)nn3)(C(=O)N(C)C)C2)=O)CC2C=CC1C2 12402,C1(N(C(CCC)=O)C)CC2CCC(C1)N2C(=O)C(C(CC)CC)N(C)C 12403,CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)CCC2CC2(C)C)CC1O 12404,C(CNC(C1CNC(=O)O1)=O)(CC(=O)NCCN(C)CCF)OC 12405,C(CC(C)(C)C(=O)NCC1CCCC(CNC(c2ccc(Cl)cc2C)=O)C1)OC 12406,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 12407,N12CCC3(CC1)COCC(O3)C2=O.c1(C(=O)NC2(OCC)CC2)cnc[nH]1 12408,C1(NC(c2ccc(CC)cc2O)=O)CC(NC(c2ccoc2)=O)C12CCOCC2 12409,CC1COC2(CCC2)CN1C(C1CC2CC1CC2NC(c1cccn1C)=O)=O 12410,C1(CC(=O)NC(C(=O)OCC=C)(C)C)C2CCCC2N1C(=O)CCc1cnoc1 12411,N1(C(C(C)=C(C)C)=O)CCC2(CC1)CN(C(C1C3COCC13)=O)CC(C)O2 12412,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2ccsc2)=O)C1)NC(=O)OC 12413,C(C(C)(C)CNC(=O)CCc1conc1C)N(C(C1(OC(C)C)CCC1)=O)CC 12414,c1(-c2ccc(C)cc2)nc(C(=O)Nc2cccc(F)c2C(N)=O)ccc1F 12415,CCC(C)(CNC(C1(CNC(=O)C(c2ccnn2C)O)CC2(CC2)C1)=O)C(N)=O 12416,O=C1CN(CC(N2CCC3CC3C2)=O)CCN1.C(CS)O 12417,CC(C)C(O)C(C)C(=O)N1CC(=CCNC(=O)CN2CCC2)C1 12418,Cn1nc(C(=O)NCC2CC(NC(=O)C(c3ccc(Cl)cc3)(C)C)C2)ccc1=O 12419,c1(CC)n[nH]cc1C(=O)NC(C1CCN(C(=O)C(O)C2CCC2)C1)C 12420,Cc1cccc(Cl)c1-n1cc(C2(O)CCN(C(=O)C(C)(F)CN)C2)nn1 12421,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(C1)CN(C(=O)Cc1ccc(Cl)s1)C2 12422,C=CCC(C(=O)NCC1COCC1NC(=O)C(C(C)(C)C)C1CC1)C(C)C 12423,CC1CC(NC(=O)C(c2cccc(Cl)c2)O)CCN1C(C1CN2CCC1CC2)=O 12424,C1(C)(CNC(CS(=O)(=O)NCC)=O)CC(F)(F)CN1C(c1cc(C(C)=O)on1)=O 12425,c1(C(=O)NCC2C(C)(C)N(C(c3ccc(O)nn3)=O)CC2)ccnc2ccnn12 12426,c1(CN(C)CC2CCCN2C(C2CCC(=O)N2C)=O)cccc2cc[nH]c12 12427,c1(CCC(N2C(CNC(Cc3c(C)ccs3)=O)CC2)=O)ccccc1C(N)=O 12428,CC1=C(CNC(=O)C(c2ccco2)NC(c2cccnc2)=O)CCCC1 12429,C1(C2CCN(C(=O)Cc3ccc(F)cc3)C2)(NC(=O)Cc2ccsc2Cl)CC1 12430,CC(C)CC(Cc1ccccc1)C(=O)N1CCCC1CC1CCN(C(=O)CO)C1 12431,C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(=O)CC2C=CCC2)C1 12432,c1(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CC2)cc(F)c(C)cc1N 12433,C1(C)(NC(=O)OC(C)(C)C)CCCC(NCC2CCN(C3CCC3)CC2)C1 12434,N1(C(COCCCN(C)C)=O)CCC2(CC(NC(=O)CSc3ccc(F)cc3)C2)C1 12435,N1(C(CCC(=O)NCC)=O)CCC(CNC(=O)Cc2cnc(C)o2)(COC)CC1 12436,c1(OC)c(C)cc(C(=O)NC(C)C(C)NC(c2cccc(CCO)c2)=O)cc1C 12437,CC1CCc2[nH]c(C(=O)NCCCCC(CO)NC(=O)C(C)(C)F)cc2C1 12438,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(=O)CN(C1CCCC1)C)C2 12439,C1(CC)CN(C)CCCN1C(C1COCC1NC(=O)C(F)C(C)(F)F)=O 12440,CC(C)CC(=O)NCC(=O)NC(c1ccccc1)CNC(=O)CSC(F)(F)F 12441,Cc1cc(C(=O)NCCCCC2CCC2)n2ncc(NC(=O)C3=CCCC3)c2n1 12442,C1(C(=O)NCC(C2CCCC2)C)CC2C=CC1N(C(=O)CC1CC(F)C1)C2 12443,C1(C(N(CCNC(=O)CSC)CC)=O)CCn2ncnc2C1 12444,N1(C(CCNC(C2=C(C)CCOC2)=O)=O)CCCC2(CCC2)C1 12445,c1(SC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12446,c1(-c2cn(C3CCN(C(=O)C(O)C4CN(C5CC5)C4)C3)nn2)ccccc1Cl 12447,C(=O)(C1CCc2cc(F)ccc21)N1CCC(CN(C(C2=NOC(C)C2)=O)C)CC1 12448,N1(C(=O)NC(C)C=Cc2cn(C)nn2)CCCC(C)(N(C)C)C1 12449,N1(C(CCS(=O)(=O)N(C)C)=O)CC2(C1)CN(C(C1(C)CCC(=O)N1)=O)CC2CO 12450,C1(NC(C2C3COCC23)=O)CN(C(=O)C=CCF)C2(CCC2)C1 12451,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12452,C1(NC(CC2(CC)CC2)=O)CN(C(=O)Cn2nccn2)CC1SC 12453,c1(OC)c(Cl)cc(CN2CC(NC(c3cc(C)ccc3I)=O)C(O)C2)cc1Cl 12454,N1(C(C=C(C)C(=O)O)=O)CC(NCc2ccc(N(C)C)cc2)CC(C)C1 12455,C(=O)(C(C)(C)C)NC(C)C(=O)NC1CC1NC(=O)C=Cc1ccco1 12456,c1(N(C)Cc2ccns2)ccc(S(=O)(=O)N2CCC3(CCOC3)C2)cc1Cl 12457,CC1CC(NC(=O)CC=Cc2ccc(F)cc2)CCN1C(=O)C1=CSCS1 12458,C(c1ccc(C)c(C)c1)=CC(=O)NC1CCCC(NC(CC=C=C)=O)C1 12459,N1(CC(=O)NCC(=O)NCC(C2CCOC2)OCC)CCCNC1=O 12460,c1(OC)ccc([N+](=O)[O-])c(C(=O)NC2CC(NC(=O)COc3csc(C)n3)C2)c1 12461,CC(CCNC(=O)CC1CCCC(C)(C)O1)N=c1[nH]cnc2cnccc12 12462,N1(C(CCN(C)CC)=O)CCCCC(CO)C1.c1(C2C(=O)N2)ccccc1 12463,CCCCCCCCC(=O)NC1CC1NC(c1ccc(C(C)(C)C)s1)=O 12464,C(=O)(C1=C(Cl)CCC1)N.c1(N)cccnc1CO.C12(CC1)C(C)NC2=O 12465,c1(SCC)ccccc1CC(N1CCC(NC(C2(C)CCC(C)C2)=O)C1)=O 12466,C1(C(=O)NCCCCCCF)C2CCN(C(c3cncc(F)c3)=O)CC12 12467,N1(C(CCSc2ccc(C)cc2)=O)CCC2CCN(C(=O)Cc3ccco3)CC12 12468,n1(CCCC)nnnc1C(c1ncc(-c2ccccc2)[nH]1)NCCC=C(C)CC 12469,N1(C(c2c(CCC)n[nH]c2)=O)CC(CNC(c2ccn(CCF)n2)=O)CC1(C)C 12470,c1(N(C)C(C2CCN(C(c3nn(C)cc3Cl)=O)CC2)=O)cc(Cl)ccn1 12471,N1(C(C(CC)SC)=O)CCC(CNC(c2cc(F)cc(F)c2OC)=O)C(F)(F)C1 12472,c1(COC(Cc2cc(C)nn2C)=O)c(C)nn(C)c1Cl 12473,c1(OC(C)C(=O)N2CC(CNC(C3CSC(C(F)(F)F)S3)=O)C2)ccc(F)nc1 12474,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cn2ccnn2)C(CO)CC1 12475,c1(C(=O)NCC2(C(=O)NCc3ccc(C)c(F)c3)CC2)cc2cc[nH]c2cn1 12476,C1(C(N(C)Cc2c(CNC(CSC)=O)cccc2)=O)CCOCC1(C)C 12477,C1(NC(c2cc(C)[nH]c2C)=O)CC2CN(C(C34CC(CC(F)F)(C3)C4)=O)CC2C1 12478,c1(NCCC2N(C(CN(CCC)C)=O)CCCC2C)nc2cc(C)ccc2o1 12479,CC(C)C(C)(C(N)=O)NC(C1CC2CC1CC2NC(=O)CN(C)C(C)C)=O 12480,C1(OC)CC(NC(=O)C=CBr)CN(C(=O)CC2CCSCC2)C1 12481,C(=O)(CCCC(=O)Nc1nccs1)NC1C(CNC(C2CC=CC2)=O)CCC1 12482,Cc1nn(C)cc1CNC(C1CCC(C(=O)NC2CCC(N)CC2)CC1)=O 12483,CC1(C(=O)NCC2CC(NC(c3cccc(CO)c3)=O)C2)CC2CC2C1 12484,Cc1ccc(CC(=O)N(C(=O)C(C)(C)c2ccns2)C)s1.C1CN1C(C)C 12485,N1(C(CCc2c(C)cccn2)=O)CCC(CNC(C2CCCOC2)=O)C(C)C1 12486,C=CCC(CC(C)C)C(=O)NCCCC(O)C(N1CC(CO)CC(C)(C)C1)=O 12487,C#Cc1ccc(C(=O)NCCC2(NC(c3cn(C)nc3C#N)=O)CCC2)nc1 12488,N1(C(C(C)(C)C)=O)CCCC(C)(C(=O)NC2CC2(C)C)C1 12489,C(C1=NOC2CN(C(=O)Cc3cccc4c3CCC4)CC12)NC(CC(=C)C)=O 12490,CC1CN(C(=O)C(C)(C)CNC(=O)C2=COCC2)CCS1=O 12491,C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(C(=O)NC(CC)C(C)(F)F)F)C1 12492,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12493,N1(C(c2ccc(C)nc2C(C)C)=O)CCOC2(CCN(C(C3CC3F)=O)CC2)C1 12494,C1(C(=O)NCC2CC(NC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12495,C1(NC(=O)C=C2CCOCC2)CC2CC1CN(C(C1CCCCC1)=O)C2 12496,CC1(C#N)CCN(C(=O)CCC2(NCCC3(C(=O)N)CC3)CCCC2)C1 12497,N1(C(c2cn(CC(C)(C)O)nc2)=O)CCCCCC1N=c1ccc(C#N)n[nH]1 12498,CC1CN(C(C2(c3cccs3)CCCC2)=O)CC1NC(C1(C)CC1(C)C)=O 12499,CON1CCC(C(=O)NC2CC(CC(=O)N(C3CCC3)C)C2(C)C)CC1 12500,C1(NC(CCNC(=O)NC)=O)COC2C(NC(=O)Cc3ccc(F)cc3Cl)COC12 12501,C(=O)(C(C)(C)C(C)O)NCCn1cc(C(N(CCCC)CC(C)OC)=O)nn1 12502,c1(CSCCC)ccc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)cc1 12503,N1(C(C(C2(O)CCC2)NC(CCCSC)=O)=O)CC2CCC(C1)C2C#N 12504,C#CCC(C(=O)NCCCSC)N(C(=O)C(=Cc1cn[nH]c1)C)C 12505,C1(CSC)CCN(C(=O)CCOC2CN(C(=O)C(C)CN(C)C)C2)C1 12506,CN1CCN(C(c2sccc2COCC(=O)OC2CCCC2)=O)C(C2CC2)C1 12507,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(C(CC)(CC)CC)=O)C 12508,C1(c2nnnn2CCSc2ccccc2)(NCC2(CC)CC2)CCCSC1 12509,c1(C(=O)OC)ccc(OC)c(C)c1N(C(C(C)OC1CCCO1)=O)C1CC1 12510,C1(C)(N(C)C)CCCN(C(=O)C(c2ccnn2C)NC(=O)COC(C)(C)C)C1 12511,N1(c2c(C(=O)OC)n(C)nn2)CCCC(C)(C(=O)NC(C)(CO)C(C)C)C1 12512,CC1CCCC(CC(=O)N(C2CCCN(C(c3cnc(N)cn3)=O)C2)CCO)O1 12513,c1(CN(C(c2ccccc2)C(=O)Nc2ccccc2)CC(C)C)ccncc1 12514,c1(C(=O)NCC(C)NC(C(CC)n2cncn2)=O)cnc(C)n1C 12515,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12516,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(c1ccc(Cl)o1)=O 12517,Cn1cc(C(F)=CC(=O)NCC2C=CCN2C(=O)CC2CCCCO2)cn1 12518,N1(C(C=CCCC)=O)CCCC(C(=O)OCCNC(=O)CC(C)SC)(COC)C1 12519,N#Cc1ccc(C(N2CCC(O)C(O)C2)C(=O)NCC2CCCO2)cc1F 12520,c1(C(N2CCN(C(=O)Nc3cccc(C)n3)C3C2C3)=O)nncc2c1CCCC2 12521,N1(C(C=NOC)=O)C2CCC1CC(NC(c1nc(Cl)sc1C(C)C)=O)C2 12522,c1(CNC(C(C)=CC)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCCCC1)C2 12523,C1(F)(C(=O)NCC(C)NC(c2cc(-c3ccccc3Cl)no2)=O)CCCOC1 12524,C(CCC(=O)NCCC1(C)CN(C(=O)C(n2cc(Cl)cn2)C)C1)NC(C)=O 12525,c1(OC)nc(Cl)ccc1C(N1CCC(NC(c2ncccc2C)=O)CC1C)=O 12526,N1(C(CCCn2cc(CC(C)(C)CO)nn2)=O)CC2CC2(CN2CCOCC2)C1 12527,CCCCCC(CC)C(=O)NCCN(CCSC)C(c1c[nH]c2cccc(C)c12)=O 12528,N1(C(c2cc(OC)n[nH]2)=O)CCC2(C(=O)NCC3CC(N(C)C)C3)CC2C1 12529,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12530,c1(C2(CNC(C(=O)NC)C)CC(=O)C2)ccc(Cl)cc1 12531,C(C(CC(F)(F)F)NC(c1cnn(C)c1)=O)NC(c1cnc(C(C)C)s1)=O 12532,N1(C(C(CC)OC2CCCC2)=O)C2CCC1CC(CNC(=O)C(F)F)C2 12533,C(=O)(N1CCCc2nncn21)C1C2(CCN(C(c3cc(OCC)no3)=O)C2)C1 12534,CC(C)CC(C)(CNC(c1c[nH]ccc1=O)=O)NC(C1CN(C)CC(C)O1)=O 12535,C(N=c1nc2c(c[nH]1)COCC2)C1(NC(c2ccc(C)c(F)n2)=O)CC1 12536,C1(NC(C=C(C)C2CC2)=O)CN(C(C23CCCC(C2)OC3)=O)C2CCCCC12 12537,C(CCS(=O)(=O)c1ccc(F)cc1)NC(=O)NC1CCC(C#C)C1 12538,c1(C(=O)NC2CC(O)C2C(=O)NC2CCCS2)cccc(N2CCCCC2)c1 12539,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1ccnc(S)c1)=O 12540,C1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C2CC2)CCS(=O)(=O)C(C)C1 12541,Cc1nn(CC(=O)NCc2cn(C3CCOCC3)nn2)cc1[N+](=O)[O-] 12542,C1(C(N2CCC(O)(C(C)NC(=O)COC3CC3)C2)=O)CS(=O)(=O)CC(=O)N1 12543,c1(NCC2C(C)CCN(C(=O)C(C)CC3CCCC3)C2)ncnc2cnccc12 12544,C1(NC(=O)C(=O)NCCOc2ccc3ccoc3c2)C2C3CC4C1C1C2CC3C41 12545,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCCc1ncnn1C 12546,C1(C)(CNC(CC=C)=O)CN(C(c2coc(COC)n2)=O)CC1C 12547,N1(C(c2ccn(CC)c2C)=O)CCCC(C2CCN(C(c3c[nH]c(=N)o3)=O)C2)C1 12548,C(=O)(C(F)(F)CCC(=O)N1CCC1CNC(c1cnc2n1CCS2)=O)OC 12549,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1CNC(=O)CC12CCCC1C2 12550,c1(C(N2CCC(C(N3C(CC)CCC3)=O)C2)=O)cccc2c1nc(O)n2C 12551,Cc1csc(C(C)C(=O)NCC2(C(N)=O)CN(C(C3CC34CC4)=O)C2)n1 12552,c1(C(=O)OC(C)C(=O)N2CC(CC3CC3)C2)cc(Br)cs1 12553,N1(C(COCC(=C)C)=O)CCCC2(NC(c3ccc(C(C)C)c(F)c3)=O)CC12 12554,N1(C(CC2(C)N(C(c3cc(CCC)[nH]n3)=O)CC2)=O)CCC(C)(C#N)CC1 12555,C1(c2nc(CC)on2)CCCN(C(=O)CCCn2cccn2)C1.c1c[nH]c(=N)o1 12556,c1(C(N2CC(C)(C(=O)OC)C(C)C2)=O)cc2c(F)ccc(Br)c2[nH]1 12557,c1(C(N2CC(NC(C(F)OC)=O)C(O)C2)=O)sc2[nH]cnc(=O)c2c1C 12558,C1(C(N2C(CCNC(C3(CC)CCC3)=O)CCCC2)=O)CCOC(=O)CC1 12559,Cc1ccn2ncc(C(N3CCN(C(=O)CCC4CC4(F)F)CC3CO)=O)c2n1 12560,N=c1[nH][nH]c2cc(C(N3CC4CC3C4NC(=O)CCc3ncc[nH]3)=O)ccc12 12561,CC(C)(CCCO)NC(C1CSCCN1C(C1CC(F)C(=O)N1)=O)=O 12562,c1(C(N(CCCCCNC(c2ccc(Cl)o2)=O)C)=O)cc2n(n1)CCCNC2=O 12563,C1(C(=O)NCC(=O)NCC(C)NC(=O)OC)CCCC(F)C1 12564,c1(C(=O)NC2CCC(NC(C3(CCC)CC3)=O)C2)ccnc(C2CC2)n1 12565,c1(C(=O)OC)cncc(C(N2CC=CC2CNC(c2ccoc2Cl)=O)=O)c1 12566,CN1CC(NC(=O)CCOCCCNC(C2CCC(C#N)C2)=O)CC1=O 12567,C12(NC(C3OCCN(CC)C3)=O)CC(CNC(=O)CP(C)(C)=O)(C1)OC2C 12568,N1(C(C=C(CCN(C)C)Cl)=O)CC2C(CNC(=O)CNS(=O)(=O)N(C)C)C2C1 12569,C1(C)(C(N(C)Cc2c(C)nsc2)=O)CCCN1C(=O)CC1CCCSC1 12570,C(=O)(N1CCCc2ccnn21)C1N(C(C2(C)C(C)CCC2)=O)CC(C)(C)C1 12571,C(C(=O)NC(C1CCC(CC)O1)=O)(C(C)C)NCC1CCCC12CC2 12572,c1(CC)cc(CC(=O)NCCN(C(=O)CCCc2cncs2)CC)on1 12573,CCCCCCCC1CN(C(=O)CNC(=O)CCCn2cc(C(C)(C)CO)nn2)C1 12574,C12CCN(C1)C(=O)C1(CC1)CN(C)C(=O)N2.CCC(C)OC1COC1 12575,N1(C(C2CNC(=O)N2)=O)CC(NC(=O)COC2CC2)C(c2ccc(F)cc2)C1 12576,C1(C(=O)NCCC(C)NC(=O)CC2(C)CCCC2)CCN(CCO)C(=O)C1 12577,C(C(O)CC(=O)NCC1(C(N)=O)CN(C(=O)CSc2cccc(F)c2)C1)N(C)C 12578,O=C1CCC(CCC(=O)NC2CC2CNC(=O)COc2ccccc2O)CN1 12579,c1(C(=O)NC(CC)CNC(=O)C(CSC)OC)cn(C)nc1-c1ccccn1 12580,Cc1cc(C(N2CC3C(NC(=O)C(O)Cn4cncn4)C3C2)=O)sc1C 12581,N1(S(Cc2cccc(OC)c2)(=O)=O)CCN(C(=O)C(C)C(C)=O)CC(C)(C)C1 12582,c1(C(=O)NC2CN(C(c3cnc(N)nc3)=O)CC(O)C2)nccc2ccsc12.CO 12583,Cc1cc(Cl)c(NC(C2CSCCS2)=O)cc1O 12584,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12585,C1(C(=O)NCc2cn(CCNC(C3(SCC)CC3)=O)nn2)CCCCC1F 12586,CC1C(C)C1(Br)C(=O)NC(CNC(C1(C#N)CCC1)=O)C1CCC1 12587,Nc1c(F)ccc(F)c1C(=O)NCC1CCCC1NC(=O)CN1CCOCC1 12588,C(=O)(CCCCCC#N)NC(COC)CC(=O)N1CCCCC1CF 12589,Cc1cc(Cl)cc(NC(C2CCN(Cc3ccnn3C)CC2O)=O)c1O 12590,C(N=c1[nH]c(NC2CCCn3ccnc32)nc2ccccc12)c1cc(C)ncn1 12591,S(=O)(=O)(c1cnccc1C(=O)Nc1cccc(CCOC)c1)N(CC)CC 12592,c1(C(n2ccnc2)CNC(=O)Nc2sncc2Br)ccccc1 12593,N12CC3CCC1CN3N(Cc1cccc(C)c1)C(c1cncnc1)C2=O.CC 12594,c12cc3cc(Br)cc(c3o1)OC2.n1(C(=O)O)c(=O)ccn(-c2ccccc2)c1=O 12595,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12596,c1(C(N(CC(CC)NC(=O)CCC2CC=C(C)CC2)CC)=O)cccc(C)c1F 12597,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(N(C(=O)CSC(C)(C)C)C)C2C1 12598,c1(C(=O)NCC2CCN(CCOC)C2)c[nH]c(C)c1Cl 12599,CN1CCCC2CN(c3cc(N(CCC(C)(C)C)C)ncn3)CCC12 12600,CCN=c1[nH]cc(C(=O)NCC(C)CN(C(=O)Cn2cc(CO)nn2)C)s1 12601,N1(C(Cn2ccc(C)cc2=O)=O)CCC(C)N(C(=O)Cc2cn[nH]c2)CC1 12602,C(=O)(C1=C(Cl)CCOC1)N1CCCC(C)C1C(=O)NOCCC1CC1 12603,N1(C(c2nn(C)c(O)c2)=O)CCN(C(c2cc(O)ncc2F)=O)C(CC(F)F)C1 12604,c1(C(N(CCCC(=O)NCC(C)N(C)C)C)=O)c(O)cccc1F 12605,c1(C(=O)NC(C)CNC(c2ccc(N)cc2)=O)cc2ccc(O)nc2s1 12606,N1(C(c2cccc(N)c2)=O)CCOCC(F)(CNC(c2cc(Cl)no2)=O)CN1 12607,CCC(CN=c1cc(NCCN2CCCCC2C)nc[nH]1)OC 12608,CC#CCCC(=O)NCc1cnn(C)c1C(=O)NCC1CCOC1 12609,C1(NC(C2CC(CC)C2)=O)CN(C(=O)CCC2CC2)CC1c1ccnn1C 12610,c1(C(N2CC(OC)C(CNC(=O)C(C)C#N)C2)=O)cc2n(n1)CCO2 12611,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(c1cn(C)cn1)=O 12612,c1(NC(CC)=O)ccc(C)c(NC(=O)Nc2ncc(Br)cc2N)c1 12613,C1(COCC(=O)NC2CC2CNC(=O)C2CC2)CC(N2CCCC2)C1 12614,c1(C(=O)NC2CC(NC(CCN(CC)CC)=O)C2)nnc(S)n1C 12615,N1(C(c2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(c1ncsc1C)=O)C2 12616,c1(NC(C2CCCN(C(=O)OCC)C2)=O)cc2ccccc2nc1C(F)F 12617,c1(C(=O)NCCCC(=O)NC(C)CN(C)C(=O)C2CC2)ncn(C)c(=O)c1Br 12618,Cc1cnn2ccc(C(=O)NC3(CNC(c4cn(C)c(C)n4)=O)CC3)nc12 12619,C1(NC(CC2CC(SC)C2)=O)CN(C(c2cc(C)ccc2Cl)=O)C2(CCC2)C1 12620,N1(C(CCP(C)(C)=O)=O)CCC(C2(NC(=O)Cn3cccn3)CC2)C1 12621,C(=O)(C(O)P(C)(C)=O)NCCC(C)NC(c1cncc(C(C)(C)C)c1)=O 12622,N1(C(c2ccc(OC)s2)=O)CC(CO)C2(C1)CN(C(C1(C#N)CCSCC1)=O)C2 12623,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)N(C)Cc1cn(CC)nn1 12624,CC(C)S(=O)(=O)CC(=O)N1CC2(COC(CNC(c3ccon3)=O)C2)C1 12625,c1(C(=O)NC23CC(CNC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12626,C(=O)(C(F)(CNC(=O)C(=O)NC1CC1)C(C)C)NCc1ncc(CC)[nH]1 12627,Cn1cc(C(C(=O)NCCCC2CCC2)NCc2cccnc2)cn1 12628,C(CCCCC(C(=O)NCC1CCOC1)N1CC(C)(C)C2COCC12)OC 12629,O=S(=O)(c1ccccc1N1CC(O)CC(F)C1)NCCOC1CC1 12630,C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CC(C)C(NC(=O)Cn2nnnc2C2CC2)CC1 12631,C1(C(C)C)CN(C(=O)Cn2nc(O)ccc2=O)CCN1C(c1cc(O)nn1C)=O 12632,c1(CNC(c2n(CC(C)(CO)CO)ncc2)C(F)(F)F)cccc(S(=O)(=O)CF)c1 12633,C12(C(=O)NC3CCCCN(C(=O)CC45CCC(CC4)C5)C3)CC1Cc1c[nH]nc12 12634,C(N=c1[nH]c(=NCC2CC2)[nH]c2ccc(Cl)cc12)c1cccc(OCCOC)c1 12635,c1(N(CC(COC)(F)F)C)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12636,Cn1cc(C=CC(=O)NCCCC2(C(=O)NCC3CC3C3CC3)CC2)nn1 12637,C1(N(C(C(CC)NC(C)=O)=O)CC)CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 12638,C1(CNC(CCCSC)=O)(CO)CCN(C(c2csc(Cl)c2)=O)CC1 12639,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12640,C1(C(N(CCCNC(=O)CC2(C)CC2)CC)=O)C(C(F)(F)F)C1[N+](=O)[O-] 12641,C=C(F)CN=C(NC(C)C)NC1CC(=O)N(c2cccc(C(F)(F)F)c2)C1 12642,N1(C(C2(O)CN(C(C(C)NC(CC)=O)=O)C2)=O)CCc2ncn(C)c2C1 12643,c1(C(=O)OC)c(NC(=O)CCC(C)(C)N(C)C)sc2c1CCC(C)C2 12644,C(=O)(C(C(F)(F)F)C(F)(F)F)NCCC1N(C(C2CCC(C)(C)O2)=O)CCSC1 12645,C(=O)(C(C)(C)C(O)C(C)C)N1CCC(C#C)(C(=O)NCc2noc(C(N)=O)n2)C1 12646,C(=O)(C(C)(F)C(CC)CC)NCC1(CNC(C(CC=C)c2ccccc2)=O)CC1 12647,C1(NC(=O)C(N2CCCC(c3ccnn3C3CC3)C2)=O)CCCS(=O)(=O)C1 12648,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(N)=O 12649,C1(C2CN(C(c3n[nH]cc3C(F)(F)F)=O)C2)(NC(C2C(CC)CCC2)=O)CC1 12650,c1(C(=O)NCC2C(C)CCN2C(=O)CC2CC(C)(C)C2)ncc(N)cc1Cl 12651,c1(C(=O)NCC(C)NC(=O)C(C)Sc2ccccc2)cccnc1O 12652,c1(CNC(c2scc(C(=O)OC)c2)=O)nc(C2CC2)n(C)n1.C1C(C)(C)N1 12653,C1(OC)CCC12CC(C(=O)NCCC1(NC(c3coc(C#N)c3)=O)CCC1)C2 12654,C(CC(=O)N=c1cc[nH]c(CCCO)c1)NC1(c2c(OCC)cc(C#N)cc2)CC1 12655,C1(CCNC(c2cnn(CCC)c2C)=O)CCN(C(=O)CN(C)CCO)C(C)C1 12656,C1(CC)CCN(C(c2coc(C3CC3)n2)=O)C1CNC(C1CCC(CO)CC1)=O 12657,CCCC(C)(C)CC(=O)N1CC2CCC2(CCNC(c2cc(C)ncn2)=O)C1 12658,c1(C(=O)NC2(CN(C(C(N3CCCC3=O)C)=O)C)CC2)cc(=O)cc[nH]1 12659,CN=c1ncc(Cc2cn(CCC(N3CC4CC4C3CO)=O)nn2)c[nH]1 12660,C1(NC(C(C)=C2CCC2)=O)CN(C(c2cnn(CCO)c2C)=O)CCC1C 12661,N1(C(C(c2scc(C)c2)C)=O)CCC(C)(NC(c2coc(C(F)(F)F)c2)=O)C1 12662,C1(NC(C(C)OCC#C)=O)CCC(N(C(C2(OCC)CC2)=O)CC)C1 12663,N1(C(CC#C)=O)CCc2cc(CNC3COC(C)C3)ccc2C1 12664,C(=O)(CC(O)CC(C)C)NCC(F)(F)C(=O)NCC(CCC)C(=O)N.C(C)=O 12665,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12666,c1(C(=O)NCCOCCC(=O)N(C(C)CC)C)ccc(C(F)F)o1 12667,c1(NC(=O)OC)ccc(Cl)c(C(=O)NC(=O)C(C)Sc2ccccc2Cl)c1 12668,c1(CC)cc(C(=O)NCC2CCCC2C(=O)NC2CC(O)CC2O)ncn1 12669,c1(C(N2CCCCC2C(=O)Nc2ccc(I)cc2)=O)cc(F)cc(Br)c1Cl 12670,C(=O)(C1=CCC(NC(c2cc[nH]n2)=O)C1)N1CCC(C)(O)C1 12671,C1(C(=O)NCCNCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12672,N1(C(C(CCC)O)=O)CCC(C(F)(F)F)CC1CNC(c1nn(C)cc1SC)=O 12673,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12674,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12675,C=CC(CC)CC(=O)NCCCCC1CN(C(C2CN(C)CC2O)=O)C1 12676,c1(CN2CC(C)C(NC(C3(C#N)CC4CC4C3)=O)C2)cn2c(Br)cnc2s1 12677,Cc1nn(C)c2ncc(C(=O)NCC3C4CN(c5nc(Cl)c(C#N)s5)CC34)cc12 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12784,C(=O)(C1=NOC(NC(=O)CC(=O)N(C)C)C1)NC(C)CCSC.COC 12785,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12786,c1(C(=O)OC)ccoc1C(=O)NCCCCCNC(c1ccnn1CC1CC1)=O 12787,c1(C(C)C)ccc(CNC(=O)N(C)CC2CCCN2Cc2ccccc2)cc1 12788,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2)CC)[nH]1 12789,c1(C(N2C(CNC(C3C(C=C)C3)=O)CC(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 12790,N1(C(C(C2CC(C)(C)C2)OC)=O)CCC2(CCC(NC(=O)CC(F)(F)F)C2)C1 12791,C=CCCCCC(C)Nc1ccc(NS(=O)(=O)CC2CCCCC23CC3)cn1 12792,c1(C(=O)OCCCCC=C)[nH]cc2c1CCCC2 12793,N1(C(C2CCN(C(=O)NC)CC2)=O)CCC2(CCC2)C(CNC(=O)C(C)SC)C1 12794,c1(C(=O)NCCN(C)C(c2cnc3n2CCCCC3)=O)cc(O)c2ccoc2c1 12795,C(=O)(C#CC1(C)CC1)NC(C)C(=O)NCC(CNC(=O)CC(C)(C)C)(C)C 12796,c1(C(=O)NC2CC3(CC(NC(c4scnc4Cl)=O)C3)C2)cc2ccccn2c1 12797,c1(C(N(CCC)CCNC(=O)CSC(C)(C)C)=O)ccc2c[nH]nc2n1 12798,C12(S(C)=O)CCN(C1)C(=O)NC(CO)COC2=O.C(C)(C)(C)NC(=O)NCC 12799,CC(C)(C)CCCC(=O)C(=O)N1CCCC(Cn2cc(C3(O)CCOC3)nn2)C1 12800,C1(CNC(CSC(=N)N)=O)CC2CC2N1C(=O)CCOCC(F)F 12801,N1(CCOC)CCC(N=c2[nH]c(N3CCSC(C(C)(C)C)C3)nc(=N)[nH]2)C1 12802,c1(COC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CNc1nccs1 12803,c1(SC)cccnc1C(=O)NCC1CC2CC2N1C(=O)CCc1cscn1 12804,C1(NC(C(C)c2ccsc2)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12805,c1(CNC(C2N(CC)CCC2)=O)nnc2n1CCN(C(C1Cc3nccn3C1)=O)C2 12806,N1(C(C(C)SC(C)C)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 12807,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12808,C1(CCC(=O)N(CC#C)C)CCCN(C(=O)CCC(C)OC(C)=O)C1 12809,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(NC(C1(N(C)C)CC1)=O)C2 12810,c1(C(CNC(C2CCCO2)=O)NC(c2cc(C3CC3)[nH]n2)=O)ccc(F)cc1 12811,c1(C(N2CC(C)C(CNC(c3cc(Br)no3)=O)C2)=O)cnc2c(n1)CCCC2 12812,c1(OCC(=O)NC(CC)CNC(C2CC2C(F)F)=O)ccc(Cl)cc1C 12813,N1(C(CNS(C)(=O)=O)=O)CCCC2(CCCCC2NC(C2(C)CSC2)=O)C1 12814,C1(C(N2CC(N(C(c3ncsc3C3CC3)=O)C3CC3)C2)=O)CCCC2(CCC2)C1 12815,C1(C(=O)OC)CCCN(c2ccc(NC(c3ncc(I)cn3)=O)cn2)C1 12816,CC1C(=O)CCC1CC(=O)N(C)CCN1CCN(C(=O)CC2CNC(=O)C2)CC1 12817,C(C(C(C)(C)C)NC(=O)CCCn1cccn1)NC(C(C)NC(N)=O)=O 12818,N1(C(C(C)OCCC#C)=O)CCN(C(=O)CCNC(=O)COC)CC(C)(C)C1 12819,Cc1cc2[nH]c(C(=O)NC3CC4(C3)CC(Nc3ncc(F)cn3)C4)cc2o1 12820,C1(C(=O)NCC2C3CN(C(COCCCC#C)=O)CC32)CCC(S(N)(=O)=O)CC1 12821,C1(CO)CCOC12CCCC2.C1C(OC(C)C)CC(=O)N1.C(C1C(=O)N1)OC 12822,N1(NC(c2c(C)c(Br)ccc2)CO)CCC12CC(C#N)C2 12823,C(=O)(C(CC)CC=C)NC(CCCCNC(c1cc(CC)[nH]n1)=O)C 12824,N1(C(c2n(C)cnn2)C(=O)NCCC#N)CCOC(c2cncnc2)C1 12825,Cc1cc(C(N2CC(NC(=O)CCS(C)(=O)=O)C(C)C2)=O)cc(N)c1 12826,CC1=C(C(=O)NC(C)C(C)SC)Cc2ccccc2O1.C(=O)(CS(C)(=O)=O)N 12827,c1(C(CC)NC(=O)C(=O)NC2CCC(C)(C)NC2)cccc(C#N)c1OC 12828,C1(C(=O)NC(C2CCN(C(C3(C)ON=C(C)C3)=O)CC2)C)CCCC2(CCC2)O1 12829,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12830,C#CC1CN(C(=O)CCC2CCOCC2)CCN1C(C1CN2CCN1CC2C)=O 12831,N1(C(CCC=C)=O)CC2CN(C(c3cccc4cncn34)=O)CC2C1 12832,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(c2cc(Br)nn2C)=O)C1 12833,N1(CC(N)=O)CC(CN=[N+]=[N-])C(C(F)(F)F)C1.c12ccn(n1)CC(=O)NC2 12834,c1(C(=O)NCC2C(C)(C)CO2)cccc(Cl)c1.C12CCCN(C1)C(=O)CCC2 12835,C1(C(C(=O)NCCCCCC)C)CCN(Cc2cncs2)CC1 12836,Cn1nc(C(N2CC3CC2(C(N2CCC(C)(F)C2)=O)C3)=O)cc1O 12837,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(C(C)C)OC 12838,CCCC(C)(CC)C(=O)NCC1CC(C(=O)NCC2(CN(C)C)CC2)=NO1 12839,C1(SC)CN2CC1C2=O.c1(CCC(=O)NC2CC2c2cccnc2)ccncn1 12840,CCC(CC(=O)NCCCC(=O)N1CC(C)(CCO)C1)C1CC1 12841,c1(C(N(C2CN(C(C(C(C)C)N3CCC3)=O)C2)C)=O)cc2c([nH]1)CCC2 12842,C1(CCCCCC)CCCC1(c1nnnn1C1(C)CC1)NCC 12843,CC12CN(C(=O)C(=O)NCCCC(F)F)CC1(CO)C2 12844,c1(C(=O)NC)ccc(CC(=O)NCC2CCN(C(C3(CF)CCC3)=O)CC2)cc1 12845,CC(CCCCNC(=O)CCc1cc(Cl)no1)NC(c1coc(Cl)c1)=O 12846,c1(N(C)CC2CN(C)C(=O)C2)ncccc1S(=O)(=O)N1CCC(CF)C1 12847,C(CC(C(C)(C)C)NC(C1CC2CC2C1)=O)N(C(c1c(C)cncn1)=O)C 12848,O=C(C1=CCCN(CC(N2CCCC2)=O)C1)NCCn1ccc2ccccc12 12849,C1(NC(C2CCCC(OC)C2)=O)CCC2(CC1)CCN(C(=O)C1=CCCCC1)C2 12850,C(=O)(C(O)CC(N)=O)NCC1(C(N)=O)CN(C(C2(OC)CCC(C)C2)=O)C1 12851,C#Cc1ccc(CC(N2CCCOC(CNC(=O)OC(C)(C)C)C2)=O)cc1 12852,CC(C)CC(O)C(=O)N(C)CCOCCN(C)C(c1ccc(-c2cccs2)o1)=O 12853,C(=O)(C(CO)C(C)(C)C)N1CC(C(=O)N(C2CCCCC2)C2CC2)(COC)C1 12854,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12855,C1(NC(CCNc2c(OC)cccc2)=O)CCC(C)N(C(=O)C2=CCSC2)C1 12856,C1(C(C)(C)C)C(=O)N1.c1(CCCSC)cn(Cc2ccoc2)nn1 12857,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12858,C1(CC(=O)N(C)CC2CCN(C(c3ncn(C)n3)=O)C2)CCC(=O)C1C 12859,N1(C(c2c(C)cccc2)C(=O)N(C)C)CCN(CC(F)(F)F)CC(CO)C1 12860,CCC(O)C(F)(F)C(=O)N1CCN(C(=O)C#CC(=O)NCCOC)CC(CO)C1 12861,N1(C(C=C(C)C(C)C)=O)CCC2CCC12CNC(c1ccc(O)c(F)c1)=O 12862,c1(C(=O)NC2C3(CN(C(C4(OC)CCCC4)=O)C3)CC2)cc2c(s1)CCSC2 12863,C1(c2n(CCOC)nc(-c3ccnn3C)n2)CCc2n[nH]cc2C1C 12864,c1(NC(c2nnnn2C2COC2)(CNC(C)=O)C)cc(Cl)ns1 12865,C1(Br)(C(N(CCN(C(=O)C2=CC(C)(C)C2)C(C)C)C)=O)C(C)(C)C1(C)C 12866,C(O)(C(=O)NCC(CN(C)C)NC(=O)CC=CC(C)(C)C)SC 12867,C1(NC(c2cc(C(C)(C)C)sc2)=O)CCN(C(C2COCC(C)(C)O2)=O)CC1O 12868,Cn1cc(C(=O)NCC2CCCCN2C(=O)Cn2ccccc2=O)n(C)c1=O 12869,C(=O)(CC(C)(C)C(F)F)N(C1(CO)CCC1)C.N12CC(C(O)C1)C2=O 12870,c1(C(=O)NCCCN(C(=O)C=C2CC2)CC)cc2cc(C)ccc2o1 12871,C1(CNC(C=C(C)C(C)(C)C)=O)C2CCC(C2)N1C(C1(C)CC2CCC1C2)=O 12872,C12(NC(c3coc(Br)n3)=O)CCC(n3cc(-c4ccns4)nn3)(CC1)C2 12873,N1(C(C(C)OCC(=O)NC)=O)CCC(CO)(NC(=O)CN2CC=CC2)CC1 12874,n1(CCC(=O)NCC(C)NC(c2cc(C(=O)NC(C)(C)C)no2)=O)cc(Cl)cn1 12875,Cc1[nH]nc(C(C)C)c1C(N1CCC(CCC(C)O)CC1)=O 12876,C#CCC(C(=O)N1CCC1c1ccccc1)NC(=O)C(CC)NC=O 12877,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12878,N1(C(C2(NC(c3ccc(C)n3C)=O)CCCC2)=O)CCOC(C)(C)CC1 12879,c1(C(=O)NCC(CNC(CCCC)=O)C(F)(F)F)cc(N=S(C)(C)=O)ccn1 12880,c1(C(N2CCN(C(c3ccccc3)=O)C(C(F)F)C2)=O)cc([N+](=O)[O-])n[nH]1 12881,c1(NC(=O)NC2C(C)(C)C2)cccc(CN2CCOCC2)c1 12882,C(C)(CCC(=O)NCc1nc(CNC(c2ccccc2O)=O)cs1)OC 12883,c1(C(N2CCN(C(c3c(CC)cns3)=O)C(CO)C2)=O)ccc2ccoc2c1 12884,C1(CCN(C)CC)CCCC1(C)C.C(=O)(C(C)O)NCCCOCCOC 12885,C1(NC(=O)NCC(C2CCOCC2)(C)C)CC2(C1)CC(F)(F)C2 12886,c1(C(N2C(C(=O)NC3CCCC3)CC(=C)C2)=O)cc(C)ccc1O 12887,C1(C(N2CCC(C(=O)OC)C2C)=O)CNC(=O)CN1C(C1CC(C)(C)CN1C)=O 12888,Cc1cc(NCCCNC(C2(O)CCCC(C)CC2)=O)n2ncc(C)c2n1 12889,C#Cc1c[nH]nc1C(=O)NCC=CCNC(C1CCC(NC(C)=O)CC1)=O 12890,C(CCCC#N)(C(=O)NC1CCCC1)N(C(CC=C)CO)C 12891,C1(C(N2CCCC(CN(C)C(c3cc(CO)ncn3)=O)C2)=O)CC2(CCCC2)CO1 12892,C1(NC(=O)OC(C)(C)C)CC(C(=O)NCc2ccno2)C12CCC2 12893,c1(CCCOC)cn(CC2CCCN2C(c2cc(-c3ccns3)on2)=O)nn1 12894,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC)CC12 12895,c1(N2CC=CC(NC(C3C(CC)CCC3)=O)C2)ncnc2sc(C)nc12 12896,C=CC1(C(=O)NC(CO)C2CC2)CCN(C(=O)Cc2cccnc2)C1 12897,c1(C(=O)NCC(CNC(CCn2ncc(C)c2)=O)C)cncc(N)c1C 12898,CCCCC(F)(F)C(=O)NC(C)CN(C)C(C1(Br)CC1(F)F)=O 12899,c1(NC(C(N2CC(C)N(CC(=O)NCC(F)F)CC2)=O)=O)cccc([N+](=O)[O-])c1 12900,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12901,N1(C(C(CCCOC)NC(C2CC=CCC2)=O)=O)CC=CC12CCCCC2 12902,N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(CCO)CC1(C)C 12903,N1(C(C(C)SC)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)F)C1 12904,C(C(CC(C)C)C(=O)NC(C)(C)C(F)(F)F)CCC(=C)Cn1ccnc1.C1(=O)CN1 12905,N1(C(c2c(C)c[nH]n2)=O)CC(C)CN(C(C2(C)CC(O)CN2C)=O)CC1C 12906,C(=O)(C1CC(NC(c2c[nH]c3ncc(Br)c-3c2)=O)c2ccccc21)OCC 12907,c1(C(=O)NC2CCCN(C(=O)NCCCC(C)C)C2)cccc2c1NCC(C)C2 12908,c1(C(=O)NCC2N(C(C(C)CC3CCC3)=O)CCCC2C)nccc2occc12 12909,c1(C(N(CCCNC(C2CCC(C(F)(F)F)CC2)=O)C)=O)ncn2c1COCC2 12910,C12(C(N3C(CN(C(=O)CCc4cn(C)nc4C)CC)CCC3)=O)CCN(CC1)C2 12911,c1(NC(C)CCNC(c2ccnc(CO)c2)=O)cc(O)nc(=O)n1C 12912,c1(C(N2C3CC(NC(C(COC)OC)=O)C(C3)C2)=O)ccc(C)c2ccccc12 12913,N1(C(=O)Nc2ccc(CC)s2)CCC(CN(C2CCN(C)CC2)C)CC1 12914,N1(C(Cc2scc(C)c2)=O)CCN(Cc2ccc(O)cc2C)CC1C(C)CN(C)C 12915,c1(C(N2CCC(CN(C(=O)CCS(N)(=O)=O)C)C2)=O)cc(N(C)C)nc(Cl)c1 12916,N(C)(C1CCCc2ccccc21)C(C1Cc2n(CC)ncc2CC1)=O 12917,C1(NC(CCC2CC(CC(N)=O)C2)=O)(CNC(=O)CNC=O)CC2CCC1C2 12918,C1(OC)CCCCC1C(=O)N(C)CC=CC(=O)NCc1nc(SC)ns1 12919,c1(C(=O)NC2C(OC)CN(C(c3cccc(F)c3C)=O)C2)cc(N)c(C)cc1F 12920,N1(C(c2ncn(CCNC(C(C)C3CCCC3)=O)c2)=O)CC(C(N)=O)C2(CC2)C1 12921,N1(C(CN(C(Cc2nc(=N)[nH][nH]2)=O)CC2CC2)=O)CCCN(C2CC2)CC1 12922,c1(C(C)Nc2c(CC)n[nH]c2)cc(Cl)ccc1OCCNC(=O)OC(C)(C)C 12923,c1(C(C)C)nnc2n1CC(NC(=O)CNC(c1ccc(O)cc1)(C)CO)CC2 12924,Cc1cc(C)c(C(=O)NC2CC3CC(C2)N(C(=O)Cn2nccc2C)C3)c(S)n1 12925,C#Cc1ccc(OCC(=O)NCC(=C)CCNC(C2(F)CC=CCC2)=O)cc1 12926,c1(COC)nc(Cl)cc(=NC(C)C2CCN(C(C3CCCC4C3C4(F)F)=O)CC2)[nH]1 12927,N1(C(C2(COC)CC2)=O)CCC(C)C(NC(=O)CC(c2cccc(N)c2)C)C1C 12928,C1(CC)C(C(N2CCCC2C(=O)NC2CC(CSC)C2)=O)C1(C)C 12929,CC1CC(NC(=O)CC=CC(C)(C)C)CN1C(c1cc(N2CCOCC2)ccn1)=O 12930,N1(C(C2(CNC(C(COC)(C)OC)=O)CCCO2)=O)CC2CCCCC2C1C 12931,C(=O)(C(F)C(=O)NC1(C)CC(NC(C2(C)CC2)=O)C1)OCC 12932,c1(C(=O)NCC2C(NC(C(C)OC)=O)C2)sc2ccccc2c1Cl 12933,CC1CCCCC1(C)NC(=O)Cn1cc(C2CCC2)nn1.N12CCC(C1)C2=O 12934,N1(C(C(C)CNC(c2cc(C(F)F)[nH]n2)=O)=O)CCC2CCN(C)CC12 12935,Nc1ncc(N)cc1C(N1CCC(NC(C2CC2(Cl)Cl)=O)C(F)C1)=O 12936,C1(NC(C(CCC)NC(N)=O)=O)CN(c2ccncn2)CC(F)(F)C1 12937,c1(C(=O)NC2C(NC(c3ccc(NC)cn3)=O)CC2)cnc(O)c(F)c1 12938,Cc1ccc2c(c1)c1ccc(o1)c(=O)sc1n2ccn1.C1C(=O)N(C)C1 12939,c1(C(=O)NC2CCC(NC(C(C(C)C)SC)=O)CC2)cc(C)c(=O)n(C)c1 12940,N1(C(c2c(CC)scc2)=O)CC2(C)CN(C(=O)COC(F)(F)F)CC2(C)C1 12941,Cc1csc(C=CC(=O)NCC2COCCN2C(=O)CC(C)c2cnn(C)c2)n1 12942,C1(C(N2CC(N(C)CCO)C2)=O)(CC)CCOC1.C(C)(C=O)NCC 12943,C1(C(=O)OC)COC2(CCN(C(C3(C)CCN(C(=O)OC(C)(C)C)C3)=O)CC2)C1 12944,c1(SC(CNC(C2(COCC(=O)NC3CC3)CC=CC2)=O)C2CC2)ccccc1 12945,Cc1ncc(C=CC(=O)NC2CC(NC(c3coc(CO)c3)=O)CC2O)s1 12946,C(c1cccnc1)=CC(=O)NC1CN(C(=O)Cc2ccc(C(=O)O)nc2)C1.CCF 12947,c12cc(ccc1F)N(C)C2=O.CC1OC(=O)NC1C(=O)NCC1(COC)CC1 12948,CCC(O)C(F)(F)C(=O)N1CCCC(CCC(=O)N(C2COCC2(C)C)C)C1 12949,CCCCC(O)C(C)C(=O)N1CC(O)(C(C)(C)CNC(=O)Cc2cnoc2)C1 12950,C1(CN(C(c2ncn(CC)c2)=O)C)CN(C(c2cnc(S)n2C)=O)CCO1 12951,c1(OC(CC)C)cc(C(N2CC(N(C)Cc3cscn3)C2)=O)ccn1 12952,c1(C2(C)CCN(C(C(=O)NC(C)(C)C)CC3CCC4CC34)C2)cc(Cl)ccc1Cl 12953,c1(OC)ccc(Br)c(CN2CCCCC2CCC2CCC2)c1OC 12954,C1(C(=O)NC2CC(C)(C)N(C(=O)Cc3csc(Cl)c3)C2)CCCN2CCCCC12 12955,c1(C(=O)NC(C)CN(C)C(C2(c3ccccc3)CCC2)=O)snc(O)c1Cl 12956,C(C(=O)N1CC2C(CC(=O)NC(C)(C(N)=O)C3CCCC3)C2C1)(C(C)(C)C)N(C)C 12957,Cc1cnc(C(=O)NC2CCCC(NC(C3(N(C)C(C)=O)CC3)=O)C2)nc1 12958,c1(C(=O)NC(CNC(C(C2CCCCC2)C)=O)C(C)C)nc(=O)n(C)[nH]1 12959,N(C1CCOc2ccc(F)cc21)C(c1nccc(-c2ccc(N)cc2)c1)=O 12960,C(=O)(CC(C)CC(C)C)N1CCC(CNC(c2c(CC)scn2)=O)(COC)C1 12961,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCC12CN(C(=O)C(C1CCCCC1)O)C2 12962,C(C(O)CCNC(=O)C(Cc1ccoc1)C(=O)NC1CC1)OC 12963,N1(C(CC2CC(=C)C2)=O)CCN(CC(=O)NCC(=O)Nc2cn[nH]c2)CC1 12964,N1(C(C=CC(C)C)=O)CCC2(C1)CN(C(=O)C(N1CCC(C)C1)=O)CCO2 12965,N1(C(c2cc(CCOC)on2)=O)CCC2(CCCN2C(=O)CP(C)(C)=O)C1 12966,CN1CCC(C(=O)NCC(C2CC2)NC(C2CCN(c3ccccc3)C2)=O)CC1 12967,c1(C(=O)NC(CNC(C(n2ccc(C)n2)C)=O)CO)cnn2cc(C#N)cnc12 12968,C1(CC)CCC(C(N2CCCCC2C(C)NC(=O)Cc2ncc(C)o2)=O)CC1 12969,C12(CNC(C(C)NC(COC)=O)=O)CC1CN(C(C1(F)CCCCC1)=O)C2 12970,N1(C(CNC(C(CC)C)=O)=O)CC(F)CC1CNC(C1CCCC(OC)C1)=O 12971,c1(COC)cccc(C(N2CCC2C(C)O)=O)n1.c12c[nH]c(c1)C(=O)NC2 12972,N1(C(CC2(O)CCCN(C)C2)=O)CCC(CNC(c2cccnc2)=O)C12CCC2 12973,C1(CN(C(CN(C)CC)=O)C)COCCN1C(=O)CCCc1csc(C)n1 12974,c1(N(C)CCn2c(C)cc(C)n2)ncccc1S(=O)(=O)N1Cc2ccncc2C1 12975,c1(CC(=O)NC(CC)C(=O)c2ccccc2)cn(C)c2ccc(F)cc12 12976,N1(C(C=CC(C)NC(C2CCCS2)=O)=O)CC2(CCNC(=O)O2)C1 12977,c1(N(C)C)ncc(CC=CCNC(=O)NC(=O)CCC2CCCCCC2)cn1 12978,C(CNC(=O)CC(Cl)Cl)(C(=O)NC(C1=CCCC1)C1CC1)N(C)C 12979,C#Cc1ccc(C(N2CCOC(C(C)NC(C3CCC4(CC4)C3)=O)C2)=O)c(C)c1 12980,c1(NC(C=CCNC(c2c(CC)nn(C)c2)=O)=O)ccc2occc2c1 12981,c1(C(CNC(C2CNC(=O)C2)=O)NC(CN(CCC=C)C)=O)ccccc1OC 12982,C(=O)(C(C)(C)CC(F)F)NC1C(OC)CN(C(=O)CN2CCCCC2C)C1 12983,C(=O)(C1COc2ccc(F)cc21)NCC1(NC(C2C(C)(C(F)F)C2)=O)CCCC1 12984,CCCCC(CC)C(=O)NC12CCC(CNC(=O)CC(F)(F)F)(C1)OC2 12985,c1(C(=O)NCC(CNC(c2nc(CC)sc2)=O)OC)cccc2c(C#N)c[nH]c12 12986,c1(OCCOC)nnc(Cl)cc1NCc1cccc(F)c1OC 12987,CCC(C)CCC(O)CC(=O)NC(C1CCN(C(=O)CS(=O)(=O)C2CC2)C1)C 12988,C=C(C)C(C)(C)C(=O)NC1CC1NC(C1CCN(C(c2cccnc2)=O)CC1)=O 12989,c1(C2CC(C(=O)NCC3CCN(C(COC)=O)C3)C2)ccc2c(c1)OCO2 12990,N1(C(CCP(C)(C)=O)=O)CCCC2CN(C(c3cc4ccccc4cn3)=O)CC12 12991,c1(C(=O)NC(CNC(CCOCCC)=O)C2CCC2)cc2cc(C)ccc2[nH]1 12992,C(C)(CCC(=O)NCCCn1cc(-c2csc(-c3ccoc3)n2)nn1)SC 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13063,C(=O)(C1=CCC(C)CC1)NC1CCN(C(CCCn2c(C)nc(C)n2)=O)C1CC 13064,C1(n2cccn2)(C(=O)OC)CCN(C(=O)NCCOCCOC)CC1 13065,CC(=O)CCCC(=O)N1CCCC(NC(c2ccc(C(F)(F)F)cc2F)=O)C1 13066,c1(C(=O)NC2CCCC(N(C)C(c3ccsc3Cl)=O)C2)ccc2nn[nH]c2n1 13067,C1(NC(C2ON=C(CC)C2)=O)C(C)CCN(C(c2cnc3ccccn23)=O)C1C 13068,c1(C(C(=O)NCC)N(C)CCC2CC2)ccc(OC(F)F)cc1 13069,C1(CC)CN(C(=O)Cn2cc(Cl)cn2)CCC1NC(=O)C(F)(F)C=C 13070,C12(CCCC1)C(=O)NCC2.C(=O)(CCSC)NCC1(CNC(=O)CO)CC1.CC 13071,N1(CC(=O)NC2CC(C)(NC(=O)CC3CC4CC4C3)C2)CCC(=O)NC1=O 13072,N1(C(C(C)C(C)O)=O)CCC(NC(C2(O)CCC2)=O)C(c2ccccc2)C1 13073,N1(C(C(C(C)C)(C)O)=O)CC(NC(c2ccc(F)s2)=O)CC(C)(C)C1 13074,N1(CCNC(N(C)Cc2cnn(C3CC3(F)F)c2)=O)CCc2ccccc21 13075,c1(Nc2ncc(C#C)cn2)ccc2c(c1)CN(C(=O)C(C)OCCC=C)CC2 13076,C#CC(CNC(=O)CC1(CNC(C2CCO2)=O)CC1)CC1CC1 13077,N1(Cc2n(C)ncc2)CC2(C1)CC1(C3CCC3)CC(c3nn[nH]n3)(C1)C2 13078,NS(=O)(=O)c1ccc(NNC(=O)C(=O)NC2CC2F)s1 13079,N1(C(CCCCC#C)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)CC2CO 13080,C1(NC(CCCSC)=O)CCOC(CNC(=O)C(C)N=[N+]=[N-])C1 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13150,C(CC(=O)N(CC(C)NC)C)C(=O)C(F)C1CCOC1.C(C)(C)(C)OC(CC)=O 13151,N1(C(C(C2CC2)NC(c2ccc(NC)cc2)=O)=O)CC2(CCC(O)CC2)C1 13152,c1(CNC(C2CC2)=O)noc(-c2ccccc2)n1.C1(CNC=O)CCC1C(F)(F)F 13153,c1(NC)ccnc(C(N2CCC(CNC(=O)CCC(C)c3ccccc3)C2)=O)c1 13154,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13155,N1(C(C(CC)NC(N)=O)=O)CCC(N=c2cc(C)nc([N+](=O)[O-])[nH]2)CC1C 13156,N12CCC(CC1)CN(C(=O)Cn1ncnn1)CC2.C(=O)(CCc1cscn1)N 13157,c1(CC)ccc(C(N2CCC(NC(=O)C(C)=C3CCC3)C(CO)C2)=O)cc1N 13158,c1(C(=O)NCC(O)CNC(c2ncnn2-c2cccs2)=O)ccnc(Cl)c1 13159,Cc1cccc(C(=O)NCC(C)N(C)C(c2ccc(CCF)cc2)=O)c1C 13160,N1(C(c2ccc(C=C)cc2)=O)CC=C(CC(=O)NCc2cccc(F)n2)CC1 13161,C1(CNC(c2nn(CC)c(O)c2)=O)(NC(c2cc(Br)n[nH]2)=O)CCCCC1C 13162,c1(C(N(C(C)CNC(=O)C(C2CC2)N(C)C)C)=O)cc2ncccc2o1 13163,c1(CC(N2C(CNC(=O)Cc3ccno3)CCC2)=O)ccc2ncsc2c1 13164,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13165,C1(C(N(CC(C)(C)NC(C(CSC)OC)=O)C)=O)CC2CCC(C1)N2C1CC1 13166,C(C(C)C(=O)NC1CCC1)NC(CCNC(C)=O)=O 13167,C1(C(=O)Nc2ccc(I)c(Cl)n2)C2CCCC1CN(C(C1(O)CC1)=O)C2 13168,c1(C(=O)NC(CNC(CCCc2[nH]c(=N)sc2)=O)C2CC2)ccc(CCO)cc1 13169,C=CCC(CC=C)C(=O)NCC(O)CNC(c1cccc(I)c1)=O 13170,N1(C(=O)NC(C)(C)C)CC(CO)CC1C.c1(CC(=O)OC)cn(CCO)nn1 13171,C1(CC(=O)NCCc2ccsc2)CCN(C(=O)C=Cc2cnccn2)CC1 13172,c1(C(=O)NC(C(C)NC(c2c(CC)nco2)=O)C)ccc(F)cc1OC 13173,C1(C(C)OC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCCC2)CC1 13174,N1(C(C2C(=C)C2)=O)C2CCC1C(NC(c1cccn1C1CCCC1)=O)C2 13175,C1(C(N(C)Cc2cccc(Cl)c2)=O)CN(CC(=O)NN2CCC2CO)CC1F 13176,N1(C(c2c(CC)nns2)=O)CC(C(=O)NC(C)(C)CCCO)C(F)(F)C1 13177,N1(C(CCNC(C2=CCCC2C)=O)=O)CCCN2CCCC2C1 13178,Cc1cnc2n1CCC(C(=O)OC(C)(C)C)C2.C1C(c2ccccc2)C(=O)N1 13179,CN1CCN(C(c2cc(O)ncn2)=O)C(C(N2CCCC(OC3CC3)C2)=O)C1 13180,c1(CC)cc(C(N2CCCCC2C2CCN(Cc3[nH]c(C)nc3C)C2)=O)ncn1 13181,C(=O)(CCc1cnco1)NCCN(C(N1CCCC1)=O)CCOC.O=CCOC 13182,N1(C(c2cc(OC)no2)=O)C(CNC(=O)C(C)CO)CC2COCC12 13183,c1(-c2cc(C)c(=N)[nH]c2)n[nH]c(=NC(=O)NCC2(CN(C)C)CC2)s1 13184,C(N=c1[nH]cc2c(c1C#N)CCCC2)C(C)C(N1CCNC1=O)=O 13185,C(CCCC(=O)N1CCCCO1)NC(CCCCOCC)=O 13186,CC(C(CO)NC(c1csnc1-c1ccccc1)=O)NC(c1ncccn1)=O 13187,C(CS(=O)(=O)C1=CCC2CC2C1)N(C)C(=NCc1cnn(C)c1)NCC1CCOC1 13188,C12(C(=O)NCC(CCN(C(C3(CN(C)C)CC3)=O)C)O)CCC(C1)C2(C)C 13189,CC(C)CC(O)CC(=O)N1CCCCC(N(C(=O)C(F)(F)C2(O)CCC2)C)C1 13190,C#Cc1c[nH]nc1C(=O)NC1CC1NC(=O)Cc1ccccc1CSCC 13191,N1(C(C=Cc2ncn(C)c2)=O)CCC(F)(CNC(=O)CC2CCC(=O)N2C)CC1 13192,c1(C(=O)NCC2C(NC(C3N(CC)CC3)=O)CC2)nnc(O)c2ccccc12 13193,N1(C(C2CC=CCN2C(=O)C(O)CN2CCCC2)=O)CC2C=CCC(C2)C1 13194,c1(C(=O)NC2(C3CCCN3C(=O)Cn3ccnn3)CC2)cn2ccnc2cn1 13195,C1(C(N(C2CCN(C(C(C(C)SC)O)=O)CC2)C)=O)CCCC(C#N)C1 13196,Nc1ccc(C(N2CCCC2CCNC(=O)C#CC2CCC2)=O)nc1C(F)(F)F 13197,C(C(O)CNC(=O)CN(CC(C)(C)C)C)N(C(=O)CC1CCCO1)C 13198,C1(NC(C2(CC)N(C(c3n[nH]c(CC)c3C)=O)CC=C2)=O)CCC(C)CC1C 13199,C1(N(C(CNC(=O)NC)=O)C)CN(C(=O)CC2CCCOC2)CC1F 13200,CC1CC(=O)NC1C(N1CCC(CCCNC(=O)Cc2cccc(O)c2)CC1)=O 13201,c1(OCCOC)ccc(NC2COC3CC2C3)cc1 13202,c1(NC2(CNC(c3cncc(NC)c3C)=O)COC2)ncnc2cc(Br)ccc12 13203,C(=O)(C1CCCc2sccc21)N.CN1CCC(C2(O)C(NCC)(CO)CC2CCC)C1.CO 13204,Cc1cccc(C(C)NC(=O)C(C2CCC2)N(C(=O)C)C)n1.C1CC1 13205,N1(C(C(CC(C)C)CNC(c2ccon2)=O)=O)CC2CCOC(=O)C2C1 13206,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13207,C1(NC(CNC(=O)OCC=C)=O)CCN(C(=O)C2=CCCCO2)CC1C 13208,c1(C(=O)NCCN(CCOC)C(C2CCSC2)=O)ccnn1-c1ccncc1 13209,c1(CC(=O)NCC2CCO2)ccc2nonc2c1.C12CCCC1CNC2=O 13210,C1(CNC(=O)CC2CCO2)(NC(=O)CC23CCC(CC2)C3)CCCCC1 13211,c1(SCC2N3N(CC3)C2)cc(Cl)c(O)cc1F.c1(CCC=O)ccc(Br)cn1 13212,C#Cc1ccc(C(=O)NCCCC2CCCCN2C(=O)COC2CCC2)c(F)c1 13213,CC(C)C(F)(CNC(C1CCCN1C1CC1)=O)C(=O)NCC(C)(C)CN=[N+]=[N-] 13214,n1(CC(N2CCN(C(=O)C3=CCOCC3)CC2C2CC2)=O)ccc2cccnc12 13215,C1(C(=O)NCCC(CNC(c2cc(OC)n[nH]2)=O)O)CCS(=O)(=O)CC1 13216,C(CC1=CCN(C(c2ccc(F)c(F)c2N)=O)CC1)NC(C(=Cc1cnc[nH]1)C)=O 13217,c1(OCC)ncnc(OCC(=O)OC)c1C(N1CCC1)=O.C1(OC)CCOCC1 13218,c1(C(=O)OCC)nnn(C)c1CNC(c1cscc1Cl)C 13219,C1(C(=O)NC(CC=C)C(=O)OCC)CNC(=O)CN1C(=O)Cc1ccco1 13220,c1(CC)ccccc1-c1cn(N2CCOCC2C2(c3ccc(Cl)cc3)CC2)nn1 13221,C1(CNC(c2cc(C)[nH]c2C)=O)CCCC2CCCCC12 13222,Cc1ncccc1C(N1CC(C(N)=O)(CNC(=O)CC2CCCC(C)O2)C1)=O 13223,c1(C(=O)NCC(CC)NC(C2NC(=O)CC2C)=O)ccc(N)cc1O 13224,C1(C(=O)NCCOCCC(=O)NC(CC)C2CC2)CCC1C#N 13225,c1(-n2c(C(CC)OC)nc(-c3ccc(Cl)o3)n2)cc(F)c(F)c(F)c1 13226,N1(C(C(c2scc(C)n2)C)=O)CC2(CCC2)CCC1CNC(C1CCOC1)=O 13227,C1(CC#C)(C(=O)NC(CC(F)(F)F)C2CC2)CCN(C(C2C=CCS2)=O)C1 13228,c1(OC)cc(C)nc(NC2CC(NC(=O)COCc3nnc(C)o3)C23CCC3)n1 13229,O=C1NCCCCC1S(=O)(=O)NCCCCCCCCN 13230,N1(CCNCC(CNC(c2cnn(CCCC)c2C)=O)CO)CCS(=O)(=O)CC1 13231,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13232,C1(NC(C(C)=C(C)C)=O)CCC(NC(=O)C(C2CCOCC2)C)C1 13233,Cc1ncc([N+](=O)[O-])cc1NC(=O)C(=O)N(C)Cc1cc(F)c(F)c(F)c1 13234,O=CN1CCCN(C(=O)CC(CNC(C2CC2(Cl)Cl)=O)C2CCC2)CC1 13235,c1(C(=O)NCc2cccc(NC(C3CCC(=O)NC3)=O)c2)coc2c1COC2 13236,C(CC)(CCCO)NC(C1(CC=C)CN(C(=O)C(C#N)CC)C1)=O 13237,c1(OC)ccc2[nH]ccc2c1C(=O)NCCC1(OC)CN(C(=O)C2=CCCS2)C1 13238,C(=O)(C(C)(C(C)C)OC)NC(CC=C)CNC(=O)Cc1n[nH]c(C)n1 13239,c1(OC(C(N2CC(NCc3cncc(C(C)=O)c3)C2)=O)C)ccc(C)cc1Cl 13240,C=CCC(C)(C)C(=O)N1CC(OC(CCCNC(COC(C)=O)=O)C)C1 13241,Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)N(C)C)=O.C1C(=O)N1 13242,c1(CC)nn(C)cc1C(=O)NCC1(NC(C2CC(C)OC(C)C2)=O)CC1 13243,CC1(C)C(C(=O)NCC(F)(F)Cl)C2CCCN(C(=O)CC3CCOC3)C12 13244,Cc1ccc2ccc(C(=O)NCC(O)CN(C)C(C3C(F)(F)C34CC4)=O)nc2c1 13245,CC1CCN(C(C2CN(C)CCO2)=O)CCN1C(c1ccn2ccccc12)=O 13246,C(CN=c1[nH]c(=NCC(C)c2ccccc2)[nH]c2c1COC2)n1c(C)ncc1 13247,CC(CO)(C(=O)NC1CCCSC1)NC(=O)C(C1CCOCC1)F 13248,N1(C(CC=C)=O)CCOC(Cn2cc(CC(c3ccccc3)O)nn2)C1 13249,c1(COC)cnc(NC(=O)NCC(c2ccccn2)C)nc1 13250,CC1CN(C(=O)C(=O)C(F)(F)F)CCC1NC(=O)CCC1CC1(F)F 13251,C1(CC(=O)N(CC(C)NC(=O)CCCCCn2cnnn2)C)CCS(=O)(=O)CC1 13252,C(=O)(CCCNCCC(F)(F)F)N(C)CC1CC(C#N)C1 13253,CC1CC2CN(C(C3CC3F)=O)CC2N1C(=O)C(O)CC(N)=O 13254,C1(OCC2N(C(C3(OC)CC3)=O)CCC2)CCN(C(C23C=CC(CC2)C3)=O)CC1 13255,C1(NC(C(c2nccc(CC)c2)N2CCC2C2CCCC2)=O)CCCCCCC1 13256,CCC(C(=O)NCCOC1CN(C(c2occc2Cl)=O)C1)OC 13257,C1(C(=O)NCC2(O)CN(C(C(C)=C(CC)C)=O)C2)CCN(CC(F)(F)F)C(=O)C1 13258,C1(NC(C(C)OCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13259,N1(CCF)CCC(CNS(=O)(=O)CC2CCOC2)CC1 13260,CCCCCC(C)CC(=O)NCC1(C(N2CC3OCCOC3C2)=O)CC(C)(C)C1 13261,C1(C(=O)NC2CCC(CNC(=O)CCN3CCCC3)C2)CC2(CCOC2)C1 13262,C(=O)(CC(C)C(C)(C)NC(=O)C(O)C(C)CC)N(CCCCC=C)C 13263,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCCN(C(c2cc[nH]c2)=O)C1 13264,c1(OC)cc(COC(=O)CN2CCCCC2)c(NC(=O)CCC2CCOC2)cn1 13265,c1(C(=O)NCC2(F)CC(NC(C3C(OC)CCC3)=O)C2)oc(CO)nc1C 13266,C1(NC(c2ccnc(C)n2)=O)C2CC1CN(C(=O)C(C)Sc1ccccn1)C2 13267,CC1CCC(CNC(=O)C(O)C(F)(F)F)CN1C(c1cnc[nH]1)=O 13268,CC(C#N)CCC(=O)N1CC(CNC(C2CC3C=CC2CC3)=O)C(C)(C)C1 13269,C1(C)(CNC(c2cc(CNC(C(CC)SC)=O)no2)=O)C=CCCC1.C(N)=O 13270,C1(N(C)C(C2CC(=O)N(C3CC3)C2)=O)CCN(C(C2C(C(=O)NCC#C)C2)=O)CC1 13271,c1(COC(C(=O)OC)C2CC2)cnc(N2CCC(NC(=O)C(CSC)OC)C2)s1 13272,C1(C(=O)NCC(C(C)C)O)CN(C(C2CSC2)=O)CC1(C)C 13273,c1(CC)nn(C)c(N2C3CCC2CC(NC(c2nccn2CC)=O)C3)c1[N+](=O)[O-] 13274,C(=O)(C(CO)C(C)C)NCC(C)N(C(Cc1cccc(C(C)C)c1)=O)C 13275,c1(OC)ccc(C(=O)NCCNC(=O)CC2CCCC(C)C2)nc1Br 13276,N1(C(CC(C(C)=O)(C)C)=O)CCCC2(CCN(C(=O)C(O)C(C)(C)C)CC2)C1 13277,C1(NC(c2c(C)cno2)=O)CCC(CNC(=O)Cc2csc(Br)n2)CC1 13278,CC(C)C(CNC(=O)CCn1cccc1)C(=O)NC(C)(C)CC1CCCC1 13279,Cc1c(CC(=O)NC(C(=O)N(C)Cc2ccnn2C)C2CC2)ncn1C 13280,N1(C(COCC(C)C)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13281,N1(C(C(CC=C)OC)=O)CCC(C)C(CC(=O)N(CCC(N)=O)CC)C1 13282,C1(C(=O)NCC(CCC)C)(CNC(c2nc(O)sc2C)=O)CC12CCC2 13283,C1(SCC)CC2(C1)CC21CCC1.c1(N(C=O)CC2(C(=O)OCC)CC2)cn(CC)nn1 13284,c1(OC)cc(NC2CC(=O)OC2(C)C)c([N+](=O)[O-])cn1 13285,N1(Cc2c(-c3ccc(OC)c(OC)c3C)n[nH]c2)CCC(C2CCN(C)CC2)CC1 13286,N1(C(C(CC)N(C)C)=O)CC2CCC1C(C(N1CCC(c3ccccc3)C1)=O)C2 13287,C(C)(C(=O)NC1(CCNC(=O)CNC(C)=O)CCC1)NC(=O)OC 13288,C1(C(N(CCN(C(=O)C(O)CC(N)=O)C)C)=O)CSc2ccccc2O1 13289,c1(OCC)ccc(F)cc1C(=O)N(C1CCC(C(N)=O)CC1)CC(=O)O 13290,C(C)(CCC(=O)NCCCOCc1cc(C(N(CCCSC)C)=O)no1)COC 13291,c1(CC(=O)NC(C)C(CO)NC(c2ccoc2)=O)cccc(OC(F)(F)F)c1 13292,N1(CC(=O)NC2CCC2NC(C2(F)CC2)=O)Cc2ccccc2C1 13293,Cc1nc(O)nc(O)c1CNC12CCCC1N(C(=O)CCS(N)(=O)=O)CC2 13294,N1(C(C(CC)(C)C#N)=O)CCCN(C(c2ccn(C3CC3(F)F)n2)=O)CC1C 13295,CC1CCC(c2nc(-c3ccc(COc4ccccc4)cc3)nn2CCF)OC1 13296,C1(C(=O)NC2C(NC(C(c3ccccc3)OCCC(C)C)=O)C2)CCCCCC1 13297,c1(C(=O)NCC(CC)NC(c2ccn(-c3cccc(F)c3)n2)=O)cccnc1C 13298,C12(CCNC(=O)OC3CCN(C(C)C)CC3)CCCCC1C2(F)F 13299,c1(-c2scc(C)n2)nc(C(=O)NNC(=O)OC(C)(C)C)nn1C 13300,N1(C(CN(C(C)C)C)=O)CCC(C(C)(C)CNC(=O)CC2NC(=O)NC2=O)CC1 13301,CC1CC(NC(=O)CC2CCC3(CC2)CC3)CCN1CCN1CCCCCC1=O 13302,CC(C)CC(C)(CNC(C1(O)CCC1)=O)NC(C1CC(=O)NC1=O)=O 13303,C1(NC(CCc2n(C)ncc2)=O)C2CC3C(C2)C13C(=O)NCc1nccc(O)n1 13304,C1(OCC(N2CC(C(=O)NC)C2)=O)CCCCC1C.c12cnn(c1)CCNC2=O 13305,C1(CNC(C2(C(C)C)CCC2)=O)CC(NC(=O)C=CC2CCOC2)CCO1 13306,CCC(CC(=O)NC(CN(C)C)C(=O)NCC1(O)CC2C=CC1C2)CC(C)C 13307,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)N(C)C)NCCCOCC=C 13308,N1(C(=O)OC(C)(C)C)CCC(C(N2CC3CC3(C(F)F)C2)=O)C(C)(C)C1 13309,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CNC(=O)N3C)=O)CCO2)c(C)n1 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13328,N1(C(C(c2scc(C)n2)(F)F)=O)CC(NC(c2cc(Cl)ccc2F)=O)CC(O)C1 13329,N1(CCOC)CCCC(CN(C(=O)Cc2c[nH]nc2C2CC2(F)F)C2CC2)C1 13330,N1(C(C(C)CC2CC2)=O)CC(CNC(=O)CCc2ccc(F)nc2)CC1(C)C 13331,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13332,c1(C(N(CC(CC)OC)C)=O)cn(C)nc1C(C)C.C1(=O)CCCC2(CCC2)C(=O)N1 13333,Cc1ncn(C2CN(C(c3coc(NC(N)=O)n3)=O)C2)c1C 13334,C1(CC(N2CC(C3(NC(C4CC(C)(C)C4)=O)CC3)C2)=O)CCCC2(CC1)OCCO2 13335,c1(COC(c2ccccc2C(F)(F)F)=O)nc2ccc(F)c(F)c2[nH]1 13336,c1(CC(=O)N(CCC(C)NC(COCC(=C)C)=O)C)ccc(S(=O)C2CC2)cc1 13337,C#CCC(C)(C)C(=O)N1CCOC(CCNC(=O)Cn2ccc(C)c2)C1 13338,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13339,c1(C(N2CCC(C(CO)NC(CCC=C(C)C)=O)CC2)=O)cc(S(C)(=O)=O)cs1 13340,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13341,c1(CCC(=O)NCCCC(C)NC(C2(F)CCCCC2)=O)nc2ccccc2[nH]1 13342,N1(C(c2cnc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13343,c1(C(C(=O)OCC)NC(c2cc(Br)cs2)=O)ccc(OC)nc1OCC 13344,Cc1ccc2[nH]c(C(=O)NCCOCC(=O)NCCN(C)C)cc2c1C 13345,Cc1nc(C(C)(F)F)ccc1C(N1CC(NC(C23CCCC2C3)=O)C(C)(C)C1)=O 13346,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)CC1O 13347,c1(-c2n(C)cnc2)ccc2c(c1)CN(Cc1ccccc1I)CC2 13348,C(=O)(CC(C1CC1)NC(=O)CN1CCCCC1)OC.C12C=CCN1C2=O 13349,N1(c2nnc(C(CC)(C)C)o2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13350,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(C)N1CCC1 13351,C1(OCc2onc(CC)n2)CC2N(C1)C(=O)CCCOC2=O.C1(OCC)CCC1 13352,Cc1cc(NC(C2(C)CC(O)CN2C)=O)ccc1NC(c1snc(C)c1N)=O 13353,C=CCCCCCC(=O)NCC(CCCC)NC(=O)C(N1CCCCC1=O)C 13354,N1(c2n(CC(=C)C)c(-c3ccc(CC#N)o3)nn2)CCCC(SC)CC1 13355,C1(NC(C(C)(F)C(F)(F)F)=O)CCCC2CN(C(=O)C=CC(=O)N(C)C)CC12 13356,C#CC1(C(=O)NC(c2ccncn2)C)CCN(C(=O)C=Cc2nccs2)C1 13357,Cc1noc(C(F)(F)F)c1C(=O)NC1CC1CNC(=O)CCc1cnccn1 13358,c1(SCc2cn(CCCC(=O)NCC(C(C)(C)C)O)nn2)c[nH]c(=N)nc1O 13359,C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C=C(CCC)CCC)CC1C 13360,C(=O)(C(CCSC)NC(=O)CCC(C)N(C)C)N1CC(C#C)C1 13361,C(=O)(C(C)NC(C1(C(F)F)CC1)=O)N(C(CC1CC1)C(=O)OC(C)(C)C)C 13362,C1(CCCOC)(CNC(c2coc(O)n2)=O)CCCC1.C1(=O)C(C2CCOC2)N1 13363,c1(SCC(=O)NCC(C2CC2)NC(COCCCC(C)C)=O)ccc([N+](=O)[O-])cc1 13364,NS(=O)(=O)CCCC(=O)NCC1CCCCN1C(=O)CCN1CCCCC1 13365,N1(C(C(C)NC2C3CCCCC23)=O)CCC12CC(NC(=O)C(C1CCOCC1)O)C2 13366,C1(CNC(C=CC(=O)OCC)=O)CN(C(=O)CC(C)(C)c2ccccc2)CCO1 13367,C(CC(C(C)(C)C)NC(c1cnn(C(C)(C)C)c1N)=O)N(C(C(CC=C)C)=O)C 13368,c1(C(=O)NCC2CN(C(c3c(C)nncc3)=O)CC23CC3)cnc2[nH]nnc2c1 13369,c1(C(=O)NCC#CCNC(Cc2cc(C)on2)=O)nc2c(s1)CN(C)CC2 13370,C1(SC)CN(C(=O)CCc2cncs2)CC1NC(=O)CN1CCCCCC1 13371,C(C)(C)(CC(=O)N(C)CCN(C(=O)CC1CCC1(F)F)C)c1cncc(SC)c1 13372,c1(C(N(C(C)CN(C(=O)CCCCc2cnc[nH]2)C)C)=O)cnc2ncccn12 13373,c1(CN2C(C(N3CCC(Cc4ccc(Cl)cc4)C3)=O)CC2)cccc(O)c1 13374,C#Cc1cnn(CC(=O)NCC2CC2CNC(c2ccc[n+]([O-])c2)=O)c1 13375,C#CCC(C)(C)C(=O)NC1CCC(CNC(C2CCCOC2)=O)C1 13376,c1(C(N2CC3(CO)CCC2CC3)C(=O)NCC2CCOC2)ccc2cc[nH]c2c1 13377,c1(CC)nn(C)cc1C(C(=O)NC1(C)CC1)N(C(C)C)CC1CCCCC1 13378,C1(c2n(C(C)C)cnn2)CCN(N2CCC(CCc3ccccc3)C2)C1 13379,CC(C(C(=O)N1CC(C)(N)C(C)C1)N1CCCC(O)C1)C(C)(C)C 13380,C1(F)(C(N2CC(N(C)C)C(F)C2)=O)CCN(C(c2ccccc2C(N)=O)=O)C1 13381,c1(N2CC3CC(N(C)CCNC(=O)C4CC4)C3C2)nc(Cl)nc2ccccc12 13382,C=CCCCC(=O)NCCS(=O)(=O)Cc1cn(CCN2CCCC2=O)nn1 13383,c1(C(N2CCN(C(CC(C)(C)F)=O)CC2CCO)=O)cc2ccncc2cc1F 13384,c1(CC(=O)NC2CN(C(c3cn(CC)nn3)=O)C3C2C3)cc(C)ccc1OCC 13385,C(N=c1[nH]c(=NCC2COCCC2(F)F)c2[nH]ccc2[nH]1)c1c(N)cccc1F 13386,C(=O)(C(F)(F)CO)NCc1cc(C(=O)NCCCCCSC)n[nH]1 13387,C(=O)(CC(C(F)F)n1ccnc1)N1CC(O)(CC(N2CCC2Cn2cccn2)=O)C1 13388,c1(CNC(C(n2cc(-c3ccccc3CN)nn2)C)=O)cccc(C(F)(F)F)c1 13389,c12nccc(Br)c1OCCN2.CCC(Cn1cncn1)N(C)C 13390,c1(C(N(CCCCN(C(=O)Cc2ccn(C)c2)C)C)=O)csc(C(C)(C)C)n1 13391,C1(CC)(NC(=O)CCOCCN(C)C(C2CCN(C)C2)=O)CC(C)(C)C1 13392,C(C(CC(C)C)C(=O)N1CC=C(C(=O)NCC2CCC(C)CO2)CC1)OC 13393,C1(C)(C)CCC2CC2C1.S1(=O)(=O)CC(=O)NCCCC2(CC2)NC1=O.CC(C)(C)N 13394,N(C(=NCC1CCCO1)NC1CC(c2ccc(F)cc2)C1)CC1(C)CCC1 13395,c1(OC)ccc(C(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)c(C)n1 13396,CC(C)C(C#N)C(=O)NCCN(C(=O)CC1CC1C1CC1)Cc1ccccc1 13397,c1(CN2CC(F)(C(=O)NC34CC(C(N)=O)(C3)C4)C2)cccc(O)c1 13398,CC#Cc1ccc(C(N2CCN(C3CCCO3)CC2)C(=O)NCC2CC2)cc1 13399,C(CC1=CCCCC1)N(C(c1cc(C(F)(F)F)cs1)C(=O)NCCC)C 13400,N1(C(c2cnc(C)nc2C2CC2)=O)CC2CC1CCN2C(=O)CC(C)(C)C 13401,c1(C(=O)NC(C)CNC(c2conc2-c2ccccc2)=O)ccc(C(F)F)nc1 13402,N1(C(CCC)=O)CCC(C)CC1NC(=O)C(c1cnn(C)c1)C 13403,O=C(C1=CCCSC1)NCCCCCCNC(C1COCC1C(F)F)=O 13404,C1(CNC(COC2(C)CCCC2)=O)CCCCN1C(C1(C2CCC2)CC1)=O 13405,c1(C(N(C)CCOCCNC(C2CCC23CCC3)=O)=O)cc2cccnc2cn1 13406,C1(NC(CSc2n[nH]c(=NC)s2)=O)COCCN(C(C2CCCC(F)(F)C2)=O)C1 13407,N1(C(C)C(=O)NCCCn2ncnn2)CCN(c2ccccc2)CC1 13408,C(=O)(CCN(C1CCCC1)C)N(CC(C)N(C(CC1(CSC)CC1)=O)C)C 13409,C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(=O)CN2CCCC2)CC(C)O1 13410,C1(NC(CC2N(C(C)C)CCC2)=O)CN(C(=O)CCOC2CCOCC2)CC1C 13411,c1(C(=O)NC2CCN(C(CC(C)CF)=O)C23CC3)ncnc2c1CCC2 13412,c1(NC(C(C)(C)NC(c2c(C)ncs2)=O)=O)ccc2nncn2c1 13413,c1(CNC(C(C(C)(C)C)O)=O)ccc2c(c1)CN(C(=O)C1=CCCOC1)C2 13414,N1(C(C2(C)N(C(C)C)CCC2)=O)CCC(C(=O)NCCOCCF)C(C)(C)C1 13415,c1(C(=O)NC(C2CCCC2)CNC(C2C(C)=C2)=O)c(C)cc(C#N)cc1C 13416,CN1CC=C(C(=O)N2CCC2CNC(=O)CC2CC3(COC3)C2)C1 13417,c1(C(N2CC(C(N)=O)(CNC(C(C)n3cncn3)=O)C2)=O)ccnc2[nH]ncc12 13418,c1(OC)ccc(-c2cc(NC(C3(CSc4ccccc4)CC3)=O)ccn2)c(C)c1 13419,Cc1[nH]nc(Cl)c1C(=O)NCCCCNC(C1CCCCC1OC(F)F)=O 13420,N1(C(C(CC)(CC)CO)=O)CCOC2(CCCN(C(=O)CCCC3CC3)C2)C1 13421,c1(C(C)C)ccc(C2CC2C(=O)NOCCN(C)C)cc1 13422,c1(C(=O)NC2C(NC(CCC=C)=O)C2)ccc(NC=O)cc1.C1CCN1 13423,Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(F)CNC(c1c[nH]c2cccnc12)=O 13424,C(=O)(C(C)(C)C(C)NC(C1CCCCC1O)=O)NC(c1cccc(C)n1)C 13425,C1(C(=O)NCC2(C)CC(NC(C3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13426,c1(CNC2CCC(C(N3C(COC)COCC3)=O)CC2)cc2ccccc2s1 13427,N1(C(C2CCSCC2)C(=O)NCCOCC)C2CCC1CC(C(C)(C)C)C2 13428,C1(NC(C2(C)CCN(C(c3ccc(C(F)(F)F)nc3)=O)C2)=O)CCC(F)(F)CC1 13429,CC(C)(O)C(C)(C)C(=O)N1CCCC1CNC(C1OCC2CCCC12)=O 13430,C1(C)(OCC(=O)N(C2(NC(=O)CCCC3CCCC3)CC2)C)CCCC1 13431,C(=O)(CC(CC)N(C)C(c1ccn(C)c1C)=O)N(CC=C)C1CC1 13432,c1(C(=O)NCC(C)NC(CC(C)C(F)F)=O)cc2ccc(Br)cc2s1 13433,C(=O)(C#Cc1ccccc1)N1CC2C(C(=O)Nc3cc(OC)cc(F)c3)C2C1 13434,C1(C(=O)NC2CC(C(F)F)(NC(C(C3CCC3)CC)=O)C2)CC(C)CC(C)C1.O 13435,CC#CCC(C)NC(=O)C(C1(O)CCC1)NC(=O)CC(C)c1ccco1 13436,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(N)cnc1Cl 13437,c1(C(N2CC(NC(=O)C(F)C3CCC3)(CO)C2)=O)cncc([N+](=O)[O-])c1 13438,C1(C(F)(F)F)(C(N2CC(NC(CC3(C)CCCC3)=O)C2)=O)CC2CC2C1 13439,C1(C(=O)NC2CC(NC(C=C(C)C)=O)CC2O)C(F)(F)C12CCC2 13440,c1(C(N(CCCNC(C(C)OCC)=O)CC)=O)ccc2nccnc2c1 13441,C(C1=CCCOC1)NC(C(c1cccs1)NC(c1cc(CO)on1)=O)=O 13442,N1(C(C=C(C)C)=O)C2CCC1C(CNC(=O)C(F)F)C2 13443,Cn1ccc(C(=O)NC(C2CCOC2)CNC(c2ccsc2)=O)c1C1CCC1 13444,C(C)(C)(CC(=O)NCc1ccccn1)NC(COCC(C)C)=O 13445,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCCO3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13446,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)CC1(c2ccccc2Cl)CC1 13447,N1(C(C(C)OCC=C)=O)CCSCC1C(N1CCC(CF)CC1)=O 13448,C#CC1(NC(=O)CC2CN(C(=O)CCN(C3CCC3)C)CCO2)CC2CCCC12 13449,C12(NC(C(C)SC(C)C)=O)CC1CN(C(c1cc(-n3cccc3)ccn1)=O)C2 13450,C(=O)(C(CC(C)C)N(C)C)NCC(=O)NCc1cncc(C)c1 13451,N1(C(C2C(C)=C2)=O)CC2CC2(CNC(c2ccc(CC(C)C)cc2)=O)C1 13452,n12cc(cn1)S(=O)(=O)N(C)C2.N1(CC)CCC(O)CC1C 13453,N1(C(c2c(C)nc(O)cc2)=O)CC2CCCC1(CNC(C1(CO)CCCC1)=O)C2 13454,N1(C(C(n2c(C)ccn2)C)=O)CCCC(N(C)C(c2ccnc(N(C)C)c2)=O)C1 13455,CCCCCC(C)CC(=O)NC1CC(NC(C2C(C(F)(F)F)C2C)=O)C1 13456,C(=O)(CC(C)(C)O)N(C(C(N1CC(C(=O)NC)C1)=O)C)C 13457,Cc1cc(C(=O)N(CC(C)C(=O)N2CC(N(C)C)C2)N(C)C)cn1C 13458,C(=O)(C(CC(C)C)N(C)CC1(O)CCSC1)NC(CC)C 13459,C1(C(=O)NCC2N(C(c3c(C)cnnc3)=O)CCN(C)C2)CCc2cnnn2C1 13460,C(=O)(CCCCC(=O)N1CC(NC(=O)CC2C(C)(C)C2(C)C)CC(C)(C)C1)OC 13461,c1(CNC(CCN(C(=O)CC2CC(C)=NO2)CC#C)=O)cccc(F)n1 13462,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)SC2CC2)CC1)NC 13463,C1(CN(C)C(C2(C)CCC2)=O)CCCN(c2nc(Cc3ccccc3)ns2)C1 13464,C1(C)(CNC(C2N(CC)CCCC2)=O)CN(C(=O)CCCCC2CC2)C(C)(C)C1 13465,C1(N)(C(=O)NCC(=O)Nc2cc(CC)ncn2)CCC(C)(C)CC1 13466,CC1CCC(OC(c2ccc(-n3cncn3)c(F)c2)=O)C(=O)N1 13467,c1(OC)ccc(C(=O)NCC2(C)CCCN2C(c2cnc(C)[nH]2)=O)c(N)c1 13468,Cn1nc(Cl)c(C(N2CC(CNC(=O)CSc3nncs3)C(F)(F)C2)=O)c1Cl 13469,N1(C(C2(CCC)CCOC2)=O)C2CCC(C2)C1CC(=O)N(C(C)CCC)CC 13470,Nc1ccc(C(=O)NCC2(NC(=O)C=Cc3cccnc3)CCOCC2)nc1N 13471,c1(C(=O)NCCC(C)NC(c2cc(F)c(F)c(F)c2)=O)cc2n(c1)CCCC2 13472,CCC(CC(=O)NCCC1CC(NC(C2CCCSC2C)=O)C1)c1ccccc1 13473,c1(C(C(=O)O)N(CC)Cc2cc(Cl)sc2Cl)ccc(Br)cc1F 13474,C1(C(=O)NCC2C(NC(c3c(C)nc(C)nc3)=O)CC2)CCCCC12CCC2 13475,C(=O)(C1CCCc2nncn21)NC1(C)CCN(C(=O)Cc2cccnc2Cl)C1 13476,c1(CN2CCC(O)(n3cc(-c4cccc(C(C)C)c4)nn3)C2)cc(Br)ccc1Br 13477,C1(NC(c2cc(Cl)cnn2)=O)C2CCC1N(C(=O)Cc1cccc(F)c1O)C2 13478,N1(C(C(COCC)C)=O)CCN(C(c2cnn(C)c2C2CC2)=O)CC1C(C)C 13479,N1(C(CC=C)=O)CC(C(c2cnn[nH]2)OC)C(C)C1.C12(COC1)CC(=O)N2 13480,c1(C(C)(C)C)cccc(C(=O)NC2CCC(CNC(=O)CCc3cscn3)C2)n1 13481,C1(NC(c2c(Cl)cnc(CC)n2)=O)COC2(C1)CN(C(=O)C=Cc1ccc[nH]1)C2 13482,N1(CC(=O)OCC)CCCC(F)(NCCCCN(CCCSC)C)C1 13483,N1(Cc2cccc(C#N)c2)CC2CC(NC(=O)CCCc3cccnc3)CC2C1 13484,CON(CCC(=O)NOCCOCCSCCC(F)(F)F)C(=O)C1=C(Cl)CCC1 13485,N1(C(C2C(CC)OCC2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)(F)F)C1C2 13486,N1(C(c2cn(C)nc2)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C12CCC2 13487,N1(C(C(=O)NCC)=O)CC(F)(CNC(C2(CC)CC2(F)F)=O)C1 13488,N1(C(C(C)=CC=C)=O)CCC(NC(=O)CN(C)C(=O)C2CC2)C(F)C1 13489,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-c2ccncc2)ccn1)=O 13490,N1(C(Cc2c(C)ncs2)=O)CC2(CCC2NC(=O)CC2COC(C)(C)CO2)C1 13491,c1(C(N(CCNC(=O)C(C)=C2CCC2)CC)=O)cnn(-c2ccncc2)c1C 13492,c1(C(N(C2CCCC2)CCCNC(C2C(C)(C)CC2)=O)=O)cc[n+]([O-])cc1 13493,c1(OC(C2CC(N(C)CC)C2)=O)ccc(F)cc1Br.C1(SCCNCC)CCCOCC1 13494,C(N=c1[nH]cnc2ccc(O)cc12)C1CCC(NC(C23CC=CC(C2)OC3)=O)C1 13495,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13496,CC12COCC1CN(C(C1CNC(=O)CN1C(=O)CC1=CCCCC1)=O)C2 13497,N1(C(C2(CN(C)C)CCCN2)=O)CC2CC(F)(F)C2C1 13498,N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)CCc2nccs2)C(C)CC1C 13499,C1(CC)CCCC(N=c2nc3sccc3c(NCC3=CCN(C)CC3)[nH]2)C1 13500,c1(C(=O)NC(CC)CN(C(=O)CSCc2cccnc2)C)cn(C)nc1C(C)C 13501,C1(NC(C(C)Cc2ccco2)=O)CN(C(=O)C=Cc2ccccc2)CCC1C 13502,Cc1nn(C)c(Cl)c1C(=O)NCC1CC2CC1CN2C(=O)CC1CC2(CC2)C1 13503,Cn1nc(C(F)F)cc1NC(=O)NCCC(O)C(=O)NC1CCCCC1 13504,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13505,N1(C(c2c(C)ccnn2)=O)CC2(CC(NC(C34CC3COC4(C)C)=O)C2)C1 13506,c1(C(=O)Nc2c(OCCOC)cc(C(=O)OC)cc2)cc2n(n1)CCCN2 13507,C(=O)(C(F)(CNC(c1cnns1)=O)C(C)C)NC(CC(=O)OCC)C 13508,c1(C(=O)OC)[nH]c(=NC2CCCCCN(C(C3(O)CC3)=O)C2)sc1C 13509,C1(CNC(C2CN(CC(C)C)C2)=O)CN(C(=O)C(C)N2CCCC2)CC12CCC2 13510,c1(N2CCCC(C)(C(=O)NC)C2)nc(SCC(OC)OC)nc2sccc12 13511,CC(CCCC(=O)N(C)CCO)NC(=O)CC.c1(C2(C)CC2)ccccc1F 13512,C1(C)(CNC(C2CCCC(C)C2)=O)CCCN(C(c2cccc(F)c2)=O)C1 13513,c1(C(=O)NCCN(C(=O)CCC2CC2(F)F)CC(C)O)cnn(C)c1 13514,c1(CC)[nH]ccc1C(=O)N(CC(=O)N(C)C(C1CCC1)C)C1CC1 13515,c1(CCCC)ccc(C(c2nnnn2C)NC(c2cncs2)C)cc1 13516,Cc1csc(C(=O)NCCCn2cc(C3CCN(C)C3)nn2)c1C 13517,C1(C(N2CCOC(C(F)F)CC2)C(=O)NCCCOC)Cc2ccccc2O1 13518,N1(C(C(C)(C)C(F)F)=O)CC2COCC(C1)C2NC(=O)CC1CCOC1=O 13519,C1(C(=O)NCC2C(CNC(CSCC(=O)OC)=O)C2)CC(C(C)C)=NO1 13520,c1(CC)ncc(C(=O)NC(CNC(C2CC3C=CC2O3)=O)CCOC)c(O)n1 13521,C1(CC(=O)NCC(N2CCCCC2)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)C1 13522,C1(OC)CCCN(CCOc2ccccc2)C1.C1(Cc2ccccc2)C(=O)N1 13523,Cc1cc(C(=O)NC(C2CCN(C(=O)C#CC(=O)N(C)C)CC2)C)ccn1 13524,C1(N(C(=O)C=CC2CCCO2)C)CCCN(C(C2CCOCC2)=O)CC1 13525,c1(C(N(C)CC2CCCN2C(c2cc(Br)c[nH]2)=O)=O)ccc(C#N)cn1 13526,c1(C(=O)NC(CNC(C2C(OCC)C2C)=O)C)cnc2c(c1)nnn2C 13527,n1(C(CC)C)nc(CCOCC(F)(F)F)nc1-c1ccccc1OC 13528,Cc1coc(C)c1CNC(=O)C(C)N(C(=O)Cc1ccccc1)C1CC1 13529,c1(OC)cnc(Br)cc1NC(C1CC1NCc1c(I)ccnc1OC)=O 13530,C(=O)(C(F)C(C)(C)O)OCCc1nnc(SCC(C)C)s1 13531,c1(CC(=O)NC2CC(NC(=O)C(F)=CC3CC3)C2)noc2ccccc12 13532,Cc1cc(C(=O)NC2CCCC(NC(C3C4(CC4)C34CC4)=O)C2)cc2ccsc12 13533,C(=O)(N1CCCc2ccnn21)C12CC(NC(c3n(C)nnc3)=O)C(OC1)C2 13534,C1(CC(N2C(CNC(c3cn(CCO)nn3)=O)CC2)=O)CC(=O)c2ccccc2C1 13535,C#Cc1ccc(C(=O)OCC(C)C(C)NCCC(C)F)nc1 13536,C1(CNC(CCCOC(C)C)=O)CCN(C(=O)C(C)Sc2ccccc2)CC1C 13537,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13538,N1(C(CN(C(COC)=O)C)=O)CC2CC(C(=O)NC3CCCN3C(C)C)C(C2)C1 13539,C1(NC(CSCCNC(c2cn(CC)nc2)=O)=O)CCCC12CC2 13540,C1(NC(Cn2ncn(C)c2=O)=O)CCN(C(=O)CCc2cnc(O)[nH]2)CC1O 13541,C(=O)(C(C)(CC)C(N)=O)N1CCCC(N(C(=O)COc2cc(F)ccc2F)CC)C1 13542,n1(CCOC)cc(C(=O)NCC(O)CCNC(=O)CSCC(N)=O)c(C)n1 13543,C(=O)(CCCOCC(c1ccccc1)C)NCCNC(C1(CSC)CC1)=O 13544,C=C1CC2(C1)CN(C(=O)C(CC(C)C)N(C(=O)CC#N)C)C2 13545,C1(C(=O)NC2(C(C)C)CCC2)CCC2(CC2)N1C(c1cnc(O)o1)=O 13546,N1(C(C(C)CC2CC2)=O)CCCC(C(=O)NC(C)(C)C(F)(F)F)CC1 13547,C1(C)(CC)NC(=O)N(CC(=O)OCCOc2ccc(Cl)cc2C(C)C)C1=O 13548,c1(COCC)cn(CC(=O)NOCC2CCN(C)C2)nn1 13549,CCC(CC(C)C)C(=O)NCC1CN(C(c2ccc(C#N)nc2O)=O)CCO1 13550,CC1CCC(C(=O)N(C)Cc2nnnn2C)N1C(c1ccn(C)n1)=O 13551,N1(C(c2[nH]c(=NC)sc2)=O)CC(N(C(=O)C(C)SC(C)C)C)C(C)(C)C1 13552,C=CCCCC(C(=O)N1CCN(C(=O)C2=CC(C)(C)C2)CC1)c1ccccc1 13553,Cc1ncc(C(=O)NC2C=CCN(C(c3c(C)noc3C3CC3)=O)C2)cc1C#N 13554,CCCCCC(CC)C(=O)NC1CC2(C1)CC2NC(=O)CN1CC(=O)NC1=O 13555,c1(C(=O)OC)c(F)ccc(-c2cnc(-c3cccc4c3OCO4)c(C)c2)c1F 13556,N1(C(c2cnc(OCC)s2)=O)CCCC(O)(CNC(=O)C2=C(Cl)CCOC2)CC1 13557,Cc1cc(NC(c2ccc(CNC(c3cnns3)=O)s2)=O)c(O)cc1F 13558,c1(CC)ccnc(C(=O)NCC(C(=O)Nc2c(OC)noc2C2CC2)OC)c1 13559,C12(CNC(C3(CO)CCC3)=O)CC1CN(C(=O)COC1CCC1)C2 13560,N1(C(C(CCC(C)C)N(C)C)=O)CCCC2C1CCCCN2C(=O)CC1CC=CC1 13561,C(=O)(C(F)C(F)(F)F)NC(CC1CCN(c2cc(CC)ncn2)CC1)C1CC1 13562,N1(Cc2c(C(=O)O)cc(Cl)cc2)CCCC2C1CCN2C(=O)CN1C(=O)C=CC1=O 13563,N1(C(=O)CNCc2ccc(Br)cc2F)CCCc2c(C(F)F)cccc21 13564,N1(C(C(C)C)=O)CC(C(=O)Nc2c(-c3cccc(F)c3)noc2C)CC12CCC2 13565,C1(CC)C(NC(=O)C=C(C)CN(C)C)CCN1C(c1ccncc1C(F)F)=O 13566,c1(OC)cncc(C(=O)OC2CCN(c3nccc(-c4cccc(C)c4)n3)C2)c1 13567,CCC(CC(=O)N1CC2CN(C(c3c[nH]nc3-n3cnnn3)=O)CCC12)C(C)C 13568,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13569,C1(CNC(c2c(C)nsc2C)=O)C(C)CCCN1C(c1ccc(C)cc1F)=O 13570,C(C(C)(C(C)C)C(C)C)NC(C1CN(C(C2(CO)CCCC2)=O)CC(C)O1)=O 13571,c1(C(=O)NC(C)CC(C)NC(C2(C)CC(F)(F)C2)=O)ccc2cc[nH]c2c1F 13572,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1[N+](=O)[O-] 13573,c1(C(N(CCNC(C(N)=O)=O)C2CC2)=O)cc2c(O)ncnc2cn1 13574,c1(CC)nccnc1C(N1CCCCC1CN(C)C(C1(C)CCC(=O)N1)=O)=O 13575,C(C(C)(C)CNC(C1CCCN1C)=O)N(C(=O)C(=O)C1CCCC1)CC 13576,c1(C(=O)N(C(CNC(C2CN(C(C)=O)C2)=O)C)C(C)C)ccc(C)c(Br)c1 13577,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)CC1CN(C)CC1O)=O 13578,C1(NC(Cc2c(C)ocn2)=O)CCN(C(c2cccc(C(C)(C)C)c2)=O)C(C)C1 13579,Cc1conc1CC(=O)N(CC(=O)N(C)Cc1cccnc1)CCO 13580,c1(OC)cc(Br)cc(C(=O)NC2COCCC2NC(=O)Cn2cncn2)c1N 13581,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2o1 13582,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)CC2COC(C)(C)C2)C)cc(O)n1 13583,c1(C(=O)NCC2CC3COCC23)ccccc1OC1CCOC1 13584,c12cccc(c1)C(=O)NCCS2.c1(C(N(C)SC)=O)cnc(S)[nH]1 13585,c1(CNC(=NC)NC2CC(OC(C)C)C2)ccccc1Cl.C1CO1 13586,Fc1ccc(F)c(-c2ccc3nc[nH]c3c2F)c1F 13587,C(=O)(C(C)(C)C(N)=O)NCCC1C(C)CN(C(=O)COCc2cccnc2)C1 13588,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cnc(O)cc2C)cc1C 13589,Cc1cc(C(=O)NC2CCCN(C(C3CCN(C)C3)=O)C2)cc([N+](=O)[O-])c1O 13590,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13591,C(=O)(C1=CCCOCC1)NC(C(=O)NCC(C1CC1)OC)C1CCOC1 13592,C1(C(=O)NC(CNC(c2scc(C)c2)=O)CO)CCCN(C(C)C)C1 13593,C(=O)(C(C)(C)CNC(=O)C=C1CCC1)N(CCCC)CCOC 13594,n1(CC(C)NCCCC(C)(C)CO)cnc2c(cnn2C)c1=O 13595,N1(C(c2c(CC)c[nH]n2)=O)CCC2C(C(=O)NC(c3noc(C)n3)CC)C2C1 13596,CN1C(=O)Cc2ccc(C(N3CC4(CCC4)CC3CNC(=O)CCC#N)=O)cc21 13597,CCCCCCCC(CC)NC(C1CCN(C(c2cccc(O)c2F)=O)C1)=O 13598,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13599,CCCC(O)(CNC(c1c[nH]nc1C1C(C)CCN1C(=O)C(C)C)=O)CCC 13600,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13601,C=CC(F)(F)C(=O)NCC(O)CC(=O)N(C)CC1CCOC1C 13602,c1(C(=O)NCCNC(c2cnn(CC)c2C2CC2)=O)ccc2[nH]c(=N)sc2c1 13603,C1(CNC(Cc2cn(C)nn2)=O)COCCN(C(c2cnn[nH]2)=O)C1 13604,c1(C(=O)NC(CC(C)NC(c2c(OC)ccs2)=O)C)ccc(-c2cccs2)cn1 13605,C1(C(N2C(C(=O)NC3CCCC3F)CC(OC)C2)=O)CC2(CCC2)CO1 13606,N1(C(CNC(CNC(c2n(C)cc(Cl)c2)=O)=O)=O)CCOCC(C)(F)C1 13607,Cc1nc(CC(C)C)oc1C(=O)NCC(O)CCNC(C1(C)CC(F)C1)=O 13608,C1(COC)(NC(=O)CC(c2cccc(Br)c2)C)CCCNC1 13609,N1(C(C(C)n2ccnn2)=O)CC(C(=O)NCc2ccnc(F)c2F)C2(CCC2)C1 13610,N1(C(=O)OC(C)(C)C)CCc2nc(C(=O)NC3CCC=CCC3)cn2CC1 13611,c1(C(=O)NCC2(CNC(=O)C(C3CCOC3)OC)CC(=C)C2)cnc(C)n1C 13612,Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C2=CCC(C)CC2)cc1C 13613,Cc1cc(CC(=O)NC(CNC(=O)Cc2[nH]cnc2C)C(C)C)n(C)n1 13614,C1(C2CCC2)(C(=O)NCC(C)N(C(=O)COc2cccnc2)C)CC1(F)F 13615,C1(CNC(C(C=C)C)=O)CN(C(c2cc(C)cs2)=O)CC12CC2 13616,O=C1CCC(S(=O)(=O)N(CC(O)CC2CN(C(=O)C3=C(Cl)CC3)C2)CCO)CC1 13617,Cc1nnc2n1CC(CNC(=O)CCn1cncc(Br)c1=O)CC2 13618,C1(CC)CC(C(N2CCCC2(CNC(C2CCOCC2)=O)COC)=O)CC(=O)N1 13619,Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(C(F)F)cs3)=O)C2)cnc1O 13620,C12(C(N3CCC(NC(COCCCCOCC#C)=O)C3)=O)CC(C1)C(C)O2 13621,CCCC(C)C(=O)NC(C)(C)C(=O)NC(c1ccc(Cl)cc1)CCC(=O)NC 13622,c1(-c2onc(C(=O)NCC(C)NC(=O)C(C)(C)c3cncnc3)n2)cccc(Cl)c1 13623,c1(CC)sccc1C(=O)N(C(C)C(C)OC)CC 13624,C1(CC(=O)NC(CCN(CCOc2cc(C)on2)C)=O)CC(O)C1(C)C 13625,N12CCN(C(C)C1)C(=O)c1noc(C(=O)OCC)c1CC2=O.C1(CC)(CC)CC1 13626,C1(CNC(C2(C#C)CCCC2)=O)CN(C)CCN1C(c1cc(CC)on1)=O 13627,C(C(CC(=O)NC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)C(F)(F)F)N(C)C 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13646,C1(CNC(CCCOCCC)=O)CC2CCC1N2C(=O)C(N)=O 13647,CN1CCn2cc(C(N3CCCC4CN(C(C5(C)CC5)=O)CCC34)=O)nc2C1=O 13648,C(=O)(C(C)S(=O)(=O)C(C)C)NCCCCC(C)NC(c1c(C)onc1Br)=O 13649,N1(C(=O)CC2CC2)CC2CC(C(N3CC(CC45CC(C4)C5)C3)=O)(C2)C1 13650,CC1CC(NC(c2c[nH]c(Br)c2)=O)CN1c1cc(C(F)F)ncn1 13651,C1(C(=O)NCCC2(NC(CSCCC)=O)CCC2)COC(C)C1 13652,N1(C(c2ncn(C)c2)=O)CCCCC(NC(C2OCC3CCCC23)=O)C1 13653,CCCCCCCCNC(=O)CCNC(=O)CNC(=O)C(C)C#N 13654,C1(NC(c2c(OC)ccs2)=O)CC2CCC1CN(C(=O)CN(C)C(N)=O)C2 13655,c1(C(N(CCN(C)Cc2noc(C(C)(C)C)n2)C)=O)ccc2c(c1)N(C)C(=O)CO2 13656,C1(C(C)C)(NC(c2ccc(NS(C)(=O)=O)cc2)C)CNC(=O)C1 13657,C(=O)(CCCC(OC)OCC)NC(C1CN(CCC)C(=O)C1)=O 13658,C1(NC(c2ncc(Cl)cn2)=O)CC12CCN(C(c1ccc3cc[nH]c3c1)=O)CC2 13659,c1(-c2onc(C)n2)ccnc(Nc2cc(NSC3CCCCC3C(N)=O)ncn2)c1 13660,C(=O)(C(CO)NC(=O)CC1CCOC1C)NC(C)CCF 13661,c1(C(=O)NCC(CNC(CCSC)=O)O)c2c(nn1C)CCNC2 13662,c1(C(=O)NCCNC(C2C(C(N)=O)C2)=O)ccnc2ccc(O)cc12 13663,c1(C(N2CC(CNC(C3CC3F)=O)CC(C)(C)C2)=O)ccc2c(c1)NS(=O)(=O)C2 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13682,N1(C(CC(CC)C)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)C2CC12 13683,C1(NC(=O)CNC(=O)C2CC2)CCCC(NC(c2c(Cl)cncc2Cl)=O)CC1 13684,C1(C2CCCN(C(C3C=CCC3)=O)C2)(NC(=O)CN2CC3CC3C2)CC1 13685,C1(C(=O)NCC(C(C)O)O)CCCN1NC(=O)c1c[nH]c2cccnc12 13686,C1(C(N2C(c3cc(OC)n(C)n3)CCC2)=O)CCN(S(=O)(=O)N(C)C)CC1 13687,Cc1cc(CNCC2COCCN2C(C2CC(O)CN2C)=O)c(O)c(Br)c1 13688,N1(C(c2c(C)nns2)C(=O)NC2CCC2)CC(C#N)(c2ccccn2)C1 13689,C1(CC=C)(C(=O)NCC2CCN(CC)C2)CCCN1C(c1nonc1N)=O 13690,c1(N2CCCC(CN(C)C)C2)nc2ccccc2nc1NCC1CCC1(F)F 13691,c1(NC(C=Cc2c(Nc3cc(OC)cc(F)c3)cccc2)=O)ncc2cn[nH]c2n1 13692,c1(N2CCOCC(CC)C2)nc(=NCCc2cc[nH]n2)[nH]c2c1CC(C)CC2 13693,C=C=CCC(=O)NC(C(=O)NCc1cnn(CC)c1)C1(C)CC1 13694,c1(Nc2cccc(Br)c2)cc(C(=O)O)nc(C(F)(F)F)c1.CC1CC1 13695,C1(CC(N2CCC(C(C)NC(=O)CC3CC4CC4C3)C2)=O)CCCNC1=O 13696,C1(O)(CN(C)C(c2sncc2Br)=O)CCN(C(c2c[nH]cc2C2CC2)=O)C1 13697,c1(C(=O)NC2C(C)CN(C(=O)C(C3CCOCC3)C)CC2)c(F)ccc2occc12 13698,N1(C(C(CSC)OC)=O)CCCC(C2CCN(C(=O)C3CCc4nccn43)C2)C1 13699,N1(C(c2onc(COC)n2)C)CC(NC(c2cccc(Cl)c2C)=O)C(C)(C)C1 13700,C1(C(N(C(Cc2ccc(OC)c(Br)c2)C(=O)O)C)=O)CCc2nccn2C1 13701,N1(C(c2ccc(N(CCCC)C)cc2)=O)CC2CC1CCN2C(=O)CCS(C)=O 13702,C1N=C2N=c3sccc3=C(N2)N(C)C12CCC(C)CC2.C(COC)SC 13703,C=Cc1cc(C(N2CCC(NC(=O)CCSCCCC)C2CC)=O)cc(F)c1 13704,c1(NC(NC2CCN(CC)C2)=S)ccc(C2CCNCC2)cc1 13705,c1(C(=O)OC)cccc(CNCCC2CCCN(Cc3ccccc3)C2)n1 13706,C#CCC(CC(=O)Nn1cnn(C)c1=S)NC(c1cnc(O)o1)=O 13707,c1(N2CC3C(CNc4ncc(CC(=O)OC)[nH]4)(C3)C2)cc(F)c(C)cn1 13708,C1(NC(C=C(C)C(F)F)=O)(CO)CC1(C)C.C1(=O)CCOCCCN1 13709,C1(NC(CCC=CC(C)C)=O)CCCC(N(C)C(c2csc(C(N)=O)n2)=O)C1 13710,c1(NC(=O)NCC(CNC(=O)Cc2nnc(O)s2)OC)ccccc1C 13711,c1(NC(C(=O)NC(C)CCn2cncn2)=O)ccc(I)cc1Br.C(C)(C)(C)O 13712,C(C)(CCCNC(=O)COCCOCCO)N.C1CCC1C(=O)OC 13713,C1(SCC(N2CC(C(C)NC(=O)CCc3nncs3)C2)=O)CCS(=O)(=O)C1 13714,C1(NC(CN2CCC(=C)C2)=O)CCCC(NC(c2cccc(C(C)C)n2)=O)CC1 13715,CC1(CNC(C2CCC(=O)N2)=O)CCN(C(C2CCCN2N=O)=O)C1 13716,C1(C)(NC(CCSCC)=O)CCN(C(C2CCCC2(C)C)=O)CC1 13717,CC1CN2CCC1C2.c1(CN(C(=O)NCc2cnns2)C)ccccc1 13718,c1(C(CNC(C(C2CCCCC2)SC)=O)(C)NC(C)=O)ccc(Br)cc1 13719,N1(C(C(C)SC(F)(F)F)=O)CCC(CNC(c2scnc2C(C)(C)C)=O)C1 13720,C1(CNC(c2c(OC)cccc2)=O)CN(C(C2CCCS2(=O)=O)=O)CCC1(C)C 13721,Cc1nnc2n1CCC2(C)C(=O)NC1CCC(N(C)C(C2CCOC2)=O)CC1 13722,C(CCSC)(C(=O)NCC1(C(C)(C)O)CN(C(c2scc(C)c2C)=O)C1)NC(C)=O 13723,CCC(C)C(C(=O)NCC(=O)N(C1CC1)CC1CC1)OC.C12(CC1)CC(=O)O2 13724,CC1CCC(F)(C(=O)NCCCCCCn2cc(COC3CCOC3)nn2)CC1 13725,c1(C(N2CCC(CN(C)C(c3ccc(N)cn3)=O)C2)=O)cc(F)n(C)n1 13726,C(CNC(C1OCCC1C)=O)(C(=O)NC(C)(C)CC1CCOC1)OC 13727,C(=O)(CCCC(=O)NC1CC(C)N(C(=O)COc2cccc(F)c2)C1)OC 13728,C(C(CN=c1[nH]c(N2CCC(C)(C)CCCC2)nc2c1CCCCC2)OC)OC 13729,CC1C2CC(C2NCc2ccccc2)N1C(=O)CC(C)(F)F 13730,N1(C(C(CC(C)=O)C)=O)CCC2CN(C(c3ccncc3C(F)(F)F)=O)CC12 13731,N1(C(Cc2ccn(C)n2)=O)CC2CC(C(=O)Nc3ccccc3C(C)(F)F)C1C2 13732,N(C1CCCn2ncnc21)C(C(C)NC(C1CN(C2COC2)C1)=O)=O 13733,N1(C(N=c2cc(CCCCCCC)[nH][nH]2)=O)CCCC2CC(C)CCC12 13734,C(CC1=CCN(C(c2nc3cnccc3s2)=O)CC1)NC(CCN(C)CC)=O 13735,Cc1nc(NCc2cc(Cl)ccc2N)cc(=NCc2ccn(-c3ccccc3)n2)[nH]1 13736,C1(C(=O)NCC2C(NC(=O)CC34CC(C3)C4)CCC2)CCCN1c1ncccn1 13737,c1(C2C3CCN2CC3)nc2ccc([N+](=O)[O-])cc2[nH]1.C1(C(F)(F)F)(CO)N=N1 13738,CN(CCCC(=O)N1CCOC(CCCNC(C2(C)COCCO2)=O)C1)N=O 13739,n1(CC)ncc(C(=O)NC2CN(C(C3CC3(C)Br)=O)CC2F)c1C 13740,C1(NC(CNC(=O)NC)=O)CCN(C(=O)CNC(C2(n3cccn3)CC2)=O)C(C)C1 13741,CC(O)C(C)(C)C(=O)NC1CC(NC(c2cc(C(F)F)no2)=O)C1 13742,c1(NC(C(C)OCC=C)=O)[nH]nnc1C 13743,C1(C)(SC)CCC1(C)C(=O)NC1CN(C(c2cccc(C)c2)=O)C1 13744,c1(C(N(C2CC(C(N3CC4CCC3CC4)=O)C2)C)=O)cc(I)c(O)c(I)c1 13745,N1(C(C2CCC(COC)C2)=O)CCC(C)(NC(C2(c3cccc(C)c3)CC2)=O)C1 13746,N1(C(c2ccc(OCCCC)nc2)=O)CCC(COC(=O)CCC(C)O)C1(C)C 13747,CCC(O)CC(=O)NCCN(CC)Cc1cnc(C)s1 13748,C(=O)(CC(=O)NC(C1(C(N2CCC(C(C)(C)C)C2)=O)CC1)C)NCC#C 13749,Cc1cccc2cc(C(N3CC(N(C(=O)CCF)C)C3)=O)oc12 13750,C(C(C)C(C)C(=O)NCC1CN(C(c2ccc(F)c(SC)c2)=O)C1)OC 13751,Cc1[nH]n(-c2ccc(Cl)cc2)c(=O)c1CC(=O)OCC(C#N)C(C)C 13752,C1(CC(=O)OC)(NC(c2scc(C)c2Br)=O)CCCS(=O)(=O)C1 13753,N1(CC)CCCCC1C(=O)N(CCC(C(C)C)NC(=O)CCc1cc(C)[nH]n1)C 13754,C1(C)(C(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)(C)C)CCC(C)=C(C)C1 13755,c1(C(N(CC(C)O)CCNC(c2cc(CC)ncc2)=O)=O)ncnc2ccsc12 13756,c1(OC)cc(C(F)(F)F)cnc1-c1cncc(SC)c1.c12cccc(c1)CN2 13757,c1(C(=O)NCC(Cc2ccccc2)NC(C2C(=C)CC2)=O)cccc(C2CC2)c1 13758,C1(NC(C(C(C)C)N(CC)CC)=O)(NC(=O)C(C)N=[N+]=[N-])CCC(F)(F)CC1 13759,CC1CCN(C(=O)CSC2CC2)CCN1C(C12CC(CO)(C1)OC2C)=O 13760,CC12CC(C(=O)NC3CCOCC3NC(c3ccc(CO)cn3)=O)(C1)C(C)(C)O2 13761,N1(C(CS(CC)=O)=O)CCC2(CCCC2CNC(c2n[nH]c(C)c2O)=O)CC1 13762,c1(N2CCC(N(C(=O)Cc3c[nH]ccc3=O)C)C2)cc(Cl)nc(C(F)(F)F)n1 13763,N1(C(CSCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13764,N1(C(CNC(C)=O)=O)CCC(C2(CNC(C3CC3C)=O)CCOCC2)CC1 13765,c1(CC)nc(C)c(CC(=O)NCC(C(C)C)NC(C2CCCC23CC3)=O)c(C)n1 13766,N1(C(CC(CN(C)C)O)=O)CC(N(C(=O)Cc2cncc(O)c2)C)C(C)(C)C1 13767,N1(C(c2cc(C)sn2)=O)CCC(O)(CCNC(C2(CO)CCOC2)=O)C1 13768,N1(C(c2c(CNC(c3ccc(C(F)F)o3)=O)c[nH]c2)=O)CCN(C2CC2)CC1 13769,C1(C(=O)NCC2CN(C(C3C(C)CC(C)O3)=O)C2)CCC2CC(C)CN2C1 13770,c1(C(COCCC)NS(=O)(=O)CCOC)nccn1C 13771,N1(C(CC2CC(CC)C2)=O)CCCC(CNC(C2CCN2CC)=O)CC1 13772,C(=O)(C(C)CS(C)(=O)=O)NC1CC(CNC(C(C2CCC(C)CC2)CC)=O)C1 13773,C1(CC=C)CCCC1NC(=O)C(C)(C)NC(=O)C=C=C(C)C 13774,C#Cc1cc(NC(C2CC(=O)C2C(C)(C)CC)=O)ccc1C 13775,N1(C(C)=O)CCC(C)(C(=O)N(CCC(C)NC(=O)CCC2CCCCCC2)C)C1 13776,C1(CNC(c2ccsc2)=O)CC(F)CN(C(C2(NC(C=COCC)=O)CC2)=O)C1 13777,CCCCC(C(=O)NC1CC(CNC(=O)C(C)(C)C2CCCC2)C1)C(C)C 13778,N1(C(C(=O)NCC(CO)NC(C=C(C)C(C)C)=O)=O)CCCC(C)C1.C1C=CC1 13779,N1(CC)CCP(C)(=O)CC1.C12CCC(CC1)OC2=O.c1(S)ccccc1C=O 13780,c1(C(N(C)CC2CCCN2C(C2C(C)(C)OC2(C)C)=O)=O)ncsc1S(N)(=O)=O 13781,N1(C(C23CCCC2C3)=O)CCC(c2ncc(C(=O)O)[nH]2)C1 13782,C1(C2(O)CCN(C(=O)CC3(O)CCC3)CC2)(NC(CCc2ncc(C)[nH]2)=O)CC1 13783,C(C)(C)(C(=O)NC(CNC(c1nncn1C1CC1)=O)CC)OCC 13784,CNS(=O)(=O)NC(=O)CCC1CCCN1C(C1(C2(F)CCOC2)CC1)=O 13785,c1(C(N(c2ncc(C)c(C)n2)C2CC(N)C2)=O)noc2cc(Cl)ccc12 13786,C12(NC(c3ccc(CC)s3)=O)CCC(C(=O)NCCNC3CCCC3)(CC1)C2 13787,Cn1ccc2cc(C(N3C4CCC(C4)C3C(N3CC4(CCCCC4)C3)=O)=O)cnc12 13788,N1(C(=O)OC(C)(C)C)CCC(F)(NCC(C2CC3CCC2C3)O)C1 13789,c1(CCNC(C(=O)NCCOCC(=C)C)=O)noc(CC)n1 13790,c1(C(N2CCC(CNC(C(C)=C3CC3)=O)CC2C)=O)cc2cc(C)c(C)cc2o1 13791,N#CC12CCC(C(=O)SCCl)(CC1)CC2.c12nc(cs1)CN2 13792,c1(-n2ccc(C)n2)cccc(C(=O)NCC2(C)CC2(F)Cl)c1 13793,C1(CC)CN(C(C(=O)NC2CC2)C2CCC2)CC=N1 13794,N1(C(Cc2cncc(C)c2)=O)CCC(C)C(NC(=O)CC(O)C2CC2)C1 13795,CC1C(C(=O)NCCCc2ccnn2C)CCN1C(=O)CCC1CCCCO1 13796,N1(C(C(CC)SC)=O)CCCC2C(CCCN2C(c2cccc3[nH]ccc23)=O)C1 13797,Cc1nn(C)c(C)c1C(=O)N.c1(C(=O)NC(CCC)CC(C)C)cccc(Cl)c1F 13798,c1(C(C)=O)ccc(C(=O)NC(CNC(C2(CC3CC3)CC2)=O)CC)c(F)c1 13799,N1(C(C(c2cnn(C)c2)C)=O)CC(CC(=O)Nc2cnc(O)c(F)c2)C2(CC2)C1 13800,N1(C(C(C)NC=O)=O)CCC(C(=O)N(CCC=O)CCO)=C(F)C1.OC 13801,c1(OC)cc(C(=O)N(C)CCN(C(=O)C(F)=C2CCC2)C)[nH]n1 13802,c1(C(N2CC3C(NC(CN(C4CC4)CC)=O)(C3)C2)=O)cc2cn[nH]c2cn1 13803,C(=O)(CC1=NN(C)C(=O)C1)N(CC(CC)NC(=O)C(F)CC1CC1)C 13804,C(=O)(CC(F)(F)C(C)C)N1CCCC(N(C(C(CCCOC)C)=O)C)CC1 13805,N1(C(c2cnc3[nH]nnc3c2)=O)CC(C2CCCN(C(C3CCOC3)=O)C2)C1 13806,Cc1noc2nc(=NCC3CC(c4ccccc4)=NO3)[nH]c(O)c12 13807,C(=O)(C(F)C(C)CC(C)(C)C)NCCSCC(=O)NCC1C(C)CCCC1 13808,c1(C(=O)NCC2C(C)CCN2C(C2CN(C(N)=O)C2)=O)nn(C)c2ccc(F)cc12 13809,c1(CC(=O)NCC(CNC(c2[nH]cc(C)c(=O)c2)=O)O)ccc2c(c1)OCCO2 13810,N1(C(c2ccc(F)c(F)c2)=O)CC2CN(C(c3cccc[n+]3[O-])=O)CC2C1 13811,C1(NC(CCCc2cc(C)no2)=O)CN(C(c2cn(C)nc2C)=O)CC1C 13812,C1(C(=O)NCCSCC)CC2(CC(NC(=O)CC(=O)NC)C2)C1 13813,c1(N2CC(C)OC3(C2)CCCC3)ccc(S(=O)(=O)NCC2CCCN(C)C2)cc1Br 13814,C1(C(=O)NC2C(CNC(CC(C)(C)OC)=O)CCCC2)CCC2(CC1)CC2(F)F 13815,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)C(C)=CC)C1(CC=C)CCOCC1 13816,C(CC1=CCCCC1)NC(c1c(CNC(C2(C(F)(F)F)CC2)=O)ccs1)=O 13817,c1(-n2nnc(C)c2CN2CCN(C)CC2c2ncc[nH]2)cc(Cl)c(F)cc1Cl 13818,C1(NC(c2c(CCC)n[nH]c2)=O)CC12CCN(C(C1CCNC(=O)C1)=O)C2 13819,C1(C)(CC(=O)NC(C)CCNC(c2cc(Cl)c[nH]2)=O)Oc2ccccc2O1 13820,CC1CCN(C(C2(CN(C)C)CC2)=O)CC1CNC(c1ccc(F)cc1)=O 13821,Cc1ccc(C(C)C)c(OCC(=O)NCC2CC2NC(c2cnnc(O)c2)=O)c1 13822,Cc1sncc1C(=O)NC(C)C(C1CCCCC1)NC(c1csc(Cl)n1)=O 13823,c1(C(=O)NC2(CNC(C(C=C)O)=O)CCCC2)cn(C)nc1-c1ccc(Cl)cc1 13824,C1(C)(Nc2c(Cl)cnc(SC)n2)CCN(C(c2nccc(C#N)n2)=O)CC1 13825,C1(C)(C(N(CC(CNC(C2C(OC)CCC2)=O)C)C)=O)CCC(=O)NC1 13826,N1(C(CCc2c(=N)[nH]cnc2)=O)CC2CCN(C(=O)C=CC(=O)N(C)C)CC12 13827,N1(C(C(C)Oc2cccnc2)=O)CC=CC(C(=O)NCC2(C)CC2(C)C)C1 13828,N12CCC(C)C(C1)CN(C)C(=O)CSC1N(CCC1)C2=O.CCC=CC=O 13829,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(n2cc(CCC#C)nn2)C(O)C1 13830,c1(C(=O)NC2C(C)CCN(C(=O)Cn3nccn3)C2)cc(C#N)ccc1Cl 13831,c1(C2C(C)(C)C(O)C2)ccc(S(=O)(=O)Oc2ccc(C(F)(F)F)cc2)cc1 13832,c1(COC)cnc(OC)c(C(=O)NCC(C)CNC(c2coc(Cl)n2)=O)c1 13833,C1(c2n(CC(C)C)nnn2)(NCc2cnc(N(C)C)nc2C)CC(C)SC(C)C1 13834,C1(C(C)NC(C2CC(n3cnnc3)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13835,N1(C(C2C(C)C2(F)F)=O)CCCC12CCC(NC(c1n[nH]c3c1COC3)=O)CC2 13836,c1(C2CCN(C(C3CCC(c4ccccc4)C3)=O)C2)cc(Br)ncc1Br 13837,N(C(=NCC(C)OC)NC(C1CCCCC1)CC)Cc1ccc(CCCC)cc1 13838,c1(-c2cn(CC(=O)NCc3ccc(OC)cc3)nn2)cc(Cl)c(C)cc1Cl 13839,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnc2)=O)C1 13840,c1(C(=O)OCC)cc(F)cc2c1CCN(C(C1CCCN1C(=O)CC#N)=O)C2 13841,C1(C(N(CCCC)CCCC)=O)CCN(C(=O)c2ccc(CO)o2)O1 13842,Cc1cnc(C=CC(=O)N(C2CCOC2)C(C)C2CC2)[nH]1 13843,N1(c2c(OC)cncn2)CCCCCC(NC(=O)CC2C=NN(C)C2=O)C1 13844,C#CCCCC(C)C(=O)N(C)CCOCCNC(=O)CCc1cocn1 13845,C(c1ccccn1)=CC(=O)N(CCOC)CCNC(C1CCOC1C)=O 13846,Cc1cc(C(=O)NCC2C(C)CCCN2C(=O)C(C#N)=CC2CC2)cc(F)c1C 13847,O=C1CC2C(C(=O)NC3CCC3)C2C1.c12csc(c1)C(=O)NC2 13848,C(=O)(C(C)C(C)(C)C)NC(CNC(C1C(OCC)C1)=O)CO 13849,N1(c2c(C)c(Cl)ncn2)CC2(CCC(NC(=O)C(CO)NC(=O)OC(C)C)O2)C1 13850,CC1CC(NC(=O)CC2CNC(=O)C2)CN1C(=O)Cc1ccnc(Br)c1 13851,C=CCC(C(=O)N(CC(C)CNC(c1cc2ncccc2s1)=O)C)C(C)C 13852,Cc1cc(=NCc2cnn(CCO)c2)[nH]c(N(C)Cc2ccoc2)n1 13853,c1(OCC)cncc(C(=O)NCCC(COC)NC(c2cn(C)c(C)n2)=O)c1 13854,CCC(CN(C1CC2(CCC2)C12CCC2)c1ccc(OC)cc1)(CC)C(=O)OC 13855,N1(C(CCC#C)=O)CC(NC(=O)CCc2cccnc2C)CC12CCCCC2 13856,C(CC(CC)C(=O)NC1CCCCC1C(=O)N(C(C)CC)CC)=CC 13857,c1(SC)cc([N+](=O)[O-])nn1C.c1(OC)cnc(C(N2CC3(C2)NC3)=O)cn1 13858,C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)CCOCC(F)(F)F)C1(C)C 13859,c1(CC)nc(C)c(C(=O)N(CC(C)(C)CNC(=O)CCn2nc(C)cc2C)C)o1 13860,CN1CCC(C(N2CC3(CCN3C(=O)C=CCn3cncn3)C2)=O)CC1=O 13861,CCC(C)C(O)C(C)C(=O)N(CCC(=O)NCC1CC1)CCCO 13862,c1(C(=O)NC2CCCN(C(C3(C#N)CC(C)C3)=O)C2)cc2c(nn1)CCC2 13863,N1(C(=O)NC2C(SCC)CCCC2)CCC2(CCCN(C)C2=O)C1 13864,Nc1nccn2ncc(C(=O)NC3CCC(O)CN(C(=O)CSC4CC4)C3)c12 13865,C1(N2CC(n3ncc(NC(C(C)(F)F)=O)c3)C2)CCCCN1O 13866,CC1(C)CC(C)(C)C1CNCCN1CCN(C(=O)OC(C)(C)C)CC1 13867,CC1CCCCC1C(=O)NCC1(CNC(=O)C(F)(F)C2(O)CCC2)CC1 13868,c1(C(=O)NC2CCCC(C(N3CCCCC3)=O)C2)ccc2c(c1)CCCS2(=O)=O 13869,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13870,C1(C(N(CCN(C(C)C)C(c2ccc(CC#N)cc2)=O)C)=O)C2CC2C2CC12 13871,C1(CNC(c2ccn(CCOC)c(=O)c2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O 13872,c1(-c2c(CC)nco2)nc(C2CCCC2)nn1C1CCSC1 13873,C(=O)(C1=C(C(C)=O)N(CCF)C(=O)NC1c1cc(Cl)c(F)cc1F)OCC 13874,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13875,c1(C(N2CCCC(NC(c3ccc(CF)cc3)=O)CC2)=O)cn2ccnc2cn1 13876,c1(C(=O)NC(C2CN(C(C3(OC)CCC(C)C3)=O)C2)C)ccc2cc[nH]c2c1 13877,C#Cc1cc(C(=O)N(C)CCN(C(=O)C(c2ccc(F)cc2)F)C)cc(F)c1 13878,CC#CCCCC(=O)NC1(C2CN(C(=O)CC=CCC)C2)CC1 13879,c1(C(N(CC)Cc2nccn2C)=O)occc1CNC(=O)CC1CCSC1 13880,C(=O)(C(CSC)NC(c1cn(C(C)(C)C)cn1)=O)N(CCOCCO)CC 13881,C(N1CCC(CCC2CCCO2)CC1)n1n(C)c(=O)cc1 13882,c1(C(=O)NCC2CCC(NC(=O)C(c3ccccc3)F)C2)ccc(O)nc1Cl 13883,Cn1c(C(=O)NCc2cncc(C(=O)NCC3CCOC3(C)C)c2)cccc1=O 13884,CCCCC(C)CCC(=O)N1CCC(C)(C)C(C(=O)NCC2CCCOCC2)C1 13885,c1(C(N2CC(CN(C)C(c3cnn(C)c3C3CC3)=O)C2)=O)n[nH]c2c1COC2 13886,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(C)(C)SC)CC1C 13887,Cc1cc(C(=O)NCC2(NC(=O)Cc3cnoc3)CC2)cc(F)c1C 13888,C(=O)(CC(C)C(C)(C)NC(C1CNC(=O)N1)=O)N(CC(C(C)C)OC)C 13889,CC(C)C(CNC(C1C2CCCCCC12)=O)C(=O)NCCC1(O)CCC1 13890,c1(-c2cc(CN3CCC(C(=O)O)(CC)C3)sc2)ccc(OC)cc1Br 13891,c1(N(C)C)ccc(Br)cc1C(N1CCC(C)(CNC(C2(O)CCC2)=O)C1)=O 13892,C1(C(N2CCC(CNC(C(C)OCC(C)C)=O)C2)=O)CCC2(CC1)CNC(=O)C2 13893,Cc1cnc(C)c(C(N2CC(N(C(=O)CC(C)C3CC3)C)C3(CC3)C2)=O)c1 13894,N1(C(CC2N(C)CCCC2)=O)CCCC(C)(CNc2cc(C#N)ncn2)C1 13895,C1(C(=O)NCC(=O)NC(C)C)CC(C)C1.C1(NC(=O)COCO)CCCC1 13896,CCCC(O)C(=O)NC(C(=O)N1CCC(CN(C)C)C1)C(C)C 13897,c1(C(=O)OC)[nH]c(=NCC(C)CNC(=O)C(O)Cc2cnc[nH]2)sc1C 13898,CCCCCCC(C)C(=O)NC1CC(C(=O)NCC(O)C2(Cl)CC2)=CC1O 13899,Cc1c[nH]nc1C(=O)NC1CN(C(C2(COC3CCOCC3)CC2)=O)C1 13900,N1(C(C2CC(=C)C2)=O)CC2CCCC2(NC(=O)Cn2nc(C)c(Br)c2C)C1 13901,CC1(C)C(c2ccc(Br)cc2)CCN1C(=O)NC1CCC(F)C1 13902,c1(C(=O)NC2(C(=O)NCC(C)Cn3ccnc3)CC2C)cc([N+](=O)[O-])n[nH]1 13903,C1(C(=O)NCC2CCN(CC)C2)CSCCN1C(=O)CCN(C)CCO 13904,N1(C(CN(C2CCOCC2)C)=O)CCC2(CCCCN(C(=O)COCC3CC3)C2)C1 13905,c1(CN2CCN(C(N3CCCC(c4ccccc4)C3)=O)CC2)ccc(F)c(F)c1 13906,c1(CC(=O)NC2C(O)CCN(C(CCCCC#C)=O)C2)cc(Cl)cc(Cl)c1O 13907,n1(C(C)C)nc(C2CC2)cc1S(=O)(=O)NC(C1CN(C(C)C(N)=O)C1)=O 13908,c1(C(N2CC(C(N3CCCC(c4cc[nH]n4)C3)=O)C2)=O)c(F)cc(Cl)cc1F 13909,C1(C(=O)NCCC(=C)CNC(c2c[nH]nc2-n2cnnn2)=O)CC2(CCC2)C1 13910,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 13911,C(=O)(C1=NOC2(CCN(c3nccc(Br)n3)C2)C1)Nc1cc(C)cc(C)c1 13912,C1(C(=O)NCC(C(C)C)NC(c2csc(C(F)F)n2)=O)CC(=O)N(C)C1 13913,c1(NC2OCCN(CC(C(C)C)O)C2)ccc2sccc2c1 13914,N1(C(c2ccc(CCC)cc2)=O)CCC(F)CC1C(N1CCN(C)CC1CC)=O 13915,C(CC1=CCCCC1)N(C1CN(C(c2c[nH]nc2C#N)=O)CC1C=CC)CC=C 13916,C(=O)(C(C)(C)CF)N(C1CCN(C(C2CCN(C)C2=O)=O)CC1)C 13917,c1(C(=O)NC2CC(CCNC(Cc3n(C)nnc3)=O)C2)ccc(N)cc1O 13918,c1(C(=O)NCC(CNC(C2CCC(O)CN2C)=O)OC)cc(C)c(Cl)cc1F 13919,Cn1c(NC(=O)Nc2ccc(OCCO)cc2)nnc1-c1ncccn1 13920,c1(NCC2(C)ON=C(C)C2)[nH]c(=NC(C)C2CCCC2)nc2sccc12 13921,N1(C(=O)Cn2cnnn2)CC2CC(N=c3ccnc(C4CCCC4)[nH]3)CC1C2 13922,C(=O)(CCNC(=O)CCc1cnco1)NC1(CCC)CC1 13923,c1(OC)cc(C)ccc1C(NC(=NCc1nonc1C)NC1CCC1)C 13924,C(c1ccc(Cl)cc1Cl)=CC(=O)N(C1CCCN(C(C)=O)C1)C 13925,C(=O)(C(CCNC(=O)C(CC1CCC1)OC)OC)NCCCC#C 13926,C1(C2(CC#N)CCC2)(C(=O)OC(C)(C)C)CCC1.CC1CCC(=O)N1 13927,C1(CNC(C(CC)NC(=O)CCCOC(C)=O)=O)CC2(CCC2O)C1 13928,C(c1cc(F)c(O)c(F)c1)=CC(=O)NC1(CC=C)CN(C(C2CC2(C)C)=O)C1 13929,S(=O)(=O)(CCC(=O)NCC1COCCN1C(C1COCC1C(N)=O)=O)NC 13930,N1(C(CCOC(C)C)=O)CCC(NC(c2ccc3nc[nH]c3c2)=O)C2(CCC2)C1 13931,C=Cc1ccc(C(N2CCCC(CNC(=O)CC3CCS(=O)(=O)C3)CC2)=O)cc1 13932,c1(CNC(C2CCC(C3CC3)N2C(C2CCCC2O)=O)=O)cccc2cc[nH]c12 13933,Cc1c(Cl)cc(CN2CCCC(C(=O)NC3CCS(=O)(=O)C3)CC2)cc1Br 13934,c1(C(N2CCN(C(CNC(C)=O)=O)CC2C(C)C)=O)c(C)cc(Br)cc1C 13935,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 13936,c1(C(=O)NCC23CC(NC(CN(CCC)C)=O)(C2)C3)ccc2cccnc2c1 13937,C1(CC=C)(NC(C2(CC3CC3)CC2)=O)CCN(C(=O)CCC2(C)CC2)CC1 13938,N1(C(Cc2n[nH]c(=NC)s2)=O)CCCC12CCCN(C(c1cnncc1O)=O)C2 13939,c1(C(=O)NCCCCNC(c2nn(C)c(C3CC3)c2)=O)cccc(Cl)c1[N+](=O)[O-] 13940,n1(CC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 13941,c1(OC)cc(C)c(C(=O)NCCC2CCN(C(C3CCN(C)C3)=O)C2)c(C)c1 13942,C1(C)(CC)CCCN(C(c2ccc(C(N)=O)cc2)C(=O)NCCOC(C)C)C1 13943,C1(NC(c2cc(C(C)C)no2)=O)CCCC(N(C(=O)C(=O)NCC(F)F)C)C1 13944,CCC(N)C(C)(C)C(=O)NC1(c2nnnn2C(C)(C)C)CC2CCC1CC2 13945,N1(C(C(CCCC)(C)F)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)OCC)C1 13946,C(c1ccc(OC)c(Cl)c1)=CC(N1CC2C(NC(COC(CC)C)=O)C2C1)=O 13947,c1(CC(=O)N(C(C)CCNC(=O)C(N2CCCCCC2)C)C)cccc(F)c1O 13948,C(=O)(CCCCC(F)(F)F)NCC(CCOC)NC(c1cn(CC(N)=O)nn1)=O 13949,N1(C(COc2c(CCNC(CC(C)F)=O)cccc2)=O)CC(O)CCC1C 13950,c1(OC)ccccc1CNCC1CCCN1C(c1ccc(C)cn1)=O 13951,N1(C(C(CC=CCC)C)=O)C(C(N2CCCC2C(C)(C)O)=O)CCC12CC2 13952,C1(C(=O)NCC2CC(=C)C2)CC(F)CN(C(c2cccn2C)=O)C1 13953,Cc1cccc(C(=O)NCCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 13954,c1(CN2C(C(=O)Nc3ncc(CC)s3)COCC2)coc2cc(N)c(SC)cc12 13955,CC1=C(C(=O)N2CCC(NC(=O)CC(O)CC(C)C)C(O)C2)C(=O)OC1(C)C 13956,c1(CC2CC(C(=O)NCCNC(=O)NC3CC3)C2)ccc(F)c(O)c1F 13957,C(=O)(CCN=c1cc(C(F)(F)F)nc(Cl)[nH]1)N1CCCC(NC(C=CSC)=O)CC1 13958,c1(C(=O)NC(C2(C(=O)NCC3CC3CNC(N)=O)CC2)C)cccc[n+]1[O-] 13959,N1(C(C(C=CC)O)=O)CCC2CC12C(=O)N(C)CCN1CCCC1=O 13960,N1(C(CN(c2n[nH]c(O)n2)C)=O)CCN2CCNCC2C1 13961,C(=O)(C(C)(C)C(F)(F)F)N1CC(O)(C(C)N(C(=O)CN2C(C)CCC2C)C2CC2)C1 13962,N1(CC(N2CC(NC(C(F)=CCC)=O)C(CO)CC2)=O)C(=O)NC(C)(CC)C1=O 13963,c1(SCCC(c2cnc(C)[nH]2)NC2COCC2C(N)=O)ccc(Br)cc1 13964,c1(C(N2CCCCC2CNC(C2(CF)CC2)=O)=O)cc2c[nH]nc2s1 13965,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 13966,C(=O)(CCCCCCCCC(=O)OCC)NC(CN(C(C1CC(OC)C1)=O)CC)C 13967,C1(N(C(CNC(=O)OC)=O)C)(CNC(c2cnc[nH]2)=O)CCCCCC1 13968,c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCCCC3)CC2)c(Cl)n1 13969,C(C(C(=O)NCc1ccccc1)N(C1CCCCC1O)C)(C1CCC1)OC 13970,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)C(C)C)C1 13971,C1(CNC(C(CC)OC)=O)C2CN(C(C3CC3c3cccnc3)=O)CC12 13972,N1(C(=O)NCc2snc(C(C)(C)C)n2)CCCC(=CC(=O)O)C1 13973,CC1(NC(C2(C(F)F)CC(O)C2)=O)CCN(C(c2cccc(C3CC3)n2)=O)C1 13974,Cc1cc(CNC(C23CC(NC(=O)CCc4cccnc4)(C2)C3)=O)n(C)n1 13975,CCCCC(O)C(C)C(=O)N1CCN(C(=O)Cc2cc(C)[nH]n2)CC1CCC 13976,c1(NC(C2CC(=C3CC3)C2)=O)ccc2c(c1)COC2 13977,c1(CC)ccc(C(=O)NC(CNC(C2CNC(=O)N2)=O)CC(C)C)cc1CC 13978,c1(CC(=O)Nc2ccn(Cc3cn(CC(CC)C)nn3)n2)cc(C)nn1C 13979,c1(C(=O)Nc2nc(CNC(C3N(C)C(=O)CC3)=O)oc2)ccc2nc(O)[nH]c2n1 13980,N1(C(CSCC(=O)N(C(c2cccc(C)n2)C)CC)=O)CC(C)(C)C1C1CC1 13981,Cc1c(C(N2CC3CC(C2)CN(C(C2CCOC2C)=O)C3)=O)nn2c1OCCC2 13982,C1(C(=O)NC(c2ccccc2)CNC(=O)C=C2CCSCC2)CCCC(=O)N1 13983,c1(OC)c(F)ccc(-c2ccc(CN3CC(N)C3)c(F)c2)c1F 13984,c1(-c2nc(C(C)OC)nn2-c2cccc(OC)c2)onc2ccccc12 13985,c1(NC(c2n(CCCC(=O)OC)nnn2)(C)CCOC)ccc2c(c1)CCCS2 13986,c1(C(=O)NCC2CN(C(CNC(CC)=O)=O)C2)ccc(OC)cc1C 13987,c1(C(=O)NC23CCN(C(C4(CCN(C)C)CC4)=O)CC2C3)ccc(S(C)=O)cc1 13988,C12C3CC4C1C4C3C(=O)N2.C(CCCC(=O)N1CCCC(OCCO)C1)OC 13989,Cc1nc(CC(=O)NCCn2cc(C3CC3CO)nn2)c(Br)s1 13990,c1(C(=O)NC(C2(O)CN(C(=O)CC3CCNC3=O)C2)C)ccccc1OCC(N)=O 13991,N#Cc1cnn(CC(N2CCN(C(c3cnnc(O)c3)=O)C3CC23)=O)c1N 13992,c1(N(C)C)ncc(NC(=O)NC(CCc2ccco2)Cc2cccs2)cn1 13993,C(c1cccc(O)c1)=CC(=O)NCC(C)(F)CNC(C1(N(C)C)CCCC1)=O 13994,N1(C(=O)NC23C(C)OC(C)(C2)C3)c2c[nH]nc2CCC1C(F)(F)F 13995,CCCCCS(=O)(=O)CC(=O)NCC1(F)CN(C(c2cc(F)ccc2OC)=O)C1 13996,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)N1CCOC(CO)C1 13997,C1(CC=C)(NC(c2cnn[nH]2)=O)CCCN(C(C2C3CCCOC23)=O)C1 13998,c1(C(=O)NCCNC(C(=CC2CCC(C)CC2)C)=O)ccc2c(c1)CN(C)CC2 13999,c1(C(N2C(CNC(C3C(C)C3c3ccccc3)=O)CC2)=O)nccnc1Cl 14000,C1(CNC(CCc2cc(C)on2)=O)CCC(F)(CNC(c2ccoc2C)=O)CC1 14001,N1(C(COCCC(C)C)=O)CCCC(C(C)NC(c2n[nH]c(C(C)C)c2Cl)=O)C1 14002,C(=O)(C(C)(C)C(N)=O)NCCCC(C)NC(=O)C(C)c1ccco1 14003,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14004,CC1CN(C(c2coc(Br)c2)=O)C(C)CN1C(=O)CSC(F)(F)F 14005,c1(CCC)cccc(C(=O)N(CCCNC(C2C3CN(C)CC23)=O)C)c1 14006,c1(C(=O)NCCNC(=O)CN=C2NS(=O)(=O)c3ccccc32)ncc2c(F)cccn12 14007,CC(C)C(C(=O)N(CC(O)CN(C)C(c1ccc(Cl)cn1)=O)C)n1cncn1 14008,C1(CNC(=O)Cc2ccccc2CO)CN(C(c2cccc[n+]2[O-])=O)CC12CC2 14009,C12(NC(CCCC3C(C)C3)=O)CCC(C(=O)NC34CC=CC(C3)OC4)(CC1)C2 14010,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14011,C1(C2(O)CN(C(=O)Nc3cccc(OCC(C)C)c3)C2)(C(=O)NCC=C)CC1 14012,C(=O)(CCCCCCNC(=O)C=Cc1cnccn1)N1C(COC)CCCC1 14013,CCCCC(C)CCC(=O)N(CC(=O)N(CC(O)COC(C)C)CCO)C 14014,c1(COC)ccccc1-c1ccc(N2CCN(C(=O)CCC3CC3)CC2)nc1 14015,C1(CCCC)CN(C(c2csc(C)n2)=O)CCN1C(c1cn(CC2CCC2)nn1)=O 14016,c1(C(=O)NCCC(CNC(=O)Cc2ccc(Br)s2)OC)cccc(C)n1 14017,N1(CCC(=O)O)CCc2c(NC(c3cccc(C(F)(F)F)c3)=O)cccc2C1 14018,C1(NC(CCCSC)=O)CN(C(=O)CNC(=O)COCC2CCC2)CCC1(F)F 14019,C12(C(=O)NCCCCNC(c3cn(C)nc3Cl)=O)CCC(CC1)C(C)(C)O2 14020,c1(C)ccc(C=CC(N2CCCC2CNC(C2C(C(C)(F)F)C2)=O)=O)o1.C1(N)CC1 14021,CC1CC(C(=O)Nc2cnccc2I)N(Cc2cccc(F)n2)C1 14022,Cc1c(N2CCCC2)nc(Cl)nc1N1CCCC(CSC2CCCC2)C1 14023,N1(C(c2c(C)nn[nH]2)=O)CCC(N2CCN(C(c3cccnc3Cl)=O)CC2)CC1 14024,CN1CCC(C(=O)NOCCCF)(NC(C2CCCC2F)=O)C1 14025,c1(C(N2CCOCC2C2CCOCC2)C(=O)NCC)cc(Br)c(O)nc1C 14026,N1(C(c2cc(C(C)C)ncc2)=O)CC(C)CCC1CNC(c1ccc(F)o1)=O 14027,c1(NC(C(CC)C2CC2)=O)ccc(C(C(=O)OC)N(C2CC(C(=O)OC)C2)C)cn1 14028,N1(C(COCC(=O)NC)=O)CCCCC(N(C)C(c2nnn(C(C)C)c2C)=O)C1 14029,c1(CNC(c2c(C)cc(C(F)(F)F)n2C)=O)n[nH]c2c1CN(C(=O)C1CC1)CC2 14030,N1(C(CCC(=O)NC)=O)CCN(C(c2ccc(Cl)c(Cl)c2C)=O)CC(O)C1 14031,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(C1(c3ccno3)CC1)=O)CCO2 14032,c1(C(C(=O)NCC(C)N(C)C(c2cn(C)nn2)=O)(C)F)ccccc1F 14033,CS(=O)CCC(O)C(=O)NC1CC(CNC(c2cncc(F)c2Cl)=O)C1 14034,C1(C2(O)CN(C(C3CC3c3ccncc3Cl)=O)C2)(CNC(c2cn[nH]c2)=O)CC1 14035,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CCN(C(c2n(CC=C)ccc2)=O)C1 14036,CC1CN(C(c2c(N)cc(F)cc2F)=O)CC(C)N1C(C1CC(N(C)C)C1)=O 14037,c12ncnc(c1C)N1CC3CC3(C1)CN2.Cc1cccc(C(N2CCCC2)C)c1 14038,CC(C)C(C(=O)N1CC(CCNC(C2C(C)(C)C2(F)F)=O)C1)NS(C)(=O)=O 14039,Cc1nn(C)cc1C(N1CC(CNC(=O)CC2CC(C3CC3)C2)C1)=O 14040,C(=O)(C(CC(=C)C)NC(c1c[nH]nc1OC)=O)NCCCCCC=C 14041,C1(C(=O)Nc2cn(CC#C)nc2)CN(C(C2(CCOC)CC2)=O)CCO1 14042,C1(O)(CCNC(=O)COc2ccccn2)CCN(C(=O)C(C2(O)CCCC2)F)C1 14043,C=CCC(CC)C(=O)N(C1CN(C(c2ccnn2C)=O)CC1(C)C)C 14044,C1(N(C(CN2CCC(OC)C2)=O)C)CCN(C(c2coc(C3CCC3)n2)=O)CC1 14045,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14046,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14047,N1(C(C2N(C(c3cc(C)c(C)o3)=O)CCCC2)=O)CCC2(COC(=O)N2)C1 14048,N1(C(C(C)NC=O)=O)CC(O)(CCNC(=O)C(c2ccsc2)C)C1 14049,C1(N(C(CCC=C)=O)CCO)CCCN(C(=O)CC2CC(N(C)C)C2)C1 14050,C(=O)(C(S(C)(=O)=O)C1CC1)NCCC(C)NC(C(Cn1ccc(C)n1)C)=O 14051,C1(C)(CC(=O)NCC(C)=CC(N2CCCC2CCCO)=O)CC(C)(C)C1 14052,N1(C(CN(C(=O)C=Cc2cn(C)nn2)CCC)=O)CCC(CN=[N+]=[N-])CC1 14053,N1(C(c2cc(C)ns2)=O)CCC2CC2(C(=O)NCc2ncccc2F)CC1 14054,Cc1nsc(C)c1C(=O)NCC1CCCN(C(C2CCC(CO)O2)=O)C1 14055,N1(C(C(=O)Nc2c(OC)cccc2)c2cscn2)CCCC(=O)C1C 14056,c1(C(N(CC(Cc2ccccc2)NC(=O)CO)C)=O)c[nH]cc(F)c1=O 14057,c1(C(=O)NC(CC)CNC(C2CCN2CC)=O)ccc2ncccc2c1 14058,c1(OCC)cc(NCC(=O)NCCCCCNC(c2c[nH]ccc2=O)=O)ccn1 14059,c1(C(N(C)CCN(C)C(C2(C(F)(F)F)CCCC2)=O)=O)ccnc(OCCO)c1 14060,N1(C(C(C)=O)=O)CCC(C(=O)NCCNc2ccn(C(C)(C)C)n2)C1 14061,c1(C(=O)NC2C3CC(CNC(C(C)OCC)=O)(C3)OC2)cnn2cccc(C)c12 14062,N1(C(c2scc(C)c2C)=O)CC2CC(C(=O)NC(c3ncc(Br)cn3)C)(C2)C1 14063,C1(S(C)(=O)=O)(C(=O)NCC2CCCN(C(C=CS(C)=O)=O)C2)CCCC1 14064,N12CC3CC(CC1C3)C2=O.Cc1ccc(C(C)NC(C23CCC(CC2)C3)=O)cn1 14065,C#Cc1ccc(NC(C2CCNC2c2ccccc2)=O)cc1C 14066,CC(C)C(O)C(=O)N1CC2CC1(CNC(=O)CC1CC3(CC3)C1)C2 14067,c1(C(N(C)C)=O)cccc(NC(=O)C(N2CCOCC2c2ccc(F)cc2)=O)c1 14068,C1(NC(c2c(OC)ncc(C)c2)=O)CN(C(=O)C(O)c2ccsc2)CC1C1CC1 14069,C1(C(=O)Nc2cnc(O)c(F)c2)CN(c2ccnc(C3CC3)n2)CC2(CCC2)C1 14070,c1(C(C)C)ncc(N(C(=O)C(F)(F)F)C)[nH]1.C1C(C)(C)Cn2cc(nn2)COC1C 14071,c1(OC(C(N2C(CNC(c3c(CSC)ncs3)=O)C=CC2)=O)C)cccc(C)c1 14072,N1(c2c(OCC)cnc(Cl)n2)CCC(C2(NC(c3ncsc3NC)=O)CC2)C1 14073,CC1CCCC(C)N(C(=O)CC2(NC(c3ncc[nH]3)=O)CCC2)C1 14074,CC(O)C(C(=O)N(C1CC1)CC1CCN(C(c2ncoc2C(N)=O)=O)CC1)N(C)C 14075,C1(CC(=O)NC2CCCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)C2)CCS(=O)(=O)CC1 14076,N1(CC)C(=O)CCC1CC(=O)NC1CC12CC(NC(=O)CCC1CCCC1)C2 14077,N1(C(C2(C)C(C)(C)C2)=O)CCC(CC(=O)NCC2CC3C=CC2O3)CC1 14078,N#CC1(C(=O)NC2CCCC(C(=O)NCc3ccncc3F)C2)CC12CCC2 14079,Cc1cccnc1C(=O)Nc1ccc(C(=O)OCCN=S(C)(C)=O)nc1 14080,c1(C(N2C(C)(CC(N3CCCC(O)(CCO)C3)=O)CC2)=O)ccc2[nH]ccc2n1 14081,c1(OC)ccc2c(c1)NC(C(N1CCC3CCN(C(=O)C=CC4CC4)C3C1)=O)C2 14082,C1(C(C2CC2)NC(CCc2onc(C)n2)=O)CN(C(=O)CCCNC(N)=O)CCO1 14083,N1(C(CC(C=C)C)=O)CCC(CNC(c2cccc(CC3CC3)n2)=O)C1(C)C 14084,c1(C(C)C)cc(CNC(=O)Nc2ccoc2CN(C)C)on1 14085,C1(O)(C(C)CNC(c2cnc(O)o2)=O)CCN(C(c2ccc(F)cn2)=O)C1 14086,N1(C(c2c(COC)scc2)=O)CCC(CNC(c2ccc(C)s2)=O)C(CC)C1 14087,Cn1cc(S(N)(=O)=O)cc1CC(=O)NC1CCC(=O)N1CC(F)F 14088,CCCCCCCNC(c1cc(C(=O)OC)cc(C)c1)=O.CC1(CC)C(=O)N1 14089,C1(NC(c2cc(CCOC)on2)=O)CC12CCN(C(=O)C(F)OC(F)(F)F)CC2 14090,C(=O)(C1=CC(C)(CC)C1)N1C(C(=O)NCC(CC=C)(C)C)CSCC1 14091,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14092,CC(CCNC(C1CN(C(c2cccc(F)c2)=O)CC1C(C)C)=O)CC(C)(C)C 14093,N1(C(C(C(C)O)N(C)C)=O)CC(NC(c2ncccc2N(C)C)=O)CC2(CC2)C1 14094,N1(C(=O)Nc2cc3n(n2)CCCO3)C2CCC(CO)C1CC2 14095,CCCC(C)(O)C(=O)N1CCCC1C1(NC(c2ccc(=O)n(O)c2)=O)CC1 14096,c1(C(N2CCC(CC=C)(NC(c3nnn(C)c3C)=O)C2)=O)cc(C)c(C)nc1C 14097,C1(NC(COCCC)=O)CC1C1CCN(C(C2CCc3nnn(C)c3C2)=O)CC1 14098,N1(C(C(C)OC)=O)CC2CCCN(C(=O)C(C)Cc3cccc(C)c3)C2C1 14099,c1(CCC(=O)NC2CCC(Nc3c(SC)cccn3)C2)coc2ccccc12 14100,N1(C(Cc2ccc(C)nc2)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(CCO)C1 14101,N1(C(C2C(NC(CC3(CC)CCC3)=O)CCO2)=O)CCC2(COC(=O)N2)C1 14102,C1(O)(CCC)CCN(C(c2cc(C(N)=O)co2)C(=O)NC(C)CC)C1 14103,c1(CC(C(=O)OC)NCC2CCC3(CNC3)O2)c(F)ccc(Br)c1F 14104,c1(C(N2CCC3(C(CC(=O)O)CCC3)C2Br)=O)ncc(Br)c2ccc(F)cc12 14105,c1(C(=O)NC23C(CN(C(CC4CCC(OC)CC4)=O)C2)C3)cc(C)ncc1C 14106,N1(C(C2CCC(C)O2)=O)CC2C(C(=O)NCc3ncc(Cl)cn3)C2C1 14107,c1(C(=O)NC(CC(F)(F)F)c2ccccc2)cn2c(n1)COCC2 14108,c1(C(N2CC(NC(CC3CC(OC)C3(C)C)=O)(CO)C2)=O)ccc(Cl)c(N)c1 14109,N1(C(C)=O)C=Cc2ccccc2C1CC(=O)NC1(n2cc(CCCO)nn2)CC1 14110,c1(SC)ccc(C(=O)NCC(C)NC(=O)CS(=O)(=O)C2CC2)cc1[N+](=O)[O-] 14111,C1(C)(NC(C(C2CC(F)(F)C2)OC)=O)CCN(C(C2CC2c2ccccc2)=O)C1 14112,CCCC(O)(CCC)CC(=O)NC(C)CN(C)C(C1CCn2nccc2C1)=O 14113,N1(C(c2c(C(C)C)nco2)=O)C2CCC1C(CC(=O)NC1(C)CCC(C)C1)C2 14114,CC1CCC(CC(=O)NCCN(C(=O)CC2(C#N)CC2)CCOCCO)C1 14115,C(CN(C)C)(CC(C)C)NC(C1C(NC(c2cnc(C)s2)=O)C1)=O 14116,C1(F)(C(=O)OCC)CN(C(=O)Cc2c(F)ccc(Br)c2F)CC12CC2 14117,c1(C(=O)NCc2cn(CCC)nn2)cccc(F)c1C.C1(C)C(=O)O1 14118,c1(C(N2CCCC2)=O)ccc(-c2cn(C3C=CCCC3)nn2)nc1 14119,C1(C(=O)NCC(C)NC(COCCCC)=O)CCCCC1F 14120,Cc1ccc2sc(C(=O)NCC3C=CCN3C(c3cc(O)ccc3C)=O)cc2c1 14121,C1(NC(C#CC(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)C2(CCCCC2)C1 14122,N1(C(c2ccc(SCC)cc2)=O)CC2CC(C)N(C(C3COCC3COC)=O)C2C1 14123,N1(C(c2ccc(OC)c(Br)c2)=O)CCC2(CCN(Cc3nc(O)n[nH]3)C2)C1 14124,O=C(C1CCc2cccnc21)NC1CN(C(c2cccc(CO)c2)=O)CC1O 14125,C1(C(CC)C)CCN(C(=O)C(C2(O)CCC2)NC(=O)Cc2cccs2)CC1 14126,C(N=c1[nH]c(=NC2CCC(C)C2)[nH]c2c(F)cccc12)c1cccc(NCC)c1 14127,c1(CC(=O)NCCN(C(C)=O)CC)nc(C2CCOCC2)no1.C1(=O)C(C)(C)N1 14128,C(=O)(C(C(C)NC(C1CCC(=O)CC1)=O)C(C)C)N1CCC(CCCC)C1 14129,C(C(C)(C)CNC(c1cc(C)ns1)=O)NC(CCOCC)=O 14130,C#CCCCCCCNC(C1CC(C)CN(C(c2c[nH][nH]c2=N)=O)C1)=O 14131,Cc1cc(C(=O)NCC2CCCC2NC(C2CC23CCOCC3)=O)ccc1[N+](=O)[O-] 14132,CON1CCC(C(=O)NC2CCCC2(C)COC)CC1.C12CC(C1)N(C)C(=O)C2 14133,c1(C(=O)NC2C(NC(C3C(C#C)C3)=O)CC2)cccn1CC#C 14134,N1(C(C(C)(F)F)=O)CCC2CC2(NC(=O)CN2CCCNS2(=O)=O)CC1 14135,c1(C2(C)CC2)nocc1C(=O)NCC1(NC(c2cc[nH]c2)=O)CCC1 14136,C#CCCCCCC(=O)NCC(CC(C)C)NC(c1cncc(Cl)c1C)=O 14137,N1(C(c2cc(OC)ns2)C(=O)NC2CCN(C(C)=O)CC2)CC2CCCC2C1 14138,CC(C)CC(O)C(=O)NCC1CC(F)CN1C(=O)C1=CCCCC1 14139,C12(C)CN(C1)C(=O)CSC(CC)(C)O2.C12CC1NC2=O.C(C)(C)(C)OC(C)=O 14140,c1(OC)cccc(CCC(=O)NC2CCCCN(C(=O)C(C)(C)CF)C2)c1F 14141,c1(SCC(=O)NC2(CNC(C(N3CCCC3=O)C)=O)CCC2)nccn1C 14142,C1(C(=O)NC2C(NC(CNC(=O)OCC=C)=O)COCC2)CC2CCCC2C1 14143,N1(c2ncnc(OC)c2C)CCOC2CN(C(c3nc(Cl)ccc3F)=O)CC12 14144,CC1CC=CCC1C(N1CC(NC(c2ccccc2C(C)(F)F)=O)C(F)C1)=O 14145,c1(C(=O)NCC2C(C)(C)C2)ccc(Cn2cccn2)n1C 14146,c1(CNc2ccc(CC(=O)OC)cc2)cc(OC)ccc1N 14147,N1(C(CC2CC(OC)C2)=O)CCC2C(NC(=O)CC3CN(C)CC3O)CC12 14148,c1(OC)cscc1C(N1CCC(CCNC(C2CC2F)=O)C1)=O 14149,N1(C(C(C)OCC#C)=O)CCC(=CCNC(=O)Cn2ccc(C3CC3)n2)CC1 14150,c1(CC)conc1CC(=O)NC(CN(C)C)C(=O)N1CCCC1C(C)O 14151,c1(OC)cccc(-n2nc(-c3ccsc3)nc2C2CCCN2C)c1 14152,C=CCCCCCCCC(=O)OCCOC1CC(O)C1(C)C 14153,C1(C(N(CC(C)Nc2nnn(C)n2)C)=O)(SC)CCOCC1.C1CC(=O)N1 14154,N1(C(C2(C(C)=O)CC2)=O)CC(C(=O)NC(c2ccc(O)cc2)C)C(F)C1 14155,c1(OCC)ccc(C(=O)NCCN(C)C(c2ccccc2C2CC2)=O)cc1N 14156,N1(C(COCCOCC)=O)CCC(CNC(C2CC2c2cccc(C)c2)=O)CC1 14157,c1(C(=O)NCC2CCCN2c2ncc(Br)cn2)cc2ccc(O)cc2[nH]1 14158,C=CCC(C)C(=O)NC1(CCOC)CCN(C(c2ccc(N(C)C)nc2)=O)C1 14159,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14160,CCCCCCCNC1CCCC1C(=O)NCC.c12ccc(cc1)c(=O)[nH]2 14161,C#Cc1ncc(F)cc1NCC(=O)OC(c1ccc(Cl)cc1)C 14162,c1(NCC)cc([N+](=O)[O-])ccc1SCc1nc(C(=O)OC)nn1-c1ccccc1 14163,c1(OC)c(Cl)ccc(C(=O)NC(C)C(C)NC(=O)CN2C(=O)CN(C)C2=O)c1F 14164,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14165,N1(C(C(CC)c2ccccc2)=O)CC2(CC(NC(c3c(C)ncn3C)=O)CO2)C1 14166,Cc1[nH]nc(Cl)c1C(=O)N(C)CCC1CCCCN1C(C1C2(CC2)C12CC2)=O 14167,CC1CN(C(=O)Cc2nn(C)cc2Cl)CC1CNC(c1scnc1C1CCC1)=O 14168,C1(NC(CC(C)NC(=O)Nc2ccccc2)=O)CCCC(C)C1C 14169,C(=O)(C1=NNC(=O)CC1)N(CCCNC(c1cc(C)cc(C)c1)=O)CC 14170,c1(C(=O)NC2C=CCN(C(C3C(C(=O)OC)C3)=O)C2)cc(F)ccc1C(F)(F)F 14171,N1(C(C(CCC)CC2CC2)=O)CCC2(CCCN(C(=O)C(F)COC)C2)CC1 14172,c1(C(c2nnnn2C2CCOC2)C(CC)OCC=C)cn(C(C)C)nn1.C1(CO)CC1 14173,c1(N2CCCC3(NC(c4cnsc4)=O)C(C2)C3)ncnc2sc3ccccc3c12 14174,N1(CC=O)CCN(C(=O)CCC2CC2(F)F)CC1.C1(NC)CC(C)(C)C1 14175,C(C#Cc1ncccn1)NC(=O)Nc1cc(C(F)(F)F)ccc1Br 14176,C1(C(=O)OC)CCC(c2ccccn2)(NC(=O)NCC(F)(F)CCl)C1 14177,N1(C(CC2C(C(=O)OC)C2(F)F)=O)CCOC(C)(CNC(=O)C(=O)NC2CC2)C1 14178,Cc1cc(=NC(=O)NCCC2COc3ccccc3O2)c(-c2ccc(F)cc2)c[nH]1 14179,c1(OC(C)C(=O)N2CCC2CNC(c2cc(Br)[nH]n2)=O)ccccc1O 14180,N1(C(=O)CCc2cc(Br)ccc2F)CCC(F)C(NC(=O)CCCC2CCC2)C1 14181,c1(N(C(C)C)C)cccc(CC(=O)Nc2coc(-c3ccccc3Cl)n2)c1 14182,c1(N2CCN(C(=O)NCC3C(CC)OCCC3)CC2)nc(C2CC2)ncc1C 14183,N1(C(c2c(CC)nns2)=O)CCCC(F)(C(N2CCCC2C(C)(C)C)=O)C1 14184,c1(C(=O)NC2CC(NC(C(C(C)C)N(CC)CC)=O)C2)cc(F)cnc1O 14185,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14186,c1(C(C)NC(CC2OCCN(c3ncnc(C)c3F)C2)=O)cccc([N+](=O)[O-])c1 14187,c1(N2CCN(C)C(CNC(=O)CCc3ccc(F)nc3)C2)ncc([N+](=O)[O-])c(=N)[nH]1 14188,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CC=C(Cl)Cl)CC2C1 14189,O=C(C1CCCc2ncnn21)NCC1(F)CCN(C(c2cc(Cl)ccc2Cl)=O)CC1 14190,Cc1cnc(Cl)c(-c2nc(CNC(C)C)cs2)c1 14191,c1(C(=O)NCC2(CCNC(CC(COC)C)=O)CC2)cnn2ncccc12 14192,C1(OCCC)CCC(CC(=O)NC2CN(C(=O)C=CCF)C2)CC1 14193,C1(NC(=O)NCCc2nc(CSC)sc2)CC2(CCN(CC(C)(C)C)C2)C(=O)O1 14194,c1(NC(C(c2cccc(Cl)c2)NC(CSC)=O)C)ncc(C#N)cc1F 14195,C1(CCNC(c2csc(S)n2)=O)CCCCN1C(C1(C2CC2)CC1)=O 14196,n1(CC(=O)OC)cc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cn1 14197,C1(CC(c2n(C)nnn2)NC2(C3C(C)(C)C3(C)C)CC2)CC(F)(F)C(=O)N1 14198,N1(C(c2c(CNC(CC(CC)O)=O)cco2)=O)CC2CCCC(O)C2C1 14199,C(=O)(CC(C)CC(C)C)NCC(C(=O)N(CC(CC)O)CC)C(C)C 14200,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14201,O(S(=O)(=O)c1cccc2c1OC(C)C2)CC(C)=O.OC(F)F 14202,CC1(C)OCC2CC12C(N1CC(O)CC1C(N1CCC2(CCC2)C1)=O)=O 14203,Cc1n[nH]c(C)c1CC(=O)NC1CCC(CNC(c2cnsn2)=O)C1 14204,CCCC(=O)NCC(=O)NCC(F)CNC(=O)Cc1cccs1 14205,C1(CNC(c2cccc(CC)c2)=O)CN(C(c2sccc2C#N)=O)CCC1CO 14206,N1(C(CCCC)=O)CCC2(CCC(N(C(=O)C=Cc3ccco3)CC)C2)C1 14207,N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(=O)CC3(O)CC3)C1C2 14208,c1(C(N(CCCCCCNC(COC)=O)C)=O)cccc(SC)c1[N+](=O)[O-] 14209,C#Cc1cncc(C(c2nnnn2C2COC2)NC(CCC)c2cccs2)c1 14210,N1(C(c2c(C)sc(O)n2)=O)CCC2(CC1)CC(NC(c1ccc(O)nn1)=O)C2 14211,N1(C(CSc2n(C)cnn2)=O)CCC(C)(C)C(NC(=O)CSC(F)(F)F)C1 14212,c1(C(N2CC(C(N(c3ccc(C)cc3)CCC)=O)C(C)C2)=O)nc(OC)c(C)s1 14213,C1(C(=O)NCC2N(c3snc(COC)n3)CCCC2)CCC2(CCC2)OC1 14214,c1(C(=O)NCC(C)N(C(C2(OC)CC2)=O)C)cc(S(=O)(=O)CC)ccc1F 14215,CC1CC(c2cn(Cc3nnco3)nn2)CCN1C(C1CS(=O)(=O)C1)=O 14216,N1(CC(=O)NC(c2ccccc2)C)CCN(c2ncc(C(N)=O)cn2)CC1 14217,Cc1n[nH]c(C)c1CCC(=O)NCC1CC1NC(c1coc(N(C)C(C)C)n1)=O 14218,c1(OC(C)C(=O)N(C)CC2CCCN2C(=O)CCc2cnn[nH]2)ccccn1 14219,N(C1c2ccccc2CC1CNC(=O)C(O)P(C)(C)=O)C(CCOC)=O 14220,c1(OC)c(C(=O)NC2CC(C)CN(C(c3cnc(C)c(N)c3)=O)C2)cccc1Cl 14221,C1(C(N(CCN(C(c2ncccc2F)=O)CC)CC)=O)CC12CCCCC2 14222,N1(C(CCC=CC(C)C)=O)CCN(C(C2CCCN2C2CCOCC2)=O)CC1C 14223,N1(C(C(C)=C2CC2)=O)CCC2C(CCCN2C(=O)Cn2cnnn2)C1 14224,C(S(=O)CC(=O)N1CCC(N(C(N)=O)Cc2nc[nH]n2)CC1)c1cn(CC)nc1 14225,C1(C(=O)OC)CN(C(c2sncc2C)CNC2CCCCC2)CC(C)C1 14226,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14227,C1(NC(c2occ(C(N)=O)c2)=O)C2CC(CN(C(C3C4COCC34)=O)C2)C1CO 14228,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CCCOC)nn1)=O)N(C)C 14229,N1(C(CC2OCC(C)(C)OC2)=O)CC2=C(C1)CN(C(C1CN(C3CCC3)C1)=O)C2 14230,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C)CNC(C2CCO2)=O)CC1 14231,Cc1ncc(C#N)cc1NC(=O)C(O)CCNC(C1C2CCCCCC12)=O 14232,N1(C(C2=CCN(C(c3c(C)n(C)cc3)=O)C2)=O)CCC(O)C(C)(C)C1 14233,CC1(C)CC(NC(C2CN(c3ncc(O)cn3)CCN2)=O)CC(C)(C)O1 14234,C1(C(=O)NCCCN(C(=O)Cc2nn(C)cc2Br)CC)CC2CC(=O)C1C2 14235,N1(C(Cc2ccc(C)cc2Cl)=O)CCC(CNC(=O)Cc2ncc(C)o2)C12CCC2 14236,Cc1cc(F)c(CC(=O)NCC2CC(C)N(C(c3cnn(C(C)C)c3)=O)C2)cc1F 14237,C1(C#N)(C(=O)NCC(CNC(c2c(C(=O)OC)cccn2)=O)OC)CCCCC1 14238,c1(N2CCC(COC)(NC(=O)CN3CCCCC3C)CC2)ccn2nccc2n1 14239,C1(C2CCC2)(NC(c2ccn(C(C)C)n2)=O)CC1.C1CC(=O)NCCS1 14240,c1(CNC(C(c2c(OCCC)ccc(F)c2)(F)F)=O)cccc(F)c1C#N 14241,C1(CNC(CCOCCC)=O)CC(F)(F)CN1C(=O)C(c1ccn(C)n1)C 14242,c1(OC)cccc(CC(=O)NC2CC(O)(CNC(=O)Cc3ccc(Cl)nc3)C2)c1F 14243,N1(C(C(C)=C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14244,C1(N(CCC)C(c2ccc(CC)o2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 14245,C12CC3(CO1)CN(C3)C(CCC)C(=O)NC2.C(C)(C)(CN(C)C)N 14246,c1(-c2cn(CCCCC)nn2)cc(C)nc(C)c1.N12CCN(CC1)CC2=O 14247,c1(C(=O)NCC(C)N(C(=O)Cc2cn(C)nn2)C)ccc2ncnn2n1 14248,Cc1nnc2n1CC(C(=O)N(CC(O)CNC(c1nccnc1N(C)C)=O)C)C2 14249,C1(C(N(C2CN(C(C=C(CC)CC)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14250,C#Cc1cccc(C2CC2C(=O)NC2(CNC(c3ccc(F)c(Cl)c3)=O)CCC2)c1 14251,c1(C(N2CCC(CN(C(Cc3c(C)ccnc3)=O)C)C2)=O)cc2ncccc2o1 14252,C=C(C)C(CC(=O)N(C1CCCN(C(=O)CNC(C2CCCC2O)=O)C1)C)OCC 14253,C1(NC(c2ncc(OC)cn2)=O)CC(N=c2[nH]nc(-c3ccon3)s2)C1(C)C 14254,C12(CN)CN(C(=O)C(C)(C)n3ccc(C4CC4)n3)CC1CCO2.CC12CC(C=O)(C1)C2 14255,C1(OC)CCC(CC(=O)NCC2CC(C)N(C(=O)Cc3c(C)n[nH]c3C)C2)CC1 14256,C(=O)(C1=CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1)NC(CC#C)CC#C 14257,C1(CC(=O)N(CCC(=O)NCCC(C=C)C)CC)CCC(C)(C)O1 14258,C12(NC(COc3c(C)nn(C)c3C)=O)CCCC1CN(C(c1ccc(Cl)cn1)=O)C2 14259,c1(NC(C(=O)N(c2nc(C)c(Br)cc2Br)CC)=O)nc2cc(Cl)ccc2o1 14260,C1(CC(=O)NCc2c(CC)noc2C)CN(C(c2nc(C)ccc2F)=O)CCC1C 14261,C(c1ccc2[nH]ccc2c1)=CC(N1CCC(NC(C2CC2(Cl)Cl)=O)(CF)C1)=O 14262,c1(C(C)(C)C)csc2ncnc(NCCc3cn(CCCc4ccco4)nn3)c12 14263,c1(C(=O)NC2CC2F)cc(F)cc(Cl)c1.C12CC(F)(C1)CNC2 14264,CCCC(C(=O)NCCN(c1ncnc(=N)[nH]1)CC)S(N)(=O)=O 14265,c1(C(=O)NC2CC3CC(NC(c4cncc(C)c4)=O)C2C3)nc2ccccc2[nH]1 14266,c1(C(N2CC(N(C)C)C(C)(C)C2)=O)coc2c1CN(C(C1CCCC(O)C1)=O)C2 14267,C1(C)(C(N2CC(C(C)NC(C=CC=CC)=O)C2)=O)Cc2ccccc2N1 14268,C1(C(=O)NCC(F)F)CCNC2(CCCCCC2)C1 14269,Cc1cc(NC(=O)CO)n(CC(C2(O)CN(C(C(c3ccnn3C)F)=O)C2)C)n1 14270,CCC(O)C(F)(F)C(=O)NCC1(O)CC(NC(=O)CN2CCCCCC2)C1 14271,C1(NC(c2c(OC)c(F)ncc2)=O)CC2(CCN(C(c3scnc3C)=O)C2)C1 14272,N1(C(C(C2CCN(Cc3ccccc3)CC2)=O)=O)C2CCC1CN(C(=O)CO)CC2 14273,N1(C(C2CCC(OC)C2)=O)CC2CCCC(NC(c3cc(N)nc(Cl)c3)=O)C2C1 14274,C(N=c1nc(N2CCCC(C3(C)CC3)C2)c2c([nH]1)CCC2)c1ccc(C)cc1F 14275,C1(C(=O)OC)C2CC1N(C(=O)CC1CCN(C(C3OCCOC3C(C)C)=O)C1)C2 14276,c1(C(N2CCC(C3CCCN3C(=O)CC3CC3)C2)=O)ccc(Br)c(O)n1 14277,Cn1nnc2cc(-c3nc(CC(C)(C)C)nn3Cc3ccc(Cl)cc3Cl)cnc12 14278,Cc1cc(N)n2ncc(C(=O)NC3CN(C(=O)CSC(C)C)CC34CCC4)c2n1 14279,CC(C)CC(C)(O)C(=O)NC1CCCC(CC(=O)N(CC(O)CO)C(C)C)C1 14280,c12cc(F)ccc1NC(=O)C1CC21.C1(C(C)=O)CCCN(Cc2cncn2C)C1 14281,C1(OC)CC(NC(C2(C)CCCN2C(=O)C(C)OC)=O)C1(C)C 14282,O=C(C(O)C(F)(F)F)N1CCC(O)C1C(=O)NCCC1CC1 14283,CCC(C#N)C(=O)NC(C)CN(C)C(c1cc(C(F)F)nn1C)=O 14284,c1(NC2CCCN(C(C(C)(C)OC)=O)CC2)cc(=O)n(C)c(=O)n1C 14285,c1(C(C)C)c(F)ccc(CN2CCC3(CC3C(=O)NCC(N)=O)C2)c1F 14286,C(C(CC(C)C)C(=O)N(C1(COC)CCCC1)C)NC(C1CC=C(C)CC1)=O 14287,C1(C(=O)OCC2N(C(=O)OC(C)(C)C)CC(O)C2)Cc2c[nH]cc2S1(=O)=O 14288,c1(NC(=O)NC2C(c3ccc(C)o3)C2)cccc(N=c2cc[nH]cc2)c1 14289,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C2C1 14290,C1(CCNC(CSC)=O)CCN(C(c2noc3cc(Cl)ccc23)=O)CCC1(F)F 14291,C1(NC(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CCCC#N)CC1F 14292,N1(C(CCC)=O)CC2(CCCCCC2)C1.CCCCC(O)C(=O)OC 14293,O=C(C(O)C1CN(C(C2CC2c2ccco2)=O)C1)NCC(O)CC1CCCC1 14294,C1(C(=O)NCCC2N(C(CCN(CCC)C)=O)CCOC2)CCC(C)=C(C)C1 14295,N1(C(CCC#CC)=O)CCCC2(CCC(NC(c3ccnc(S)c3)=O)C2)C1 14296,C(=O)(C1=NOC2(CCC2)C1)N(CCCC(=O)NCCOCC(F)F)C 14297,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4CCC3C4)[nH]2)C1 14298,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)N(C(CNC(C(CC)NC(N)=O)=O)C)C 14299,S(=O)(=O)(c1ccc(Cl)cc1)NC(C(=O)NC(c1ccc(C(F)(F)F)cc1)C)CO 14300,c1(C(=O)NC(c2nocc2C2CC2)C)cc(-n2cc(-c3cc[nH]n3)nn2)nn1C 14301,c1(C(=O)NCC2N(C(C(C(C)C)OC)=O)CC2)cc(Cl)cc2cccnc12 14302,C12(NC(C(C)(C)O)=O)CC(CNC(c3cccc(F)c3O)=O)(C1)OC21CCC1 14303,C(=O)(CC(C(F)F)NC(=O)CCn1ccc(C)n1)NCCC1ON=C(C)C1 14304,Cn1ncc2cccc(CNC(N3CCC4CNCC4C3)=O)c12 14305,CC1CCN(C(=O)C(C)CC2CC2)CCN1C(=O)Cc1ncsc1Br 14306,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCCC(N)=O)N(CC(C(C)C)O)C 14307,c1(C(N2CC(NC(c3cc(CC)ncc3)=O)C(O)C2)=O)oc2ccccc2c1Cl 14308,c1(C(C)C)cccc(F)c1C(=O)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 14309,C#CCCCCC(=O)NC(CC1CC1)C(=O)NC(C)(C)C(N)=O 14310,c1(C(N(CCC(C)NC(C(CSC)C)=O)C)=O)cnc(O)nc1O 14311,Cc1ccc(C(=O)NCC2COCCN2C(c2ccc(F)o2)=O)c(Cl)c1 14312,C=CCC(CO)NC(=O)CNC(c1ccc(C2CCCO2)[nH]1)=O 14313,C1(CCNC(C2CC23CCC3)=O)CCN(C(C2CN(c3nncs3)C2)=O)CC1 14314,C1(C(C)CNC(=O)C(=O)N(C)C)CCCN(C(=O)C=CC(=O)OC(C)(C)C)C1 14315,C1(CNC(CCCC#C)=O)COC(C(F)(F)F)CN1C(=O)Cn1ccc(C)n1 14316,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14317,c1(C(=O)NC2C(NC(c3c(C)n4c(s3)ncc4)=O)C2)cc2c(s1)CC(C)CC2C 14318,c1(N2CCCC(C(C)NC(CC=CC=C)=O)C2)nc2ccccc2s1 14319,n1(CC)c(C(=O)N(C(CC)C(=O)NCc2ccnc(OC)c2)C)cnc1O 14320,c1(CC)nn(C)cc1CNC(C1CCN1C(=O)CSCC(=O)OC)=O 14321,c1(C(N2CC(NC(C(C)OCC=C)=O)CC23CCC3)=O)nn2c(c1C)OCCC2 14322,CCC(CC)(CC)C(=O)N1CCC(N(C(=O)Cc2csc(C3CC3)n2)C)C1 14323,C#Cc1ccc(C(=O)N(CCCNC(c2c[nH]c(=N)nc2CC)=O)CC)nc1 14324,C(CNC(=O)CCc1ccc(Cl)cc1Cl)(CC(F)(F)F)NC(C(CC)C)=O 14325,c1(C(=O)OC)cccc(OC)c1NS(=O)(=O)c1nc[nH]n1.C(C)=O 14326,c1(OC)ccc(S(=O)(=O)NCc2ccccc2NS(=O)(=O)C(F)(F)F)cc1Br 14327,C(CCCCCCNCC1CCOC1)(C=O)C1CCC(C(=O)OC)C1.OC 14328,N(C1CCCn2ncnc21)C(C1C2CN(C(=O)C3=C(Cl)CCCC3)CC21)=O 14329,CN1N=CC(CC(=O)NC2CC(CCC(N3CCOCC3CO)=O)C2)C1=O 14330,CC1=C(C(=O)NC2(CO)CN(C(C3C(C)(C)C3(F)F)=O)C2)CCCO1 14331,c1(-n2cc(COCC)nn2)nc(CCCO)nn1Cc1ccccc1F 14332,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC(F)F)cn2)=O)CC1C1CC1 14333,C(c1ccc(Br)cc1)=CC(=O)N(CC(=O)OCC)C 14334,N1(C(CC2(OCC)CC2)=O)CCCC1S(C)(=N)=O 14335,N1(C(C=CC(=O)NC2CC2)=O)CCC2(CC1)CN(C(C1CCOC1)=O)C2 14336,C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC1N(C(c2cc(OC)ns2)=O)CCC1 14337,CC1CC(NC(c2cccc(Br)c2)=O)CCN1C(=O)CC1CCCCN1C 14338,C#CC1CCC(CN(C(=O)C(C)NC(=O)COCC)C2CC(C)C2)CC1 14339,C12(C(N3CC(CN(C(=O)Cc4ccc(O)cc4)C)C3)=O)CCCC1OCC2 14340,C1(O)(CN(C(COCCC)=O)C)CCN(C(C2C=CC=CC=C2)=O)CC1 14341,C(CC(C(=O)Nc1csnc1C)NC(C)=O)NC(=O)Cc1ncoc1C 14342,C1(C(=O)NC2C(CCC)C2)CCCN(C(c2ccccc2N(C)CC)=O)CCC1 14343,C(C(C)(C)CC(=O)NC1CCCCC1CC(=O)Nc1cnc(CO)nc1)SC 14344,c1(C(N2C(C)CC(NC(C3CC(=O)NC(=O)N3)=O)C2)=O)ccc2c(c1)OCCC2 14345,c1(COC(C(=O)N(CC(C)NC(C(C)NC(C)=O)=O)C)C)ncc(C(F)F)s1 14346,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14347,c1(C(=O)NC2C(NC(C3CCCOC3)=O)CC2)ncccc1OCCOC 14348,Cc1nn(C)c(C(=O)NN2CCN(C(=O)N(C(C)CC(C)C)C)CC2)c1I 14349,c1(C(N2CC(CCC)C(NC(=O)CCC=CBr)C2)=O)cc(C)cc(O)n1 14350,C(=O)(C(C)(CC)CCCCCC)NCCC(CNC(c1n(C=C)nnc1)=O)O 14351,C1(CCCNC(c2cnn[nH]2)=O)CCN(C(=O)Cc2cncc(C(F)F)c2)CC1 14352,N1(C(C2(CC(C)C)CC2)=O)CCN(C(=O)Cc2cc(C)nn2C)CC1.C(C)N 14353,C1(C)(CNC(COCCOCC)=O)CCCN1c1ncncc1Br 14354,c1(C(=O)NC(CN(C(C(CC#C)C2CCCCC2)=O)C)(C)C)cc(C)ccc1N 14355,c1(CNC2c3cc(OC)sc3CC2)nc(O)c2c3c(sc2n1)CCCC3 14356,N1(C(CC)=O)CCCCC(CNC(c2cn(Cc3ccccc3)nn2)=O)C1 14357,O=S(=O)(c1ccc2nc(N3CCCC3c3ccc(Br)s3)ccc2c1)N1CC2CC2C1 14358,c1(NC2CCC(C(N3CCCC(C(=O)OCC)C3)=O)CC2)ccccc1S(C)=O 14359,C1(c2nc(-c3ccc(COC(C)C)cc3)nn2-c2ncnn2C)C(C)CCCC1C 14360,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CCC1 14361,c1(NC(CCC)C)cc(=NCCc2cnc3ncccn23)[nH]c(COC)n1 14362,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14363,CONC(=O)CN(C1CN(C(=O)C(C2CCCOC2)OC)C1)C 14364,C1(SCC(C)=O)CC(=O)N(C)CC1CCC(C)C 14365,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14366,N1(C(=O)C(F)=CC2CC2)CCN(C(=O)CCC(F)(F)F)C2CC12 14367,C1(OCCOC)CCN(N2CCN(S(=O)(=O)C3CC3)CC2)C1c1cccnc1 14368,CC(CC#N)N=c1cc[nH]cc1S(=O)(=O)NCC1(OC(F)F)CCCCCC1 14369,N1(C(C2C(CNC(CCCN=[N+]=[N-])=O)OCC2)=O)C(CO)CCC12CCC2 14370,c1(C(=O)NC2C(C(N(CC(=O)OCC)C(C)C)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 14371,c1(CC)cccnc1C(=O)NCCC(O)CNC(C1CNC(=O)N1)=O 14372,c1(C(=O)OCC(=O)NC(C(=O)N(C)C)C2CC2)cnn(CCO)c1 14373,C(=O)(C(C)CC(C)C)N1CC(O)(C(C(=O)NC(C(=O)OC)(C)C2CC2)F)C1 14374,c1(CNC23CC(C(=O)NCCNCCO)(C2)C3)cc(Br)cc(F)c1F 14375,N1(C(Cn2c(C)ncc2)=O)CC2C(C(=O)NC(C)C(C)CO)C2C1 14376,c1(C(=O)NC(C2(O)CCN(C(COCC(=O)OC)=O)C2)C)nsc2ccccc12 14377,N(C(=S)N1CCC1CCc1ccc(OCC)cc1)CC=C 14378,Cn1cc(C(=O)NCC23CC2CN(C(c2cnc(C(F)(F)F)cn2)=O)C3)c(Cl)n1 14379,CCC(C)(COC)CNC(=O)C(O)CNC(c1cncc(O)c1)=O 14380,C(C)(C)(CC(=O)NC(C)CC(C)NC(=O)CCCCc1cnc[nH]1)OC 14381,C1(C(N(CCOCC=C)C)=O)CC(N=[N+]=[N-])CN1C(C1C=CCC1)=O 14382,C12CN(CC1O)Cc1ccc(cc1)C(=O)N2.c1(CC)ccn(CC(=O)O)n1 14383,c1(OC)cc(F)c(C(N2CCC(NC(c3cnn4ccn(C)c34)=O)C2)=O)cc1N 14384,c1(C(N(C2CCCN(C(=O)Cc3ccsc3)C2)CC)=O)cc(C)nc(OC)n1 14385,N1(C(C2CCC(SCC)CC2)=O)CCC(NC(=O)C2=CCCCC2)CC(C)(C)C1 14386,N1(C(C(C)OC2CCCCC2)=O)CCC(C)C(NC(=O)C(C)(C)CF)C1 14387,CCC(CC)C(=O)N(C)CC1CN(C(c2ncn(C(C)(C)C)n2)=O)CCO1 14388,c1(C(=O)OC)cnn2c1CN(C(C1CC1CNC(=O)CN(C)C)=O)CC2 14389,N1(C(CC(=C)C)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC2C1 14390,c1(CN(C(C2C(C(=O)OC)C2)=O)CC=C(C)C)ccccn1 14391,C#Cc1cccc(C(=O)NC2CCN(C(c3[nH]c(C)cc3C)=O)C(C)C2)c1Cl 14392,c1(N2CCC(CC(CC)C)CC2)nc2c(c(=NC3CCSC3)[nH]1)CCCCC2 14393,C(C(CO)(CO)NC(c1cncnc1)=O)N(C)C(C12COCC1C2)=O 14394,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14395,C1(NC(C(CC(=O)OC)C)=O)CC2CCC1CC2NC(=O)CC1(CS(C)(=O)=O)CC1 14396,c1(C(=O)NC23C(CN(C(C(C)CF)=O)C2)C3)cccc2c1OCCO2 14397,C1(C(N2CC(CNC(c3cc(OC)no3)=O)(COC)C2)=O)CCCCN1C(C)C 14398,C(CC(C)(C)C(=O)N1CCCC(N(C(=O)Cc2csc(Br)n2)C)C1)OC 14399,C1(NC(C(CCCOC)NC(c2cc[nH]n2)=O)=O)CCCCCC1(C)C 14400,N1(C(C)=O)CCCC(N(CCC#N)CC2CCN(C(=O)OC(C)(C)C)C2)C1 14401,N1(C(CC=C)=O)CCCN(C(=O)C(C)OCCCC)C(C)C1 14402,N=c1cc[nH]cc1C(=O)NC1CCCC1NC(c1ccnc(OCCO)c1)=O 14403,C1(O)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14404,c1(CC(=O)N(CCN(C(C2C(OC)CCC2)=O)C(C)C)C)c(C)nc(O)nc1C 14405,Cc1nc(CNC(C2CC2c2ccco2)C)sc1C(=O)O 14406,Cc1c[nH]cc1C(=O)NCCOCCNC(C1CC1C(C)(C)C)=O 14407,C12(CNC(C=CC(CC)C)=O)CC(CNC(=O)CC(C)F)(C1)C(C)(C)O2 14408,C1(N)(C(=O)NCCc2nc(OC)ccc2F)CCCN(CC)C1 14409,CCCC(CC)CCC(=O)NC1CCC2CCN(C(c3coc(C)n3)=O)C1C2 14410,CCCCS(=O)(=O)NC(C)C(=O)NC(CNC(c1ccc(C2CC2)nc1)=O)CO 14411,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14412,c1(CCC)nc(-c2coc(C)n2)n(CCS(C)(=O)=O)n1 14413,N1(C(=O)COC2CCC2)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14414,N1(C(CN2C(C)CCC2)=O)CC=CC(NC(c2ccn(C)n2)=O)C1 14415,N1(C(C(c2ccccc2)SC)=O)CCOC2(C1)CN(C(c1cnn(C)c1F)=O)C2 14416,C1(NC(Cc2c(SC)cccc2)=O)CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 14417,C1(C2CN(C(=O)CNCc3ccccc3)C2)(NC(CC2CCN(C)C2=O)=O)CC1 14418,c1(C(N2CC(N(C(c3c(C)snn3)=O)C)C(O)C2)=O)cncc(N=[N+]=[N-])c1 14419,c1(C(N2CCC(C(CC)O)C2)=O)cccnc1N(c1ccccc1)c1ccccc1 14420,C1(C(N(CC(C)NC(=O)CN2CCC(C(N)=O)CC2)C)=O)CCCC1S(C)(=O)=O 14421,c1(C(N(C2CN(C(=O)C(C3CC=CCC3)F)C2)C)=O)cncc2nc[nH]c12 14422,C=Cc1ccccc1N(C(=O)CC(=C)C)c1nnnn1Cc1cccs1 14423,Cc1c(C(=O)NCCCC(C)NC(=O)CCC2CCCC2)cc(C2CCC2)n1C 14424,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14425,N1(C(C(=O)N(C)C)=O)CCC2CCN(Cc3nc(-c4ccccc4)n[nH]3)CC12 14426,C1(O)(C(C(=O)NCC(COCC(=O)Nc2c(C)scc2)C)N(C)C)CCCCC1 14427,C1(C(=O)NC(CSCC(=O)NC)=O)CCC(C(F)(F)F)O1 14428,CC1CN(C(C2CC3COCC3C2)=O)CCC1CNC(c1c[nH]c(C(N)=O)c1)=O 14429,c1(CC(N2CC3(CC(CNC(C(C)(C)C4CC4)=O)C3)C2)=O)csc2ccccc12 14430,Cc1cc(C(N2CC(F)CC2C(=O)N(C)CCN(C)C)=O)cc(O)c1 14431,N1(C(CCSC)=O)CC2(C(=O)NC3CC(CCC(N)=O)C3)CC1CO2 14432,N(C1CC2(CN(C(=O)C=CCO)C2)n2ccnc21)C(C1C2C(=O)C3C(C2)C31)=O 14433,C1(C(N(CCNC(c2nc(CCOC)oc2)=O)C)=O)CCc2nnc(O)n2C1 14434,Cc1cccc(OC(=O)CCC(C)C(F)(F)C(F)(F)F)c1.C1(=O)CO1 14435,CCCCC(C(=O)N1CCN(C(c2cc(CO)on2)=O)CC1CC)N(C)C 14436,c1(C(C(=O)Nc2ccc(C#C)nc2)(C)C)ccc2ccccc2c1 14437,C(=O)(C(C)S(N)(=O)=O)NC1CCN(C(CCSc2ccc(C)cc2)=O)CC1 14438,C(=O)(CC1C(=O)Nc2ccccc21)NCCC(CNC(C(C)(C)CC(F)F)=O)O 14439,C1(C2CCNCC2)(C(=O)NC(C)CCc2ccccc2)CCC1 14440,C(=O)(C(C)CC(C)(F)F)NC(CN(C)Cc1c(C)cccc1C)C 14441,C1(NC(C(=O)NC(c2cccnc2Br)C)=O)CCCN2CCSCC12 14442,C(=O)(CCCCC(N)=O)N(C1CCCN(C(C2CC23CC(O)C3)=O)C1)CC 14443,CC1OC2(C(=O)NC3CC(O)(CNC(=O)CN(C)C)C3)CCC1CC2 14444,c1(SC)nc(N2CC=CC(NC(=O)Cc3ccc(C)s3)C2)[nH]c(=N)n1 14445,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14446,c1(C(=O)NC2CC(NC(c3c(-c4cn(CC)nc4)n[nH]c3)=O)C2)cc[n+]([O-])cc1 14447,c1(C2C(=O)N2)ccc(O)cc1.Cc1ccc(NC(N2CC(F)(F)C2)=O)o1 14448,C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC2(CCN(C(=O)C=CCF)CC2)C1 14449,C1(C(N2C(C(C)(C)O)CC2)=O)CCC(CNC(c2ccsc2Cl)=O)O1 14450,c1(OC)ccncc1CC(=O)NC1COCC1NC(c1cnn(CCO)c1)=O 14451,c1(C(N2CC3(CCN3C(C3CCOC3)=O)C2)=O)cc2n(c1)CCOC2 14452,c1(C(=O)NCC(C)N(C(=O)CC2C=NN(C)C2=O)C)coc2c(Cl)cccc12 14453,C1(N(C(=O)CC2(C)CC2(F)F)C)CCC(NC(=O)COc2cccc(Cl)c2)CC1 14454,c1(C(C)NC(c2c(C)n[nH]c2)=O)ccc(CC(=O)C2CC2)cc1.c1(C=O)c[nH]c(Br)c1 14455,C1(C(=O)NC(c2ccccc2)CNC(c2n[nH]c(C)c2O)=O)CC12CCCCC2 14456,C1(=O)C(CCC)N1.C(=O)(C(C)C=C)N(CC(=O)NCC#C)C 14457,C1(CNC(=O)C=Cc2cn[nH]c2)(NC(C2CC3CC3C2)=O)CC2CCC1C2 14458,c1(N(C(=O)CCC(N)=O)C(c2ccc(O)cc2)C)ccc(N2CCOCC2)nc1 14459,C(CC(F)(F)CC)NC(CC1CC(C(=O)NCc2onc(COC)n2)C1)=O 14460,CCC(CC(=O)NC1(c2ccccc2)CC(NC(c2cccc(F)c2)=O)C1)OC 14461,c1(C(N(C2CCN(C(CSC)=O)C2)CCO)=O)cc(C)nc(N2CCCC2)n1 14462,C1(NC(c2c(C)ncs2)=O)CCCOC12CCN(C(=O)CC1CC=CCC1)CC2 14463,N1(C(CC(C(C)C)C)=O)CCN(C(c2noc3ccccc23)=O)CC(CO)C1 14464,C1(NC(C2C(C(C)C)C2)=O)C=CCCC1C(=O)NCc1cn(C(C)C)nn1 14465,CC1CN(C(=O)CCCC2CC2)CC1CNC(c1cc(-c2ccns2)on1)=O 14466,C1(CNC(c2ccnn2CCF)=O)CN(C(C2CC2[N+](=O)[O-])=O)C2(CCC2)C1 14467,C(=O)(C(C)(C)CC(C)C)NCCSCC(=O)NCC1N(CC)CC1 14468,N1(C(CCOC)=O)CCCC1C(C)(C)CNC(C1C(C)C1(F)F)=O 14469,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14470,c1(CCC)ccccc1NC(=O)C#CCNC(=O)C(C)CO 14471,C1(Nc2cncc(SC)c2)CCCC(NC(=O)NC2CCCCC2CO)CC1 14472,C12(C(N(C)CC3CCN(C(CC=C(C)C)=O)C3)=O)CCCCC1OCC2 14473,c1(CC)nnc(CCNC(=O)C(C2CCN(C(=O)C(C)(C)SC)C2)F)s1 14474,CC1N(C(C2CCN(C(c3n[nH]c4c3COC4)=O)C2)=O)CCC1(C)C 14475,CSC1=C(C(=O)NCCC(C)NC(c2ccc(C)cn2)=O)CCCC1 14476,Cc1cn(CC(F)(F)F)[nH]c1=NC(=O)N1CCN2CCCCC1C2 14477,c1(C(=O)NCCC(=C)CNC(c2ccc(N)c(Cl)c2O)=O)nsc2ccccc12 14478,c1(C(C)OC(CC(=O)NCCC(C)(C)NC)C)cccc(C)n1 14479,O=C(CCCC1CCCCC1)N1CC(Nc2nnc(-c3ccncc3)s2)C1 14480,C(CCN(C)C(C1CCC1(C)C)=O)(C(C)(C)C)NC(C(C)NC(C)(C)C)=O 14481,N1(C(c2ccc(C)n2C)=O)CCCC2C1CCCN2C(=O)C(F)F 14482,c1(C(=O)NC(CN(C(=O)CC(C)C(F)(F)F)CC)C)cnn2ccncc12 14483,c12nc(nc(=N)[nH]1)NC(=O)C1CN2C1.C(C(F)(F)F)SCNC(=O)OC(C)(C)C 14484,C1(C(N(C2CCCCC2)CCNC(C(CCC)F)=O)=O)CCc2nc[nH]c2C1 14485,N1(C(C(C(C)C)NC(COC)=O)=O)CCCC(C)(CNC(c2ncc(C)s2)=O)C1 14486,c1(C(N(C(CNC(c2cc(C)on2)=O)C)C)=O)ccc(NC2(C)CCCO2)cc1 14487,c1(OCC(N2CCC(CNC(=O)C(CO)c3ccccc3)C2)=O)cccc(Cl)c1 14488,CCCN=C(NCCc1cccnc1N1CCS(=O)(=O)CC1)N1CCC(CF)C1 14489,c1(C(N(CC(CC)NC(c2cnn3ccn(C)c23)=O)C)=O)cc(C)n(C)c(=O)c1 14490,C1(C)(C(C)(C)C)CC(C(N2CC(NC(=O)CCc3cccs3)C2)=O)C1 14491,c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C)cccc(C#CC2CC2)c1 14492,C1(CNC(Cc2cnc(C)[nH]2)=O)CCCCC1NC(=O)C(C)C1CCCC1 14493,c1(C(=O)NCC(CNC(CCCCC#C)=O)(C)F)ccc2cccnc2n1 14494,CCCCN=C(NC1CCCC(COC)C1)N1CCC2CCN(C)C(=O)C2C1 14495,C1(C(=O)NCCC(C)(C)N(C)C)(CNC(CCCSC)=O)CC2(CC2)C1 14496,N1(C(CC(=C)Br)=O)CC2CCC(CNC(=O)CCCCCC)(C2)C1 14497,C(=O)(C1SCCc2sccc21)N1CCOCC(CNC(C=CCOC)=O)C1 14498,N1(C(CCCOCC)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC1C1CC1 14499,c1(C(=O)NC2CN(C(C3CCCCO3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 14500,c1(CN=C(NCC(C)OC)NC2CCCCCCC2)cc(C(F)(F)F)c(Br)nc1Br 14501,CC(C)CCCCCC(=O)N1CCC(O)(CNC(=O)C2=CC3C=CC2C3)C1 14502,C(=O)(C(O)C(C)(C)C)NCC(C)N(C)C(c1nn(C)c(Cl)c1Br)=O 14503,Cc1cc(Br)cnc1C(N1CCCC1C(C)O)C(=O)NCCC#N 14504,C(=O)(C(C)C(=O)NCc1ccc(C(=O)NC2CC(=O)N(C)C2)nc1)OC 14505,c1(C2C(CNC(=O)NC(C)C(F)F)C2)cccc(Cl)c1Cl 14506,Cc1ccc(F)c(CNC(C2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)CC2)=O)c1F 14507,C(=O)(C(F)C(F)(F)F)NCCC1N(C(c2cc(C(C)(F)F)ncc2)=O)CCCC1 14508,CCC(CCCO)NC(c1sccc1CNC(=O)CC(CC)SC)=O 14509,N1(C(c2c(C)onc2)=O)CC(C)(C)CCC1CNC(=O)C(C#N)C(C)C 14510,Cc1cnccc1C(C(=O)NCC(C)C)N(CCN1CCCCC1)C 14511,N1(C(C2N(C(C)=O)CCCC2)=O)CC(NC(c2cc(C)cnn2)=O)CCC(O)C1 14512,c1(CC(CC)NC(=O)N(C)CC2CCCO2)ccc(F)cn1 14513,N1(C(c2ccc(CC)cn2)=O)C(C(=O)NC2CCCC2COC)C2CC(O)C1C2 14514,C(=O)(CC(CNC(=O)C(C)(C1CC1)OC)OC)NC(C(=O)OCC)CC 14515,C#Cc1cccc(C(=O)NCCC2(C#N)CN(C(=O)OC(C)(C)C)C2)c1Cl 14516,N1(C(c2cncc(C(=O)OC)n2)=O)CCCN(C(=O)C2=COCC2)CC1CO 14517,N1(C(=O)CN2CCNC2=O)CC2(CC(NC(c3cncnc3)=O)c3nccn32)C1 14518,C(=O)(CCC(F)(F)F)N1C(CC)C(C(=O)NCC2(Cl)CC2(F)F)CC1 14519,N1(C(c2cn(C(C)C)nc2)=O)CCC(C=CC(=O)N(C2(C)CCC2)C)CC1 14520,CC1CCC2CCCN(C(c3nnn(C(C)C)c3C(F)F)=O)C2C1 14521,C=CCCN=C(NCCOc1ccc(F)cc1)NCC1(C)CC1(F)Cl 14522,C1(N(C)C(c2cnc(O)o2)=O)CCN(C(c2cc(Br)n(C)n2)=O)CC1 14523,N1(C(C(OCC)OCC)=O)CCN(C(c2cc(O)cc(=O)o2)=O)CC1CC(F)F 14524,CC(C)(C(=O)NCCNC(c1csc(C(F)(F)F)n1)=O)C1CCCOC1 14525,C(=O)(C(CC(F)F)NC(=O)C=NOC)N(CCCC)CC 14526,c1(CC(N2CC(C)(NC(C(=O)OCC)=O)C2)=O)c[nH]c2cc(OC)ccc12 14527,c1(C(=O)NCCCN(C)C(c2ccc(-c3ccccn3)o2)=O)n[nH]cc1I 14528,C=C1CC2CC1CN2C(=O)CC1CC(C)N(C(c2cnn(C)c2C=C)=O)C1 14529,c1(NC2C(NC(C(N3CCCCC3)C)=O)CS(=O)(=O)C2)ccc2nnnn2n1 14530,C=C(C)C1CCC(C)(O)C(NC(c2ccc3ncccc3c2C)=O)C1 14531,N(C(=NCCCOC1(C#N)CCOCC1)NCC1CC1c1ccccc1)CCOC 14532,C1(NC(CC2C(N)CCC2)=O)CCCC(F)(F)C1 14533,c1(C(=O)NCC2CCN(C(C(C)SC)=O)C2)sc2ccccc2c1Br 14534,CC(C)CC(C)(CNC(c1ccc(C2CC2)nc1)=O)NC(C1CC12CCC2)=O 14535,Cc1cc(=O)oc(C)c1C(=O)NC(C)(C)CNC(=O)CCC=CC(C)C 14536,C1(NC(C(C)(F)F)=O)CCC2CCN(C(c3ccc(NC4CC4)nc3)=O)C1C2 14537,c1(CC)cc(C(=O)NCC2CC2CNC(=O)COCc2cc(C)no2)c(C)o1 14538,CC1CCCN1CCc1cn(C2CCC(c3ncc(C(=O)NC4CC4)s3)C2)nn1 14539,C1(C#N)(C(=O)NC(C2CN(C(c3cc(CO)ncn3)=O)CCO2)C)CCOCC1 14540,Cc1ccnc(N2CCC3C(C(=O)Nc4ccc(Br)cc4C)C23)c1[N+](=O)[O-] 14541,Cc1cnc2n1CCN(C(=O)C(C)(C1CC1)N(C(=O)CCc1cn(C)nn1)C)C2 14542,C(=O)(C1CCc2nccn21)N1CCCC(C(=O)NC2(C)CS(=O)(=O)C2)CC1 14543,C(=O)(C1=C(Cl)CCOC1)N1CCN(C(C2CCN(C(=O)NC)CC2)=O)C2C1C2 14544,C(c1cnccn1)=CC(=O)NC1CC1NC(C1(N2CCOCC2)CC1)=O 14545,CCC(CC(=O)NC1CCCC(C(=O)NCCC(C)(C)OC)C1)OC 14546,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2n[nH]cc2c1)=O)C1CC1 14547,CC1(C)C(NC(=O)CC2CC(F)(F)C2)CC1CC(=O)NCC1CCC(F)(F)C1 14548,Cn1nccc1C(=O)NCC(O)CNC(c1cc(-c2ccncc2)[nH]n1)=O 14549,CC1CC2(CC(NC(C3CC(O)CN3C(c3ccc(O)c(F)c3)=O)=O)C2)C1 14550,C=C1CCN(C(C2CC3(CCO2)CC3)=O)C(C(=O)NCC2C=CCCC2)C1 14551,N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CCCC(C2(NC(C3CC3(C)C)=O)CC2)C1 14552,c1(C(=O)NCCCOCCNC(C(C)SC(C)C)=O)cc(Cl)cnc1NC(N)=O 14553,c1(CN(C=O)C(c2nnc(C3CCCOC3)o2)C)ccc[n+]([O-])c1 14554,N1(C(c2cnc[nH]2)=O)CC(NC(C2CCN(c3cc(F)ncn3)CC2)=O)C(O)C1 14555,C(=O)(CCC(=O)N(C)C)NC(C1CN(C(C2(C(O)C(F)(F)F)CCC2)=O)C1)C 14556,C(C)C(=O)NC1(CCOCCN(CCC)C(C2(C)CC2)=O)CC1.C(C)(C)(C)OC 14557,c1(CC(C(=O)NCC(CNC(c2nnc(CC)s2)=O)O)F)ccc([N+](=O)[O-])cc1 14558,C1(C(N2CC3C(CNC(C(c4ccc(C)o4)C)=O)C3C2)=O)CC2OC(=O)OC2C1 14559,C12(NC(=O)CONC(=O)C(F)C3(O)CCOCC3)CCCC1C2(F)F 14560,Cc1ccc2nc(C(N3CC(O)CC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14561,C(=O)(CC(CC)C(C)(C)C)NCCCCNC(CC(C=C)CCC)=O 14562,N1(C(c2cn(CC=C)nn2)=O)CC2=C(C1)CN(C(C1(CCC)CCC1)=O)C2 14563,C(CNC(C1CC2CC1CC2O)=O)(CC(F)(F)F)NC(=O)C=Cc1ccoc1 14564,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14565,C12(CNC(CCNC(N)=O)=O)CCCCC1N(C(=O)CCc1cn[nH]c1)CC2 14566,n1(CC(=O)NC2C3CN(C(c4cccc(C(N)=O)n4)=O)CC23)ncccc1=O 14567,C(C)(CO)(C(=O)N1CCC(C(C)CNC(=O)Cn2ncc(Cl)c2C)CC1)OC 14568,C1(CNC(c2ncn(CC)c2)=O)CCCCN1C(=O)CCn1ccnn1 14569,N1(C(c2nc(COC)sc2)=O)C2CCC1CN(CCN1C(=O)CCC1=O)CC2 14570,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1C(F)F)=O)C2 14571,C1(NC(Cc2cc(CN(C)C)no2)=O)CN(C(C2CC2F)=O)C2(CCCC2)C1 14572,C1(N(C)C)CCCCC1NC(=O)C(C1CCN(C(C2CCNC2=O)=O)CC1)O 14573,c1(CNCCN(C2CCCCC2)C(C=CC(C)(C)SC)=O)cn2c(n1)CCCC2C 14574,CN1CCCC(C)(Sc2ccc(F)cc2)C1.N12CC3CN(CC13)c1nc2ns1 14575,N1(C(C2(CC)CCCC2)=O)CC(CC(=O)N(C)Cc2cnn[nH]2)C(C)C1 14576,N1(C(c2c[nH]c(C)c2Br)C(=O)OCC)CCN(CCCOC)C(CC(=O)OC)C1 14577,c1(CN2CCN(C(c3c(C)nc(C(C)(C)C)s3)=O)CC2C)cc2ncccc2[nH]1 14578,C#CCCCCCC(=O)NCC(CCOC)NC(=O)CC1C(=O)NN=C1C 14579,C#Cc1cc(C(N2CCCCC2CNC(=O)C(O)Cc2cnc[nH]2)=O)ccc1Cl 14580,N1(C(C2CCC(=O)CC2)=O)CCC(C(=O)NC2CC(O)C2)C12CCC2 14581,C12CCCN(C1)C2=O.c1(CC2N(C(C)=O)CCC2)ncccc1Br 14582,c1(C(N2CCC(NC(C3CCN(CC4CC4)CC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 14583,c1(C(=O)NCC2CCN(C(c3nc(C)n(C)c3)=O)CC2)c(F)cncc1Cl 14584,c1(C(=O)NCC(CC)(C)NC(=O)C(C2CCOCC2)N(C)C)cc(C#N)c[nH]1 14585,C#Cc1cccc(NC(C2(NC(=O)COC(C)CC)CC2C)=O)c1 14586,c1(C(=O)OC(C)(C)C)ccc(C(N(C(C)CC(=O)OCC#N)C)=O)cc1.C=O 14587,CCC(C)(CC)C(=O)NCC(C)(CO)NC(c1cnc(C(C)OC)s1)=O 14588,S(=O)(=O)(c1ccc(Br)cc1N1CC=C(C(C)(C)C)CC1)N1C(C)CC(C)C1 14589,c1(OC)ccncc1C(=O)NCC1(C(C)NC(c2cc(F)cs2)=O)CC1 14590,C1(OC)CC(C)CN(C(=O)CC(C)CNC(C2CCOC2(C)C)=O)C1 14591,c1(C(=O)N(O)Cc2cccc(Cl)c2)cc2c(cc1Br)OCCO2 14592,CC1CN(C(C2(Cl)CC2(C)C)=O)CC1NC(c1ccnnc1O)=O 14593,C#Cc1cnn(C)c1NC(N1CCCC1CC)=O 14594,C1(C(=O)NCC(CC(C)C)NC(=O)COC2CCOC2)CCc2nnn(C)c2C1 14595,N1(C(C2C(NC(C(C(CC)CC)F)=O)C3CCC2C3)=O)CC2(CNC(=O)OC2)C1 14596,c1(CC)cc(CNC(C(=O)N2CCC(C)CC2)C(C)C)ccc1Cl 14597,c1(C(N(CCCN(C(c2[nH]cc(C(=O)OC)c2)=O)C)C)=O)ccc(OC)nc1 14598,C1(C(=O)NC(CC)CNC(c2conc2C(=O)OC)=O)C2COCC12 14599,N1(C(CC(C)F)=O)CCC(NC(=O)CCOCC(F)(F)C(F)F)C(C)C1 14600,C1(C(=O)NC2(CCNC(c3c(C)cco3)=O)CCCC2)CC1C1CC1C 14601,c1(C(=O)NC(CNC(=O)C=CBr)C2CC2)cc(Cl)ccc1F 14602,CC(C(=O)N(C1CN(CC(=O)N(C(C2CC2)C2CC2)C2CC2)C1)C)C(C)(C)C 14603,C1(CN(C(C)=O)C(=O)C2CC2)CCCCC1Nc1cccc(F)c1 14604,c1(CC)cccc(C(=O)N(C)CCN(C(c2ccc(CC)o2)=O)C(C)C)c1O 14605,c1(C(N2C(CN(C)Cc3cc(CCCC)no3)CCC2)=O)cc(F)ncc1OC 14606,c1(C(=O)NCCN(CCCCCC)C(=O)CN2CCC(O)CC2)cc(C)ncc1C 14607,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14608,Cc1sc(C)c2sc(C(=O)NCC3CCCCN3C(=O)COC3CC=CC3)cc12 14609,N1(C(C)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1C1CC1.c1(C(=O)OC)ccon1 14610,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14611,S(=O)(=O)(c1cnc(NCC2CN(C)CCO2)c(Cl)c1)N(C(CCSC)C)C 14612,C(=O)(C(CC(C)(C)C)NC(c1cocc1C)=O)NCC(CC(=O)OC)O 14613,N1(C(c2c(CC)nn[nH]2)=O)CCN(C(C2C3CN(C)CC23)=O)CC1C1CC1 14614,CCC(C)CCC(O)CC(=O)NCCNC(=O)C(C)(O)COC 14615,C(C1CCCN1C(=O)Cc1cccs1)=CC(=O)NC1CCC1 14616,N1(C(C(C)NC(C)=O)=O)CCCC(C)(CNC(=O)COC2CC(F)(F)C2)C1 14617,N1(C(c2ccc(F)c(C)c2O)=O)CCCN(C(c2ccc(CO)cc2)=O)CC1C 14618,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14619,CC1(CNC(=O)CP(C)(C)=O)COCCN(C(c2cc(C#N)ccn2)=O)C1 14620,c1(C(N2C3CC(NC(=O)CC4CCCCO4)(C3)C2)=O)cnc2occc2c1 14621,C#CCC(CC(=O)N(C)Cc1csnn1)NC(=O)Cc1cnns1 14622,c1(CC(=O)NCCCCCNC(C2CC2CF)=O)cc(O)cc(Br)c1 14623,Cc1nn(C)c(C)c1C(C)C(N1CCC(O)(CNC(c2c(Cl)nsc2Cl)=O)C1)=O 14624,C(C1CCC(C)CC1)=C(C)C(=O)NCCC1CC(NC(c2oc(C)cc2C)=O)C1 14625,C(C(C(=O)N(C(COC)COC)C)NC(C1CC1F)=O)SC 14626,C1(CNC(c2[nH]cc(C)c2)=O)C2CC1N(C(c1ncccc1F)=O)C2 14627,C(=O)(C1=CCC(C)CC1)N(C)CC1CCCN(C(CCc2cccc(C)c2)=O)C1 14628,c1(OC)cc(C(=O)N(CCC(C(C)C)NC(C2CC2C)=O)C)c2c(c1)CCCC2 14629,c1(CCC(=O)NCCN(C(=O)CSCc2ncccn2)CC)ccc(Cl)cc1 14630,C(C)(CO)(CCF)NC(C(=O)N(CCCC(C)C)CCO)=O 14631,Cc1c(C(N2CCCCC(NC(=O)Cc3ccns3)C2)=O)[nH]c2c1C(=O)CCC2 14632,C1(C)(C(=O)NC(C)CC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)CCC(C)(C)CC1 14633,N1(C(c2ccccc2)=O)CCC2(CCN(C(=O)NC(c3cccc(F)c3)=O)CC2)C1 14634,C#CC1(C(=O)N(C(CCO)C(F)F)C)CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 14635,CC1=C(C(=O)N2CCCC2C(N2CC(C(C)C)C2)=O)SCCO1 14636,N1(C(CCC(=C)Cl)=O)CC2(CCN(C(=O)Cn3ccc(C)n3)CC2)CC1C 14637,C(c1ccc(C2OCCO2)o1)=CC(=O)N(C)CCNC(C1CC(O)(C(F)F)C1)=O 14638,c1(CC(=O)NC2CN(C(C(C)(F)OC)=O)CC2n2ccnn2)ccn2cncc2c1 14639,CC1=C(CC(=O)OCc2cc(C)ccc2OC(F)F)c2ccccc2C1 14640,C(=O)(CCCC(C)(C)C)NC1C(C)C1C=CC(N1CCNC(=O)C1CCO)=O 14641,CC1OCC2(CCN(C(CCC3OCCO3)C(=O)NC)C2)O1 14642,C(=O)(CC(C)(C)C(=O)NCC1C2CN(C(=O)C(CSC)OC)CC12)OC 14643,N1(C(COC(C)(C)CNC(=O)CCC2CCCC2)=O)CCOC(C#N)C1 14644,C1(NC(=O)CC2(CO)CC2)CC2CCC(C1F)N2C(=O)CCCc1ccccc1 14645,CC(C)(C)CC(C(=O)NCC1CCCNC1=O)NC(=O)C1=COCCC1 14646,c1(NC2CC(NC(c3n[nH]c(C)c3C)=O)C2)nccc(C(F)(F)F)c1[N+](=O)[O-] 14647,C(=O)(CCCC#CC)NCC(CC=C)NC(=O)Cn1cc(CN(C)C)nn1 14648,N1(C(c2nnc(CC)o2)=O)CC(CNC(=O)Cc2ccsc2C)CC1(C)C 14649,Cc1cc(C(N2CCOC(CNC(C3(C#N)CC3(C)C)=O)C2)=O)nn1C 14650,C(=O)(CC(F)(F)C(C)(F)F)NC(C1CCN(C(N)=O)CC1)C 14651,N1(C(C(CC(C)(C)C)(C)C)=O)CCc2sccc2C1CNC(C1CC=CCC1)=O 14652,c1(-n2c(C(C)(CCC#N)N3CC(NCCC)C3)nnn2)ccc2c(c1)OCO2 14653,C(CCN=c1[nH]ccc(=NC2CC3(C2)CC3(F)F)[nH]1)N(CCN(CCN(C)C)C)C 14654,C(c1ccc(OC)cn1)=CC(=O)NC1(CO)CCN(C(C2(OCC)CCC2)=O)C1 14655,N1(C(C(C(C)C)NC(C)=O)=O)CCC(C)C(NC(c2snc(O)c2Cl)=O)C1 14656,CCC(CCCO)N=c1cc(F)nc(C2(C)CC2)[nH]1 14657,CC(O)(CC(=O)N1CCCCC1CNC(c1cc(Br)cs1)=O)C(F)(F)F 14658,C1(CNC(c2ccc(CO)o2)=O)CN(C(=O)CN2CCCCC2)C2CC12 14659,c1(C(N2C(C)(C(=O)Nc3ncc(Br)cc3I)CCC2)=O)cc(F)ccc1Br 14660,S(=O)(=O)(c1ccc(C)c(C(=O)NC(CNC(=O)Cc2cnn(C)c2)CO)c1)NC 14661,c1(NC2c3nnnn32)ccc(NCC)cc1.C1(CCC)(COC)CCC1 14662,N1(C(C2C(=O)NCC2)=O)CC2CN(C(=O)C=CC(F)(F)F)CC(F)(F)C2C1 14663,c1(C(N2CCC(NC(C(C)N3CCC3)=O)C23CC3)=O)cn2ccnc2cn1 14664,Cc1cc(N2CCN(C)C(C)CC2)ncc1S(=O)(=O)N1CCOCCC12CCC2 14665,c1(OCC)cncc(CC(=O)NCC(CO)NC(c2ncoc2CC)=O)c1 14666,N1(C(c2c(C)ccs2)=O)CCC2(NC(=O)C(c3ccc(Cl)s3)=O)CC2C1 14667,C1(CC(F)(F)F)(CN2CCC(NC(=O)CCC3CCCCO3)C2)CCNC1=O 14668,C#Cc1ccc(OCC(=O)NC2CCCN(C(c3cc(F)ccc3C)=O)CC2)cc1 14669,CC(C)C(F)C(=O)NC1CCC(CCNC(=O)CCCc2ccsc2)C1 14670,C(=O)(C(O)CCCOC(=O)CCc1ccc(Nc2cscn2)nc1)OCC 14671,C(CC(=O)NCC1CC1Cl)(C(F)F)NC(C1(Cl)C(C(C)=O)C1)=O 14672,C1(NC(C(CO)NC(C2CN(C)C(=O)CC2)=O)=O)CCc2ccccc2C1 14673,C1(S(N)(=O)=O)(C(=O)NC2CC(CNC(C(C)SC3CCCO3)=O)C2)CCCC1 14674,N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(c3csc(O)n3)=O)C2)C1 14675,N1(C(c2c(C)nc(CNC(C3CCO3)=O)o2)=O)CCN(C)CC1CCO 14676,N1(C(c2ncccn2)C(=O)NCCCSCC)CCC(O)CC1c1ccccc1 14677,C#CCC(C)(C(=O)Nc1cc(CO)ccc1C)NC(c1ccc(OC)nc1)=O 14678,c1(C(=O)NC(CC=C)CNC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14679,c1(OC)ccc2c(C)c(C(=O)NCc3ccc(-c4ccon4)cc3)[nH]c2c1 14680,O=C(C1CCCc2scnc21)NC1CC2(C1)CN(C(C13CCCCN1CCC3)=O)C2 14681,CC(C)(C)C(CNC(C1CCN1C(C)(C)C)=O)C(=O)Nc1ccc2nc[nH]c2c1 14682,CC(CCCC(=O)NC1CC(C(C)C)C1)NC(c1ccc(Cl)cc1)=O 14683,Cc1nccc(C(=O)NC2(C(=O)NCc3ccc(Cl)cc3)CCN(C)C2)n1 14684,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14685,Cc1ccc(C)c(C(=O)NC(C)C(C)NC(c2ncccc2C)=O)c1 14686,N1(C(C(=O)NCCOC)C(C2CCC2)OC)CCCC(C2CC2)CC1 14687,Cc1ccc(C(N2CCC(O)(C(F)F)CC2)C(=O)NC2CC2)c(F)c1F 14688,Cc1ccc(NC(=O)CN(C)C)cc1C.C1(O)(C(F)(F)F)CNC(=O)NNC1=O 14689,C=CCC(C)(CC)C(=O)NCC1(O)CCCN(C(c2csc(CC)n2)=O)C1 14690,c1(NC)nc(N2CCC(c3ccc(C(CF)OC)cc3)CC2)nc2c1ncn2C 14691,c1(CCc2n(CCOC)nc(-c3ccc(Cl)s3)n2)cccc(C#CC2CC2)c1 14692,CC(C(=O)NCC1CC(NC(c2cc(CCCO)on2)=O)C1)C(C)(C)C 14693,C1(NCC(C)(C)OCC(=O)N(C(C(C)C)C)C)COC(=O)N1C 14694,CSC1=C(C(=O)NCC2CCCCN(C(=O)C#CC3(C(F)(F)F)CC3)C2)CCCC1 14695,c1(CC(=O)NC2CC(NC(=O)CCn3ccnn3)CC2O)c(O)ncnc1O 14696,c1(C(N2CCC(NC(C3C(C(N)=O)C3)=O)C2)=O)cccc2nscc12 14697,N1(C(C(C(C)C)OCC)=O)CCN(C(=O)CCC2CCC2)CCC1C 14698,N1(C(COC)=O)CCOC2CCN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14699,C(=O)(CCC(=O)NC1(C(=O)NC2CCN(C(C)=O)C2)CC(CO)C1)OC 14700,c1(C(=O)NC)ccc(CN2CCCC2C2CCCN2C(C2CC(C)(O)C2)=O)cc1 14701,CCCCN=C(NCC1CCOC1)NCC1CC2CCC2C1 14702,c1(COCC(N2C(NC(COC(C)C)=O)CSCC2)=O)ccccc1C(F)F 14703,c1(C(C)NC(C2CCN(Cc3ccc(C)s3)C2)=O)ccc(F)cc1 14704,n1(CC(=O)NC2CCC2NC(=O)CC2(CO)CCCCC2)nc(O)ccc1=O 14705,c1(C(=O)NCC2N(C(C(N3C(=O)CCC3=O)CC)=O)CC2)cn(C)c(C)cc1=O 14706,N1(C(c2c(CC)c(C)sc2)=O)CCN(C(=O)C(C)(C)CC)CC1CS(C)(=O)=O 14707,C1(CC#C)(C(N2CCCC2C2(NC(c3ncoc3C)=O)CC2)=O)CCCCO1 14708,N1(C(CN(C(CC)C)C(C)=O)=O)CCCC(C)(C(N2CCC(n3ccnn3)C2)=O)C1 14709,C1(C(=O)NCCN(CCC)C(C2(F)CCOC2)=O)C2CCC1(C)C2(C)C 14710,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14711,CC1=C(C(=O)NCC(CNC(=O)C(C)(C)C2CCOCC2)OC)C(=O)OC1(C)C 14712,C1(C(N2CCOCC(CO)C2)=O)CCCCN1N=O 14713,C1(C(=O)NCc2cc(NC(CNC(CN(C)C)=O)=O)ncc2)C2C3CCC(C3)C12 14714,N1(C(C(c2cccnc2)OC)=O)CC(NC(=O)CC(C)CF)C2(CCOCC2)C1 14715,C1(F)(CNC(C2(CC)CCC2)=O)CCCN(C(c2ccon2)=O)CC1 14716,C(CC(C)(C)C(F)(F)F)NC(=O)NC1(CC(=O)O)CN(C(c2ccccc2)C)C1 14717,CON(CCC(=O)NCc1ncc(CO)o1)C(=O)C(C)(C)c1ccno1 14718,CCCCCC(=O)NC(C1(O)CCCCC1)CNC(c1ccc(Br)cn1)=O 14719,O=C1CC(=O)NC(C(=O)NCc2cc(C(=O)NCC3CC3(Cl)Cl)n[nH]2)C1 14720,C1(NC(c2ccn(C)n2)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)CC1O 14721,Cc1ccc(F)cc1CC(=O)NC1CC(C)N(C(c2cc(C(F)F)nn2C)=O)C1 14722,C1(C(=O)NC(CNC(c2cnc(C)o2)=O)(C)Cn2cccn2)C(C)(C)C1(F)F 14723,N1(C(c2cccc3[nH]ncc23)C(=O)NC2CC(CC)C2)CCC2CCC(C1)N2C 14724,N1(C(C2(OC)CCCCCC2)=O)CCC2(CCN(Cc3nc(SC)cc(O)n3)C2)C1 14725,C1(C(N(C(CNC(COCC=C)=O)C2CC2)C)=O)CCCC(C)(C)C1 14726,C(CCN=c1cccc(S(=O)(=O)NC2COc3cc(F)ccc32)[nH]1)(C(C)C)OCC 14727,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14728,N1(CC(=O)NC(CNC(CC2N(C(C)=O)CCC2)=O)C(C)C)CCN(C)C(=O)C1 14729,N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(=O)C(F)C2CCOC2)C12CCCC2 14730,C1(C(=O)NC(=O)CC2(O)CCCC2)CC(F)CN1Cc1cccc(F)c1 14731,C1(NC(CC2(CNC(C(CC)(C)O)=O)CC2)=O)CS(=O)(=O)CCO1 14732,C1(C(=O)NC(c2nnc(C)s2)C)CN(C(=O)CC2(C)CCCCC2)CC1F 14733,c1(CN=c2scc(CC(=O)NC3CNCCC3(F)F)[nH]2)cc(F)c(F)c(F)c1 14734,C1(S(C)(=O)=O)(C(=O)OC(c2nc(-c3ccccc3)no2)C)CCCC1 14735,C12(NCCN)CC(C#N)(C1)C2.C1(C(C(=O)CC2CCCO2)=O)CCCCC1 14736,c1(OCC#C)ncccc1C(=O)NC12CC1CN(C(c1ccn(C(F)F)n1)=O)C2 14737,C1(C(N(c2oc(O)nc2C)CC)=O)CCCCN1C(=O)CCCC1CCCC1 14738,CC1CCN(S(=O)(=O)CC(=O)NCC(C2CC2)NC(C2(C)CCCO2)=O)CC1 14739,C(C)(CNC(c1nc[nH]c1C(C)(C)C)=O)(CNC(=O)C(C)=C(C)C)OC 14740,c1(C(C)(C)NC(c2c(C)ncs2)=O)cccc(CNC(=O)CC2(C)CC2)c1 14741,N1(C(c2c(CC)csc2)=O)CCC(C)C(N(C)C(c2csc(N(C)C)n2)=O)C1 14742,C(=O)(C(C)CNC(C1CC1(C)C)=O)N1CC(CSC)C1 14743,c1(NC2(C)CCN(C(C(C(C)(C)C)NC(C)=O)=O)C2)nc(C)c([N+](=O)[O-])cc1Cl 14744,N1(C(C(C(C)(C)C)C2CC2)=O)CC23CCCCC2(C1)CN(C(=O)C(=O)N(C)C)C3 14745,C1(CNC(CC=C)=O)CC2(CCOCC2)CN1C(c1cc2cc(Br)sc2[nH]1)=O 14746,C(N=c1[nH]c(=N)[nH]c(=NC2COCC2n2ccnc2)[nH]1)c1cccc(C)c1 14747,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14748,N1(C(C(CC)NC(C)=O)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1F)CCO2 14749,C1(CC(=O)Nc2n(CCC)ccc2)CN(C(=O)COC(C)=O)CC(C)(C)O1 14750,N1(C(CCCN(CCC)CCC)=O)CC(CNC(=O)CCC(C)(C)F)CCC1C 14751,C1(C(=O)NC2CC(c3ccccc3)(NC(C=CC=CC)=O)C2)C2CCCOC12 14752,C(=O)(C1=CC2(CCN(C(c3csc(=N)[nH]3)=O)C2)C1)N(C)CCC1CCOCC1 14753,c1(NC(C23CC(NC(CC(C)(C)C(F)F)=O)(C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] 14754,C(=O)(C(CCC(N)=O)n1cc(CC)nn1)OC(=N)O.C(CCC(C)CO)NCC 14755,c1(CC)nn(C)c(CC)c1C(=O)NC1CCCCC1NC(C1CC(O)C1)=O 14756,C1(NC(CC2(C=C)CC2)=O)CN(C(c2cn(CC)nn2)=O)CCC1F 14757,c1(OC)ccc(C(N2CC(CCNC(C3CCSC3)=O)C2)=O)c(OC(F)F)c1 14758,c1(C(=O)NC2CCC(NC(C(CC=C)(C)C)=O)C2)cccc2nccn12 14759,Cc1cc(NC(=O)C(F)CC2CN(C(=O)CC(C)n3cccc3)C2)sn1 14760,Cc1c(C(N2CC(NC(C3CCCO3)=O)CC2C)=O)sc2ccccc12 14761,c1(C(CNC(=O)C(N2CCC(CO)C2)=O)OC)cccc(Br)c1C 14762,c1(NC)cnncc1C(=O)NCC(c1ccc(Cl)cc1)NC(c1cncs1)=O 14763,C1(CC(=O)NC23CC2CN(C(=O)CCCN(C)C)C3)(OC)CCCCC1 14764,C(c1cccc(Cl)c1)=C(C)C(=O)NCCC1CC(NC(C2(C)CCN(C)C2)=O)C1 14765,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14766,CC1CCC(C)(C)N1C(c1cnc(CNC(C2CC23CCCC3)=O)nc1)=O 14767,C1(C#N)(C(N(CCC(C)NC(c2ccc(F)cn2)=O)C)=O)CC12CCCC2 14768,Cc1ncn(C)c1NC(C1CCN1C(C1CC(F)(F)C1)=O)=O 14769,N1(C(C(CCC)C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14770,CC1(C)CC=C(c2cc(C(=O)N=c3[nH]nc4[nH]ccn34)cc3[nH]ncc23)CC1 14771,CCC(CC)C(C)C(=O)NCCCC(=O)N(C1CC(O)C1(C)C)C 14772,c1(OCCC(=O)NCCC2CCN(C(CN(CCOC)C)=O)C2)ccccc1C 14773,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14774,C=C(C)C1OCCC1C(=O)N(CCCNC(=O)COCCSC)C 14775,c1(C(=O)NCCN(C(C2CSCCS2)=O)CC)cnn(CCOC)c1C 14776,CC(C)(CCC(=O)N1CC(C(=O)NCC2CCC(CO)O2)C2(CC2)C1)[N+](=O)[O-] 14777,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)C(c2cnn(C)c2)C)C1 14778,c1(C(=O)NCC2CC(NC(CCC(C)(F)F)=O)C2)ccc2c(c1)CCCS2 14779,C(=O)(CC1OCCc2sccc21)N1CC(C)(NC(c2cc3sc(Cl)cc3[nH]2)=O)C1 14780,CC1OCCC1CNC(=O)C=Cc1ccsc1.C12CCC(C1)NC(=O)CC2 14781,C1(NC(=O)CC2CSCCS2)CCCC(CNC(c2ccoc2)=O)C1 14782,c1(C2N(C(c3cc(C4CC4)no3)C(=O)NCCOC)CCC2)cccc(Cl)c1 14783,Cc1cnc(NCCCCC2CC2C)c(S(=O)(=O)NCCCCS(C)=O)c1 14784,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14785,c1(OC)ccc(C(N2CCN(C(=O)C=CC(C)(C)C)C(CCOC)C2)=O)nc1Cl 14786,C1(C(N2C(C3CCN(C(CN(C)C)=O)C3)CCC2)=O)CC2(CC2)CN1C 14787,c1(OC)cnc2ccccc2c1C(N1CC(C)C(C(=O)O)C(C)C1)=O 14788,CC1(C(=O)NC2CCN(CC(=O)NCCC#N)C2)Cc2ccccc2C1 14789,c1(NC(C2CCN(C(c3ncccn3)=O)CC2O)=O)ccc(I)c(F)c1 14790,O(C1CCCc2cc(Cl)ccc21)CCCOC(C1(C#N)CCOCC1)=O 14791,C1(C(N2CC(O)(C(C(N3CC(OCC(C)C)C3)=O)F)C2)=O)CCOC(=O)CC1 14792,CC#CCC(C(=O)NCCC(O)CCO)NC(=O)CN(C)CC 14793,CCC(C)C(O)C(=O)N(C)CCSC(CC)(CO)CO 14794,CCC(C)C(=O)C(=O)NC(C(=O)NCCCN1CCCCC1=O)C1CC1 14795,N1(C(C(N2CCOCC2)C)=O)CC23CCCC2(C1)CN(C(C1CC(F)(F)C1)=O)C3 14796,c1(C2(CC(N3CC(C)C(F)C3)=O)CC2)ncnc2c1c(Br)cn2C 14797,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14798,C1(CNC(C(C)=C2CCCC2)=O)CCCCN(C(=O)CC(C)N(C)C)C1 14799,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)C2CC2)=O)C(O)C1 14800,C1(C(=O)NC2C3CN(C(c4c(C)n(C)nn4)=O)C2C3)CC12CCS(=O)(=O)CC2 14801,Cc1cccc(CCNC(c2c[nH]nc2CCNC(=O)Cn2cc(C)cn2)=O)n1 14802,c1(C(=O)NC(C2CCCO2)C(=O)NC(C#C)(C)C2CCOC2)c[nH]nc1[N+](=O)[O-] 14803,Cc1ccc(C(N2CCC(C(=O)NCc3ccoc3)CC2)=O)cc1C#N 14804,c1(C(c2n(CC(C)C)nnn2)NCC2CCCOC2)cc(Br)ncc1F 14805,N1(C(C2(C)CC2)=O)CCCC(O)(C)C1.C(=O)(C)N(C)OCC.C(=O)(C1CC1)N 14806,C(N=c1[nH]c(N2CCCN3CCCC3C2)nc2c1SCC2)C1CCC(C)(C)CO1 14807,C1(NC(CCC(C)O)=O)CC2CCCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 14808,c1(C(N2CCC(CCCCCCC(=O)N)CC2)=O)ccc2nncn2c1.CC(=O)N 14809,C1(C(=O)NC2(CO)CN(c3cc(C(C)=O)ncn3)C2)CCC(C)(C)CC1 14810,c1(C2(C(N(C)CCNC(=O)CCC3CC3(C)C)=O)CC2)cccnc1Cl 14811,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCO2)CCC1 14812,c1(C(N(CC(C)NC(c2c(CC)nn(C)c2)=O)C)=O)ccc(COC)c(F)c1 14813,CC(CC(N)=O)C(=O)NCC1(C)CN(C(=O)CC2CCCCCCC2)CCO1 14814,C#CC1(NC(=O)N(CC(C)(F)C(C)(C)F)CCOC)CCC(C)CC1 14815,c1(CC(=O)N(CC(=O)NCCC(C)C2CC2)CC)ccoc1C 14816,C(=O)(C(C(C)C)S)N(CCC)CCNC(c1csc(C(=O)NC)n1)=O.C(C)(C)O 14817,C1(C(C)C)CCN(C(c2ccc(I)cc2)C(=O)NCC(F)F)C1C 14818,Cc1ccc(-c2nc(C(=O)N(CC(O)CNC(=O)Cc3cnsc3)C)cs2)cn1 14819,C(=O)(C(COC1CCN(C(n2cc(Oc3cccnc3)cn2)=O)C1)CC(C)C)NC 14820,C1(NC(c2ncc(C)c(Cl)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC1N=[N+]=[N-] 14821,Cc1ccc(NS(C)(=O)=O)c(C(N2CCC(CNC(C3CC3(C)C)=O)C2)=O)c1 14822,N1(C(CC(C)SC)=O)CC=C(CNC(=O)C(c2ccc(F)cc2)(C)F)CC1 14823,C1(NC(COCCNC(C2C(C)OCCO2)=O)=O)CC2(C1)CC(O)C2 14824,N1(C(C2(SC)CCC2)=O)CCC(C(N2CC(C(C)O)C2)=O)CC1(C)C 14825,c1(C(=O)NC2C3N(C(C(C(C)C)F)=O)C(CC3)C2)ccc2c(c1)C(=O)OC2(C)C 14826,S1(=O)(=O)CCC(=O)NC2(CCCCC2)N1.CC(F)(F)C(=O)NCCOC1CCOC1 14827,C(=O)(CC1OCc2ncccc21)N1C2CCN(C(CCNS(C)(=O)=O)=O)C2CCC1 14828,N1(C(c2c(C)nn(C)c2)=O)C(C(=O)NOCCF)CCC12CC2 14829,N1(C(C(C2CCOCC2)NC(C2=NOC(C)C2)=O)=O)CCc2nocc2C1 14830,C1(NC(CCC)=O)CC(NC(c2oc(CC)cc2C)=O)C12CCOCC2 14831,CC1CC(CNC(=O)C(C)c2ncco2)CN1C(=O)Cc1cccc(Br)c1 14832,N1(C(c2cc(C)c(N)cc2Cl)=O)C2CCC1C(C)C(NC(=O)C(F)=CC1CC1)C2 14833,c1(C(N(CC(CC)NC(=O)Cn2cc(CO)nn2)C)=O)cccc2nn(C)nc12 14834,c1(C(=O)NC2C(CNC(C(CCC)OC)=O)CC2)cc(F)c(C)cc1N 14835,Cc1c(NC(=O)CC2CC(C)N(C(=O)Cc3cncnc3)C2)cccc1Cl 14836,C1(C(=O)NCC2N(C(CC(CC)(C)C)=O)CCCC2)CCOC2(CCCCC2)C1 14837,C1(CC(=O)NCC(C)(O)CNC(=O)C(O)c2ccsc2)CCC2(CCCC2)CC1 14838,C(=O)(C#CC1CCC1)NC1(C)CC(NC(=O)CCC2CC2(Cl)Cl)C1 14839,C(=O)(C1=C(Cl)CCCC1)NC(C)(CNC(c1cnn(CCN(C)C)c1)=O)C1CC1 14840,N1(C(C2(C#C)CC2)=O)CCOC2(CCN(C(c3cn(C)nn3)=O)C2)C1 14841,c1(C(=O)NC2CC(CCNC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14842,C(=O)(CC(O)CC(C)C)NC1CCCC(NC(c2n(CC=C)ccc2)=O)C1 14843,C(C(F)C(=O)NC(=O)CC1(C)CC1)SCCOC.C(C)(C)(C)OC(NC)=O 14844,C1(C(=O)NCC2(CCNC(CNC(CCC)=O)=O)CC2)CCCN2CCCCC12 14845,CCCCC(C(=O)NCC(O)CN(C)C(c1ccnc(O)c1F)=O)N(C)C 14846,c1(C(N(C2CCN(C)CC2)C)=O)ccc2[nH]nc(-c3cccc4ccsc34)c2c1 14847,Cc1ccc(=N)[nH]c1C(N1CCN(C(c2ccc(C(C)C)o2)=O)CC1C)=O 14848,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(C3SCCS3)=O)C2)C1 14849,N1(C(c2n(CCC)ncc2)=O)CCC(C(C)NC(=O)CCC#N)CC1 14850,N1(C(C(C)Br)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14851,CC(CC(=O)NC1C=CCN(C(c2sccc2CN(C)C)=O)C1)CC(F)(F)F 14852,C1(NC(c2ccc(CNC(CSCCC)=O)s2)=O)CCC(C(N)=O)CC1 14853,C1(c2nnnn2C2CCCC2)(C(=O)NSCC=C=C)CCOC(C(F)(F)F)C1 14854,CC1CC(CCNC(c2cncnc2)=O)CCN1C(=O)CSCC(F)F 14855,c1(CCC)cc(C(=O)N(C2CCCN(C(C3(F)CCCC3)=O)C2)CC)c(C)o1 14856,c1(OC)cc(C(=O)NC2(CNC(=O)C3=C(C)OCC3)CC2)c(Cl)cn1 14857,c1(C(N2CC=CC(C(=O)NC(CCCC)C)C2)=O)cc(C#N)oc1C 14858,N1(C(c2c(C)cncn2)=O)CCCC2C1CCN2C(c1ccc(Cl)cn1)=O 14859,CC(C)(F)CC(=O)N1CCC(CCCCCNC(=O)CCc2csc(=N)[nH]2)CC1 14860,Cc1ccc(C(=O)NCC(C)NC(c2csc(C3CCCO3)n2)=O)nc1 14861,S(=O)(=O)(c1cccc(F)c1)CCNC(C)CNC(=O)CCc1cnc[nH]1 14862,C(=O)(C(C(C)C)NC(=O)COCc1nc[nH]n1)NCC(C#C)CC 14863,C1(CNC(c2ccc(Cl)s2)=O)CN(C(=O)CSC(F)F)CC12CCC2 14864,N1(CCCC(=O)OCCS(C)(=O)=O)CCc2c(F)cccc21 14865,c1(SC)ncc(CN(c2nccc(N(C)CC3CCCS3)n2)C)cn1 14866,N1(C(C(C)NS(CC)(=O)=O)=O)CCCCC(CNC(C2(C)CC2)=O)C1 14867,C(C(CNC(C1(C(F)(F)F)CC(O)C1)=O)C(F)(F)F)NC(C(n1c(C)ncc1)C)=O 14868,N1(C(c2c(C)nco2)=O)CCCCC1CCNC(=O)C(C)OC1CCOC1 14869,c1(CCCC(=O)N(C2CCN(C(C3CN(C(N)=O)C3)=O)C2)CCO)ccc(O)c(F)c1 14870,C(CCCC(CO)NC(=O)CCc1cncc(F)c1)NC(c1c[nH]c(=NC)o1)=O 14871,C1(NC(CCc2cncc(OC)c2)=O)CN(C(c2sccc2F)=O)C(C)(C)C1 14872,Cc1ccc([N+](=O)[O-])c(C(N2CC3CC2CN3C(c2cnn(C(F)F)c2)=O)=O)c1 14873,c1(SC)nc(Cl)c(NC(C2CC23CCN(Cc2cc(F)c(Br)cc2F)C3)=O)c(Cl)n1 14874,C1(CC(N2C(CNC(c3cnc(C)s3)=O)C=CC2)=O)CC2(CCC2)CO1 14875,Cn1ncc(NC(c2conc2C2CCC2)=O)c1-c1cn(C(C)(C)C)nn1 14876,CN1CC2CCN(C(C3(CCNC(c4c[nH]ccc4=O)=O)CCC3)=O)C2C1 14877,c1(CCC(=O)NC(CCc2c[nH]c(=N)[nH]2)=O)ccccc1.C(C)(C)CC1CC1 14878,c1(C(C)C)cccc(C(=O)NCC(C)N(C)C(c2cnc(C3CCC3)s2)=O)c1 14879,C1(C(C)C)CCC(c2nc(-c3ccc(C(F)F)cc3)nn2C2CCSC2)CC1 14880,c1(C(=O)NC2CC(C(=O)NC(CC)CO)OCC2)c(F)ccc(OC)c1N 14881,c1(N(CCCOC)C(C)C)nc(C)nc2ccccc12 14882,C1(CC(=O)NCC2(NC(CSCC(C)C)=O)CC2)CC2(CCC2)CO1 14883,Cc1ccc2ncc(C(=O)NCC3(NC(=O)CN4CCC(CO)CC4)CC3)n2c1 14884,c1(N2CCN(Cc3cccc(C(=O)NCC)c3)CC2)cc(C#N)ccc1N 14885,CCCCCC(O)CNC1(c2nnnn2CC(F)F)CCC(C)C1 14886,C#Cc1ccc(C2CCN(C3CCN(C(c4cn(C5CC5)cn4)=O)C3)CC2)cc1 14887,C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(C2CC(F)(CF)C2)=O)CC1 14888,C(=O)(CCc1ccco1)N(CC(=O)NCCSC)C 14889,c1(C(=O)NCCCCN(C(CC(C)C(F)F)=O)C)nsc2c(Cl)cccc12 14890,c1(C(=O)NC2C(NC(C(C)OCCCC)=O)CC2)cnc2c(ccn2C)c1 14891,C1(C(N2CCC(OC)(CNC(C)=O)CC2)=O)CC2(CCNC2=O)C1 14892,CCCC(CCC)C(=O)NCC1CCCN(C(C2CCC(OC(F)F)CC2)=O)C1 14893,c1(CC(CNC2(CCC)CCC2)C)ccccc1C(F)(F)F 14894,c1(C(=O)NC2(C)CCN(C(CCC(C)OC)=O)CC2)cccc2ccoc12 14895,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14896,O=C1C=COC2(CCN(C(c3ccc(-c4cn[nH]c4)cc3)=O)CC2)C1 14897,C1(N(C(c2c(CCC)n(CC)nn2)=O)C)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 14898,C=CCCCC(=O)N1CCCC1(C(C)C)Cc1cn(C2CCCC2O)nn1 14899,c1(OC)ccc(Cl)c(CN2CCCCC2CNC(=O)C(C)(C)C2CC2)c1 14900,Cc1nc(C)c(C(N2CC(NC(c3scnc3C(C)C)=O)C(O)C2)=O)s1 14901,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(C2CCC=CCC2)=O)C1 14902,c1(C(=O)OC)cncc(C(=O)NC2CN(C(C3(F)CC3)=O)CC2C)c1 14903,N1(CC)CCOCC1CC(=O)NCC1(F)CC(NC(c2cccc(CO)n2)=O)C1 14904,CN1CCN(C)CC(C(N2CC(C3CN(C(C4CCCN4N=O)=O)C3)C2)=O)C1 14905,C1(CSC)CCN(C(c2ccc(C(=O)NOCC(C)C)n2C)=O)CC1 14906,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CCO.C12C=CC(C1)C(=O)N2 14907,N1(C(CC2C(NC(CCC=C)=O)CCC2)=O)CC(C2=NOC(C)C2)C1 14908,N1(C(CCNC(=O)OC)=O)CCC2(CCC(NC(=O)CCCF)C2)C1 14909,C1(CC(=O)N(C(C)CCNC(C2(C(F)(F)F)CCC2)=O)C)OCCC1C 14910,c1(N2C(CCOC)CCC2)cc(C)nc(CO)n1.n12cc(nn1)C(=O)NC2(C)C 14911,c1(C(=O)NC)cccc(C(=O)NCC(O)CNC(=O)CC2CC(=O)NC2=O)n1 14912,C1(C(N(C)CCN(C(=O)CCCN2CCCC2)C)=O)CCc2nncn2C1 14913,C(CCC(N)=O)(C(=O)NC1CCN(C(=O)COCC(C)(C)C)CC1O)NC(C)=O 14914,N1(C(c2c(CC(C)C)n(C)nc2)=O)CCOC(C)(CNC(=O)CC2CCOC2)C1 14915,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCn2cc(Br)cn2)CC2(CC2)C1 14916,N1(C(c2ccc(C#C)cc2)=O)CC(NC(=O)CSc2nncn2C)CC2(CC2)C1 14917,c1(N2CCC(C(c3cn(C(C)C(=O)N(C)C)nn3)(C)C)C2)ccnc2ccc(F)cc12 14918,c1(CN(C=O)CCc2ccccc2I)scc2c1OCCO2 14919,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(c1cn(CCO)nn1)=O 14920,C(CCN(C)C(c1nn[nH]c1Cl)=O)(C(C)C)NC(C(C)SCc1ccccc1)=O 14921,N1(C(c2cccc(OC)n2)=O)CC(C(=O)NC(c2ccc(F)cc2)C)CC(F)C1 14922,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 14923,c1(CNC(C(CC)N(C)C(c2ccnnc2O)=O)=O)cc(O)ccc1F 14924,C12(CNC(C(c3ccccc3)C)=O)CC(CN1C(c1nocc1C(C)(C)C)=O)C2 14925,c1(OC)ccc(F)c(C2CCN2C(=O)C(F)OC)c1NC(C1CCCCO1)=O 14926,C=CC1(C(=O)N(C)CC2CCOC2)CCN(C(c2ccsn2)=O)C1 14927,c1(C(=O)NC2CN(C(CC3CC(=O)C3)=O)CC23CC3)cncc2c(Cl)cccc12 14928,Cn1cnnc1SCC(=O)NC(Cn1cncn1)C(=O)NC1CCOC1=O 14929,Cc1cnc(-c2noc(CC3(O)CCCC3)n2)nc1 14930,c1(OC(C)C)ccc(NC(c2cc(N3OCCNC3=O)ccc2F)=O)cc1F 14931,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 14932,Cc1cc(F)ccc1NC(=O)C(=O)NCc1cccc(C(N)=O)c1 14933,C1(CN2C(c3cn(C(C)CS(N)(=O)=O)nn3)CCC2)CN(C)CCN1C 14934,C(=O)(N=c1sccn1Cc1ccccc1)c1cccc(C2CC(CO)C2)c1 14935,Cc1cccc2cc(C(N3CCC4(C3)CN(C(=O)C3CC3)CCO4)=O)nn12 14936,C1(NC(CC(=O)NCC#C)=O)CN(C(=O)C(C)(C)c2ccccc2)CC12CC2 14937,C1(CC=C)(NC(=O)COCCC)CCN(C(c2cnc(SCCC)s2)=O)C1 14938,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 14939,C1(NC(C(C)=C2CCCC2)=O)CCC(N(C(=O)C(c2cnn(C)c2)O)C)CC1 14940,C(=O)(C1=NNC(=O)CC1)N1CC(C)(C)C(NC(=O)Cc2ccc(F)cn2)C1 14941,c1(OC)cc2c(cc1S(=O)(=O)N1CCCC(CC3CCCC3)CC1)OCC2 14942,C1(C)(CNC(C2(COCC)CC2)=O)CCN(C(=O)Cc2ccon2)CC1 14943,C=CC1CN(C(=O)CC(C)NC(=O)C(C)OC)CC1O 14944,c1(CC)n[nH]cc1C(=O)NC1CC(O)C1CC(=O)NCCSS(C)(=O)=O 14945,N1(C(Cc2n(C)c(S)nn2)=O)CC(NC(C23CC2CNC3=O)=O)C2(CCC2)C1 14946,c1(NC(COCCOC)=O)cc(C)ccc1CNC(=O)C(C(C)C)n1cnnc1 14947,C1(NC(C2CN(C(C)C)C(=O)C2)=O)CC2(CCN(C(C3CC3(C)C(C)C)=O)C2)C1 14948,N1(C(C(C)CO)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 14949,C1(C)(C(=O)NC(C)CNC(c2cn(C3CC3)nn2)=O)CC(c2ccccc2)=NO1 14950,N1(C(C(C2CCN(C(=O)NCC=O)C2)F)=O)CCCc2ccccc2CC1 14951,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 14952,c12ccccc1OCCCNC2.c1(COC)cc(C2(C)CC2)on1 14953,c1(C(N(CC(C)NC(c2cc(=O)n(C)o2)=O)CC)=O)csc2ccccc12 14954,c1(C(=O)NCCCNC23CC2CCC3(F)F)c[nH]ccc1=Nc1ccccc1 14955,N1(C(Cc2n(C(C)C)cnn2)=O)CC2(CC2)CC1CNC(c1nccn1C)=O 14956,c1(C(N(CCCCCNC(CCC(=C)Br)=O)C)=O)cc2c[nH]nc2s1 14957,C1(CNC(C(C)n2cccc2)=O)CC(F)(F)CN1C(c1cc(Cl)cnn1)=O 14958,c1(C(C)C)nc(C(=O)NCC(O)CCNC(=O)Cc2ccc(Cl)s2)co1 14959,Cc1nn(Cc2ccccc2)cc1C#N.c12cc(cs1)NC(=O)OCC2 14960,N1(C2CCN(C(C(CSC)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 14961,c1(C(N2C(C)CCC(CNC(c3cnn[nH]3)=O)C2)=O)cc2c(o1)CCCC2 14962,c1(C(=O)NCC=CCNC(C(C)NS(C)(=O)=O)=O)sc(F)cc1Cl 14963,S(=O)(=O)(CCC(=O)NCCNC(=O)C(F)(F)c1cscn1)NC 14964,CC1(C)CC(C)(C(=O)NOCC2CCOC2COC)CN1C(c1cnc(=N)[nH]c1)=O 14965,C(=O)(C(C)CC(F)(F)F)NCCC1N(C(c2n(CC)ncc2)=O)CC(OC)C1 14966,C(C(C)CN=c1c(C#N)c[nH]c2cccc(C)c12)NC(c1cc(C)nn1C)=O 14967,c1(C(=O)NCC23CC(NC(CC4CCC(C)CO4)=O)(C2)C3)coc2ccccc12 14968,CN1CCCC(C(=O)Oc2cccs2)C1=O.c12csc(n1)OC2=O 14969,c1(OC)cc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)COC(F)F)c(F)c1 14970,C(CO)(C(=O)NC1CC12CCC2)NC(=O)CN1CCC1CF 14971,c1(CCN2CCOCC2)ccc(C(N2CCCC2CC(=O)OC(N)=O)=O)cc1 14972,C1(N(C(CN2C(C)CC2)=O)NC(CC(=O)N(C2CC2)C2CC2)=O)CCOC(C)(C)C1 14973,C(=O)(C1CCCc2nc[nH]c21)NC1(C)CN(C(C2CCN(C3COC3)C2)=O)C1 14974,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)Cc3cc[nH]c3)CC2)cnc2cc[nH]c2c1 14975,C1(CNC(c2ccc3ncccn23)=O)CCCC(F)(F)CC1 14976,CC#CCCC(=O)NC1CN(C(c2cnc(N3CCOCC3)s2)=O)CC1C 14977,c1(CCC)nc(C)c(C(=O)NCC2CCN(C(C3(C)COC(=O)C3)=O)CC2)o1 14978,c1(C(=O)NC(C)C(C)(C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 14979,C1(NC(C(C(C)C)O)=O)CN(C(=O)C=CCF)CCN1C 14980,C1(NC(c2c(CC)cno2)=O)CC2CCC(C1)N2C(=O)C(C)Sc1ccccc1 14981,c1(C(=O)NCC23CC(CN2C(C2C=CCCC2)=O)C3)cnc2sccn2c1=O 14982,c1(C(=O)NC2C(NC(c3cncc(C)c3)=O)CC2)ccc2c(c1)SCC(=O)N2 14983,c1(N(C(=O)Nc2ccccn2)C(N2CC3CC3C2)C2CC2)ccccc1 14984,C1(C(N(CCC)CCNC(=O)C(CC)(CC)CO)=O)Cc2cccc(C)c2O1 14985,C(N=c1[nH]cnc(Cl)c1CO)C1C(C)CN(C(c2cc(C(F)(F)F)on2)=O)CC1 14986,CCCC(C)(C)C(=O)N1CC(CNC(=O)CCc2nnc(C)n2C)C(O)C1 14987,N1(C(c2nn(C)c(Cl)c2Cl)=O)CCN(C(C2CCNC2=O)=O)CC12CC2 14988,C(C)(C)(CCCCC(=O)N1CCN(C(C2(F)C3CCCC23)=O)C2(CCC2)C1)OC 14989,c1(CC)nc2c(C)csc2c(=NCC2CCCN2C(=O)C(C)NS(=O)(=O)CC)[nH]1 14990,CCS(=O)(=O)CCn1cc(C(=O)N(C)CCNC(=O)C(F)(F)F)cn1 14991,N1(CC)CCCC(N(C(CCC(=O)NC(=O)CC23COC(C)(C2)C3)=O)CC)CC1 14992,C1(N(C)C(C2CC(C)(C)O2)=O)CCCCN(C(c2cc[nH]c2C2CCCC2)=O)C1 14993,C1(NCCN2CC(NC(CCNC(C(C)(C)C)=O)=O)C2)C(Cl)(Cl)C12CC2 14994,N1(C(C(CC)NC(=O)OC)=O)CC(F)CC1CNC(C1CC2CC2C1)=O 14995,CC(CS(C)(=O)=O)C(=O)N1CCCCC(NC(c2ccc3ncnn3n2)=O)C1 14996,C1(NC(COCC=C)=O)COC2(CCCN(C(c3ccc(N(C)C)cc3)=O)C2)C1 14997,C1(C(N(C2CCN(CC)C2)C)=O)CCN(C(=O)Cc2ccn(C)c2)C1(C)C 14998,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC2C(C(=O)Nc3c(F)cncc3F)(C2)C1 14999,N=c1[nH]nc(SCC(=O)NCC2CCCN2C(c2ccnn2CCF)=O)s1 15000,C1(CNC(C(C)OCCCC)=O)CN(C(=O)CC2(O)CCOCC2)CCO1 15001,N1(C(CCSCCC)=O)CCN(CCNC(=O)C(C)C(C)O)CC1 15002,c1(CC(CNC(=O)CSC(F)F)N(C)C(C2CCCO2)=O)ccccc1 15003,N1(C(c2nc(CNC(C3(C#N)CCCO3)=O)oc2)=O)CCN2CCC1C2 15004,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(NC(CSCC(C)C)=O)C2)C1 15005,C1(NC(C2CN(C(=O)NC)C2)=O)(CO)CCCCN(C(=O)Cc2ccno2)C1 15006,CC1CCC2CN1C(=O)c1cccnc1CNC2=O.n1(CCN(C)C)cncn1 15007,c1(C(=O)NC2CCCC2NC(C2CCCCC2O)=O)cnc2nccn2c1 15008,CC1CC(NC(c2ncc[nH]c2=O)=O)CN(C(c2ccn(CC#N)n2)=O)C1 15009,N1(C(CC=CCC)=O)CC2(CC2)CC1CNC(=O)C(C#N)CCC 15010,c1(C(C(=O)NCC=C)N(C(CF)CF)C2CC2)cncc(Br)c1C 15011,N1(C(C2(c3cccc(C#C)c3)CC2)=O)CC2CC(NC(=O)CCC3CC3)CC1C2 15012,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15013,C1(NC(=O)C(c2cccc(F)c2)O)CCCN(C(c2ccc(F)s2)=O)C1 15014,N1(C(c2c(CC)noc2)=O)CC2(CNC(c3ccn(C)n3)=O)CC(F)(C1)C2 15015,c1(OC)cccc2c(N3CC(CO)(NC(=O)Cc4cnsc4)C3)ncnc12 15016,C1(C(N(C(C)C)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15017,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=C(C)C(F)F)C2 15018,N1(CCOC)CCC1C(=O)NOCC(O)CO.C1C(=O)N1 15019,C(C1=CCN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)CC1)NC(C1CC1F)=O 15020,CCCCCC(F)C(=O)NCC1CCCCC1C(=O)NCc1ccc(OC)cc1 15021,C1(CC=C)(C(=O)NCc2csc(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15022,CC1(C)COCC(C(=O)NC(c2ccccc2)CNC(C2(CO)CC2)=O)O1 15023,c1(C(=O)OCC)cc(NC(=O)COC(c2csc(C3CC3)n2)=O)cn1C 15024,N1(N2C(C)CS(=O)CC2)C2CC1CN(C(=O)Cc1ccccc1O)C2 15025,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15026,C=C=Cn1ccccc1=NC(=O)C1CC12CN(c1cc(F)cc(F)c1)C2 15027,CS(=O)(=O)c1ccccc1C(=O)NCC1(O)CCN(C(=O)Cn2ccnn2)C1 15028,N1(C(C(C)OC)=O)CC(F)(F)CC1CCNC(=O)C(C)NC(c1ccccc1)=O 15029,C1(C)(NC(C2(COC)C=CCN2C(=O)CN(C)C(=O)OC)=O)C(C)(C)C1(C)C 15030,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15031,c1(SC)ccccc1C(=O)NC1CC1NC(=O)C(C)(C)CO 15032,C1(NC(=O)CCF)CCN(C(c2ccnn2CC(F)(F)F)=O)CC1CO 15033,c12cc3ccc(nc3s1)C(=O)NN1CCCCCN2CC1.C1(CC)(CC2CC2)CC1 15034,C(=O)(C(C)(C)CC(C)(C)C)N(C1CCN(C(c2ccnnc2C)=O)C1)CC 15035,C1(NC(c2[nH]nc(N(C)C)n2)=O)CC2CC2N1C(=O)CNC(=O)Nc1ccsc1 15036,c1(C(=O)NCCOCCCN(C)C(c2cnc(O)o2)=O)cc(Cl)ns1 15037,c12ccccc1CNC(=O)C2.CCS(=O)(=O)Cc1cn(CC23CCCC2C3)nn1 15038,Cc1cc(-c2ccc(N(C)C)c(-c3nccn3CCO)c2)c(O)cc1F 15039,C1(C(=O)Oc2ccc(CO)cn2)CCC2(CC1)CN(C(=O)OC(C)(C)C)CCO2 15040,c1(C(=O)NC2CCC(NC(C3CC3CF)=O)C2)cncc(C2CC2)c1 15041,c1(N2CCCC(C)C2)nc2cc[nH]c2c(=NCC(C)(C)C(C)C)[nH]1 15042,C1(C(=O)OCC)CCC(C(F)F)(NC(=O)CC2CCNCC2)CC1 15043,c1(NCC2CC(C)CC2)nc2ccccc2nc1NCc1ccc(S(C)=O)cc1 15044,C1(CNC(Cc2ccc(C)o2)=O)CCN(C2CN(C(=O)CC(C)(C)C)C2)CC1 15045,C#Cc1cnn(C)c1C(=O)NCCC1CSCCN1C(C1CCCN(C)C1)=O 15046,CCC(C(=O)OCC(F)(F)F)N1CCCC1=O.C1(=O)CO1 15047,CC(O)C(C(=O)NC(C(C)(C)O)C1CC1)NC(c1ccc(O)cc1)=O 15048,c1(-c2n(CCOC)nc(-c3ccc(OCC)nc3)n2)cc(Cl)c2cnn(C)c2n1 15049,c1(C(N(CC(C)NC(=O)CC2COCCO2)CCO)=O)cnn(C)c1 15050,C1(CC(=O)NCCC2(N(C)C)CC2)CC(CNC(C(C)C)=O)C1(C)C 15051,N1(C(C2(C)C(C)C2)=O)CCC(C(c2ccccc2)NC(C2CCC23CCC3)=O)CC1 15052,C1(CF)C2CNCC12.C1(C)(CF)CC1 15053,C1(C(C)OC)(CNC(C2CCCC2)=O)CN(OC)C1.C1(C2CCC2)(C(=O)OC)CC1 15054,CC1(C)CN(C(c2csc(S)n2)=O)C(CNC(=O)Cc2ncc(Cl)s2)CO1 15055,c1(SCC(=O)NC2CC(NC(C3COCCC3(F)F)=O)C2)ccc(F)c(F)c1 15056,S(=O)(=O)(c1cccnc1NCC1CCCS(=O)(=O)C1)NCCOC(C)C 15057,Cc1ncccc1CC(N1CCC(NC(=O)COCCCN=[N+]=[N-])C1)=O 15058,C(=O)(C(c1ccccc1Cl)=CC(C)C)N1CCC(C(C)NC(CCN(C)CC)=O)C1 15059,N1(CC2CCCN(CC)C2)CCN(CC(=O)NCC(C)Cc2ccccn2)CC1 15060,CC(CCc1ccccc1)C(=O)N1CC(F)CC1C 15061,N1(C(C(CCC)CC)=O)CC(C2CCCN(C(c3cnc4cccnn34)=O)C2)C1 15062,C1(NC(C(C2CC2)OCC)=O)CCC(F)(CNC(c2cc(CO)[nH]n2)=O)C1.C1CC1 15063,C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 15064,CCCCC(C(=O)NCC1COCC(C)O1)NC(c1ccc(F)cn1)=O 15065,CC1CN(C(C2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)=O)CCS1=O 15066,N1(C(CCCC#C)=O)CCN(C(=O)CCc2cccc(O)c2)C2CC12 15067,c1(C(N(CCOC)CCNC(C2CCC2C)=O)=O)csc(Br)n1 15068,C(=O)(CCCN=C(NCc1ccc(O)cc1Cl)NCC(C)C)OCC 15069,c1(C(C)C)ncc(C(=O)NCCc2cc(C(=O)NCCCO)no2)cn1 15070,CC1CN(C(=O)CC)CC(CCNC(c2ccc(-c3ccon3)cc2)=O)O1 15071,C=CCCCC(=O)NC1(C(N)=O)CN(C(=O)CN(c2ccccc2)C)C1 15072,c12ccc(cc1)C(=O)NC(C)C2C.C1(C)(NC(CC)=O)CC(C(=O)OC)C1 15073,c1(NC2CCCC(NC(=O)OC(C)(C)C)C2)cc(O)c2ccccc2n1 15074,C1(N(C(C)C)C(C2CCCCC2)=O)CCC(C(C2OCCC2C)=O)CC1 15075,c1(C(N2CC(C(N)=O)(CNC(CC(CC)C)=O)C2)=O)ncc2[nH]ncc2n1 15076,C(C)(C)(C(C(=O)Nc1cccc(OC)c1Br)C(C)C)OC(CC(=O)OCC)=O 15077,C1(NC(C(CCCOC)C)=O)CCCCN(C(=O)Cc2cccc(C)c2)CC1 15078,Cc1cccc(NC(C2CN(C(c3ccc(CC(=O)O)cc3)=O)CCO2)=O)c1O 15079,c1(C(N2C(C)(C(=O)Nc3ccc(I)c(Cl)n3)CC2)=O)cccc2[nH]ncc12 15080,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)CC1 15081,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(=O)Cc3ccn(C)n3)C2C1 15082,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCC2(CC1)CC2NC(=O)CSCC(N)=O 15083,N1(C(C2(C#N)CC2)=O)CC2(CC2)CC1CNC(C12COC(CF)(C1)C2)=O 15084,N1(C(CCC=CC(C)C)=O)CCC(=CCNC(C2CC=CCN2C)=O)CC1 15085,C1(OC)CN(C(=O)C(C)=CC2CC2)CC1NC(c1ccc(F)s1)=O 15086,c1(CCCC(=O)NCCN(C)C(c2ccc(F)c(N)c2)=O)c[nH]c2ccccc12 15087,N1(C(c2c(C)cc(Cc3ccncc3)cc2C)=O)CC2CC(C1)c1ccccc12 15088,Cc1cc(C(=O)NC2CCN(C(C3CC3F)=O)CC2F)c(C)n1-c1cnn(C)c1 15089,C1(C(N2CC(C(C)NC(C(C)OC3CCCCCC3)=O)C2)=O)CCCCS1(=O)=O 15090,C12(NC(=O)CCCc3cccnc3)CC(C1)N(C(c1cscc1F)=O)C2 15091,C1(CNC(CN(C)CCO)=O)CC2COCC2N1C(C1(C(F)F)CCOCC1)=O 15092,C(C)(C(=O)NNC(=O)C(C)O)n1cc(OCn2c(C)ncc2)nn1 15093,C(CCC(CO)NC(c1coc(C2CCC2)n1)=O)NC(=O)CCCF 15094,c1(OC)cc(OC)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15095,Cc1cccc(O)c1C(=O)NCC1CC(NC(=O)Cc2cn(C3CC3)cn2)C1 15096,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15097,c1(OCC)cnc(CNCC2(c3cccnc3CC)CC2)cn1 15098,C1(C(N(CC(C)C(=O)NCC(C)(O)C(F)F)C)=O)CC2(CC(=O)C2)C1 15099,C(C(C(=O)NC(c1csc(C)c1)C(=O)O)OC)OC 15100,C1(C(N(CC(=O)NC2CC2)C)=O)CC12CC(NC(=O)CCOCC(F)F)C2 15101,CCCCCS(=O)(=O)NC(CCCCSC)c1nnnn1CCCOC 15102,Cc1c(NC(=O)N(C)CCOC(F)(F)F)cnn1C1CC(N)C1 15103,N(C1C(=O)Nc2cccc(Cl)c21)C(c1ccc(-c2ccc(C)cn2)cc1)=O 15104,N1(C(CC2(COC)CC2)=O)CC2CC2C1CNC(c1cncc(C(F)(F)F)n1)=O 15105,c1(CCCNC(Cn2cc(CCS(C)(=O)=O)nn2)=O)ccc(Cl)c(C(F)(F)F)c1 15106,N1(C(N2CCCC(F)(C(=O)OC)C2)=O)C(C)C2CCCCC2C1 15107,CC1(C(N2CC3C(NC(=O)C=CC4CCOCC4)C3C2)=O)CCCCNC1=O 15108,c1(OC)ccc(Cl)c(C)c1C(N1CCC2(NC(c3cc(C4CC4)[nH]n3)=O)CC2C1)=O 15109,CCCC(O)CC(=O)N(CCN(C)C(c1c(F)ccnc1F)=O)C(C)C 15110,c1(C(N2CCC(NC(CC(CC)SC)=O)(CF)C2)=O)ncc(F)c(OC)n1 15111,c1(C(N2C3CN(C(c4cc(SCC)ncc4)=O)CC32)=O)ccc2ccccc2c1 15112,c1(C(=O)NCC2(C)CCN(C(CSCCCC)=O)CC2)ccc(F)cc1[N+](=O)[O-] 15113,Cc1ccc(-c2cc(C(N3CC(NC(C45CC(F)C4C5)=O)C3)=O)c(C)o2)cc1 15114,c1(SC(C(N2CCC(NCC3(C=C)CCC3)C2)=O)CC)ccc(C#N)cc1.C(C)=O 15115,C(=O)(C=CS(C)=O)N1CCC(N(C(CNC2CCC(=O)N2C)=O)C(C)=O)C1 15116,CC1(C)CCC(C(=O)NCC#CC(=O)NCc2c[nH]nc2C2CC2)CO1 15117,c1(C(=O)NCC(=O)NC2(C)CC(C(=O)NCC(=O)NC)C2)cccc(F)c1 15118,N1(C(C2CCC2)=O)CCC(CNC(CC(C)Cn2cccn2)=O)(CN(C)C)CC1 15119,C1(n2cc(CCC(C)(C)C)nn2)CC2CCC(C1)S2.C1(C)CCOCC1 15120,Nc1cc(C(N2CCCC3(NC(C4CC=CC4)=O)CC3C2)=O)cc(F)c1O 15121,C1(c2ccccc2)(C(=O)NCC(C)NC(c2cc[nH]c2)=O)CCCC1 15122,C1(NC(c2cc(C(C)C)n(C)n2)=O)CCC(C)N(C(c2ccc(Cl)cc2O)=O)C1 15123,c1(CCNC(C2CSCCN2C(c2cocn2)=O)=O)ccccc1F 15124,c1(C(N2CC(C(C)(C)O)(CNC(C3C(C)(CC)C3)=O)C2)=O)ccc2cc[nH]c2c1 15125,C1(C(=O)NC2(CNC(C3CCS(=O)(=O)N3)=O)CCCC2)CC2COCC(C1)C2 15126,C1(CC(N2CC(O)(CNC(=O)C(=O)NCC3CC3)C2)=O)CCCCCO1 15127,CC(c1cnn(C)c1)=CC(=O)NC1CC(O)CN(C(=O)CSc2cn[nH]c2)C1 15128,C#CCCC(O)C(=O)N1CCN(C(=O)COCCCC)CC1C(F)F 15129,c1(C(=O)NCC2(NC(C(CC)NC(N)=O)=O)CCCC2)cnn(C)c1Br 15130,C1(CCNC(C(C)SC)=O)CCCN(C(C23CCN(CC2)C3)=O)C1 15131,C1(CNC(C=C(C)Cl)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 15132,N1(C(COCCC#C)=O)CC(C2CCCCN(C(c3cc(Cl)ccc3F)=O)C2)C1 15133,N1(C(C(CC)=CCCC)=O)C(C(=O)NCC2CCN(C(C)C)C2)CC2CC12 15134,N1(C(C)=O)CCN(C(C(=O)NCCCF)C2CCC2)C(CCO)C1 15135,CC1(CNC(C2OCCC2C(F)F)=O)CCN(C(c2csnn2)=O)C1 15136,C(=O)(NNC(=O)C(C)(O)COC(=O)Nc1ccccc1)c1c(Cl)ccc(OC)c1 15137,C(CCN=c1ncc(O)c[nH]1)N(C)C(C1CC1CCSc1ccccc1)=O 15138,Cn1cccc1C(=O)NC1(CCNC(C2CCN(c3ccncc3)C2)=O)CCC1 15139,C(C)(CC(C)NC(C1CC1OC(C)=O)=O)NC(C1C(CCC)C1)=O.C(C)(C)(C)O 15140,N1(C(C2CC(NC(C)=O)C2)=O)CCC(F)(C(N2CCNC(=O)C2)=O)CC1 15141,C1(C)(C(=O)NCC2(CN(C)C(C3(O)CCCC3)=O)CC2)CCCCNC1=O 15142,CCCCC(CN=c1[nH]cc(CC(C)C)c(O)n1)NC(c1nn(C(C)C)cc1C)=O 15143,C=CC(C)(C)C(=O)NCCC(C1CCN(C(=O)C(F)C2CC(OC)C2)CC1)O 15144,N1(CC)CCC(CNC(=O)NC(CC2CCCO2)C(=O)OC)C1 15145,C1(CC)CCOC1C(=O)NCCOC1CN(C(c2nnn(C)n2)=O)C1 15146,C1(NC(C(CC)(C)C)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15147,c1(NCCP(OCC)(C)=O)ncc(S(=O)(=O)N)cc1Cl.C(S(C)(=O)=O)C1(CCC)CC1 15148,C1(C(C(=O)N(CC)Cc2ccncc2)F)CCN(C(c2sccc2Cl)=O)C1 15149,C(=O)(C(CO)C(C)(C)C)NC(CCNC(CNC(C)=O)=O)C(C)C 15150,C1(CC=C)(NC(C2CC2C(N)=O)=O)CCN(C(=O)C(c2cccnc2)C)CC1 15151,c1(C(=O)NC2CC(CCNC(C3N(CCC)CCC3)=O)C2)c(N)cc(F)cc1Cl 15152,C1(NC(C2(OCC)CCOCC2)=O)Cc2ccccc2N1.C12(O)CN(C1)C(=O)C2 15153,C(=O)(C#CC1CCOCC1)N(C)CCNC(=O)COC(C)(C)C(F)(F)F 15154,CC(C)(CCC(=O)N1CC(O)CC1NCCn1cc(C2CC2)nn1)c1ccon1 15155,c1(SC)nc2ccccc2[nH]1.N12CCN(C3CC13)C(=O)Cc1cnccc1C2=O 15156,c1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CC=C2)ccc(Br)c2cn[nH]c12 15157,c1(CNC2CCC(NC(CC3N(C(C)=O)CCCC3)=O)C2)ccc(F)nc1C 15158,N1(C(C(CCCC)C)=O)CCC2(CCCCN(C(=O)C(C3CCOCC3)C)C2)C1 15159,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15160,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15161,c1(C2(C(=O)OC)CCC2)cccc(C(=O)Nc2cccc(-c3ccncc3)c2)c1 15162,c1(C(=O)NC2CCCC(NC(Cn3c(C)ccn3)=O)CC2)cnn2c1CC(F)(F)C2 15163,c1(CC(C)(C)C)nc(-c2cc(-c3cccnc3)no2)n(C2CCS(=O)(=O)C2)n1 15164,C1(Nc2c(CC)ocn2)=CC=NC=CC=C1S(=O)(=O)N1CCS(=O)(=O)C(C)(C)C1 15165,C1(C(N2CC(NC(C(C)CS(C)=O)=O)C2)=O)CCC2(CC1)NC(=O)NC2=O 15166,CCCC(C)(C)C(=O)NC1CCN(C(c2cnn(C(C)C)c2)=O)CC1 15167,Cc1cc(C(=O)N(C(C)CCNC(c2cc(C(N)=O)no2)=O)C)n(C(F)F)n1 15168,C(=O)(C(O)CC(C)(C)C)NC(C(C)C)(C)CNC(=O)C1=CC(C)(C)C1 15169,c1(CC)cccnc1C(=O)NC1CN(C(c2ncoc2C(C)(C)C)=O)C1 15170,N1(C(c2[nH]ccc2C2CC2)=O)CCC2(CCCN(NC(=O)C=CCF)C2)CC1 15171,C1(O)(C(C)NC(C2CNC(=O)N2)=O)CN(C(=O)CCc2nc(O)n[nH]2)C1 15172,C(=O)(C1=NOC2(CCC2)C1)NCC(CO)(CO)NC(C(c1ccc(F)cc1)C)=O 15173,N1(C(C2CC(=C)N2)=O)CC2(CCN(Cc3ccc(OC)c(OC)c3C)CC2)C1 15174,Cc1cnc(C(N2CCCC2(C)CNC(=O)CC2CCS(=O)(=O)CC2)=O)c(C)c1 15175,Cc1cc(C)c(NC(C2CCCN2C(c2cnc(Cl)cc2I)=O)=O)c(Br)n1 15176,Nc1nc(C(N2CCC(NC(=O)Cn3cnnn3)C2C2CC2)=O)ccc1Br 15177,C(=O)(CC(C)CC(C)C)N1C2CN(c3c(F)cnc(OC)n3)C(C2)C1 15178,C(=O)(C#CC1(C)CCCO1)N1CC(CNC(CC2C(C)CCC2)=O)OCCC1 15179,c1(CNC(C2CCC(CNC(C3C(C(C)(F)F)C3)=O)O2)=O)ccc(F)nc1 15180,c1(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC(F)C2)cccc2c1CCC2 15181,C(=O)(CCCCCN=[N+]=[N-])NC.Cn1ccnc1C1CC1 15182,C12(CC(C)NC(c3cnn(CCNC(=O)C(N)=O)c3)=O)CCC(CC1)C2 15183,c1(CNC(C(=O)NC(C(C)(C)C)Cc2ccccc2)=O)cnc2[nH]ccc2c1 15184,Cc1ccc2oc(C(=O)NC3CC4CCC(C3)N4Cc3ccc(C#N)s3)cc2n1 15185,c1(OC)ccc(-n2cc(C(=O)N(C)CN3CCCC(SC)C3)nn2)c(OC)c1 15186,C1(NC(C(C)SC)=O)CC2CCCC(C1)N2C(=O)CCc1nnc(C2CC2)o1 15187,CC1(C)CN(C(c2cnc(Br)s2)C(=O)NC2CC(F)(F)C2)CCS1=O 15188,C(=O)(C1=NOC(CNC(C2CCCN(C(=O)CC(C)(C)O)C2)=O)C1)OC 15189,C1(O)(C(=O)OC)CN(C(CC2C=CCC2)C(=O)NC2CCOCC2)CC1O 15190,N1(CCC)C(=O)NC(c2ccc(O)cc2CC)C2=C1C1(CCSC1)NC2=O 15191,C1(O)(C(C)CNC(c2cnn(CC(F)F)c2)=O)CCN(C(C2CCCS2)=O)C1 15192,CCC(CNC(=O)C(CC)N(C)C)(CC)C(=O)N(CC(N1CCCCC1)=O)C 15193,N1(C(CC2(C)N(C(C3CCCN(C)C3)=O)CC2)=O)CC23CCC2(COC3)C1 15194,C1(N(C(CCSC)=O)C)CCCCC1N(C(=O)C(O)COCc1ccccc1)C 15195,CC1(C)CC(NC(C2CC(C)(C)OC2(C)C)=O)CN(C(c2c[nH]ccc2=O)=O)C1 15196,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15197,CCCC(CNC(=O)CC1CCC(C)(C)O1)C(=O)NCC1OCCC1(C)C 15198,c1(C(N2CCC(C(CNC(C3C4CCCC34)=O)F)CC2)=O)cccc2cncn12 15199,C1(CC)(NC(c2csc(C(=O)NC)c2)=O)CCCN(C(c2sccc2Cl)=O)C1 15200,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15201,CC1CC=CCC1C(N1CCCC(CC(=O)NC2CCNC(=O)C2)C1)=O 15202,C1(C(CC(=O)OC)NC(=O)CSc2n[nH]c(C)n2)CCC(F)(F)CC1 15203,c1(C(N2CC(CNC(=O)CCNC(N)=O)CC(C)C2)=O)n[nH]c2cc(Cl)ccc12 15204,C(=O)(CC(C)(O)C(F)(F)F)NCCC1CC(OC)CN1C(=O)CSCC(N)=O 15205,C(=O)(C(S(C)(=O)=O)C1CC1)N1CC(N(C(COC(CC)(C)C)=O)C2CC2)C(C)C1 15206,C1(C2CN(C(C3C(Cl)(Cl)C34CC4)=O)C2)(NC(=O)OC(C)(C)C)CC1.C1CCO1 15207,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15208,C1(CC(=O)NCC(CC)(C)NC(=O)CC(C)COC)CCC=CCC1 15209,CC1CN(CCC(=O)NC2CCC2)C(c2ccccc2)CO1 15210,N(C(=NCCc1ccc(F)cc1)N1CCN2C(=O)OCCC2C1)CC(=C)F 15211,C(CCOCCO)(C(=O)NC1(C2CC2)CC1)NC(c1cnc(C)s1)=O 15212,C1(CC)C(C(=O)Nc2cccc(N(C)C)c2)CCCN1C(c1cn[nH]c1)=O 15213,O=C1CN(CC(N2CCCC2CNC(c2cc(C3CCC3)on2)=O)=O)C(=O)N1 15214,N1(C(CN2CCN(C)CC2)=O)CC2(CC(NC(=O)C(O)CF)CO2)C1 15215,C12(C(=O)NC34CC(NC(c5cnn(CCF)c5)=O)(C3)C4)CC(CCF)(C1)C2 15216,C1(CNC(Cc2c(C)nn(C)c2)=O)CN(c2nncs2)CCN1C 15217,c1(N(CC(c2cccc(I)c2)O)C)ccc(C#N)nn1 15218,c1(C(=O)Nc2nn[nH]n2)ccc2nc(-c3cnn(C4CCOC4)c3)cn2c1 15219,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15220,c1(C(N2CCCC(C)(C(N3CC(O)(C(C)C)C3)=O)C2)=O)cnc2cc(Cl)ccn12 15221,CCC(C(=O)N1CC(O)CC1(C)C(N1CCCC2(C1)N=N2)=O)C(C)C 15222,c1(OC)c(Br)ccc(C(=O)NCc2c(C)n[nH]c2C)c1F.N12CCC1(C)C2=O 15223,C(=O)(CCCN=[N+]=[N-])NCCCN(C(C1N(CCC)C(=O)CC1)=O)CCO 15224,N1(C(C(COC)COC)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)NC1)=O)C3 15225,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC(O)C3)C2)=O)cnn1C 15226,c1(CC(=O)N(C(C)CNC(=O)CC2OCCOC2(C)C)C)coc2ccccc12 15227,C1(C(=O)NCC(C2(O)CN(C(c3c(C)onc3)=O)C2)(C)C)CC2CCC1C2 15228,CC(CNC(=O)COCCN(C)C)(CO)NC(c1cnoc1C1CCC1)=O 15229,c1(CCC=C)ccc(CC(=O)NC2CCCC2CCNC(=O)CC=C)cc1 15230,C(C1=NOC2CN(C(c3csc(C4CCC4)n3)=O)CC12)NC(c1cnsn1)=O 15231,c12ccc(Cl)cc1c1cn(nn1)c1ccsc1c(=O)[nH]2.Cc1ccc(CO)cn1 15232,S(=O)(=O)(c1nc(NC2CCCCC2CO)ccc1Br)N1CC2CN(C)CC2C1 15233,C1(CNC(c2c(C)nn(C)c2C)=O)CN(C(=O)Cc2csnn2)C2CCN1C2 15234,c1(C(=O)NCC2(OC)CN(C(=O)Cc3cncc(C)c3)C2)n[nH]c2c1CC1CC21 15235,N1(C(CCC2(C)CN(C(C(C)OCC#C)=O)C2)=O)CCCC12CCOC2=O 15236,CC1(NC(=O)Nc2ccccc2-c2ncn[nH]2)CCCN(C(=O)Cn2ncnn2)C1 15237,c1(C(N(CC(C)NC(=O)C(C)(C)N2CCCCC2)CC)=O)c[nH]cc(C)c1=O 15238,C(=O)(CS(=O)(=O)C1CCCC1)N1CCCC(NC(C2C3CCCCCC23)=O)C1 15239,c1(C(C)C)cccc(CC(=O)NC(C2CCCCN2C(C2(C)CC=CC2)=O)C)c1 15240,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15241,c1(NCCCCNC(c2cc(CCC)[nH]n2)=O)ccc(S(C)(=O)=O)cn1 15242,c1(C(N2CC3N(C(c4ccc(OC)o4)=O)C(CC3)C2)=O)cn2cccc(Cl)c2n1 15243,c1(C(=O)NC(CC)(C)CNC(C2(C)CCC(=O)CC2)=O)ccnc2c1cnn2C 15244,C1(NC(COCCC)=O)CCN(C(=O)CC2CCCN(C(C)=O)C2)CC1F 15245,C(=O)(C1(Cl)C(=O)N(C)c2ccccc21)N1CCC(COCCCOC)CC1 15246,C12CN(C(=O)C3CC3)CC1C(=O)N2.C1(NC(C2C=CCC2)=O)CCCO1 15247,c1(NC(C2(NC(C3CCC(N=[N+]=[N-])C3)=O)CC2)=O)cc[nH]c2nccc1-2 15248,C1(NC(C2C(C)OCCC2)=O)CCSC12CN(C(C1CCCCC1N=[N+]=[N-])=O)C2 15249,C1(C(C)NC(=O)N(C2(O)CCOC2)C2CC2)CCN(C(=O)OC(C)(C)C)C1 15250,c1(OC)cc(O)ncc1C(N1CC(C)(NC(=O)CC2CCN(C)C2=O)C1)=O 15251,C1(NC(C2C(C(=O)OC)C2)=O)CC2(C1)CC(C(=O)N(C)CC1CC1)C2 15252,C1(CCC)CN(C(c2cn(C)nc2C2CCC2)=O)CCN1C(=O)CCF 15253,c1(SC)ncc(C(N2CC(CNC(c3cnn(C)c3S(N)(=O)=O)=O)C2)=O)c(O)n1 15254,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(C(=O)NOCC1CCCO1)C2)=O 15255,C1(COC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)CC(=O)N(C)C 15256,c1(SC)cc(C)ccc1C(=O)NC(CNC(=O)C(C)(O)C(C)C)C1CC1 15257,C1(C(N(CCNC(c2cc[nH]c2)=O)CC)=O)Cc2ccccc2O1 15258,N1(C(CC(COC)(C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCS(C)(=O)=O)C3 15259,N1(C(C)=O)CCCCC1c1ccc[nH]1.N1(C)CCNC1=O 15260,C1(NC(C(CC)N(C)C)=O)CN(C(C2CCC(OC)CC2)=O)C2(CCCC2)C1 15261,S(=O)(=O)(C1CCOC1)NC1CCCN(CC(c2ccccc2)=O)C1 15262,c1(C(N2CCC(C)CC2CNC(C2CCCC2(C)C)=O)=O)ncn2ccccc12 15263,N(C(=NCCC(C)(O)C(F)(F)F)NCc1cc(C)ccc1F)C(CC)C 15264,Cc1ccc(S)cc1Cl.C1(C(=O)CC)CCN(C(=O)c2nocc2C)O1 15265,C(=O)(CS(=O)(=O)CC)N1CC(CCCCNC(c2cn(CC=C)nc2)=O)C1 15266,N1(C(CN(CCOC)C)=O)C(CNC(c2nc(Cl)ccc2F)=O)CC2COCC12 15267,c1(C2(CN)CC2)cc(NC(c2cncc(C(F)(F)F)n2)=O)cc(Br)c1 15268,c1(N2CCCC(CC)C2)nc(=Nc2cccnc2C)[nH]c2c1ncn2C 15269,C=C(C(=O)N1CCC(CC(=O)Nc2c(-c3ccccc3)noc2C)C1)C(F)(F)F 15270,N1(C(CSc2nc(C)[nH]n2)=O)CCN(C(=O)CC(O)C2CCCC2)C2CCC12 15271,N1(C(=O)Cc2ccc(F)cn2)CCCCCC1CO.N12CCC1C(=O)NCC2=O 15272,c1(C(N2C(C(C)NC(C3CC(SC)C3)=O)CCC2)=O)cc(N)ccc1Cl 15273,c1(C(=O)NCC(C)CNC(C2CC23CC(O)C3)=O)cnc(-c2ccccn2)nc1 15274,C#CCCN=C(NCc1ccnc(Cl)c1)N1CCC(C2CC2)CC1 15275,C#CCCCC(=O)N1CC(NC(c2sc(Br)cc2Cl)=O)C(C)C1 15276,N1(C(C=C2CCC(C)C2)=O)CCCC(CCNC(=O)CCc2cccs2)CC1 15277,N1(C(C(CCC)NC(N)=O)=O)CCC(F)(F)C(CNC(c2cc(CC)sn2)=O)C1 15278,c1(C(=O)N)ccncc1O.C12(O)CN(C1)C(=O)c1cn(nn1)C2.C1(C)CCCCC1 15279,C(=O)(C(C)(COC)CC)NCC(=C)CCNC(=O)Cc1csc(Br)n1 15280,c1(OC)ccc(NC(c2sccc2Cl)=O)c(OC(F)F)c1 15281,Cc1cccn2c(C(N3CCCC(NC(c4cccn4C)=O)CCC3)=O)cnc12 15282,C(=O)(CC(C)(C)CN(C)C)NC(C(C)NC(c1csc(C)c1C)=O)C 15283,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C)C(CNC(c2n[nH]c(C)c2C)=O)C1 15284,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15285,c1(C(N2CC3C(CNC(CS(=O)(=O)N(CC)CC)=O)C3C2)=O)cn2nc(C)sc2n1 15286,c1(NC)ccc(N2CCC(C(c3ccccc3Cl)NC(C)=O)CC2)nn1 15287,C1(C(N2CC(C(C)NC(c3c(SC)n(C)nc3)=O)C2)=O)CN(C)C(=O)CCO1 15288,C1(C(=O)NCC2N(C(c3cc(C#N)no3)=O)CCCC2)CC(C2CCCC2)C1 15289,C#CCC(C)(C(=O)NCC1CCCSC1)NC(=O)CCc1cncn1C 15290,C1(C)(C(=O)NCC(CNC(C(CC)C2CCC(=O)N2)=O)F)CC(C)(C)C1 15291,C(CCC(C)(C)C(=O)NC(CNC(c1cc(CC)n(C)n1)=O)C)OC(F)F 15292,N1(C(c2n(C(C)C)ccn2)=O)CC2C(CNC(=O)Cc3cn[nH]c3)C2C1 15293,c1(CC(=O)OC)ccccc1NC(C1CC1)=O.C1(C=O)CCC1C#N 15294,c1(CNC(C(c2ncn(CC)c2)N(CCCCC(C)C)C)=O)ccc(Cl)c(Cl)c1 15295,C1(CC)CN(C(=O)CC(C)(F)F)CCC1NC(c1cccc(C2CC2(F)F)c1)=O 15296,c1(C(N2CC(C)C(NC(=O)C(C)(C)CN(C)C)C2)=O)nc(Cl)ccc1F 15297,c1(CCNCCC(CN(C(C(=O)NC(C)=O)=O)C)C)cccc2ncsc12 15298,c1(CNC(c2scc(C#N)c2)=O)c(Br)sc2ccccc12 15299,n1(CC)ccc(C(=O)NCC2(C(N3CC(O)(CC(C)C)C3)=O)CC(C)(C)C2)c1C 15300,C1(CNC(C(CNC(c2ccnc(O)c2)=O)N(C)C)=O)CC2(CC2)C(=O)O1 15301,Cc1ccc2c(CC(=O)N(C)CCOCCNC(C3(C)CCCC3)=O)c[nH]c2c1 15302,N1(C(C2(C)CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)C(F)CC1CCCC1 15303,Cc1nn(C)c2ncc(C(N3CC4CCN(C(=O)C(F)C(C)(C)O)C4C3)=O)cc12 15304,n1(C(CC)C)nnnc1C(C(C)(C1CC1)OC)NC(COC(C)(C)C)C1CC1 15305,C1(C(=O)NCc2noc(C)c2C)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15306,N1(C(CCOCCC)=O)CCN(C(C2COCCC2(F)F)=O)C(C)C1 15307,N1(C(c2c(CNC(C(CC)CN(C)C)=O)ccs2)=O)CC(C)(C)C2COCC12 15308,c1(C(=O)OC)nn(C)nc1C(=O)NCC1CN(C(c2ccc(C)n2C)=O)CC1C 15309,C=CCC(C)(CNC(C1(CNC(C2CCCC2O)=O)CC1)=O)CO 15310,N1(C(CCn2cc(C(C=C)(C)O)nn2)=O)CCN(C(C)=O)CC(C)C1 15311,C1(NC(c2c(O)ccc(OC)c2)=O)C2CC3CN(C(=O)C(C)OC)C1C3C2 15312,CC1(C(N2CCC(NC(c3cccn4ccnc34)=O)C2)=O)CCCC(F)(F)C1 15313,C1(CCC(=O)NCCCN(C(C2(CO)CC=CCC2)=O)C2CC2)CCC(=O)NC1 15314,C12(C(=O)NCC(CNC(C(C)Cc3ccco3)=O)F)CC(C1)C(C(F)(F)F)O2 15315,c1(NC(=O)NC(c2nnco2)C)cn(C(F)F)c(=O)nc1O 15316,C1(NC(c2cccc([N+](=O)[O-])c2)=O)CC12CCN(Cc1cncc(Cl)c1)CC2 15317,C1(C#N)(C(N(C2CN(C(CC(C)SC)=O)C2)C)=O)CC1(C)C 15318,C#CCC(C)(CNC(C1(NC(C2CC=CCC2)=O)CCCC1)=O)CO 15319,N1(C(c2cnc(C)s2)=O)CCC(C)C(NC(C2CC(n3cnnc3)C2)=O)C1 15320,N1(C(C(CC)=CC)=O)CCC(C)C1C(=O)N(CC(F)Cl)C 15321,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15322,C1(CNC(=O)CC=C(C)C)CCOC1SCC(=O)N(CCOCCO)CC 15323,O=C(NN1C(=O)NC2(CCC2)C1=O)c1c[nH]c2c(F)cc(Cl)cc12 15324,C1(CNC(=O)CN2C(=O)CNC2=O)CC(F)(F)CN1C(C12COCC1C2(F)F)=O 15325,c1(CC(=O)N(CC(CC)NC(C2CCC(=O)NC2)=O)CC)cn2cccc(C)c2n1 15326,C(=O)(C(C(C)C)NC(=O)C=CCl)NC(CN(C(CCCOCC=C)=O)CC)C 15327,c1(OC)ccnc(NC2CC2CNC(c2ccnc(Oc3ccccc3)c2)=O)n1 15328,Nc1c(C(=O)NCCNC(=O)CSc2cnn(-c3ccccc3)c2)cccc1Cl 15329,Cc1cncc(C(=O)NCCC(C)CCNC(c2coc(C3CCC3)n2)=O)n1 15330,c1(C(=O)NCC2(N(C(C(C3CC3)SC)=O)C)CC2)ccc(Cl)o1 15331,Cn1nc(C(=O)NC(C(=O)NC2CCOC2=O)C2CC2)cc1F 15332,N1(C(CCC(=C)C)=O)CCOC2(CCN(C(c3cccc(Br)c3N)=O)C2)C1 15333,c1(C(=O)NC)nc(NC(=O)NCC2COCC2C(=O)OC)nn1C 15334,N1(C(Cc2nc(C)sc2)=O)CC(CC(=O)Nc2ccnc(C3CC3)n2)OC(C)C1 15335,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2[nH]ccc2C)=O)CC1)NC(=O)OC 15336,c1(CC(N2CC(CC(C)(C)C)C2)=O)c[nH]ccc1=O.c12cn(nn1)CC2 15337,c1(C(=O)NCC(=O)NC(CNC(C(C)OCC(C)C)=O)C)ccccc1F 15338,c1(NC2CC(NC(c3cncnc3)=O)C2)ccc2cc[nH]c2n1 15339,CC(C)(C)C(CCO)NC(=O)CCC1CCN(C(=O)C2=COCCC2)C1 15340,Cc1ccc(CCCCC(=O)N(C)CCNC(C2CCSC2)=O)cc1 15341,C1(CNC(CCCOCC)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 15342,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15343,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2O)cccc2nn[nH]c12 15344,C(=O)(CCNCCC1(SCCOC(=O)COCCOC)CCC1)NC 15345,c1(OC)cccc(OC)c1CCC(=O)NC1CCS(=O)CC1 15346,c1(C(=O)NC23CCN(C(CCCCCC)=O)CC2C3)cn(CC)c2ccccc12 15347,C1(CC(N2CC3C(c4c(OC)cccc4)(C3)C2)=O)NC(=O)CN(C)C1=O 15348,CC(C)CC(CNC(c1cnn2cnnc2c1)=O)C(=O)N(CCC#N)C 15349,c1(C(=O)NCCCC(C)NC(=O)Cc2csc(Cl)c2)ccc2cccnc2c1N 15350,C12(C=O)CC=CCN1CCC2.c1(N)cncnc1.C1(=O)CN(C2CC2)N(C)CCN1C 15351,N1(C(c2c[nH]c(=NC)o2)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15352,C1(NC(c2occc2Br)=O)C2CN(C(=O)Cc3cccc(O)c3)CC12 15353,N1(C(C(C)O)=O)CC2(CCC(CNC(C3C(=O)CC3C(F)(F)F)=O)O2)C1 15354,c1(C(N(CC(=O)NC(CN(CCCC)C)C)C)=O)cccc(C)c1N 15355,N1(C(C=CC(c2ccccc2)C)=O)CC(NC(=O)CC2(O)CCCC2)CC(C)(C)C1 15356,CCC(CC)(C(=O)N1CCC(N(C)C(c2cc(C(N)=O)co2)=O)CC1)C(C)C 15357,N1(C(COCCCC#C)=O)CCC(CNC(C2CCC23CCC3)=O)C12CCC2 15358,C1(CCOC)(C(N2CCC(CNC(=O)CCCF)C2)=O)SCCCS1 15359,Cc1nc(C(N2CCC(C3CCCCN3C(c3cn(C)nn3)=O)C2)=O)c(C)s1 15360,C12(C(=O)NCC3C(C)(C)C(NC(c4cc(Cl)no4)=O)C3)CC=CC(C1)OC2 15361,O=C1CC(CC(=O)NCC2C(OC(=O)NC3(CCc4ccccc4)CC3)C2)CN1 15362,CCCCC(CN(CCC)CCNC(c1nn(C)nc1Br)=O)CC 15363,Cc1cc2ncc(C(=O)NC(C)(CNC(=O)C(C#N)C3CC3)CC(C)C)cc2[nH]1 15364,n1(CCNC(c2n(CCCSC)nnn2)C(C)(C)OC)nc2ccccc2n1 15365,c1(CC(CC)C)nc(C2CCC2(F)F)n(-c2cccc(F)c2)n1 15366,Cc1cc(N2CC(C)N(C(C)C)C2)nc(NC(c2ccccc2C)C)n1 15367,C1(NC(C(C)(O)C2CCC2)=O)CN(C(c2cnc(C(F)(F)F)nc2)=O)CCC1F 15368,c1(NC(C2(SC)CCOC2)=O)nc(C)ccc1F 15369,CC1(C)CN(CC(=O)NC2COCC2CNC(=O)CCOC2CCCOC2)C1 15370,CS(=O)c1ccc(F)c(C(N2CCCC(CNC(=O)CC(F)(F)C(F)F)C2)=O)c1 15371,C(=O)(CCCC(=O)NCC1CC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)OC 15372,C1(C(=O)NC2C(NC(c3occ(C)c3)=O)COC2)CC2CCCC(C1)C2 15373,N1(C(CC(=C)Br)=O)CCC2(CC1)CN(C(=O)C(c1ccc(C(F)F)cc1)O)C2 15374,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15375,c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccc(Cl)s2)=O)ccnc(O)c1 15376,C(=O)(C(C)(C)C(C)(C)O)N(CC(C)C(=O)N1CCC(C(F)(F)F)C1)C 15377,Cc1ccc(CC(=O)N(CCN(C)C(c2n[nH]cc2C)=O)C(C)C)c(F)c1F 15378,c1(C(=O)NC(C)CCNC(c2cccc(C(C)(F)F)c2)=O)ccc2[nH]ccc2n1 15379,C(=O)(C1CCC(=O)c2cccn21)N1CC2(CC(NC(C(C)CC(C)(C)C)=O)C2)C1 15380,c1(CC(C)NCc2cnc(C(F)(F)F)s2)ccc(Cl)nc1 15381,c1(OC)ccc(CC(=O)Nc2ccc(-c3ccc(CC#N)nc3)cn2)cc1Cl 15382,N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(CO)C1 15383,c1(C(=O)NCC(n2cc(COCc3cccc(Cl)c3)nn2)C)ccccc1C(F)F 15384,C1(C(=O)NCCN(C(C2(OC)CCC2)=O)C)CCC2(CCC2)CO1 15385,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)C2)C)cc2n(c1)CCCC2 15386,N1(C(CC[PH](C)(=O)=O)=O)CCC2CCN(C(=O)CCc3ccsc3Cl)C2C1 15387,N1(C(C(C)CN(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)CC12CCC2 15388,C1(O)(C(C)C)CN(C(=O)CCC2(NC(=O)C(C)Cn3ccnc3)CCC2)C1 15389,c1(NCC2(OCC)CCOC2)ccnc(O)c1 15390,C1(C(=O)NC2CCC(CN(C)C(C3CCSC3)=O)CC2)CCc2nnn(C)c2C1 15391,Cc1nnc(NC2CC(CCNC(=O)C(n3ccc(C(F)(F)F)n3)C)C2)nc1C 15392,c1(C(=O)NCCOCCNC(C(C)CN(c2ccco2)C)=O)ccc(O)cn1.C=O 15393,C(CCN=C(NCC(c1ccccc1)CO)NCC1CN(C2CC2)C1)OC 15394,N1(C(c2ccc(CCCC)cc2)C(=O)NCC(=O)OC)CCC(F)(F)C(C)C1 15395,CN=c1[nH]cc(C(=O)NCc2ccnc(N3CCN(C(=O)CNC=O)CC3)c2)o1 15396,CCCCCCCCCCCCC(=O)NCC(C)N(C(=O)CC(C)n1ccnc1)C 15397,CN1CCC(O)(CNC(c2ccc(CNC(=O)C(=O)C(C)(C)C)cn2)=O)CC1 15398,Cc1cc(C(N2CCN(C(=O)C(N(C)C)N(C)C)CC2CF)=O)n2nccc2n1 15399,c1(NC(c2c(CC)c[nH]n2)=O)ccccc1CC(=O)NCC1(CCO)CC1 15400,CCCC(C(=O)NCCCN(C(c1ccn2cccc2c1)=O)CC)C(C)C 15401,c1(CC)cc(CCC(=O)N(C2CCN(C(=O)Cc3cc(C)no3)C2)CC)oc1C 15402,CC1CN(C(C)C(=O)NCC2CCCCC2)CCN1C(C1CCCCN1C)=O 15403,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)C(C2CCCCCC2)C)c1 15404,c1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)cc(C)n(C)c1 15405,C(=O)(C(CN=[N+]=[N-])NC(=O)CC1CC1)NC(c1ccccc1)C 15406,C(CCOCC)(C(C)C)N(C(C=CCC)=O)C(=O)CC1CNC(=O)O1 15407,N1(C(c2cc(CC)oc2C)=O)CC(C2CN(C(c3c[nH]nc3C3CC3)=O)C2)C1 15408,N1(C(c2ccc(CCC)[nH]2)=O)CCC(C(C)NC(c2ccccc2C)=O)CC1 15409,Cc1c(F)ccc(C(=O)NCC2CCN(C(=O)CC3CC4CC4C3)C2(C)C)c1F 15410,C(=O)(C(O)CC(F)(F)F)NC1CC(C(=O)NC2(C(N)=O)CC2)CC1O 15411,c1(C(=O)NCC2(OC)CN(C(=O)C(F)CC(C)C)C2)ccc2oc(C)nc2c1 15412,N1(C(C(CNC(c2cn(CCC)nn2)=O)OC)=O)CCC(O)C(F)C1 15413,c1(CC(=O)NC(CC=C)CNC(=O)CC2COCCO2)cc(O)nc(O)n1 15414,C#CC12CCC(C(N3C4CCCC3CN(C(=O)C(C)OCC)C4)=O)(CC1)CC2 15415,c1(OCC(=O)OC)ccc(C)cc1C(c1nnnn1C1CC1)NCCOC 15416,C1(NC(CCOc2c(CC)cccc2)=O)CC(F)CN(C(=O)C(F)C2CCC2)C1 15417,S(=O)(=O)(c1cc(NC(=O)C(C)S)ccc1O)NC(CC)C(N)=O 15418,c1(OC)ccccc1NC(=O)CC1(O)CC1.C1(OCC(=O)NC)CCCCC1C 15419,N1(C(CCCC(=O)OCC)=O)CC2CC3CC2C1C3NC(c1coc(C)c1)=O 15420,c1(C(N(CCCCNC(C2(Cl)CC2(C)C)=O)C)=O)ccn2c1CCCC2 15421,C(CC(C)(C)c1ccccc1)N(C)Cc1ncn(C2CCC2)n1 15422,c1(C(=O)Nc2n(C(C)(C)C)cc(C#N)c2)ncnc2c1ncn2C 15423,Cn1nc(C(=O)NCC2COCC2NC(C2CC=CCO2)=O)c2c1CCOC2 15424,c1(C(N2CCC(C(C)NC(=O)COCC3CC3)C2)=O)ccccc1-c1cn[nH]c1 15425,C1(n2nnnc2C2CC2)(NCC2N(C(CCC3CCC(C)O3)=O)CC2)CCOCC1 15426,C1(CC)CCN(C(c2cccc(=O)o2)=O)C1C(=O)NCC1(F)CCOC1 15427,C(N=c1[nH]c(=NCCC23CCCC2C3(F)F)[nH]c2c1CCC2)c1c(Cl)ccc(Cl)c1 15428,c1(CC)cc2scc(Cl)c2[nH]1.C12(C(=O)O)CC(OC)CN1C2=O 15429,N1(C(c2c(C)sc(O)n2)=O)CC2(CC2)CC1CNC(c1nccc(Cl)c1Cl)=O 15430,CC(CNC(=O)CC(C)(C)C#N)C(F)C(=O)N(C)Cc1cccnc1O 15431,C1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)CN2CCCN1CC2 15432,C1(C(=O)NCCC(=O)N(C)C)CCN(C(C2(O)CCSCC2)=O)CCO1 15433,c1(C(N(CC(O)CNC(=O)Cn2ncn(C)c2=O)C)=O)ccccc1CO 15434,N1(C(C)C(=O)NC(c2ccccc2)=O)CCOc2ccc(-c3cccc(Br)c3)cc21 15435,c1(C(=O)NCC(CNC(=O)C(C2(O)CCCC2)F)F)ccc(Cl)cc1O 15436,C12(CNC(COC3C(NC(C(N4CCOCC4)C)=O)C3)=O)CCC(CC1)CC2 15437,Cc1oc(C)c(C(N2CCC(N(C(=O)Cc3cccc(F)c3)C)C2)=O)c1Br 15438,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C(F)C1 15439,C1(CC)(CNC(=O)C(F)CC2CN(C(C3(C)CC4CC4C3)=O)C2)CCCCO1 15440,N1(C(C2CCCCN(CCC(=O)NC)C2=O)=O)CC2COCC(C1)C(=O)N2 15441,C1(C)(C(=O)NCCN(C(C(C)Cc2cnn(C)c2)=O)C)CCC(=O)NC1 15442,N1(C(CN(C(C(C)C)=O)C)=O)CC=CC(NC(=O)CC2CCC(C)(C)O2)C1 15443,C1(NC(=O)CC2C=CCC2)CC(F)(CNC(c2cc(C(F)F)cs2)=O)C1 15444,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CN(C)C(c1nc(Cl)cs1)=O 15445,C(=O)(CCS(C)(=O)=O)N(C(C)C(=O)NCC1CCCCC1O)C1CC1 15446,CC(C)(C(=O)N1C2CCC1C(CO)C2)C(F)c1ccccc1 15447,C(c1ccccc1Cl)=CC(=O)NC1CN(C(C(C)(C)OCC)=O)CC1SC 15448,c1(C(=O)NCC2CCCC(NC(CC3(C)CC3(Cl)Cl)=O)C2)ccc2nsnc2c1 15449,CC1(C)CCC(C(N2CCCC(n3cc(COc4ccncc4)nn3)C2)=O)C1 15450,C1(NC(C(CC=CC)NC(=O)CC2CCC(=O)C2)=O)CC2CCC(C1)N2C 15451,CC1CCC=C1C(=O)NCC=CCC(=O)NCC(=O)NC(C)C 15452,C(=O)(CCC(=O)N(C1C(CCC)C1)CC)OC.C1(=O)CCCn2ccnc2CN1 15453,N1(C(C2(NC(C)=O)CCCC2)=O)CCC2(CC(NC(c3ccc(C#C)s3)=O)C2)C1 15454,C(c1ccncn1)=CC(=O)NCc1cc(C(=O)NC(C)CO)on1 15455,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15456,c1(CC(=O)NC(C)CCN(S(C)(=O)=O)C)ccc2oc(O)nc2c1 15457,C(=O)(C(C)(O)C(C)(O)C(=O)O)N1C2CN(C(C(C)CN)=O)C(CC2)C1 15458,c1(C(=O)NCC2CN(C(CC)=O)C3C(O2)COC3)cc2cccnc2cc1F 15459,Cc1ccc(C(=O)N(C2CCN(C(c3cnc(O)o3)=O)C2)CCO)nc1O 15460,n1(CC(=O)NCC(CC)NC(=O)C(O)COC)cnc(-c2ccccc2)n1 15461,C#Cc1cc(C(=O)NC(C)CNC(C2CC23CCCC3)=O)cc(N)c1 15462,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOC(C)C)=O 15463,C(=O)(C(F)(F)C=Cc1ccccc1)N(C1(C)CCC1)CC(F)(F)F 15464,N1(C(C2(C(C)NC(c3ccc(O)nn3)=O)CC2)=O)CCCN(C)CC1 15465,c1(CNC(C(COCC2CCOCC2)=O)=O)cc(C2(C3CC3)CC2)n[nH]1 15466,N1(C(c2nn(CC)c(C)c2)=O)CC2CC(NC(=O)CNS(=O)(=O)CC)C1C2 15467,CC1(C(=O)NCCC2(O)CCCC2)CCCN(C(c2ccc(C#N)cc2)=O)C1 15468,C1(CC)C(NC(=O)C(C)CN2CCCC2)CCCN1C(C1CCC(O)C1)=O 15469,N1(C(c2cnc(C)s2)C(=O)NCCC)CCCC(c2ccc(Cl)nc2)C1 15470,CC1(O)CCCN(C(C2(CNC(=O)Cc3cn[nH]c3)CCOCC2)=O)C1 15471,C#Cc1ccc(C(=O)NC2C3CC2N(C(=O)Cn2ncnn2)C3)nc1 15472,c1(C(=O)NC2CC(CNC(COCCC#C)=O)C2)cc(Br)c(OC)cc1C 15473,c1(-c2cccc(-c3c(C)cccc3)c2)ccncc1S(=O)(=O)NCC(C)O 15474,N1(C(C(C=CCCC)O)=O)CCN(CCNC(=O)C(C#N)CC)CC1 15475,c1(C(=O)NC2C(CNC(=O)CCCOC3CC3)CC2)ccc(C2CC2)cc1Cl 15476,C1(NC(c2ccnc(C(C)C)n2)c2nnnn2CCCF)CCC2(CCC2)CC1 15477,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCC2C(O)CC12)=O 15478,C12(CC)COC(C(=O)NC(C)CCCNC(=O)Cc3cccc(Cl)c3)(C1)C2 15479,C1(NC(CC=C(C)C)=O)CN(C(C2CCCN2C(=O)C2CC2)=O)C2CC12 15480,CCCC(C(O)C(=O)N1CCCC(CCO)C1)NC(C1CCCCO1)=O 15481,N1(C(C2CC(NC(=O)Cn3ccnn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15482,c1(CN2CC3C(C(N4C(C)C=CC4)=O)C3C2)cc2ccccc2o1 15483,O=C(C1=CCCOC1)N1CC(n2ccc(CNC(C34CCC3C4)=O)c2)C1 15484,CCC(C)CC(CO)NC(=O)Cn1cc(CSc2ccncc2C(F)(F)F)nn1 15485,C(=O)(C(CC1CCCO1)C(F)(F)F)N1CCCC1.Cc1nn(C)c(C)c1N 15486,CC(N)CCCC(=O)N1CCN(C(c2ccc(-n3cnnn3)cc2)=O)CC1C1CC1 15487,Cc1cc(CC(=O)NC2CCC(NC(C3NC(=O)CC3C)=O)CC2)ccn1 15488,c1(NC(C(N2C(CNC(C(CCC)F)=O)CC2)=O)=O)c(C)cccc1C 15489,N1(C(c2cn(CC)nc2)=O)CC2CN(C(c3ccnc(C)c3)=O)CC12 15490,CC(C)C(C#N)C(=O)NC1(C(=O)N(C)CC2CC(O)C2)CSC1 15491,C1(O)(C(N2CCN(C(=O)CSc3ccc(Cl)c(F)c3)CC2)=O)CN2CCC1CC2 15492,c1(CC(=O)NCCCCCCCNC(CSCC#C)=O)ccc(F)c(Cl)c1 15493,N1(C(CCCCC=C)=O)CCC2C(C1)CN2C(C1CCN(CC(F)(F)F)C1)=O 15494,CCC(O)C(C)(C)C(=O)N(C1C2CN(C(C)=O)CC12)C1CC1.C(=O)CCC(F)(F)F 15495,Cc1cnc(C(=O)NCC2CN(C(c3cccnc3)C)CCO2)cc1C 15496,C1(C(=O)NCc2cccc(C)n2)(COC)C=CCN1C(c1ccccc1O)=O 15497,c1(NC(CNC(C(c2ccc(F)cc2)(C)C)=O)C2CC2)ncnc(O)c1Br 15498,C12(C(=O)NCCOCCOCCNC(c3c(C)noc3C)=O)CCCC(F)(C1)C2 15499,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1cnc(C(F)(F)F)n1 15500,C=CC(C)C(C)C(=O)N(CC(C)(C)CNC(=O)CC1(C(=O)OC)CCCC1)C 15501,C=C(F)C1(CC(=O)NC2CC(NC(C3(OC)CCC(C)C3)=O)C2)CCC1 15502,N1(C(CC2CCCC(C)C2)=O)CC2(CNC(c3coc(C(N)=O)c3)=O)CCC1CC2 15503,c1(CC(=O)NCC2(F)CCC(NC(=O)CC3CC3)C2)ccc(O)c(Cl)c1 15504,c1(OCC)ccc(CCC(C)NC(=O)COC(C2(OCC)CCC2)=O)cc1 15505,O(N1C(=O)c2ccccc2S1(=O)=O)C(C)C(=O)OO.C1CCCC1 15506,N1(C(C(C2CC2)OC)=O)CC(F)(F)CC1C(=O)NC(C)CN1CCCCC1 15507,c1(C(=O)NC2CC3CN(C(C(C)=C(C)C)=O)CC32)cnc2[nH]ncc2c1 15508,C#Cc1cncc(NC(C2CNC(=O)CN2C(=O)C2=COCC2)=O)c1 15509,C1(CNC(CSC(C)(C)C)=O)CCC2(CN(C(c3cc(N)ccn3)=O)C2)O1 15510,S(=O)(=O)(c1ccc(C(=O)O)c(C#N)c1)NC(C)CCCCCO 15511,c1(C(N2CCC(C(C)NC(C(n3cc(C4CC4)cn3)C)=O)C2)=O)c(O)cccc1Cl 15512,C1(C)(C(N(C(C)C(=O)NCc2[nH]nnc2CC)CC)=O)CCC(C)C1 15513,C1(CC(=O)NCC23CC(NC(C(N(C)C)C4CC4)=O)(C2)C3)CC(O)C12CCC2 15514,c1(C(C(=O)NCC(C)(C)C)N(CCOC)CC)scc2c1OCCO2 15515,c1(OC)ccc(-n2nc(Cc3nc[nH]n3)nc2COC(F)F)cc1 15516,c1(C(=O)NCC(CC)(C)NC(=O)C=Cc2cocn2)noc2c1CCCC2 15517,N1(C(C(c2nncn2C)C)=O)CCCC(C2CC2NC(C2(C3CC3)CC2)=O)C1 15518,CCC(C)(C)C(O)C(=O)NCC1CC(C)CN(C(=O)C(F)(F)CO)C1 15519,c1(C(=O)NC2C3CC(NC(C4C(CC)C4)=O)CC32)ccc2nc(C)sc2c1 15520,c12ccc(cc1)CN(C)C(=O)C2.C1(NC2(C(=O)OCC)CC2)CNC(=O)N1 15521,N1(C(c2n(C(C)C)ncc2Cl)=O)CCCC(NC(c2cc(=O)n(C)cn2)=O)CC1 15522,C12(CCCO1)C(=O)NCc1cc(on1)C(=O)N2.C1CCC(O)C1.COC 15523,CCCC(C)(CO)NC(=O)CN(CC(C)C)C(c1cc(OC)ns1)=O 15524,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15525,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15526,c1(CC(N2CC(Nc3ncnc(CC)c3F)C(C)C2)=O)noc2ccccc12 15527,CC1CCCC(O)(C(=O)NC2CC(C)(Nc3ncc4c(n3)COC4)C2)CC1 15528,CCCCC(O)C(C)C(=O)NC1CCOC(C(=O)NCc2occc2C)C1 15529,C(=O)(CCCCC(C)(C)OC)N1C(C(C)(C)NC(CCC=CCC=C)=O)CCC1 15530,Cc1cc(C(=O)NCCC(C)(C)NC(=O)C(=O)N(C)C)nn1CC(F)(F)F 15531,CC1CCCCC1N1CCCC(NC(c2cc(I)cn2C)=O)C1 15532,c1(N2CCN(CC(=O)NC(COC)C)C(=O)C2)ccnc2cc(Br)nn12 15533,CCCC(CCCNC(=O)CCCOC)NC(c1cc(F)ccc1N)=O 15534,c1(C(N2CCN(C)CC2CNC(C2CN3CCN2CC3)=O)=O)n[nH]c2cccnc12 15535,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15536,C1(C(=O)NCC2CN(C(=O)CCc3ccc(F)cc3F)C2)CC2(CCC2)CCO1 15537,O=S(=O)(c1c[nH]ccc1=NC1CCC(C2CCC2)C1)N1CC2(CCC2)OC1 15538,C=C(C)CCC(C)(c1nnnn1Cc1ccccc1)NC(c1ccc(Br)cc1)C 15539,N1(C(C2CC(=O)N2)=O)CC2CCC1C(C(N1CCCCC1CCC(=O)O)=O)C2 15540,Cn1ccnc1SCC(=O)NCCCC1(NC(CCOCc2ccco2)=O)CC1 15541,C1(NC(C(CO)NC(C(CC#C)O)=O)=O)CCC(N=[N+]=[N-])CC1 15542,N1(C(CC(C=C)C)=O)CCc2sc(CNC(=O)Cn3cnnc3O)nc2C1 15543,C1(CCN)CNCCN1C(c1cnccc1Cl)=O 15544,CC1CCCCCC1NC(=O)CC1CCCCN1C(=O)COC1CC1 15545,c1(OC)cc(NC(C2CC(F)CN(C(=O)C(N3CCCCC3)C)C2)=O)cc(Br)c1 15546,c1(-c2ccc(CSCC(C)(C)O)cc2)ccc(F)c2ccoc12 15547,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CC)c2C)=O)C1 15548,C=C1CCN(C(=O)Cc2ccco2)C(C(=O)NOCCOCCO)C1 15549,C(=O)(C(C)(C)C1CCCCO1)NC(CN(C(COCC)=O)C)C 15550,CCCCC(C(=O)NCC(C)(C)CN(C)C(C1CC1CF)=O)C(C)C 15551,C1(OC)CN(C)C(C)(C(=O)NC2CC(CNC(c3ccncc3N)=O)C2)C1 15552,C12CCCCC1C(=O)NC2.c1(C(C)NC(C(SC)SC)=O)ccccc1O 15553,C(=O)(C(O)CCC(F)(F)F)N1CCN(C(c2c(CC)nns2)=O)C2C1C2 15554,CC(C)C(C(=O)N(C)CC1(COC)CCC1)NC(=O)CC1CCOC1=O 15555,c1(OC)cc(C(=O)NC(CCNC(C2C(F)(F)C23CC3)=O)C(C)C)cc(OC)n1 15556,C#CCC(C(=O)NC(CO)CC=CC)NC(c1cnc(CC)nc1)=O 15557,c1(Sc2c(N(CCN(C)C)C)[nH]cc2)nccc(-c2ccnn2C)n1 15558,C#Cc1ccc(C(=O)N(CC(=O)NCc2ccco2)C(C)C)o1 15559,C=C(F)C1(CC(=O)NCC(C)NC(=O)CCCC(=O)OC(C)(C)C)CCOCC1 15560,n1(CC)cc(C2(C(=O)NC3CCCC3N)CC2)cn1 15561,C=CCC(CN(C(=O)CC1CCCOC1)C1CC1)C(=O)NCP(C)(C)=O 15562,C1(CNC(c2nc(COC)oc2)=O)CN(C(=O)Cc2ccccc2C)CCCO1 15563,c1(N2CC(C(C)NC(=O)COCC(F)F)C2)c(Cl)cc(F)cc1Br 15564,c1(CN2C(C(=O)NC(CCC)C)CC3(CC3)C2)c(F)cc(Br)cc1Br 15565,C1(C)(C(=O)NCCN(C(c2cc(CC)c(C)s2)=O)C2CC2)CCC(=O)N(C)C1 15566,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)C2)[nH]1 15567,C1(CC(=O)NCC2(C(=O)OC)CCC2)CCN(C(=O)C(C)O)CC1 15568,C(CCCCCNC(C1COCCO1)=O)NC(=O)COC1CCOCC1 15569,CCCC(C(=O)OC1CCN(C(C2CC2OCC)=O)C1)NC(=O)OC(C)(C)C 15570,N12CC(C(O)C1)N(C)C(=O)c1ncoc1C2=O.c1(CC)cc(=O)cc[nH]1 15571,c1(OC)cc(=NC(=O)Cc2nc(C(=O)Nc3n[nH]cc3Cl)cs2)[nH]o1 15572,N1(C(C2C(C)C2)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15573,c1(C(CC)=O)ccc(NCC(C)CNC(C2CCOCC2(C)C)=O)c([N+](=O)[O-])c1 15574,CC(CNC(=O)CCC(C)N(C)C)C(F)C(=O)NCCc1cc[nH]n1 15575,C(=O)(C(CCCCCN)C(=O)O)N1CC(C)N(c2ccc3c(c2)CCCC3)CC1 15576,C1(C(=O)Nc2cc(-c3ccncc3)cnc2O)CC(C(=O)O)C(O)C1O 15577,N1(C(C2CC(NC(C3N(C)C(=O)CC3)=O)C(O)C2)=O)CCC(F)(F)C(O)C1 15578,c1(C(=O)NCCC(C)NC(c2c(C)scc2)=O)cc2cnccc2[nH]1 15579,C(=O)(CCC1=CCCCC1)N1CCN(C(CC(C(C)C)O)=O)C(CO)C1 15580,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15581,CCC(CNC(C1CC(C)CCN1C(=O)CSCC(N)=O)=O)(CC)CO 15582,C1(C)(C(=O)NCC2C(C(=O)NCCC(C=C)(C)C)CCCC2)CCC2CC2C1 15583,C12(CC(=O)NCC(F)CO)CCC1CN(C(c1cc(CCO)on1)=O)C2 15584,Cc1cc(=NCc2csc(Br)c2)[nH]c(=NCc2conc2C)[nH]1 15585,Cc1ccc(CC(=O)NC2COCC2NC(c2snnc2C2CC2)=O)c(Cl)c1 15586,c1(NC(Cn2cc(CNC(C(C)SCC=C)=O)nn2)=O)cccc2c[nH]nc12 15587,Cc1ncsc1C=CC(=O)NCCN(C(=O)CS(=O)(=O)NC1CC1)C 15588,C1(CNC(C(CC)N(CC)CC)=O)CCN(C(c2cncc(OC)c2)C#N)CC1 15589,c1(C(=O)NC2CCN(C(=O)CC3CCC4CC4C3)C2)ccc2cc[nH]c2n1 15590,C1(C(=O)NC2CC2NC(=O)Cc2ccn(C)n2)(COC)CCCO1 15591,C1(OC)CC(C(=O)NCCCSC)N(C(=O)CCCc2cccs2)C1 15592,c1(CNC2CCC(C(=O)Nc3c(OC)nnc(Cl)c3)CC2)c(F)ccc(F)c1O 15593,C1(NC(CNC(C)=O)=O)C2CN(C(C3CCCN3Cc3nnn(C)n3)=O)CC12 15594,N1(C(=O)COC2CC(F)(F)C2(C)C)CCOc2ccccc21.CC1C(C)(C)N1 15595,C1(C(N2CC3C(C)(C)C3C2)=O)CC2C=CC1N(C(c1cccc[n+]1[O-])=O)C2 15596,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15597,N1(C(=O)NCc2cccc(OCC)n2)CC2CC(C)(C)C2C1CO 15598,Cc1ccc2ncc(C(N3CCC4(CC(NC(C5C=CCCC5)=O)C4)C3)=O)n2c1 15599,c1(C(N2CCC(NC(c3cncc(CC)c3)=O)C2C)=O)c(C)cc(F)cc1Br 15600,CC1CN(c2nnnn2C2CCCN(CC3CCCCC3)C2)CCC1NC 15601,N1(C(C2CN(C(c3cccnc3F)=O)C2)=O)CC2C(C1)C2(F)F 15602,N1(C(C2(C)CC=CC2)=O)CC(C)CN(C(c2ccc(C3CC3)cn2)=O)C(C)C1 15603,N1(C(C2CC(CNC(CC#N)=O)OC2)=O)C(CO)CCC1C1CC1 15604,C#CCC(O)C(=O)NC(C(=O)NC1CC(CC(N)=O)C1)C1CCOC1 15605,C1(NC(C(F)=CC)=O)CC2CCC1CN(C(c1cc(C(F)(F)F)ccc1C)=O)C2 15606,c1(C(=O)NC2C(C)(CN(C(C3C(=C)C3)=O)C)CCC2)c(S(C)(=O)=O)cnn1C 15607,CS(=O)(=O)CC(=O)N1CC(F)CC1CNC(C1CC=CCO1)=O 15608,CC(CCCCCO)NC(c1nnnn1C(C)C)(C1CCCCC1)C 15609,c1(C(=O)NC2C(OC)CC2)cnn(CCNC(=O)CC2CC(COC)C2)c1 15610,Cc1cnccc1CC(=O)NC(C)CN(C(=O)C(C)NC(c1cccs1)=O)C 15611,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]nnc1C1CC1)=O 15612,C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)Cn2ccnc2)CC1S(C)(=O)=O 15613,N1(CCSC(=N)N)CC(C(=O)NCc2cccc(Cl)c2)C(C)(C)C1 15614,CN1CC=C(CNC(=O)CONC(C2(C)C(C)(C)C2(C)C)=O)CC1 15615,C(CNC(=O)CCCF)(CC(=O)N(C)CC1(C)CCCO1)OC 15616,CCCCC(COC)NC(C1(CF)CCN(C(=O)C=CC(F)(F)F)C1)=O 15617,C1(C(N(c2cn(CC)nc2)C)=O)COCCN(C(=O)CC2CC2C2CC2)C1 15618,c1(C(=O)NCC2N(C(=O)C3=CCCS3)CCC(C)C2)cnc2ccoc2c1 15619,C1(C(=O)NC2(Oc3ccccc3)CC2)CCCC1CNC(C1CCOC1C(F)F)=O 15620,N1(C(C(C)C(C)(F)F)=O)CCOC2(CCCN(C(=O)Cc3csc(S)n3)C2)C1 15621,N1(C(C2(CC=C)CCN(C(c3ccc(CC#N)cc3)=O)C2)=O)CCC=C(CO)C1 15622,C1(CN(C(c2cc(CNC(CCCC)=O)no2)=O)C)CCCCCC1 15623,C1(C(C)C)CN(C(c2cc(-c3ccco3)c[nH]2)=O)CCN1C(C1COCC1C)=O 15624,Cc1nnc2n1CCCC2C(=O)N1CCCC1CNC(c1ccn2c1CCCC2)=O 15625,c1(C(=O)NC2C3CN(C(c4cnc(C(C)C)[nH]4)=O)C2C3)ccc2c(c1)CCC=C2 15626,c1(C(=O)NCC(CNC(=O)CO)OC)cnn(-c2ccccc2Cl)c1C(C)C 15627,C(=O)(C(C)(C)C)N(CCn1cc(C2CC(C)CO2)nn1)CCC(C)=O 15628,Cc1cc(CN(C(=O)CCCCN(C)C)C)cnc1C.C12CN(CC13CC3)C2=O 15629,Cc1cn(C)cc1C(=O)NCCC(C)NC(C1CCCCO1)=O 15630,C(=O)(CCC(CF)CF)N1CC2C(NC(c3n[nH]c(C)c3Br)=O)(CC2)C1 15631,c1(CCC)nc(C)c(C(=O)N(CCC)CCN(c2ncc(NC)cn2)C)s1 15632,c1(CC(=O)NC2C(CC(C)(C)C)CN(C(C3CCCS3)=O)C2)ccc(Cl)cc1F 15633,c1(SCC2(NC(=O)NCc3ccc(C)cc3)CC2)cnc2[nH]c(C)nc2c1 15634,C(CCN=c1[nH]c(=NCC(C)SC)[nH]c2c(F)cccc12)COCC=C 15635,C(CCCC1CCCC1)NC(C1(CNC(C2(CCOC)CC2)=O)CCC1)=O 15636,CC1CC(C(=O)NCC(O)C(=O)NC(c2nn[nH]n2)C2CC2)CN1C 15637,c1(C(=O)NCC2(C)CCC(NC(CCC(C)OCC)=O)C2)cnc(C)nc1CC 15638,N1(C(CCC2C(C)(C)C2)=O)CC2CCCC2(CNC(C23CC2C3)=O)C1 15639,c1(C(C(N2C(C(=O)NCC=Cc3cnc[nH]3)CCC2)=O)O)ccc([N+](=O)[O-])cc1 15640,C12(CN(C(C3CCCCC3)CC)CC)COC(CNC)(C1)C2 15641,C1(NC(CC(C2CC2)NC(C)=O)=O)CCCN(C(c2cc[nH]c(=N)c2Cl)=O)C1C 15642,c1(C(N2CC(=C(CNC(C(C)Cc3cnc[nH]3)=O)F)C2)=O)ccc([N+](=O)[O-])s1 15643,C(=O)(C(O)C(F)F)N1CCC(C(C)(C)NC(c2cc(C(=O)OC(C)(C)C)on2)=O)C1 15644,c1(C(=O)NCCCNC(C2N(C(C)C)CCC2)=O)cc(Cl)cc2[nH]ccc12 15645,N1(C(=O)NCc2cc(C#N)c(F)nc2N)CC(F)(F)Oc2cccc(F)c21 15646,N1(C(c2ccc(C(=O)OC)s2)=O)CCC2(CCCN(C(=O)C(O)P(C)(C)=O)C2)C1 15647,N1(C(c2c(C)cco2)=O)CC2(CC(NC(=O)C(F)C3CCC3)CO2)C1 15648,N1(CC2C(C)(C)CCO2)CCCC(n2cc(CN3CCCC3CO)nn2)CC1 15649,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15650,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15651,Cc1cnc(Br)c(NC(C2CC23CN(Cc2nc(Br)cs2)C3)=O)c1 15652,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15653,c1(OC)ccc(C)cc1C(N1CC2(C1)CN(C(=O)CCC1CCC(=O)NC1)C2)=O 15654,C1(NC(CC(C(C)C)OCC)=O)CC2CCC(C1C)N2c1ncc(I)cn1 15655,C1(O)(CNC(c2nn(C)c(F)c2)=O)CCN(C(=O)CC2CCCC(=O)N2)CC1 15656,N1(C(CCC(=C)Cl)=O)CC(NC(c2cnn(C3CCC3)c2C)=O)CCC1C 15657,NS(=O)(=O)c1cc(C(=O)NC2(c3ccc(C(F)(F)F)cc3)CC2)cs1 15658,c1(CNC(c2ccccc2)C#N)cccnc1-c1cccnc1 15659,N1(c2cccc(SC(C)CCn3cccn3)c2)c2ccccc2C(C)(C)C1 15660,C1C(C)(C)NC(=O)CCNC(=O)C=CC(=O)N1C.C(=O)(CO)NC1CC1 15661,N1(C(=O)NCc2cc(C(C)C)no2)CCOC(C)C1 15662,N1(C(=O)CON2CCOCC2)CCC2(NC(C3CCCN3C3CC3)=O)CCCC12 15663,c1(C(=O)NC2(CCNC(C3CC(C)(CC)C3)=O)CCCC2)cncc2c1CCC2 15664,c1(C(=O)NCC2N(C(C3CC(C)(C(=O)OC)C3)=O)C3C(C2)C3)cccc(Cl)c1C 15665,CC1CCCC1(C(=O)N(C)Cc1cncnc1)NC(=O)CCc1cn(C)nn1 15666,CCC(CC)(CCNC(C1CCC1C)=O)NC(=O)Cc1ccc(C)c(Cl)c1 15667,C1(C(=O)NC(C(C)C)CNC(C2CCC(=O)N2)=O)CC(=O)N(C2CCCC2)C1 15668,N1(C(c2c(C)nccc2)=O)CCC(CO)C(NC(=O)C(C)(C)C2CCOCC2)C1 15669,Cc1cc(F)c(F)cc1C(=O)NC1CN(Cc2ccc(F)c(O)c2)CC1F 15670,Cc1cc[nH]c1C(=O)NCC1CC(C(=O)NC(c2ccnn2C)(C)C)C1 15671,C1(C(N2CCCC(OCC)C2)=O)CCN(C(C2CCCSC2C)=O)C(C)C1 15672,CCCCCCN(CCc1c[nH]nc1OC(c1cc(C2CC2C)on1)=O)CC 15673,N1(C(C(C=C)CC)=O)CCN(C(=O)Cc2c(C)cccc2F)CC(O)C1 15674,c1(C(=O)NCCCCNC(=O)C(F)C2CCOC2)ccc2c[nH]nc2c1 15675,C1(NC(=O)C=C2CCC2)CCN(C(c2ccc(C3(O)COC3)cc2)=O)CC1 15676,N1(C(CCCC#CC)=O)CCN(C(C23CCCCC2OCC3)=O)CC(O)C1 15677,c1(NC(CC(CC#C)NC(=O)C(C)C(C)OC)=O)ccc(C)c(C#N)c1 15678,c1(CNC(CN(C(c2ccc(C#C)o2)=O)C2CC2)=O)cc(C)ccc1O 15679,CCC(CC(=O)N(CCC(C)NC(=O)CCCc1cccs1)C)C(F)(F)F 15680,Nc1cnc(C(F)(F)F)cc1C(=O)NC1CC1NC(c1cccn(C2CC2)c1=O)=O 15681,S(=O)(=O)(c1cnoc1C)Nc1cccc(N2CCC(CC(=O)OC)C2)c1C 15682,C1(O)(CCNC(c2c(C)ncs2)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 15683,C1(C(N2CC(CC)OCCC2)=O)CC(N=[N+]=[N-])CN1C(C1CCC(=O)N1C)=O 15684,N1(C(C(C)(C)F)=O)CC2CN(C(c3cccc(Cl)c3F)=O)CC12 15685,c1(OC)cc(CCC(=O)NC23CC(NC(c4ccc[nH]4)=O)(C2)C3)ccc1O 15686,c1(C(N2CC3CCN(C(C4(C)CC4)=O)C3CC2)=O)cccc(C2=CCOCC2)c1 15687,CC(C)C(C)CN(CCC(=O)N(C)CCOCCCN(C(=O)CC1CCC1)C)C 15688,C12(NC(c3ccc(C)cc3C)=O)CCC(CN(C(=O)CCC3CC3)C1)C2 15689,C1(c2cn(CCOCCOCC(=O)Nc3ncccn3)nn2)CCCCCC1 15690,C1(C(C(=O)NC2CCC2)N(C2CCCOC2)C)CCC2CC2C1 15691,C(=O)(C1CCCc2ncnn21)NCC1N(C(c2c(C)[nH]c(=NCC)s2)=O)CCC1 15692,N1(C(C)(C)C)CC(C(=O)NCC2(C)CCCN2C(C2CC3C=CC2C3)=O)CC1=O 15693,CC(C)CC(O)CNC(c1ccc(CNC(=O)CCN(C)CCO)cn1)=O 15694,C(CC(F)=C(F)F)CNC(C1(SC)CN(C(CCC=CCC=C)=O)C1)=O 15695,c1(CC#N)cccc2c1CN(C(c1ccc(Cl)cc1)c1ccnc(OC)c1)C2=O 15696,c1(OC)nsc(CNCC(c2cccc(Br)c2)C)c1Br 15697,C1(NC(CC)C(=O)NCC)(Cc2ccccc2)CCCN(Cc2cnccc2C#N)C1 15698,N1(C(c2cc(CCC)on2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15699,N1(C(C(C)OCC)=O)CCCCC1CNC(C12CCC(CC1)C2)=O 15700,c1(N2CCN(c3n(CC(C)F)nnn3)CC2)cc2c(cc1Br)OCCO2 15701,Cc1ccc(C(F)C(=O)NCCOCCCN(C)C(c2cncc(N)n2)=O)cc1 15702,C1(C(N2CCC(CNC(c3c(C)nn(C)n3)=O)C2)=O)CCCC2(CC2)C1 15703,C1(NC(COC(C)C)=O)C=CC(C(=O)N(CC(C)O)CCc2ccccc2)C1 15704,c1(C(=O)NC23C(CN(C(c4cnnc(Cl)c4)=O)C2)C3)c[nH]c2cc(F)c(F)cc12 15705,c1(C(C)C)ccc(C(=O)NCC(C2CCC2)NC(=O)C=Cc2cnccn2)nc1 15706,c1(OC)ncc(Br)cc1C(N1CC(CC(=O)Nc2cc(C(=O)OC)ccn2)C1)=O 15707,c1(CN(C2C(C)CCNCC2)C(c2ccn(C)c2)=O)ccc([N+](=O)[O-])cc1I 15708,c1(NC(C2C3CN(C(CCC#C)=O)C2C3)=O)cc(Cl)nnc1Cl 15709,C1(C(=O)NC(C(C)C)(C)CNC(c2ccn(C3CCC3)n2)=O)CCCCCCC1 15710,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(OCC(C=O)NC(=O)OC(C)(C)C)C1.OC 15711,c1(CC(N)=O)ccc(C(=O)NC(c2ccc(Br)cc2)c2cncnc2)cc1 15712,N1(C(C=C2CCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15713,C(CC(F)F)(C(=O)N1CCC1c1ccccc1)NC(CCc1onc(C)n1)=O 15714,C1(C(N2CC(C(C)(C)O)OCC2)=O)CCCN(C(c2ncc(F)cc2F)=O)CC1 15715,CC(c1ccccc1)=CC(=O)NCC1CN(C(C2(C(F)(F)F)CC2)=O)CCN1C 15716,c1(CC)cnc(CNC(=O)C(c2cnn(C)c2)NC(c2cc(C)c[nH]2)=O)[nH]1 15717,CC(C)CC(C(=O)NCC(C)(C)CCNC(C1(C#N)CCCO1)=O)C(C)C 15718,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15719,C(CCS(=O)(=O)C(F)F)N(C1CC(C)(C)OC1(C)C)C 15720,c1(CC(=O)NC2CC(CNC(C3N(CC)CCOC3)=O)C2)cnn2c1CCCC2 15721,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15722,c1(CNC2CCCC(C(N(C)C)=O)C2)cc([N+](=O)[O-])c(O)cc1F 15723,N1(C(=O)CC2(C3CC3)CC2)CC2ON=C(CNC(C3(CO)CCOCC3)=O)C2C1 15724,c1(NCC(CC)Cc2ccccc2F)ncnc(NCc2nc(C)cs2)c1C 15725,n1(CC)nc(C2CC2)cc1C(=O)NC1COCCC1NC(=O)CNC(C)=O 15726,C1(S(N)(=O)=O)(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)CCCC1 15727,C1(C(N2CCC(NC(CCOCCC)=O)C23CC3)=O)CCc2cnc(C)n2C1 15728,CC1(CCCO)CCCN1C(=O)Cc1cnccn1.C1(=O)CCN1CCO 15729,C=CCC(C(=O)NC1CCCCCC1)C(C)C.C1(C)C(=O)N1 15730,c1(CC(=O)NC2(C)CC(NC(c3coc(C(N)=O)c3)=O)C2)ccc(CC(N)=O)cc1 15731,C(=O)(C1COc2ccc(F)cc21)N1CC(C)(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15732,c1(CC(=O)N(C)CC2CCCN2C(=O)C(C)(O)C2CC2)cnn2c1OCCC2 15733,c1(C(=O)OC)ccc2nc(N3CCC(OCCN)C3)sc2c1.C1(C)(O)CCOCC1 15734,c1(C(C)NC(C2CN(C(=O)C(F)CC)C2)=O)ccc(NC(=O)COC(F)F)cc1 15735,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15736,N1(C(C2(C=C)CC2)=O)CCC(C2(CNC(C3CCC(=O)N3)=O)CCOCC2)CC1 15737,c1(C(=O)NC(c2ccccc2)CO)cc(F)c(O)cc1F.N12CCN(CC1)CC2 15738,C=C(C)C1OCCC1C(=O)NC1CC2(C1)CC2NC(=O)CCc1ccc(C)o1 15739,c1(OC)ccc(OC)c(CC(=O)NCCCC(C)CCNC(=O)CC2CC2(C)C)c1 15740,c1(C(N2CCN(C(CCC3N(C(C)=O)CCC3)=O)CC2)=O)ccc(F)c(Br)c1F 15741,CC(C)C(CNC(c1cn(CC2CC(CF)C2)nn1)=O)NC(C1CC12CCC2)=O 15742,c1(C(N2C(CNC(C3CCCS3)=O)CCCC2)=O)ccc2ncsc2c1 15743,C1(C(=O)NCC(O)C(C)O)(NC(COC(C)C)=O)CCCC1 15744,N(C(=NCCF)NC1CCC(c2ccc(Cl)cc2F)C1)C1CCN(CCOC)CC1 15745,N1(CCNC(c2c(OC)nsc2)=O)CCC(NC(=O)C#CC(=O)N(C)C)CC1 15746,C1(NC(C=CC)=O)CCN(C(=O)CCOc2ccccc2C(N)=O)C(C)C1 15747,c1(Cc2scc(C(=O)NC3CN(C(c4ccc(C)s4)=O)C3)n2)c[nH]c(=N)cc1C 15748,C(=O)(CC(C)CC(C)(C)C)NCC=C(C(=O)N(CCCCCCC)C)C 15749,C12(CNC(c3n(C)ccc3)=O)CCCC1CCN2C(c1csc(C2CCC2)n1)=O 15750,CC(CN=c1nc(N2CC3(CCC3)CO2)c2c([nH]1)COC2)c1nccs1 15751,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15752,C1(NC(C(COC)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15753,CCC(C(=O)N1CCCC1CC(=O)NC(C)C1CC1)NC(N)=O 15754,C(c1ccoc1)=CCN(C(=O)CC1CCN1C(=O)COCC1CCOC1)C 15755,N1(C(C(C)SCC)=O)CC2CC1CCC2NC(c1c[nH]c(C(N)=O)c1)=O 15756,Cc1cccc(OC(C)C(N2CC=CC(NC(=O)C(F)C3CCOC3)C2)=O)c1C 15757,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15758,C1(CNC(C(C)c2cccs2)=O)CCN(C(=O)C(c2cc(CO)on2)=O)CC1 15759,Cc1ncc(-c2ncc(CNC(C(C)(C)C)c3ncccn3)s2)o1 15760,N1(C(=O)OC(C)(C)C)CCCCC1c1nc(CCC2CCC(O)CC2)no1 15761,c1(C(=O)NC(CC(C)C)C(=O)N2CCC(N3CCCCC3)C2)ccn2ccccc12 15762,C#CCCCC(C)C(=O)N1C(C(=O)NCCCOC)CCC12CC2 15763,C(=O)(C(C)CN(C)C(C1CCSCC1)=O)NC(C)Cc1ncco1 15764,C1(NC(=O)NCC(S(C)=O)OC)CCNCCC1c1ccccc1 15765,C=CCC(F)(F)C(=O)N1CCN(C(C2CCN(OCC3CC3)CC2)=O)C(CF)C1 15766,N1(C(C)=O)CCc2ccc(N(C(C)CNC(=O)C(=O)NCCN(C)C)C)cc2C1 15767,N1(Cc2ccc(C#N)s2)CCC2CN(C(c3cc(Br)ncc3Br)=O)CC2C1 15768,c1(OCC(N2C(CO)CC(NC(C=C(C)C(C)(C)C)=O)C2)=O)ccc(C)c(C)c1 15769,N1(c2nccc(C)n2)CCC2(CCC(NC(c3cc4c([nH]3)CCC4)=O)CC2)C1 15770,CC1CC2CCC(C1)N2C(=O)C(C)N(C(=O)C(C#N)C(C)(C)C)C1CC1 15771,C=C(C)CN=c1[nH]c(=NCc2ccc(S(C)=O)cc2)c2ccc(F)cc2[nH]1 15772,N1(c2n(CC(=C)C)c(CC3CC=CCC3)nn2)CCCC2CN(C)CCC12 15773,c1(CC(=O)NCC2CCN2C(c2coc(Cl)n2)=O)cnc2c(=O)[nH]ccn12 15774,CCCCCCC(=O)N1CCCC(n2cc(COC3CCCNC3=O)nn2)C1 15775,Cc1ccc(C)c(C(=O)NCc2cc(C(N3CCC4CC34C)=O)on2)n1 15776,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C=CI)C2 15777,c1(C(=O)OCC)cc2c3c(OC(=O)CCCSC)cccc3ccc2[nH]1 15778,c1(C(N2CC3C(C(N(C(C)CC(N)=O)C)=O)(C3)C2)=O)c(O)cccc1F 15779,C1(NC(C2C(CC)OCC2)=O)(CNC(=O)Cc2nonc2C)CCOCC1 15780,C1(C(=O)NCC2COCC(C)O2)CCC(C)(C)N(C(c2ccc(C#N)[nH]2)=O)C1 15781,C1(NC(COCCN(C)C)=O)CCN(C(c2cc(C#N)cn2C)=O)C12CC2 15782,C1(C(N2CC(CNC(c3cnc4ccsc4c3)=O)C2)=O)CC2CCCCN2C1 15783,C1(NC(CSCCOC)=O)(NC(=O)COc2cccc(C)c2)CC2CCC1C2 15784,c1(OCC)cc(C(=O)NC(C)CC2CN(C(=O)CSSC)C2)[nH]n1 15785,C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)COC(C)C)CC1 15786,N1(C(CN(C(C(COC(C)=O)C)=O)CCO)=O)CC2(C1)CN(C)C2 15787,c1(OCC)ccccc1C.n1(Cc2cn(CCC(=O)NC3CC3)nn2)c(O)nnc1O 15788,C1(C(=O)NCc2cc(C(N3CCC(CCC)C3)=O)sc2)CCC2(CC2)C1 15789,CCCCC(=O)C(=O)NCCN(C(=O)C(C)Oc1ccc(Cl)cc1Cl)C 15790,C(C1CC1)(C1CC1)=CC(=O)NCC1(CNC(C2C(CC)CCC2)=O)CCCC1 15791,C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(CC2(C=C)CCOCC2)=O)CCCC1 15792,N1(C(c2cccc(C(C)C)c2)=O)CC2CCC1CN2C(=O)C(C)(C)F 15793,c1(C(=O)O)c[nH]cc(-c2ccc(CN3CCN(C(=O)C(C)C)CC3)cc2)c1=O 15794,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCN(C(=O)C(O)Cc1ccc(Cl)cc1)C 15795,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)NC(C)Cc1cccs1 15796,c1(C(=O)NCC2CCN(C(CCCOCCOC)=O)CC2)nccc2n[nH]cc12 15797,CCCCCC=CC(=O)N(CC(O)CNC(=O)Cc1cscn1)C 15798,C1(CNC(=O)CCC2CCC2)(CO)CCCN(C(=O)Cc2c(F)cncc2Cl)C1 15799,C(c1cccc(O)c1)=CC(=O)NC(CC1CN(C(c2cccc(C)n2)=O)C1)C 15800,C1(NC(C2N(CC)CCC2)=O)CCC12CCCC2.c12cc([nH]n1)S2 15801,O=C1CCC(CC(N2CCC(O)(C(F)F)C2)=O)CN1 15802,N1(C(Cc2c(C)nc(C)s2)=O)CC(C)CN(C(c2cn(CCO)nc2C)=O)C(C)C1 15803,C(=O)(CC(C)CC(=O)NCC1=CCN(C(C2CNC(=O)N2)=O)CC1)OC 15804,c1(C(N2CCC(CNC(C3N(C)CCC3)=O)C23CC3)=O)cc2cc(O)ccc2[nH]1 15805,N1(C(C2C(CNC(CCCOCC)=O)CCO2)=O)CC(=O)NCC1C(N)=O 15806,C1(C(=O)NC(CC(=O)OC(C)(C)C)CC#N)CC2(CCCCC2)C1 15807,C#CCC(C)(CC)C(=O)N1CCCC1CNC(C1CC12CC(F)(F)C2)=O 15808,C1CCCCC(=O)N1.C1(CC(=O)OC)CCCCN1C(=O)C=CC(=O)N(C)C 15809,Cc1cnccc1C(C)NC(=O)Nc1cc(CCO)nn1C(C)(C)C 15810,C1(NC(=O)C=Cc2ncc[nH]2)CC2CC1N(C(=O)CC1(c3ccc(F)cc3)CC1)C2 15811,C1(NC(C2C(NC(CC)=O)CCC2)=O)CCC(NC(C2SCCCS2)=O)CC1 15812,N1(C(C(C(C)C)CO)=O)CCCc2c(CN=c3[nH]c(Cl)ncc3F)cccc21 15813,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(CC=CCC)=O)CC1 15814,c12cccc(c1C)C(=O)NCCCN2C.c1(C(=O)OCC)cccnc1CC 15815,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)OC 15816,Cc1csc2ncnc(N3CC(NC(c4cnccc4F)=O)CC(O)C3)c12 15817,c1(CCOC)n[nH]c(=NCCCN(C)C(C2CCCC2Sc2cccc(Cl)c2)=O)s1 15818,c1(C(=O)OCC)ccc2c(c1)CCN(c1nccc(N3CCCC3)n1)C2 15819,c1(N2CC(C(N)=O)(CNC(c3c(C)noc3C)=O)C2)ncnc(Cl)c1C 15820,O=C(C1=NOC(CNC(C2CCCS2)=O)C1)NCCC12CC(CO1)C2 15821,c1(CC(N2CC(CCNC(C)=O)C2)=O)c(N)nc(C)nc1O 15822,C(C(C)CC(F)(F)F)NC(C1N(C(CCCOCC(C)C)=O)CSC1)=O 15823,Cc1csc(C(C)C(=O)NC(C)CN(C(=O)Cc2cccnc2)C)n1 15824,N1(C(C(C=C)(C)O)=O)CC2(C1)OC1(C)CC2(NC(c2nn(C)nc2C(F)(F)F)=O)C1 15825,C1(CCCn2cc(NC(CCOC)=O)nn2)CCCC=C1Br 15826,C1(NC(=O)Cc2nncs2)CCN(CC(=O)Nc2ccccc2)C(SC2CC2)C1 15827,c1(C(=O)Nc2cccc(NC(C=Cc3cc(C)no3)=O)c2)ccccc1S(C)(=O)=O 15828,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nonc1N)=O 15829,N1(C(C(=C(C)c2ccco2)CC)=O)CCCC(NC(=O)C(C)(C)CC2CC2)C1 15830,Cc1cc(=NC(=O)C=C2CC(C(=O)Nc3nnc(C#N)s3)C23CCOCC3)[nH]o1 15831,N1(C(c2n(CC)ccc2)=O)CCC(CC(C)NC(=O)COCC2CCOC2)CC1 15832,c1(C(N(C2CCC(NC(C(CCC)OC)=O)CC2)C)=O)cc(OC)cnc1F 15833,Cc1cc(C(=O)N(C(C(=O)NCC2(C)NC(=O)NC2=O)C2CC2)C)nc(O)n1 15834,C1(C2CCN(C(=O)CCc3cccs3)C2)CCCCN1C(=O)CC1CCCOC1 15835,CC1CC(C)N(C(=O)CC(C)(C)C)CCN1C(=O)Cc1nc2cc(Cl)ccc2s1 15836,c1(CNC(C)(C)C)ccc2c(c1)CCC2NC(=O)NCc1cc(C)cc(F)c1 15837,c1(C(=O)NC(CNC(c2c(C)nc(CC)s2)=O)CO)cnc2[nH]cnc2c1 15838,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15839,C12(C(N3CCC(C(C)NC(c4nccc(S)n4)=O)C3)=O)CCC(CC1)OC2.C 15840,C1(NC(c2cc(F)c[nH]2)=O)CC2CC1N(C(c1cnc(O)cc1O)=O)C2 15841,n1(C(CC)CC)nc(CC2CCCCC2)nc1-c1nc(-c2ncccn2)n(C)n1 15842,C1(C(N=c2nc(CCC)[nH]s2)=O)CCN(C(c2ccccc2Cl)=O)CC1(C)C 15843,Cc1cn(C)nc1C(=O)NCC1(F)CN(C(C2CCCC(F)C2)=O)C1 15844,c1(NC(C2N(C(Cc3cccc(OC)n3)=O)CCOC2)=O)ccc2cnoc2c1 15845,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15846,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(c2coc(Cl)n2)=O)CCC1O 15847,c1(C(=O)Nc2c(CC)nnn2C)ccc(C(=O)OC)c(Cl)c1 15848,Cn1ncc2c1CCN(C(C1(C)CCN(C(=O)C(O)CC3CCCC3)C1)=O)C2 15849,c1(C(=O)NCC2C(NC(C3(SC)CCC3)=O)COC2)cc(C)c[nH]1 15850,C1(CN(C(CC)=O)C(C2CCCC2)=O)CC(O)CN1C1CCCC1 15851,C(N=c1[nH]c(NC(N2CCCC2=O)C2CCCCC2)nc2c1SCC2)C1(C)CC1 15852,c1(OCC)nc(NC2C3CN(C(=O)CCN(S(C)(=O)=O)C)CC23)ncc1C 15853,N1(C(C2C(C#N)C2)=O)CCC(C(=O)NCC2CC23CC3(F)F)(CO)CC1 15854,N1(C(C(c2n(C)ncc2)O)=O)CCCC2(CC(NC(=O)C(C)(C)CF)C2)C1 15855,c1(CC(N2CCCC3COCC23)=O)ccc([N+](=O)[O-])cc1 15856,C(C(O)C(=O)NC1CC(CNC(C2(CCN3CCOCC3)CC2)=O)C1)N(C)C 15857,Cc1ccc(SC(C)C(=O)NC2CCC(NC(C3CCC(CO)CC3)=O)C2)cc1 15858,C1(NC(c2c[nH]cc(C)c2=O)=O)CN(C(c2cnc(C#N)s2)=O)C2CCCCC12 15859,N1(C(Cc2c(CC)cccc2)=O)CCC(C2CCN(C(=O)C(F)C(C)C)C2)CC1 15860,C(=O)(C(CCC)S(N)(=O)=O)NC(CCC)CCCNC(=O)Cn1nc(C)c(Cl)c1C 15861,C1(F)(C(=O)NCC(CNC(C2(CC3CCC3)CC2)=O)CO)CCCOC1 15862,c1(C(=O)NC(C(C)NC(=O)C=CC2CC2)CO)cccc2ccncc12 15863,C=CCC(C)(C(=O)N1CC(O)(C2CCCN2C(=O)CCc2ncc[nH]2)C1)N(C)C 15864,N1(C(c2c[nH]ccc2=O)=O)CCC2(CC1)CN(C(C1CCCC1)=O)CCO2 15865,C1(c2n(C(CC)(C)C)nnn2)(NCc2ccc(C(F)(F)F)c(Cl)c2)CN(C)CC1C 15866,c1(NC(C2(O)CCC(CC)C2)=O)ccc(NC(=O)CCCC(C)=O)c(C)c1 15867,N1(CC(=O)NC(C)CC(C)NC(=O)CCc2nc[nH]n2)CCCOC1=O 15868,c1(C(N2CCCC(NC(c3nc(SC)nc(O)c3)=O)C2)=O)ccc(F)c(C#N)c1 15869,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15870,C1(C2(O)CN(C(c3n[nH]cc3C)=O)C2)(CNC(C2CCCC(OC)C2)=O)CC1 15871,c1(C(=O)NC(CC)CNC(C2(CO)CC2)=O)ccc2c(n1)NC(=O)CO2 15872,c1(C(=O)NC2CN(C(C3CCC(F)(F)C3)=O)C2)cnc2cccnc2c1 15873,c1(C(=O)OC)ncnn1C1CCN(Cc2cscc2OC(C)(C)C)C1 15874,C#CCC(C)(C(=O)NCC1CC(CCC)C1)NC(c1nc(C)ccc1C)=O 15875,N1(C(c2cn(CC=C)nn2)=O)CCC(C)C(CNC(c2cn(CC3CC3)nn2)=O)C1 15876,C1(NC(CCCCN(C)C)=O)CCCC12CN(C(C1CN3CCCC1C3)=O)C2 15877,CON1CCC(C(=O)NC2(CNC(=O)CCCC3CCCC(=O)N3)CCC2)CC1 15878,c1(CNC(Cc2nc(CN)sc2)=O)cccc(Oc2ccc(F)cc2)c1 15879,C1(NC(c2ccc(C)cc2N)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)CC1C1CC1 15880,C1(N(C)C(c2ccc(-n3cccc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15881,c1(C(N(C2CCN(C(C(C=C)(C)O)=O)C2)C)=O)csc2cncn12 15882,CCCCCCC(C(=O)NCC(C)C)N1CCN(C(=O)C(CCC)C(C)C)CC1 15883,CC(CC(=O)NC1(C2CCN(Cc3cc(C(C)(C)C)n[nH]3)C2)CC1)C(F)(F)F 15884,CC1CCOC1C(=O)NC1CC1NC(c1cnns1)=O 15885,CN1CCCCC1CC(=O)NCc1ccnc(C(=O)NCCC2CCCN2C)c1 15886,C1(C(N2C(CNC(c3c(C(=O)OC)scc3)=O)CCC2)=O)CC2C=CC1O2 15887,N1(C(C2C(C)C2)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15888,Cc1cc2c(C(=O)N(CCNC(c3csc(C#N)c3)=O)C(C)C)cccc2o1 15889,C(CC1(CO)COc2ccccc21)N(C)Cc1cc2ccccc2oc1=O 15890,O=C1C=C2CN(C(C3CSCCN3Cc3cnc4n3CCOC4)=O)CCC2S1 15891,C1(C)(NC(C(C(C)(C)O)NC(=O)CN2CCNC2=O)=O)CCCC(C)(C)C1 15892,C1(Cn2c(NCC)ccn2)C2CCC(C2)N1C(=O)C(C)SC.C(=O)C(C)(C)C 15893,C1(NC(=O)CCCn2ccnc2)CN(C(=O)Cn2[nH]cnc2=N)CC2(CCC2)C1 15894,C1(C(=O)NCC2(F)CN(C(CC(N3CCCCC3=O)C)=O)C2)CCOCC1(C)C 15895,Cc1nc2cc(F)ccc2cc1C(=O)NC(C)CNC(c1ccnn1C)=O 15896,S(=O)(=O)(c1ccc(NCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 15897,c1(-c2cccc(CN3C(C4C(CO)C4)CCOCC3)c2)c[nH]c2ccc(Cl)cc12 15898,C1(N2C(CNC(c3cc(OC4CCOC4)ncn3)=O)CCC2)CCC(=O)NC1=O 15899,CC1(C)CC(NC(=O)C(C)(C)CCF)CN(C(c2cnc(C3CC3)o2)=O)C1 15900,C1(NC(CCNC(COC)=O)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 15901,N1(C(C2N(C)C(=O)CC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 15902,C(C#CC(F)(F)F)CNC(C(C)SC1CCCN1C(C1(C(N)=O)CC1)=O)=O 15903,N1(C(C2CCC(C)C2)=O)CCC2(CCN(C(C3(O)CCOCC3)=O)CC2)C1 15904,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 15905,Cn1c(C(F)F)nc2cc(C(=O)NC3CCC34CN(C(C3(C)CC3)=O)C4)cnc12 15906,Cc1cc(F)cc2[nH]c(C(N3CCC(N(C)C(c4ccc(F)cc4)=O)C3)=O)cc12 15907,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 15908,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 15909,C1(CCNC(CCCN(C(=O)C(F)C(C)(F)F)C)=O)CCC2(CC1)CC2 15910,c1(CC(N2CC(C(C)NC(c3ccc(Cl)[nH]3)=O)C2)=O)n[nH]c2ccccc12 15911,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ncccn2)cn1 15912,S(=O)(=O)(c1ccccc1)NCC(N1C(C(=O)N(CC2C(C=C)C2)CC)CCC1)=O 15913,NCCC(C(N)=O)NCCCNC(=O)NC1CCN(C(F)(F)F)CC1 15914,C(=O)(C(CC(C)C)NC(=O)CC1CNC(=O)O1)N(C(CC)C1CC1)C 15915,N1(C(C(C=C)(C)CCOC)=O)CC2CCC(C1)C(NC(C1CC(C)(CC)C1)=O)C2 15916,C1(CC(=O)N(C)CC2CCN(C(C(C3CCC3)OC)=O)CC2)CCC(C)(C)CC1 15917,N=c1[nH]c(N2CCC(NCCCOc3ccccc3)C2)nc2ccccc12 15918,N1(C(c2c(C)coc2)=O)CCCCCC(NC(=O)C(c2ccc(F)cc2F)C)C1 15919,C1(C(=O)NCCC2(NC(=O)C=CC3CCOC3)CCCC2)CC12CCOC2 15920,CC(O)C(C)C(=O)NC1CCCCC1NC(=O)CCc1cncc(N(C)C)c1 15921,C1(OC)CCN(C(=NCCSC)NCCSCCC(F)(F)F)C1 15922,C(=O)(CC(C)(O)C(F)(F)F)N(CC(C)NC(CCC(=C)Cl)=O)CC 15923,C1(OC)CC(CCNC(=O)CCCN(C)C)N(C(C2CC2CC(C)C)=O)C1 15924,C1(NC(C(C=C)(C)CC)=O)CCN(C(c2ccc(OCOC)cc2)=O)CC1(C)C 15925,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 15926,c1(C(N2CCCC(CC(N3CCOCC3)=O)C2)=O)noc2c1CC(F)(F)CC2 15927,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 15928,c1(CN(C(CCc2c(C)cccc2)=O)C)ccc(S(=O)(=O)C(F)(F)F)cc1 15929,c1(C(=O)NC2(C(=O)NC(CCSC)CO)CC(CO)C2)cc(C(N)=O)ccn1 15930,N1(C(C2C(C)C2)=O)CCCCC(NC(=O)CCC(=O)NCN2CCCC2=O)C1 15931,c1(C(=O)NC2CC(NC(CC(=O)OC)=O)C(O)C2)ccc2ncncc2c1 15932,n1(CCN(C(=O)CCC(C)(C)F)C)ccc(=NC(=O)CCC2CC3CCC2C3)[nH]1 15933,N=c1cc[nH]cc1CNc1ccccc1C(=O)Nc1cncc(N(C)C)c1 15934,c1(OCC(=O)N(CC(C)(C)NC(C(CCCC)C)=O)C)ccc2c(c1)CCCC2 15935,C(CC(C(=O)N1CCC(CCOC)C1)NC(c1cncn1C)=O)=CC 15936,CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CN(C)CCC1O 15937,c1(C(=O)NCC2(COC)CCCN2C(c2scnc2Cl)=O)cc2ccccn2n1 15938,S(=O)(=O)(c1cccc(N(CC=C(Cl)Cl)Cc2ccccc2)c1)N1CC(C)OCC1 15939,C(=O)(CS(N)(=O)=O)NC1CC(CCNC(C(CC2CCC2)OC)=O)C1 15940,c1(C(N2CC(C)CC(NC(CC3(OC)CC3)=O)C2)=O)cc2n(n1)CCCN2 15941,C1(NC(C(C)(C)SC)=O)CCC(C)N(C(=O)C=CC(C)=O)C1 15942,C1(C(N2CC(CNC(c3ccn(CCF)n3)=O)C2)=O)(CC)CCOC1 15943,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnnc3)C2)C(C(F)(F)F)C1 15944,C12(C(=O)NC3CC(NC(C4CCCS4)=O)C3)CCC(O)C1CC2 15945,C1(CN(C(=O)CC2(O)CC2)C)CN(C(=O)CCc2ccc[nH]2)CC12CC2 15946,CC1CCC(C(N)=O)CN1C(C1(C)CC1C(F)(F)F)=O 15947,C(c1cccc(Cl)c1)=CC(=O)NC1CC1.CC1(F)CNC(=O)CC(=O)NC1 15948,C1(c2c(OC)cccc2)CCN(C(c2ncc(Cl)n2C)C(=O)NC2CC2)C1(C)C 15949,CC(C)(C)C(C(=O)N1CCC(O)CC1C1(CN)CC1)c1cc(F)cc(F)c1 15950,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 15951,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CCC2)=O)c1O 15952,N(C(=NCC1CCC(=O)NC1)NCc1ncccc1C(N)=O)C(CC)C 15953,C1(NC(=O)COc2ccc(Br)cc2Cl)CCCN(CCO)C1=O 15954,C1(CC(=O)OCC)CCCN1C(=O)C(C)NC(C1(COC)CCCC1)=O 15955,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(CO)nc2)=O)CC1)CCC 15956,N1(C(c2nc(C#C)sc2)=O)CCC2(CCN(C(=O)C(C)NC(=O)COC)C2)C1 15957,Cc1cc(C(=O)NC(C2(C(=O)NCC3C4CCCCC34)CC2)C)sc1C 15958,CC1CC(NC(=O)C(C)CCCO)CCN1C(c1ccc(OCC2CC2)nc1)=O 15959,c1(C(=O)NC(CC(C)NC(C(CN(CC)CC)F)=O)C)cc(S(N)(=O)=O)sc1C 15960,N1(C(C2CC(C)N2C(c2ccc3[nH]ccc3c2)=O)=O)CC2(CCN(C)CC2)C1 15961,C(CCC(=O)NCCC(C)NC(=O)C(C)OCCC(C)C)=CCC=C 15962,C1(CNC(N(CC)CC)=O)CC2CCCN2C1.c12cc(Br)c(o1)CCNC2=O 15963,CC(C)C(C(=O)NC(C)CCN(C)C)NC(C1(CO)CC(C)(C)C1)=O 15964,CC1C(NC(=O)Cc2cnccc2Cl)CCCN1C(c1c[nH]nc1C(C)(C)C)=O 15965,c1(C(=O)NCC2CCN(C(C(C)C3CC3)=O)C23CC3)cccc2ncnc(O)c12 15966,C1(CNC(C2CCN(C)C2)=O)CN(C(c2ccc(Br)nc2O)=O)CC1(F)F 15967,[N-]=[N+]=NC1CN(C(C2C3CC4C(C3=O)C24)=O)CC1CNC(c1sccc1F)=O 15968,N1(CC)CCC(N=c2[nH]c(N3CC4CCC3C4)nc3cccc(F)c23)C1 15969,C1(CNC(CC(C)F)=O)CN(C(=O)C=CC2CC2)C2COCC2O1 15970,C=CCCN=C(NCCC(C)F)NC1CCOC(C(C)C)C1 15971,c1(NC(C)=O)ccc(C(=O)NC2CC2NC(=O)CCc2cnc(C)nc2O)c(Cl)c1 15972,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(C1(CO)CCOCC1)=O)CO2 15973,c1(C(=O)OC)nc(C(=O)N(C)Cc2csc(C3CC3)n2)cs1 15974,CN1CCN(C(=O)C2=NOC(CNC(=O)CN3CC(=O)NC3=O)C2)CCC1=O 15975,C(=O)(C1CCSc2ccccc21)NCCN(c1nc(NC)nc(C)c1I)CCC 15976,CN1CC(O)CC1C(=O)NCCN(C(=O)CCCc1ccsc1)C 15977,CC1(C)CCC(CC(=O)NC2CN(C(=O)COc3ccc(F)cn3)C2)CC1 15978,C=C=CC(C)C(=O)NCc1c[nH]nc1C(=O)NCCOC1CCCC1 15979,Cc1cc(CC=O)c(C)s1.C(=O)(CCCNS(C)(=O)=O)NC(CC1CNC1)C 15980,c1(CCC)cccc(C(=O)NC2(CNC(c3cc(OC)nn3C)=O)CC2)c1 15981,c1(C(=O)NCC(CNC(c2c(C)n(C(C)C)nc2)=O)C)cc(S(N)(=O)=O)cn1C 15982,c1(C(=O)NC2CCCC(N(C(CC=CC)=O)C)C2)c(F)cc(OC)cc1Cl 15983,C1(NC(CCSCCC)=O)CC(O)CN(C(c2cnc(CC)s2)=O)C1 15984,C(=O)(C1CCc2c(Cl)cccc21)N1CCC(CN(C(C2CCC(C)CC2)=O)C)C1 15985,C(=O)(CC(=O)NC1CCC1NC(c1nnc(C(C)C)s1)=O)NC 15986,c1(-c2cn(CC3N(C(C4(C#N)C(C)C4)=O)CCC3)nn2)ncn2ccccc12 15987,C1(NC(CC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1Cl 15988,C1(C(N2CC(NC(=O)OC)C2)=O)CN(C(=O)C(C)(C)N(C)C)CC1F 15989,C12(C(=O)NC(CCO)C3CCCC3)CC(CCO1)N(C(C13CC(C1)C3)=O)C2 15990,CC(CC(N)=O)C(=O)N1CC(CNC(c2cnn(CCC(F)(F)F)c2)=O)C(O)C1 15991,c1(C(=O)OCCNC(C2CC(C)OC2=O)=O)cccc(OCC2(C(C)C)CC2)c1 15992,c1(C(=O)NC(C2CN(C(c3sccc3Cl)=O)C2)C)ncoc1C1CCCCC1 15993,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)CC1O 15994,Cn1cc(C(=O)NC2COCC2CNC(=O)CCc2cn[nH]c2)c(C2CC2)n1 15995,CC1=C(C(=O)NC2CCN(C(=O)C(C)OCCC(C)C)C(C(C)C)C2)CCC1 15996,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 15997,C1(N(C(Cc2cn(CC)nn2)=O)C)CCN(C(c2ccnc(OC)n2)=O)CC1C 15998,c1(CC)cccc(-n2nc(-c3nccs3)nc2-c2coc(CN(C)C)c2)c1 15999,CCCCS(=O)(=O)NCC(=O)NCC1CCN(C(C(=O)NC)(C)CSC)C1 16000,CC1=C(C(=O)N(CCCNC(c2cnccc2OC(C)C)=O)C)CCC1 16001,N1(C(C=C(C)CN(C)C)=O)C2CCC1CC(C(=O)Nc1cnc(C)nc1C)C2 16002,CC1(NC(C2CC(NC(=O)NCc3ccccc3)C2)=O)CCC(=O)NC1=O 16003,C(CNC(=O)CCn1ccnc1C)(CC(C)C)NC(C1C(CCC)C1)=O 16004,O=C(CC(O)CNC(C1CC12CC2)=O)NC1CCC(O)C1 16005,c1(C(N(CCN(C(C2CCC(C)O2)=O)C)C)=O)csc2ccccc12 16006,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)COC3)=O)CC2)C1 16007,c1(C(=O)NC2CC(CCNC(=O)CC3CC4CCC3C4)C2)cccc2sncc12 16008,C1(NC(c2c[nH]c(Br)c2)=O)CN(C(=O)C(F)=CC2CC2)C2CCCCC12 16009,C1(NCC(=O)Nc2c(C)scc2)CC2(C1)CN(C(=O)C(C)Cc1ccco1)C2 16010,Cc1cc(C(=O)NC2CN(C(C3CCS(=O)CC3)=O)CC2C)n2nc(C)cc2n1 16011,C(=O)(C(F)(F)C(C)O)NC1(C)CC(NC(C(CCC)O)=O)C1OC 16012,C1(NC(c2cc(C)cc(C)c2)=O)CN(C(c2ccc(O)cc2F)=O)C2CCCC12 16013,CS(=O)(=O)c1ccc(C(=O)NCC2CCCCN2C(=O)C(c2ccccn2)O)o1 16014,CCCCCC(O)CC(=O)NC(c1cn(C)nn1)CNC(c1cc(Cl)c[nH]1)=O 16015,c1(SCC(=O)NC2C(C)CN(C(=O)C(C3CC3)C3CC3)CC2)ccc2c(c1)CCC2 16016,C1(NC(C(C2CCN(C(c3c(C)[nH]cc3)=O)C2)C)=O)CCOC(C(C)C)C1 16017,C(CC1CC1)(C(=O)NOCCn1ccnc1)NC(C1CC2CCC1O2)=O 16018,C(=O)(C(CC)(CC)OC)N1CCC(N(C(c2cc(C3(C)CC3)on2)=O)CC)C1 16019,N1(C(CCNC(COC)=O)=O)CCC(O)(CNC(=O)CNC(=O)CC(C)(C)C)C1 16020,N1(C(C=CCOCCOC)=O)CC2CC(O)C1C2NC(C1CC(n2ccnn2)C1)=O 16021,C(=O)(C1=NNC(=O)C1)N1CC(CCCNC(C(C(C)C)OC)=O)OCC1 16022,c1(C(=O)NCC2(C(=O)NCc3ncc(C)nc3)CC2)cccc(O)c1C 16023,CC(C)CCC(=O)C(=O)N1CCC(C(C)C(c2cc(C(C)(F)F)ncn2)=O)CC1 16024,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(N)(=O)=O)c(C)s1 16025,C1(NC(CC2(C(=O)OCC)CCCC2)=O)CCN(C(c2cnsn2)=O)C(C)C1 16026,Cc1ccc(CN(C)CC2CCCN(C(=O)C=Cc3ccn(C)c3)C2)cc1 16027,c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)CO)cc(N)c(Cl)c(O)n1 16028,CCC(CC)CCC(=O)NCC1CC2CCCC2N1C(=O)CS(=O)C(F)(F)F 16029,C1(C(=O)NC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16030,C1(NC(C(CC)SCc2ccccc2)=O)CN(C)CCN1C(C1C(C)CC1C)=O 16031,C1(SC)CCN(C(=O)CONC(=O)C=Cc2ccoc2)CC1O 16032,CCCCCCCCNC(=O)C(=O)NC(C)CNC(=O)CC1CC(SC)C1 16033,c1(CCNC(c2n(C)cnc2Br)=O)nc2c(o1)CCSC2 16034,C1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)CCn2ccnc2C1 16035,c1(C(COC)NC(=O)C(c2ccnn2C)O)ccccc1F 16036,C1(CC(C)NC(c2cc3ncccc3o2)=O)CC2CCC(C1)N2C(=O)CCF 16037,N1CCC(C)CC1C(=O)NC(COC)C(C)C.C1(CC=O)(CC)CCC1 16038,C(C1CCc2nccn21)NC(C(CC(=C)C)ONC(=O)C(F)=C(C)C)=O 16039,c1(C(=O)NC2C(CNC(C=CCCC)=O)C2)cn(C)nc1-c1ccnn1C 16040,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16041,C1(CN(C(=O)C(C)(C)c2cncs2)C)CCCN1C(=O)CCn1ccnc1 16042,c1(C(N(C(C(=O)NCCC2CCCC2)C2CCCO2)C(C)=O)C)ccc(C)cn1 16043,Cn1ccc2c(C(N3CCN(C(=O)CC(C)(C)C(=O)OC)C(CF)C3)=O)cccc12 16044,C1(C(C)C)CN(C(=O)C(C)CN2CCCCC2)CCN1C(=O)CCCCC1CC1 16045,n1(CCNC(C23CC(C)C2C3)C)cc(C(F)(F)COC(C)=O)cn1 16046,C1(NC(=O)CC2CC2(Cl)Cl)CN(C(c2cccc(OC3CCC3)c2)=O)CC1F 16047,C12(C(=O)NC(CNC(c3ccco3)=O)CO)CC(=O)C1C2 16048,N1(C(C(CC)(C)C)=O)CCN(C(c2cc(C)n(C)n2)=O)C(CC(C)(C)C)C1 16049,c1(OC)cc(C(=O)N(C)CC2CN(C(=O)C(C)C(C)O)CC23CC3)nnc1C1CC1 16050,C(=O)(C(C)(C)C(=O)NC(C1(O)CCN(C(C2CCCCC2O)=O)C1)C)OC 16051,C(c1ccc(F)c2ccccc12)=C(C(=O)N(C1CC1C)CCOCC)C#N 16052,C12(CNC(CCCCN(C(=O)C(=O)NS(C)(=O)=O)C)=O)CCCN1CCC2 16053,C(CCCCCNC(=O)C(=O)NCC(F)(F)F)NC(CNC(C)=O)=O 16054,c1(C(=O)NC(C2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)C)cc(F)cc(F)c1N 16055,CS(=O)CCC(=O)NC(CNC(=O)CCSc1ccccc1)C1CC1.C1(C=O)CCC1 16056,CC(C)CCCC(C)C(=O)N1CC2(CC(C(=O)NC3(C)CCCC3(F)F)CO2)C1 16057,C(=O)(CCS(N)(=O)=O)N(CCCNC(c1cnc(C2CCC2)o1)=O)C(C)C 16058,c1(NC(C(C2CN(C(c3cc(CCC)[nH]n3)=O)C2)O)=O)ccc(C)c(C)c1 16059,c1(C(=O)NC2CC2NC(c2cnsn2)=O)cccc(-c2nc(=O)o[nH]2)c1 16060,C1(C(=O)NCc2cn(CC)nc2)(CNC(c2sc(F)cc2C)=O)CCCCC1 16061,CC1CC(C(=O)NC(C(=O)Nc2cncc(C3CC3)c2)c2ccco2)=NO1 16062,CC(C)(C)C(C(=O)NCCc1nc[nH]n1)NC(c1ccnnc1)=O 16063,c1(C(N(C2CCC(NC(C3CC34CC(O)C4)=O)CC2)C)=O)ccc2[nH]ccc2c1 16064,CC1CCCN1CC(N1CCC(n2cc(C3(O)CC(C(F)(F)F)C3)nn2)C1)=O 16065,n1(CC(=O)NCCC2N(C(c3ccc(OC)s3)=O)CCC2)cc2ccccc2n1 16066,c1(C(C)C)cccnc1NC1CC(C)N(C(c2ccc(Br)o2)=O)C1 16067,n1(CCC)nc(C)cc1C(=O)N(CCCN(C(=O)C(C)CC)C)C 16068,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16069,Cn1cc(C(=O)NC2CCCCC2NC(c2nccs2)=O)c2ccccc12 16070,c1(CC)ccc(OC2(COCC(=O)OC)CN(C(C3C=CC=CC=C3)=O)C2)cc1 16071,c1(C(N2CCCC(N(C)C(C3CCS(=O)(=O)N3)=O)CC2)=O)ccc2nc[nH]c2n1 16072,CC1(C)CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)CNc1ccc(O)cc1 16073,C1(C(=O)OC)CCCC12CCCN(CC1CC3(CC3)CN1)C2 16074,C#CCC(C(=O)N1CCCC1(C)CCCNC(=O)CC1(N(C)C)CCC1)C1CC1 16075,c1(C(N2CCOC(CCO)C2)C(=O)NC(C(=O)OC)C)ccncc1Cl 16076,C1(CNC(C2C(C)=C2)=O)CCC2(CCN(C(c3cccc(N)c3C)=O)CC2)O1 16077,CC(C)CC(C(=O)NC(=O)NC1CCC1Oc1ccc(F)cc1F)N(C)C 16078,c1(CC23OCC(CNC(C=C(C)C(C)C)=O)(C2)C3)ncnc2cccc([N+](=O)[O-])c12 16079,CC(C(=O)NC(CNC(c1ccc(C2CC2)o1)=O)CCO)C(C)(C)C 16080,C(CC(F)(F)CO)NC(C1CC=CCN1C(C1CC(O)C(F)C1)=O)=O 16081,C1(C(C(=O)NC(CCCC)C)N(CCOC)CC2CCCO2)CCCCCC1 16082,c1(C(N2C(C)(C)CC(NC(C3CC(C)(C)CO3)=O)C2)=O)cc2ccccn2n1 16083,N1(CCCC)CCCCC1C(N1CC(NC(c2cc(C)on2)=O)CC1C)=O 16084,CC(O)C(=O)N1CC(N(C(C2CCCO2)=O)CC2CC2)C1 16085,c1(C(N2CCCC(C(N(C)Cc3c(C)occ3)=O)C2)=O)cc2ncccc2[nH]1 16086,n1(CC)nnnc1C1C(C2CC2)C(=O)O1.C(CN)(CCOC)NCC 16087,C(=O)(CC(C)C(=O)NCC1CC(C)CN1C(=O)COCCCN=[N+]=[N-])OC 16088,c1(C(C(N2CC(O)(CNC(C(C)N3CCC3)=O)C2)=O)O)ccc(Cl)cc1Cl 16089,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CC(c1c(C)ccc(F)c1)O 16090,C1(C)(C(=O)NC(CCCNC(c2c(CC)n(C)nn2)=O)C)CC2(C1)CC2(F)F 16091,c1(NC(=O)OC)ccc(F)c(C(=O)NCCC2CCN2C(=O)NCC2CC2)c1F 16092,c1(C(=O)NCC23OCC(NC(C4C(=C)CC4)=O)(C2)C3)cc([N+](=O)[O-])ccc1Cl 16093,C(=O)(CC1OCCc2ccccc21)NC(=O)NC(C)CN1CC=CC1 16094,N1(C(C=CC(C)NC(C2CCC(C3CC3)C2)=O)=O)CCCCCCCC1 16095,C1(CC(=O)N(C(CN(C(C(C)NC(COC)=O)=O)C)C)C)COCC(C)(C)O1 16096,C1(NC(c2cnn(CCO)c2)=O)CN(C(=O)CC2OCCCO2)C2(CCCC2)C1 16097,C(=O)(C#CC1CCCOC1)N1CCOCC(C)(Cn2cc(C(C)(C)C)nn2)C1 16098,N1(C(C2CC(=C)C2)=O)CC2C3CCC(C2C1)N(C(=O)COc1ccc(Cl)cc1)C3 16099,N1(C(C(c2ccn(C)n2)(C)C)=O)CCC12CN(C(C1CC1(C)Br)=O)C2 16100,C1(NC(C2(OC)CC2)=O)COCCC1NC(c1scc(C)c1C(=O)OC)=O 16101,n1(CC)c(C)cc(C(=O)NC2CC(NC(c3sccc3COC)=O)C2)c1C 16102,C(=O)(CCCC(C)C)N(C(C(CC)O)=O)C1CCC(N2CCCC2)C1 16103,N1(C(C(C)OCCCC)=O)CC2(NC(=O)CCn3c(C)csc3=O)CCC1C2 16104,C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2c(C)nn(C)c2C)=O)C(CF)C1 16105,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CNC(=O)CCCc2csc(=N)[nH]2)C1 16106,c1(C(=O)NC2CCCN(C(=O)C=Cc3cnccn3)C2)cccc2nc(Cl)sc12 16107,c1(C(CC(=O)N2CC(NC(C3C(CCC)C3)=O)C2)C)ccc(F)c(F)c1 16108,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16109,N1(C(c2snc(C(=O)OCC)n2)C)CCC(=O)N(C)CC1 16110,Cc1noc(C)c1C(C)C(N1CCN(CCCNC(C2CCC2)=O)CC1)=O 16111,N1(C(C(CCC)OC)=O)C2CCC1CC(CN(C(=O)C(C)=C1CC1)C)C2 16112,O=c1c(C(F)(F)F)c[nH]c2ccccc12.c12ccccc1-c1cn(nn1)CCO2 16113,CC1CCN(C(C2(c3ccccn3)CC2)=O)C1CNC(=O)C=Cc1ccncn1 16114,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC)CCC1C 16115,C1(N(C(C(C)OC(C(c2ccc(C)cc2)OC)=O)=O)C)CCN(C)C1(C)C 16116,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16117,C(C)(C(=O)NNC(=O)C12CNCC1C2)OCC(=O)OC 16118,N1(C(C(CCC)O)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC1c1ccc(F)cc1 16119,Cc1cnc(C(=O)NCC(F)CNC(c2cn3ccnc3s2)=O)c(C)c1 16120,C1(NC(CCc2n(C)c(S)nn2)=O)CCN(C(=O)C2=CCOC2)C12CC2 16121,N1(C(C(C)C2(O)CCC2)=O)CCCOC(CNC(=O)CC(O)C2CCCC2)C1 16122,C1(C(N(C)CC2CC(=C)C2)=O)CCN(C(=O)CCCCOCCC)C1CC 16123,C=CCC(CNC(=O)C(C)N=[N+]=[N-])C(=O)NC(c1nnc(C)o1)C 16124,N1(C(C(c2ccccc2F)C)=O)CC2C(NC(C3CC3C(C)O)=O)C2C1 16125,C1(CNC(C(c2ccc(CC)s2)=O)=O)CCCCN1C(=O)CCN1CCCC1 16126,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(C1CCCOCC1)=O 16127,c12ccc(cc1Cl)NC(=O)C(=O)NCC2.Cc1cnccc1C(C)OC1CCCC1 16128,C(CC(N)=O)(C(=O)NC(CC=C)C(=O)OC)NC(c1ccc(C#C)o1)=O 16129,C1(c2n(CCCC)nc(C)c2)NC(=O)N(CC2CCCO2)C2=C1C(=O)NC2(C)C 16130,N1(C(=O)C=CC2CCCO2)CC(NC(C2CCCCCC2)=O)CC2(CCC2)C1 16131,c1(SC)cccc(NC(=O)Cc2csc(Cl)c2)c1 16132,N1(C(C(F)=CCC)=O)CCC2C(CCCN2C(=O)CC2CCCCN2C)C1 16133,C1(SCC)CC(C)=NO1.C1C(=O)NCC=CC(=O)N1CCO 16134,N1(C(C(C)Cc2ccco2)=O)CCC2CN(C(c3cc(F)ccc3Cl)=O)CC2C1 16135,C(C(O)(CNC(=O)CNC(=O)CCn1ccnc1C)CO)OC 16136,Cc1ncc(C(N2CC=C(CNC(C3CCC4C3C4(F)F)=O)CC2)=O)cc1C#N 16137,c1(NCC(C)N(C(=O)C#CC2CCCCC2)C)cccc(SC)c1[N+](=O)[O-] 16138,N1(CCC(N2C(CNC(Cn3c(=N)scc3)=O)CC2)=O)CCN(CC2CC2)CC1 16139,c1(COC(C(=O)NCC(C)CN(C)C)C2CCCO2)ccccc1 16140,C1(NC(C#CC(C)C)=O)CN(C(=O)C(C2CCOCC2)F)CC12CCOCC2 16141,C(CC(C)C(=O)N1CC(C)(NC(C2(C(=O)OC(C)C)CC2)=O)C1)SC 16142,C=CC1(C(=O)N(CC)CC2CCOC2)CCN(C(c2ccccc2CC#N)=O)C1 16143,N(C1CCCc2occc21)C(C(CC(C)C)NC(C1CCC(=O)O1)=O)=O 16144,c1(OC(F)(F)F)cc(C(=O)NCC(C2CC2)OC)ccc1F.C1(=O)CC(C)O1 16145,Cc1cc(C)n(C(C)C(=O)N(C2CC(NC(C3CCC(F)(F)C3)=O)C2)C)n1 16146,c1(NC(C)=O)cc(F)ccc1C(=O)NC1CCCC(NC(=O)Cn2ccnn2)C1 16147,N1(C(C2CN(C(C)(C)C)C2)=O)CCN(C(=O)CC2(C(F)(F)F)CCC2)C(CF)C1 16148,Cc1ccc(C)c(OCC(N2CC(NC(=O)C(F)(F)CO)OC(C(F)(F)F)C2)=O)c1 16149,Cc1cc(N(C)Cc2cc(C#N)cs2)nc(=NCCc2ccc(CO)cc2)[nH]1 16150,c1(C(=O)NC2C(C)CN(C(c3ccnc(F)c3)=O)CC2)cc2c(F)cccc2[nH]1 16151,c1(-c2ccc(C(=O)NCc3cncs3)cc2)cc[nH]c(=O)c1CCO 16152,N1(C(C(C2CCN(C(C(C)SC)=O)C2)F)=O)CCC(C)(C)C(CO)C1 16153,c1(C(N(CCNC(=O)C(C)=C2CCCC2)CC)=O)ccc(F)nc1 16154,C12(NC(CC3(CSC)CC3)=O)CCCC1N(C(c1cn(C)nc1SC)=O)CCC2 16155,c1(CC)cccc(C(N2CC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)c1 16156,C1(C(C)NC(C(C)=C(CC)C)=O)CCCN1C(=O)CCNC(N)=O 16157,CC1CCN(C(c2cn(C)nc2C(C)(C)C)=O)CCN1C(C1CNC(=O)C1)=O 16158,CC1CC(CNC(c2cn(Cc3ccccc3)nn2)=O)CN1C(=O)CNC(=N)N 16159,c1(CNC2CCC(NC(c3cnc(O)[nH]3)=O)C2)ccc(F)cn1 16160,N1(C(CN(C(C)=O)C)=O)CCC(F)(C(=O)NC2CCCC2CF)CC1 16161,c1(C(=O)NCC2(C)CC(NC(C3N(C(=O)OC)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16162,c1(Cn2cc(CNC(C3CC(OC)C34CCC4)=O)nn2)c(F)cc(F)cc1F 16163,C1(NC(C(C)n2cccn2)=O)CN(Cc2ccccc2CCBr)CC1C#N 16164,c1(C(N2CC(C)C(NC(=O)Cc3ccc(Cl)cc3)C2)=O)cnc2cc[nH]c2c1 16165,N1(C(C)=O)CCCc2cc(Br)c(NC(CC)CCCC(=O)NCC)cc21 16166,C1(NC(C(C)SC)=O)CCN(C(c2ccc(OCCOC)cc2)=O)C1C 16167,C#Cc1ccc(C(N2CCN(C(=O)Cc3cn[nH]c3)CC(O)C2)=O)c(F)c1Cl 16168,c1(C(=O)NCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CCCC2)cc(O)cc(=O)o1 16169,C1(CC(=O)NCCN(C(=O)CC(C)(C)C2CC2)CCC)CC(O)C1(C)C 16170,CC1(C)CCN(C(=O)CCC)CC1C(N1CCCCC1CC(N)=O)=O.C(C(N)=O)S 16171,CCCCCC(C(=O)N(C(C)CNC(=O)CCCc1ccccc1)C)C(C)C 16172,N1(C(C2CN(C(C(CCC)=CCC)=O)CC(C)C2)=O)CCC(=O)N(C)CC1 16173,C(C(CC(C)C)C(=O)N1Cc2cncnc2C1)NC(C1(COC)CCOC1)=O 16174,c1(C(=O)OCC)cc(=NC(=O)C2(c3nccc(=N)[nH]3)CCC2)[nH][nH]1 16175,c1(C(=O)NC23CC(CNC(C(C)N(CC(F)(F)F)C)=O)(C2)C3)snc2ccccc12 16176,C1(NC(c2c(C)ncnc2)=O)CC2CC1N(C(c1ccc(F)cc1Br)=O)C2 16177,c1(C(=O)NCC2C(NC(c3cc(CCOC)on3)=O)C2)cccc(F)c1C 16178,C=Cc1cccc(C(N2CCC3(CC3C(=O)NCCc3ccnc(O)c3)C2)=O)c1 16179,C1(CCC)CN(C(c2ncccc2Br)=O)CC1NC(C1COC(=O)C1)=O 16180,c1(N2C(CNC(=O)Cc3ccc(F)cn3)CCCC2)nc(C2CC2)nc(Cl)c1C 16181,C1(NC(N2CC(CCNC(CCOC)=O)C2)=O)CCCC1O 16182,C(=O)(C(C)CC(F)(F)F)NC1CN(C(c2cc(C)cc(N)c2)=O)C1 16183,CCS(=O)CC(=O)N1CC(CNC(c2ccnn2C2CCCCC2)=O)C(C)C1 16184,N(C)(C1CCCCCc2ccccc21)c1cc(NCC(C)F)nc(C(C)C)n1 16185,N1(C(C(C)CF)=O)CCC2CCN(C(=O)CSC(F)(F)F)CC2C1 16186,c1(NC(C2N(C(C3(CC)COC3)=O)C3C(C2)C3)=O)ccc(Cl)cc1C 16187,c1(C(=O)NCCC2N(C(CCCCOC)=O)CCCC2)cnc(N)c(Cl)c1 16188,C1(CNC(=O)N(C2CCN(CC#C)CC2)C2CC2)CCC=CCCC1 16189,C(CCC(=O)NNC(=O)c1ccc(F)cc1Br)OC 16190,c1(COC2CC(NCC(C3CC3)OC)C2)cnc(OC)nc1 16191,c1(N2C(C)CC(NC(C3CC(F)(F)C3)=O)C2)ncnc2sc3c(c12)CCC(C)C3 16192,Cn1nncc1CC(=O)NC1(C)CN(CCC(=O)NCC(O)COC(C)C)C1 16193,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16194,c1(OCC)cccc2[nH]cc(CC(=O)N(C(=O)NC3(O)CN(C(=O)CO)C3)C)c12 16195,C1(C(=O)NC2(CF)CCN(C(c3c(C)nsc3N)=O)C2)CCc2ncncc2C1 16196,C1(NC(c2c(C)cc(Br)o2)=O)CN(C(C2CC2F)=O)CC1S(C)(=O)=O 16197,C1(C(=O)NC(C2CN(C(c3csc(CO)n3)=O)CCO2)C)CCC(N=[N+]=[N-])CC1 16198,C1(C2CN(C(C3CC(=O)C3)=O)C2)(SCC)CC1.c12ccc(cc1)C(=O)NC2(C)C 16199,c1(C(=O)NC(CNC(=O)Cc2cnccc2Cl)CO)cc(Cl)c([N+](=O)[O-])[nH]1 16200,N1(C(Cc2n(C)nnc2)=O)CCN(C(c2nn(C)cc2Cl)=O)C(CS(C)(=O)=O)C1 16201,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(O)CC1 16202,CCCCC(C(=O)N1CCC(N(C(=O)CSc2cc(F)ccc2F)C)C1)C(C)C 16203,N1(CC(=O)N(C(C(=O)N(CCC2CC2)CC)C2(C)CC2)C)CCNC(=O)C1 16204,C1(C(=O)OC)CC12CCN(c1nnc(-c3ccc(C)o3)n1CC(C)C)CC2 16205,N1(C(C(C#N)C2CC2)=O)CCC2(CCC2)C(CNC(C2CCC23CCC3)=O)C1 16206,c1(CC(=O)NC(C(C)NC(COCC#C)=O)C)nc(C)sc1C 16207,C(=O)(CC(C)C(F)(F)F)N(C(C(=O)N(CC(C)C)CCO)C)C1CC1 16208,c1(CC(=O)NC(CNC(C(C)OCCOCC)=O)C)cc(N)c(O)c(F)c1 16209,Cc1cnc(C(N2CCC(CCNC(c3cnc(N)c(Cl)c3)=O)C2)=O)cc1Cl 16210,C1(C2CC2)(NC(CCCC)=O)CCN(C(c2ccc(-n3ccnc3C)cc2)=O)C1 16211,c1(C(=O)NCC2(F)CCN(C(CC(C)N(C)C)=O)C2)cnc2[nH]nc(O)c2c1 16212,N1(C(=O)CCC2CCOCC2)CC2=C(C1)CN(C(c1cnc3ccnn3c1)=O)C2 16213,O=C(CC(F)(F)C(F)(F)F)NC1CCC2(CC1)CN(C(c1ccccc1O)=O)C2 16214,C1(CC(=O)NC(C2CC=CC2)C)CC(F)CN1C(=O)Cc1csnn1 16215,C(=O)(CCC(CC)NC(C1C(C)C1C)=O)NC(C#C)CC1CCCC1 16216,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16217,C1(C(N2CC(OC(CC)=O)CC2=O)=O)CCCN(c2nncs2)C1C 16218,C1(CNC(CCSCCCC)=O)CC(C)CN(C(=O)C(F)C2CCOC2)C1 16219,CC1=C(C(=O)NC2CCCC(NC(c3c(N)cnn3C)=O)CC2)CCCC1 16220,C1(CC(=O)NC(C2N(C(Cc3c(C)n[nH]c3)=O)CCC2)C)Cc2ccccc2N1 16221,C1(C(=O)NC(CCNC(c2ccc(C(C)=O)c(F)c2)=O)C)CC2(C1)CC1(CC1)C2 16222,C1(CNC(c2ccc(N(C)C)cn2)=O)CCCCN(C(C2CCCC(O)C2)=O)C1 16223,c1(NC(C2CCN(C(C3C(=C)C3)=O)C(CC)C2)=O)cccc2cnccc12 16224,c1(C(CNC(C(CC)CCCCCC)=O)(F)F)ccc(F)cc1F 16225,C(CS(=O)(=O)N=S(C)(C)=O)OCCCC 16226,C1(C)(CNC(CN2C(C)CC2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)C(C)(C)C1 16227,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CC3CCCCO3)C2)C1 16228,C(C)(CNC(=O)C(C)(C)CF)(C(C)C)NC(CCn1ccc(C)n1)=O 16229,C(=O)(C(F)C(C)(F)F)N1C(C(N(CC(C(=O)NC)C)C)=O)CCC12CC2 16230,c1(OC)ccc(C)c(NC(c2ncncc2-c2ccc(O)cc2SC)=O)n1 16231,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)C(C1CC1)N(C)C 16232,CC(=O)CCCCC(=O)N1CCC(NC(=O)CC(=O)OC(C)(C)C)CC(O)C1 16233,N1(C(CC2CC(C)(C)C2)=O)CCC2CC1CN(C(=O)C(C)(C)F)C2 16234,S(=O)(=O)(c1cccc(C(N2CCS(=O)(=O)CC2CCO)=O)c1)NC(C)CC1CC1 16235,c1(C(=O)NC2CN(C(C3CC34CC4)=O)CCC2F)cc2ccnc(Cl)c2s1 16236,c1(C=O)ccc(C2=CCN(N(C)C)CC2)cc1.C1CC1 16237,c1(C(=O)NC2CCCC2C)ccccc1C=C1CN(C)C1=O.CC(C)CCO 16238,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16239,C1(CC(=O)N(C2CC(NC(=O)CCOc3cccnc3)C2)C)OC(C)(C)OC1=O 16240,N1(CCN(C(=O)C(F)=C2CCCC2)C)CCN(C(C2CC(CF)C2)=O)CC1 16241,Cc1cc2ccc(C(N3CCC(F)(F)C(C(=O)NCCSC4CC4)C3)=O)cc2o1 16242,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16243,N1(C(CCCC=C)=O)CCN(C(C2CC(=O)CCO2)=O)C2COCC12 16244,C(=O)(C(F)(F)C(O)C(C)C)NC1CC(NC(c2cccc(SC)c2)=O)C12CCC2 16245,C1(NC(CNC(=O)NC)=O)CCCC1O.c1(CNC(=O)C2CC2)ccc(CO)nc1 16246,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16247,c1(C(N(C2CCN(C(C34CC3C4)=O)C2)CC)=O)cccc(CSC)n1 16248,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OC(C)(C)C)C2)=O)c1O 16249,c1(C(=O)NC2(CC=C)CN(C(=O)C#CC3CCCO3)C2)cccc2c1OCCC2 16250,N1(CCC(C)=O)CCC2C(CCCN2C(=O)CSSC)C1 16251,C(CC(C)n1cccn1)N(C)C 16252,C1(NCc2nc(C)sc2)CC2(CCN(C(c3cc(N)nc(Cl)c3)=O)CC2)C1 16253,C1(O)(CCNC(Cc2ccc(OC)cc2)=O)CCN(C(=O)Cc2cnns2)CC1 16254,c1(OCCOC)ccnc(N2CCC(CNC(c3cnnn3C)=O)(OC)C2)n1 16255,N1(CC(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC=C2)CCCCS1(=O)=O 16256,N1(C(c2nccc(SC)n2)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)COC)C2 16257,C(=O)(NN1CCCC(C(=O)OCC)C1)C1CCCN(C(CCC(=C)C)=O)CC1 16258,n1(CC)cc(Cl)c(C(=O)NCC(C)N(C(=O)CC(CC)C2CC2)C)n1 16259,C1(C(=O)NCC23CC(CNC(c4n(C)cnc4)=O)(OC2)C3)CC12CCC(=O)CC2 16260,C1(C(C)C(=O)N(C2(C)CC2)C)CCN(C(C2CC(=O)C2)=O)C1 16261,C(CCCCNC(=O)Cn1ncnn1)NC(C=CC(C)(C)SC)=O 16262,N1(C(C(CC)(C)C)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C)COC)C1 16263,N1(C(c2cnn(CC)c2C)=O)CCC(NC(=O)CCn2ccccc2=O)C(C)C1 16264,N1(C(C2(OC)CCOCC2)=O)CC2(CCN(C(=O)CC3(C)CCC3)CC2)C1 16265,C1(NC(c2cnc(OC)nc2)=O)CCN(C(=O)CCOC2CCOC2)CC1(C)C 16266,Cc1cc(Cl)ncc1C(=O)NCC1CC(NC(c2nc(Cl)c(Cl)s2)=O)C1 16267,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16268,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16269,N1(C(CC2N(C)CCCC2)=O)CCN(C(=O)CCCF)C(c2ccccn2)C1 16270,c1(OC)ccc2cc(C(=O)NC3CCCC(NC(=O)C(C)S(C)(=O)=O)C3)n(C)c2c1 16271,N1(C(C2C(C)(Br)C2)=O)CCC(C2CCCN2C(=O)CCc2ccc(F)cc2)CC1 16272,ClC1=NC(NNC(=O)NCCC(F)(F)F)C(c2ccccc2)=CC=C1 16273,c1(C(N2C(C(C)NC(C(=O)N(C)C)=O)CCC2)=O)nccc2cccnc12 16274,c1(C(=O)NC2CCN(C(c3cc(Cl)sc3Cl)=O)CC2)cc(Cl)nc2ccccc12 16275,c1(NCCOCCCC)ccc(S(=O)(=O)NCC(CO)C(C)(C)C)cc1Cl 16276,c1(-c2cn(CCN(C(=O)CC3OCCC3(C)C)CC)nn2)ccc(Cl)cc1Cl 16277,c1(C(=O)NCCOCCNC(C2(C)CNC(=O)C2)=O)cc(Cl)cc(F)c1F 16278,N1(C(C(C=C)O)=O)Cc2ccccc2C(CNC(=O)C(F)=C2CCCC2)C1 16279,c1(CC)ncc(C(=O)N(CC(C)NC(c2cn(CC3CNC(=O)O3)nn2)=O)C)s1 16280,C1(NC(CC2(OC(C)(C)C)CC2)=O)CN(C(c2cn(CC(N)=O)nn2)=O)CC1O 16281,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16282,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(C(C(C)CO)=O)C(C)C1 16283,c1(CC(=O)NC2CN(C(COCCSC)=O)CC2F)cnc2c(=O)[nH]ccn12 16284,N1(C(C2CC(OC)C2)=O)CC(CNC(c2cc(CO)[nH]n2)=O)C(C)C1 16285,CCCCCCCCC(F)C(=O)NC(C)CNC(c1cnc2[nH]c(O)nc2c1)=O 16286,c1(COC(N(C)C)=O)ccc(N(C2CC(F)(F)C2)C2CC2)c(F)c1 16287,C12(CNC(C=CSC)=O)CCC(CC1)N(C(c1cc[nH]c1)=O)C2 16288,c1(C(=O)NC2(CF)CCN(C(C(CCC)OCC)=O)C2)cncc2ccsc12 16289,c1(C(N2CC(C)C(NC(=O)CC3CC4CC4C3)C2)=O)n[nH]c2c1CC(C)OC2C 16290,c1(CC(=O)NC(CNC(CCCn2ncc(C)c2)=O)C(C)C)cccc(C)c1F 16291,C(=O)(CC(C)CNC(c1ccccc1-n1cc(NC(=O)C(C)(C)F)nn1)=O)OC 16292,c1(CCCC(=O)N(CCNC(c2cnc[nH]2)=O)C2CC2)cc2ccccc2o1 16293,c1(NC(C2N(C(c3ccc(OCCC)o3)=O)CC(O)C2)=O)c(C)ccnc1C#N 16294,c1(C(=O)NC2CCCC2CNC(c2ncc(F)cc2F)=O)cn2cnnc2cn1 16295,C1(NC(=O)CCN2CCCC2=O)CCCCN(C(=O)C(C2CCCCC2)O)CC1 16296,C1(C(=O)NC2(CC=C)CCC2)C2CCC(C2)N1C(=O)Nc1cc(NC)ccc1Cl 16297,N1(C(CSCC#C)=O)CC(C(=O)NC23CCC(CC2)OC3)OC(C)C1 16298,c1(NC2C(C)CN(C(c3c[nH]ccc3=N)=O)C2)nc2c(cc1Cl)C(=O)OC2 16299,c1(OC)ccnc(OC)c1C(=O)NCc1ncoc1CCNC(C1(C)COC1)=O 16300,Cc1ccc(F)cc1C(=O)NCC1C2CN(C(=O)C(C(CC)N(C)C)N(C)C)CC12 16301,C1(NC(=O)C(C2CCCCC2)O)CC2CC1N(C(c1c[nH]nc1F)=O)C2 16302,C1(CC#C)(C(=O)NC2CN(C(=O)Cc3ccnn3CC)C2)CCCCO1 16303,N1(C(CNC(=O)C2CC2)=O)CC(C(=O)NC23CCCC2C3(F)F)C(C)(C)C1 16304,c1(C(=O)NC2CCC(NC(=O)C(F)=C3CCC3)C2)ccc(CO)c(Cl)c1 16305,C(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2ccc(Cl)cc12)c1[nH]nc(SCC)n1 16306,c1(C(=O)OC)ncc(N(C2CCN(C(C3CCCC(C)(C)O3)=O)C2)CC)nc1C 16307,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16308,C#CCCCCCNC(C1CN(C(=O)C(CC)OCC)CC1CC)=O 16309,N1(C(c2n(CC)nc(C)c2)=O)CCCCC(CCC(=O)NCC2CC(CF)C2)C1 16310,N1(C(c2oc(Br)cc2-c2ccccc2)=O)CCC(C2CC2(F)F)C1 16311,CCC(F)(F)C(=O)NCc1ccccc1N1CCN(C(C2(C#N)CC2C)=O)CC1 16312,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16313,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16314,N1(C(=O)COc2ccc(Cl)cc2Cl)CC(=O)NC2CNCCC12 16315,C1(CNC(c2occc2Br)=O)CC2COCC2N1C(C1CCc2c[nH]nc2C1)=O 16316,N#Cc1ncn(CC(=O)NCC2CCC(NC(=O)Cc3ccn(C(F)F)n3)C2)n1 16317,C(CNC(c1cccc(-n2cccn2)c1)=O)(CC(C)C)NC(c1c(C)con1)=O 16318,c1(-c2ccccc2)ncc(CNCCn2ccnn2)cn1 16319,N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 16320,C(C(C(=O)O)C1CC1)SCCOCCC(C)C1CC1 16321,c1(C(N2C(C)CCC(NC(c3c(C)nccc3)=O)C2)=O)ccc2cnncc2c1 16322,c1(C(=O)NC2CC(CCNC(c3cncc(C#C)c3)=O)C2)cc(S(C)(=O)=O)cs1 16323,N1(C(Cc2cn(CC)nn2)=O)CCC2(CCC2)C(CNC(c2cn[nH]c2)=O)C1 16324,C(=O)(C(CNC(=O)CCc1nccn1C)CC(C)C)NCC1(C(CC)=O)CC1 16325,C(=O)(C(C)CC(C)C(C)=O)N1C(CNC(c2n(C(CC)C)ncc2)=O)CCCC1 16326,Cc1cc(N2CCCCCCC2)nc(N2CCC(SC(F)F)C2)n1 16327,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16328,C(=O)(CCCC(C)(F)F)N1CCC(CCNC(C(C)(C)CF)=O)C1 16329,C1(CNC(c2c(C)noc2)=O)CN(C(c2c[nH]c(Br)c2)=O)CCC1C 16330,C1(CCC(=O)NCC2CC(NC(C(C)C3CCC3)=O)C2)CCCCO1 16331,c1(C(=O)NC(C)CCCCNC(=O)C(C)(O)c2cccs2)cn(C)c(=O)nc1O 16332,Cc1nn(CCC(=O)NCC2(O)CCN(C(c3n[nH]c(C)c3Cl)=O)C2)c(C)c1C 16333,N1(C(CC2CC(C)(C)OC2)=O)CCC2CN(C(=O)Cc3ccon3)CC2C1 16334,C1(CNC(c2scc(OC)c2OC)=O)CCC(C)CN1C(C12CC(C)(C1)C2)=O 16335,N1(CC)Cc2ccccc2C(C(=O)NC2CCN(C3CCCC3)CC2)C1 16336,Cc1cc(C(N2CCOC(CCNC(c3cc4occc4s3)=O)C2)=O)cc(F)c1 16337,c12cc(cc(O)n1)COC2=O.C(CC(=O)NC(C)(C)C)(OCCC)OCC 16338,Cc1cc(C)c(C(=O)NC2CC(NC(=O)C(O)CC(F)(F)F)C2)c(O)n1 16339,C(C(c1nnnn1CCC1(C)CC1)Nc1ccccc1C)(C(C)C)OC 16340,CC(C(CO)NC(=O)CC)NC(C1CC1c1ccccc1)=O.C(CN(C)C)OC(C)=O 16341,C1(C)(CNC(CCc2c(C)ncs2)=O)COCCN(C(=O)C(C)C(F)F)C1 16342,N12CC3CCC3(C1)NC2=O.C(CC(O)c1cccs1)N(C)C 16343,C1(O)(C(=O)NC(CCOC)CNC(=O)C(c2ccnn2C)O)CCC(C)CC1 16344,c1(N2C(COC)CCC2)nc(OCNCCCC2CCS(=O)(=O)C2)cc(C(F)(F)F)n1 16345,Cc1ncc(C(N2CC3(CCN3C(=O)Cc3ccoc3)C2)=O)c(Br)c1Cl 16346,C(=O)(C#CC1CCOCC1)N(C)CC1CCCN1C(c1cc(F)cnc1Cl)=O 16347,C12(C(N3CCC(CN(C)C)C3)=O)CC(CO)(CN1C(=O)CCOCCN(C)C)C2 16348,c1(CC(=O)NCC2CN(C(C3(C(F)F)CC3)=O)CCCO2)cn2ccsc2n1 16349,C1(NC(C(CC2CN(C(C3CCN(OCC)C3)=O)C2)F)=O)C(C)CCC1C 16350,Cc1ccc2cccc(C(N3CCC(N(C)C(c4c(C)nsc4C)=O)C3)=O)c2n1 16351,C1(OC)CCCC(CC(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16352,CC1CN(C(=O)Cc2nnc(O)s2)CC(C)N(C(=O)Cc2cc(Cl)ccc2Cl)C1 16353,c1(CC(=O)NCC2C(NC(C(C)OC)=O)C2)cc(C)nn1C 16354,C#CCC(O)C(=O)NCC1C=CC(NC(=O)Cc2csc(Cc3cccs3)n2)C1 16355,N1(C(C(C2CCC2)OCC)=O)CCCC(C)(CNC(c2ccc(=O)n(C)c2)=O)C1 16356,C(=O)(NNc1cc(F)ccc1N1CCOCC1)NC(c1cc2c(cc1)OC(C)C2)=O 16357,C1(NC(c2cc(CC)ncc2)=O)CN(C(=O)CNC=O)CC1(F)F 16358,c1(C(N2CC(c3cn(CC(C)(C)O)nn3)(O)C2)=O)ccc(S(N)(=O)=O)cc1 16359,c1(CN(CCNC(C(CSC)C)=O)C(C)=O)cccc(Cl)c1.C1(=O)CCCN1 16360,C(=O)(CC(C)(CNC)C(F)(F)F)NC1CC(NC)CN(C(c2c(CC)nc[nH]2)=O)C1 16361,c1(COC)ccc(-c2ccc(C3(C(=O)N(C4CC(O)C4)C)CC3)cc2)cc1 16362,Cc1nnccc1C(=O)NC(C1CCCN1C(c1cccc(NC(N)=O)c1)=O)C 16363,C(Cc1ccccc1)(C(=O)N1CC(O)(CCNC(=O)Cc2nc[nH]n2)C1)NC=O 16364,c1(C(=O)NC2C3CN(C(c4n(CC)ccc4)=O)C2CC3)nc(C)c(N)cc1C 16365,C(CC(C(=O)NC(C)COC(F)(F)F)NC(=O)Cc1ccccc1F)=CC 16366,C1(NC(c2ccc(CSC)cc2)=O)CC2CN(C(C3(C)CCCC3)=O)CC12 16367,C1(CNC(COC(CC)CC)=O)CCCN(C(c2nnsc2C)=O)CC1 16368,N1(C(=O)Cn2cc(C3CC4C=CC3C4)nn2)CCC(OC)CC1.C12CN(C1)C(=O)C2 16369,Cc1ccc(I)cc1C(=O)OC1CC(NC(=O)OC(C)(C)C)C1 16370,N1(C(C(C)O)=O)CCCC2(C1)CN(C(C1C3(CC3)C13CC3)=O)CCO2 16371,c1(C(N2CC(N(C)C)C(CNC3CCCS3)C2)=O)ccc2sc(O)nc2c1 16372,Cn1c(C(=O)NCCCCCNC(c2n[nH]cc2Cl)=O)c2n(c1=O)CCCC2 16373,CCCC(C)CC(C)(c1nnnn1C(C)C)Nc1ccc(C(=O)N(C)C)c(C)c1 16374,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16375,CC(CC(C)(C)C)C(F)C(=O)N(C)CC1CCCN1C(=O)CCc1cscn1 16376,CC1CCN(C(=O)CC(=O)N(C)C)CC1NCC1CCN(C(=O)CC2(O)CC2)CC1 16377,CCCC(CC)CC(=O)N1CC(CNC(=O)COCCc2cccs2)(OC)C1 16378,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(NC(c3csc(Cl)n3)=O)CCCCCC12 16379,c1(C(=O)NC2Cc3ccccc3C2)cc2c(NC3CC3)cccc2[nH]1 16380,C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(CNC(c2ccc(C)s2)=O)=O)CC1C 16381,Cc1cccc(Cl)c1C(=O)NCCCC(C)(C)NC(=O)CN1CCC(C)C1 16382,CCCC(CNCc1nnnn1Cc1cc(C(N)=O)co1)CCO 16383,S(=O)(=O)(c1cc(C(=O)Nc2ccc3c(c2)CCO3)ccc1F)NC(C)C 16384,c1(OC)ccc(C(N2CCCC(C)(CNC(C3(C(N)=O)CCC3)=O)C2)=O)cc1Cl 16385,CC1CC(C(N2CCCC2CNC(c2cncs2)=O)=O)CC(C)C1 16386,c1(CNC(C2CC2Cl)=O)cccc2c1CN(C(c1ccn3nnnc3c1)=O)C2 16387,c1(C(=O)NCC2CC(NC(C(N3CCC(C)CC3)C)=O)C2)ccc2nc(O)[nH]c2c1 16388,N1(C(C(c2scc(C)n2)(F)F)=O)CCCC(N(C(=O)CCOCCC2CC2)C)C1 16389,c1(NC(COCCOCCOC)=O)nc(CNC(=O)C=Cc2ccc[nH]2)cs1 16390,CC(CC(C)(C)C)NC(C1OCCC1NC(=O)CCc1nc(O)n[nH]1)=O 16391,C(=O)(CCCCCF)N1CCC(C)(CCNc2c(CC)cccc2)C1 16392,c1(OC)ccnc(CC(=O)N(CC(C)(C)CNC(C2CC2c2ccco2)=O)C)n1 16393,N1(C(C(C)(C)C#N)=O)CCN(C(c2ccc(F)nc2F)=O)C(CCO)C1 16394,C1(OCC(=O)NCC2C(NC(c3cnc(C)o3)=O)CCC2)CCC(C)CC1 16395,N1(C(C(C(C)C)C)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 16396,N1(C(c2n(C)ncc2Br)=O)CC2CCC2(CC(=O)NOC2CCOCC2)C1 16397,C1(C(=O)NC(CCCNC(CSCCN(CC)CC)=O)C)Cc2ccncc2C1 16398,c1(C(C)SC2CC=CC2)cn(C(C2CC2(C)C)C)nn1 16399,C1(CNC(c2c(C)scn2)=O)CC2CCC1N2C(C1(C)CC(F)C1)=O 16400,CC(CC1CC1)C(=O)N(CC(C)(C)NC(=O)C(C)n1ccnc1)C 16401,C1(C(=O)Nc2csc3ccccc23)(N(C)C)OCCc2ccccc21 16402,CS(C)(=O)=NC(=O)C(=O)C(C1CC(c2ccccc2)(N)C1)=O.C1CN1.C(C)(=O)O 16403,C1(NC(C(COC)OC)=O)CN(C(C2CSCN2C(C)=O)=O)CCN1C 16404,O=C1NCC2(CCN(C(=O)C3=CCN(C(=O)CC4C=CCCC4)C3)CC2)N1 16405,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(C1CCC1)C 16406,N1(C(C=C(C)C)=O)Cc2nccn2CC(NC(=O)CN(C)C2CC2)C1 16407,C(c1cccc(C(F)(F)F)c1)=CC(=O)NCC1(O)CN(C(C2C(C)CC2)=O)C1 16408,c1(OC)ccc(C(=O)N(C(C)CNC(c2ncc(N)nc2C)=O)C)c(Cl)c1 16409,Cc1cc(C(=O)NC(C)(C)CC=CC(=O)NCCCO)n[nH]1 16410,CCC(CC(=O)N1CCC1CNC(c1ccc(CSCC)s1)=O)c1ccccc1 16411,N1(C(CCN(CC)CC)=O)CC2(C1)SCCC2NC(c1ccc2occc2n1)=O 16412,CC(CN(C)C(c1cccc(OC(F)(F)F)c1)=O)N=c1ccnc[nH]1 16413,c1(OC)cc(Br)cnc1C(=O)NCC(C1CC1)NC(c1cnn2c1OCC2)=O 16414,c1(C(=O)NC(C)CNC(=O)C=Cc2cc[nH]c2)cc2cc(Cl)cc(Cl)c2[nH]1 16415,c1(C(N2C(C)CC(NC(CCCOCCOC)=O)C2)=O)nc[nH]c2nccc1-2 16416,C1(NC(c2occ(OC)c(=O)c2)=O)CCOC2(CCOCC2)C1 16417,N1(C(Cc2ccc(C(C)=O)s2)=O)CC(NC(C2(CO)CC2(F)F)=O)CC2(CC2)C1 16418,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16419,n1(CCNC(C(C)C2(O)CCC2)=O)ccc(C(=O)NC2(C(O)CO)CC2)c1 16420,CC1CN(C(C)CCN2CCOCC2=O)CC1Cc1ccccc1 16421,CCCCCC(C1CCC1)NC(=O)NC1CCOCC1C(=O)OC 16422,C(=O)(CCCCCCn1cc(-c2cscc2C)nn1)NC(C(CC)C)C 16423,C(C)(C)(CCN=c1[nH]cnc(C)c1C#N)NC(c1cn(CC)nc1C)=O 16424,CC(C)(C)C(C(=O)N1CCC(C(C)(C)O)C1)C1CCOC1 16425,C#CCN(OC)C(=O)C1(CONC(C2CCC3C2C3(F)F)=O)CCCCC1 16426,C1(CNC(C2N(C)CC2)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CC1C(F)(F)F 16427,CC(CCCNC(=O)CNc1ccccn1)NC(=O)CC1CC1 16428,C(=O)(C1=CCCCCC1)NCc1c(CCNC(=O)CC2NC(=O)NC2=O)ocn1 16429,c1(COC(C)C(=O)NC(C2(O)CN(C(c3cc(Cl)no3)=O)C2)C)ccc(F)cc1 16430,Cn1cc(C(=O)NCCCNC(c2cn(C3CCOC3)cn2)=O)c(Cl)n1 16431,CCC(CC(F)F)C(=O)N1CCC(CN(C(=O)C(C)c2ccco2)C)C1 16432,c1(SC)nc(C)c(CCC(=O)NCC23CCCC2CCN3C(=O)C(C)C)c(O)n1 16433,C(C(=O)NNC(=O)C1CN(C(=O)OC(C)(C)C)C1)n1cc(-c2c(C)ccnc2)nn1 16434,N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)CC2(C)CCS(=O)(=O)N2)CC1C 16435,C(=O)(CC1=CCCCC1)N1CC2C(CNC(c3ccc(C(=O)O)cc3O)=O)(CC2)C1 16436,c1(C(N2CC3C(C(=O)NC4C5CCCCCC45)(C3)C2)=O)sc2ccccc2c1Cl 16437,Nc1nc(C(N2CC3(NC(=O)CCC(=O)N(C)C)CC2C3)=O)ccc1O 16438,C1(c2nc(C)sc2)CCC(CNC(N2CCOCC2c2ncnn2C)=O)CC1 16439,c12csc(=Nc3ccnn3C)n1CCN(CC)c1cccc-2c1.S(C)C1CC1 16440,N1(C(C2(OC)CS(=O)(=O)C2)=O)CCC(NC(=O)CCc2cnn[nH]2)C(CO)CC1 16441,C(C1=CCN(C(c2coc(CC3CC3)n2)=O)C1)NC(C(C)OC)=O 16442,CCC(C)(C)C(=O)NC1(CNC(=O)CC2CCC(C)(C)O2)CCOC1 16443,c1(C(=O)NC23C(CCN(C(CCOCC)=O)CC2)C3)cc(Cl)c(OC)c(Cl)c1 16444,C1(C2CCCN(C(=O)CN3CC4CC4C3)C2)(NC(C2(OC)CCOCC2)=O)CC1 16445,CN1CC(C)(C)CC1C(N1CCC(NC(c2ncc(F)cn2)=O)C1)=O 16446,N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)CC2CC(O)C2(C)C)C(CCO)C1 16447,N1(C(C2CC3CC3C2)C(=O)NC)CCn2ncc(CN(C)C)c2C1 16448,N1(C(c2ccn(COC)n2)=O)CCC(C)C(NC(=O)CCCCOC)C1 16449,c1(C(=O)OCC(=O)N(C2CC(=O)NC2=O)CC)cccc(O)c1Cl 16450,N1(C(C(C)OCC#C)=O)CCOC(CNC(=O)CCN2CCN(C)CC2)C1 16451,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(O)C(C)C)CC2)=O)nc1C 16452,C1(CCC)CN(C(C2ON=C(C)C2C)=O)CC1C(=O)NCc1nc(CO)n[nH]1 16453,CCC(C)(CNC(=O)COC1CC(NC(=O)CC2CCCCO2)C1)CC 16454,C1(O)(C(=O)NC2CC(NC(Cc3ccn(CC)n3)=O)C2)CCCC(C)(C)CC1 16455,Cc1ocnc1C(N1C(C(=O)NC(C)(CO)C2CCCC2)CC1C)=O 16456,N1(C(C)=O)CCCC1C(N1CC(O)(C(C)NC(=O)C(C)(C)c2ccnn2C)C1)=O 16457,C(=O)(C1=NOC(C)C1C)NCCCCNC(C(c1ccccc1)OC(C)C)=O 16458,CN1CC(N=c2nc3sccc3c(NCCN3CCCC(O)C3)[nH]2)CC12CCC2 16459,c1(OC)nccc(I)c1C(=O)NC1CCC(NC(c2ccc(OC)cc2Br)=O)C1 16460,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C2CN(C(c3cc(C)[nH]n3)=O)C1C2 16461,CC(C)(CC(F)C(=O)NCCC1CCSC1)NC(C1CC12CC2)=O 16462,c1(C(N2CC(NC(C3(CCO)CC3)=O)CC(O)C2)=O)ccc2ncccc2n1 16463,c1(C(=O)NC2(CNC(=O)CC3CCCC(O)C3)CCCCC2)cn2c(n1)CCC2 16464,C(=O)(CCCN=c1nccc[nH]1)NC(C)CN(C)C(C1CC(OC(F)F)C1)=O 16465,C1(CNC(c2coc3c2COC3)=O)CN(C(=O)C=CBr)C2CCN1C2 16466,c1(N(C2(c3n(CCCC)nnn3)CCOC2)C)ccc(N(C)C)c(F)c1 16467,c1(C(C(=O)NCC)N(C)CC23CC(C2)C3)ccnc(O)c1.C1(C(=O)N)COCC1 16468,C1(NC(C2(OCC)CCC2)=O)CCC2CN(C(C3CN4CCN3CC4)=O)CC2C1 16469,C1(N(C(c2cc(C)c(-c3ccc(F)cc3)s2)=O)C)CN(C(=O)C(F)F)CC1(C)C 16470,C1(NC(C2(C(=O)NC)CC2)=O)CC2CCC1CC2NCc1cc(Cl)ncc1OC 16471,N1(C(CCC#C)=O)CCC2CC(C(N3CCC(F)(CO)CC3)=O)C2C1 16472,C(C)(C)(C(C)CC(=O)NCCCN(C(=O)CCS(C)=O)CCC(C)C)OC 16473,N1(C(C2CC3CCC2N3C(C2CCCC(=O)N2)=O)=O)CC2(CNC(=O)N2)C1 16474,C1(NC(c2n(C(C)C)ncc2Cl)=O)CN(C(C2CN(C)C2)=O)CC1(C)C 16475,Cc1nnccc1C(=O)N(C(CNC(c1cccc(C(F)(F)F)n1)=O)C1CC1)C 16476,N1(C(c2nc(C(C)C)oc2)=O)CCC2CN(C(=O)CCCCCCCBr)CCC12 16477,C1(C(F)(F)F)(NC(=O)NC(c2ccc(C)cc2)CC(=O)OCC)CCCCC1 16478,Cc1nn(C)c(N)c1C(N1CCOC(CC(N2CC(C)C2(C)C)=O)C1)=O 16479,CC1(C)C(C(=O)NCC2CN(C(=O)Cc3ccno3)CCO2)C1(C)C 16480,NC(CC(=O)N1CCCCC1CCc1ccccc1F)C(=O)O 16481,c1(OC(F)F)ncc(C(F)(F)F)cc1F.c12ccc(F)cc1SCc1nnnn1-2 16482,Cc1cnc2n1CCC(N1CCCCC1CCC#N)C2 16483,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(c2ccnc(C)c2)=O)c(F)n1 16484,S(=O)(=O)(c1cccs1)NC(C1CN(C(C(C#N)NCCC(=O)OC(C)(C)C)=O)C1)=O 16485,N1(NC(C(C)n2ccnc2)=O)CC2CCC1(CO)C2.C123CC(C1)(C2)CC(=O)N3 16486,C(C(C)(O)CC(=O)NCC1CC(NC(c2nc(C)n(C)c2C)=O)CCO1)OC 16487,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)C(C)(C)C)c1C 16488,c1(C(=O)NCC2CN(C(c3cn(CC=C)nc3)=O)CC2C)cccc2c1NCC2 16489,O=C1CN(C(c2cocn2)=O)C2CCN(C(=O)CSC(F)(F)F)CC2N1 16490,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16491,c1(C(=O)NCC(C(C)C)NC(C2(CCF)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 16492,c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16493,C1(C(N2C(CNC(C3(CCOC)CCC3)=O)CC(O)C2)=O)CCCCN1N=O 16494,N1(C(=O)CC2(CO)CC2)CC2CN(C(C3(c4cccs4)COC3)=O)CC2C1 16495,C(=O)(C(F)(F)c1nccs1)NC(C1CCCN1C(c1nnn(C)n1)=O)C 16496,N1(C(C2(CCC)CCC2)=O)CC(N(C)C(c2cccc(F)c2C)=O)C(C)(C)C1 16497,C(=O)(C1=NOC(C)C1)NCC(C(C)C)NC(C1C(CC(C)C)C1)=O 16498,NS(=O)(=O)c1cccc(NC(=O)Nc2nc(C(F)F)cs2)c1 16499,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)N(CC=CC)C1CC1 16500,C1(OCC)CC2(C1)CC2C(=O)N(CCCCCNC(C12CCC(CC1)C2)=O)C 16501,C1(C(=O)NC2(C(=O)NCCc3ncc(C)cn3)CCC2)CC2(CCC2O)C1 16502,N1(C(N(c2nc3ccccc3o2)CC(C)C)=O)CCc2cccc(C#N)c21 16503,CN=c1[nH]c(C(N2CC(CCNC(C3CCN(CC(F)(F)F)CC3)=O)C2)=O)cs1 16504,c1(OCC)ccc(C2(C)C(F)(C(=O)NCCCO)CC2)cc1Cl 16505,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)N(C)C)NC(C1CCSC1)C 16506,C1(O)(CCNC(CSS(C)(=O)=O)=O)CCN(C(=O)Cc2sccc2Cl)C1 16507,N1(C(C(C(C)C)(C)C)=O)CCCC(NC(C2CC=CC2)=O)C(F)C1 16508,C=CCC(CC(=O)Nc1ccccc1CCO)NC(c1ccc(C#N)cc1)=O 16509,C(=O)(C(C)CCCOC)N1CCC(CC(C)NC(COCC(C)C)=O)CC1 16510,c1(SC)c(OC(F)(F)F)cccc1NC(C1CCN(C(=O)C(C)S(N)(=O)=O)C1)=O 16511,c1(CC)nccnc1C(=O)NCc1sc(=N)[nH]c1C.C12=CC(=O)N(CC1)CC2 16512,C1(C(N2C(COCC)COCC2)=O)CC(F)CN(C(=O)Cc2cc(F)ccc2F)C1 16513,N1(C(C2C(C)OCCC2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16514,S(=O)(=O)(c1ccc(OC(F)(F)F)c(Cl)c1)N1C(C(=O)NCCC)CCCCC1 16515,C(=O)(C(O)CC(C)C)NC1C(CNC(Cc2c(OC)ccnc2)=O)C1 16516,N1(C(c2c(C#N)scc2)=O)CCCCC(CNC(=O)Cn2cccc2)C1 16517,c1(CSN2C(=O)C(c3ccc(-c4ccco4)cc3F)CC2)cc2n(n1)CCCO2 16518,N1(CC)CCC(N(C2CCN(c3ncccn3)CC2)C(=O)OC)CC1 16519,C1(C(N2CCC(C(N(C)Cc3cccnc3O)=O)(CO)C2)=O)CCOC(=O)CC1 16520,C#CC1CCN(C(=O)C(CCCOC)NC(=O)C(C(C)OC)N(C)C)CC1 16521,c1(C(=O)NCCC2COCCN2C(C2CCCC2)=O)cc2nc[nH]c2cn1 16522,N1(C(C(CCC)NC(C)(C)C)=O)CCCC2(CC1)CNC(=O)C2 16523,CC1(C)CC(NC(c2ccc(-c3cccs3)o2)=O)CN(C(c2cccnc2)=O)C1 16524,N1(C(C2(C)C(CC)CCC2)=O)CCc2nc(CNC(=O)CCCC3CC3)sc2C1 16525,N1(C(=O)Cn2cc(-c3cscn3)nn2)CC(CO)OC2(CCOC2)C1 16526,c1(C(=O)NCC2(COC)CN(C(C3CC3Cl)=O)C2)noc2ccc(Cl)cc12 16527,N1(C(c2c(C)oc(CNC(=O)Cc3ccn(C)c3)n2)=O)CCc2nc(O)[nH]c2C1 16528,S(=O)(=O)(c1cc(Cl)sc1C(=O)N(C1CC(NC(C2CCCO2)=O)C1)C)NC 16529,c1(OC)cc(C)sc1C(=O)NC1CCC(NC(c2cnccc2C)=O)C1 16530,CC1CN2CCN1C(C(=O)NCCCCCNC(=O)CCC(F)F)C2 16531,C1(OC)CCC2(C(=O)NCCC(C)(C)NC(c3cccc(OC)n3)=O)CCC12 16532,C(C(C)(C(=O)N1CC(C)(N(C)C)C1)NC(c1ccc(C)nc1)=O)SC 16533,c1(NC(C2(CNC(c3cc[nH]c3)=O)CCCC2)=O)cccc(C2CC2)c1 16534,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16535,C1(C2(O)CCC2)(C(N2CCN(C(c3ccoc3)=O)CC2)=O)CC1 16536,C1(C)(CNC(C(C)OCCOCC)=O)CN(Cc2nccnc2Cl)CCO1 16537,CCC(C(=O)NCCC1CCCN1C(=O)C(C)ONC(=O)OC(C)(C)C)N(C)C 16538,n1(CCCCCC)nc(CC2(CC3CCCC3)CC2)nc1-c1cn(CC)nc1C 16539,N1(C(C(CC)F)=O)CCCC(C)(NC(c2cnncc2C)=O)C1 16540,Cc1c(C(=O)NC2CCC2C(=O)NCC(C)CN(C)C)cccc1-c1ccncc1 16541,N1(CC(=O)NCC2C=CC(NC(CSCCC)=O)C2)CCS(=O)CC1 16542,c1(C(N(C)CC2N(C(CN3C(C)CCCC3)=O)CCC2)=O)cccc2ccsc12 16543,C1(C(=O)NC(CC=C)CNC(=O)Cn2cc(Cl)cn2)C2CC3CC(C2)CC1C3 16544,c1(C(N2C3CC(CNC(C(CC#C)C4CC4)=O)C2CC3)=O)ccn2ccccc12 16545,C1(NC(CC2(C)CCCC2)=O)CCOCC1NC(c1ccccc1)C1CC=CC1 16546,c1(CC(=O)NCCCNC(C(C2CCOC2)OCC)=O)sc(O)nc1O 16547,C1(C(N(C(C)CNC(=O)OC)CC)=O)CCN(C(=O)C=Cc2csc(C)n2)CC1 16548,N1(C(c2cn(CCC(=O)N(C)C)nn2)C2CC2)CCCc2ccccc21 16549,C1(C(C)C)CCCN(CC(=O)NCC(=O)NCc2ccc(CO)cc2)C1 16550,CCCCN=C(NCCc1ncc(C)cn1)NCC1CCCSC1 16551,CC1OCCC1(F)CC(=O)NC1(CCNC(c2ccn(C)c2)=O)CCC1 16552,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16553,C12CCN(C1C(C)C)CC1CCCC1C(=O)N2.c1(C(C)C)nc(C(F)(F)F)cs1 16554,C1(CC=CC)CCCN(C(=O)CC(C)(C)NC(=O)C=C(C)C(C)(C)C)C1 16555,CCCCCC(C(=O)N1CCC(NC(c2cccc(Cl)c2)=O)C1C)C(C)C 16556,C1(C(N2CC(F)(CNC(C(CC)Sc3ccccc3)=O)C2)=O)CCCCN1CC 16557,N1(C(c2cc(C)nn2C)=O)CCC(C2CC2)C1CNC(c1cnc(F)cc1C)=O 16558,CC(C)(F)CC(=O)NCC1COC(CNC(c2cnc(O)o2)=O)C1 16559,C(=O)(C1=NN(c2ccccn2)C(=O)CC1)N1CC(CS(N)(=O)=O)C(O)C1 16560,CS(=O)CCC(O)C(=O)NC12CC(NC(=O)C=Cc3cccs3)(C1)C2 16561,CCCCCC(O)C(C)C(=O)N1CC(CNC(C2Cc3nccn3C2)=O)C(O)C1 16562,c1(C(C)NC(=O)C(CC2CCOCC2)NC(=O)C(C)n2cccc2)ccccn1 16563,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16564,N1(C(c2ccc(C(C)=O)o2)=O)CCCC(CCC(=O)N(C2CCCC2C)C)C1 16565,c1(NC(=O)NC(c2ccccc2)C2CCCC2)nccc(-c2cnccn2)n1 16566,C1(NC(C(CNC(=O)C(F)=CC2CC2)N(C)C)=O)CCC(O)C(O)C1 16567,C1(CNC(CC(C)c2ccccc2)=O)CCCCC1NC(C1(N(C)C)CC1)=O 16568,Cc1oc(C)c(C(=O)NCc2ocnc2C(=O)NC2CCCC(O)CC2)c1C 16569,C1(C(N2C(C)(CNC(=O)C=CBr)CCC2)=O)CCCC12CCC2 16570,C1(CCNC(CCCC=C)=O)CN(C(=O)CCCC#N)CCCO1 16571,N1(C(c2c(SC)ccs2)=O)CCCCC1CNC(=O)C(C)(C)c1cnco1 16572,C1(NC(C2C(OCC)C2)=O)CC2CC(C1)CN(C(=O)CC(C)(C)CN(C)C)C2 16573,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 16574,C(=O)(CCCC(C)NC(C1(C#N)CC1(C)C)=O)Nc1cccc(OC)c1 16575,C#CCC(C)(CNC(C1C=CCN(C(=O)CC(C)n2cccc2)C1)=O)CO 16576,N1(C(CC(C)SC)=O)CCCC(C)(C(=O)Nc2cccc(F)c2)C1 16577,c1(OC)ncc(C(=O)NCCN(C(c2ccc(Br)cn2)=O)C(C)C)c(C)n1 16578,Cc1c(C(=O)NCC(C2CCOC2)NC(=O)C2=CCCCO2)nc2sccn12 16579,C1(CNC(C2C(CC)CC2)=O)CN(C(C2CC(n3cnnc3)C2)=O)CCC1C 16580,C=CCC(C(=O)N1CCCC1CCNC(C1(N(C)C)CCCC1)=O)C(C)(C)C 16581,c1(CC(N2CC(C)(CNC(c3cc(Cl)ccc3Br)=O)C2)=O)cn2ccccc2n1 16582,CCCC(C(=O)NC(C)CNC(C1(C)CN(C(=O)OC(C)(C)C)C1)=O)S(N)(=O)=O 16583,CC1CN(C(=O)Cc2ccccc2C2CC2)CC1NC(=O)CCN(C)CCO 16584,C1(C(N(C(C)CNC(=O)C=C(Cl)Cl)C)=O)C2CCC1(c1ccco1)C2 16585,S(=O)(=O)(c1ccc(Cl)cc1)N1CC(NC(C(C)NC(CCC(=C)Cl)=O)C(C)C)C1 16586,CCCC(CCCNC(c1nocc1C)=O)NC(c1ccc(COC)nc1)=O 16587,C1(CC)CN(C2CC(C)OC(C)C2)CCN1C(=O)NC1CCCCC1 16588,c1(C(=O)NC(CC=C)C(=O)NCC2CC3C=CC2C3)cc(O)cc(=O)o1 16589,C1(C(=O)NC2CC(C)(NC(=O)CCC=CBr)C2)CCC2(CCC2)CC1 16590,C1(C(=O)NC2CCC(NC(C3C(C(=O)OC)C3(F)F)=O)C2)CC2CC1C1CC21 16591,CC(C)(C)C#CC(=O)NCC1CCCN(C(C2CCC(=O)N2C(C)=O)=O)C1 16592,c1(C(N2CCC(NC(CCC(C)N(C)C)=O)C(F)C2)=O)cn2cccnc2n1 16593,N1(CC(=O)N(CCOC)CCNC(c2cnn(CC3CC3)c2)=O)CC(C)(C)C1 16594,Cc1ccccc1C1CC1C(=O)NC1CC(NC(c2ccnc(S)c2)=O)C1 16595,c1(C(CNC(c2n[nH]cc2Cl)=O)NC(C=NOC)=O)cccc(F)c1 16596,C1(NC(C(CSC)OC)=O)CCC(NC(=O)CC2(O)CCCCC2)CC1 16597,C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(C(CC2CC2)OC)=O)CC(F)C1 16598,CC1CCCN1CC(=O)N(CC(=O)NC(c1cnn(C)c1)CO)CC(C)O 16599,C1(CNC(c2n(C)ncc2)=O)CC2CC2N1C(c1cc(CO)n(C)n1)=O 16600,N1(C(c2cn(CCCC(c3n(C)ccc3)=O)nc2)=O)CCC(O)CC1 16601,c1(CN2CCCC(C(=O)NC(CC(=O)OCC)C)C2)cnc2[nH]ccc2c1 16602,Cc1nc(C)c2c(n1)CCCC2NCC(=O)NC1CCCC(N)C1 16603,CC(C)C(C)(F)CNC(C1CC(C)N1C(=O)CCCNC(N)=O)=O 16604,c1(CCC)ccc(C(C(=O)NCCCSC)N(C)Cc2cncn2C)cc1 16605,C(=O)(CCC(C)NC(=O)CC1(NC(C)=O)CC1)NC1(CC=C)CCCC1 16606,c1(C(N2CCCCC(CNC(CCC#C)=O)C2)=O)ccc2cccc(OC)c2n1 16607,C1(F)(CNC(c2c(CC)con2)=O)CCN(C(c2c(C)nsc2N)=O)CC1 16608,c12cccc(F)c1C(=O)N2.N1(CC(C)NC(=O)CSC(=N)N)CCOCC1 16609,N1(Cc2c(C)nn(C)c2)CCCC2CN(C)CCC12 16610,Cc1cc(C(=O)NCC(C)N(C)C(c2csc(CO)n2)=O)cs1 16611,CCCC(C(F)(F)F)c1nnc(C2CN(CCN(S(=O)(=O)CC)CC)C2)o1 16612,c1(OCCOC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccccc2)C)cn1 16613,C1(C(N2CC(NC(C(CC(=O)NC)C)=O)C2)=O)CCS(=O)(=O)C2(C1)CC(CO)C2 16614,CC1(F)C2CCC(C2)C1c1nc(=O)o[nH]1 16615,C1(C)(NC(CC(=O)NCC)=O)CCCN(C(C23CCC(CC2)C3)=O)C1 16616,c1(C(N2CC(CC(CNC(C(C)CC(F)F)=O)(C)C)C2)=O)c(O)cc(Cl)cc1F 16617,N1(C(C2CCC23CC(F)(F)C3)=O)CCC(CO)C12CCC2.C(CO)OC 16618,C1(NC(CS(CC)=O)=O)CC1C1CCCN(C(=O)COCCF)C1 16619,c1(C(=O)NC2CC(NC(c3[nH]nnc3C3CC3)=O)C2)cccc(F)c1C1CC1 16620,C(=O)(C1=CCCOCC1)NCC(C1CCN(C(c2n[nH]c3c2CCSC3)=O)C1)C 16621,c1(OC)cc(Cl)c(CN2CC3C(C2)N3C(c2ncco2)=O)cc1OC 16622,C1(c2noc(N3C(=O)CCC3=O)n2)(C(N2CC3C(OC)C3C2)=O)CCS(=O)(=O)C1 16623,c1(OC)nc(Cl)ccc1C(N1CCC(CNC(c2ccc(Cl)[nH]2)=O)(OC)C1)=O 16624,c1(S)cc(=O)c(-c2ccccc2F)co1.n1(C2(CC)CC2)cc(C(=O)N)nn1 16625,C(=O)(CCC(=O)NN(C)C)NCC(C)(C1(C(N)=O)CC1)NC(c1c(C)occ1)=O 16626,C(=O)(CCS(=O)(=O)CC(C)C)N(C(CNC(c1c(CCC)occ1)=O)C1CC1)C 16627,C1(O)(C(N2CCCC(CN(C)C(c3ccnnc3Cl)=O)C2)=O)CCCC(C)CC1 16628,C(C(=O)N1CCC(N(C(=O)Cc2ccno2)CCO)C1)(C(C)C)N(CC)CC 16629,CCC(CC)(CC)C(=O)NC(c1ccccc1)C(C)NC(=O)C(C)(C)F 16630,c1(NC(C2C(NC(=O)Cc3nccs3)CCC2)=O)ccc(N2CCCC2=O)cc1 16631,C1(CC)CN(C(C23CC(OC)(CO2)C3)=O)CCN1C(=O)CCOCC(F)F 16632,c1(CN(C(=O)CCN(C(=O)CCC2CC2(F)F)C)CC)n[nH]c2c1CCC2 16633,C(=O)(C(CCF)NC(C1C(NC(=O)Cn2ncccc2=O)OCC1)=O)OC 16634,C(CCC(=O)NCC(C)(C)N(C(=O)CC1CC=CCC1)C)OCCOC 16635,c1(NC(c2ccc(CNC(CN(CC(=O)NC(C)C)C)=O)o2)=O)cnn2ccsc12 16636,N1(C(c2c(N)cccn2)=O)CCC(C2CCCN(C(C3CCCO3)=O)CC2)CC1 16637,c1(C(C)NCC2C(C)(C)C2(C)C)ccc(Cl)cc1F 16638,CC1(C)CCC(=CC(N2CC(O)(c3ccnn3CC(=O)N(C)C)C2)=O)CC1 16639,c1(CCC(=O)N(C2CCN(C(C3CN(C(C)C)C3)=O)C2)CC)n[nH]c(=N)s1 16640,C12(C(=O)NCC3N(C(C4CCCC4)=O)CCN(C)C3)CC(C)(C1)OC21CCC1 16641,c1(OC)cc(C(N2CCCC2CCC(=O)NCc2cnn(C)c2O)=O)n(C)n1 16642,C1(OC)C2CC3CN(C(c4ccc5c(c4)COC5)C(=O)NCCCF)C1C3C2 16643,C1(NC(CC(=O)OC)=O)CN(C(=O)C(C)C=Cc2ccccc2)CC1O 16644,c1(CCC(N2C(C3(NC(C(CSC)C)=O)CC3)CCC2)=O)csc2ccccc12 16645,C(=O)(C(CCC)N(C)C)NC(c1cn(CC(=O)NC)nn1)CCC 16646,Cc1cc(F)cc(C(=O)NCCCCCNC(c2nc(C)n(C)n2)=O)c1N 16647,CC(C)C1=NOC(C(N2CCN(CCNC(=O)CCc3cc(Cl)no3)CC2)=O)C1 16648,n1(C(CC)C)nnnc1C(C1(C(C)C)COC1)NCC1(CO)CCCC1 16649,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16650,c1(OC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16651,N1(C(C(C)O)=O)CCN(C(=O)C=C(C)C(F)F)CC(COCCCC)C1 16652,c1(CCNC(C2CCC3(CCC3)CC2)=O)nc2cccnc2[nH]1 16653,C(=O)(C(O)CC(N)=O)NCCC(=O)NC(C)C(CO)NC(c1ccco1)=O 16654,c1(C(N(C(C)C)CCNC(C23CC4CC2C3C4)=O)=O)nccn2nccc12 16655,c1(C(=O)NC(CCCNC(C(CSC)C)=O)(C)C)ccc(C(C)=O)cc1F 16656,N1(C(C(=O)NC(CC2CCN(CC)CC2)=O)C)CCCCCC(C(=O)O)C1 16657,c1(CN2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)cc(F)cc(F)c1F 16658,Cc1cnc(C(N2CC(C(=O)NC3(C)CCSC3)C(C(C)C)C2)=O)cn1 16659,C1(C(N2CCCC(NC(CCC(C)C)=O)C2C)=O)CCC2(CCC2)CO1 16660,N1(C(CC2CN(C(c3c(OC)nsc3)=O)CC2C)=O)CCC(=O)N(C)CC1 16661,N1CCSCC1(C)C.Cc1cc(C(N2CCCCC2=O)C=O)c(C)s1 16662,c1(C(=O)OC)cncn1CC(=O)NC(C)C(C)NC(c1ccc(CN(C)C)o1)=O 16663,CCCCC(O)CC(=O)Nc1ccc(NC(C2COC(=O)N2)=O)c(C)c1 16664,c1(CC(=O)NC(CC=C)CNC(=O)Cc2conc2C)ccc(O)nc1 16665,c1(C(=O)NC2(C)CN(C(c3c(C(=O)OC)coc3)=O)C2)c[nH]c(=O)cn1 16666,N1(C(CC2N(C)CCOC2)=O)CC2CC(NC(=O)C3=COCCO3)CC1C2 16667,c1(C(=O)NCCOC(CNC(C2C(C=C)C2)=O)(C)C)ccc(C)nc1N 16668,c1(CC)nc(C(=O)NC(C)C(C(C)C)NC(c2ccnn2CC(F)F)=O)c(C)o1 16669,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cc(OC)no3)=O)CC12 16670,C(=O)(CC(C)C(C)(C)NC(=O)C=C(C)COCC)NC1(CC=C)CCCC1 16671,C(C1CCCN1C(=O)C(SC)SC)=CC(N1C(C#C)CC1)=O 16672,c1(C(=O)NC(CNC(C(CCC)C(C)C)=O)(C)CO)cc(O)nc2cnccc12 16673,C(C1=NOC2CN(C(C3(C)CCCC3)=O)CC12)NC(C1(COC)CC1)=O 16674,c1(C(N2CCCC(CNC(C(CCC)C)=O)C2)=O)cc(F)ccc1NC 16675,C1(NC(c2c(C)ccn2C)=O)COC2(CNC(=O)CSc3n[nH]c(C)n3)CC1C2 16676,C1(C(=O)NCC2C=CCN2C(c2cnc(C3CC3)s2)=O)C(Cl)(Cl)C12CC2 16677,c1(C(N2CCOC(CCF)C2)C(=O)NCCC#N)cncc(C2CC2)c1 16678,S1(=O)(=O)c2ccc(c(F)c2)N2CCCC(C2)N1.C=C1CC(CN(C)C)C1 16679,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(=O)C=Cc3ncc[nH]3)CC2)C1 16680,C(CC1=CCN(CCOc2cccc(Cl)c2)CC1)NC(c1n(C)cc(Cl)c1)=O 16681,CC1=C(C(=O)N2CCC(O)(C(C)NC(C3(C)CC=CCC3)=O)CC2)CCCO1 16682,CN1CCC(C(=O)NCC2CCC2NC(c2ccc(CO)s2)=O)CC1=O 16683,n1(CC)cc(C(=O)NCCN(C)C(c2cc(N)c(Cl)c(O)n2)=O)c(O)nc1=O 16684,c1(-c2nnc(COC(C)C)n2C2CCNCC2(C)C)cc(Cl)cc2c1OCC2 16685,CC1CC2(CC(C(=O)N(C(C)CCNC(c3sc(=N)[nH]c3C)=O)C)C2)C1 16686,c1(C(CC)NC(=O)N(CC)Cc2cc(N(C)C)ccn2)cc(F)c(F)c(F)c1 16687,Cc1nc2cccc(C(N3CC(CNC(c4ccc(=N)[nH]c4)=O)CC3C)=O)c2[nH]1 16688,N1(C(c2nc(Cl)sc2Cl)=O)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16689,N1(CCOCCOC)CCC(NC(c2snnc2C)C)CC1 16690,c1(C(=O)NCC2(C(C)NC(COCC=C)=O)CC2)ncn2c1CCC2 16691,C1(CC(=O)NCC2CCCN2C(=O)CN2CSCC2=O)CCCCO1 16692,c1(C(N2CC3N(S(C(C)C)(=O)=O)C3C2)=O)cccc(Br)c1O 16693,C1(C(=O)NCC2N(C(c3n[nH]c(C)c3F)=O)CCC2)CCC2CCCCN12 16694,N1(C(COCCCC)=O)CC2CCN(C(C3(CCCF)CC3)=O)CCC2C1 16695,N1(C(C(N2CCC(O)CC2)C)=O)CCCCC(NC(c2cncn2C2CC2)=O)C1 16696,c1(CC(N2CC(NC(=O)CC3C4CC5C(C4=O)C35)C(CO)C2)=O)ccc(F)cc1Cl 16697,N1(CCC(=O)OC)CCCC2(CN(C(c3ccccc3C(F)F)=O)CCO2)C1 16698,N1(C(C(C)CN2CCOCC2)=O)CC2CC(NC(=O)C=Cc3nccs3)CC1C2 16699,N1(c2nnc(C(C)C)o2)CCC2(CCN(C(=O)CC(C)C3CC3)C2)C1 16700,N1(C(c2nc(OC)c(C)s2)=O)CCN(C(C2(C3CC3)CC2)=O)CC(CO)C1 16701,C(=O)(C(CO)C(C)(C)C)NC(C(=O)NCC(C(=O)OC)C)C 16702,N1(C(c2c(C)n[nH]c2)=O)CCCC(O)(CCNC(=O)C(O)C(F)(F)F)C1 16703,C=CC(C)CC(=O)N1CCC(O)(CN(C(=O)CNC(=O)CC(C)(C)C)C)C1 16704,C(CNC(C1(S(C)(=O)=O)CCC1)=O)(C(C)C(C)C)NC(c1cc(CCC)[nH]n1)=O 16705,c1(C(=O)NCCC2CC(NC(c3cc(F)cs3)=O)C2)nnc(C(F)(F)F)s1 16706,C1(NC(=O)NC(c2cccnc2)COC)CC(c2ccncc2)CN1 16707,c1(C(N2CC(CNC(C=C(C)Cl)=O)C3(C2)CC3)=O)cncc(N=[N+]=[N-])c1 16708,C1(NC(C2CC(CCC)OCC2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC(C)(C)C1 16709,N12CC3CN(C3C1)Cc1cc(Cl)cnc1OC(=O)CC2=O.C(COC)OC 16710,C1(C(=O)NC2CN(C)C2)CC12CN(C(c1cc(=O)cco1)=O)C2 16711,c1(OC)cc(C(=O)N(CCCNC(=O)COC2CC2)C2CC2)cc(Cl)n1 16712,c1(CC)ccc(C(=O)N(C)CCN(C)C(c2ccccc2CS(C)(=O)=O)=O)cn1 16713,c1(CNC2C(C(=O)Nc3cnn(CCC)c3C)C2)cc(Br)cc(F)c1O 16714,c1(C(=O)NC2CC(O)CN(C(c3ccnc(Cl)c3O)=O)C2)cnc2nccn2c1 16715,N(C(=NCCCC(C)(C)C)NC1CCC1)CC1C(C)COCC1 16716,C1(NC(C(=Cc2cccs2)C)=O)CC2(CCN(C(=O)CCc3n[nH]c(=N)s3)C2)C1 16717,C1(NC(c2n[nH]cc2Cl)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16718,C1(C(=O)NCCC(C(=O)NCCCSC)OC)CCCCN(C)C1=O 16719,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16720,C(CCCCC(=O)N1CC(n2cnnn2)C1)N(C(=O)Cn1cc(C#N)cn1)C 16721,O=C(N=c1[nH]cc(C2CCC2)s1)N1CCOCC1C1CCOC1 16722,C(=O)(C1=NOC2(CCN(C(c3cc(C)cnc3F)C(=O)NC3CC3)CC2)C1)OC 16723,C1(CNC(C2C(CC)C2)=O)CC(C(C)(C)C)CCN1C(=O)CCCc1nccs1 16724,N1(C(c2nccc(C#C)c2)=O)CC2CN(C(c3cc(C)cc(F)c3)=O)CCC12 16725,N1(C(=O)C=CSc2ccccc2)CCN(C(=O)Cc2csc(Cl)c2)C(CCO)C1 16726,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 16727,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(CC2CC(CC(C)(C)C)C2)=O)C1 16728,CC1CC(N(C)C(C2CC(NC(c3ccns3)=O)CCO2)=O)CC(C)C1 16729,CC(CC(C)(C)C)C(=O)NCCNC(C1(OCCF)CCC1)=O 16730,Cc1ccc(C(C)NCC2(CO)CCCCO2)cc1C1CC1 16731,CN1CCOC(C(=O)NCC(C2CCC2)NC(c2cnc(C3OCCO3)s2)=O)C1 16732,C#Cc1cnc(C(=O)NCC(C)CNC(=O)C(C)(CC2CCC2)OC)c(C)c1 16733,C1(=O)CCC(C(C)C)NC(=O)C(=O)C(C(=O)N2CCCC2)O1.C(C)(C)(C)OOC 16734,c1(CN2CCC(C)(N(C)C(C3CCC(C(=O)O)CC3)=O)C2)c(C)sc(C)c1N(C)C 16735,N1(C(c2ccc(NC)o2)=O)CCC(N(C)C)C2(CC2)C1 16736,N1(C(C=CCC)=O)CCC(C2CCCN(C(c3cc(C(F)(F)F)nn3C)=O)C2)C1 16737,N1(C(C(C)=CC)=O)CC2CC(C1)C(CO)C2NC(=O)C(C)(O)c1ccccc1.C1CC1 16738,c1(NC)ccc(C(=O)NC2CC(NC(=O)C(C(C)C)n3cncn3)C2)cc1 16739,C=Cc1cnn(C)c1C(=O)NC(C1CN(C(=O)C(C)NC(=O)C(C)(C)C)C1)C 16740,c1(C(=O)NCCNC(C2(n3cnnn3)CCOCC2)=O)cc2n(n1)CC(F)C2 16741,CC1CCN(C(=O)Cn2cnc(C#N)n2)CCN1C(=O)CC1CC2(CC2)CO1 16742,CC(C)(C(=O)N1CCC1CNC(c1cnc(S)nc1)=O)C1=CCS(=O)(=O)CC1 16743,c1(C(=O)NCC2C(CNC(C(c3cccc(C)c3)O)=O)C2)ncc(Cl)cc1F 16744,c1(C(N2C(CC(N3CCC(NC(C)=O)C3)=O)CCC2)=O)ncnc(O)c1F 16745,C1(C(N)=O)CCN(CC(=O)NCCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)CC1 16746,N(C1c2ccccc2CC1NC(=O)C(C)CS(C)(=O)=O)C(CC(CCC)(C)C)=O 16747,C(=O)(C1=CS(=O)CCC1)N(C(C)CNC(c1cn(C(C)C)nn1)=O)CC 16748,c1(C(N(CC(CC)NC(=O)Cn2nnc(C)n2)CC)=O)cccc(O)n1 16749,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16750,c1(OCC)cc(CO)c(-c2csc(C(=O)NCCCN(C)C)c2)cn1 16751,Cc1ccc(N)c(C(N2CCC(C(F)(F)F)C(NC(C3(CCO)CC3)=O)C2)=O)c1 16752,c1(NC(N2CCN(CCc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16753,c1(C(N2CCN(CCCNC(C(C=CCCC)O)=O)CC2)=O)cc(Cl)ncc1N 16754,C1(C)(CC)C=C(C(=O)NC2CN(Cc3c(C(=O)OC)nccc3)CC2C)C1 16755,C1(C(N(CC(C)O)CCNC(C(CC(C)C)N(C)C)=O)=O)CCC2C(C1)C2(F)F 16756,c1(OC)cc(C(N2CCCCC2C2CCN(C(=O)CC(C)=C(C)C)C2)=O)ncn1 16757,Cc1cc(C(=O)NCC(C)(O)C(=O)O)ccc1S(=O)(=O)N1CCOCC1 16758,N1(C(CCC)=O)CCCC1(C)CNC1CC(NC(=O)CC)C1.C(C)=O 16759,C1(C(N)=O)(NC(C)=O)CCN(C(=O)NN2CCC(Cc3ccccc3)C2)C1 16760,C(=O)(C1CCCc2nn[nH]c21)N(C)CCNC(c1cccn1-c1cnccn1)=O 16761,c1(C(N2CC(NC(c3cnc(Br)s3)=O)C(F)C2)=O)c(F)cc(C2CC2)cc1F 16762,C1(C(=O)NC2(c3ccc(F)cc3)CC2)CC2CC2N1C(=O)NCc1cnc(Cl)s1 16763,c1(C(C(=O)NCC(F)F)N(C)Cc2nc(CC)sc2)cc2c(s1)CCOC2 16764,C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccco1)N1CC(NC(N(C)C)=O)C1 16765,c1(CNC2CCC(NC(c3cnn4c3CCC4)=O)C2)ccc2c(c1)CCO2 16766,N1(C(c2ncc(C(=O)NC)nc2)=O)CC2CCN(C(=O)COC(C)=O)C2C1 16767,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(SC)o1)=O)C(COC)C 16768,c1(COC)nc(N(CCCCO)C)cc(N2CCCC(c3ccccn3)C2)n1 16769,N1(C(C(C2CC2)OCC)=O)CCN(C(c2c([N+](=O)[O-])cnn2C)=O)CC(C)(F)C1 16770,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16771,c1(COC(C(CC#C)c2ccccc2)=O)nn(C)c2c1CCC2 16772,C(=O)(CCCN(C)C)N(C(C)CNC(=O)C(C)(c1ccccc1)N(C)C)CC 16773,S(=O)(=O)(c1ccc(N2CCC(O)C(F)C2)c(C#N)c1)NC(c1cccs1)C 16774,c1(OC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F.C(C)(=O)N 16775,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16776,C(=O)(CCCCCO)NC1CC(C(=O)NC(c2ccc(Br)c(F)c2)C)C1 16777,C1(C(=O)NCC2CC23CC3(F)F)CCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 16778,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(C2(CC(F)F)CCC2)C)CCC1 16779,CC1CCC(O)C(C2CCCN2CC(=O)NC2CCOCC2)C1 16780,CC1CCc2[nH]nc(C(=O)NC3CC(NC(c4cc[nH]n4)=O)C3)c2C1 16781,CC1(C)C(C(=O)NC2(CNC(=O)Cc3csc(C(F)(F)F)n3)CCOC2)C1(C)C 16782,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(Br)cnc2O)=O)cc1N 16783,c1(C(N(C)Cc2cn(C)nn2)=O)cncc(N(C)C)c1.C1(=O)C(C2(O)CCC2)N1 16784,c1(OCC(=O)NCCCOc2cscc2Br)cccc(F)c1 16785,CCC(CCCC(=O)NC1CN(C)CC(F)(F)C1)NC(c1cnn(C)c1N)=O 16786,c1(CC)ccc(OCCC(=O)NC(C)C(C)NC(C2CCCCC2)=O)cc1 16787,c1(C(N2CC(C(C(=O)NC(C)(C)CC3CCCO3)(C)C)C2)=O)cn(C2CC2)cn1 16788,C1(C(=O)OC)CCN(C(C2C3CCCC23)C(=O)NC2(C)CC2)C(C)C1 16789,N#Cc1c(NC(=S)NC2(CO)CCOC2)ccnc1Br 16790,c1(CNC(c2cnn(C)c2N)=O)c(Cl)ccnc1F 16791,C1(C(=O)NCCC=C=C)CN(C(=O)Cc2ccccn2)CCN1C 16792,C1(=O)C(CC(C)C)N1.C1(CC)(CC)CCN1C(c1nnsc1C)=O 16793,c1(-c2nc(CCc3c(C)con3)n(CC(F)F)n2)ccc(F)c(C)c1 16794,C1(C(=O)NC2C(C#C)CCC2)C2CC3C(C2NC(C2CCCC(CC)C2)=O)C13 16795,c1(C(=O)NC2CCC(NC(c3ccc(Cl)o3)=O)C2)cc2ccc(F)cc2o1 16796,Cc1[nH]nc2c(C(N3CC4(CNC(c5c[nH]nc5Cl)=O)CCC3C4)=O)cccc12 16797,c1(-n2cc(C(C)N(C)C(c3nn(C)nc3Br)=O)nn2)cc(F)cc(F)c1 16798,N1(C(C(C)=C(C)C)=O)CC2CC(NC(=O)C=Cc3ccoc3)C1C2 16799,C(C)(C(C)(C)C(=O)NC1COC(C(F)F)C1)NC(c1cccc(CC)n1)=O 16800,N1(C(CCC=CC(C)C)=O)CC2CC(C)N(C(=O)Cc3ncc[nH]c3=O)C2C1 16801,c1(OC)ccccc1C(=O)NCC(CNC(=O)Cc1sc(SC)nc1C)OC 16802,C#CC1(OCC(=O)NCC(=O)NCc2noc(C(C)C)n2)COC1 16803,n1(CC(=O)OC)cc(CNC(=O)NCC2CC(N3CC(O)C3)C2)nn1 16804,CCC(C)CCC(=O)N1CC(C(=O)NCC(=O)OC(C)C)CC1(C)C 16805,N1(C(C2CCC(CNC(CCC(=O)NC)=O)O2)=O)CCCCCC(N(C)C)C1 16806,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(C1(C(F)F)CC1(F)F)=O)CO2 16807,C#CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C=CCN(CC)CC 16808,c1(NC(C2CCC2C(=O)NCCN2CCOC2=O)=O)cc(O)ccc1F 16809,c1(OC)cccnc1C(N1CCC(O)(CCNC(=O)C(F)(F)C2CC2)C1)=O 16810,C(=O)(C(C)C(O)CC(C)C)N1C2(CNC(Cc3c(C)ocn3)=O)CC(C1)C2 16811,C1(C(C(=O)NCCCOCC(C)C)NC(C(=O)OCC)=O)CC=CCC1 16812,c1(C(C)(C)C(=O)OC2COCCC2=O)ccc2nc(O)[nH]c2c1 16813,C1(C(=O)NCC2CN(C(C(C)(C)c3ccns3)=O)C2)CCCC2C1C2(F)F 16814,C1(=O)CCC(=O)N2CCN(CC2)CCN1C.CCC(C(=O)OCC)n1cncn1 16815,N1(C(c2c(C)nn[nH]2)=O)CCC(C(=O)NC(C2CCCCO2)C)=C(F)C1 16816,c1(C(N(CCOC)CCF)=O)conc1C(C)NC(=O)C(C)N(C)C 16817,C=CCC(F)(F)C(=O)NC1CN(C(c2nn(C)cc2Cl)=O)CC1CO 16818,c1(C(=O)N(CC2CCC(NC(C(CCC)(C)O)=O)CC2)CC)cccc2c1OCC2 16819,c1(C(N(CCNC(CC2C(CC)C2)=O)CCOC)=O)cnn(C(C)C)n1 16820,CC1(C)CCC(NC(=O)NC2CC(=O)N(CCc3cccnc3)C2)OC1 16821,C1(n2c(-c3ccnn3N3CCCCC3)nc(C3CCOC3)n2)CCC(F)(F)CC1 16822,C1(NC(C2N(C(c3nn(C)c(F)c3)=O)CSC2)=O)CCCC(O)C1O 16823,N1(C(c2nc(CCCCC)sc2)=O)CCCC(CNC(=O)COC)C1 16824,C1(C(=O)OC)CCC2(CCN(c3ncnc4sc(C)nc34)CC2)O1 16825,C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)NC(=O)Cc2nc(C)sc2C)C1 16826,C12(C(=O)NC(CC)CN(C)C(C3CC(C)(C)C3)=O)CC1COC2(C)C 16827,C1(NC(CCNS(CC)(=O)=O)=O)CC2CC(C1)N(C(c1c(C)coc1C)=O)C2 16828,C1(F)(C(C)NC(C2CN(c3cn(CCCOC)nc3)C(=O)C2)=O)CC2(CCC2)C1 16829,C1(CC(=O)OC)CCC2(CCC2)C1NC(=O)CC(=O)NC(c1ccc(C)cn1)C 16830,c1(CSCC(=O)NC2(C3CCCN3C(c3cnsn3)=O)CC2)cccnc1 16831,c1(OC)cccc(C2=NOC(C(=O)OCC#N)C2)c1.C1CCCC1 16832,c1(NCC23CC(C(=O)Nc4ccn(CC)n4)(C2)C3)ncc(C)cc1I 16833,C(=O)(NNc1cc(Br)ccn1)c1scc(-c2cc(C)c(C(=O)N(C)C)nc2)n1 16834,C1(CNC(C2(C#C)CCC2)=O)(COC)CCCN1C(=O)C(CO)N(C)C 16835,CC1(CNC(=O)CCOC2CCCOC2)CCN(C(C2(C)CC=CCC2)=O)C1 16836,CC(O)CC(C)(C)CNC(c1csc(-c2ccccc2)n1)C 16837,CC(C(=O)NCC1CCC(NC(C2C=CC=CC=C2)=O)CC1)C(F)F 16838,N1(C(C(C(C)C)SC)=O)CC2CCCC(NC(=O)CCc3cn(C)nn3)(C2)C1 16839,C(=O)(CC=C(Cl)Cl)NCC1(OCC#C)CN(C(=O)C=Cc2cnc(C)s2)C1 16840,c1(C(N2C(CN(C(C3CCCOC3)=O)CC)CCCC2)=O)c(N)cc(C)cc1F 16841,C12(NC(c3cnccn3)=O)CCOCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 16842,N1(C(CN(CC(C)(C)C)C)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CC2)C1 16843,N1(C(c2cnc(C)[nH]2)=O)CCC2(NC(c3nccc(Cl)c3F)=O)CCCCCC12 16844,Cc1ccc(SCCC(=O)NC2CCCN(C(c3cccc(CF)c3)=O)C2)cc1 16845,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16846,c1(NC(C2CC3CC3N2Cc2cc(O)cc(Cl)c2)=O)ccc2cnccc2c1 16847,c1(C(=O)NC(CC)CN(C(C2CCCS2)=O)CC)cnc2[nH]c(C)nc2c1 16848,C1(OC)CC(NC(=O)CC2(C)CCN2C(c2scc(C)c2C)=O)C1(C)C 16849,N1(C(c2cc(CCC)on2)=O)CCCC(C2(NC(=O)C(F)n3ccnc3)CC2)C1 16850,C(c1cccc(C#N)c1)=CC(N1CCN(C(C(CC)N(CC)CC)=O)C2C1C2)=O 16851,c1(C(=O)NC(CC=C)CNC(=O)C(F)(F)COCC)ccc(N(C)C)cc1 16852,C(=O)(C1=NN2CCC(C)N=C2N1)N(C1CCN(C(C(CC=C)CC)=O)C1)CCO 16853,c1(C(=O)NCCCNC(CC2(OC)CC2)=O)cc(=O)n(-c2ccccc2)[nH]1 16854,c1(C(=O)NC(C2(C(=O)NC3CCN(C)C3=O)CCCO2)C)ccccc1CO 16855,C(=O)(C(F)CC(CC)CC)N(C(C)C(N1CCC2(C=CCO2)C1)=O)CCC 16856,C1(NC(C(CCC)(C)C)=O)CCC2CC1CN2C(c1ccc(F)cc1OC)=O 16857,c1(OC)cc(CN2CCCC(C)(C(=O)O)C2)ccc1OCCO 16858,c1(C(c2nnnn2CC2CCCO2)NC2CC=C(C)CC2)cccc(C)c1O 16859,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1cccnc1C 16860,c1(C(=O)NC2(CF)CCN(C(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16861,c1(C(=O)NC2CCN(C(C(COC)C)=O)CC2F)nc2cnccc2s1 16862,CS(=O)(=O)c1ccc(Cl)c(C(=O)N(C2CC2NC2CC2)C(=O)CN2CCOCC2)c1 16863,C1(NC(C(CC)NC(N)=O)=O)CCC2CN(C(C3CCN(OC)CC3)=O)CC2C1 16864,C1(C)(C(N2CC(OCC(=O)N(CC(C(C)O)O)C3CC3)C2)=O)CCN(C)CC1 16865,C(=O)(C1CCCc2nc[nH]c21)NCCCCN(C(=O)CNC(C1(C)CCC1)=O)C 16866,C1(C(=O)NCCC2COCCN2C(C2CCSCC2)=O)Cc2ccccc2O1 16867,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16868,N1(C(c2n(CC)nc(C3CCCC3)c2)=O)CC2CCC(NC(=O)OC)CC2C1 16869,c1(C(=O)NC(CC)CN(C(=O)COCC(C)C)C)cc(C)nn1C1CC1 16870,c1(C(=O)NC2C(NC(C3(CCC)COC3)=O)CCC2)c(C)cc[nH]c1=N 16871,c1(C(N2CCC(C(C)(C)NC(=O)CCN3CCC3)CC2)=O)ncc(Cl)cc1F 16872,C1(CC)(CNC(C2CC2c2cncs2)=O)CN(C(=O)CC2CCOCC2)C1 16873,c1(C(=O)NC2C(NC(CC(C)C3CCC3)=O)CCCC2)ncc2cc(Cl)ccn12 16874,N#Cc1cncc(CC(=O)NC2(CO)CCN(C(c3cnsc3)=O)C2)c1 16875,C(=O)(C#CC(C)(C)CNC(=O)Cc1cn(C)cn1)NC(C(=O)OC)CCF 16876,c1(C(=O)NC2CC(OCC(=O)N(C3CCSC3)C)C2)cnoc1C1CC1 16877,C(=O)(C(C)(C)C(C)NC(=O)COc1cc(C)on1)NCCOCCC#C 16878,c1(OC(c2cc(OC)ns2)C(=O)N(C)CC2OCCN(C)C2)ccccc1Cl 16879,N1(CC(=O)Nc2cccc3ccccc23)CCn2cccc2C1c1ccncc1 16880,C(N=c1[nH]c(C2CC2)ccc1C(=O)O)C1CCN(C(C=NOC)=O)C1 16881,C1(CN(C)C(C2CC3C=CC2C3)=O)COCCN1C(=O)Cn1cc(Cl)cn1 16882,N1(CC)C(=O)CCC1C(=O)NCC12CC(NC(C3CCC34CCC4)=O)(C1)C2 16883,C1(NC(=O)Cc2ccc(Cl)cc2Cl)CC2CC(C1)N(C(=O)C(F)n1ccnc1)C2 16884,c1(C(=O)NCC2N(C(CNC=O)=O)C3CCC2C3)cc2c(F)cc(Cl)cc2[nH]1 16885,C1(CNC(c2cnc(CC)o2)=O)CCN(C(=O)CC2C=CCC2)CC1C 16886,c1(CN2CCC(C(=O)Nc3cc(Cl)cnc3Br)C(O)C2)ccc(F)c([N+](=O)[O-])c1 16887,C#CCCCCCC(=O)N1CC(C2CC2C(=O)NCCCCCCCCC=C)C1 16888,c1(C(=O)NCC2N(C(C)=O)CC(C(F)(F)F)OC2)ccc(F)cc1C(C)=O 16889,c1(NC(c2cccc(NC(CN(C)C)=O)c2)=O)ccc(CN2CCCC2)c(F)c1 16890,N1(C(c2c(C)[nH]nc2C(C)C)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 16891,C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(C)C)C(=O)Nc1cc(C)cc(O)c1 16892,C1(C(=O)NCCOCCNC(c2n[nH]cc2Cl)=O)CCC2(CCOCC2)CO1 16893,c1(OC)ccc(C(C(=O)N(C(C)CNC(c2cocn2)=O)CC)OC)cc1 16894,C1(C(=O)NC2CC3CNCC23)CC2(CCCCC2)CN1 16895,c1(NCC2(NC(C3(CF)CCC3)=O)C(C)CCCC2)ncc2c(n1)CCOC2 16896,c1(C(=O)NC2C(C)CCN(C(=O)CCCCN(C)C)C2)sc2nccnc2c1N 16897,CC(C)(C)C(C)(C)C(=O)NCC1CCC(C(N2C3C=CCC2CC3)=O)CO1 16898,N1(C(c2cc(C)on2)=O)CC(C)CCC1CNC(=O)CCC(=O)c1ccc(C)s1 16899,C1(NC(c2cc(C)c(O)cc2)=O)CC2CCC(C1)N2C(=O)CCCc1cnn[nH]1 16900,C(Cc1ccco1)(C(=O)NC1CCCC1NC(=O)C=CSc1nc[nH]n1)N(C)C 16901,c1(C(N2CC(NC(=O)C(C)(F)F)CC(C)C2)=O)cc2c(Br)cccc2c(=O)o1 16902,c1(N(C(=O)NC(C)CCCc2ccccc2)C)ccc(F)cc1 16903,C1(NC(=O)C=CC2CC2)CCC1C(=O)NCC(c1cnc[nH]1)O 16904,c1(OCCC(=O)NCC2COCCN2C(c2cccc(F)n2)=O)cccc(F)c1 16905,Cc1ccc(S(=O)(=O)NCc2cnc3c(c2)COCC3)cc1[N+](=O)[O-] 16906,c12ccc(cn1)N(C)C2.C(=O)(C(=O)NC(=O)NCC(=O)OC(C)(C)C)OCCCC 16907,C12CCCC3(CN(C3)C1=O)O2.C#CC(C)(C)C(=O)NC1(C(O)C(F)(F)F)CC1 16908,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 16909,C(=O)(CC(C)CC(C)C)NC1C(CC(=O)N(C(CCC(C)C)C)C)CCC1 16910,C(=O)(C(CCC1CCC1)NC(=O)NCc1cnsc1)OC 16911,Cc1ncccc1C(N1CCC(F)(CNC(=O)C(C)(C)CN(C)C)C1)=O 16912,c1(CCCC(=O)NC(CNC(C2CCC(C)C2)=O)CO)ccc(F)cc1 16913,C1(C)(C(=O)NCCN(C(CC2CC(=C)C2)=O)CC)CCOCC1 16914,C12(C(=O)OC)CCCC1(C(=O)N(C)CCNC(C1CC1(C1CC1)COC)=O)C2 16915,C12(CCSCC(N3CC(C(=O)OCC)C3)=O)CC1CNC2=O 16916,Cc1coc(C2CC2)c1C(=O)NCCN(C(=O)COC1CCOC1)C1CC1 16917,c1(C(N2C(CNC(CS(C)(=O)=O)=O)CCCC2)=O)c(Cl)ccc(F)c1F 16918,C1(C(C)NC(c2ccsc2)=O)CC(NC(=O)CN(C2CCC2)C)C1 16919,c1(CNC2(N3C(=O)OCC3)CC2)cn(C2CC2)nc1C1CCCOC1 16920,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 16921,C1(CN(CC(=O)NC(c2ccccc2)CC)C)(OC)CCOCC1 16922,C1(CC(=O)NC(C)CO)CN(C(=O)CC2(O)CCC2)C1 16923,CC(C)C(N=[N+]=[N-])C(=O)NCc1cc(C(=O)N(C)C(c2cccnc2)C)no1 16924,C(=O)(C#CC1CCCCC1)N1C(C2(C(N3C(C)C(=O)N(C)CC3)=O)CC2)CCC1 16925,c1(CNC(C(C(C)C)NC(C2CC(C)(C)CCO2)=O)=O)cncc(C#N)c1 16926,C1(SC)CN(C(=O)CCOC2CCN(C)CC2)CC1NC(C1CCS(=O)(=O)C1)=O 16927,CCCC(O)CC(=O)NC(C)(C)CNC(=O)CCc1ccc(C(C)C)cc1 16928,Cc1nc(=N)[nH]cc1C(N1CCN(C(C2CC2C)=O)C(c2ccccc2)C1)=O 16929,C#CCC(CC(=O)NOCCC(F)(F)F)NC(=O)C=Cc1nc(C)cs1 16930,N1(C(=O)C=Cc2ccsc2)CC2CN(c3ncncc3F)CC2C1 16931,c1(OC)cccc(C)c1NC(=O)CCCCCNC(C1NC(=O)OC1C)=O 16932,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2cc3c(C)[nH]nc3s2)=O)CC12CCC2 16933,N1(C(C(CC(C)C)O)=O)CCC2(CCC1)CN(C(C1CCCN(C(N)=O)C1)=O)C2 16934,c1(C(=O)NC(C)C(CO)NC(=O)CCc2ccnn2C)cncc(Br)c1 16935,CC1N(C(C2CCCN(C(c3nc(=N)cc[nH]3)=O)CC2)=O)CCC1(C)C 16936,N1(C(=O)Cc2ccncc2Cl)CCN(C(c2cccc(Br)c2)=O)C2CC12 16937,C1(CCC(=O)NCC(C)NC(C2CC(C)(C)C2)=O)CCCC(O)C1 16938,N1(C(c2scc(C)c2Cl)=O)CC(C)CCC1CNC(=O)C(C)CC(F)F 16939,C(=O)(CCC(=O)NC(C)(C)CC(=O)N1CCCCC1C(C)C)NCC 16940,C12(C(N(CCCNC(CCC=C(C)C)=O)C)=O)CC3CC1C2C3(F)F 16941,N1(C(c2n(C(C)(C)C)ncc2)C(=O)NC2CCC2)CCC2OC(=O)OC2C1 16942,c1(C(N(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)CC)=O)cncc2ccccc12 16943,c1(OC)cc(C(=O)N(CCCN(C)C(C2(C)CC=CC2)=O)C)on1 16944,C1(CC)CCN(C(C2CC(N(C)C(C34CCC(CC3F)C4)=O)C2)=O)CCO1 16945,N1(C(Cn2c(C)ncc2)=O)CCC(NC(C23CC2CNC3=O)=O)CC1C 16946,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)CC2COC(=O)C2)cc1Br 16947,c1(NCC(C(=O)OC)O)nc2nc(C(F)(F)F)ccn2n1 16948,C(=O)(C(C)(C)C(=O)NCC1(F)CCCN(C(=O)CC2CC(C)(C)CCO2)C1)NC 16949,c1(C(N2C(C)CC(CNC(c3cncc(F)c3)=O)CC2)=O)nn(C)c2c1CCC2 16950,C1(C(=O)NCCC(O)CNC(c2cnccc2C)=O)(COC)CCCCC1 16951,N1(C(CCCC2C(C)C2)=O)CCN(C)CC1C(=O)N(CCO)CC1CC2CCCC12 16952,C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(N(C(=O)CC2CCCC23CC3)C)C1)=O 16953,C1(C(=O)NC2(C(=O)NCCCc3cc(C)no3)CC(F)C2)CC(C)CCO1 16954,C=CC(C)CC(=O)N(CCNC(=O)C(n1ccc(C2CC2)n1)C)CC1CC1 16955,C1(C(=O)NC2CC(C(C)NC(c3cccc(C4CC4)c3)=O)C2)CC2CCCC2C1 16956,c1(C(N2C(C(N=c3ccn(C)[nH]3)=O)CC(F)(F)C2)=O)cc(Cl)cc2nc[nH]c12 16957,N1(C(CCC#CC)=O)CCCC(CNC(=O)C(C2CCCCCC2)C)C1C 16958,N1(C(CC)=O)CC(N=c2nc3scnc3c(NCCS(C)=O)[nH]2)CC12CCC2 16959,CC(O)C(C(=O)NCCCC(C)NC1CC1)NC(C1(C(=O)OC(C)(C)C)CC1)=O 16960,CC(C)C(CN(C)C)C(=O)NC12CCC(CC1NC(=O)CC1CCOCC1)C2 16961,c1(C(=O)NC(C)C(CO)NC(c2ncoc2C(F)(F)F)=O)cc(=O)n(C)cn1 16962,c1(C(=O)NCC(C2CC2)NC(CC2C(C)(C)CCO2)=O)cc(S(C)(=O)=O)ccn1 16963,C1(NC(C2N(CC)CC2)=O)CCCC(CC(N2CC(C(N)=O)C2)=O)C1 16964,C(=O)(C(C(C)(C)C)c1ccccc1)N(C)CC1C(O)CCN1S(=O)(=O)c1cccs1 16965,C(=O)(C(C)CC(C)(C)C)N1C(Cn2cc(-c3c(C)nc[nH]3)nn2)CCC1 16966,N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CCCN2C)=O)C(C)C1 16967,C1(CC(=O)NCCCN(C(CNC(=O)NCC=C)=O)CCOC)CCCSC1 16968,C(=O)(C(O)CC(F)F)NCCN(C(CCCc1scc(C)n1)=O)C 16969,N1(C(C=C(CCC)CCC)=O)CCN(C(=O)CC2CCC(=O)N2)C(CC)C1 16970,c1(C(N2CC(C)(NC(=O)CN3CCOCC3)C2)=O)ccnc(C(C)(F)F)c1 16971,C1(Nc2cc(N(C)CC3COCCOC3)ncn2)CCN2CCCC12 16972,c1(C(N(c2ccccc2)S(CC)(=O)=O)=O)ccc(C#N)n1C 16973,c1(CCC(=O)NC2CC(CNC(CCSC)=O)C2)cc(Br)ccc1OC 16974,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCN(C(c2cscc2C)=O)CC1C(C)C 16975,c1(-c2cn(CC(=O)Nc3ccc(N4CCC4CO)nc3)nn2)c(F)cccc1Cl 16976,c1(CCCNC(=NC)NCC2COC(=O)N2)cc(Cl)ccc1Cl 16977,C#CCC(O)C(=O)NC1CN(C(=O)CCSc2ccccc2)CC1CO 16978,Cn1cncc(C(N2CCC(Cn3cc(Cc4ccncc4)nn3)CC2)=O)c1=O 16979,C1(NC(c2ccc(CC)o2)=O)CCC2(CCN(C(=O)CCNS(=O)(=O)CC)C2)C1 16980,S(=O)(=O)(c1cccc(N2CCC(O)C2)n1)N(C)Cc1ccc(C)c(C)n1 16981,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 16982,N1(C(C2C(COC)C2)=O)CCN(C(=O)COCC2CC2)C(CCO)C1 16983,C(=O)(N=c1cc(Cl)nc(C)[nH]1)c1c(C(=O)OC)nc(C(F)(F)F)cc1 16984,N1(C(C(Cc2cn[nH]c2)NC(CC2(OC)CCC2)=O)=O)CCC2(CC2)C1 16985,C1(C(=O)NCC2CN(C(C3C(C#C)C3)=O)C2)(NC(C)=O)CCCC1 16986,c1(NCCC(=O)N(c2c(C)cccc2C)C2(C)CCCN2)ncc2c(ccn2C)n1 16987,N1(C(c2c[nH]c(=NC)o2)=O)CC(C(=O)NCCC(=O)NC)C2(CC2)C1 16988,C1(NC(c2cccnc2Cl)=O)CC2CC1CN(C(C1(n3nccn3)CC1)=O)C2 16989,Cc1nc(NC2CCCN(C(=O)Cn3nnnc3C(C)C)C2)cc(Cl)n1 16990,c1(C(=O)NCCCN(C(c2c[nH]c(C#N)c2)=O)CC)ccc2c(c1)COC2 16991,c1(C(COC(C)C)NC(C(=O)Nc2cc(C)c(C(=O)O)s2)=O)ccc(F)cc1F 16992,C(=O)(C1=C(Cl)CCC1)NCCC(C)(C)NC(c1ccn(CC)c1C)=O 16993,CC(C)C(O)C(F)(F)C(=O)N1CC(CN(C(=O)CC2CCC2)C)C1 16994,c1(N2CCC(NC(c3cn(CCCC)nn3)=O)C2)ncnc2ncn(CC)c12 16995,C(=O)(CC(F)(F)F)N(c1cccc(-c2noc(CC3(c4ccccc4)CC3)n2)c1)C 16996,CC1=C(C(=O)N2CCC(F)C(NC(=O)Cc3cnc(C)o3)C2)S(=O)(=O)CCO1 16997,N1(C(C2C(C(C)C)CCC2)=O)CCN(CC(=O)NCCn2cccn2)CC1 16998,C1(CC)CCN(C(C2CC(C#N)(OC)C2)=O)C(C(=O)NCCc2nccn2C)C1 16999,N1(C(C2(C)COC2)=O)CCC(C#N)(NC(c2ccc(Br)cn2)=O)C1 17000,C=CCCCCC(=O)N(C1CN(C(C2CC2C)=O)C(CC)(CC)C1)C 17001,N1(C(c2ccc(C3(C)CC3)cc2)=O)CCN(C(=O)CCCF)C(CO)C1 17002,Cn1cnc(C=CC(=O)NCCC2COCCN2C(=O)CCCc2ccsc2)c1 17003,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(Cc3ccc(Cl)nn3)CC2)C1 17004,Cc1ccc(-n2cc(CNC3CCC(NC(c4csc(C)c4C)=O)C3)nn2)cc1 17005,c1(C(N2CCC(COC)(CNC(C3CCC3)=O)CC2)=O)nccc2ccn(C)c12 17006,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17007,C#CCC(C)C(=O)NC(CNC(c1cnc(C(C)OC(C)(C)C)s1)=O)CC(C)C 17008,c1(CC(N2CC(CNC(C3C(C(=O)OCC)C3)=O)C2)=O)ncc(F)cc1F 17009,C1(CNC(=O)CC2CCOCC2)CCN(C(C2CC3(CCC3)C2)=O)CC1O 17010,C(=O)(CC(CNC(C)=O)CC(C)C)N(C)CC1CCN(c2cc(OC)ncn2)C1 17011,C1(NC(=O)CCCCCn2cc(C3CCOC3)nn2)CCNCC12CCC2 17012,C1(CNC(=O)Cc2cccs2)CCC1C(N1CCC1C(N)=O)=O 17013,C(=O)(C(C(C)C)NC(=O)CN1CCC(=O)CC1)NC1(CC)CC1 17014,c1(C(N2CCCC(N(C(C3C(C)C3)=O)C)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17015,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17016,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17017,C(=O)(CCOCC(O)C1CC1)N(C)N(C)C(C1(OC2CCCC2)CC1)=O 17018,c1(C(c2nnnn2C)NCC2(C(=O)OC)C=CCC2)ccc(C)c(F)c1 17019,c1(Cn2cc(C3(C)N(C(c4[nH]c(=NC)sc4)=O)CCC3)nn2)ccc(F)cc1Cl 17020,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17021,CCCC(CCC)CC(=O)NC1(C(=O)NCCCC(C)CO)CCSC1 17022,Cc1oc2ccccc2c1C(N1CCCC(CNC(C2(C)CCNC2=O)=O)C1)=O 17023,N1(C(C(n2ccnn2)C)=O)CCC(C)(C)C1C(=O)N(CCCCCO)C 17024,c1(OC)ccc(NC(=O)CC2CN(C(c3ccc(C)cc3)=O)CCC2C)c(C)c1 17025,c1(OC)ccc(F)c(CC(=O)NCCC(C)NC(=O)C(F)CC2CCCCC2)c1 17026,C(c1cccc(F)c1F)=CC(=O)Nc1c(OCCOC)cc(Cl)cc1 17027,c1(C(=O)N(c2cn(-c3cccnc3)nn2)CCC2CCCO2)ccc(Cl)cc1 17028,N1(Cc2nc(C(CCC(=O)OCC)C)sc2)CCS(=O)(=O)C2COCCC12 17029,C1(CC(=O)NCC2CN(C(c3nc(COC)sc3)=O)C2)CCCCC1C 17030,c1(COCC(=O)NCC2C=CCN2C(=O)CCC2CCCO2)ccccc1Cl 17031,c1(C(C)(C)NC(=O)NCCC23CC(CO2)C3)ccc(O)cc1F 17032,CCCCCCCCCC(=O)N1CCC(O)(CNC(c2csc3nccn23)=O)C1 17033,c1(NCCc2c(C)ncs2)cc(N(C)Cc2cccc(F)c2)ncn1 17034,c1(C(=O)NCCCN(C(C2(C=C)CC2)=O)CCO)cccc(CSCCOC)c1 17035,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(C3CC3)c2)=O)CCCO1 17036,c1(C(N(CC(C)NC(=O)CCc2nnc(C(F)F)o2)C)=O)ccc2occc2c1 17037,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17038,CC1(C)CC(NC(C2CCC(OC(F)(F)F)C2)=O)CN1C(=O)Cc1cncs1 17039,C1(C(=O)NCc2nc(C)on2)CCC=CC1NC(c1csnn1)=O 17040,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17041,Cc1ccc(C(=O)N(C2(C(=O)NC=O)CC2)C)c(F)c1.C(C(C)C)C(C)C 17042,c12cccnc1C(=O)N2.C1(CNC(C2(CCC)CC2)=O)CC(CC)(CC)C1 17043,CC(CCS(=O)N=c1nc2scnc2c(N2CCC(S(=O)(=O)C(F)F)C2)[nH]1)C1CC1 17044,CC1CN(c2nnc(C(F)F)s2)CC1NC(c1cccc(N(C)C)c1)=O 17045,c1(CC(=O)NCCC2CN(C(=O)C=CCO)C2)ccc(Cl)c(F)c1 17046,c1(CC(=O)NCCNC(C(c2c(OC)cccc2)C)=O)nn(C)c(=O)n(C)c1=O 17047,C#Cc1ccc(C(=O)NC(CN(C)C(c2cnn(C(C)(C)C)n2)=O)CC)c(C)c1 17048,C1(NC(=O)CCCC2CCCC2)CCN(C(C2CC(CC3CC3)C2)=O)CCC1(F)F 17049,CC1CCN(C(C2CCCC(O)C2)=O)C1CNC(=O)CC(O)c1ccccc1 17050,C1(C(=O)NCc2nc(C)c(Br)cc2)CCC2(CN(C(=O)CC(C)O)C2)O1 17051,C1(CN(C(CCN(CCC)C)=O)C)CN(C(C2COCCN2C)=O)CCO1 17052,Cc1sc(C2CCN(C(c3ccc(C)s3)C(=O)NCCCF)CC2)nc1C(=O)O 17053,C1(C(=O)Nc2ccc(C3CC(=C)CN3C(C)=O)cc2)CCOC12CCOC2 17054,c1(OC)cc(O)c(CN2CC3(CC3)CC2C(=O)NCc2ccc(C)o2)cc1Cl 17055,C1(C(=O)OC)COCC2(CCN(C3CCC(C(=O)OC)CC3)C2)O1 17056,c1(C(=O)NC(C)(C)CCNC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17057,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17058,c1(OC)nc(N2CCC(F)(C(=O)Nc3cccc(-c4nnco4)c3)C2)ncc1Br 17059,C1(CNC(CNC(CC)=O)=O)CN(C(=O)C(C)(C)N(C)C)CC12CCC2 17060,CCC(C(=O)N1CC(O)(C(C)(C)C(=O)OC)C1)C(C)O 17061,CC1CC(NC(c2cc(CO)on2)=O)CN1C(c1cnc(-c2ccccc2)s1)=O 17062,CC(C)(C)C(CN(C(=O)C(O)CC#N)C1CC1)CO 17063,C1(NC(=O)Cn2cc(Cl)cn2)CN(C(C2CC(CF)C2)=O)CC2(CC2)C1 17064,c1(C(=O)NCC(C(C)C)NC(=O)C=CBr)cccc(C2CC2)c1Cl 17065,C(c1c(C)noc1C)=C(C)C=O.C(CCN)N(C)C(C(C)(C)C)=O 17066,c1(NC)cc(N2CCC(CCNC(=O)CC(C)(C)OC)(OC)C2)ccc1[N+](=O)[O-] 17067,CCCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)CCc2nnc(C)n2C)C1 17068,CC(C)C(C(=O)NCC(C)(CO)NC(c1csc(Br)n1)=O)N(C)C 17069,c1(C(N2CC(NC(C(C)=C(CC)C)=O)C3(C2)CC3)=O)nc2cccnn2c1Br 17070,N1(CCNC(=O)CCOC)CCN(C(C2CC2NC(COCC=C)=O)=O)CC1 17071,c1(C(=O)NCC2CCCC(NC(CSC)=O)C2)c(C)ccc(N)c1C 17072,C1(CNC(CCOCCC)=O)CN(C(c2cc(OC)ccn2)=O)CC1(C)C 17073,C1(NC(C=CSC)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCC12 17074,C1(F)(CNC(COCCC)=O)CC(NC(c2occc2C2CC2)=O)C1 17075,C(=O)(CC(CC)CC)NC(CSCC)C(=O)NC(c1cnn[nH]1)C 17076,CCC(CC)CC(F)C(=O)NC1(C)CCC(C(N2CCCN(C)CC2)=O)C1 17077,c1(C(N2C(C(N(C)CCC3CCCC3)=O)C=CC2)=O)ccncc1F 17078,C1(C(NNC(=O)N(c2c(C)cc(Br)cc2F)CC(C)C)=O)CCc2ccccc2C1 17079,N1(CC(C)N(CC)CC)CCC(NC(c2sccc2C2CC2)=O)CC1 17080,c1(OC)c(Cl)cc(Cl)c2c1CCN(c1ccc(S(=O)(=O)N3CCCC3)c(Br)c1)C2 17081,C#CCCCCCCC(=O)NC1(C)CN(C(C2CC3C(C2)C3(F)F)=O)C1 17082,N1(C(CCOC)=O)CC2CCCC(CNC(=O)C=CS(C)=O)(C2)C1 17083,c1(CNC(C(C)N(C(=O)CCC(N)=O)C)=O)cccc2occc12 17084,c1(-c2nc(C3OCCN(C)C3)nn2-c2ccccc2)coc(S(C)(=O)=O)c1 17085,C(C(C)(C)CCNC(c1ccnc(O)c1)=O)NC(c1cn(CC=C)nc1)=O 17086,C(=O)(C(F)(F)C1=CCOCC1)N1CCC(CNC(Cc2n(C)ncc2Cl)=O)CC1 17087,C(c1cn(CC(=O)N(C(C)CN(C(=O)C2=CCCC2C)C)C)c(=O)nc1O)=CC 17088,S(=O)(=O)(c1cccnc1N1CC2NC(=O)OC2C1)NCC(c1ccsc1)N(C)C 17089,C1(C(N2C(C)CN(C(=O)CC#N)C(C)C2)=O)=CC=CC=CC=C2N(C=C1)C2=O 17090,N1(C(CSC)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 17091,CN1CCN(C(=O)COc2cccc(CO)c2)C(CNC(c2cccnn2)=O)C1 17092,c1(NC(C2C3CN(C(CCCSC)=O)CC32)=O)ccc2ncnn2c1 17093,c1(CCNC(C2(O)CN(C(C(C)(C)C)=O)C2)=O)ccccc1O 17094,c1(C(N(C(C(=O)NC(C)Cc2nc(CO)n[nH]2)C2CC2)C)=O)cc(C#N)cs1 17095,N1(C(C2(CCNC(C3CCCC(C)C3)=O)CC2)=O)CC2(CCC(=O)NC2)C1 17096,c1(OC)ccccc1C(O)C(=O)NC1CCC1CNC(c1ccc(Cl)cn1)=O 17097,C12(C(N3CC4(CN(C(CC(=O)NCC)=O)C4)C3)=O)CC=CCN1CCC2 17098,c1(C(c2nnnn2C2CCOC2)NC(c2ncc(C)s2)C)cc2ccoc2cc1C 17099,N1(C(C2(COC)CCCO2)=O)CCCC(N(C(=O)CCN2CCC2)CCO)C1 17100,N1(C(CCC#C)=O)CC2=C(C1)CN(C(=O)CCCCNC(=O)OC(C)(C)C)C2 17101,C(C)(C)(CC(=O)NCc1ncccc1C(N1CC(C)(CO)C1)=O)OC 17102,c1(C(N2CCN(C)CC2)=O)cccc2nc(C(=O)NC3CCCNC3)cn12 17103,n1(CC)cnc(C(=O)NC(C2CCCN2C(=O)C(F)=CC2CC2)C)n1 17104,C(=O)(CCCC(F)(F)CO)NCC1(NC(C(CCCC)N(C)C)=O)CC1 17105,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1F 17106,S(=O)(=O)(c1cccc(F)c1)N(C(C)C(=O)Nc1ccccc1)C1CC1 17107,N1(C(CN(C(C)=O)C)=O)CCCC(CN(C(=O)CCc2ccnc(OC)c2)C)C1 17108,n1(CCOC)ncc(C(=O)NCC(C2CCC2)NC(C2C3CCN2CC3)=O)c1C 17109,N1(C(C2(CC)CC(F)(F)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3)C14)=O)C2 17110,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ncn3)=O)C2CC1 17111,N1(C(C2CC(C3CC3)=NO2)=O)CCC2C(CCCN2C(C2CCCC2)=O)C1 17112,c1(COC(C2C(=C)CN2C(=O)OC(C)(C)C)=O)cnc(F)c(C)c1 17113,c1(C(=O)NC2C(C)CN(C(C34COCC(C3)C4)=O)C2)cccc(C2CC2)c1Cl 17114,C1(NC(C2(CC)CC2)=O)CCC(CNC(=O)COCC2CCCOC2)C1 17115,c1(C(C)(C)NCC2CC(OC(C)=O)C2)ccccc1C(=O)O 17116,Cn1nc(O)cc1C(N1CCOCC1CNC(c1ccc(CCF)cc1)=O)=O 17117,C(N=c1nc2[nH][nH]cc-2c(O)n1)C1(NCc2cccc(OCCC)c2)CC1 17118,c1(C2(CC(=O)NC3C=CCN(C(Cn4nc(C)oc4=O)=O)C3)CC2)c(Cl)cccc1Cl 17119,CC(C)CC(CNC(=O)CCc1cn(C)cn1)NC(C1CC(CF)C1)=O 17120,N1(C(C2CCCC(C#N)C2)=O)CCC=C(C(=O)Nc2cnn3cccc3c2)C1 17121,Cc1c(Cl)ccnc1C(N1CCCCCC1CNC(C1(F)CCCCC1)=O)=O 17122,C(C)(C)(CC(F)C(=O)N1CC2CC2C2CC12)NC(C1C(C(=O)OC)C1)=O 17123,CCCC(C)(C)CC(=O)NC1COC2(C1)CN(C(c1ccn(C)c(=O)c1O)=O)C2 17124,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17125,C1(C(N(C(C)CNC(=O)C2=CCCCC2)C)=O)CCCC2(CCC2)C1 17126,N1(C(CCCOC(C)(C)C)=O)CC=CC(C(=O)NCc2sccc2F)C1 17127,CC1CC(NC(=O)C(c2ccccn2)O)CN1C(c1cc(C(N)=O)cs1)=O 17128,c1(SC)ccc(CC(N2CCCC2C(=O)NCc2cc(CO)no2)=O)cc1 17129,C1(C(=O)NC(C2(O)CCCCC2)C(N2C(CC)CC(O)C2)=O)CN2CCN1CC2 17130,C(=O)(Nn1c(C)nc2ccccc12)c1nccc(COCC)c1 17131,c1(N2CCOCC(C(C)C)C2)nc(N(CCCCO)C)c2c(F)cccc2n1 17132,Cc1ncccc1CC(=O)NC(C(=O)NC(C)CO)C1CCCO1 17133,N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C3CCC(N(C)C)CC3)=O)CC2C1 17134,C(C(=O)NCC(C)(O)CO)(C(C)C)N(C(COC)=O)C 17135,c1(N(C2CCN(C(C(C)C3CCCO3)=O)C2)C)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 17136,CC(C(=O)N(CC(=O)NC(C)Cc1cn[nH]c1)CC1CC1)N(C)C1CC1 17137,CCCC(C)(CC)C(=O)NC1CCN(c2ccccc2)NC1=O 17138,c1(C(N2CC3C(C(=O)OC(C)(C)C)C3C2)C(=O)NC)ccc(C#N)cn1 17139,c1(CC(=O)NCC2CC(NC(=O)CC3CC4(CC4)C3)C(O)C2)ccc(F)cc1F 17140,CC(C)(O)C(C(=O)NCCOCCCO)NC(c1scnc1Cl)=O 17141,N#Cc1cccc(-c2cscc2C(=O)O)c1 17142,c1(OC)ccc2c(NC(=O)CC3CCCN3Cc3cnn(C)c3C)ccnc2c1 17143,N1(CC(=O)N(CC)CC)CCN(C2CCN(C(C3CC3(F)F)=O)C2)CC1 17144,N1(C(C2C(COC)C2)=O)CC2CCN(C(c3cnc4c(c3)COC4)=O)C2C1 17145,c1(C(C)C)ccc(F)c(C(N2CCC(NC(c3ccnc(O)c3)=O)C2C)=O)c1 17146,C(C)(C(C(=O)NCCC1CC(C)C1)C(C)C)NC(C(C)=CC)=O 17147,c1(CN2CC(CC)OCC2)ccc(C)c2c1CCC2 17148,N=c1cc(CCC(N2CCN(c3ccccc3)CC2)=O)cc[nH]1.N1(CCC)CCNCC1 17149,Nc1cc(C(=O)NCC2(CNC(=O)CC3C=CCCC3)CC2)ccc1Cl 17150,C1(C)(CNC(CC(CC)C)=O)CCC(NC(=O)CCNC(c2ccco2)=O)CC1 17151,c1(C(=O)NC2C(NC(CC(C)CF)=O)CCCC2)n[nH]c2c1COCC2 17152,C(=O)(CCS(N)(=O)=O)N1CC(OCC)C(CNC(c2conc2C)=O)C1 17153,c1(CC)nc(N2CC=CC(NC(c3cc(CCOC)on3)=O)C2)c(F)c(Cl)n1 17154,c1(CNC(C(CC)F)=O)cnc2sc(C)nc2c1 17155,C=CCCCC(C(=O)OC)NCC(c1ccc(OC)cc1)C1CC(F)(F)C1 17156,N1(C(C=C(C)C(=O)O)=O)CCc2nc(-c3sc(C)nc3C)sc2C1 17157,c1(OC)[nH]nc(CC(=O)N(CC(=O)O)Cc2ccccc2)c1Br 17158,C(CC(F)F)(C(=O)N(CCCc1cccs1)C)NC(C1OCCN(C)C1)=O 17159,C1(SCC)CCCN(C(=O)CCc2cnc(C3CCC3)o2)C1.c12nc(Cl)c-1s2 17160,C#Cc1ccnc(C(=O)NCC2(O)CN(C(c3cnn(C(C)(C)C)c3N)=O)C2)c1 17161,N1(C(C(Cn2ccnn2)NC(c2ccc(C)nc2O)=O)=O)CCc2cncnc2C1 17162,C(=O)(C(C)CCCC(C)C)N1C(C(=O)NCCCC)(COC)C=CC1 17163,CN1CC(=O)N(CC(=O)NC2CCCCC2CNC(c2nccc(Cl)c2F)=O)C1=O 17164,C(=O)(CC(CC(N)=O)CC(C)C)NC(CN(C(c1c(C)nco1)=O)C)(C)C 17165,C(=O)(CCCCCF)N1C(CN(C(C2CCCN2C(=O)C(C)C)=O)CC)CCC1 17166,N1(C(C(CCSC)O)=O)CC(CNC(c2c(F)cccc2F)=O)CCC1C 17167,C(=O)(C1=C(c2ccccc2)CCC1)NC1CC(C)(NC(=O)Cc2cc[nH]n2)C1 17168,c1(C(N2CC(N(C(CCN(C)CC)=O)C)C(F)C2)=O)cn2cccc(C)c2n1 17169,CC1CC(C(=O)N2CCC(C(=O)NC3(C)CCCC3O)C(O)C2)=NO1 17170,c1(C(C)(C)F)ccc(F)c(C(=O)NCC2COCCN2Cc2cccnc2O)c1 17171,N(C(=NCc1ncnn1C)NC1CCCCC1)C(C)C(F)F 17172,C1(O)(CNC(c2cncc(F)n2)=O)CCN(C(=O)CCc2ccc(F)cc2)CC1 17173,Cc1ccc(C)c(C(=O)NCC2CCCC2C(=O)N(CC(C)C)CCO)n1 17174,c1(OCC)ccc(SCCC(=O)NC2CCC(CNC(=O)CCC(C)=O)C2)cc1 17175,C(=O)(C(C(C)C1CCOCC1)N1CCC(C)(O)C1)NCCCN(C(C)C)C(N)=O 17176,Cc1nc(C2CC2)nc(C)c1C(=O)NCC1(C(N)=O)CN(C(c2ccoc2Cl)=O)C1 17177,CCCCCC(C)(CC)C(=O)NCC(C)(C)CNC(=O)C(n1cc(Cl)cn1)C 17178,C12(C(N(CCCCN(C)C(C3CC(=O)CO3)=O)C)=O)CC3CC(CC1C3)C2 17179,C(C)(C)(CCNC(C1CC(OC)C1)=O)NC(c1cnc(NCC2CC2)s1)=O 17180,Cn1c(O)nc2ccc(C(=O)NCCC3CCN(C(C4(C)CC4(C)C)=O)C3)cc12 17181,C=Cc1cnn(C)c1C(=O)N(CC(CO)(CO)NC(c1ccc(C(N)=O)cn1)=O)C 17182,c1(CC)cnn2ccc(C(=O)NCCN(C(=O)C(C)CCCNC(C)=O)C)nc12 17183,C1(C(=O)NCCN(C2CCCCC2)C(c2cocn2)=O)(OC)CC(CF)C1 17184,C1(CC)C(NC(C2CCCSC2)=O)CCCN1C(=O)CNC(c1cscn1)=O 17185,C(CCN(C)C(C1CC2(C1)CC(F)C2)=O)(C(C)(C)C)NC(CC(=O)OCC)=O 17186,c1(CCONC(c2cc(F)c(C)cc2C(N2CCCC2)=O)=O)c[nH]c2ccccc12 17187,CC1=C(Br)CCN(C(C2CCC(c3nc(C)no3)CC2)=O)C1 17188,CC(C)(CCC(=O)N1CC2(C1)CN(C(=O)C(F)F)C2)c1ccccc1 17189,CC=CCC1N=C2C=C(C=C(C(F)(F)F)O2)C1=O.C(F)F 17190,Cc1sc(C(=O)N(O)Cc2ccccc2)nc1I 17191,c1(C(=O)NCCN(CCC)C(c2nnc(C)s2)=O)ccc(-n2cncn2)nc1 17192,N1(C(C2NC(=O)CC(C)C2)=O)CCC(NC(=O)CCCC2CC2)C12CCCC2 17193,c1(N(CC(C)CNC(=O)COC2CCCC(C)C2)C)nc2cc(F)ccc2o1 17194,CCC(CC)CC(F)C(=O)N1CCCC1C(=O)NCc1n[nH]cc1C1CC1 17195,CC(C)C(C(=O)NCC1CC1CNC(=O)C(c1ccccc1)F)NC(N)=O 17196,c1(C(C)Sc2cc(C)on2)nc(-c2ccoc2)nn1Cc1csc(Cl)c1 17197,CCC(C)C(C(=O)NCC1(CNC(=O)CC2CSC2)CC12CCC2)N(C)C 17198,N1(C(C(CCC)OCC)=O)CC2CCC(C1)N2CC(=O)Nc1cccc(C)c1 17199,C1(CNC(C(CC)(C)CO)=O)N(C(c2nc(C)ccc2F)=O)CCCC1(C)C 17200,CC(F)(F)C(C)(C)C(=O)NC1CC=C(C(=O)N2CCCC2C2CCCC2)C1 17201,C1(C)(C(=O)NC2CCN(C(CCCCCOC)=O)CC2OC)CC(C)OC(C)C1 17202,CC(C)C(O)C(=O)N1CC=CC1(C)C(=O)N(C)CCC1CN(C)C1 17203,C(=O)(C(C)S(=O)(=O)CC)N1CC(NC(Cc2ccn(CC)n2)=O)(CF)C1 17204,N1(C(c2ncc(C(=O)C(F)(F)F)cn2)=O)CCCc2cncc(Br)c21 17205,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17206,c1(CNC(c2scc(CNC(=O)COCC3CCCO3)c2)=O)cnnc(O)c1 17207,CC(C)(C)CCCC(=O)NCC1CN(C(=O)CCOc2cc(F)cc(F)c2)C1 17208,CCC(Cc1ccccc1)(CCn1cc(C2(C)CCCO2)nn1)C(=O)O 17209,c1(CNC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17210,C(=O)(C(CCOCC)NC(=O)C(C)OC1CCCC1)N(CC#C)C.C=C1CC(CCO)C1 17211,c12ccc(nc1Cl)CN(C(CC(=O)OC)=O)CCNC2=O.C(C)(C1CC1)NC1CC1 17212,C1(CNC(=O)CC2(O)CCOCC2)CCC2(CN(C(=O)C(F)CC3CC3)C2)O1 17213,c1(NCc2cc(C)ns2)nc(=NCCOCCC2CC2)[nH]c2cc[nH]c12 17214,c1(C(=O)OC)cc(=NCC(C2CC2)N(C(=O)C(c2cnn(C)c2)O)C)[nH]c(C)n1 17215,c1(CC(C)C(=O)NC(c2cccc(Cl)c2)CNC(=O)C2CC2)ccc(F)c(F)c1 17216,C(=O)(C1=NN(C)C(=O)CC1)NCC(CCOC)NC(c1c(C)cccc1Cl)=O 17217,c1(NC(CN(C)C(C2(F)CCCCC2)=O)(C)C)nc2c(cc1C#N)CCOC2 17218,Cc1cc(C(N2CC(CNC(C3(CO)CCC3)=O)C(O)C2)=O)cc(Br)c1C 17219,NS(=O)(=O)c1cc(C(=O)NC2CC(CNC(C3CCCSC3)=O)C2)cs1 17220,C1(C(N2CC(C)(CC=C)C2)=O)(C(C)C)CCN(C(C2CCC2C)=O)C1 17221,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CNC(C(C)Nc3ccccc3)=O)(CC2)C1 17222,N1(C(C2CC(OC)CN2C(C2CCC(=O)O2)=O)=O)CCC2(CNC(=O)O2)C1 17223,c1(C(=O)NCC(=C)CCNC(=O)CSS(C)(=O)=O)cnc(OC)cc1C 17224,C1(CCC)CCC(C(=O)NC2CCC(NC(=O)C(F)C(C)C)C2)CC1 17225,c1(CC(N2CCC(N(C(=O)C=C(C)C)CC)C2)=O)cnccc1Cl 17226,c1(C(N2CC(N(C)C(C3CCCC3C(F)(F)F)=O)C2)=O)cc(OC(F)F)n(C)n1 17227,c1(C(N(CCCC)CC(N)=O)=O)ccc(CNC(C2CCCS2)=O)nc1 17228,N1(C(C(C)Cc2ccccc2)=O)CCCN(C(c2ccn(C)c2)=O)CC1 17229,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2ccncc2)=O)c1 17230,C1(COCC)CCN(c2ccnc(NCCOC3CCCCC3)n2)CC1 17231,C(=O)(CC(C)(C)CNC(C1CCC(=O)CC1C)=O)N1CC(C)(CC)C1 17232,c1(C(N2CCCC(NC(C3(C)CC3(Cl)Cl)=O)CC2)=O)ccc2c(n1)COCC2 17233,C1(C(=O)OC)CC(NC(=O)C(C)Cc2cccc(C)c2)CCN1 17234,C1(NC(c2ncn(CC)c2)=O)CCN(CC(=O)NC2CCS(=O)(=O)CC2)C(C)C1 17235,c1(C(=O)NCCC2CC(C)N(Cc3ccncc3)CC2)cc2c(cc1N)OCO2 17236,C1(NC(C(CN(C)C)c2ccccc2)=O)CN(C(C2CC(O)C2)=O)CCC1C 17237,C1(CC(=O)NC(C=C)(C)CC)CCN(C(C)=O)C1(C)C 17238,N1(C(C2(CC=C)CCC2)=O)CCCCC1.C1(=O)C(C)OCCCCN1.C(C)C 17239,C(=O)(C(F)CC1CCOC1)N(CC(=O)NCCc1nc(O)n[nH]1)C1CC1 17240,N1(C(C2C(C=C)C2)=O)CC(NC(c2ccc(C(N)=O)cn2)=O)C2(CCC2)C1 17241,c1(C(=O)NC2C(CNC(c3c(CC)ocn3)=O)CC2)c(Cl)cccc1Cl 17242,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CO)CCCO2)=O)C(C)(C)C1 17243,c1(N2CCOCC(CC)C2)ccc(S(=O)(=O)NC2CCSC2(C)C)cn1 17244,CC(C)(C)CC(C)(C)C(=O)NCC1CC1CNC(=O)CCn1cc[nH]c(=O)c1=O 17245,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17246,c1(NC(C=CC(N2CCC(OCCS(C)(=O)=O)C2)=O)=O)sc(F)cc1Cl 17247,c1(SC)cc(C(=O)NCC2CC2NC(=O)CS(=O)(=O)NC(C)(C)C)c(C)o1 17248,c1(OC)cc(Br)ccc1CC(N1CCC(NC(C2CCS(=O)(=O)CC2)=O)C1)=O 17249,C1(NC(=O)C(c2cc(F)ccc2F)F)CC2CCC(C1)S2(=O)=O 17250,n1(CC=C)cc(C(=O)NC2CCC(C(N3CCC3C(=O)N(C)C)=O)C2)cn1 17251,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17252,c1(OCc2ccc(C(=O)NCC(CO)NC(CC(C)O)=O)o2)cccc(Cl)c1 17253,C1(C(=O)NC2(CN(C)C)CCCCC2)CN(C(c2cnco2)=O)CC12CCC2 17254,C1(NC(c2nc(COC)oc2)=O)(CF)CCN(C(C2CC(N3CCOC3=O)C2)=O)C1 17255,CCCCCCCC(=O)N1CC(F)(C(=O)Nc2cc(F)ccc2OC)C1 17256,c1(C(C)(F)F)cccnc1C(=O)O.C1C(=O)N(CC#N)CCN1 17257,c1(CC)cnn2c1CCC2.C1C(C)(C)CNC(=O)C(=O)N1CC.C(COCCO)S 17258,Cc1sc(Cl)c(C(=O)NCCOC2CN(C(=O)CCC3CCN(C)CC3)C2)c1C 17259,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17260,N1(C(C(COCC)C)=O)CCC2C1CCCN2C(c1cccc2ccnn12)=O 17261,C1(NC(C(C2CN(C(=O)Cc3ccsc3C)C2)OC)=O)COCCC1(F)F 17262,C1(C(=O)NCCNCCCO)CC12CCN(Cc1ccc(I)c(O)c1)C2 17263,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17264,N1(C(c2ccc(C)nc2C)C(=O)NCC2CCCO2)CCc2ccccc2C1C 17265,c1(SC)ccc(C(C)=O)cc1NC(C1CN(C(C2CN(C(C)=O)CC2O)=O)C1)=O 17266,CC1CCCC(NCCCCNC(=O)Cc2csc(Cn3cccn3)n2)CC1 17267,N1(C2CCN(C(C=C(C)C3CC3)=O)C2)CCN(C(=O)C(c2cnn(C)c2)C)CC1 17268,C1(NC(CCn2ncn(C)c2=O)=O)CC(NC(C2(S(C)(=O)=O)CC2)=O)C12CCC2 17269,N1(NC(CONC(Cc2ccc(=N)[nH]c2)=O)=O)CCC2(CC(F)C2)C1 17270,C#CCCCCC(=O)NN1CCOCC1.c12ncoc1CC1C(CC1)NC2=O 17271,c1(C(N2CCN(C(CNC(c3scc(C)c3)=O)C)CC2)=O)ccc(O)nc1C 17272,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nnnn2C1 17273,c1(C(=O)NC2CCC(C(=O)Nc3nc(C(=O)OC)c(Br)s3)C2)cc(O)cc(O)c1 17274,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(C(C)C)s2)=O)CCC1CO 17275,c1(C(N(CCNC(C2C(OC)C2)=O)C)=O)c(F)c(C)cc(N)c1F 17276,N(C1CCc2c(Br)cccc21)C(C(C(CC)CC)F)=O 17277,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17278,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17279,c1(C(=O)NCCNC(CN(C)C(C2CCC2)=O)=O)cc(C(=O)N)co1.C1CC1 17280,C=C(C)CCCNC(=O)COC(C)(C)CNC(C1(CCCC)CC1)=O 17281,O=C(C1=C(F)CN(C(C2(F)CCOC2)=O)CC1)NCc1nn[nH]n1 17282,c1(C(=O)NC2CC(C(C(N3CCC(NC(C)=O)C3)=O)F)C2)nn(C)cc1C 17283,N1(C(CN(S(C)(=O)=O)C)=O)CCOCC1N(C(=O)COC1CCOC1)C 17284,O=C1COc2ccc(C(=O)NC34CC3CN(C(c3cnc(Cl)s3)=O)C4)cc2N1 17285,c1(CNC(=O)NC(c2ccc3c(c2)CCC3)(C)C)cc(Cl)c([N+](=O)[O-])[nH]1 17286,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17287,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17288,CCCC(O)(CCC)CC(=O)N1CC2(CCC(CNC(=O)Cc3cc[nH]n3)O2)C1 17289,C(c1cnn(C)c1C)=CC(N1CC=CC(NC(c2ccc(NC)cc2)=O)C1)=O 17290,c1(C(=O)NCC2C(CNC(c3ccc(SC)s3)=O)C2)cnnc2ccccc12 17291,c1(C(=O)NCC2CCC(C(N3CSCC3C(=O)OCC)=O)C2)cccc(F)c1 17292,C(=O)(C1CCCc2nncn21)N(CCN(C(=O)C=Cc1ccco1)C)C 17293,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17294,c1(C(=O)NCC(CC)NC(c2nn(C)nc2Br)=O)cnc(C)n1C 17295,N1(C(c2cc(CCC)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17296,CC1CN(C(c2ccc(S(N)(=O)=O)o2)=O)CC2(CCN(C(C3(C)CCC3)=O)C2)O1 17297,c1(COC)c(C(=O)NCCC2CN(C(c3csc(=N)[nH]3)=O)C2)oc2ccccc12 17298,C1(C(=O)NCc2ccc(F)[nH]2)C2C3CC4C5CC(C1C35)C24 17299,C1(C)(NC(c2ncn(C(C)C)c2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17300,c1(C(=O)NC2C=CCN(C(CCN(C)CC)=O)C2)c(C)[nH]c2ccc(F)cc12 17301,N1(C(c2c(C)csc2C)=O)CCCN(C(=O)C=CCCc2ccccc2)CC1 17302,S(=O)(=O)(c1csc(C(N2CC(n3ccnn3)C(O)C2)=O)c1)NC.C1C(=O)O1 17303,c1(C(=O)NCCCCNC(c2c(CC)ncs2)=O)cnc2ncccn12 17304,c1(C(N2CC3C(CNC(c4n(CC)cnn4)=O)(C3)C2)=O)ccc2c(c1)CCCC2 17305,CC(O)CC(C)CNC(=O)Nc1cccc(OCC(F)F)n1 17306,CN1C(=O)Cc2ccc(-c3cccc(-c4nccn4Cc4cc(Br)cs4)c3)cc21 17307,N#Cc1cc(N2CC3(CN(C(c4ns[nH]c4=O)=O)C3)C2)nc(C2CC2)n1 17308,C1(CNC(CC(C)(C)N(C)C)=O)CN(C(=O)CC2CCCO2)C(C)(C)C1 17309,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17310,C1(C(=O)NC(C#C)C)CN(C(c2cn(C)nc2OC)=O)CC1(F)F 17311,c1(NC(CNC(CC2C(OC)COC2)=O)(C)C)ncn(C)c(=O)c1Br 17312,c1(C(=O)NCC2CC(NC(CCCCN(C)C)=O)C(O)C2)ccc(O)c(F)c1F 17313,N(C(=NCCC(=O)N1CCOCC1)N1CCC(C(=O)OC)C1)CC1(C)CCCO1.N(C)C 17314,c1(Cc2cn(C(C(=O)NC(CC)CCCO)C)nn2)cc(Cl)ccc1Cl 17315,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(c1ccc(F)cn1)=O 17316,C(CCCC(=O)NC(C)(C)C(=O)N(C(C)Cc1cn[nH]c1)C1CC1)OC 17317,C1(C(C2(C)CC2)=O)CC2CCC1C1CN(NC(Cc3cc(CC)no3)=O)CC21 17318,C1(C(N2CCCC(NC(Cn3c(C)cc(C)n3)=O)C2)=O)CCc2nnn(C)c2C1 17319,c1(C(N2CCN(C(C3(c4ccc(F)nc4)CC3)=O)C3CC23)=O)cn2ncccc2n1 17320,N(C1CC(F)(F)c2ccccc21)C(=O)CC1CCSCC1 17321,Cc1nc2cc(C(=O)NCC3(C)COCCN(C(C4CCC(=O)C4)=O)C3)[nH]c2s1 17322,CCC(CCCC(=O)NCc1csc(C)c1)NC(=O)C(C)OCCOC 17323,C1(CC(=O)NC2(COC)CCN(C(=O)Cc3cnoc3)C2)CC(C)CC(C)(C)C1 17324,c1(CC(=O)NCC(C)CN(C)C(C2CCC2C#N)=O)cc(C(F)(F)F)no1 17325,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17326,c1(C(=O)NC(C)(C)CCNC(c2sccc2F)=O)cccc(Cn2cncn2)c1 17327,CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(F)(F)CC)C(c2ccccc2)C1 17328,C=CC1COCCN1C(=O)C(CC(C)C)N(CCNC(=O)C(CC)CC)CC 17329,CC1CCC(CCC(=O)NC(C2CCCC2)C2CCCC2)O1 17330,c1(CN2CCCC(C(=O)Nc3cccnc3S)C2)cccc2ncccc12 17331,C(=O)(CCCC(C)(C)C)NC(CCN(C(C1N(S(CC)(=O)=O)CCC1)=O)C)C(C)C 17332,Cc1ccc(CNC(C2C3CC3CN2C(=O)CCC2CC2C)=O)nn1 17333,N1(C(C(C=C)CC)=O)CC2(C1)CN(C(=O)CCn1ccc(C)n1)CC2CO 17334,c1(C(=O)NC2CCCC(NC(Cn3c(C)cnc3)=O)C2)nnn2c1CCCC2 17335,c1(CN2CC(NC(CS(=O)(=O)N(C)C)=O)C(F)CC2)ccc2c(c1)OCCCO2 17336,N1(c2n(C)ncc2)CCN(C(=NCCOC(F)F)NCC2CC2)CC1 17337,Cc1cc(C(=O)NCCC(C(C)C)NC(=O)C(C)(C)C2CC2)c([N+](=O)[O-])c(O)n1 17338,C1(NC(C2(CCCC)CC2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3)COC1C2 17339,c1(C(N(C(CNC(C(CC=CC)C)=O)C2CC2)C)=O)cc2occc2s1 17340,C(C(=O)NC(C1CCCC1)CNC(=O)C(O)C(F)F)(C(C)C)OC 17341,N1(C(C=CC)=O)CC2CCN(C(c3scc(C)c3C(N)=O)=O)C2C1 17342,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(O)CCCCC4)C3)=O)ccnc12 17343,Cc1cc(C(N2CCC(C)C(NC(=O)COCCN(C)C)C2)=O)nnc1C 17344,CCCCCC(CC)C(=O)N(C1CCCCC1NC(c1cnc(C)nc1C)=O)C 17345,C(c1ccc(F)c(F)c1)=CCCC.c1(NC(=O)NOC)ccc(F)cc1C 17346,c1(CC)nn(C)cc1C(=O)NC(C)(C)C(C)NC(=O)CCc1cn(C)nc1C 17347,Cc1cc(C)c(S(=O)(=O)N2CCC(CC(N3CCNCC3)=O)CC2)c(F)c1 17348,O=C1Cc2ccc(C(=O)NC3(c4ccc(Cl)c(Cl)c4)CCC3)cc2N1 17349,N1(C(c2cc(CNC(C)=O)on2)=O)CCCC(C(C)C(=O)NC2(C)CCCC2)C1 17350,C1(C)(NC(c2c(C(C)NC(c3sccc3Cl)=O)ccs2)=O)CCCOC1 17351,C1(C(=O)N(CC(NOCC2(CCC=C)CC2)=O)C(C)C)CC12CCCC2 17352,C(=O)(C(C)(C)CC(C)(C)C)NC(C)CC(C)NC(C1CCN1S(C)(=O)=O)=O 17353,CCC(C(=O)N1CCC(C(C)(C)NC(C2CCC(N(C)C)CC2)=O)C1)C(C)C 17354,Cc1sc(O)nc1C(N1CC(C(N)=O)(CNC(=O)Cn2cnnc2)C1)=O 17355,CC1OCC2(CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)C1N1CCCC(F)C1 17356,CC1C(C)CCN1C(=O)C(F)C1CC(NC(=O)CCCNC(N)=O)C1 17357,N1(C(C2(CC(=O)OC)CC2)=O)CCN(C)C(CNC(=O)C(n2ccc(C)n2)C)C1 17358,c1(OCC(=O)OC)ccccc1N(C1CCCC1)Cc1cscn1 17359,C(CCSC)(C(=O)N(CC(O)CC(=O)Nc1nc[nH]n1)CCOC)OC 17360,CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)CC(C)(O)C1CC1 17361,CC(C)(C)CCCCC(=O)NC1CN(C(c2c(N)cccc2F)=O)CC(C)(C)C1 17362,C(C)(CCC(=O)NCC1CCCC1C(=O)NC1(CCO)CC1)OC 17363,c1(CC)nc(Cl)[nH]c(=NCC(C2CC2)NC(C2(S(C)(=O)=O)CC2)=O)c1Cl 17364,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(c2cc(OC)n[nH]2)=O)CC1(C)C 17365,CC1CC(NC(=O)CC(F)(F)F)CN1C(C1CC2CCC1O2)=O 17366,c1(CC)ccc(C(=O)NCC2CCCN(C(=O)C(C#N)CC)C2)cc1C(F)(F)F 17367,C1(NCCC2N(C(CCC(=O)NC3(C)CC3)=O)CCSC2)CCCC(F)(F)CC1 17368,N1(C(C=CCC)=O)CCC(NC(c2cc(C(C)=O)c[nH]2)=O)CC1 17369,C12(CNC(=O)NCc3[nH]cc(C)c3)CCCC(C)(C1)OC2 17370,c1(SCC)cncc(C(=O)N(CCNC(=O)CCC2(N)CC2)C(C)C)c1 17371,C1(CCNC(CCOCC)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17372,N1(C(c2n(CC)ccc2)=O)CC(NC(c2cc(-c3ccccc3)co2)=O)C(C)C1 17373,N1(C(CCSC)=O)CCCC2CN(C(c3cccc4ncn(C)c34)=O)CCC12 17374,N1(C(CSS(C)(=O)=O)=O)C2CCC1CC(NC(c1cc(Cl)no1)=O)C2 17375,c1(NC(CCC(C)NC(=O)C=CC2CCOCC2)=O)cccn2ncnc12 17376,CC1(C)CCC=C1C(=O)NCC12CN(C(=O)CC3SC(=N)NC3=O)CC1CCO2 17377,CN=c1cc(C(=O)NCC(c2cn(C(C)C)nn2)(C)C)c(Br)c[nH]1 17378,C1(CNC(C(C)C2CCC2)=O)CN(C(=O)COCc2ccnn2C)CCN1C 17379,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCNC(c1cc(F)c(OC)c(F)c1)=O 17380,c1(C(=O)NC2CCN(C(c3ncc(OC)cn3)=O)C2CF)ccc2nc[nH]c2c1 17381,C1(COC)CCC(C(=O)NCC2CC2CNC(C2(OC)CCCC2)=O)CC1 17382,C=CCCC(O)CN(C)C(C1CC(F)CN1C(=O)C=C1CCCCC1)=O 17383,C1(NC(c2c(C)[nH]cc2)=O)CC2CC1N(C(=O)CNC(c1cccnc1)=O)C2 17384,c1(CC)ncc(CN(C(C2CN(C(C)C)C2)=O)Cc2ccccc2F)cn1 17385,c1(C(=O)Nc2ccc(-c3ccn(C)n3)nc2)c(OCCF)sc2c1CCC2 17386,c1(NC(N(C)CC2CCN(C(C3(C)CCC(C)C3)=O)C2)=O)cccc([N+](=O)[O-])c1 17387,c1(C(N2C(CN(C)C(C3CC3F)=O)CCC2)=O)cn2c(n1)COCC2 17388,CC1(C(=O)NC2C=CCN(C(=O)CSC3CCCCO3)C2)CS(=O)(=O)C1 17389,Cn1cnc2[nH]c(C(N3CCC4CCCC34CNC(c3ccsc3Cl)=O)=O)cc12 17390,C12(CNC(C(CCC)CCC)=O)COCCN1CCN(C(=O)C(C)CSC)C2 17391,CC1CCC(C(=O)NCCC(O)CNC(c2ccnn2Cc2ccccc2)=O)O1 17392,c1(C(=O)NCC(CO)NC(=O)Cn2ccccc2=O)ccc2nc(O)nc(O)c2c1 17393,N1(C(=O)CCN2CCOCC2)CCOC2CN(Cc3cc(Cl)cnc3Br)CC12 17394,C12(NC(CC(C)C3CC3)=O)CCCN(C(=O)COc3ccccc3F)CC1C2 17395,N1(C(C(C)OC)=O)CCCC(CNC(C2CC3CC3CC2C)=O)CC1 17396,C1(NC(CCC(=O)NC)=O)CCN(C(=O)CS(=O)(=O)CCOC)CCC1CO 17397,C(=O)(C1=CS(=O)CCC1)NCCC1CCN(C(c2c(C)c(Br)ccn2)=O)C1 17398,c1(C(=O)NCC(CCC)NC(c2coc(C(N)=O)c2)=O)cc(F)c(C)cc1Cl 17399,c1(C(=O)NC2C(CNC(c3sccc3CO)=O)CCCC2)cc2ncccc2s1 17400,Cc1cc(F)c(C(=O)NCC(C)(C2CC2)NC(C2CN(c3cscn3)C2)=O)c(Cl)c1 17401,C(=O)(C(C)(C)S(C)(=O)=O)NCC(C)(C)CCNC(C1CC1C(N)=O)=O 17402,c1(CC(=O)O)ccc(-c2nnc(C3CCCC3)o2)c(Cl)c1 17403,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17404,c1(C(=O)NCC2N(C(C3(CC)CCCO3)=O)CCCC2)noc2cc(Cl)ccc12 17405,Cn1cc(CCC(=O)N2CCC2CC2COC(=O)C2)cn1.c12cn(nn1)C2 17406,N1(C(CONC(C(C)c2cc(C)no2)=O)=O)CC2CCCC(O)C2C1 17407,CC1(CC(=O)NCC(C2CCC2)NC(=O)C(F)=C2CCC2)CC1(F)Cl 17408,N1(C(C=CC(=O)OCC)=O)CCN(C(=O)C(O)Cn2cncn2)CC2(C)CCCC12 17409,c1(C(=O)NC2CC3(CC(C(=O)NCc4ccc(C)cn4)C3)C2)ccnc([N+](=O)[O-])c1 17410,N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCOC2CC2)CCC1C 17411,C1(O)(NC(COCC(C)C)=O)CCN(C(c2ccnnc2)=O)C1 17412,CC1CCN(C(c2coc(CC3CC3)n2)=O)C(CNC(=O)CSc2nc[nH]n2)C1 17413,c1(C(CC)NC(=O)NC(C2CCCO2)C)cccc(C#N)c1 17414,C#CCC(CC#C)C(=O)N(C)CCN(C(=O)CNSc1ncc[nH]1)C 17415,c1(C(N(CCC(N2CC(C)SCCC2)=O)CC2CC2)=O)ccc([N+](=O)[O-])cn1 17416,c1(C(C)N(C)C(=O)NCC(C)C#N)cccc(C(F)(F)F)c1 17417,C1(NC(c2c(CCC)n(C)nc2)=O)CN(C(=O)CSc2nc[nH]n2)CC(C)(C)C1 17418,N1(C(=O)C=Cc2cscn2)CCCN(C(=O)CC2CCC3(CCC3)O2)CCC1 17419,N1(C(c2cc(CC)on2)=O)CC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2C1 17420,C12(NC(c3cc(C(F)(F)F)ccn3)=O)CCC1CN(C(C1CCCCC1O)=O)C2 17421,c1(CC(=O)NCCN(CCC)C(C23CC(C#N)(C2)C3)=O)ccccc1Cl 17422,C(=O)(C#CC1CCC1)NC(CCOCC)C(=O)N(C1CCOC1)C 17423,c1(OC(C)C)ccc(Cl)c(F)c1CN1CCC(CCC(=O)NC(C)(C)C)C1 17424,c1(CC)ccc(C(=O)O)cc1F.n12cc(nn1)-c1ccc(s1)NC(=O)C2C 17425,c1(CC(=O)N)nccn1C(C)(C)C.C(C)(C)(C)OCCCCN(CCOC)C 17426,c1(C(N2CC(C(=O)NC(CCCC)C)C2)=O)ccnc2cc[nH]c12 17427,c1(C(=O)OC(C)C)ccc(C(=O)NC(C)(C)CNC(=O)CCc2ccccc2)nc1 17428,C1(NC(N2CC(OCCN(C)C)C2)=O)CCN(c2ncccn2)CC1 17429,c1(C(=O)OC)ccnc(N(CCCNC(c2occc2F)=O)CC2CCCC2)n1 17430,C(CC(C)CCNC(c1nocc1Br)=O)NC(C1CC(OC)C1)=O 17431,C(=O)(CC1=NNC(=O)C1)N1CC(N2CCN(C(C3(OCC)CCCC3)=O)CC2)C1 17432,N1(C(C(CC=CC)CC)=O)CC(CNC(=O)CCc2cn[nH]c2)CC12CCC2 17433,C1(C)(C(=O)NCCNC(C(C)(C)C)=O)CCNC1=O 17434,C1(C(N2C(C)(C(N3CCCC(CCOC)C3)=O)C=CC2)=O)CC2CCCC2C1 17435,C1(NC(C(C(CC)O)C)=O)CCN(C(c2cc(Cl)no2)=O)CC12CCC2 17436,c1(C(C(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)(F)F)ccc(Br)cn1 17437,c1(C(N2CCCC2c2ccsc2)C(=O)NC(C)C)ccc(C(=O)N(C)C)cc1 17438,C(=O)(C(C)(C)C(=O)NCC(O)CNC(=O)CNC(c1cc(Cl)cc(Cl)c1)=O)NC 17439,CC1(C)CCCC(C(=O)NC2CN(C(c3cccnn3)=O)CC2(C)C)C1 17440,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17441,N1(C(C(C)N(C)C)=O)CCN2CCN(C(=O)C(F)=C3CCC3)CC2C1 17442,N1(C(c2cnc(OC)c(Cl)c2)=O)C2CCCC1CN(C(=O)C#CC(C)(C)C)C2 17443,c1(C(=O)OC)ccc(-n2nc(C3CC34CC4)nc2-c2ncccc2Cl)cc1C 17444,c1(C(=O)NC(CNC(=O)CCc2ccsc2)C2CC2)occc1C(C)(C)C 17445,c1(C(N2CC(CNC(c3c(CC)csc3)=O)OCC2)=O)cc(C)cc(C)c1N 17446,c1(C(N2CCC2CO)=O)ncncc1N1C(=O)C2(CCCC2)CC1.C1(CO)CC1 17447,CC1CCCN(C(=O)C(c2cnn(C(F)F)c2)=O)C1CCNC(c1ccsc1)=O 17448,c1(NCC2(C)N=C(C)SC2)ncccc1S(=O)(=O)NCC1(C)CC1(C)C 17449,C1(CNC(=O)COCC2CCOC2)CC2CCC(C1)N2C(=O)C=Cc1cnc[nH]1 17450,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)O)c(O)cccc1F 17451,CCCCC(F)C(=O)NC1CC(OCC(N2CCC(C(F)(F)F)C2)=O)C1 17452,c1(CN(C)C)cccc(CNC(C2CCC(CNC(=O)CC3CCC3)C2)=O)n1 17453,CCC(CC(=O)N(CC(=O)N(CCCn1ccnc1)C)CC1CC1)CC(C)C 17454,C1(F)(C(=O)NCC(CCC)OC)CCN(C(=O)CN(C(=O)C(C)C)C)C1 17455,C(=O)(C(O)CC(C)(C)C)NC1(CN=[N+]=[N-])CCN(C(COCC(C)C)=O)C1 17456,C(=O)(C1=C(Cl)CC1)N(C1CC(CNC(=O)CCc2nc(-c3cccs3)no2)C1)CC 17457,C1(C(=O)Nc2n(C)c(S)nn2)CC2(CCCCN2C(=O)COCP(C)(C)=O)C1 17458,N1(C(CCC)=O)CCCC(N(C(=O)C(c2cc(Cl)cc(Cl)c2)(C)C)CC)CC1 17459,c1(NC(CSc2cccc(C)c2)=O)cccc(C)c1CN 17460,CN1CCC=C(C(=O)NC(CC2CC2)C(=O)NCCCCc2ncc[nH]2)CC1=O 17461,c1(C(N2C(CNC(C(C=C)(C)CC)=O)CC(F)C2)=O)cc(S(=O)(=O)NC)oc1C 17462,C(C(=O)N(CCCNC(=O)C(C1CCCC1)C1CC1)C)(C1CCCO1)OCC 17463,C=CCC(C(=O)NC1(CCSC)CN(C(=O)C(C2CCCCC2)O)C1)NC(C)=O 17464,N1(C(C2CN(C(C)=O)C2)=O)CC(NC(=O)Cc2csc(C)n2)CC1.C1(CN)CC1 17465,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17466,Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCC(O)CNC(=O)C(C)C(C)(C)C 17467,C1(C#N)(C(=O)NCC(c2ccc(F)cc2)N(C)C(c2cncs2)=O)CC12CCC2 17468,CON(CCC(=O)Nc1ccc(C)cc1)C(=O)C1(C#N)CCOC1 17469,N1(C(c2cnc(CC)s2)C(=O)NC(C)C)CC(C(N)=O)CC(c2cnn(C)c2)C1 17470,CC(C)CC(C)(C)CNC(C1CCN(C(=O)C2C=CCC2)O1)=O 17471,C1(NC(C(C)OCc2ccoc2)=O)CN(C(C2C3CCCC23)=O)C2(CCC2)C1 17472,c1(C(N(C)Cc2ccc(S(C)=O)cc2)=O)c(F)c(F)c(O)c(F)c1F 17473,c1(OCC)cc(C)[nH]c(=NCC2CN(C(c3nn(C)cc3Cl)=O)C2)n1 17474,C1(C)(CNC(CCCc2cn(C(C)C(=O)O)nn2)=O)CCC(=O)N1 17475,CC1(C)C(NC(C2(n3cncn3)CC2)=O)CCN1C(c1ccnc(NC)c1)=O 17476,c1(C(N2C(C)(C(=O)Nc3ccc(O)c(C)c3C)CC2)=O)c(F)cccc1[N+](=O)[O-] 17477,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17478,C#CCC(CC(F)F)C(=O)N(CC(C)(C)C(=O)NC1CC2(C1)CC(C#C)C2)C 17479,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(c1cccc3oncc13)=O)C2 17480,C1(NC(c2cc(OC)n(C)n2)c2n(CCCC)nnn2)CC2(CCOC2)C1 17481,N1(C(Cn2ncc(C(C)(C)C)c2)=O)CCN(C(C2(CF)CCC2)=O)CC1CCO 17482,N1(C(CC2C(C)CCO2)=O)CCC(CO)(CNC(=O)CN2CCOCC2=O)C1 17483,c1(C(=O)NC2C(CNC(c3c(CC)[nH]cc3)=O)CCCC2)nn(C)c(N)c1C 17484,Cc1nc(CN(C(=O)C(CNC(C2CC3CC3C2)=O)N(C)C)C)n[nH]1 17485,Cc1ccc(-c2ccnn2C)cc1C(=O)NC(C)Cc1ncc(Br)cn1 17486,N1(C(c2cc(C)nnc2)=O)CC2CCC2(CCNC(c2cc(F)ccc2O)=O)C1 17487,C1(NC(c2cnc(CCCC)s2)=O)CCCN(C(c2cscc2F)=O)C1 17488,N1(C(c2cc(C)c(Br)s2)C(=O)NCCSC)CCC12CCN(C)CC2 17489,c1(C(N2CCC(O)(C(C)NC(=O)C3=CCCC3(C)C)CC2)=O)cc(F)cc(N)c1F 17490,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17491,Cc1cc(Cl)ccc1C(N1CC(CNC(=O)CSCc2cccs2)C1)=O 17492,C1(NC(c2c(CCC)nco2)=O)CC2CCC1(NC(c1ccnn1C)=O)C2 17493,C1(NC(c2ccnnc2O)=O)CC(CO)N(C(c2csc(Cl)c2)=O)C1 17494,Cn1cc2c(n1)CCC(C(N1CCC(NC(=O)C=Cc3ccc(Cl)cc3)C1)=O)C2 17495,N(C1CCOc2ccncc21)C(C(N1CCC(O)(CC)CC1)=O)=O 17496,C1(C(=O)N(CCCNC(C2CC2CF)=O)C)(NC(C)C)CC1 17497,N1(C(CCC(C)=O)=O)CCCCCC1CNC(=O)CC1NC(=O)NC1=O 17498,CC1CN(C(c2coc(-c3cccs3)n2)=O)CCN1C(=O)CCc1cc(Cl)no1 17499,c1(NC2CN(C(c3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17500,CC(C)C(C)CC(=O)NC(CC1CCC1)C(=O)N1CC(c2cnsc2)C1 17501,CC(C)(C)C(CNC(=O)CC1CC2CCC1C2)C(=O)N1CCC(C(F)F)CC1 17502,C12CN(C3(CCC3)C1)C2=O.C=Cc1cncc(C(=O)NCC2(N(C)C)CC2)c1 17503,C(=O)(C1=C(CC)OCCC1)NC(CC#C)(C)C(=O)Nc1cccc(CO)c1C 17504,C1(C(=O)NCC(CNC(c2c(C)n(CCO)cc2)=O)C)Cc2cccc(C)c2O1 17505,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17506,c1(CCNC2CCCN(CC)C2)ccccc1S(N)(=O)=O.C1(=O)CCCC(=O)N1 17507,c1(C(N(CC(C)N(C)C(C2CCC(=O)N2)=O)C)=O)coc2c(F)c(Cl)ccc12 17508,CC1CCOC(C(=O)N(C)CCNC(c2cccc(-c3cnc[nH]3)c2)=O)C1 17509,c1(CCC(=O)N(C)CC2C(c3cncc(C(=O)OC)c3)(F)C2)ccc(C)cc1C 17510,C(=O)(CCC(=O)c1ccc(Cl)cc1)NC(CC=C)CNC(C1(COC)CCC1)=O 17511,c1(NC(C2N(C(C(CC)N(C)C)=O)CCC2C)=O)ccc(OC)c(F)c1 17512,C1(C(=O)NCC2CN(C(c3cnncc3O)=O)CC2O)CC12CCSCC2 17513,N1(C(CN(C(=O)OC)C)=O)CCCC(NC(=O)CCc2cncc(F)c2)C(F)C1 17514,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17515,N1(C(Cc2cc(OC)no2)=O)CC(CNC(=O)C(=O)N=S(C)(C)=O)CC(C)(C)C1 17516,N1(C(c2c(C#N)ccs2)=O)CC2CC(C1)C2NC(=O)CNC(c1ccncc1)=O 17517,CC1CCN(C(C23CC(CN(C(c4cc(C(N)=O)[nH]n4)=O)C2)C3)=O)CC1CO 17518,N1(C(=O)CCc2ccsc2)CCC(CNC(C2(F)CCOC2)=O)C1 17519,C1(C(N2CCC2c2ncc(C)s2)=O)(CC)CCN(C(C2CC(F)(CF)C2)=O)C1 17520,C1(C(=O)NC2(C)CC(NC(c3ccc(CN(C)C)cc3)=O)C2)CC2(CCO1)CC2 17521,C1(OC(C(=O)NC(C(CO)NC(C(C)=C(C)C)=O)C)C)CCCCCC1 17522,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCS1 17523,C(=O)(C1=CC2CCCC12)NCC=CCNC(c1cc(C)c(Cl)s1)=O 17524,N1(C(c2cc3ncccn3n2)=O)CCC2C(C1)CN2C(=O)C1=CCCOCC1 17525,N1(C(=O)NCC2(C)CC2)CCc2c1ccc(F)c2Br 17526,C1(NC(C)=O)CN(C(c2cccc(NCS(=O)(=O)C(C)C)c2)=O)C(C)(C2CC2)C1 17527,c1(OC)cc(NC(=O)CNC[Si](C)(C)C)c(F)cn1 17528,C(=O)(CCC(C)N(C)C)N(CC(C(=O)NCC(COC(C)C)(C)C)C)C 17529,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cn(C3CC3)nc1C)=O)C2 17530,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NCC(C)C2CCC2)nc1)OC 17531,C(=O)(C#CC1CCCCO1)NC1C(NC(c2cc3n(n2)CCCC3)=O)COC1 17532,C(C#Cc1ccc(F)cc1)N1C(Cn2cc(CCCOC)nn2)CCC1 17533,C1(C2CCCN(C(C3CC3(C)Br)=O)C2)(NC(C(C2CCOC2)OC)=O)CC1 17534,c1(CC)ccc(OCC(=O)N(C2CCN(C(C3(C)COC(=O)C3)=O)C2)C)cc1 17535,c1(C(N(C(CNC(CC2C(C(C)=O)C2(C)C)=O)C)C)=O)n[nH]cc1[N+](=O)[O-] 17536,C1(CCNC(C(N2CCOCC2)C)=O)CCC(NC(c2nccn2C(C)C)=O)C1 17537,c1(CN(C(c2n(C)ncc2C2CC2)=O)CC2CC2)cc(=O)oc2ccc(O)cc12 17538,c1(OC)cc(C(=O)Nc2csc(C)n2)c(NC(c2ncc(F)cc2OC)=O)cn1 17539,C(C)(CO)(C(=O)NCCN(CCc1ccccc1)C(c1cnc(S)nc1)=O)OC 17540,N1(Cc2ccc(C(=O)OC)cc2)CCC(C#N)(OC)C1.c12ccc(cc1)CN2C 17541,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17542,Cc1nc2ccc(C(N3CC(N(C)C(C4CC4(C)C)=O)C4(CC4)C3)=O)cc2s1 17543,c1(SC)cc(C(=O)N(C2CCC(NC(=O)C(c3cncn3C)O)CC2)C)n(C)n1 17544,C(=O)(C(O)C(C)(C)C)NC1(C2N(C(CCN(CC)CC)=O)CCCC2)CC1 17545,N1(C(=O)Nc2ccc(OCCC)nc2)CCN(C)c2ccccc2C1 17546,Cc1ccc(O)c(NC(c2cc(CNC(C3(CN(C)C)CC3(C)C)=O)cs2)=O)c1 17547,N1(C(CSC)=O)CCC2(CCCC2NC(=O)Cc2ccccc2C2CC2)CC1 17548,CC1(C#CC(=O)NCC2CC(CNC(=O)Cn3cnnn3)CO2)COC1 17549,Cc1cc(C(=O)N(CCCN(C)C(C2NC(=O)C3CC23)=O)C)nn1C(C)C 17550,Cn1cnc2nc(N3CCc4nccc(Cl)c4C3)nc(N3CCCC(F)CC3)c12 17551,c1(CC)cccc(NC(C2CCN(C(c3snc(C)c3N)=O)C2)=O)c1O 17552,c1(CCC)ccnc(OC)c1NC(=O)C(=O)NCc1ccc(Br)c(F)c1 17553,c1(CC(=O)N(C(C(=O)NCC(O)C=C)c2ccoc2)CC)ccc(O)cc1 17554,Cc1cc(C)n(C2CCCN(Cc3nnc(C4CC4C)o3)C2)n1 17555,Cc1cc(=O)oc(C)c1C(=O)NC1CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 17556,N1(C(c2cnn(CCCC)c2C)=O)CCCCC(CNC(C2(F)CCOC2)=O)C1 17557,c1(C(CC)(C)C)ccccc1C(=O)NCC(C)CNC(c1cn(CC)nc1C)=O 17558,CN(S(=O)(=O)NC(=O)Nc1cncs1)c1cccc(F)c1.C1(=O)CO1 17559,N1(C(C2CC(OC)CN2C(=O)C(C)C(O)C(C)C)=O)CC2CN(C)CC2C1 17560,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17561,C12(C(=O)NCC(C)NC(c3cn(CCC)nc3)=O)CCC(F)(CC1)C2 17562,CCC(CC(=O)N(CCCN(C)C)C1CC1)NC(=O)COCCCN=[N+]=[N-] 17563,C(CCN(C)C(C1CCS(=O)(=O)N1)=O)(C(C)(C)C)NC(Cc1c(C)occ1)=O 17564,N1(C(c2cc(Cl)cc(C)c2O)=O)CC2CN(C(=O)CN(C3CCSC3)C)CC2C1 17565,N1(C(C2C(C(=O)OC)C2)=O)Cc2ccccc2CC1C(N1C(C)CCC1C)=O 17566,c1(C(=O)NCC(=O)NCCN(C(c2n[nH]cc2F)=O)CC2CC2)cccc(F)c1 17567,CC12CC(C(=O)N(C3CC3)CC3CCOCC3)(C1)C2 17568,c1(CNC(=O)Nc2c(SC)cc(Br)cc2)ccc(F)c2[nH]ncc12 17569,O(C1CCCc2ccccc21)CC(=O)N(C1CN(C(c2c(CC)cno2)=O)C1)C 17570,C(C1c2ccsc2CCN1C(=O)CC(C)CC)NC(COCC(=C)C)=O 17571,N(C)(C1CCc2c(Cl)cccc21)C(c1c(C)[nH]nc1CO)=O 17572,N1(C(C(C=C)(F)F)=O)CCC(C2CC2)(CNC(=O)CN2CCSCC2)C1 17573,c1(C(=O)NC(c2nccn2C)C)cccnc1CNC(=O)C(O)CC1CCCC1 17574,c1(C(=O)NCC(C2(O)CCN(C(=O)CNC(N)=O)C2)C)cc2c(cn1)OCCO2 17575,Cc1ccc(O)c(C(=O)NCCCNC(c2cc(-c3c(C)noc3C)no2)=O)c1 17576,C12(C(=O)NCC(CC)NC(=O)C(C)OC3CCCCC3)CCC(C1)C(C)(C)O2 17577,N1(S(C)(=O)=O)CCCC(C(=O)NC2CC(O)(CNC(=O)C(F)OC(F)(F)F)C2)C1 17578,c1(C(=O)NCC(CCC2C(C)(CC(Cl)Cl)CC(=O)N2)(F)C)c(Cl)ccc(O)c1N 17579,C=CC1(C(=O)N(C)CCC2CCCN2C)CCN(C(=O)COCCCOC)C1 17580,c1(C(N2CC(CC)(NC(=O)C(C)(C)F)C2)=O)cc(C)c(OC(C)C)c(C)c1 17581,C1(C(N2CCC(C(=O)NCCC(=O)NCCC)CC2)=O)CCC(=O)N(C)C1 17582,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(C)=O)c(F)c1 17583,C1(NC(CN(C)C)=O)CCN(C(c2cc3nccnc3cc2F)=O)CC(C)(C)C1 17584,N1(C(CC(C)C2CC2)=O)CCC(F)(F)C(NCc2c[nH]nc2C(F)(F)F)C1 17585,C1(OC)CCC2(C(=O)NCC(O)Cn3cccn3)CC12.N12CC(C1)OCC2=O 17586,C(=O)(C(C)(C)CCS(C)(=O)=O)N(C(C)CNC(c1c(O)cccc1Cl)=O)C 17587,c1(C(=O)NCC(C(C)C)NC(C2CC3C(C2)C3(F)F)=O)ccc2ncnn2c1 17588,Cc1coc(C)c1C=CC(=O)N(C)CCN(C(=O)CC(C)c1cccnc1)C(C)C 17589,C1(CCN2C(CNC(=O)CCOC3CCOCC3)CCC2)CCCCC1(F)F 17590,C1(NC(CN2C(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCO)c1)=O 17591,C(=O)(C1=CC2CCC=CCCC12)NCC1(CC(=O)NC2(C(F)F)CCCC2)CC1 17592,C(c1ccccc1F)=CCNC(N(C)Cc1cccc(-c2cnn(C)c2)c1)=O 17593,CC(C(=O)NCCCCN1CCN(C(=O)C(C)(C)C#N)CC1)S(C)(=O)=O 17594,C1(NC(CC2(OC)CC2)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)C2)=O 17595,c1(C(N2CCN(C(Cn3ncc(C)c3)=O)C(CO)C2)=O)c(C)[nH]c2ccccc12 17596,C(c1ccc(C(C)(C)C)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17597,c1(Cc2nc(N3CCC(NC(c4c[nH]c(=O)cn4)=O)C3)sn2)ccc(Cl)cc1 17598,c1(C(=O)NC2C(C(=O)OC)CCC2)ccc(C)cc1C(=O)N(C)CCNC(C)=O 17599,C12(C(N(C)Cc3cscn3)=O)CCC1CN(C(=O)C=CC1CCOCC1)C2 17600,CC1=C(C(=O)N(C2CCN(C(=O)CCCc3cc(C)no3)C2)CCO)CCO1 17601,C(=O)(C(F)(F)c1ncc[nH]1)NC(C)C(=O)NCC(c1ncccn1)N1CCCC1 17602,C(c1ccc(O)cc1)=CC(=O)NCc1cc(C2CCCC2)on1 17603,CC1(C)CN(C(C2CCC(F)CC2)=O)CC1CNC(C1(CCF)CC1)=O 17604,C1(CC)(NC(=O)Cc2cnoc2)CCN(C(=O)CCCC2CCOCC2)CC1 17605,C1(O)(C(C)NC(C2CC23CCC3)=O)CCN(C(=O)Cc2cc(Br)cs2)C1 17606,C1(CNC(c2c(C)nsc2)=O)CCCCN1C(=O)COCCCN=[N+]=[N-] 17607,C(=O)(CCCC(C)(C)C#N)N1CC(NC(Cc2ccn(C(C)C)n2)=O)C(C)C1 17608,c1(SCC)nc(C)c(CC(N2CCCC(NC(c3ccc(CO)o3)=O)C2)=O)s1 17609,c1(C(=O)NCC)ccc(N)c(C)c1Cl.C1CC(=O)N2CC(C2)CC(C)N1CC 17610,c12c(nc(C)nc1Cl)S2.c1(C(=O)NC(C)CCN(C)C)coc(C(N)=O)c1 17611,c1(OC)c[nH]nc1C(=O)NC(C(=O)NCCN1CCCC1C)C1(C)CC1 17612,Cc1cn(C)cc1C(=O)NCC1C=CC(C(=O)NCCCSCCO)C1 17613,C1(c2cn(C3CCN(C(c4cc(C5CC5)no4)=O)C3)nn2)CN(OC)CC1.C1CC1 17614,C(=O)(C(C)(C)C(C)C)NC(COC)CC(=O)N(C)Cc1nncn1C 17615,N1(C(C2C(C)(Br)C2)=O)CC2(CCC2)CC1CNC(c1cnn[nH]1)=O 17616,c1(C(N(C(c2ccccn2)C)C)=O)c[nH]n(C)c1=O 17617,CC(C(C)(C)NC(C1CSCCS1)=O)NC(=O)COc1ccon1 17618,Cc1nc(N2CC(O)(C(C)NC(C3CC34CCC4)=O)C2)c2cnn(C)c2n1 17619,Cc1nc(C2CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)n[nH]1.C1(=O)CC(C2CC2)CN1 17620,N1(C(c2ccc(C)cn2)=O)CCC2(NC(c3cccc(C(N)=O)c3N)=O)CC2C1 17621,c1(CC)cc(=NC(C)CC(C)NCC)[nH]c(C)n1.C1(=O)C(C)O1.C(C(C)C)O 17622,C1(C)(C(N2CC(O)(CN(C(=O)Cc3n[nH]c(=N)s3)C)C2)=O)Cc2ccccc2C1 17623,N(C1CCCc2c1cnn2-c1cccc(F)c1)C(C1CC(C(C)C)C1)=O 17624,N1(C(C(C)CNC(=O)NCCC)=O)CC2C(C(=O)Nc3ccc(F)cc3)C2C1 17625,C1(NC(Cc2c(C(=O)OC)scc2)=O)C2CN(C(c3cc(SC)n(C)n3)=O)CC12 17626,C1(CC(=O)NCc2cc(C)ns2)CN(C(=O)CCc2cncs2)CCO1 17627,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17628,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17629,N1(C(C2CC(=O)NCC2)=O)CC(NC(=O)CCc2cnco2)C(F)(F)C1 17630,CCCC(C)(C)C(=O)NC1CC=CCC1C(=O)NCC(=O)N1CCCO1 17631,c1(Nc2scc(CC(=O)NCCN3CC(=O)NCC3)n2)cc2c(s1)COCC2 17632,C(=O)(C1=C(Cl)CCCC1)NCC1(C(=O)NCC(C(C)C)C)CCC1 17633,CC(CC1CCCCC1)CN=c1[nH]c2c(c(=NCc3ccncn3)[nH]1)SCC2 17634,C12(C(N3CCC(C4CC4)(NC(C=NOC)=O)C3)=O)CCCC1CC(=O)CC2 17635,C1(C(=O)OC)C2CCC(C2)C1CC1CCCO1.C12(CC1)N(C)OCC(=O)NC2 17636,N1(C(c2cc(C(C)C)n[nH]2)=O)CCN(C(=O)C(C)c2ccco2)CC(C)(C)C1 17637,C1(C(=O)NCCOCCC(=O)NCC(C)(O)CC)CCCC2(CC2)C1 17638,CC1CC(C)C1C(=O)NCCCNC(=O)C(C)(C)F 17639,Cc1ccc(C(=O)NCCC2CCN(C(C3CCOC3=O)=O)C2)c2ncccc12 17640,N1(C(C2(COC)COC2)=O)CCCC(O)(CNC(c2cn(C3CCC3)nn2)=O)C1 17641,N1(C(=O)CNC(F)(F)F)CCc2sc(S(=O)(=O)N3CC=CC(CO)C3)cc2C1 17642,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17643,C1(CNC(C(=Cc2ccccn2)C)=O)CCN(C(=O)C(C)(C)C(F)F)CC1C 17644,C(CCCC(C)(F)F)NC(C(C1(C)CC1)NC(C(c1ccnn1C)C)=O)=O 17645,CCCCC(C)C(=O)N1CC(C(C)(C)NC(=O)CCOCC(F)F)C(O)C1 17646,Cc1c[nH]c(C#N)nc1=NCCNC(C12COCCN1C(=O)COC2)=O 17647,C1(NC(C(C)NC(=O)C2CC2)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)C12CC2 17648,c1(C(=O)NC(c2cn(C(C)C)nn2)CCC)ccc(Cl)cc1-n1cnnn1 17649,N#CC1CN(C(=O)N(c2ccsc2)CCCO)CC12COC2 17650,c1(C(C(=O)NCCCCCC)N(c2ccccc2)CC)ccc(OCC)cc1C 17651,CC(C)C(O)CC(=O)NC1CCN(C(c2csc(C3CC3)n2)=O)CC1O 17652,C1(CNC(CC#N)=O)CN(C(=O)Cc2nc[nH]c2Br)CC12CCC2 17653,c1(C(c2nnnn2CCC2CC2)N(CCCCC=C)CC)ccccc1[N+](=O)[O-] 17654,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccns1)=O 17655,C1(CCN(C(c2cc(CC(C)C)[nH]n2)=O)C)NC(=O)NC1=O 17656,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17657,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17658,C(=O)(C(CC=C)CC(C)C)NCC1C2CN(C(c3nccc(C#C)c3)=O)CC21 17659,c1(C(N2C(C(=O)NCC(C)CO)C=CC2)=O)cc(F)ccc1O 17660,C1(NC(c2ccc3oncc3c2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 17661,n1(CC2CC(NC(C(c3ccccc3)C)=O)C2)cc(C2C3COCC23)nn1 17662,c1(C(N2CCC(NC(CNC(C(CC)CC)=O)=O)C(O)C2)=O)ccc(P(C)(C)=O)o1 17663,c1(SCC(=O)NC2CC(CCNC(c3[nH]cc(CC)c3)=O)C2)ccc(C)cc1C 17664,C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1CC(F)CN1C(C1(C)CCNC1=O)=O 17665,O(NC(=O)C(C)(C)C1CCCN1C(=O)CN1CCCCC1)CC.C(C)(=O)O 17666,C1(NC(CC(CC)C)=O)CC(CNC(C2(CC3CC3)CC2)=O)C12CCC2 17667,c1(OC)cnc(C(N2CCCC2CCCNC(=O)C(n2cc(Cl)cn2)C)=O)nc1 17668,N1(C(CC2N(C(c3nn(CC)c(C)c3)=O)CCOC2)=O)C2CCC1CN(C)CC2 17669,C1(C(=O)NC2CC(CC(N3C(C(=O)NC)C=CC3)=O)C2(C)C)CC(C2CC2)=NO1 17670,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17671,C(=O)(C(CNC(=O)C1=CC2(CCOC2)C1)CC(C)C)N1C(CC)COCC1 17672,c1(SCc2cn(CC(=O)NCC)nc2)ccnc2ccccc12 17673,C12(NC(c3c(NC(C)=O)c(F)ccc3)=O)CCCCC1CN(C(=O)C1=CCCC1)C2 17674,N1(C(=O)COCc2sccc2Cl)CC2(C1)CN(C(=O)CC1CCCOC1)C2 17675,N1(C(CC)=O)Cc2ccccc2CC1CNC(=O)C(C(C)C)NC(=O)NC1CC1 17676,NC(=O)CCCC(=O)N1CCC(C2OCCCC2C(=O)Cn2nnnc2Br)CC1 17677,CC1CCN(C(c2cncc(-c3nnco3)c2)=O)CC1c1ccc(F)cc1 17678,CCC(C)CCCCC(=O)NC(CC(=O)N(C)Cc1ncco1)C(C)OC 17679,CN1CCN(c2ccc(C(N3CC(NC(c4ccoc4)=O)C(O)C3)=O)cc2)CC1 17680,c1(C(N2CC(O)CC(NC(CCc3nc(=N)[nH][nH]3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 17681,c1(OC(C)C(N2CCC(CO)C2)=O)ccc(CC(C2NC(=O)OC2C)=O)cc1F 17682,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(=O)Cc2ccsc2Cl)C1C 17683,CN1CCC(OCC(=O)NCC(O)CNC(=O)Cc2ccc(Br)cc2)CC1 17684,C1(C(N(CCCC#C)CCOC)=O)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17685,C1(C(=O)NC(C(C)C)CCNC(=O)C=Cc2cnn(C)c2)CCC2(C1)CC2(F)F 17686,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(C)O)C1 17687,C(=O)(CCCC(c1nnnn1CC)NC(=O)C(C)(C)CSc1ccccc1)OC 17688,C(=O)(CCS(=O)(=O)N1CC2CC2(CNC(c2sccc2I)=O)C1)OC 17689,C1(F)(CNC(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 17690,c1(C(=O)NCC(CNC(Cn2c(C)nnn2)=O)(C)C)cccc(OC2CCC2)c1 17691,c1(CC(N2CCCC(n3cc(-c4ccn(C)n4)nn3)C2)=O)ccc2nn[nH]c2c1 17692,C(=O)(CCCNC(C1CCN(C(=O)CC(=O)N2CCCC2)C1)=O)OCC 17693,C1(F)(CN(C(=O)CSS(C)(=O)=O)C)CC2CCC(C1)N2C(=O)CC1CS(=O)(=O)C1 17694,Cn1cnc(NC2CC(NC(C3CC34CC(C)(C)C4)=O)C2)cc1=O 17695,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(c1)CCC2 17696,c1(N(C)C)cccnc1C(=O)NCCC1(CNC(=O)C(C)(C)c2cncs2)CC1 17697,C1(C)(C(=O)NC2CC(N(C(=O)COCC3CC4CCC3C4)C)C2)NC(=O)OC1(C)C 17698,S(=O)(=O)(c1cnc(NCC(C)(C)CS(N)(=O)=O)c(Cl)c1)N1C(CC)CCCCC1 17699,NS(=O)(=O)c1ccsc1C(N1CCC(CO)C(NC(c2cn[nH]c2)=O)C1)=O 17700,c1(C(N2CCC(C(C)C(=O)NC3CCSC3)CC2)=O)ccc2c(c1)CCCO2 17701,c1(C(N2CCC(N3CCN(C(C(C)OC)=O)CC3)C2)=O)c(C)cc(O)nc1C 17702,N1(C(C(CCC)O)=O)CC2(CCC2NC(C2(OCC)CCCCCC2)=O)C1 17703,Cc1ccc(CC(=O)NCCC2(NC(C3CC(OC(=N)O)C3)=O)CC2)o1 17704,c1(OCC)ccc(CC(N2CC(N(C(=O)CCc3cn(C)cn3)CC)C2)=O)cc1 17705,C1(C(=O)NCC(CNC(=O)CCc2nc(C3CC3)no2)CO)(OC)CCCSC1 17706,c1(C(=O)NC2C=CCN(C(C(c3ccn(C)n3)(C)C)=O)C2)ccc2cc[nH]c2n1 17707,C1(NC(c2nc(-c3cn(C)nc3)oc2)=O)CCCCN(C(C2CC(F)C(=O)N2)=O)C1 17708,N1(C(CC(C)OC)=O)CCCC(CC(=O)Nc2cccc(-n3cc(C)cn3)c2)C1 17709,c1(C(=O)NCC(C)(C(C)C)NC(c2c(C)nccc2)=O)oc2ccccc2c1C 17710,C1(NC(CC2CC(C)C2)=O)CCCC1CNC(C1CS(=O)(=O)C1)=O 17711,C1(C)(C(N(C2CN(C(=O)CCc3cocn3)C2)C)=O)CCCCNC1=O 17712,CC(C#N)C(=O)N(CC(O)CN(C(=O)CN(C)C(=O)Cc1ccccc1)C)C 17713,C1(CC#C)(C(=O)NCCCO)CCN(C(=O)CNC(=O)OCC)C1 17714,N1(C(C2C(CC(C)C)C2)=O)CCC2CN(C(=O)CN3C(=O)C(C)C(C)C3=O)C2C1 17715,N1(C(COCC#C)=O)CCC2CCCN(C(c3ccccc3Br)=O)C2C1 17716,c1(C(=O)NC2CN(C(CCCOCCOC)=O)C(C)CC2)cc(O)cc(C#N)c1 17717,Cn1cnc(C=CC(=O)NCC(=O)NC2COCCOC2)c1 17718,n1(CC(=O)NC23CN(C(C(C=C)O)=O)C(COC)(C2)C3)cc2ccccc2n1 17719,c1(C(=O)NC2CCCC(NC(CC3C(C)(C)C3)=O)C2)c[nH]cc(F)c1=O 17720,c1(N2CCCC(O)(CS(=O)(=O)NC)C2)nc2ccccc2n1C 17721,Clc1ccc(C(c2nnnn2CC2CC2)NC23CC(C2)C3)cc1Cl 17722,c1(CC2OCC(C)C2)cccc(NC(=O)N(C2CSC2(C)C)C)c1 17723,C1(C)(CC)CC(NC(=O)Cn2cc(C(c3c(C)cccc3C)O)nn2)CCO1 17724,C1(C(=O)NCC2(F)CCN(C(C3(CC(=O)OC)CC3)=O)C2)CN(CP(C)(C)=O)C1 17725,C1(c2cn(CCN(C)CC)nn2)CN(C(=O)Cc2csc(C)c2C)CC1C 17726,c1(CCC(=O)NC2C(CC(=O)OCC)CCC2)cc(F)ccc1C 17727,N1(C(c2ccc(N(CCC)C)cc2)=O)CCN(C(C2CC(CF)C2)=O)C(CC)C1 17728,c1(OC)cncc(C(=O)NCC(C(C)C(C)C)NC(c2sccc2C#N)=O)c1C 17729,c1(C(N2C(C)CN(C(=O)C=CCN3CCOCC3)CC2)=O)cn2cnnc2cn1 17730,N1(C(=O)C=Cc2ccccc2)CCC(F)(C(N2CCC(CO)C2)=O)CC1 17731,C(c1cccs1)=C(C)C(=O)NCCN(C)C(c1conc1C1CCCO1)=O 17732,c1(C(=O)NCC2CN(C(CCCCOC)=O)C(C)(C)C2)cc(C)c(C#N)c(C)c1 17733,C=CCC(C(=O)N1CC=CC1CN(C)C)NC(=O)CC(C1CC1)C1CC1 17734,C1(CNC(CSCC=C)=O)CN(C(C2COC(=O)N2)=O)CCC1C 17735,CN1CC(NC(C2CC(F)(F)CN2C(C2CCCC2O)=O)=O)C2(CC2)C1=O 17736,C=C(C)C(C)(C)C(=O)NC(C1CCCN1C(c1coc(C(F)F)n1)=O)C 17737,CC1CC(C(=O)NCCC2CCN(c3nccc(CO)n3)C2)CCN1C 17738,N#CC1(C(=O)O)CC(NC(=O)NC(c2ccc(Nc3ccccc3)cc2)CF)C1 17739,N1(C(C2N(CC)CCC2)=O)CCC(C(C)C)C1CNC(=O)Cn1cnc(C#N)n1 17740,C1(C(=O)NCC2CC(CNC(C(Cc3ncn(C)c3)O)=O)C2)Cc2nccn2C1 17741,c1(OC)ccc(NC(=O)C(CCN(C)C)NC(c2cc(C(C)C)on2)=O)cc1O 17742,C1(CCC)CN(C(=O)C=CBr)CCN1C(C1CCC1(C)C)=O 17743,c1(NC(CSCC(=O)N(C)CCc2ccccn2)=O)ccc(Cl)cc1 17744,C(=O)(C1CCc2c[nH]nc21)NC1(CCCC(=O)Nc2cccc(O)c2)CCC1 17745,C1(C(=O)NCC2CCN2C(=O)C(F)(F)CC2CCCO2)CCC([N+](=O)[O-])CC1 17746,CCC(CCOC)N.C12CC(C1)NC1(CCC1)CC(=O)C(=O)C2 17747,Cc1nc(O)nc(O)c1CC(=O)NCc1cccc(NC(=O)Cn2cncn2)c1 17748,c1(SC(c2cn(CC(CNC(=O)C(C)OC)OC)nc2)C)ccccc1 17749,C1(C(=O)NCCCCNC(C(c2cccc(OC)c2)C)=O)OCCOC12CCC2 17750,N1(C(c2n(C(C)C)ccn2)=O)C2CCCC1CN(C(C1CCCS1)=O)C2 17751,CC1C(NC(c2ccc(N(C)C)s2)=O)CCN1C(=O)CC(F)(F)F 17752,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CO)CCC3)=O)C2)CC1 17753,N1(C(c2c(C)nn[nH]2)=O)CCC2C(CCN2C(c2cccc3nccn23)=O)C1 17754,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)C=CCCC2)C1 17755,N1(C(C(CC=C)CNC(C2CC(=O)NC(C)C2)=O)=O)CC(C)(C)C12CCC2 17756,Cc1csc(C(=O)NC2(CCCNC(=O)C(F)F)CC2)c1Cl 17757,c1(C(=O)NCC(CC=C)NC(c2csc(=N)[nH]2)=O)nn(C)c(Cl)c1Cl 17758,C1(C(=O)NC2CC(CCOC)C2)C=CCN(C(=O)C(CCOC)OC)C1 17759,C1(C)(CC(=O)NCC(C(C)C)OC)CCN(C(=O)C(C2CC2)OC)C1 17760,C1(NC(c2cn(C)nc2-c2ccoc2)=O)CCN(C(=O)C(Cl)=CCl)CC1F 17761,O=C1NC2CCC1CN(S(=O)(=O)c1ccc(N3CCCC(C(F)F)C3)nc1)C2 17762,C1(O)(CC(=O)NCC(CC=C)NC(=O)CCc2cccnc2F)CCCCCC1 17763,N1(C(=O)Nc2cccc(OCC)c2)CCC(NC(=O)COC)C(C)(C)C1 17764,C1(OC)(OC)CN(C(c2ccn(C(F)F)n2)C(=O)Nc2cccnc2)C1 17765,c1(CN(C2CC2)CCOCCO)cccc(COC)c1.CC(CC1C(=O)N1)NCC 17766,c1(C(=O)NC(C)CN(C(=O)C(O)CC2CCCCC2)C)cnc2[nH]ncc2c1 17767,c1(C(N(C2CN(C(C(CCN(C)C)O)=O)CC23CC3)C)=O)ccn2ccnc2n1 17768,c1(OC)ccc2[nH]c(C(=O)NCCCCCSC)nc2c1 17769,C#Cc1ccc(F)cc1C(=O)NCC(C)(C1CC1)NC(c1cn(CCCC)nn1)=O 17770,N1(C(c2c(CC)ocn2)=O)CCCC(CC(=O)NCCOC(C)=O)C1 17771,N(C1CC2(CC2)Oc2c(C)cccc21)C(CC1C(OC)CC1)=O 17772,C12(C(=O)NC(CCC=C)C)CC1CN(C(c1cc(C(=O)OC)[nH]n1)=O)C2 17773,c1(SCC)cccc(CC(=O)NCC2CCN2C(c2ccc(C(F)F)nc2)=O)c1 17774,Cc1cc(C)c(C(N2CCC(N(C)C(c3cn(C(C)(C)C)nc3C)=O)C2)=O)cn1 17775,CCCCCC(=O)N1CCC(CCOC)(NC(=O)COc2ccc(OC)cc2)C1 17776,N1(C(C2CC2C2CC2)C)CCCC(C(N2CCC(c3ccccc3)C2)=O)CC1 17777,C1(NC(CC2(C=C)CCC2)=O)CN(C(c2sc(C(F)(F)F)cc2C)=O)CC1C 17778,CC#CCCCC(=O)NCC1CCC(NC(=O)Cc2noc(C)c2C#N)CC1 17779,N1(C(C(C)SC)=O)CCC(C2CC2)(CNC(c2cccc(N(C)C)c2)=O)C1 17780,C12CCC(C)(C)CC1CNC2=O.C1(C(C)(C)C)(CO)CCN(C(c2ccc[nH]2)=O)C1 17781,C1(CC)CN(C(c2cocc2C(=O)OC)=O)CCN1C(=O)CC1CCCCC1(C)C 17782,N1(C(CC(CC#C)NC(C2CC(C)N(C)C2)=O)=O)CC2(C1)OC(=O)NC2C 17783,C1(CC)CCCN(C(=O)C(n2ccnc2C)C)C1C(=O)NC1COCC(C)(C)C1 17784,Cc1cc(C(N2CCN(C(c3cc(C)ncc3Cl)=O)CC2CO)=O)ncc1N 17785,c1(NC2CCN(C(CCc3cc(C)on3)=O)C(C)C2)ncc([N+](=O)[O-])c(C)n1 17786,c1(C(N(CC(C)NC(=O)Cc2cc(O)nc(O)n2)C)=O)cc2n(n1)CCCC2O 17787,c1(Cn2cc(COC)nn2)cc2cc(C)cc(C)c2[nH]1 17788,CC1CN(C)C(C)CN1C(=O)CNC(C1CC2CCC1CC2)=O 17789,c1(C(=O)NCC2N(C(C3(C)CCC(=O)N3)=O)CCN(C)C2)cc2ccncc2s1 17790,Cc1ccc(NC(c2ccc(-c3ccc(C)cc3)cc2)=O)c(O)c1.C12CN(C1)C2 17791,c1(C(N2C(CNC(C3CCC(C)(CC)O3)=O)CC2)=O)cc(C)nc2onc(C)c12 17792,c1(C(=O)NC2C(C(N3CC(SC)C3)=O)COCC2)ncnc(O)c1F 17793,C1(NC(CCN(CCCO)C(NC(Cn2ccc(C)n2)=O)=O)=O)CCC(=O)NC1 17794,C1(CC(=O)NCC(C)C)CC(NS(C)(=O)=O)C1.C(C(=O)NC1CC1SC)OC 17795,c1(OC)ccc(CCC(=O)NCC2(COC)CC2(F)F)cc1.C12(CC1)C(=O)NC2 17796,c1(C(=O)NCC2N(C(c3cncc(C#C)c3)=O)CC2)[nH]cc2c1CCCC2 17797,c1(C(N(C)CCC2CCCCN2C(=O)CC2CCOC2)=O)cc2sccc2[nH]1 17798,N1(C(C(=O)NC(c2ccc(F)cc2)C)c2cccs2)CCC(C)(O)C(O)C1 17799,C1(C)(C(=O)NCC2CN(C(C(c3ccc(Cl)s3)C)=O)C2)CC2CC2C1 17800,CCCC(C(=O)NCC=CCOC)N(CCCO)C.N12CC3C(C3C1)C2=O 17801,c1(C(=O)NC2C(SC)CN(C(c3cnc(O)o3)=O)C2)ccc2c(c1)NC(=O)C2 17802,C(=O)(CC1=CCN(C)CC1)NCC(C)NC(c1ccc(CN(C)C)o1)=O 17803,c1(OC)nc(Cl)ccc1C(=O)NC(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)C1 17804,c1(NCC=CC)[nH]c(=NC(CCO)CC(C)C)nc2c1ncn2C 17805,C1(CC(=O)OC)CCCN(C(=O)CCC2CCN(C(C3CCOC3=O)=O)CC2)C1 17806,C#CCC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CSc1nncn1C)C1CC1 17807,c1(N(CCN(C(C(C(C)C)OCC)=O)C)C)cc2nnc(C(C)C)n2cn1 17808,C(=O)(C1Cc2c(Cl)cccc21)N1CC(C(C)NC(c2ccc([N+](=O)[O-])n2C)=O)C1 17809,c1(NC(C=CC2N(C(N3CCC(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17810,N1(C(C(C=C)(C)C)=O)CC(NC(c2cc(C(C)C)on2)=O)CC2(CCC2)C1 17811,N1(C(c2n(C(C)C)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17812,C1(C(=O)NCC2C(CNC(=O)COC(F)(F)F)C2)Cc2ccc(F)cc2C1 17813,C1(NC(c2ncc(CC)nc2)=O)CN(C(c2cc(Cl)no2)=O)C2(CCC2)C1 17814,Cc1ccc(-n2cc(C(=O)NC(Cc3ccccn3)C(=O)O)cn2)cc1 17815,N1C(=O)c2ccccc2C1=O.n1(CCOC(C)(C)C)ccc(CCN2CCCC2)n1 17816,C1(C(=O)NC(C(N2CCC(C)C2)=O)C2(C)CC2)C2C3CCC(C3)C12 17817,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17818,c1(CC)ccc(C(=O)NCC2C3CCC(C3)N2C(C2CC23CCOC3)=O)c(F)c1 17819,c1(C(=O)NCC2C3CN(C(CC(C)NC(N)=O)=O)C2C3)cc2cccnc2o1 17820,c1(-c2ccc(SC)cc2)c[nH]c(=NCc2ccc(C(=O)O)cc2F)s1 17821,N1(C(c2c(CC)ccs2)=O)CCC(C(=O)NCC(CSC)OC)CC1 17822,Cc1ccn2c(C(N3CCOCC3CNC(=O)C(O)CF)=O)cnc2c1 17823,Cn1c(C(N2CCC(c3ccc(Cl)cc3)CC2)=O)cc2cc(C(F)(F)F)cnc12 17824,N1(C(c2n[nH]c(CC)c2C)=O)CC2CCCC2(C(=O)NCCC(C)C(C)C)C1 17825,N1(C(c2n(CC)ncc2)=O)CC(NC(c2sc(Br)nc2C)=O)C2CC12 17826,c1(C(=O)NCC=CCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17827,c1(CC)cc(C(=O)NCCNC(=O)COCc2cccc(C)c2)nn1C 17828,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17829,c1(C(C)=O)ccc(CN=c2ccc(C(=O)NS(=O)(=O)C(Cl)(Cl)Cl)c[nH]2)c(C#N)c1 17830,N1(C(CCNS(CC)(=O)=O)=O)CCCCC1CCN(C)C(C1(CCOC)CC1)=O 17831,n1(C(C)C)cc(C(=O)NCC(C2CC2)NC(C2CCCSC2)=O)c(Br)n1 17832,C(=O)(C(C)(C)C(=O)c1ccccc1)NCC(CC=C)NC(C1(SCC)CC1)=O 17833,c1(C(N(CC(C)NC(c2n(CC)ccc2)=O)C)=O)cc(Cl)ccc1F 17834,C1(O)(C(C)NC(COCC=C)=O)CCN(C(C2CCC2SC)=O)CC1 17835,c1(C(N(CC(C)NC(c2cn(C3CCOC3)nn2)=O)C)=O)cc2ccsc2s1 17836,C1(C#N)(C(=O)NC(C)CC2CCN(C(=O)C(F)(F)CO)CC2)CC2CCC1CC2 17837,C1(NC(c2ccn(CC)n2)=O)CC2CC1CN(C(=O)CN(C)C(C)=O)C2 17838,CC(CF)CC(=O)NC1CCCC1NC(c1cccnc1)=O 17839,c1(C(N(C2CCCN(C(=O)C(O)C3CCCC3)C2)CC)=O)cc2cnccc2[nH]1 17840,C1(NC(C2N(CC#C)CCC2)=O)CC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 17841,C=C1CC2(CCN(C(c3ccccc3)c3nn[nH]n3)CC2)C1 17842,c1(CC(C(=O)NCC(CO)NC(COCCC=C)=O)C)ccc(Cl)cc1 17843,CNS(=O)(=O)NCC(=O)NC(C1CCC(NC(c2coc(C(F)F)c2)=O)C1)(C)C 17844,C1(C(C)C)CCCN(c2nnc(-c3cc[nH]n3)n2CC2CCOC2)C1 17845,N1(C(CC(C2CC2)NC(COC(C)=O)=O)=O)CC(O)CC1(C)CO 17846,Cn1cccc(C(N2CC=CC2(C)C(=O)Nc2ccc(C(N)=O)c(F)c2)=O)c1=O 17847,C1(O)(CF)CCN(C(=O)CN2CCCCC2=O)CC1.C12C(CCC13CCC3)CN2 17848,n1(CC(=O)N(C2CS(=O)(=O)C2)CC(C)C)cc(Br)ccc1=O 17849,C(c1ccc(F)c2ccccc12)=CC(N1C(CNC(CCC(C)C)=O)CC1)=O 17850,c1(NC(C2CC(n3cc(CCN(C)C)nn3)C2)=O)ccc(OC(F)F)cc1Cl 17851,C(=O)(C(CNC(c1nc[nH]n1)=O)CC1CCC1)NC(C)(C)C1CCC1 17852,N(C(=NCCCN1CCc2ccccc21)N1CCC(C)C2(CCC2)C1)C(CC)C 17853,c1(C(N)=O)ccc(C(N)=O)cc1.c12cn(nn1)CCNC(=O)OC2 17854,C=CC(C)(C)CC(=O)N1CCC(N(C(=O)C(CNC(C2CC2)=O)CCC)CC)CC1 17855,N1(C(c2c(COC)nn(C)c2)=O)CCCC1C1CCCN1C(=O)Cn1ncnn1 17856,C(=O)(C1=CCC2CCC1N2C(=O)C(Cl)Cl)N(c1ccco1)C(C)C 17857,c1(OC)cc(Br)ccc1C(c1nnnn1Cc1cccc(OC)c1)NCC(N)=O 17858,c1(OC)cc(CN(C2CCCN(C(=O)Cc3ccc(Br)cc3)C2)C)c(F)cc1O 17859,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17860,C1(NC(CCNC(=O)NC)=O)CC2(C1)CC2NC(c1cnn(-c2ccccn2)c1)=O 17861,C1(CC(=O)N(CC)CC2CN(C(C3(CCOC)CC3)=O)C2)CCCC1C 17862,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CCCC2)ccc(C(F)(F)F)c(N)c1 17863,C1(C)(CNC(c2occ(C(C)=O)c2)=O)CCN(C(=O)Cn2cnnn2)CC1 17864,c1(-c2nc(C)on2)ccc(CNC(C2(C)CCCN2C(=O)C(C)N(C)C)=O)cc1 17865,c1(CCC(=O)NC2(CNC(CCC(CC)C)=O)CCOC2)cnc2ccccn12 17866,N1(C(=O)C(Cl)=CCl)CCC(C2CC(NC(C34CCC(CC3)CC4)=O)C2)C1 17867,c1(CC(=O)NC(CNC(Cn2c(C)ccc2C)=O)(C)CO)cnc2ncccn12 17868,CC1CN(C(c2cn(C(F)(F)F)cn2)=O)CC1(C)CNC(=O)CCC1CC1(Cl)Cl 17869,C(=O)(CCCC(F)(F)CO)NC(C)CC1CN(C(c2c[nH]nc2F)=O)C1 17870,N1(C(=O)CCc2ccc(Br)cn2)CCC(F)C(NCc2cc(O)cc(F)c2)C1 17871,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(C3CCCO3)C2)=O)C1 17872,N1(C(C(C)n2ccnn2)=O)CCC(O)C(N(C)C(c2cc3n(n2)CCO3)=O)C1 17873,CC1CC(C(=O)N(C(C)CN(C(=O)C=Cc2ccc(=O)oc2)C)C)CC(=O)N1 17874,N1(C(C2(C(=O)NC)CC2)=O)CC(NC(c2cc(C(F)F)cs2)=O)C(C)C1 17875,C1(CN(C)C(c2ccc(-c3nc[nH]n3)cc2)=O)CCCCN1Cc1ccccc1 17876,c1(OCC=C)ccccc1C(=O)NCC1(NC(=O)C(CC)SC)CCCC1 17877,CC1(C)C(CNC(c2nc(Cl)sc2Cl)=O)CCN1C(=O)CC1CCC(O)C1 17878,C1(C(C)NC(CCc2ccc(C)o2)=O)CCCN(C(C2CC=CCC2)=O)C1 17879,C1(CC)CC(NC(=O)C2=CCOCC2)CCN1C(=O)Cc1cncs1 17880,c1(CC(N2CCC(F)(C(=O)NCCSCC)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 17881,N1(C(CC2CC(CC)C2)=O)CC(C)N(C(=O)CN2CSCCSC2)CC1C 17882,c1(NC(CCC)=O)ccc(OC2CCN(C(c3ncc[nH]c3=O)=O)CC2O)c(C)c1 17883,C(C(=O)N1CC(O)(C(C)NC(=O)CC2CNC(=O)O2)C1)(C(C)C)SC 17884,c1(C(N(C2CCCC3CN(C(COC)=O)CC32)C)=O)cccc(S(N)(=O)=O)c1C 17885,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC(NC(=O)C=CC(C)C)C2(CCOCC2)C1 17886,c1(C(=O)NC2(C#C)CC2C(F)(F)F)c(F)ccn1C 17887,Cc1cccc(C(O)C(=O)NC(C)CN(C(=O)CC2CC3C=CC2CC3)C)c1F 17888,C1(NC(c2ccc(N(C)C)cn2)=O)CC2CCC1C(NC(=O)C1=CCCOC1)C2 17889,C1(C(N2C(C(N(C3CCCC3(C)O)C)=O)COCC2)=O)CC(=O)NC(=O)C1 17890,c1(NC(c2ccc(CC)cc2)=O)c[nH]c2cc(CN)cnc12.c12cc(ccn1)OC2 17891,N1(C(C(Cc2cnc[nH]2)OC)=O)CCC2(C1)CN(C(=O)C(O)C(C)C)C2 17892,N1(C(c2cc(SC)c(C)o2)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 17893,CCC1=NOC(C(=O)N(CC(C)NC(c2cnc(CC(C)(C)C)s2)=O)CC)C1 17894,c1(C(N(CC(C)NC(C2CCCCCN2C)=O)C)=O)cccc(C#N)n1 17895,C(=O)(CC1=NNC(=O)C1)NCC1N(C(c2ncc(OC)nc2)=O)CCCC1C 17896,N1(C(C2CCC(CC)CC2)=O)C(CNC(c2cncc(Cl)c2)=O)CC2COCC12 17897,N1(C(CCn2c(CC)cnc2)=O)CC2(CC(C(=O)N(C)C(C)C3CC3)C2)C1 17898,C1(Cn2cc(-c3c(C(C)(C)O)cccc3)nn2)CCN(C(=O)C(F)(F)Cl)CC1(F)F 17899,N1(C(C2CN(C)C2)=O)CCC(CNC(C2CCCS2(=O)=O)=O)CC1 17900,N1(C(C(COC)C)=O)CCOC2(CCN(C(C3CC(=O)C3)=O)C2)C1 17901,c1(C(C)OCC)cccc(C2CCN(c3cc(-c4ccccc4)ncn3)C2)c1 17902,CCCC(CCC)C(=O)NC(C)CC(C)NC(C1CC1(C)Br)=O 17903,n1(C(CC)C)cc(CN(C)CC2CN(C(=O)OC(C)(C)C)C2)c(C)n1 17904,N1(C(C=NOC)=O)CC(NC(=O)CSc2cccc(F)c2)CC2(CCC2)C1 17905,CC1CCCn2cc(C(=O)NCC3CN(C(C4CN(S(N)(=O)=O)C4)=O)C3)nc21 17906,CCC(O)(C(=O)NCCCCC(C)NC(=O)C=CC1CCC1)c1ccccc1 17907,N#CC1C2CCC1CN(C(C13CC(CO1)N(C(=O)CC1OCCO1)C3)=O)C2 17908,CN1CC(NC(=O)NCc2occc2Br)C(C)(C)C1 17909,C1(C(N2CCCC(CNCC)C2)=O)CC12CCOCC2.C(=O)(CC(C)(C)C)C(=O)CN 17910,Cc1cc(Cl)cc(NC(=O)CC2COCCN2Cc2ccc(C)c(C)c2)c1O 17911,N1(C(C(C)OCC2CCCO2)=O)CCCN(C(=O)C(C2CCCCC2)F)CC1 17912,c1(C(N(CC(CNC(C(n2ccc(C)n2)C)=O)O)C)=O)c(C)nc(O)nc1S 17913,n1(CC)nc(C(N2C(C(=O)NCCCN(C)C)CC3CC23)=O)c(I)c1C 17914,c1(-c2ccc(C(C)NC(=O)CCC=Cc3cnc[nH]3)nc2)cc(F)ccc1NC 17915,CC(C)CC(O)CNC(C1CCC(C2CC2)N1C(=O)Cn1cnnc1O)=O 17916,N1(C(C)Cc2ccc(Br)cc2)CCN(C(C2CCCCC2)=O)C(C)C1 17917,N1(C(CC(C=C)CC)=O)CC2(C(=O)NCc3cnc(C)cc3C)CC1CCO2 17918,c1(CC(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 17919,C1(C(N(CCNC(C(c2ccc(OC)cc2)CC)=O)C2CC2)=O)CSCC(=O)N1 17920,C1(N(C)C(C2CC=CCC2)=O)CCCN(C(c2conc2C2CCCC2)=O)C1 17921,c1(C(N2CCC(F)(CNC(C3CC(CC)OCC3)=O)C2)=O)cc2nc[nH]c2cn1 17922,C(c1ccc(C)c(C)c1)=CC(=O)NC(CCOC)CNC(=O)C(O)CC1CC1 17923,c1(C(N(CC(C)N(C(C(CCC)CC)=O)C)C)=O)ccc2c(c1)CN(C)CC2 17924,C=CCC(C(=O)NCC1CCC(NC(C2CCC3CC3CC2)=O)C1)C(C)C 17925,C(=O)(C(C)(F)C(F)(F)F)N(CC=CC(=O)NCCC(C(C)C)CO)C 17926,Cc1cc(Cl)cc(CNC(C2OCCN(C)C2c2ccccc2)=O)c1O 17927,C(C(CC(=O)NC1CCN(C(C2CCCS2)=O)CC1)C(F)F)N(C)C 17928,C1(NC(c2cccc(CC)c2)=O)CCCCN(C(=O)C(C(C)N(C)C)N(C)C)C1 17929,C=C(Cl)CC(C(=O)N1CCC1CO)NC(c1nnn(C)c1C)=O 17930,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cc(Cl)sc2Cl)=O)CC1)NC 17931,C1(NC(c2c(CCC)onc2C)=O)CN(C(C2(C)COCCO2)=O)CC12CC2 17932,C(=O)(C1=CCSC1)NCC(C1CCCCC1)NC(CC(C)OC)=O 17933,N1(C(CN(c2ccncc2)C)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O 17934,CC1CC(C)N(C(c2c(Br)ccnc2F)=O)CCN1C(=O)CC1CC1 17935,N1(C(C23CC(C)(C2)OC3(C)C)=O)CCC2CC(NC(c3cscn3)=O)CCC2C1 17936,C1(CCC(=O)N(CCOCCO)CC)CCN(C(=O)CN2C(=O)CNC2=O)CC1 17937,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 17938,C=CC1(C(N2CC3CC2C3)=O)CCN(C(C2CCCN3CCCC23)=O)CC1 17939,CC1(C)CC(NC(=O)NOCC(C2CCOC2)O)C1 17940,C1(CNC(C(c2cn(C)nn2)NC(=O)CCc2cnoc2)=O)C2CCC(F)C12 17941,N1(C(c2nc(N(C(C)=O)C)sc2)C(=O)NC2CC2)CCCCC12CCCCCC2 17942,C12(NC(c3n(C)ccc3)=O)CN(C(C3CC=CC3)=O)CC1CS(=O)(=O)C2 17943,C1(NC(C(C2CN(C(C3(CC)CCCO3)=O)C2)O)=O)CCCCCC1C 17944,Cn1ncc(C(=O)NCCOCCOCCNC(c2cscc2Br)=O)n1 17945,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 17946,c1(-n2cc(CCCC(C)C(=O)N3CCS(=O)(=O)CC3)nn2)nc2ncccn2n1 17947,c1(C(=O)NCC2C(C)CCCN2C(C2(N(C)C)CCCC2)=O)cccc2ccnn12 17948,Cc1oc(C(C)C)nc1C(=O)NC1CCCC1NC(=O)C(O)c1ccsc1 17949,C(=O)(C(CC)(CC)CO)N1CCC(NC(COCC)=O)C(F)C1 17950,c1(CC(=O)NCC2C(NC(C(C)OCCCC)=O)C2)ccc(Br)nc1 17951,C1(C(=O)Nc2cccc(C(F)(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 17952,Cc1ccc(C(=O)NC2CN(C(C3C4CCCCCC34)=O)C2)nc1C(F)F 17953,CC1CN(C(=O)C(C)(C)C2CC2)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 17954,C(=O)(CC(C)C(F)F)N(CC1CCC(F)(CNC(Cc2cncc(C)c2)=O)C1)CC 17955,Cc1ccc(NC(=O)C(N2CCC(C)(NC(c3cscn3)=O)C2)=O)c(C)c1 17956,C1(NC(C(=C)Br)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 17957,c1(OCC(=O)NC2CC(C)(CCNC(C3CC(=C)C3)=O)C2)ccc(Cl)cc1F 17958,CC(C)(C)CCC(F)C(=O)N1CCCC(CC(N2CC3CC3C2)=O)C1 17959,C1(N(C)C(=O)NCc2nc(-c3ccccc3)no2)CCCCC1C(F)(F)F 17960,C1(NC(C(CO)NC(N)=O)=O)COC2CN(C(c3cc(O)ccn3)=O)CC12 17961,CCC(C)(CO)C(=O)NCC(F)CNC(=O)CN1CCCCC1=O 17962,C1(C)(CC(=O)N(CC(=O)N(CCF)CCOC)CCC)CC1(F)F 17963,C1(CCN=C(NCC(CC)CC(F)(F)F)NCC(F)F)CCC2(CCCC2)CC1 17964,C1(O)(C(=O)NC2CCC(CNC(C3=NOC(C)C3)=O)CC2)CCCC(C)(C)CC1 17965,Cc1cc(C)c(CN2CCC(=CC(=O)NC3CSC3)CC2)c(C)c1 17966,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 17967,C1(N(C)C(C2(C)CC2C(F)(F)F)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 17968,c1(C(N(C)CC2N(C(COCCC#C)=O)CC(F)C2)=O)cc2c(C)cccn2c1 17969,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 17970,N1(C(CSCC=C)=O)CC(NC(=O)CCOC(C)CC(C)C)C2CCCC12 17971,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(c2ccccc2Cl)O)CC12CCC2 17972,C1(NC(C(C)=C2CC2)=O)CC(F)(F)CC1NC(c1ccc(-c2ccco2)o1)=O 17973,c1(N(C)C(C2CCC(C(=O)O)N2)=O)cc(-c2cccnc2)cn1C 17974,c1(C(=O)NCC2CCCC2NC(C2(CF)COC2)=O)cc(Cl)cnn1 17975,C1(NC(C(C)=CC2CC2)=O)CN(C(C2CCN(CC(C)C)C2)=O)CC1C 17976,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N(c1ccccc1)CC(C)C 17977,c1(NC(C2C(CC)N(C(c3cc(O)nc(O)n3)=O)CC2)=O)cc(C)cnc1C 17978,c1(C(=O)NCc2cccc(CNC(C(C=C)(C)O)=O)c2)cc2cccnc2o1 17979,C1(NC(c2cc(C)sn2)=O)CC2CN(C(C3(C#N)CC34CCC4)=O)CC12 17980,c1(NCC23CC(NC(c4ncc(C(C)C)cn4)=O)(C2)C3)cccc(Br)c1Cl 17981,C(=O)(C(C)(C)CN(C(=O)CC1CCC1)C)N(C)CC1CCN(C)C1 17982,C(=O)(CC(C(F)F)NC(C1CC(F)C1)=O)N(CCCCC)C 17983,C(=O)(C1=CCCCO1)N1CC(NC(c2c(C)oc(-c3cccs3)n2)=O)C(F)C1 17984,CC1(C)CC(CC(N2CC(CNC(c3ccc(Cl)s3)=O)C2)=O)C1 17985,C1(C(=O)NCCCC(C)NC(COCCCC)=O)CN(C(C)C)CCO1 17986,Cc1nc2c(Cl)cccc2cc1C(=O)NCCN(C)C(C1CNC(=O)N1)=O 17987,c1(C(N2CC(O)(CCNC(c3c(CC)ocn3)=O)C2)=O)c(C)cc(Cl)nc1N 17988,C1(C(=O)NCC(C)(C)CO)CCCCC1(C)NC(c1nnc(O)nc1O)=O 17989,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 17990,c1(C(=O)NC(C)(CNC(=O)C2=CCOCC2)CO)ccc2nc(O)[nH]c2c1 17991,C1(CN(C(C2N(CC)CCC2)=O)C)CCCN(C(=O)CCC(C)(C)N(C)C)CC1 17992,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(C2CC2c2ccsc2)=O)C1 17993,c1(C(=O)NC(CCC)C(=O)N2CCC(C)(N(CC)CC)C2)cc(C)nc(O)n1 17994,c1(OCC)ccc(C(=O)N(CC(C)NC(=O)Cc2nncn2C(C)C)CC)cn1 17995,N1(C(c2c(C)noc2C)C(=O)NCC(F)F)CCC2(CCOC2=O)C1 17996,CON1CCC(CC(=O)NC23CCC(CC2NC(=O)CC2CCOC2)C3)CC1 17997,N1(C(c2cccc(C(C)(F)F)c2)C(=O)NC(CC)C)CC(OC)CC(O)C1 17998,N1(C(N(S(=O)(=O)c2cccc(NCC=C)c2)C)=O)CC2CCCC(F)(F)C2C1 17999,N1(CC(N2CCC(CC(N3C(CCC)CCC3)=O)C2)=O)CCCCCC1 18000,N(C(=NCCCP(C)(C)=O)NC1CCOC1)Cc1c(OC)cccc1OC 18001,C1(CNC(C2(OC)CCCOC2)=O)C2CCCC1N(C(=O)C=Cc1ncco1)C2 18002,CN1CCC(CC(=O)NC2(C)CC(C(=O)NC3CCCC3)C2)CC1.C1CCO1 18003,CC1CCC(C(=O)N(C)CCN(C)C(c2ccc(C(C)(F)F)cn2)=O)C(=O)N1 18004,N1(C(CC2(C)CCN(C(C3N(C)CC(O)CC3)=O)C2)=O)CCN(C)C2(CCC2)C1 18005,c1(C(C)C)ccc(C#N)c(N2CC=C(CNC(=O)CCn3cccn3)CC2)n1 18006,CCC(C(C)CN(C)C)NC(=O)C(Cc1cc[nH]n1)NC(=O)CCc1ccco1 18007,c1(C(=O)N(c2ncncc2I)CC2(F)CNC2)ccc(Cl)c(F)c1 18008,C(=O)(C(O)P(C)(C)=O)N1CCCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 18009,c1(OC)c(C(=O)NC(C)CC(C)NC(c2sccc2F)=O)cc(F)cc1F 18010,CC1(C)CC(NC(C2CCC(C(=O)O)NC2=O)=O)Cc2ccsc21 18011,C1(CNC(c2coc(Br)c2)=O)CCCN(C(C2CCC3CC23)=O)C1 18012,N1(C(C2CC(CCC)C2)=O)CCCC(C)(CNC(C2(C)CCCCO2)=O)C1 18013,c1(C(=O)NC2CC(NC(c3cc(OC)ncc3F)=O)C2)cccc(C=C(F)F)c1 18014,c1(C(N2CC(NC(c3c(N(C)C)nccc3)=O)C2)=O)ccc(-n2cncn2)cc1C 18015,N1(C(CCc2nc(C)c(C)[nH]2)=O)CC2(CNC(C3C(C)(C)C3(F)F)=O)CC1CO2 18016,O=C(C1=COCCO1)N1CCCC1C1(O)CN(C(c2ccnc(CO)n2)=O)C1 18017,CC(C)C(C(=O)NCC1(C)CN(C(C2CCCCC2C(N)=O)=O)C(C)(C)C1)C(C)C 18018,C1(c2cn(C)nc2)CCC(NC(=O)C(N2CCCC(O)C2)=O)CC1C(F)(F)F 18019,C(=O)(C(C)CC(F)F)N1CCC(N(C(=O)C=CC2CCCN2C)CC#C)CC1 18020,C1(C(=O)NCC(CO)NC(C2CCCCC(=O)N2)=O)C2CCC3C(C2)CC13 18021,N1(C(CC=C=C)=O)CCC2(CCCN(C(=O)C(C3CCOCC3)F)C2)CC1 18022,C(C(C)(O)C(C)CC)NC(=O)NCC1(CC)CCCOC1 18023,Cc1ncsc1C(=O)NCC(O)CN(C(=O)C(c1ccccc1)C1CC1)C1CC1 18024,C1(N(CC(C)C)C)CCN(C(=O)CNC(C2CCOCC2)C)C1 18025,c1(C(=O)NC(CNC(CC2CC(=C)C2)=O)(C)C2CC2)nnn(C(C)C)c1N 18026,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18027,CN1C2CCCC1CN(C(=O)C(C1CCN(C(C3CN(C(N)=O)C3)=O)C1)F)C2 18028,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18029,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(C2(Cl)CC2)=O)CC1 18030,C1(=O)CC(c2ccc(Cl)cc2)CO1.C(=O)(C(C(C)C)NC(C)=O)N(C)CC 18031,n1(C(C)C)nncc1NC(N1CCC(OCC(N)=O)C1)=O.C(CF)N 18032,c1(C(=O)NCC2CCN(C(C3C(C=C)C3)=O)C2)c(-n2cnnn2)sc(C)c1C 18033,C1(S(C)(=O)=O)(C(N2CC3CN(Cc4c(SC)cc(Br)cc4)C3C2)=O)CCCC1 18034,OCCCCCN=c1[nH]c(=NCc2cc(F)ccc2Cl)[nH]c2c1SCC2 18035,N(C(=NCCC)NCCN(C)C)c1ccc(OC)c(NCCNC(=O)C2CC2)c1 18036,c1(C(C)CNC(=O)C(=O)C(=O)Cn2cnnc2)ccc(C(N)=O)nc1.NC 18037,c1(CC)nc(C(N2C(C(N3CC(O)(CCOC)C3)=O)CC2C)=O)co1 18038,N1(C(c2c(SCCN(C)C)cccc2)=O)CC2CC1CN2C(c1cnsc1)=O 18039,CC1CN(C(C2CCCC2CNC(C2CC(O)CN2C)=O)=O)CCS1 18040,Cc1nc(Cl)ccc1CNC(C1CCN(Cc2cn(Cc3cnns3)nn2)C1)=O 18041,c1(C(=O)NC2(CCNC(CCCN(C)C)=O)CCC2)cc2[nH]ccc2s1 18042,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CCOCC1 18043,c1(C(=O)NC2C(C)N(C(c3ccsc3C#N)=O)CCC2)cccc([N+](=O)[O-])c1O 18044,C1(NC(C(C(C)C)OC)=O)CCN(C(C2CCCCC2C)=O)CC1F 18045,C1(NC(c2ccc(CN(C)C)[nH]2)=O)CCCC(CNC(=O)Cn2nccn2)C1 18046,N1(C(C2(CC=C)CCOC2)=O)CC=C(C(=O)NCC(C)(C)OCCO)C1 18047,C(C(C)(C)CN(C(c1ccc(C(F)(F)F)o1)=O)CC)NC(CCSCCC)=O 18048,C1(C(N(CCCNC(c2cn(CCC)nc2C)=O)C(C)C)=O)CC(C(C)C)=NO1 18049,c1(NCc2c(C)cc(OC(F)F)cc2C)cc(F)c2cn[nH]c2c1 18050,O=S(=O)(c1[nH]c(=NCCCCCF)ccc1Br)NCC1CCCC1C1CC1 18051,N1(C(C#CC(C)C)=O)CC2CCOCC2(NC(c2ccc(Cl)o2)=O)C1 18052,C(=O)(CCCC(C)(C)C)N(C1CCN(CC2CCCCO2)CC1)CCC 18053,C1(C(CO)Nc2ccc(OCCCOC)cc2)CCCC(C)(C)C1 18054,c1(C(=O)NCC(CCC)NC(c2cnc(C3CCCO3)s2)=O)cncc(Cl)c1 18055,C1(OC)CCC(C)(C(N2CCC(F)(CNC(C3CC(CC4CC4)C3)=O)C2)=O)CC1 18056,N1(C(c2nccc(C(F)F)n2)=O)CCCCC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 18057,c1(C(=O)NC2(CNC(C(C)N3CCC3)=O)CC3CCC2C3)nnn2c1CCCC2 18058,CCC(C)(CCC(C)C)C(=O)NC1COCCC1NC(c1nnn(C)n1)=O 18059,c1(CCC(=O)NC2C3CCCN(C3)C(=O)C2=O)ccccc1C.C(C)(C)(C)OOC 18060,C1(NC(CC(COC)COC)=O)CCC2(CCN(C(C3(OC)CCC3)=O)C2)C1 18061,N1(C(CCCCCNC(=O)C=Cc2ccccc2)=O)CCCC2CCCC12 18062,CC1(C)CC(C(=O)NC2CN(C(c3cnc(-c4cccnc4)s3)=O)C2)=NO1 18063,c1(C(N(CC(C)NC(C2C(C#C)C2(C)C)=O)C)=O)c(C)nc(O)nc1S 18064,c1(OC)ccc(CC(N2CCC(NC(C3(O)CCSCC3)=O)C(O)C2)=O)cc1Cl 18065,N1(C(c2cc(CC)ncn2)=O)CCCC(C)C1CCNC(=O)CN1CC2CC2C1 18066,O=C(NOCC(F)(F)F)C(=O)NC1(c2ccc(Cl)cc2)CCOCC1 18067,CCCC(CC)CCC(=O)NCC1CC1CC(N1CC2(CCCN2C)C1)=O 18068,CN1CC2CN(C(C3CCCN(C(c4cc(Br)c[nH]4)=O)C3)=O)CC2C1 18069,c1(C(=O)NCCC2(O)CCN(C(C(C)CN(C)C)=O)C2)ccc(F)c(F)c1F 18070,C1(c2ccccc2)(C(C)NC(=O)C(F)F)CCN(C(=O)C(F)OC(F)(F)F)CC1 18071,N1(C(c2nnc(C)o2)=O)CCC(NC(=O)CCSCc2ccccn2)C12CCC2 18072,N1(C(C(CC)(C)O)=O)CCN(C(c2cc(F)cc(Br)c2C)=O)CC12CC2 18073,C1(NC(C(C)C)=O)COC2(C1)CN(C(c1[nH][nH]c(=N)c1Br)=O)C2 18074,N1(C(C(CC)(C)C)=O)CC(C(N2CC(c3nnc(C)n3C)C2)=O)CCC(O)C1 18075,CCC(CCCC(=O)NCC(C1CC1)C1CC1)NC(c1ccc(C2CC2)cn1)=O 18076,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18077,C1(NC(C2C(C)(C(F)F)C2)=O)CCCCC1CNC(=O)Cc1ccon1 18078,c1(CC(N2CC3(CN(Cc4cncc(C)n4)C3)C2)=O)c[nH]c2ccc(F)cc12 18079,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CC=CCCCCC)=O 18080,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(C)(C)C 18081,N1(C(CCN(S(CC)(=O)=O)C)=O)CCC2(CC1)CC2CNC(=O)CC(C)CSC 18082,CC1C(=O)N(C)CCN1Cc1ccc(-c2cc(F)ccc2F)nc1 18083,N1(C(CCN2C(C)CCCC2)=O)CCC(NC(=O)CC2CCC(=O)N2)C(C)(C)C1 18084,N#Cc1cc(N2CCN(C(=O)Nc3cccc4c3ncn4C)CC2)ccc1[N+](=O)[O-] 18085,C=C(C)CCC(=O)N(CCCOCCNC(=O)CCCOC1CCCCC1)C(C)C 18086,c1(C(N2CC(C)N(C(=O)CC3CCC4CC4C3)CC2)=O)cc2ncccc2[nH]1 18087,C1(C(=O)NCCC2(NC(c3n(C)nc(O)c3)=O)CCC2)CS(=O)(=O)CC12CCC2 18088,C1(NC(C(=O)OCC)=O)CCC(CCC(=O)NCCOCC(N2CCCC2)=O)C1 18089,N(C(=NCCCCF)NC1CCCC1)CC1CCCN(C(COC)=O)C1 18090,N1(C(CCCC(C)=O)=O)CC2(CCC(CNC(=O)CC3CCC4CC34)O2)C1 18091,C1(CNC(c2[nH]cc(CC)c2)=O)(OC)CCN(C(C2CC(=O)N(C)C2)=O)CC1 18092,c1(CC(N2CCC(CCN(CCO)CC(Cl)(Cl)Cl)C2)=O)cc(F)ccc1C(F)(F)F 18093,N1(C(Cc2c(C)cc(O)cc2)=O)CCN(C(=O)CCCC(C)C)CCC1C 18094,C(=O)(NNC(=O)C(C)(C)CCCCOC(C)(C)C)c1n(CCC)ncc1 18095,n1(CC=C)cc(C(=O)NCC2CCCN2Cc2csc(-c3ccccn3)n2)nn1 18096,CC1(C)C(C)(C)C1(F)C(=O)NCCCCNC(=O)COc1cc(F)ccc1F 18097,C1(OC)CCN(C(=O)Cc2ccnc(Cl)c2F)CC12CC2 18098,N1(c2ncnc(C)c2Br)CCC(F)(F)C(C(=O)NC2CCCC(O)C2)C1 18099,c1(NC)ccccc1C(=O)NC1CC(C)N(C(=O)C(C)=C2CCC2)C1 18100,C1(C(N2C(CCC)CN(C(c3n[nH]c(C)c3C)=O)CC2)=O)CCCC1S(C)(=O)=O 18101,c1(OCCCC2(NCCCNC(=O)CN(S(CC)(=O)=O)C)CC2)ccc(O)nc1 18102,c1(-c2sc3cccc(C)c3n2)ncc(Br)c(C)c1[N+](=O)[O-] 18103,N1(C(C2CCN(C)C2c2ccccc2)=O)CCC2(CC(=O)NC2=O)C1 18104,c1(C(C)C(N2CC=CC(NC(=O)Nc3cccc(Cl)c3)C2)=O)c(Cl)cccc1Cl 18105,N1(C(c2c(OC)c(Cl)ccc2)=O)CCN(C(C2CC=CC2)=O)C2CCCCC2C1 18106,C1(C(=O)NCC2C(CNC(Cc3c(C)cnn3C)=O)C2)CC2CC(=O)C1C2 18107,C1(C(=O)NCC(C)(C)NC(=O)CC2CCCNC2=O)Cc2cccc(F)c2O1 18108,N1(C(c2cn(CC=C)nc2)=O)CCC(CN)c2ccccc21 18109,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18110,c1(C(=O)NC(CC=C)CNC(C2CCCOCC2)=O)ccc(OC)cc1Br 18111,C(=O)(CC(C)C(=O)NCC(=O)OCCNC(=O)OC)NCC 18112,Cc1cc(Br)cnc1C(=O)NC(C1CCCN1C(=O)Cc1ccsn1)C 18113,CCC(CN(C)C(c1cnsn1)=O)NC(C1CCCO1)=O 18114,S(=O)(=O)(CC(=O)NC1COCC1NC(=O)CSCC1CCCO1)N(CC)CC 18115,Cc1ncc(C=CC(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(O)n1 18116,c1(C(=O)NCC(CC)NC(=O)CCC2CC(OC)C2=C(C)C)nc(O)sc1C 18117,N1(C(c2cn(C3CCN(C)C3)nn2)=O)CCCC(CN(C(=O)CC(F)F)C)C1 18118,c1(C(N2C(CNC(CS(=O)(=O)COCC)=O)CCCC2)=O)ncc(C)nc1OC 18119,Cc1cccc2c(C(N3CC(C)CC3C(=O)Nc3ccno3)=O)nccc12 18120,C=CC1(C(=O)NCc2noc(C)n2)CCN(C(C2CCCC3CC23)=O)CC1 18121,C=CCC(CO)NC(=O)COCCNC(C1CC12CC2)=O 18122,C1(CNC(C(c2cccc(F)c2)C)=O)CC(C)N(C(c2cccnc2F)=O)C1 18123,c1(OC(C)=O)cnccc1C(=O)NCC(C)CN(C)C(c1conc1C)=O 18124,c1(C(=O)NCCOC(C(C=C)O)=O)cccc(OCc2cc(Cl)no2)c1 18125,c1(OCC)cc(C(N2CC(CNC(=O)C3=CCN(C)C3)CC2C)=O)cc(Cl)c1O 18126,C1(N(C(c2cc(C)c(O)nc2)=O)C)CC2CCC(C1)N2C(C1(C)CCOC1C)=O 18127,CCCCCC(CC)C(=O)N1CCC(CNC(=O)CCC2CC2)(COC)CC1 18128,N1(C(CCc2cncc(C)c2)=O)CC2CN(C(c3ccc(C)nn3)=O)CCC12 18129,C(=O)(CC(O)c1ccccc1)N(CCC(C)NC(=O)Cc1cccnc1)C 18130,c1(CN2CC3C(C(=O)NCc4ccc(F)cn4)C3C2)cccc(O)c1F 18131,C1(C(N2CC(CNC(c3c(C)ccc(Cl)c3)=O)C2)=O)CCC(=O)CC1(C)C 18132,N1(C(C2C(C)OCC2)=O)CCC(NC(=O)CSc2cnn(C)c2)C12CCC2 18133,c1(C(N2CCC(C(C)NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)cc2c(cc1O)CCCC2 18134,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncnn3C)=O)C(O)C2)cn1 18135,Cc1cc(C(C)C(=O)N(C2CCCN(C(c3cc(C)c(C)s3)=O)C2)C)cc(F)c1 18136,C(=O)(C(C)P(C)(C)=O)N(CCOC)CCNC(=O)Cc1c[nH]ccc1=O 18137,CC1CCN(C(=O)CSc2cccc[n+]2[O-])CC1CNC(c1cn[nH]c1)=O 18138,C(CCC(C)(C)C(=O)O)N(CC(C1CCSCC1)(C)O)C 18139,N1(C(c2cccc(N)c2O)=O)CCC(CNC(=O)C(F)CC2CCC2)C(F)(F)C1 18140,Cc1ncc(C(N2CCC23CN(C(c2cn4ccnc4s2)=O)C3)=O)c(C)n1 18141,C1(NC(=O)COCCCN(C)C)CCCCC12CC2.Cc1nc2oc1C(=O)NC2 18142,N1(C(C(F)OC)=O)CCOC2CCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC12 18143,c1(C(=O)NCC(C)(CNC(c2cc(C(N)=O)co2)=O)OC)csc(C)c1C 18144,c1(C(=O)NCCNC(=O)Cc2cccc3ccoc23)cc(F)c(O)c(Cl)c1 18145,c1(CN2CC(C(N(C(C=O)C)C3CC3)=O)C2)cc(CO)ccc1OC.CN 18146,c1(OC(C)C)ccccc1NC(=O)NCC1CCCC(C(F)F)C1 18147,n1(C2(C)CC2)cc(C(N2CC(NC(c3cc(C(N)=O)c[nH]3)=O)C2)=O)nn1 18148,C1(O)(CC)CCCN(C(c2ccc(CNC(=O)CC3(C#N)CCC3)o2)=O)C1 18149,C1(CC(=O)NC(CC)CN(C(C2(CC(F)(F)F)CC2)=O)CC)CCN(C)CC1 18150,C1(NC(Cc2cc(=N)[nH]cc2)=O)COC2(CCN(C(=O)CSC3CCC3)CC2)C1 18151,Cc1ccc(C(=O)NC2CC3CN(C(C4CC4(C)C)=O)CC23)c(C2CC2)n1 18152,C(=O)(CCCCCC#N)N1C(C(N2CCC3C(C(N)=O)C3C2)=O)CC(C)(C)C1 18153,c1(C(N(C)CC2(O)CN(C(c3c(C)ccnc3)=O)C2)=O)cc(C)c(C)cc1Cl 18154,c1(C(=O)NC2C(NC(C(C)OC)=O)CC2)ccc2ncsc2c1 18155,N1(C(COc2c(CC)cccc2)=O)CCN(C(C2CCCCO2)=O)C(C2CC2)C1 18156,c1(C(N(CC(C)N(C(C2(CC)COC2)=O)C)C)=O)cccc(P(C)(C)=O)c1 18157,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18158,c1(C(=O)NCCSCC(=O)NCC2C(C)(CO)C2)cc2ccncc2s1 18159,N1(C(C(c2cn(C)nc2)OC)=O)CCN(C(=O)CCc2ncccn2)CC12CCC2 18160,N1(C(C(C2CCCCCC2)C)=O)CCC(C2(NC(C3CC4CCC4C3)=O)CC2)C1 18161,c1(CN2C(CNc3ccncn3)CCC2)ccc2ncsc2c1 18162,N1(C(CCc2ccnc(C)n2)=O)CC2(CC2C(=O)Nc2ccc(OC(F)F)nc2)C1 18163,C1(C(N2C(C(=O)OCC)CCC2)=O)CN(Cc2csc(Cl)n2)CCO1 18164,N12CC(CC1=O)C(=O)N(C)CCNC1CC2C1.c1(C(CC)CC)nnnn1CC 18165,c1(C(=O)NC(C2CCCN(C(=O)C(CC)(CC)OC)C2)CC)cncc(F)c1C 18166,c1(-c2nc(CC(C)OC)nn2C2CCS(=O)(=O)C2)cc(Cl)ncc1F 18167,N1(C(C2OCCN(C(C(C)(CO)NC(C)=O)=O)C2)=O)CCCC(C)(C#N)C1 18168,S(=O)(=O)(c1cccc(Br)c1)N1CC2(CCN(C(c3n(C)ncn3)=O)C2)C1 18169,c1(OC)cc(C(=O)NC(C(=O)NCC(CC2CC2)CO)C2CCOC2)cc(F)c1 18170,CCC(O)C(C)(C)C(=O)NOCC(=O)NOCC(N)=O.C(C)(C)(C)OC(C)=O 18171,C(=O)(C(C)C(=O)NCCCCNC(C1CCCCC1n1cccn1)=O)OC 18172,N1(C(=O)Cc2cnc[nH]2)CC2CN(C(c3ccc(F)cc3F)=O)CCC2(CO)C1 18173,c1(C(N2CC(C)N(C(C3CC4CC3C3CC43)=O)CC2)=O)ccn2ncccc12 18174,CCC(C)(C)C(O)C(=O)NC(C(=O)N(C)Cc1ccoc1C)c1ccco1 18175,c1(CC)nocc1NC(=O)C(C)N(C(=O)CC#N)CC 18176,C(=O)(C(CCCC)NC(=O)C=CCN1CCC1)N(c1cccnc1)CC#C 18177,C1(O)(CC(N2CCC(C(C)O)C2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1 18178,C1(CNC(N(C(C)C(=O)O)C)=O)CCC(c2ccccc2)CC1 18179,Cc1nn(C)c(Cl)c1C=CC(N1CC(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 18180,N1(C(c2ccc(C#C)c(C)c2)=O)CC2CCCN(C(=O)CN3CCSCC3)C2C1 18181,c1(OC)cccc(SCC(=O)NCCC2CCCN2C(C2CC(Cl)(Cl)C2)=O)c1 18182,C1(CN(C)C)CCCC(NC(=O)CCCNC(=O)CC2CC=CC2)C1 18183,CC(CCNC(c1nc[nH]c1C(C)(C)C)=O)CCNC(=O)COC1CCOC1 18184,c1(-n2cnc(NC(C(=O)NCc3c(COC)noc3)=O)n2)ccccc1F 18185,c1(C(=O)NCC(CO)NC(C2(COC)CCOC2)=O)ccc2nc(C)sc2c1 18186,C1(CC(=O)NCCCCNC(C2CC(CC(=O)OC)C2)=O)CCCC(=O)N1 18187,C1(NC(c2n(CC)ncn2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 18188,c1(C(N2CC(CCC)N(C(C3CCCC3C)=O)CC2)=O)ccc2nnn(C)c2c1 18189,CC(C)CC(Cc1ccn(C(C)C(=O)N(C2CCC(C)(C)C2)C)n1)C(=O)OC 18190,N#Cc1cc(F)cc(SCC23CCC(CC2)C3)c1N 18191,CC1C(C)N(C(=O)C=CCN(C)C)CCN1C(=O)C=Cc1ccccc1 18192,c1(C(N2CCCC(CN(C(C(C=C)(C)C)=O)CC3CC3)C2)=O)c(F)ccc(F)c1N 18193,N1(C(C2N(C)CCC2)=O)CCC(C2CC2)C1C(=O)NCC(Cl)=CCl 18194,C(=O)(CC(O)CC(C)C)N1CC(=C(CNC(c2nc(OCC)c(C)s2)=O)F)C1 18195,N1(C(c2cc(OC)no2)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C2(CCC2)C1 18196,c1(C(=O)NC2CC(C)(NC(=O)CC3CC34CC4)C2)csc2c1CCCC2 18197,Cc1nc(NCCC2CCC(C)(C)CC2)cc(=NCc2nc(Br)cs2)[nH]1 18198,c1(NC(C)=O)nc(C)ccc1C(=O)NC1CCCN(C(=O)C(F)C(C)C)C1C1CC1 18199,C(CCC(C)(C)C(=O)NCC(C(=O)OC)OC)NC(c1ncc(CC)cn1)=O 18200,c1(NC(N2C(CC)CN(CC(C)C)CC2)=O)cnc2c(S)nc(O)n2c1 18201,C(C1CN2CC1C2=O)=CC.C12(CNC(=O)C3=NNC(=O)C3)CCCC1CCC2 18202,N1(C(Cc2c(C)occ2)=O)CC(C)(C)CC1CNC(c1nn(C(C)C)cc1Cl)=O 18203,N1(C(C2CC(C)C2)=O)CC(C)(C)OCC1CNC(C1(C(F)F)CCCC1)=O 18204,C1(C)(CC)CCCN1C(=O)C=CCC(C)(C)NC(c1ncccc1N)=O 18205,CC1CN(C(=O)COCCF)CC1NC(=O)CCc1cn(C)nn1 18206,CC(CO)C(C)N=c1[nH]c2c(c(=NCCn3cnnc3C3(CC#N)CC3)[nH]1)COC2 18207,C1(CS(C)(=O)=O)CCCN1C(=O)NCC(=O)C1CC1 18208,C(=O)(CC(COC)CC(C)C)NCC1N(C(C(CCC)CC2CCCCC2)=O)CC1 18209,c1(CC(=O)NCC(C)NC(c2c(CC)nn[nH]2)=O)cc(F)ccc1OC 18210,C(=O)(C#CC1CCCC1)N(CCCNC(c1c(C)cnn1C(C)C)=O)CCO 18211,CC1(CNC(c2cc(O)ccc2OC(F)F)=O)CCC(=O)NC1.OC(F)F 18212,N1(CC)CCCC(C(=O)NC2C=CC(C(N3CC(c4cn(C)cn4)C3)=O)C2)C1 18213,N1(C(C(CSC)O)=O)CCOC(C(C)NC(=O)CCc2cc(C)co2)C1 18214,C(=O)(CS(=O)(=O)CCO)NCC1(O)CN(C(c2cnc(C)[nH]2)=O)C1 18215,CC(C)(O)C(=O)NCC=CCNC(=O)CCn1cccc1 18216,CCC(C(=O)N1CC2CC2(CNC(C2CN(C3CCC3)C2)=O)C1)C(F)(F)F 18217,CC(CCN(C(=O)CC1CCCO1)C)NC(=O)C=C1CCC1 18218,CCC(CC)(CO)C(=O)N1CCC(O)C(N(C(=O)C=CC2CCC2)C)C1 18219,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC2(C)CC=CCC2)C(C=CC)C1 18220,N1(CCNC(CC(C=C)C)=O)CCN(C(=O)CC2CCC(C)(C)C2)CC12CCC2 18221,Cc1nn2ncccc2c1C(=O)NCC1CCCCN1C(c1ccncc1Cl)=O 18222,CC(C)(C)CC(C)(C)C(=O)NC1C2CC3C1C3C2C(=O)NCCc1ncon1 18223,CN1CCCC(C)(C(N2CCC(C(=O)NC3(c4ncccn4)CC3)C2)=O)C1 18224,c1(C2C(CNC(=O)NC3CN(C(C)=O)C4C3C4)C2)ccc(F)c(F)c1 18225,c1(C(=O)NC2(CN3CCCCC3C)CN(C(CNC(C)=O)=O)C2)ccccc1C#N 18226,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18227,C=CCC(C)(C)CC(=O)OCC1CC(C(=O)NCc2cc(Br)ccc2CC)C1 18228,c1(C(N(CCNC(=O)C(C2(O)CCCCC2)(F)F)CC)=O)cnc2nccn2c1 18229,N1(C(C(C)NC(=O)C2CC2)=O)CCN(C(C)CNC(C2CCCSS2)=O)CC1 18230,C(CCN=C(NC1CCc2ccccc2C1)N1CCC=C(C)C1)SC 18231,c1(C(=O)NC(C(C)(C)C)CNC(C2CC2C#N)=O)cc(=O)c2ccc(Cl)cc2o1 18232,c1(SC)c(NC(=O)Cn2ccnc2C(N2CC(F)CC2CO)=O)cccc1F 18233,c1(-c2cccc(SCC)c2)cnc(N=c2nc(O)c(NCC3(CO)CC3)c[nH]2)c(O)c1 18234,c1(CC(=O)NCC(C)N(C)C(c2snc(O)c2Cl)=O)ccc(C2CC2)cc1 18235,C1(NC(CN2C(C)CC2)=O)CCCC1(C)CNC(=O)CCCF 18236,n1(CC)ccc(C(=O)NC(CNC(=O)C(C)n2cnnn2)CO)n1 18237,C1(CNC(c2cscn2)=O)CN(C(C2C3CCC2CC3)=O)C2(CCOCC2)C1 18238,c1(OC)cccc2cc(C(=O)NCCN(C(c3ccc(C#N)o3)=O)C(C)C)oc12 18239,c1(C(N2CCCC2=O)=O)cc2n(n1)CCC2.c1(C2(C)CC2)nccc(O)n1.C(CO)N 18240,CCCCCC(C)CC(=O)N(C(C(=O)NCC1(CN=[N+]=[N-])CC1)C(C)CC)C 18241,C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCCN(C(CCN(CC)CC)=O)C1 18242,Cc1cc(CC(=O)NC(CNC(=O)CC2CC2(Cl)Cl)C(C)C)ccc1F 18243,c1(Cn2c(C(C3CC=CC3)NC3(CC)CC3)nnn2)cccc(SC(F)(F)F)c1 18244,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CN(C(=O)CC1CC1)C 18245,CC1CN(C(C2CC(Cl)C2)=O)CCC1NC(=O)Cc1ccc[nH]1 18246,CC1CCCN(C(=NCCS(=O)(=O)N(C)C)NCC2CCCCO2)C1 18247,N1(C(COc2c(OCC)cccc2)=O)CCC(C)(C(=O)N(C)CCN(C)C)C1 18248,c1(C(=O)NC2CC2NC(c2cc(F)ccc2F)=O)ccc2[nH]ccc(=O)c2c1 18249,c1(C(N2CCC(CC(=O)Nc3c(C)c(I)ccc3)C2)=O)cccn2cncc12 18250,C(=O)(CCCCCN(C(=O)Cn1ncccc1=O)C)N(C(C)C)CCN(C)C 18251,Cc1cncc(CC(=O)NCCC2CC(C(=O)NC(C)CC3CC3)C2)c1 18252,Cn1ncc2c(N3CC4CCN(Cc5c[nH]c6ncccc56)CC4C3)ncnc12 18253,C1(NC(C2(C)CCCS2)=O)CCCCN(C(c2cnn[nH]2)=O)C1 18254,c1(-n2cc(NC(C)=O)nn2)ccccc1Oc1nccs1.C1CCOCCN1C 18255,C1(N(C(=O)CSC2CC(F)(F)C2)C)CCN(C(=O)CCn2ccnn2)C1 18256,N1(C(C2(NC(=O)CCC(=O)C3CC3)C(C)CCC2)=O)CC2(CC=CC2)C1 18257,Cc1cc(C(F)F)oc1C(=O)NCCCN(C(=O)C(c1ccccn1)C)C 18258,c1(C(N(CCN(C(CC(CC)OC)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 18259,c12cccc(c1)CNC(=O)O2.C1(O)(C(C)(C)CF)CN(C(=O)Cc2cccs2)C1 18260,C1(NC(c2ccc(S(N)(=O)=O)cc2)=O)CN(C(C2CCO2)=O)Cc2nccn2C1 18261,C=CCCC(CC)(c1nnnn1C1CC(OC)C1)NC1CCCN(c2cnccn2)C1 18262,c1(C2C(C)C2)ccc(CCC(=O)NC(C)CCNC(c2coc(Cl)c2)=O)o1 18263,C(CC(=O)NCc1ccc(Cl)cn1)(C(F)(F)F)NC(c1n(C)ccc1)=O 18264,c1(C(C(=O)N(CCN(CC)CC)CC)(C)C)cccc(C#N)c1.C12(CC1)C(=O)NC2 18265,c1(OC)c(F)c(C(N2CC3C(C(N4CCN5CCCC5C4)=O)C3C2)=O)cc(F)c1F 18266,c1(C(N2CC(C)C(NC(=O)CCOC3CCC3)C2)=O)cc(F)ccc1Br 18267,CC1CC(N(C)C)(NC(c2ccc(Cl)c(Cl)c2)c2ccc(F)cc2)CC(C)O1 18268,C(c1ccncc1C)=CC(=O)NCCc1c(CNC(CC=C(C)C)=O)nco1 18269,CC1(C)C2COC1(C(=O)NCC(C1CC1)NC(c1cc(Cl)c(Cl)[nH]1)=O)C2 18270,C1(C(=O)NCCC2CC(C(=O)Nc3cn(CC#C)nc3)C2)C2CCCC(=O)C12 18271,C12(CNC(=O)Cn3cccn3)CC(CO1)N(C(c1cnc(C3CCCCC3)s1)=O)C2 18272,c1(C(=O)NC(c2ccccc2)C(=O)N(C(C=C)C)C)cncc(C2CC2)c1 18273,c1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)cnn2cc(C#N)cnc12 18274,CC(C)(CNC(C1CC(O)CCN1C(C1CCCO1)=O)=O)CN=[N+]=[N-] 18275,c1(C(=O)NC2CC(F)CN(C(c3ccnn3CCF)=O)C2)cccc2sccc12 18276,CC(C)C(F)C(=O)NC1CCC(NC(=O)CCC2NC(=O)NC2=O)CC1 18277,c1(C(=O)NCC=CCNC(C(F)OC)=O)nc2ccccc2c(Cl)c1Br 18278,c1(-c2onc(C3N(C)CCNC3)n2)ccnc2[nH]ccc12 18279,c1(OCCOC(CNC(CCCC(=O)OCC)=O)(C)C)ccnc2c1CCO2 18280,C(=O)(C(C)(C)C(F)F)N1CCCC(C(N(CC(O)(C(F)(F)F)c2ncc[nH]2)C)=O)C1 18281,C1(NC(CCC2CC(C)C2)=O)CCCC1NC(c1ccc(Cl)s1)=O 18282,N(C1CC(C)(C)Oc2ccc(F)cc21)c1cc(C)c(C)cc1S(=O)(=O)N(C)C 18283,C1(C#N)(C(=O)NCC(C(=O)N2CC(N(CCOC)C)C2)N(C)C)CC1(C)C 18284,N1(C(=O)OC(C)(C)C)CCOC2(C1)CN(N1CCc3cc(O)c(Br)cc3C1)C2 18285,C1(NC(C(C)NC(=O)NC)=O)CC(C)N(C(=O)CCN2CCC(C)CC2)C1 18286,CP(C)(=O)c1cccc(C(=O)NCCCNC(C2CC3CCC3C2)=O)c1 18287,c1(OC)cc(CC(=O)Nc2ccc(CC(F)(F)F)cn2)ccc1F 18288,Cc1nc2nccc(C(N3CC(C)(NC(=O)CC4CC(F)(F)C4(F)F)C3)=O)n2n1 18289,C1(C(=O)NCC(C)N(C)C(c2c[nH]c3nccc-3c2)=O)CN2CCN1CC2C 18290,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NCCCCc2cnc[nH]2)C1 18291,c1(C(=O)NC(CCN(C(C=CCC)=O)C)C(C)(C)C)sc2cncn2c1C 18292,C=CC1(CC(=O)NC2(N3CCNC3=O)CC2)CN(C(=O)C(O)CCN(C)C)C1 18293,N1(C(C2C(C)(C(C)C)C2)=O)CCC2CCC(NC(C3CC(F)(CO)C3)=O)C1C2 18294,C1(O)(C(C)NC(C(=C(C)C2CC2)F)=O)CN(C(c2cn(C3CC3)cn2)=O)C1 18295,c1(C(=O)NC(CCNC(CC)=O)C)cc(C)cc2c1NCCC2C 18296,N1(C(C2C(C)CCN2C(c2ccc3n[nH]cc3c2)=O)=O)CCCCC(C)(F)C1 18297,N1(C(CC=C)=O)CC(CNC(=O)CC(O)CC)OC2(CCC2)C1 18298,c1(C(=O)OC)c(OC(N2CC(CO)C2)=O)cccc1OC.C12CCCC(C1)N2 18299,C1(C(N2CC(C(C)C)C2C(N)=O)=O)(CNC(C2CC(=O)C2)=O)CC12CCC2 18300,N#Cc1cnc(F)c(-c2csc(NC(c3ccc(Cl)c(F)c3)=O)c2)c1 18301,CC(O)C(C)C(=O)N1CCN(C(=O)C(CN(C)C)Nc2ccccc2)CC1 18302,C(c1cncc(OC)c1)=CC(=O)NCC1C(NC(C2CC(C)(CC)C2)=O)CC1 18303,N1(C(C(C(C)(C)C)SCC)=O)C(C)CC2CN(C(C3CCC3)=O)CC12 18304,n1(CC)cnc2nc(N3CCCC(OCCO)C3)nc(NCCc3ncc[nH]3)c12 18305,c1(C(N(CCNC(C(C)CC2CC2)=O)C)=O)cc2ncccc2[nH]1 18306,C(C(C)(C)C(=O)N1CCN(C(=O)CC2CCN2C(=O)OC(C)(C)C)CC1)SCC 18307,c1(C(=O)NCCNC(C2COCCN2CC(F)F)=O)cc(Cl)ccc1Cl 18308,c1(C(N2CC(NC(CN(c3ccccc3)C)=O)C3C2C3)=O)cc2occc2s1 18309,C12(C(=O)NC3C(NC(c4cncc(Cl)c4Cl)=O)CCC3)CCCN(CCC1)C2 18310,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2c(Br)cccc12 18311,C1(COC)C(C)CCN1C(=O)C=CCC(C)(C)NC(=O)CNC(C)=O 18312,c1(NCC23C(CN(C(c4ccc(C)s4)=O)C2)CCC3)nc(Cl)nc2ncn(C)c12 18313,c1(N2CCCC(C(=O)NC3(CCOC)CCOCC3)C2)ncc2c(ncn2C)n1 18314,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18315,C(=O)(CCCCCCc1ccccc1)N1CCC(NC(C(C=C)(C)CC)=O)C1 18316,c1(C(C)=O)cccc(C(=O)NC(C2(Br)CC2(F)F)=O)n1.C12(CC1)CCN2 18317,C(c1nc2ccccc2o1)=CC(=O)NC1(CO)CN(C(CC(CCC)O)=O)C1 18318,CCC(CCCC(=O)N1CCCOCC1C)NC(C1CC(C)CCO1)=O 18319,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18320,N(C1CCc2cc(Br)ccc21)c1n(CCn2ncc(C(F)(F)F)c2)nnn1 18321,N1(C(=O)OC(C)(C)C)CC1(C)C(=O)NC(=O)CNC(C)=O.C1(C)CN1CC 18322,c1(CCNC(C2(C3N(C(CNC(=O)NC)=O)CCC3)CC2)=O)cnccc1C 18323,c1(C(N2CCCCCC2)C(=O)NC(c2ccccc2Br)COCC)nc(C)sc1C 18324,N1(C(C(C)OCC2CC2)=O)CCCC(C)(CNC(c2ncccc2F)=O)C1 18325,Cc1coc(=O)n1CC(=O)NC1CCC(N(C(=O)Cn2cnnn2)C)C1 18326,C(c1ccc(Cl)cc1)=CCN1CCC(c2onc(C)n2)C1 18327,Cc1nccn1CCC(=O)NC1CC(NC(c2ncoc2-c2ccco2)=O)C1 18328,c1(NC(C(C)(C)ONC(C2(C)N(C(CC(CC)C)=O)CCC2)=O)=O)cc(C)cc(O)c1 18329,CON1CC(c2nc(-c3cncc(F)c3)nn2C2CCCC2)CC1=O 18330,C1(NC(C=CC(C)C)=O)CCCC(CN(C(c2cc(C(F)(F)F)c[nH]2)=O)C(C)C)C1 18331,C(=O)(C(CC1CCCO1)C(F)(F)F)N(C)CC1(NC(CCCCC=C)=O)CC1 18332,Cc1cc(NC(c2c(C)noc2C)c2nnnn2CC2CC2)cnn1.C 18333,CCC(C)CC(C)C(=O)NCCCOCCN(C(=O)CSc1ccc(C)nc1)C 18334,C(=O)(CCCCSC)NCCN(C(=O)Cc1cc(C)sc1C)CCC 18335,N1(C(C=Cc2n(CC)ccn2)=O)CCCCC12CC(NC(=O)CCC1CC1C)C2 18336,N1(C(c2c(=O)ccn(C)c2)=O)CCN(C(c2cncs2)=O)CC12CCC2 18337,C1(NC(c2c(C)nn(C)c2)=O)CCCCC12CCN(C(=O)COC1CCOC1)C2 18338,C=C(CNC(=O)CCCc1cnccn1)CCNC(C1CCC(C(F)(F)F)O1)=O 18339,C1(NC(c2nn(C)nc2C(F)(F)F)=O)CN(C(C2(C)CC3(CC3)C2)=O)CC1(C)C 18340,C(=O)(CC(C)C(F)(F)F)N1CCCC(F)(C(N(CCCC(=O)NC)C)=O)C1 18341,N(C1CCCc2c(F)cccc21)C(C(C1(C=C)CCOCC1)N(C)C)=O 18342,C#CC1CN(C(C2CN(C(c3ns[nH]c3=O)=O)CC2(C)C)=O)CCN1C 18343,C1(CNC(CCN(CCC)C)=O)CC(NC(=O)Cc2ccc(Cl)cn2)C12CCC2 18344,c1(C(=O)NCC(CC=C)NC(=O)C(c2cnn(C)c2)O)nc(Cl)sc1C(C)C 18345,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)cn2C)=O)C12CC2 18346,c1(C(N(C2CC(NC(=O)CCc3cccs3)C2)C)=O)ccoc1I 18347,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2CC(F)(CO)C2)=O)CC12CCC2 18348,N1(C(C(c2cc(OC)ncc2)O)=O)C2CCC1CN(C(=O)Cc1ccnn1C)C2 18349,c1(NCC)nccc(=NCCOCCN(C(=O)CCc2cc(C)cc(C)c2)C)[nH]1 18350,CC(C)C(C(=O)N(C)CC1CN(C(c2cccn2C)=O)CCO1)c1ccccc1 18351,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1)=O)C2 18352,C1(CNC(C2CCC2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC2C1 18353,n1(C(=O)O)nc(CN2CC3(C(F)(F)F)CCC2CC3)c2c1CCOC2 18354,C1(C(N)=O)CN(C(C2(n3cc(-c4cncnc4)nn3)CC2)=O)C2CCCCC12 18355,C=CC(CCC)CC(=O)NC(CNC(c1cc2c[nH]nc2s1)=O)C1CCC1 18356,Cc1nn(C)cc1C(C)NC(c1conc1C(C)NC(=O)CC1C=CCC1)=O 18357,c1(C(N2CC(CNC(c3ccc(Cl)cc3)=O)C3C2C3)=O)ccc2ccnn2c1 18358,c1(CCC(=O)NCC2CC(NC(C(CC)SC)=O)C2)ccc2c(n1)NCCC2 18359,c1(C(N(CC(C)NC(=O)CCn2ncnn2)C)=O)ccc(CN(C)C)[nH]1 18360,C(=O)(C1=CC2CCC1C2)NCC1(CC(=O)NCCc2ccc(CO)cc2)CCC1 18361,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18362,C(CCC(C(=O)NCC1(O)CCSC1)NC(=O)CC(C)C)OC 18363,N1(c2nnc(CC)s2)CCC(NC(=O)CNC(c2cscn2)=O)C(C)C1 18364,N1(C(c2c(CC)onc2)=O)CC(NC(C2COC2)=O)C2CCCC12 18365,N(C1CCc2ccccc21)C(=O)CCNC(C1CCCCC1F)=O 18366,c1(C(=O)NC2(c3ccc(OC(C)=O)cc3)CCOCC2)cnc(F)cc1C 18367,C(CCN=C(NCC(c1cnccc1C)O)NCC(C)CC)OCC 18368,C#Cc1ccc(C(N2CCCC2C(C)NC(=O)C(O)CN(C)C)=O)c(OC)c1 18369,C(=O)(CCC(F)(F)C(F)(F)F)NC(CNC(CCCCCC#N)=O)CO 18370,N1CCCC2CCN(C(=O)CC3CC3)CC12.Cn1cnc(N)c(Br)c1=O 18371,Cc1cnc(C)c(C(=O)NCCCN(C)C(c2n[nH]cc2C2CCC2)=O)c1 18372,c1(C(N(CC(C)(C)NC(=O)CCC2CCCO2)C)=O)ccc(C#N)c(Cl)c1 18373,C1(C(=O)NC(CCCNC(c2cc(C(C)C)on2)=O)(C)C)CC2(C1)CC(C#N)C2 18374,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18375,C(=O)(N(c1cccc(Cl)c1CC)CC)N(CC(=O)OC)CCC 18376,N1(C(CC2CC(OCC)C2)=O)CC(CNC(c2c(C)coc2COC)=O)C(C)C1 18377,C(C1CCCCCC1)=CC(=O)NC1CN(C(c2ccc(NC)nc2)=O)C(CO)C1 18378,C1(CC(C)C)CCN(C(=O)C(=O)NCC2CCN2C)C(C(=O)NO)C1 18379,c1(OC)[nH]c(=NCCC2CC=CCC2)nc2c1ncn2C.C(C1CN1)OC 18380,N1(CCC(C(=O)OC)OC)CCN(c2ccc(F)cc2Cl)CC1C 18381,C(=O)(C(C)C1=CCCC1)NC(CCCNC(CSCCC)=O)c1ccccc1 18382,C1(C(=O)OC)CCC(C(=O)NCc2cn(C(C)C(=O)N3CC(C(O)CO)C3)nn2)S1 18383,c1(C(C2(C(=O)O)CC2)NC(CCc2ccn(C)c2)=O)ccccc1Br.C1(C)CCCO1 18384,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1nnc(C)s1 18385,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CO)Oc2ccccc2)CC1 18386,c1(OCC)ccc2c(c1)OCCO2.N1(C(C2CC(NC)C2)=O)CCCC(C=O)C1 18387,N1(C(C2C(CCC)C2)=O)CCOC2CN(C(c3ccc(C(C)F)cc3)=O)CC12 18388,N1(C(c2c(C)ccnc2)=O)CCN(C(=O)C(C)CC(F)F)C(CCO)C1 18389,N1(C(C2(SC)CN(C(=O)Cc3cc(C)cs3)C2)=O)CCC2CCN(C)CC12 18390,c1(C(C(=O)N(CCOC)CCC(C)C)N2CCCC2)ccc(F)cc1C 18391,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18392,CC1(C)CCN(C(=O)CCC(F)F)CC1CNC(=O)CN1CCC(C(F)(F)F)CC1 18393,CC1CCCN(C(=O)CC(F)(F)c2ccccc2)C1CNC(=O)CC1(O)CCOC1 18394,S(=O)(=O)(c1c[nH]ccc1=NCc1cccs1)N(C1C(C(=C)C)OCC1)CCCOC 18395,N1(C(C2N(Cc3cc(OC)cc(F)c3)CCNC2)=O)Cc2ccc(O)cc2C1 18396,c1(OC)ccc(F)cc1C(=O)NCCC(C)(C)NC(C1CC12CC(C)(C)C2)=O 18397,C1(C(N2CCC(c3cnn[nH]3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18398,C#Cc1ccnc(C(=O)N(CCCOCCNC(=O)C(C(C)CC)OC)C)c1 18399,C(CC(=O)N1CCN(C)CC1C)(C(F)(F)F)NC(CC(OCC)OCC)=O 18400,C1(NC(c2ccon2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18401,C1(n2cc(-c3c(NC(N4CC5C(CF)C5C4)=O)ocn3)nn2)CCCCNC1=O 18402,c1(OC)cc(C(N2CC(O)(CNC(=O)CC3CCC(C)C3)C2)=O)cc(N)c1O 18403,C(=O)(N=c1[nH]nc(Cl)cc1O)c1c(C)nc(CCN=[N+]=[N-])s1 18404,N1(C(C2C(NC(C3CC(OC)C3)=O)CC=CC2)=O)CCOC(C)C1C 18405,C1(N(C(C2(C(C)C)CCC2)=O)C)CCC2CN(C(c3ncccn3)=O)CC12 18406,S(=O)(=O)(c1ccc(S(=O)(=O)NC(=O)CCCCO)cc1)N1CC(C#N)C(CO)C1 18407,C1(NC(C=C(C)I)=O)CCN(C(=O)C=C(C)C(F)F)C(C)C1 18408,C(C(C(=O)N(CCC1CC1)N(C)C)NC(c1cnsc1)=O)OCC 18409,c1(C(N2CC(C=C)C(NC(C3CCCCO3)=O)C2)=O)cc(Cl)cc2ccccc12 18410,Cc1cc2c(cc(C(N3CC4CCN(C(=O)CS(C)(=O)=O)C4C3)=O)n2CCO)s1 18411,C1(C(N(CCC#C)CC)=O)CCN(C(=O)CNC(=O)CC)CC1(C)C 18412,C12(NC(C3CN(C(=O)CCCC4CCC4)CC34CC4)=O)CCC(C1)C(O)C2O 18413,c1(C(=O)NC2CC(F)(CNC(Cc3n(C)ccn3)=O)C2)cc2cccc(F)c2o1 18414,CCC(O)C(C)C(=O)NC1CC2CN(C(c3ccc(NC(=O)NC)cc3)=O)CC12 18415,N1(C(C(C=C)OC)=O)CCC(C2(O)CCN(C(c3nn(CC)nc3C)=O)C2)CC1 18416,c1(CC)cc(C(N2CCC2CNC(=O)C2CC2)=O)nn1CCO 18417,C(=O)(CCC(C)(C)C#N)N1C(C(C(N2CC(CC)(CC)C2)=O)(C)C)CCC1 18418,C1(NC(CC2(OC)CCOCC2)=O)(CNC(=O)C(C)C(F)F)CCOCC1 18419,C1(OC)CC(NC(=O)Cc2cnccc2Cl)CN(C(c2sc(F)cc2C)=O)C1 18420,c1(CC(=O)NC(C)CCNC(c2c[nH]c(Br)c2)=O)cccc2ncccc12 18421,Cc1cccc(C(=O)NC2CC2c2ccco2)c1N.C12CCN(C1)C(=O)CC2 18422,Cc1ncn(C)c1NC(=O)NCCn1ccc(C(=O)O)c1 18423,c1(C(N2CC(CNC(C(C(C)OC)O)=O)C2)=O)cc2occc2[nH]1 18424,C1(NC(Cc2c(C)cco2)=O)CCCCCN(C(c2ccc3cncn3c2)=O)C1 18425,N1(C(C(C)O)=O)CCCCCCC1C(N1CC2CCOC2C1)=O 18426,CC(C(=O)NCC1(O)CN(C(=O)C(C)Sc2nnnn2C2CC2)C1)C(C)(F)F 18427,Cc1oc(S(C)(=O)=O)cc1C(=O)NCC1CC(O)CN1C(=O)CCOCC(F)F 18428,N1(C(C2(C)CCN(C)C2)=O)CCC(NC(c2ccc3ccsc3c2)=O)C(C)(C)C1 18429,N1(c2nnc(CC)o2)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)CC(C)O2 18430,c1(N2CCN(C(CN(C)Cc3ccc(F)cc3)=O)CC2)ncc([N+](=O)[O-])cc1F 18431,N1(C(C2=CC(C)(CC)C2)=O)CC2CCCC2(NC(c2ccn(C)c2)=O)C1 18432,N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(=O)Cn1cccc1)CCO2 18433,n1(CCC#C)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)(C)O)C3)C2)=O)nn1 18434,C1(NC(c2ccc(C)nn2)=O)CN(C(=O)CCC2CCCOC2)CCC12CCC2 18435,N1(C(C(C(C)C)n2cnnn2)=O)CC2(CCC2CNC(=O)C(=O)N(C)C)C1 18436,N1(C(CN(C2CCC2)C(C2CC(C)N(C)CC2)=O)=O)CCc2sccc2C1 18437,c1(C(=O)NCCCCN(C(C(C)OCOC)=O)C)cnn(CCN2CCCC2)c1 18438,C1(NC(c2ccn(C)n2)=O)CCCCC12CCN(C(c1cncc(F)n1)=O)C2 18439,C1(C(=O)NCC2(NC(CCNS(CC)(=O)=O)=O)CC2)CCCN1C 18440,Nc1ccc(C(=O)N(CCC(=O)NCCC(F)CN=[N+]=[N-])CCO)nc1F 18441,c1(C(=O)NC2C(C(N(C3CC(F)(F)C3)CC)=O)CC2)ccc(C2CC2)cc1 18442,c1(NC(=O)NCCNc2ccccn2)cnnc2ccccc12 18443,c1(N(C2CCN(Cc3ccco3)C2)C(C2C3CCC(=O)C32)=O)ccc2sncc2c1 18444,CONC(=O)C(C)(C)CCNC(=O)CC(C)C(=O)OC 18445,c1(C(=O)NCC2C(CNC(C(C)(C)CO)=O)C2)cc(C(F)(F)F)cc(F)c1 18446,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18447,C1(C(N(C)C)=O)CCCC(C(N2CCN(C(c3cccnc3CO)=O)CC2)=O)C1 18448,C(=O)(C1=CC(O)CCC1)N.c1(C(=O)NCC2C(CCC)C2)cc2c(o1)C2.CC 18449,CS(=O)C1CN(C(C2(NC(C3(NC(N)=O)CC3)=O)CC2)=O)C1 18450,c1(C(=O)NCC2CC(NC(=O)Cn3ccnn3)C(O)C2)coc2ccc(F)cc12 18451,C(C(C)(C)C(=O)N1CC(CC(=O)NCC2CCN(CCF)C2)C(C)C1)OC 18452,N1(C(C(C)OCOC)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18453,C1(C(=O)NCC2N(C(c3ccc(C#C)cn3)=O)CC=C2)CC2(CO1)CC(F)(F)C2 18454,c1(C(=O)OC)cc(C)c(CN2CCC(NC(=O)CNC(C)=O)CC2)cn1 18455,c1(Cn2cc(C(N3CCC(NC(c4c(C)occ4)=O)C3)=O)nn2)cn(C)nc1C 18456,c1(SC)cccc(C(=O)NCC2(CCNC(=O)C(=O)NC3CC3)CC2)c1 18457,CC1CC(C(=O)NC2CC(CN(C)C)C2)N1C(=O)C(O)c1ccsc1 18458,c1(C(=O)NCC(C(N2CC(C)(CC)C2)=O)C)n[nH]c2c1COC2 18459,C1(C(NNC(=O)C2CCN(C(=O)OC(C)(C)C)C2)=O)CCn2ccnc2C1 18460,N12CCN(CC1C)CC2=O.c1(OC)ccc(-c2cn(-c3ccccc3Br)nn2)nc1 18461,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18462,N1(C(C=CC)=O)CC(O)(Cc2nccs2)C1.C12(c3ccccc3)CC(C1)C(=O)N2 18463,N1(C(C(Cc2cc[nH]n2)NC(C2CC23CCC3)=O)=O)CCc2ncncc2C1 18464,c1(C(=O)NCC2CCN(C(c3cn(CC)nc3)=O)CC2O)cccc2c1CCN2 18465,c1(C(N2CCC(O)(CN(C(C(C)OCCC=C)=O)C)C2)=O)cnc2cc[nH]c2c1 18466,c1(CC(=O)NC2C(NC(C3(C#N)CCCC3)=O)COCC2)ccc2c(c1)CCO2 18467,N1(C(c2c(C)cc(C)s2)=O)CCC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 18468,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(N1CCC(CC(=O)Nc2nc(C)c(C)s2)C1)=O 18469,c1(COC)cc(C(=O)NC(c2ccccc2)C(=O)N(C2CCN(C)C2)C)n(C)n1 18470,C1(NC(CSC(C)C)=O)CN(C(c2cc(C3CC3)on2)=O)CC1C(F)F 18471,C(N=c1[nH]c2c(c(=NC3CC4(CC4)C3C(F)(F)F)[nH]1)CSC2)c1c(Cl)cccc1 18472,N1(C(C(C)=CC=C)=O)CCN(CC(N2CC(CO)(Cc3ccccc3)C2)=O)CC1 18473,c1(CC(=O)NC(CN(C(CN(C(=O)OC)C)=O)C)C)nn(C)c2ccccc12 18474,N1(c2ccc(C(=O)Nc3ccc(C)nc3Cl)cc2)CCN(C(N)=O)C(C)(C)C1 18475,N1(C(CC(=O)NCC2CC2)=O)CCN(C(=O)CCC2CCC(=O)NC2)CC1 18476,c1(N2CCN(Cc3c(C)c(Cl)ccc3)C(C)C2)ccnc(S(C)(=O)=O)n1 18477,C1(NC(C(=O)NC2CC2)=O)CC2CCC1CC2NC(c1cc(F)ccc1O)=O 18478,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cnc(S)n2C)=O)C1 18479,Cc1ccc(Br)c(N)c1C(N1CCCC(n2cc(-c3ccccn3)nn2)C1)=O 18480,CCC(C)C(C(=O)NCC1CC2(CC2)CO1)NC(=O)CCn1ccnc1C 18481,N1(C(CN(CCOC)C)=O)C2CCC1CC(CCNC(C1(C)CCC1)=O)C2 18482,Cc1cc(C(N2CCC(NC(C3CN(C(C)C)C3)=O)C2C)=O)n(C)n1 18483,CC1CC(CCNC(C2(F)CC2)=O)CCN1C(=O)CSCc1ccc(C#N)cc1 18484,c1(C(=O)N(CC(CC=C)NC(C2COCCO2)=O)CC)ccc2nccnc2n1 18485,C1(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)ccn2)=O)COC2(CCC2)C1 18486,CC1CCC(NC(c2cccc(CS(C)(=O)=O)c2)=O)CN1C(c1ccsn1)=O 18487,c1(CC)ccc(C)cc1C(N1CCCC1C(C)NC(c1[nH]nnc1C)=O)=O 18488,C1(C(=O)NCC2(C(=O)NCCN(C)CCF)CC(C)(C)C2)CC(=O)NC(=O)C1 18489,C1(NC(Cc2nnc(C)o2)=O)CN(C(=O)C(C)Cc2ccccc2)C2(CCC2)C1 18490,C1(N(C)C(c2ccc(CO)o2)=O)CCCN(C(c2ccc(SC(N)=O)cc2)=O)C1 18491,c1(C(=O)NC2C(NC(c3ccc(C4OCCO4)cc3)=O)COC2)ncc(F)cn1 18492,Cc1cc(C(=O)NCCCN(C(=O)CC2CCC2)Cc2cccs2)c(C)n1C1CC1 18493,c1(C2(CC3CN(C(=O)NC(c4nnnn4C)C)C3)CCC2)ccccc1F 18494,C1(C2N(C(C(=O)NC(c3ccc(C)cc3)C#C)=O)CCC2)CCC(F)(F)CC1 18495,c1(C(=O)N(C2CC(=O)NC2=O)CCC2C(=O)CCCC2)cc(F)ccc1F 18496,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18497,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2cnc(C)c(F)c2)=O)CC1CF 18498,C(=O)(CC(C)O)NCC(C)=CC(=O)N(C)Cc1nn[nH]n1 18499,c1(C(N(CC(=O)Nc2ccc(=O)n(C)c2)CCC)=O)c(C)nc(C)nc1C 18500,Cc1nccc(C(=O)NCC2(CNC(C3(C(C)C)CC3)=O)CC2)c1N 18501,c1(C(=O)NCC2C(NC(C(C)C#N)=O)CC2)c(F)ccc(F)c1Cl 18502,c1(CNC(=O)CCC2CCCN2C(=O)CC2CCC3CC23)cccnc1F 18503,N1(C(CC(C=C)(C)C)=O)CC2CN(C(c3cn(C4CCOC4)nc3C)=O)CC2C1 18504,c1(C(=O)NC(C)CC(C)Cc2cc(N3CCCC3)ncn2)cc(Cl)n(C)n1 18505,N1(C(C(C)Cc2ccnn2C)=O)CCOCC1CN(C)C(c1cn(C)nc1O)=O 18506,C1(CC(N2C(CCCNC(C(C)SC(F)(F)F)=O)CCC2)=O)SC(=N)NC1=O 18507,C(CCC(C(=O)NC(C)(C)C(C)(C)CO)NC(=O)C=CC(F)F)OC 18508,C1(NC(c2c(C)cco2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 18509,c1(C(C(=O)NC2C(CNC(c3cc(C)oc3)=O)COC2)(F)F)ccc(F)c(F)c1 18510,C(CC(F)(F)F)SCC(N1CC(C(C)NC(c2cn(C3CCOC3)nn2)=O)C1)=O 18511,c1(C(N(CCNC(C2(c3c(COC)nco3)CC2)=O)C2CC2)=O)cnn(C)c1F 18512,C1(NC(c2nn(C)c(Cl)c2)=O)CCCC12CCN(C(=O)CC1COCCO1)CC2 18513,C1(CNC(c2cc(CC)n[nH]2)=O)CCCCC1CNC(=O)Cc1cnc(CC)[nH]1 18514,C1(CNC(CCC2N(C)CCC2)=O)CC2CC2N1C(c1cc(C#N)on1)=O 18515,C(CC(=O)NCc1c(C)cccc1O)(C(F)(F)F)NC(C=CC=CC)=O 18516,N1(C(Cc2c(CC)con2)=O)CCC2CCCC12CNC(=O)C(C)S(N)(=O)=O 18517,c1(C(=O)NCCC2N(C(CCC=C(C)C)=O)CCC2)nc(O)sc1C 18518,C(=O)(C(CCF)NC(=O)CCNC(N)=O)NCC(CC)(C)O 18519,C1(C(=O)NC2C(NC(CNC(C=CC)=O)=O)COC2)CCCN(C(C)=O)C1 18520,NS(=O)(=O)c1sccc1C(=O)N(CCNC(C1COCCO1)=O)C1CC1 18521,c1(C(=O)NCC2C=CC(NC(CC(CCC)O)=O)C2)cc(F)cc2nc[nH]c12 18522,C1(C(N(C(C)COC)CC=C)=O)CSCCN1C(c1coc(CO)c1)=O 18523,c1(C(=O)OC)ccc2c(c1)N(C(=O)NC(c1ccccc1Br)C1CC1)CCO2 18524,c1(CC(c2n(CC)nnn2)NC(C(C)C)c2nc[nH]n2)ccc(SC)cc1 18525,c1(NCCC(=O)NC)cc(=NCc2cc(-c3cccc(F)n3)no2)[nH]cn1 18526,c1(C(=O)NCC(C(=O)NCCC(C=C)C)N(C)C)ccccc1C 18527,N1(C(Cc2cn(CC)nc2)=O)CCOC2(C1)CN(C(=O)CCN1CCCC1)C2 18528,C1(CNC(C(C=CC)O)=O)CN(C(=O)C=CCCC(C)C)CCO1 18529,c1(C(=O)NC2CCN(C(c3cn(CC=C)nn3)=O)C(C)C2)ccc(C)c(C)c1N 18530,CC1CCC(CNC(=O)OC(C)(C)C)N1C.c12cc(cs1)CNC1N(CC1)C2=O 18531,C1(C(=O)NC2CCC(NC(C(C)(C)OC(C)=O)=O)C2)CCC(C(F)(F)F)CC1 18532,c1(NC(C(CCF)NC(C(CSC)OC)=O)=O)cc(C)cnc1O 18533,N1(C(c2c(C)cno2)=O)CCCCC1C(C)NC(=O)Cn1cccnc1=O 18534,N1(C(CCCc2nc(C)sc2)=O)CC(C)N(C(c2nccnc2C)=O)CC1C 18535,Cn1c(C(=O)OCC(c2ccc(I)cc2)=O)ccc1C#N 18536,N1(C(c2c(OCF)cccc2Cl)=O)CC2CCC(C1)C2N1CCC(CO)C(O)C1 18537,c1(NCCc2nc(CC)[nH]n2)cc(NCc2cncc(Cl)c2)ncn1 18538,C1(NC(=O)CSC(F)F)CC(C(N2CCCC2c2nc(CO)no2)=O)C12CCC2 18539,c1(NC(C2(C)CCN2Cc2n[nH]c3ccc(Br)cc23)=O)cnc2ccc(F)cn12 18540,c1(C(OC(F)F)NC(c2n(CC=C)nnn2)c2ccn(C3CC3)n2)cccc(Br)c1 18541,N1(C(C(CC2CC2)NC(c2c(CC)cccn2)=O)=O)CC2(CC=CC2)C1 18542,N1(CCN(CCC)C(=O)NCC2CC2(F)Cl)CCCCS1(=O)=O 18543,N1(C(CC=CC=C)=O)CC2CCC(C1)N2C(c1scnc1-c1ccccc1)=O 18544,C(=O)(C(F)CC(C)(C)NC(=O)CCc1cncs1)NCc1n(C)cnn1 18545,C1(CNC(CN(C)NC(c2cc(Cl)cn2C)=O)=O)CCN(C(=O)C(C)(C)C)CC1 18546,C1(NC(C2CC(C#C)(O)C2)=O)CCN(C(c2cnnc(C)c2)=O)CC1F 18547,C(=O)(CCCC(=O)N1CCC(F)(CNC(=O)CNC(=O)CCCCO)C1)OC 18548,c1(C(=O)OCC)cc2c([nH]1)CCN(C(=O)C(N1CCCCC1=O)C)C2 18549,CC(O)C(F)(F)C(=O)N(CCNC(C1CC(O)CN1C(=O)OC)=O)CC1CC1 18550,C1(NC(C(CC)SC)=O)CCN(C(=O)C2CC2)CCC1Nc1ncccc1CC 18551,N12CC(CC(C)C1)NC2=O.c1(C(C2CCC2)OCC)ccc(C(F)(F)F)nc1 18552,C1(C(N2C(CNC(CCc3c(C)nn(C)c3C)=O)CC2)=O)Cc2cncn2C(=O)N1 18553,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18554,C1(CNC(Cc2ccn(C)c2)=O)COCCN1Cc1nnc(-c2ccco2)o1 18555,C1(CNC(c2ccc(C)[nH]2)=O)CN(C(C2CC(C)(C(C)(C)C)C2)=O)CCN1C 18556,Cc1ccccc1COC(=O)NCC(=O)NC(C)C(C)NC(c1ccccn1)=O 18557,C1(SC)CCN(C(=O)CCNC(=O)CC2(O)CCCCC2)CC1 18558,c1(C(N(CCNC(C=C(CCC)C)=O)C)=O)ccc(N)cc1CC 18559,c1(SO)cc(Br)cc2c1CCCN2C(=O)CC1(c2ccc(F)cn2)CC1 18560,c1(C(=O)NCc2nc(CNC(CCC#CC)=O)sc2)ccc(F)c(F)c1N 18561,CN1CC(NC(C2CC3C=CC2N(C(=O)CCOC2COC2)C3)=O)C2(CC2)C1 18562,CC1(C)OCCCC1C(=O)NCC1CN(Cc2ccc(F)cc2)CCCO1 18563,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18564,c1(C(C(=O)N(C2CN(C(=O)CC3CCCC(O)C3)C2)C)(C)C)cccc(C#N)c1 18565,C1(CC)CC(C2CCCCC2)=NO1.C12(CC1)CN2 18566,C12(CC(=O)N(C3CCCC3)CCNC(C(C)O)=O)CC3CC(C1)CC(O)(C3)C2 18567,c1(SCC)ccc(C(=O)NC(C)CCCNC(C2(COC)CCO2)=O)nc1 18568,CN1CC(C)(C(N2CC(C(=O)NCCN3CC4CC4C3)C(F)(F)C2)=O)CC1=O 18569,C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)Nc1ccc(C(C)O)cc1 18570,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18571,c1(CC)cccc(C)c1C(N1CCCC(O)(CCNC(=O)CC2CC2(Cl)Cl)C1)=O 18572,CC(CC(=O)NCC1(C(=O)NCC2CCCOC2)CC=CC1)n1ccnc1 18573,C1(NC(c2cn(-c3cnncc3)nn2)=O)CCCN(Cc2ccc(Cl)nc2)CC1 18574,c1(C(N2C(C(=O)NC(c3cn(C)nn3)C)CC2)=O)cc(C#N)c[nH]1 18575,c1(C(=O)NC2CC(NC(=O)Cc3cccc(Cl)c3)C2)ccc2c(c1)CC(=O)N2 18576,c1(CC)cc(C(=O)NC2CC3CC2N(C(=O)Cc2ccc(Cl)s2)C3)cn(C)c1=O 18577,c1(OC)cc(OC)cc(CC(=O)NCC2CCC2NC(C2C3COCC23)=O)c1 18578,Cc1cc(-c2ccnc(NC(c3ccccc3N(C)C(C)C)=O)n2)ccc1F 18579,N1(C(Cc2c(C)cccc2)=O)C2CCCC1CN(C(C1CCN(C)C1C)=O)C2 18580,n1(CC)cc(Cl)cc1C(N1CC(C(C)NC(c2ccc(C#N)[nH]2)=O)C1)=O 18581,N1(C(=O)CCc2nnc(-c3ccco3)o2)CC2(CCN(C(C34CSCC3C4)=O)C2)C1 18582,C1(C(=O)NC(c2c(C)n[nH]c2)C)CCN(C(c2cc(C(N)=O)co2)=O)CC1O 18583,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18584,c1(C(N(CC(C)N(C(=O)C=Cc2cccnc2)C)C)=O)ccc(=N)[nH]c1 18585,C(=O)(NNc1ccc(F)c(Br)c1)OC(C)(C)C.N12CCCC1NC(=O)N1CC2C1 18586,N1(CCNC(C(c2ccco2)OC)=O)CCC(CCNC(=O)CC2CC2)CC1 18587,C1(NC(C(C)=C(C)C)=O)CC2(CCN(C(=O)COC3CCOC3)C2)C1 18588,CCC(C)(CCNC(=O)CCCn1ccnc1)NC(=O)C(C)n1ccnc1 18589,c1(C(N(C(C)CNC(=O)CC(c2ccc(Cl)cc2)O)CC)=O)ncccc1Cl 18590,c1(OC)ccc(F)c(F)c1-c1cn(C(C)C(N2CCC(OC(C)C)C2)=O)nn1 18591,C1(CNC(C2CCS(=O)(=O)CC2)=O)CC2CCC(C1)N2C(C1CCOC1)=O 18592,C1(OC)CN(C)C(C)(C(N2CC(NC(c3cccc(SC)c3)=O)CC2(C)C)=O)C1 18593,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)C(C)SC(F)(F)F)CCCO1 18594,N1(C(COCC(=O)NC)=O)CC(=O)CC1C(=O)NCCc1ccncc1F 18595,Cc1cnccc1CCC(=O)N1CC(c2cn(CCN3CCC(F)(F)C3)nn2)C1 18596,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18597,c1(-c2nccc(C(N3C(C)CN(C)C(C)C3)=O)c2)cccc2c1OCCCO2 18598,c1(OC)ccnc(C(=O)NCC2CCC(CNC(=O)CCCN(C)C)CC2)c1N 18599,Clc1scnc1C(c1nc(C2CC2)cs1)NCc1nnnn1CC1CC1 18600,OC1COc2ccc(-c3ccc(C(=O)Nc4ncnc5[nH]cnc45)nn3)cc2C1 18601,C#CCC(C(=O)N1CCC(O)C1C)NC(=O)CSCCCC 18602,C(=O)(CCC(CC)NC(c1cc(C)c[nH]1)=O)NC(CCC)CC 18603,C#Cc1cccc(C(=O)Nc2cccc(NC(=O)C(CO)N(C)C)c2)c1 18604,C1(CNC(C2N(C)CC(O)C2)=O)CC2(CCC2)CN1C(=O)CC1C=CCC1 18605,Cc1ccnc(C(=O)NCC2(NC(=O)C=CS(C)=O)CCC2)n1 18606,C(C(F)(F)C(F)(F)F)OCC.N12CC(=O)N(C1=O)CCCCC2.C12CCN1CC2 18607,c1(CN(C(=O)CC2(N(C(=O)C=CC3CC3)C3CC3)CC2)C)nnnn1C 18608,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)CC1 18609,C=CCN=C(NCc1ccc(NC(C)=O)nc1)NCC1(C)CC1C(F)(F)F 18610,N1(C2CC(NC(CCOC)=O)C2)CCN(C(C2OCCOC2C)=O)CC1 18611,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCC(C)(C)C2)nc2c1SCC2 18612,C(=O)(C(C)(C)CC(=O)OC)N(CC(=C)CCOC)CC.C(=O)C1=CCCCC1 18613,n1(CC)cnc2c(NC3CCCC(C)C3)nc(N3CCC(CCOC)CC3)nc12 18614,c1(C(N2C(CNC(C(C)OC3COC3)=O)CC2)=O)ccc(C2CC2)cc1F 18615,CC#CC1CCN(C(C2CCN(C(=O)CC3CCC=CCC3)C2)=O)C1 18616,C#Cc1ccc(C(=O)NCC(C)(C)OCCNC(c2ccsc2CC)=O)cc1Cl 18617,c1(CC(=O)NC2C(CNC(C=CC(=O)OCC)=O)C2)ccc2ccoc2c1 18618,C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2cccc(C(C)C)c2)=O)C1 18619,CC(C)CC(C)CC(C)C(=O)NC1(CNC(=O)CN2C(=O)CNC2=O)CCCC1 18620,N1(C(CC2CC(NC(c3c(C)cc(F)s3)=O)C2)=O)CCOCC(C)C1 18621,c1(CC(=O)NC(CC2CCN(C(CCC#C)=O)CC2)(C)C)cccc(O)c1F 18622,Cc1ccc2oc(C(=O)NC3CC(CNC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18623,c1(C(=O)NC2(C(=O)NCc3cc(C)sc3C)CCCCC2C)cnc([N+](=O)[O-])n1C 18624,C(C(CNC(C1(CO)CC1)=O)C(F)(F)F)NC(C(C)(c1ccccc1)NC(C)=O)=O 18625,C(=O)(C#CC1(C)CCCO1)N(C(C)CNC(c1cnn(C)c1Cl)=O)C 18626,CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)CSC(F)(F)F)C2)C1 18627,C1(O)(CN(C)C(c2occc2CN(C)C)=O)CCN(C(=O)CCOC2CC2)C1 18628,N1(C(C2CN(C)CC(C)O2)=O)CC2(CCN(C(=O)CSC(F)F)CC2)C1C(C)C 18629,CC(C(=O)OCCC(C)(C)C)C(=O)N(C)CCN(C(=O)CCc1cncn1C)C 18630,N1(C(C(n2ccc(C3CC3)n2)C)=O)CCCC(C(N)=O)(NC(=O)CN(C)C2CC2)C1 18631,C1(C(N(C)CC2N(C(C(CSC)O)=O)CCC2)=O)CC2CCC1CC2 18632,N1(C(c2c(CN(C)C)ccs2)=O)CCCCC2(CCN(C(c3cnc[nH]3)=O)C2)C1 18633,N1(Cc2ccc(N(C)C)nc2)CCC(Nc2cnc(O)c(Cl)c2)C(C)(C)C1 18634,c1(C(CCC(=O)NCC2(OC)CN(C(CCCOC)=O)C2)=O)cc(F)ccc1F 18635,C1(CC)CNC(=O)CN1C(C1CCN(C(=O)CC2CC(OC(C)=O)C2)C1)=O 18636,C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ncccn1)=O)C(C)C)C2 18637,C1(N(C)CC2CCN(C(=O)CC=CBr)C2)Cc2nccn2C1 18638,C1(CNC(COCCC)=O)CC(NC(=O)C(C)n2ccnc2)C1 18639,N1(C(CCc2ncn(C)c2)=O)CC(NC(=O)CSc2nc[nH]n2)C2(CC2)C1 18640,O=C(C#CC1CCCC1)NCc1cc(N2CCCCC2)ncn1.C12(CC1)C(=O)N2 18641,C(=O)(C1=CCC(C)CC1)NCCCCC1CCN(C(c2nc(C)sc2)=O)CC1 18642,Nc1cccc(Cl)c1C(=O)NC1CC2CC1N(C(C1CCC3CC13)=O)C2 18643,C1(NC(C(CC)C)=O)CCC12CN(C(=O)CCC(C)(C)OC)C2 18644,N#Cc1ccsc1C(N1CCCC1CNC(c1cncc(C2CC2)c1)=O)=O 18645,N1(C(CCC2N(C)CCCC2)=O)C2CCC1CN(C(=O)C(O)CC(N)=O)C2 18646,Nc1c(C(N2CC3CC3(NC(=O)Cc3cnn(C(F)F)c3)C2)=O)ccnc1F 18647,CC1=CCC(C(=O)NCC2CC2NC(c2ccc(NC3CC3)nc2)=O)CC1 18648,c1(CNC(=O)CN(C2CCC2)C(C2CN(C3COC3)C2)=O)ccnnc1 18649,C(C(C)(C)C(=O)N1CCC(O)(C(C)C)C1)OC.n12cc(cn1)-c1cn(nn1)CC2 18650,C1(CNC(C(CC=C)NC(C)=O)=O)CN(C(c2c(Cl)n[nH]c2C)=O)CCN1C 18651,Cc1cc(C#N)ccc1C(N1CCC2(CC2NC(C2CC3(CCCC3)C2)=O)C1)=O 18652,CCCCCCCCC(C)CC(=O)N(c1ccc(OC)cc1)CCO 18653,C#CC1CCCC(NC(=O)C(CNC(C2CC(COC)C2)=O)N(C)C)C1 18654,C1(CC(=O)OC)CCC(C(=O)NC2(C)CN(C(=O)C(C(C)C)SC)C2)CC1 18655,C(=O)(C(C)CCCC(C)=O)N1CCCN(C(C2CN(CCC)C2)=O)C(C)C1 18656,N1(C(c2cc(OC)sc2C)=O)CCC(O)(Cn2cc(C3(C)CCOC3)nn2)CC1 18657,N#Cc1cc(C(=O)NCC23CC(CN2C(=O)Cc2cncnc2)C3)co1 18658,c1(OC)ncccc1C(C1CCC1)Nc1nnnn1C.C1(CC2CC2)CCC1 18659,c1(CCC(=O)NCC(C)NC(=O)CN2CSCCSC2)cccc(F)c1Cl 18660,N1(C(C(c2cccnc2)C)=O)CCC2CC(CNC(=O)CCF)CCC2C1 18661,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18662,C1(CC=C)(NC(COCCC=C)=O)CN(C(c2csc(Br)n2)=O)C1 18663,N1(C(c2cc(OC)ncc2F)=O)C2CCCC1CC(NC(C1CCC(C)O1)=O)C2 18664,c1(COC)cc2ncccn2n1.c1(C2C(=C)C2)nc2nn1-c1ccccc1C2 18665,N1(C(c2cnc(-c3cccc(C)c3)[nH]2)=O)CCCC(O)(c2cnn(C(C)C)c2)C1 18666,C12(C(=O)NC(CC)CNC(=O)COCC3CCOC3)CSC(C1)C2 18667,N#Cc1cnn(CC(=O)NC2CC3(C2)CN(C(C2(CO)CCC2)=O)C3)c1N 18668,CC1(C)CCCCC1NC(=O)NCC(C)(C)CN1CCCC1.c12cnn(c1)CC2 18669,N1(C(CCCNC(C)=O)=O)CC2(COC(CNC(=O)C(F)CC3CCC3)C2)C1 18670,S1(=O)(=O)c2ccc(c(C#N)c2)N2CC(C3(CC3)C2)N1.C(CN(C)C)SC 18671,c1(CN2C(C(N(CCC)CC)=O)CC(F)C2)ccc(C#N)cc1[N+](=O)[O-] 18672,C1(NC(C2(O)CCOC2)=O)CC2CC1N(C(=O)CSCc1cscn1)C2 18673,C12(CNC(c3c(C)ccnc3)=O)CC(C1)C(NC(=O)C(F)C(F)(F)F)CO2 18674,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)c1C 18675,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18676,c1(NC(C2CC(NC(C(CCC)C)=O)C2)=O)cc(C)ccc1CC 18677,C1(CC)COCCC1NC(=O)CC(=O)NCC(=O)NC(=O)CNC1CC1 18678,c1(C(=O)NCC(O)CNC(C2CC2C2CCC2)=O)ccc2ccc(Br)cc2c1 18679,c1(C(N2CCCC(N(C(CCCC(=C)C)=O)C)CC2)=O)ccc2n[nH]c(C)c2c1 18680,N1(C(CCN(c2ccc3cccnn23)C(C)C)=O)CCC2CCCC2C1 18681,c1(CNC(=O)NC2CCC(N(C)C)CC2)cc(C#N)ccn1 18682,C1(NC(C2(C(C)C)CCN(C(C(C=C)C)=O)C2)=O)CCN(C)C12CCC2 18683,c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2(C)C)ccc(C(N)=O)c(Cl)c1 18684,C1(C(N(CC#C)CC)=O)N(C(=O)Cc2conc2C)CC12CCCC2 18685,CCC(CC(=O)N(C1CN(C(C2CC=CCO2)=O)CCC1O)C)C(C)C 18686,C(CC(=O)NC1(C)CC(NC(=O)CC(=O)N(C)C(C)C)C1)(C(F)(F)F)OCC 18687,Cc1nnn(CC(=O)NCc2cn(CC(=O)N(CCCF)C)nn2)n1 18688,c1(CC)cc(C(=O)NC(c2ccnn2C)C(=O)NCC2(F)CCOCC2)ccn1 18689,C1(F)(C(=O)NCc2ccc(C(N=c3c(C)ncc[nH]3)=O)nc2)CCCCC1(F)F 18690,C1(CNC(C=NOC)=O)CC2(CCN(C(c3cc4n(n3)CCCN4)=O)CC2)CO1 18691,C(=O)(CCCS(C)(=O)=O)N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1 18692,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18693,CCC(CCCC(=O)NCc1cc(C)ccc1O)NC(C1CNC(=O)O1)=O 18694,c1(C(=O)O)cnc(NC2CC2)c(Cl)c1.c1(C23CC(C2)C(=O)N3)ccc(F)cc1 18695,N1(C(CCC2CC(OC)C2)=O)CCC(C)C1C(N1CC(Cc2ccco2)C1)=O 18696,Cc1cc(C(F)F)oc1C(=O)NC1CCC(C)(CNC(C2(C(N)=O)CCC2)=O)C1 18697,CCC(C)(C)C(=O)N1CCCC(CNCc2c(C(N3CCOCC3)=O)occ2)C1 18698,N1(N2CC(CC)C(C(C)C)C2)CCCC(O)(C(F)(F)F)C1.C=O 18699,N1(C(c2nsnc2O)=O)CCC(C(N2CCCC2C2CCOC2)=O)CC1 18700,c1(OC)nc(Cl)ccc1C(N1CC(C)CC1C(=O)Nc1cnc(C)[nH]1)=O 18701,Cc1cn2c(n1)C(C(=O)N1CCCC1(C)CNC(c1c[nH]ccc1=O)=O)CCC2 18702,c1(CCN(CC(C)C)C(=O)Nc2ccco2)c(F)cccc1F 18703,N1(C(C(C)NC(C2CC23CC3)=O)=O)CC2CCCC(O)C2C1 18704,O=C(C1=CCCOC1)NCCCCNC(C1CCCCS1)=O 18705,CC1CCC(C)(C(=O)NCCN(C)C(c2ccnc(OCCN(C)C)c2)=O)C1 18706,N1(CC#C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18707,c1(C(N(CCNC(CSCCN(C)C)=O)CCOC)=O)cc(CCP(C)(C)=O)[nH]n1 18708,Cc1cccc(C(=O)NCCCCCCNC(=O)CC2(C)CCCO2)c1N 18709,N1(C(c2n(C=C)ncc2)C(=O)NCc2ccccc2F)CCC2C(CCN2C)C1 18710,N#CC1(C(=O)NCC2(CCNC(C3CCCN3C=O)=O)CC2)CC2(CCC2)C1 18711,C1(C(=O)NC(C2CCN(C(C3COC(=O)O3)=O)CC2)C)CCSC(C)C1 18712,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2ccco2)C1 18713,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18714,C1(C(C)C)N(C(C2CC23CC3)=O)CC12CCN(C(c1nc(CO)sc1N)=O)CC2 18715,N1(C(c2ccccc2NC(=O)C(Cl)(Cl)Cl)=O)Cc2cccc(O)c2C1 18716,N1(C(c2cn(CC)nc2)=O)CC2(CC2)CC1CC(=O)N(C)Cc1cc(C)n(C)n1 18717,C1(NCC(c2scc(CNC(C3CCC(C(N)=O)C3)=O)c2)=O)CCCC1C1CC1 18718,c1(CC)ccc(C=CC(=O)N(C)CC2CCCN2C(c2cc(=O)cc[nH]2)=O)o1 18719,C(=O)(C1=CCOCC1)NC(C)CNC(c1ccc(OCc2ccco2)c(F)c1)=O 18720,C(=O)(CC(C(F)F)C(C)(C)C)NCC12CC(CNC(C(CCSC)O)=O)(OC1)C2 18721,Cc1cc(Cl)cc(C(N2CCCC2C(C)NC(c2ncnn2C)=O)=O)c1N 18722,Cc1cc(NC2CCSC2C)ncc1S(=O)(=O)N1CCCCCCCC1 18723,C1(C(=O)NCCc2cn(CC)nn2)CC=CCN1C(=O)C(C(C)C)SC(C)C 18724,C1(NC(CCN(CCC)C)=O)CCCCC12CCN(c1nc(Cl)nc(C)c1Cl)C2 18725,c1(CCC(=O)NC2CN(C(=O)Cc3ccsc3)C2)cccc(F)c1 18726,c1(C(=O)NC2CCC(N(C(CCOCC)=O)C)C2)cnc2cc(C)ccc2c1 18727,c1(C(=O)OCC)ccc(CC(C)C)nc1N1CC2(C(=O)OC)CC1CO2 18728,c1(C(=O)NCC2CN(C(C3C(C)CC3)=O)C2)cc(Cl)ccn1 18729,N1(C(CSC)=O)CC2CC(C1)C(CO)C2NC(=O)Cc1cccc(C(C)C)c1 18730,c1(OC)ccc(-c2ccnc(CO)n2)cc1.N1(C(Cn2ccnn2)=O)CCC(F)C1 18731,c1(CCC(=O)NC(C(C)NC(CCC(C)OC)=O)CO)c[nH]c2cccc(C)c12 18732,c1(C(N(CCCNC(C2CC(CC)C2)=O)C)=O)cc(C)ns1 18733,CC1(C)CC(=O)N(CC(N2CC(NC(C3(c4ccc(F)c(F)c4)CC3)=O)C2)=O)O1 18734,c1(C(=O)NC2(CN(C(C(C(C)C)C3CCC3)=O)C)CC2)nn(C)c(C(F)(F)F)c1Cl 18735,C1(C(=O)NCc2ccc(C(N3CCC3CF)=O)s2)C2CCCCC12 18736,c1(NCC2CC(O)C23CCC3)nccc(=NCCOC2CCOCC2)[nH]1 18737,C(=O)(CCCCCCCC1CC1)N1CC(NC(c2c[nH]c(=N)o2)=O)CC(C)C1 18738,c1(C(N2CC(c3cccc(Br)c3)(C)C2)=O)ccnc(Cl)c1N 18739,c1(NC(C(C2CCN(C(c3c[nH]c(=N)o3)=O)CC2)O)=O)ccc2ccncc2c1 18740,N1(c2ncc(C)cc2Br)CCCC2(CC(NC(=O)COCC3CC3)C2)C1 18741,C1(NC(c2ccc(C(C)(C)C)cn2)=O)CC2CC(NC(=O)C3=CCCS3)CC12 18742,C1(NC(CC2CC(OCC)C2)=O)CCOC12CCN(C(c1cnoc1C)=O)CC2 18743,C=CCCCC(=O)N(C1CCC(NC(C2(COC)C=CCC2)=O)CC1)C 18744,c1(C(N(CC(CC)NC(C(CC)C)=O)C)=O)nn2cccnc2c1Cl 18745,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(CNC(C2(C)C=CCC2)=O)CC1 18746,N1(C(C2C(OC)CCC2)=O)CCc2[nH]nc(CNC(=O)C(C)(C3CC3)OC)c2C1 18747,C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2cnc3n2CCC3)=O)CC12CCC2 18748,Cc1csc2ncnc(N3CCC(C)(C)C(NC(=O)C4=CCCC4(C)C)C3)c12 18749,C(=O)(CC(c1ccccc1)OC)N.C1(NC(C2CC(OCC)C2)=O)CC(COC)C1 18750,C1(CNC(c2c(F)cc(C)c(F)c2)=O)(NC(=O)Cc2cnoc2)CCC(F)(F)CC1 18751,N1(C(Cn2c(C)c(Cl)cn2)=O)C2CCC(C2)C1C(N1CC2CCC1C2)=O 18752,CCCC(C)CC(=O)NCCN(C(c1ccncc1CC)=O)CC 18753,c1(C(=O)NC2(CF)CCN(c3ncc(OC)cn3)C2)ccc2ncccc2n1 18754,CCN=c1[nH]cc(C(=O)NCC(F)CNC(=O)C(c2cccc(C)c2)C)s1 18755,c1(C(N2CC3(C2)SCCC3NC(=O)C(F)CC2CC2)=O)cccc2sccc12 18756,Nc1nc2ncccc2cc1C(=O)NC1CCCN(C(=O)C2=COCCO2)CC1 18757,N1(c2nc(C#N)cc(C)n2)CCc2occ(C(=O)NON3CCCC(O)C3)c2C1 18758,Cc1cc(C(N)C(=O)NCC2CC3(CCO2)CC3)cc(F)c1 18759,c1(OC)cccc(C(N2CCCC(CCc3cn(C(C)CO)nn3)C2)=O)c1F 18760,C(=O)(C(F)(F)CC(C)C)NC1C(CNC(C(=O)NC)=O)C1 18761,S(=O)(=O)(c1ccc(NCCC2COCCO2)c(Br)c1)NC(C)CC(N)=O 18762,CC1CC(NC(=O)NNC(=O)c2cn(C)cn2)CCN1C 18763,S(=O)(=O)(CCC(F)(F)F)N1CCN(C(CNCC2(C)CCC(=O)N2)=O)CC1 18764,N1(C(C2C(=C)CC2)=O)CCN(C2CCN(C(=O)Cc3ccc(C(C)=O)s3)C2)CC1 18765,c1(C(=O)NCC(C)NC(c2c(CC(C)C)nc(C)s2)=O)cc(N)cnc1C 18766,C(CC(C(=O)N1CCC(CF)C1)NC(=O)CC1CCCC12CC2)OCC 18767,C1(N(C)C(=O)Nc2ncc(C(F)F)s2)CCN(CCF)C1=O 18768,C(CC(=O)NCCCN(C(=O)C(O)Cn1cncn1)CCO)(C(F)(F)F)N(C)CC 18769,Cc1nsc(NC2CC2)c1C(=O)NCC1CCCC1NC(=O)CN1CC2CC2C1 18770,C(=O)(C1=NNC(=O)CC1)NC1(CF)CCN(C(c2c(C)n(C3CCC3)nc2)=O)C1 18771,N1(C(c2ccc(C)c(O)n2)=O)CCC2C(C1)CN2C(c1cccc2sccc12)=O 18772,C1(O)(C(=O)NCC2CCN(C(C3(CC(=O)OC)CC3)=O)C23CC3)CCCC(C)CC1 18773,C(=O)(C1=CC2(CN(C(=O)CC3CCCC(O)C3)C2)OC1)NC(c1ccnn1C)C 18774,c1(OCC)ccccc1CN(C(C1CC2CC2C1)C(=O)Nc1cnn(C)c1)C 18775,CC1(C)COc2ccc(C(=O)NC(C)(CNC(=O)Cc3nnc(O)s3)CO)cc21 18776,N(C1CCCc2ccc(F)cc21)C(=O)NNC(=O)C(F)C1CCCC1 18777,C(=O)(C(C)CCC1CCN(C(C2(C)CCCCC2)C(=O)NCCSC)CC1)OC 18778,C1(NC(C2CC(SC)C2)=O)CC2CC(C1)N(C(=O)CCCN1CCCC1)C2 18779,c1(OC)ccc(C(c2ccc(C)s2)NC(Cc2ccccc2)C2CC2)cc1Br 18780,c1(C(=O)NC2(C)CC(C(=O)NC3CC(C)OC3=O)C2)cn(C)c(=O)cn1 18781,c1(C(N(C(CN(C(C(C)NC(C)(C)C)=O)C)C)C)=O)ncc(F)c2ccccc12 18782,C1(CNC(=O)CC2CCCO2)CCCN1c1ccncn1 18783,c1(OC)cc(C(=O)NC23CCOC(CNC(=O)Cc4cn[nH]c4)(C2)C3)ccc1O 18784,C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(=O)CC2(C)CC2)CC1)CC#C 18785,c1(OC)cc(CC(=O)NCC2(F)CN(C(c3csnc3C3CC3)=O)C2)ccc1F 18786,N1(C(C(=O)NCCCOC)CCC2CCCCC2)CCOC(C2CCCO2)C1 18787,c1(C(=O)NCC(C)CNC(=O)CC2CC3C=CC2CC3)ccc2n[nH]cc2c1 18788,N1(C(c2c(OC)cccn2)=O)CCc2ccccc2C1CNC(c1ccc[nH]1)=O 18789,c1(C(=O)NCC2CC(NC(c3c(CC)ocn3)=O)C2)cc(C)c(C)o1 18790,Cc1ccc(F)c(O)c1C(N1CCCC(NC(c2cn(C3CC3)cn2)=O)CC1)=O 18791,N1(C(C2C(OC)CCC2)=O)CC2CCCC(NC(c3cccc(Cl)c3C)=O)(C2)C1 18792,C1(C(N(C(CNC(c2cc(F)ccc2O)=O)C2CC2)C)=O)CCC(=O)NC1=O 18793,S(=O)(=O)(c1cccc(OC(C)=O)c1)NC(C(=O)NCC(=O)N(CC)CC)(C)C 18794,C1(NCCC(C)(C)CO)CC12CCN(S(=O)(=O)c1ccccn1)CC2 18795,C12(C(=O)NCC3CN(C(C4C(c5ccccc5)C4(F)F)=O)C3)CCCN1CCC2 18796,N1(C(c2c(C3CC3)cccc2F)=O)CCCC(C2CN(C(C3C(C)CC3)=O)C2)C1 18797,C1(NC(c2ncc(OC)nc2)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1C 18798,C1(CC(=O)N(C(C(C(C)(C)C)=O)C(N)=O)C(C)(C)C)CCn2c(C(=O)O)cnc2C1 18799,c1(C(CC(=O)OC)NC(C(C)N(CC)CC)=O)ccc(OC)cc1 18800,C1(NC(Cc2cc(C)ns2)=O)CCCN(C(c2[nH]nc(C(F)(F)F)c2C)=O)CC1 18801,CC1(C)CC(N=c2ccnc(C(C)(C)C)[nH]2)CN(S(=O)(=O)c2ccccc2Cl)C1 18802,N1(C(c2ccc(Cl)s2)C(=O)NCCCCCC)CCC2CCN(C)CC12 18803,C(C(C)(C(=O)N(C)CC1CCCC1O)NC(=O)CC1CCC=CCC1)SC 18804,C1(NC(CCOC)=O)CN(C(c2sc(Br)nc2C)=O)CCC1CO 18805,Cc1nc(C(N2CCCN(C(=O)C(C)C3CCCC3)CC2)=O)n2c1CCC2 18806,c1(OC)ccc(NC(c2nnnn2C(C)(C)C)C2CCC2)c(OC)c1 18807,C1(NC(=O)OC(C)(C)C)CC2CC(C(=O)OC(C3COCCOC3)=O)CC12 18808,c1(C(N2C(C)CCC(NC(C(C)=C(CC)C)=O)C2)=O)cc[nH]c2nccc1-2 18809,C1(N(C(=O)C(O)CN2CCOCC2)CC)CCCN(c2ccccc2C)C1 18810,C1(NC(C(CSC)O)=O)CC2CCC1N2C(c1ccc(Cl)cc1N)=O 18811,Cc1cccc(C(COCC2(F)CC(NC(C3(CC4CC4)CC3)=O)C2)=O)c1 18812,N1(C(C)=O)CCn2ccnc21.C(=O)(C(C)N)N(CCCN(CC)CC)C 18813,C#Cc1ccccc1CC(N1CCC(NC(C2CCC(OC)C2)=O)CC1)=O 18814,C1(NC(CC(C)CF)=O)CC2CN(C(c3cc(Cl)n(C)n3)=O)CC2C1 18815,c1(C(=O)NCCN(CC(C)O)C(=O)Cn2cc(Cl)cn2)cc(C#N)cn1C 18816,c1(ON=CC(=O)Nc2cc(CNC(=O)OC(C)(C)C)sc2)cc(Cl)cc(Cl)c1 18817,N1(C(C(C)(C)SC)=O)CCC2(CC1)OCCC2NC(C1CCc2nn[nH]c2C1)=O 18818,Cc1cnc(C(N2CCC(NC(C3CC3C(N)=O)=O)C(O)C2)=O)cc1Cl 18819,n1(C(C)C)nncc1C(=O)NCc1cc[nH]c1C(=O)NCCOCCN=[N+]=[N-] 18820,c1(OC)cc(F)c(CC(N2CC(C)(NC(c3cc(C)cs3)=O)C2)=O)c(F)c1 18821,C1(C(=O)NCC(C)CN(C)C(c2ccccc2F)=O)CCCC(C)CC1 18822,Cc1ccc(NC(C2CCCN(c3ccccn3)C2)=O)cc1OCC(F)(F)F 18823,CCC(CC(C)C)C(=O)NCc1cncc(C(N2CCOC(CCOC)C2)=O)c1 18824,N1(C(C(CCC)CC)=O)CCCN(C(=O)CCSCCCC)C(C)C1 18825,N1(C(c2n[nH]c(C)c2Cl)=O)CC=C(C(C)(C)C(=O)N(C2CCN(C)C2)C)C1 18826,c1(C(=O)NC(C(C)NC(C(C)NC(=O)NC)=O)CO)ccc(O)nc1C 18827,C1(C(N(CC(C)C)CC(=O)NCC2CC2Cl)=O)CCCC(C)(C)C1 18828,c1(OCC)cccnc1C(=O)NCC1CCCCN1C(C12CCC1C2)=O 18829,N1(C(C(n2cc(Cl)cn2)C)=O)CCC2(C)CN(C(C3CCC4CC34)=O)CC12 18830,CC1(OCCc2cn(CC(N3CC(c4ncccc4Cl)C3)=O)nn2)CC2CC2C1 18831,C12(CNC(C3(CCCCNC(C(CCC)O)=O)CC3)=O)CCCN1CCC2 18832,c1(CN(C)C(C2(C)CCN(C(=O)CCc3cnc(O)[nH]3)C2)=O)ccc(Cl)cn1 18833,C1(C(N2CCCC(CC)C2)=O)CC12CCN(Cc1ncc(Cl)nc1Cl)C2 18834,c1(NC(=O)CN2CCN(c3ccncn3)C3CC23)ccc([N+](=O)[O-])cc1C(F)(F)F 18835,C(=O)(C1=CC(C)(C)C1)N1CCC(C(=O)Nc2c(CC)nn(C)c2)C1 18836,Cc1ccc(=O)n(CC(N2CCN(C(c3ccc(C)c(C)n3)=O)C(CO)C2)=O)n1 18837,N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(c3ccnnc3C)=O)C2)C1 18838,N1(C(c2c(C)csc2)=O)CCN(C(c2cccc3ncsc23)=O)CC2(CC2)C1 18839,CCCS(=O)(=O)C(C)C(=O)N1CC(N(C)C(c2c[nH]c(=N)nc2C)=O)C(C)(C)C1 18840,C1(CNCCOC(c2c(C(C)C)cccc2)=O)CC2(CCC(F)(F)CC2)C1 18841,C1(C(N(CCCNC)CCNC(C2CC2F)=O)=O)CCCN1C(=O)C(C)(C)C 18842,N1(C(C(C)=CC=C)=O)C2CCC1CC(C(=O)NC(c1cn(C)nn1)C)C2 18843,C#Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)CCCSC)C23CCC3)c1 18844,C1(=O)CC(C)CO1.c1(C(C(=O)N(C2CCNC2=O)CC)OC)ccnn1C 18845,Cc1nc(N2CC3(CCC(CNc4cc(C)c(C)c(C)c4)O3)C2)c2ccsc2n1 18846,c1(CC)ccc(C(=O)NC2CN(C(=O)C(N3CCOC3=O)C)CC23CC3)cc1F 18847,S(=O)(=O)(c1cccnc1N1CCCN(C)CCC1)NCCc1ccn(C(C)C)n1 18848,c1(C(=O)NC(CNC(CC(C)F)=O)(C)C2CCC2)cnn(CCO)c1C(C)C 18849,C(=O)(C(O)CC(F)F)N1CC(CC(CNC(CN2CCC(OC)C2)=O)(C)C)C1 18850,c1(CNC(CCC(=C)C)=O)nc2c(s1)CCN(C(C1(F)CCCOC1)=O)C2 18851,C12(C(=O)NCC(C)(CO)NC(c3c(OC)scc3)=O)CCCC1C2(F)F 18852,c1(OC)ccc(OC)c(C(=O)NC(C)CNC(C2(C(C)C)CCC2)=O)c1 18853,C(=O)(C(C)(C)CCNC(C1CC(C)(F)C1)=O)NC(C(=O)NC(C)C)C 18854,N1(C(CCCC(=O)c2cccs2)=O)CCCC2(CCCN2C(C2CC2F)=O)C1 18855,c1(C(=O)NCC(C2CCC2)NC(CC2C(C)(C)CCCO2)=O)scc2c1OCCO2 18856,C(C)(C)(CCCCC(=O)NC(C)CNC(c1sc(OC)nc1C)=O)OC 18857,C1(S(N)(=O)=O)(C(=O)NC2CC(NC(C=CCOC)=O)CC2O)CCCC1 18858,CCC(CC(=O)NCCC(C)(C)NC(=O)CS(=O)(=O)N1CCCCC1)SC 18859,c1(CN(CC(=O)NC2(CNC(C(C)NS(C)(=O)=O)=O)CC2)C)ccccn1 18860,C1(COc2c(N=[N+]=[N-])ccc(F)c2)CCC2(CCOCC2)CO1 18861,C1(C(N(C2CN(CC)C2)C)=O)CCc2c(C)nnn2C1 18862,N1(C(=O)OC(C)(C)C)CCC(CC)C(OC)C1.c1(COCCN)noc(C(C)C)n1 18863,C(CC(=O)NC(c1cnn[nH]1)(C)C)(CC(C)C)NC(c1c(CC)n(C)nn1)=O 18864,Cc1cnc(NCC(F)C2CCC2)c(S(=O)(=O)NCC2CCC(C)(C)O2)c1 18865,c1(SC)cnc2ccccc2c1.CCCC1C(=O)NCC(C)NC(=O)N1 18866,N1(C(c2cncc(C)n2)=O)CC(CNC(=O)Cc2ccc(F)cc2)CC(C)C1 18867,C#CCCCCCCC(=O)NCC=CCNC(=O)CC1(S(C)(=O)=O)CCOCC1 18868,c1(C(=O)NCC(CC)(C)NC(c2ccsc2OC)=O)cnc2c[nH]nc2c1 18869,C(=O)(C1Cc2ccc(Cl)cc21)N1CCC2(CN(C(C(CC)NC(C)=O)=O)C2)C1 18870,c1(CC(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)ccc(F)cc1F 18871,C#CCCN=C(NCCC(c1ccccc1)O)N1CCC(N(C)C)C1 18872,C1(N(C(CC=C)=O)CC)CCN(CCCc2nnc(-c3ccccc3)o2)CC1C 18873,N1(C(c2cc(C)n(C(C)C3CC3)n2)=O)CC(C)(C)OCC1CNC(=O)C=CS(C)=O 18874,C1(C(=O)NC2C3CN(C(C4CCC(C(=O)OC)C4)=O)C2C3)CN2CCN1C(C)C2 18875,N1(C(C(CSC)O)=O)CC2CC(C(=O)NCC3CCOC3C)(C2)C1 18876,Cc1ccn(C)c1C(=O)NCC(C)(C(C)C)NC(=O)C(C)n1cccn1 18877,C1(C(=O)NC(C(C)NC(=O)CSCC(N)=O)C)(CF)CCOCC1 18878,c1(OC)cc(C#N)ccc1NC(C1(C)CCN1C(c1cnc2[nH]ncc2c1)=O)=O 18879,CC(N=c1[nH]c(=NCc2nc(O)cc(O)n2)[nH]c2c1COC2)c1ccsc1 18880,c1(C(N2C(C#N)C3CC3C2)=O)cnc2ccc(-c3ccc(F)c4c3CCC4)cn12 18881,C1(NC(=O)C=CCF)CC(CNC(c2cc(-c3ccccc3)no2)=O)C12CCC2 18882,C1(c2cn(CCCF)nn2)(C(N2CC(N3CCC(F)C3)C2)=O)CCCCCC1 18883,Cc1ccc(C)c(OCCCC(=O)NCCCNC(=O)C(=O)N(C)C)c1 18884,c1(NCCNC(Cc2c(C)nn(C)c2)=O)cccc([N+](=O)[O-])c1N1CCCC1 18885,C1(=CC(=O)NC(C)CC(C)NC(=O)COC2CCCOC2)CCC(C)(C)CC1 18886,c12ccc(C)cc1CC(=O)N2.N1(C(COCCOC)=O)CC=CC1C(=O)NC 18887,C1(CC=C)(C(=O)NCC2(C)CCN(C)C2)CCCN1C(c1ccc(F)cc1)=O 18888,CC(C)C(C(=O)NCCCCNC(C1(C)CC1)=O)NC(c1cccs1)=O 18889,C1(OC)(CO)CCN(c2nc(-c3ccc(Cl)cc3Cl)no2)CC1 18890,Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2nn(C)cc2C)=O)n(C2CCC2)n1 18891,C1(C(N(CCC(=O)NCC(CC)C)C)=O)CCC2CC12 18892,C1(C(N(CC(C)C)CCCO)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CC(C)O1 18893,C(=O)(C(F)(F)C(F)F)N1C(CN(C)C(C2CC2c2ccc(F)cc2F)=O)CCC1 18894,c1(C(N(C(C)CNC(C2(C)COC(=O)C2)=O)C)=O)ccc(Cl)cc1OCC(N)=O 18895,C(CCCCCCC(=O)NCC1CCN1C(c1nc(C)oc1OC)=O)SC 18896,CCC(CC(=O)N1CC(N(C)C)C1)NC(=O)C(c1ccc(C)cc1)=O 18897,CCC(C)(C#N)C(=O)NCCC1CN(C(=O)C(F)(F)COC)CCO1 18898,N1(C(=O)NC(c2ccc(Cl)cc2)Cc2ccccc2)Cc2cccc(Cl)c2C1 18899,C1(C(=O)NCCN(C(c2cccc(C3(C)CC3)c2)=O)C(C)C)(OC)CCOCC1 18900,CCC(O)CC(=O)NCC(C)NC(C1(NC(C)=O)CCC1)=O 18901,c1(C(N2CCCCC(CNC(CNC(C)=O)=O)C2)=O)n[nH]c2ccccc12 18902,N1(C(c2cc(O)cc(F)c2)=O)CC2(C1)CN(C(C1CCC(C(=O)O)C1)=O)CCO2 18903,n1(CCNC(c2cc(C(F)F)on2)=O)cc(CCNC2CCOC2)nn1 18904,c1(C(=O)NCC2(OCC)CN(C(C3CC3C)=O)C2)cccc2nsnc12 18905,C(C(O)C(=O)NC1CCC(C(=O)OC)C1)N(CC)CC 18906,C1(OC)(CNC(=O)C(N2CCOCC2)C)CN(C(=O)C=C2CCOCC2)C1 18907,c1(CNC(COc2c(S(C)(=O)=O)cccc2)=O)c(F)c2ccccc2oc1=O 18908,c1(SC)ccc(NC(=O)C(F)CC2CN(C(C3(F)CC=CCC3)=O)C2)cn1 18909,c12cc(n(C)n1)CNC(=O)C(C)NCC(=O)N2.C(CC(C)C)OC(=O)OC 18910,N1(C(CC2N(C(C3C(C)(C)OCC3)=O)CC(O)C2)=O)CCC2(CCC(O)C2)C1 18911,c1(C(=O)NC(CN(C(c2ccc(CCC)s2)=O)C)C)cnc(OCC)cn1 18912,C1(C(N2CC(CNC(C(CC)(C)O)=O)(COC)C2)=O)CC(C)CC(=O)N1 18913,c1(C(=O)NCCC2CSCCN2C(=O)CC2CSCCS2)cccn2ncnc12 18914,Cn1cc(I)c(C(c2nnnn2CCN2CCCCC2)NC2C(C)(C)C2(C)C)n1 18915,c1(C(N(CC(O)CN(C)C(c2cc(O)nn2C)=O)C)=O)cnn2cc[nH]c12 18916,CC1CN(C)CCC1N(C)C(C1(NC(C2CC3(CCC3)C2)=O)CCCC1)=O 18917,c1(C(=O)NCCC2CCCN(C(=O)CC(F)(F)F)C2)ccn2ccsc12 18918,N1(C(C(C)OC(C)=O)=O)CC(C)(C)CC1CC(=O)NC1CCC2(CCC2)C1 18919,C1(NC(CNC(C)=O)=O)CCCN(C(c2cc(CC(C)C)[nH]n2)=O)CC1F 18920,C1(C(N2CCC(N(C)C(=O)OC(C)(C)C)CC2)=O)CC2CCC1NC2=O 18921,c1(C(=O)NCC2CN(C(C3(CC)CCCO3)=O)CC2O)cc2oc(C)c(C)c2[nH]1 18922,N1(c2nnc(C#N)s2)C2CCC1C(CNC(=O)CCC1CCCO1)C2 18923,CC(O)CCCC(=O)NCC1CCCN1C(c1cnccc1C#N)=O 18924,c1(CCN(C(=O)C(c2ccccc2)C)C(C=C)C)ccc(F)cc1F 18925,C1(CNC(C(C(C)=C(C)C)O)=O)CCN(C(c2cn(C)ccc2=O)=O)CC1(F)F 18926,CCCCC(=O)C(=O)N1CCC(C(C)NC(C2CC3C(C2)C3(F)F)=O)CC1 18927,C(=O)(C(C)CC(F)F)NCC(C(=O)N(CCC#C)C)O 18928,N1(C(C(C)OC)=O)CCOC2(C1)CN(CCc1ccc(C)cn1)C2 18929,N1(C(c2c(C(=O)OC)cco2)=O)CCN(C(C2(C)CCCS2)=O)CC1C1CCC1 18930,N1(C(c2cccc(CCN(C)C)c2)=O)CC2CCN(C(C3CCC4CC34)=O)C2C1 18931,N1(C(c2ccc(C)s2)=O)CCN(C)C(C(=O)N(C2CCCC2)C2CC2)C1 18932,C1(NC(C=Cc2nc(C)sc2)=O)CCC(O)CN(C(=O)CCc2nc[nH]n2)C1 18933,c1(CC)cc(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc1Cl 18934,Cn1c(CNC(=N)N)c(NCCC2CCCC2)c(=O)n1C1CCCC1 18935,C1(CNC(CC)=O)CN(C(c2ccc(-c3nc(C)c(C)[nH]3)cc2)=O)C(C)(C)C1 18936,C1(CC(=O)NC2CCCC(O)C2)CCC(NC(c2ccn(C3CC3)n2)=O)CC1 18937,N1(C(c2ccc(C)[nH]2)=O)CC2C3CCC(C2C1)N(C(c1ccsn1)=O)C3 18938,c1(CC)ncsc1C(=O)N(C)CC1CCN(C(=O)CSC2CC2)C1 18939,CCC(CC(=O)NC(C)(C)CCCO)C1CC1 18940,N1(C(=O)NC(c2ccc(C3(C)NC(=O)NC3=O)cc2)C)CC=C(C(F)(F)F)CC1 18941,C(CCCCC(=O)NCCOCCCO)NC(C1CC=CCO1)=O 18942,N1(CCCc2cn(CCCC(=O)O)nn2)CCCCCCC1CSC(F)F 18943,N1(C(CCOCC(C)C)=O)CCC(C)(NC(C2CCC2SC(F)F)=O)C1 18944,OCCC(N=c1nc(N2CCC(NC3CC3)C2)c2ccccc2[nH]1)c1ccccn1 18945,C(c1ccccc1Cl)=CC(=O)NCCCC(C)(C)NC(C1CC(C)OC1)=O 18946,N1(c2c(C)c(NCCS(=O)(=O)N(C)C)ncn2)CCC(C#N)(C(C)C)CC1 18947,c1(C(N2CCC(N(C)C(C3CC(C)(C)CN3C)=O)CC2)=O)nccc2[nH]ccc12 18948,N1(C(c2c(C)cncc2C)=O)CCN(C(=O)C(C)Oc2cccc(O)c2)CC1C 18949,c1(NC(=O)C=Cc2ccsc2)ccccc1OC1CN(C(=O)C(F)=CCCF)C1 18950,Cc1nc(C(N2CCC(C)(NC(=O)CC3CC4C=CC3C4)C2)=O)c2ccccn12 18951,CC1C(=O)N(c2cc(-c3nc(-c4nnn(C)n4)no3)ccn2)CCS1=O 18952,C(C)(C)(CC(=O)N1CC(CCCCCO)C1)NC(C(F)=CCC)=O 18953,c1(C(=O)NC2CCN(C(C3C4COCC34)=O)CC2F)cc2ccccc2[nH]1 18954,C1(CNC(C(C)=C(C)C)=O)CCN(C(C2CNC(=O)N2)=O)C12CCC2 18955,c1(OCC(N2C(C(C)C)CC(O)C2)=O)ccc(C2CC2)cc1C(F)(F)F 18956,c1(C(=O)NC2CCC(C(=O)NC(C#C)CCC)C2)ncc(OC)cn1 18957,CCC(C)C(CC(=O)Nc1ccc(C)nc1OC)NC(=O)C(O)CCN(C)C 18958,CC1CN(C(c2ccc(Cl)cc2)=O)CCC1CNC(C1OCCOC1C(F)(F)F)=O 18959,CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)Nc1cccc(CO)c1 18960,C#CCCCCCCC(=O)NC(C1CCN(C(=O)CSC(C)(C)C)CC1)CO 18961,N1(S(CC(C)C)(=O)=O)CC2(CCN(C(c3ccn(C(F)F)n3)=O)C2)C1 18962,c1(C(N2C(c3scc(CCOC)n3)CCC2)=O)cncc2ccccc12 18963,C1(C(N2CC(CSC)C2)=O)CC(C)N1C(C1CCC1(OC)OC)=O 18964,N1(C(C=NOC)=O)CCOC2(CCN(C(=O)C=Cc3c(F)ccc(Cl)c3F)C2)C1 18965,N1(C(c2cnccn2)C(=O)NCCCC)CCC(N(C)C)C(CC)C1 18966,c1(N2CC3C(NC(C(C)(C)C)=O)C3C2)nc(=NCC2CCCCS2)[nH]c2c1SCC2 18967,N1(C(CSCCC)=O)CCC(C)(CC(=O)NC(C)(C)CCOC)C1 18968,C(C(=O)NCCC1CC(OCC(=O)NC(C)C)C1)(C(C)C)n1ncc(C)c1 18969,c1(C(N(CCC(N2CC(C(CC)CC)C2)=O)C)=O)cn(CC)cn1 18970,CN1CC(C)(C)CC1C(N1CC(CNC(=O)CC2CCCCCCC2)CC1(C)C)=O 18971,N1(C(C(C)OC(C)C)=O)CC2(C(=O)OCC3CC4(CCC4)C3)CCC1CC2 18972,c1(C(C(=O)OC)=O)cccnc1CNC(C)CCCNC(c1cc(Cl)cn1C)=O 18973,N1(C(C(CC=CC)CC)=O)CCC(C(=O)Nc2nc(C)c(C)s2)=C(F)C1 18974,c1(CC(=O)NCC(C)CNC(=O)C(F)CC2CCCC2)cnc2c(=O)[nH]ccn12 18975,c1(NCCC(C)O)cc(=NCC(C2CCCC2)N(C)C)[nH]cn1 18976,c1(C(N2C(C(N(CC)Cc3c[nH][nH]c3=N)=O)CC2)=O)cc(Br)cnc1Cl 18977,C1(CC(=O)NCC(CN(C)C(C2CC(OC(F)F)C2)=O)O)CCNC1=O 18978,CCC(C)(C)C(O)C(=O)NCC#CCNC(C1CCC2(CC1)CC2)=O 18979,N1(C(CC(CC)C2CCC2)=O)CC2CN(C(C3CCCC(C(N)=O)C3)=O)CC(C1)O2 18980,c1(C(=O)NC(c2ccccc2I)c2ccccc2)ccc2c(c1)COC2 18981,N1(C(C(C)c2cc[nH]n2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 18982,C(=O)(C(C)CS(C)(=O)=O)NC1CC(NC(c2ccc(-n3ccc(C)c3)cc2)=O)C1 18983,C1(C(N2CCCCC(NC(CCC3(C)CC3)=O)C2)=O)CCc2ncccc2C1 18984,c1(C(=O)NC2CCN(C(=O)CSC(F)(F)F)C2)cc(F)c(F)c(F)c1 18985,C(=O)(C1=CCCN(C(c2cc(OC)cc(F)c2)=O)C1)N1CCC(C(=O)OC)C1 18986,c1(-c2nn(C(C)C)c(C3CSC3)n2)cccc2ccccc12.C1NC(=O)OC1(C)C 18987,C1(NC(C(CCOC)C)=O)CCN(C(=O)COCc2cccnc2)CC(O)C1 18988,c1(C(=O)NC(CN(C(CCC(=C)C)=O)C)C)cc2c(C)c(F)ccc2[nH]1 18989,N1(C(C(C(C)C)N(C)C)=O)C2CCC1CN(C(=O)CN1CC=CC1)CC2 18990,c1(C(N2C3C(CC(NC(C4CC4(F)F)=O)C2)C3)=O)ccc2nnc(S)n2c1 18991,N1(C(c2cc(C)c(C)o2)=O)CC2(CCC2)CC1CNC(=O)CCc1cscn1 18992,C#Cc1ccc(CCCC(=O)NCC2CCCCN(C(C3(CC)CC3)=O)C2)cc1 18993,c1(C(N2CCC(NC(c3[nH]cc(CC)c3)=O)C2)=O)ccccc1NCC1CC1 18994,N1(CC(=O)N(CC(=O)NCC(F)F)C)CCNC(=O)C1 18995,c1(CC(=O)NC2C3CN(C(CN4CC(C)(OC)C4)=O)CC32)nsc2ccccc12 18996,Cn1c(NC(C2=Cc3ccccc3OC2)c2nnnn2C2CC2)cc2ncccc12 18997,C1(C(N2C(C(C)C)CCCC2)=O)N(C(=O)CC(=O)NC(C)(C)C)CC12CCCC2 18998,C(=O)(CC(C)CCCCCC)N1CC(NC(CC=C=C)=O)C(C)(C)C1 18999,C(c1cc(Br)cs1)=CC(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 19000,c1(N(CC(=O)NCC2CCC(NC)C2)C)cccc(C#N)c1 19001,N(C1COc2ccc(Cl)cc21)C(C1C2CN(C(CNC(C)=O)=O)CC21)=O 19002,Cc1ccc(F)c(CNC(C2(C)CCCN(C(C3CC4(CC4)CO3)=O)C2)=O)c1 19003,C(C)(CCCCNC(=O)Cc1cccc(Br)c1)NC(Cc1cnc(C)o1)=O 19004,C(c1ccc(Cl)nc1)=CC(N1CC(NC(C(C(C)C)SCC)=O)(CO)C1)=O 19005,C(=O)(CCS(=O)(=O)CC(C)C)NCC1CC(NC(CSCCOC)=O)C1 19006,c1(C(=O)NC(CNC(C2(CSC)CC2)=O)C(C)C)nc(C)nn1C 19007,c1(CC(N2C(CCCNC(C(F)=CCC)=O)CCC2)=O)cc(C)ccc1OC 19008,C1(C(N2CCCC2CO)=O)CC2C=CC1CC2 19009,c1(C(=O)NCCN(C(=O)CC2CC(F)C2)CCC)ccc2nc(O)cc(O)c2c1 19010,c1(C(C(=O)NC(C)C(=O)N2CC(N3CCCC3=O)C2)O)cccc(F)c1 19011,CCCC(C)(O)CC(=O)Nc1ccc(NC(=O)CCCC2CCCCC2)cc1C 19012,N1(C(c2ccc(C)o2)=O)CCN(C(=O)C=CCN2CCCC2)C(C2CCCC2)C1 19013,N1(C(C2N(C(c3cc(OCC)no3)=O)CCC2C)=O)CCCC(N=[N+]=[N-])C1 19014,c1(C(N2C(COC)CN(C(=O)C(F)C3CC3)CC2)=O)cc(C)c(C)cc1C 19015,CC1CCCN(CCNC(=O)CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)C1 19016,N1(C(c2ccc(C(C)C)nc2O)=O)CC2CCCC2(Nc2ccnc3ncnn23)C1 19017,c1(N2CCN(Cc3cccc(C)c3I)CC2)nc2ccccc2o1 19018,c1(C(N2CCC(CNC(C(F)=CCC)=O)CC2)=O)cc(C)cc(OC)c1O 19019,N1(C(CC=CC=C)=O)CC(CNC(=O)CC2CCC(=O)N2C)C2(CC2)C1 19020,O(NC(=O)C(F)CC(C)(C)NC(=O)CN1CCOCC1)CCC(C)C 19021,C12(C(N3CC(C(C)NC(C45CCN(CC4)CC5)=O)C3)=O)CCCCC1C2(F)F 19022,c1(N2CCC(NC)CC2)ccnc2cc(C#N)ccc12 19023,N1(C(c2nn[nH]n2)C)CCN(C(=O)C(F)C2CCOC2)CC1 19024,CCC(CC(C)C)C(=O)N(CC(=O)NCC1(C(C)O)CC1)CCOC 19025,C12(CNC(c3cc(C)no3)=O)CCCCC1CN(C(=O)CCCc1cccs1)C2 19026,C#CCCCCCCC(=O)NC1CCCN(C(=O)CC(C)N2CCCC2=O)C1C 19027,C(CCCCC(=O)NCC(c1ccccc1)NC(c1ccn(C)c(=O)c1)=O)OC 19028,N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CC2CCN(C(C3CC3F)=O)CC(C2)C1 19029,C1(CCC(=O)NCC(C)(C)OCC)CCCCN(C(C2CC3(CC(=O)C3)C2)=O)C1 19030,c1(OCC)ccccc1CC(=O)NCCc1ccncc1Br 19031,N1(C(CCc2ccc(C)o2)=O)CC2(CCC2NC(C2CCCC(=O)N2)=O)C1 19032,Cc1nc(CC(=O)NCC(O)CN(C(=O)C(C)(C)CN(C)C)C)c(C)s1 19033,c1(CC)ccc(C(N2CC(NC(=O)C(C3CC3)SC)C(n3cccn3)C2)=O)nc1 19034,c1(C(N2CCC(C3N(C(CC(=O)OCC)=O)CCC3)C2)=O)cncc(N)c1C 19035,n1(COC)nc(C(=O)NC2CN(C(c3cccc(C)c3Cl)=O)CC2F)ccc1=O 19036,c1(C(=O)NC2C(CNC(=O)CCNc3ccc(Cl)cc3)C2)cccc2[nH]ncc12 19037,N1(C(C2C(CC)CCCC2)=O)CC23CCCC2(C1)CN(CC(O)C1CC1)C3 19038,CC1(C)CCC(C)(NC(=O)C(CCC2CC2)NC(C2CCCC(C#N)C2)=O)CC1 19039,C1(CNC(C2N(C(CC)=O)CCC2)=O)(NC(=O)CC(C)C(F)F)CCC(C)(C)CC1 19040,N1(C(COCC=C)=O)CC2CCC1CN2C(c1cc(CC(=O)OC)on1)=O 19041,C1(C2(O)CCOCC2)(C(N2CCC(CNC(=O)Cc3ccc(O)cc3)C2)=O)CC1 19042,C1(C(N(CC(C)CNC(=O)CCCN(C)C)C)=O)CC(C)OC(C)C1 19043,CCC(C)CCC(=O)N1CC(O)CC1CC(=O)NCC1CCOC1C1CC1 19044,c1(C(N2CC(NC(C(C)CCSc3ccc(Br)cc3)=O)C2)=O)cnn(C)c1C#N 19045,C1(NC(CC)=O)CCCC1C(=O)OC1(CO)CC(C)C1 19046,c1(OC)cc(C#N)ccc1C(=O)N(C)CCc1ccc(C)cn1 19047,C1(NC(C(C)N(C(C)=O)C)=O)CCCN(C(c2coc3c2COC3)=O)C1C 19048,Cc1n[nH]c(C)c1CC(=O)NC(Cc1ccc(F)cc1)CC(=O)NCC1CC1 19049,c1(NC(C(C2CC2)N(C(=O)CC2CCSCC2)C2CC2)=O)cc(Cl)cnc1O 19050,c1(OC)ccc(CC(=O)NC2CC3(C2)CN(Cc2cc(Cl)cc(Br)c2)C3)c(F)c1 19051,c1(C(N2CC(NC(C(CCCOC)C)=O)(COC)C2)=O)[nH]nc(Cl)c1[N+](=O)[O-] 19052,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)CC(C)(C)c2ccccc2)=O)c1 19053,C1(C)(NC(CCSC)=O)CCCN(C(=O)CC2OCCO2)C1 19054,N1(C(C2CSCCN2C(=O)NCC2CCCO2)=O)CCc2ccccc2C1 19055,c1(-c2cn(C(C)C(=O)N(C)C)nc2)cccnc1C(CO)N(C)C(C1CCC1)C 19056,N1(c2n(C(C3CCCC3)C)nnn2)CC2OC(=O)N(c3ccc(N(C)C)cc3)C2C1 19057,Cc1c(C(=O)O)sc2ccc(CN3CCNCCC3C(C)(C)C)cc12 19058,c1(SC)nc(=NCC(C)N(C)C(c2ccc3cc[nH]c3n2)=O)s[nH]1 19059,C1(CNC(COCCCC#C)=O)CCC(C(=O)N)O1.C12(CC1)C(=O)N2C 19060,c1(C(N(CCCNC(C2(C)CC(=C)C2)=O)C(C)C)=O)ccnc(C2CC2)c1 19061,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19062,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC(CCCC)CNC(c1[nH]ncc1C#N)=O 19063,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CCN(c2ccncc2)CC1 19064,C1(N2CC(C)C(NC(C3CC3c3ccccc3)=O)CC2)CCCCCCC1(C)C 19065,C(=O)(CCCC(F)F)N1CCCC(CN(C(=O)Cc2cnn(C)c2)C)C1 19066,c1(C(=O)NCC(CC=C)NC(=O)C(n2nccc2C)C)ccnc(N(C)C)c1 19067,N1(C(c2c(CC)scc2)=O)CC2CC(C1)CN(C(=O)C(C)CCO)C2 19068,N1(C(CC2CC(=O)C2)=O)CCC(CNC(c2ccc3n[nH]cc3c2)=O)C(F)(F)C1 19069,C1(C(N2CCOC(c3cccs3)C2)C(=O)NC(CC)C)CC2(CCCO2)C1 19070,NS(=O)(=O)N1CC(C(=O)NC2CCCN(C(C3CCN(C4CC4)S3(=O)=O)=O)C2)C1 19071,c1(CC)noc(C(=O)N(C2CN(C(c3cn(CC)nc3C)=O)C2)C)c1C 19072,C1(=O)C(C#N)NC(=O)C(=O)NCCC2CN1C2.c1(S)ccccc1.CC(C)(C)O 19073,C1(CNC(C(C)OCC)=O)CN(C(=O)Cc2sc(C)cc2C)CC1O 19074,c1(C(=O)NCC(C2(O)CN(C(C(C)OCC)=O)C2)(C)C)ccc(Cl)c(F)c1 19075,C1(CC#C)CCC(=O)N(CCN(C2CCN(CC(C)C)CC2)C)C1 19076,C(c1ccncn1)=CC(=O)NC1CC(NC(C2(C#N)CC2)=O)C1 19077,CC1CC(C)(C)CC1(c1nnnn1C)NCC1CCC=CCC1 19078,c1(C(=O)NCC2C(NC(C3N(CCC)CCC3)=O)CC2)ccn2c1CCC2 19079,C(CCCCC(c1nnnn1C)NCCC1CCCN1C)OC 19080,CC(c1ccccc1)=CC(=O)NCC1CC(NC(c2ncccc2F)=O)C1(C)C 19081,C1(C(=O)O)CN(C(c2cc(-c3ccco3)on2)=O)C2CCOC2=CC=CC=C1 19082,C(=O)(C(C(C)C)SCC)N1CC(C)(NC(=O)CO)C1.C=C1CC(C)(COC)C1 19083,N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(C)(F)F)C2CCCCC2C1 19084,c1(CCC)ccc(C(=O)NC2CCN(C(=O)CCS(C)=O)C2C)cc1[N+](=O)[O-] 19085,CCC(C)(CC)C(=O)NC1CCN(C(c2sc(C)nc2Br)=O)C(C)C1 19086,N1(C(c2cc(C#N)on2)=O)CCC2(CCC2)C(NC(=O)CCC2CC2CC2CC2)C1 19087,c1(C(C)C)cc(NC(=O)NC2(C3CCCC4CC34)CCC2)nn1C(C)(C)C 19088,N1(C(c2c(CC)n(C)nn2)=O)CCC(C(=O)N2CC(CC)(CO)C2)=C(F)C1 19089,c1(C(N2C(CNC(CC(CC)CC)=O)C=CC2)=O)cn(CC#N)c2ccccc12 19090,N1(C(=O)C=C2CCC2)CCN2C(=O)C(NC(c3c(C)nn(C)c3C)=O)CC2C1 19091,CC1CCC(CN)N1C(=O)NCCC=CBr 19092,C1(N(C)C(c2ccncc2O)=O)CCN(C(c2cnc(-c3ccoc3)s2)=O)CC1 19093,Cc1c(C(=O)NC2CCC(CNC(c3nccn3C)=O)C2)cnn1CCO 19094,Cc1nc2c(C)cc(NCC3(C)CCNCC3)cn2n1 19095,c1(C(N2CC(CC(C)NC(c3cncnc3)=O)C2)=O)cccc(S(C)=O)c1 19096,C1(C(=O)NC(CC(C)NC(Cc2ccc(C(=O)NC)cc2)=O)C)CC(F)(F)C1(C)C 19097,N1(C(c2c(OC)cnc(Cl)c2)=O)CCC2(CCC2)C(CNC(C2(O)CCC2)=O)C1 19098,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19099,c1(C(N2CC(CN(C(C(C(C)OC)O)=O)C)C2)=O)cn2ccccc2n1 19100,CC1CCC(C(=O)NCC2CN(C(C)C)C2)N(C(C2COCCN2C)=O)C1 19101,C(=O)(CCCCCCn1cc(C(O)C(C)C)nn1)NC.Cc1noc(C(C)C)n1 19102,C(=O)(C1COc2ccccc21)N(C(CNC(C(C)NC(C1CCCC1)=O)=O)C)C 19103,C1(CC(=O)NCCC(C)OCC#C)CCN(C(c2cscc2C)=O)C1 19104,c1(-c2n(-c3cc(F)ncc3)nc(CCn3ccnc3)n2)c(F)cc(Cl)cc1Cl 19105,C1(C(=O)NCCCCC)(COC)CCN(C(=O)C(=O)N(C)C)C1 19106,N1(CCC=C)CCN(C(=O)C(CCF)NC(C2CCC(C)O2)=O)CC1 19107,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2ccnn2CC#N)=O)CC1)C 19108,[N-]=[N+]=NCCCCCC(=O)NCCC1CCN(C(=O)C=Cc2nccs2)C1 19109,C1(N(C(C=CCNC(C2C(C)(C(F)F)C2)=O)=O)C2CC2)CC2(CCC2)C1 19110,CCC(CC)(CO)NC(C1(CCNC(=O)Cc2cn(C)nc2C)CCC1)=O 19111,CCCC(O)(CCC)CC(=O)N1CCC(NC(c2ccc3nccn3n2)=O)C1 19112,N1(C(CCN(CC)CC)=O)CC(CN(C(=O)COCCC(C)C)C)C2(CC2)C1 19113,C(=O)(C(CCC)c1ccc(Cl)cc1)NC(CNC(C=CCCC)=O)C1CC1 19114,C#CC1(C(=O)NC2C=CCC2)CCN(C(=O)CNC(N)=O)C1 19115,C1(N(c2ncc(Br)cn2)C(C2CCCOC2)=O)CC2CCC(C1)N2 19116,C(=O)(C(F)C1=CCCCC1)NCC1N(C(C2(C)C=CCCC2)=O)CCC(C)C1 19117,c1(NCC2(C)CCCOC2)nc2ccccc2nc1NC1CCC(C)(F)CC1 19118,C(=O)(NNc1ccc(S(=O)(=O)N(C)C)cc1)Nc1cccc(OCC)c1 19119,C(c1ccoc1)=CC(=O)N(C(C)CNC(=O)Cc1[nH]cnc1C)CC 19120,C1(C(NOCC)=O)CCCCN1C(=O)CN1CC2CC2C1 19121,c1(C(=O)NCc2cc(C)ncn2)coc2c1CN(C(=O)C(c1ccccc1)F)C2 19122,C(=O)(CC(CNC(C1C=CCS1)=O)OC)NC1CCN(CC)C1 19123,C(CCCCCc1ccccc1)N(C)C(=O)NC1(C)CCOC1 19124,C(C(C(C)C)NC(c1ocnc1C(F)F)=O)NC(C1(C(=O)OCC)CC1)=O 19125,C(=O)(C(CC)NC(=O)CC1(COC)CC1)N(CCCC)C.SCC 19126,C=C(Br)CC(C)(C)C(=O)NC1CCCCN(C(c2cc(CN(C)C)on2)=O)C1 19127,c1(C(C)=O)cc(C(=O)NC(CNC(c2cc[nH]c2C)=O)C2CCC2)cs1 19128,C(CCSC)(C(=O)NC(C)(C)C(C)NC(=O)COCc1cccnc1)OC 19129,c1(NCC(=O)NCC2C(NC(C3CC(SC)C3)=O)CCC2)c(F)cccc1Cl 19130,N1(C(C2(CC#C)CCOC2)=O)CCCC(CNC(C2(C#N)CCC2)=O)C1 19131,c1(COC)nc(NCC2COC(C)(C)C2)cc(=NC2CCC(F)(F)C2)[nH]1 19132,CN1CC(NC(=O)CC2CN(C(C3CC4(CC4)C3)=O)CCO2)C2(CC2)C1 19133,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)cc(C)cc2C)=O)C3)C(=O)OC1(C)C 19134,N1(C(c2c(C)c[nH]n2)=O)CC(C)CN(C(=O)CC2(C#N)CCCCC2)C(C)C1 19135,c12cccc(c1F)-c1csc(n1)NC2=O.C1(OCC)CC(SC)C12CCC2 19136,C1(CNC(c2c(CC)onc2)=O)(NC(C2CCC23CCCO3)=O)CCCCCC1 19137,CC(CC(=O)N1CCCCC(NC(=O)CCCN2C(=O)CCC2=O)C1)C(F)(F)F 19138,C1(NC(c2cc(=O)cc[nH]2)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CCC1CO 19139,CC1CCCN(C(=O)CC2CCCCCC2)C1CNC(=O)CC1CCC2CC12 19140,CCC(C(=O)OC)C(=O)N1CCN2C(C1)C(=O)NCC=CCC2=O.OC 19141,c1(CNC(=O)NC(c2cn(C)cn2)C)csc(-c2cnn(-c3ccccc3)c2)n1 19142,N1(C(CSCC=C)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 19143,c1(OC(CNCC)C2CC2)nccc(C(=O)NCCC2C(OCC)C2)n1 19144,CCCC(C)CCNC(=O)CCOC1CN(C(=O)CC2CCOC2(C)C)C1 19145,Cn1c(N2CCC(C3CC3)C2CNC(=O)C2CC2)c(C#N)c(=O)n(C)c1=O 19146,c1(C(N2CCCC2C(C)C)C(=O)OCC)ccc(OC)cc1 19147,C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CC(C)N(C(c2cc(C3CC3)[nH]n2)=O)CC1 19148,CCC(C)(COC)C(=O)NC1CCCC(CNC(c2cccc(NC)n2)=O)C1 19149,c1(OCCC)ccc2c(c1)CCC2NCC(=O)Nc1ccnc(Br)c1 19150,CC(C)(CNC(=O)CC(=O)NC1CC1)C(=O)NCCS(C)(=O)=O 19151,C1(C(=O)NCCC(CNC(=O)C(C)(C)C(N)=O)OC)CC12CCCCC2 19152,CN1CCN(C(c2ccc(C(F)F)nc2)=O)C(CNC(c2ccsc2C#N)=O)C1 19153,C(=O)(CCCCCN=[N+]=[N-])N(c1cn(-c2c(C)c(C(F)(F)F)ccc2)nn1)C 19154,c1(C(=O)Nc2scc(C3C(C)(C)CO3)n2)ccnc2ccc(N)cc12 19155,c1(NCC=C=C)[nH]c(=NCCC(C)n2cccn2)nc2ncn(C)c12 19156,Cc1nc(-c2ccco2)ccc1C(=O)NCC1CN(C(=O)C(C)(C)O)CC1C 19157,C(CCN(C)C)(CN=c1[nH]c(=NCc2csc(C#N)c2)[nH]c2cc[nH]c12)OCC 19158,N1(C(CSC(C)C)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19159,c1(CNC(C(C)NS(CC)(=O)=O)=O)ccc(CNC(=O)C(C)OC(C)(C)C)cc1F 19160,C1(C(N2CCCOCC2)=O)CCCS(=O)(=O)C1.C12CC(C1)C(=O)N2 19161,C1(C(=O)Nc2cc(C(F)(F)F)cc(F)c2)CC2CCC1N(C(=O)COC1CCC1)C2 19162,C(=O)(CCC(=O)NN(C)C)N1C(CNC(C2CCN(CC)C2)=O)CC(O)C1 19163,N1(C(C2N(C(C)C)CCC2)=O)CCOCC(C(=O)NCCS(N)(=O)=O)C1 19164,C1(C)(C(=O)NC2CCN(C(C)C)C2)C=CCN1C(c1cc(Cl)cs1)=O 19165,c1(C(N2C(C)(CNC(C3CC(C(C)(C)C)C3)=O)CCC2)=O)cc(F)c(O)c(Cl)c1 19166,c1(C(=O)Nc2c(=NC(c3ncc(C)c(O)c3)=O)[nH][nH]c2)cccc(Cl)c1[N+](=O)[O-] 19167,C1(CC)CN(C(C2C3CC4C(C3)C24)=O)CCN1C(c1cnn(CC2CC2)c1)=O 19168,N1(C(c2cc(C)c(O)nc2)=O)C2COCC1CC(NC(C1(C)CC1(F)F)=O)C2 19169,c1(CN2CC(C3N(C(C(C(C)C)C)=O)CCC3)(O)C2)ccn(C=O)n1.C(C)(C)(C)O 19170,Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3nccn3C)C2)c1N 19171,C1(C(=O)NC23CC(NC(C(C)O)=O)(C2)C3)(N(C)C)CCS(=O)(=O)C1 19172,CC1CCc2sc(C(N3CC4CCCC3C4NC(C3CCCC(C)C3)=O)=O)cc2C1 19173,C12(C(=O)NC3C(CNC(C(C)Cc4cccnc4)=O)CC3)C3C4C1C1C2C3C41C 19174,N1(C(CC2(NC(CCNC(C)=O)=O)CCC2)=O)CCC(C)C(O)C1 19175,C1(C(C)NC(C(C)OCCCC)=O)CCCN(C(c2cccs2)=O)C1 19176,c1(C(N(C2CCCCC2)CCNC(C(C2CCOC2)OC)=O)=O)c(C)ccn1C 19177,C1(NC(c2ccnc(Cl)c2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2C1 19178,C(CN=c1nc(-c2cccs2)[nH]s1)NC(CCOCCCOC)=O 19179,c1(C(=O)NC2(C)CN(C(=O)C=CS(C)=O)C2)ccc(F)c2ccoc12 19180,N(C(=NCCC12CC(C1)C2)NCC1CC(C(N)=O)C1)CC(C)C 19181,C1(C(C)O)CCC(NCCC2(C(C)(F)F)CCC2)CC1 19182,c1(OC)ccc2cc(C(=O)NC3(CO)CCN(C(=O)C=CC=C(Cl)Cl)C3)[nH]c2n1 19183,C1(NC(CC=C)=O)CC2CCC1N2C(=O)Cc1csc(C(C)(C)C)n1 19184,c1(N(CC)Cc2cccc(N)c2)cc(N2CCOC(c3nncn3C)C2)ncn1 19185,CC(C)C(C(C)NC(c1csc(Cl)c1)=O)NC(c1sccc1C1CC1)=O 19186,C=CC1COCC1NC(=O)C(C1(C)CC1)NC(=O)C(C)(C)CC 19187,c1(N(C(C(C2CCOC2)OC)=O)CCN(C)C)n[nH]cc1COCC1CCC1 19188,N1(C(c2ccn(CC)n2)=O)CCCC2(CCC2NC(C2OCCN(C)C2=O)=O)C1 19189,CCCCCCCCC(=O)NCC(c1ccccc1)CNC(C1(CC)CCC1)=O 19190,c1(-c2onc(COC(C)C)n2)ccc(OC(F)(F)F)c(Cl)c1 19191,N1(CC(=O)NC2CCC(NC(c3cncc(SC)c3)=O)C2)CCC(=O)NC1=O 19192,c1(CC(=O)NCCCOCCCNC(C(CC(=C)C)C)=O)cccc([N+](=O)[O-])c1 19193,C1(CNC(c2c(C)scc2)=O)CCCC(CNC(=O)C(C)(C)F)C1 19194,c1(C(=O)NCC(CC)(CC)NC(CSCCCC)=O)cncc(S(C)(=O)=O)c1 19195,c1(CCC)cc(C(=O)N(CCC(=O)NC2CC(CO)C2)CC2CC2)no1 19196,N1(C(C(CC)F)=O)CCC(C)C(NC(c2ccn(C3CCC3)n2)=O)C1 19197,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2C(c1coc(C(F)F)n1)=O 19198,C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2ncccc2N)=O)CC1 19199,C(=O)(C(F)C(F)(F)F)NCc1c(CN(C)C(C2CCS(=O)(=O)N2)=O)cccc1 19200,C(=O)(NNc1cc(F)c(F)c(F)c1Br)C1=C2C(CN(C)N(C)N=C2)CO1 19201,CC1CCN(C(c2cc(CNC(=O)CC3=CCCC3)no2)=O)CC1(C)C 19202,C12(C(N3CC(O)(CC)C3)=O)CC(C)(CN1C(C1NC(=O)OC1C)=O)C2 19203,C(C(C)(C)C#CC(=O)N(CC(O)COC)C)NC(CS(CC)=O)=O 19204,S(=O)(=O)(c1cccc(=NCC2(C3CCCO3)CCC2)[nH]1)NC(CC)CN(C)C 19205,CCC(CC)C(=O)N1CC(N(c2coc(-c3cccc(F)c3)n2)CC2CC2)C(C)C1 19206,C(=O)(CCC(CC)CC)NC(C(=O)N(CCCC#C)C)CCCOC 19207,C(=O)(C(C)C(C)(F)F)N(CC(C)O)CCNC(c1n[nH]c(C(C)C)c1Br)=O 19208,CN1CCN(C(=O)CCc2cccnc2)CC1C(=O)NC1(CO)CCOC1 19209,N1(C(CCCOCCOC)=O)CC2CCC1C(NC(=O)C(C(C)(C)C)C1CC1)C2 19210,Cc1ccccc1C(=O)NCCNC(CC(N)=O)=O.C12CCCN1C2=O 19211,c1(C(N2CCCC(C(=O)Nc3[nH]nc(C(N)=O)n3)C2)=O)ncc2[nH]ncc2n1 19212,Cc1noc(C2CC(NC(=O)CCn3cnnn3)C2)n1 19213,C1(N2CCC(NC(c3c(C(C)C)ncs3)=O)C2)CCN(c2ncc(Cl)cn2)CC1 19214,CS(=O)(=O)CCC(=O)N1CCC(C2CCCN2C(c2ccoc2Cl)=O)CC1 19215,C1(NC(C=CC)=O)CN(C(C2CSCN2C(C)=O)=O)CCC1F.c12ccccc1S2 19216,C(=O)(C(C)CNC(=O)C(Cn1ccnn1)NC(=O)CCn1cncn1)NC 19217,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19218,C(=O)(C(F)CCC(C)C)NC12C(NC(C3N(C(CC)=O)CSC3)=O)CC(CC1)C2 19219,C12(C(N3CCC(C)(NC(=O)CCN4CCOCC4)C3)=O)CC1CCC2(F)F 19220,C1(C(=O)NCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19221,N1(C(c2csc(C)c2N)=O)CC=C(CCNC(C2(F)CCS(=O)(=O)C2)=O)CC1 19222,CCCC(CCCNC(=O)C(C(C)O)NC(C)=O)NC(=O)CC1CC1.C(C)(C)(C)O 19223,CS(=O)c1cccc(C(N2CCN(C(=O)CS(N)(=O)=O)C3(CC3)C2)=O)c1 19224,C(CC(C)(C)C)(C(=O)N1CCC(C(=O)OC)O1)N(CC(N)=O)C 19225,c1(C(N(CC(C)CNC(=O)Cc2cc[nH]n2)C)=O)ccc2c(n1)NCC2 19226,C1(N(C(C)C)C(c2ccc(C3CCCC3)cc2)=O)CCCN(Cc2cnoc2)CC1 19227,c1(NCC(CCC=C)(C)C)ncc(S(=O)(=O)NCC(c2cnn(C)c2)O)cc1Cl 19228,c1(C(=O)NCCC2(C(=O)NC(C#C)C(C)OC)CCCC2)c(C)cccc1O 19229,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19230,N1(C(c2c(C)[nH]nc2Br)=O)CCC2(CC(NC(=O)COCC(C)C)CO2)C1 19231,C1(NC(C2(CC(=O)O)CC2)C)CCCC1CCn1cc(CCO)nn1 19232,c1(C(=O)NC2CN(c3ncnc4cc[nH]c34)CC2O)ccc2cc[nH]c2c1 19233,Cc1cc(C)c(CNC(C2CC(n3cc(-c4c[nH]nc4C4CC4)nn3)C2)=O)s1 19234,c1(C(N2CC3(CC(NC(C4CCS(=O)(=O)C4)=O)C3)C2)=O)ccc2nnnn2c1 19235,C(C(=O)NC1C2CC3C1C3C2CO)(C(C)(C)C)N(C)C(=O)OC(C)(C)C 19236,c1(OC)cccc(C)c1CNC(C1CC1NC(c1cc(OC)ccc1F)=O)=O 19237,C#Cc1cn(C)nc1C(=O)NC(C)CC(C)NC(=O)CN(C)C 19238,c1(CC(=O)NCC(CNC(c2cc(C)c(C)o2)=O)F)ccc(F)c(Cl)c1F 19239,N1(C(C(C)NC(=O)NC)=O)CC2CC(NC(c3ccnc(C)n3)=O)C1C2 19240,Cc1nc2ccc(C(N3CCCCC(NC(c4cncc(Cl)c4)=O)C3)=O)cc2s1 19241,N1(C(c2cnc(CCC)s2)=O)CCCC(CN(C(C)C(=O)NC)CC)C1 19242,N1(C(CC(C(C)C)OCC)=O)CCC2CCN(C(=O)COc3cnn(C)c3)CC2C1 19243,C1(C(N2CCN(CC)CC2)=O)CC12CCN(c1ncc(Br)c(C)n1)CC2 19244,CC(C)(C)CC(O)CC(=O)N1CC(CNC(=O)C=Cc2cnc[nH]2)C(C(F)(F)F)C1 19245,C(=O)(CCCCCCN=[N+]=[N-])N1CCN(C(COCCCC#C)=O)CC(C)(F)C1 19246,C1(CC=C)(C(=O)NC2(C3CCCO3)CC2)CCCN1C(C1CC2(CSC2)C1)=O 19247,N1(C(C(C)CC)=O)CC(O)CC1c1cccs1.C12CC(C1)C(=O)OOC2=O 19248,C1(NC(CC2CC(C)C2)=O)CCN(C(=O)CC2C=CCC2)CC1CO 19249,N(C(C)S(=O)(=O)c1ccccc1)(CCn1ncc2cc(SC)ccc12)C(C)=O.CC 19250,c1(OC)ccc(C)c(C(N2CCCCC2CNC(=O)CN2CCCC2CO)=O)c1 19251,C1(NC(=O)CSCCCC(=O)NCCCN2CCCC2=O)CC(CO)C12CCC2 19252,Cc1cc(N)cnc1CNC(C1N(C(C2CC(=O)CCO2)=O)CCC1(C)C)=O 19253,C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C(NC(CCNC(=O)NC)=O)C1 19254,Cc1cnc(C(N2CCC(NC(=O)CC(C)Cn3cccn3)C2CO)=O)c(C)c1 19255,CC(CC(C)(C)C)C(=O)NCc1cc(C(=O)NCCCC2(C)CC2)n[nH]1 19256,CC1CCN(C(c2cn(C3CC3)nn2)=O)CC1CC(=O)N(CC(F)F)C1CC1 19257,C(=O)(C(C)(C)C(C)C)N(CC(CNC(Cc1ncc(C)s1)=O)O)C 19258,C(CCCCCNC(C1CCCN1C)=O)N(C(C(F)=CCC)=O)C 19259,C(=O)(CCCCC(=O)NCC12CN(C1)NC2=O)OC.c1(CO)ccc(OC)cn1 19260,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19261,N1(C(C(C)NC=O)=O)CCC2CN(C(c3cnc(O)nc3O)=O)CCC12 19262,N1(C(C(C(C)C)OC)=O)CC(CNC(c2cccc3nn[nH]c23)=O)CC12CCC2 19263,C12(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c3cncs3)CC3CC(CC1C3)C2 19264,N1(C(Cc2c(C)noc2Cl)=O)CCCC(NC(=O)C=CC2CCOC2)CC1 19265,C12(C(=O)NC3CCN(CC)C3=O)CC(CCO1)N(C(=O)CCc1cc(C)[nH]n1)C2 19266,C(=O)(CC(=O)N(C(CNC(=O)C(C)N(C)C(=O)C1CC1)C1CC1)C)OC 19267,N1(C(C(C)NC(C2CCC2)=O)=O)CC2CCCC(NC(=O)C(C)(C)F)C2C1 19268,c1(C(=O)NC2CC(NC(c3cnc(C)[nH]c3=N)=O)C2)nccc2ncccc12 19269,CC1CCCC(C(N2CCOCC2(C)C2CC2)C(=O)Nc2ccco2)C1C 19270,CC1CN(C(=O)C(C)(O)C2CC2)CC2(CCN(c3ncnc4c3CCCC4)C2)O1 19271,C(=O)(CC(F)(F)C(F)F)N.C1(C(=O)NCCCNC2(C)CC2)CCCCC1 19272,C12(C(=O)NCC(C)N(C(C3CC3C(F)(F)F)=O)CC)CC3CC1C2C3O 19273,N1(CC(=O)N(C(c2cn(Cc3nnc(C)o3)nn2)C)C)CCCC(C(C)O)C1 19274,C(=O)(CCC(=O)NN(C)C)N1CCCC(C2(NC(C(CCCOC)C)=O)CC2)C1 19275,Cc1cc(N2CCC3(C)C(F)(F)C3(C)C2)ncc1S(=O)(=O)NCC1CC1C1CCC1 19276,C1(C(F)(F)F)(NC(C2(OC)CCC2)=O)CCCC1.C1(C(C)C)(CC)CC1C(=O)NC 19277,c1(C(N2CCCC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2nonc12 19278,N1(C(=O)NCCCN(C(C)C)C)CCS(=O)(=O)CC1c1ccc(C(F)(F)F)cc1 19279,N1(C(C(=O)N(CC(CC)(C)CO)C)=O)CC=C(CO)CC1.n12cc(nn1)C2 19280,C(=O)(C(CC1CCCC1)NC(=O)C(CO)OC)NCC#CCC 19281,C(=O)(C#CC1CCCO1)N1CCC(NC(c2c[nH]c3nccc-3c2)=O)CC1 19282,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19283,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 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19353,C1(C(=O)NC2(CNC(c3c[nH]nc3-c3ccoc3)=O)CC2)OCCOC12CCC2 19354,O=C(CC1CCOC1=O)NOCCOCCNC(C1CC1C(F)(F)F)=O 19355,C(C(C)(C)C(=O)NCC1CCC(CC)CC1)NC(CCSCCC)=O 19356,O=C1NCCc2cc(C(c3cccnc3)NC(c3cnn[nH]3)=O)ccc21 19357,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(CO)ccc2Cl)=O)C1 19358,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19359,CC(C(=O)NCC1(C)CCCN1C(=O)CCCC1CC1)S(N)(=O)=O 19360,CC(=O)CC(C)(C)C(=O)NCC1(CNC(=O)CCCn2ccnc2)CC1(F)F 19361,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19362,C(=O)(CC(C)CNC(=O)CCOCCOC)N1CCC(CC#C)CC1 19363,c1(C(N2CCC(C)(C(N(C)Cc3ccn(CC)n3)=O)C2)=O)ccc(C)cc1C 19364,C1(C(=O)NCC(=C)C)CC2CC1CN(C(=O)CCC1OCCO1)C2 19365,N1(C(C(C)=CC(C)(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCc1cncs1 19366,N1(C(Cn2c(C)cc(C)n2)=O)CCN(C(c2n[nH]c(C)c2O)=O)CC(CO)C1 19367,c1(CC)c(C(=O)N(C)CCNC(c2cn(C(C)(C)C)nc2C)=O)nnn1C 19368,c1(OC)ccc(C(=O)NC(C)CC2CN(C(C3(n4ccnn4)CC3)=O)C2)cc1O 19369,C1(NC(C2C(C=C)C2)=O)CCCCN(C(=O)C=Cc2ccc(C)o2)C1 19370,N1(C(CCC)=O)CCN(CCC2(C(=O)NC)CC2)CC1c1ccccc1 19371,N1(C(c2n(C=C)ncc2)=O)CCC(CNC(=O)CC(C(F)(F)F)OC)C(F)(F)C1 19372,CC1(NC(c2cc(C3CC3)ns2)=O)CCN(C(C2CCCC(F)CC2)=O)CC1 19373,C1(C(=O)NC(C(=O)NCC(=O)OCC=C)CC2CCC2)CCCCCCC1 19374,N1(C(C(c2ccccc2)(C)NC(C2(N=[N+]=[N-])CC2)=O)=O)CC=CC(O)C1 19375,c1(CC)onc(OC(C2CN(C(=O)Cc3ccc(C4CC4)o3)CC2C)=O)c1C 19376,C(C(O)C(=O)N(CC(C)N(C(=O)C(CN(C)C)N(C)C)C)C)=CCCC 19377,c1(C(=O)NC2CCC(C(N(CC)CC3CCCO3)=O)CC2)nnc(O)nc1O 19378,c1(CC)nc(C)ncc1C(=O)N(CC(C)NC(c1cn2ccsc2n1)=O)CC 19379,CCC(CC)(C(N)=O)NC(=O)C(C)N(C)C(C1CC(=O)CC(=O)C1)=O 19380,C(C)(C(C)CC(C)C)(c1n(CC=C)nnn1)NCc1ccc(COC)o1 19381,c1(OC)cc(C(=O)NCCC2CCN(C(c3ccc(Cl)cn3)=O)CC2)nc(C)c1 19382,C1(N(C(Cc2nc(C)sc2)=O)CCO)CCN(C(=O)CC2(O)CCOC2)CC1 19383,Cc1nc(NCC2CCCCN2C(C23CCOC2CCOC3)=O)c(Cl)cc1C#N 19384,C1(CNC(COCCCC)=O)CC2(CCN(C(c3cc(C4CC4)ns3)=O)CC2)C1 19385,N1(CCCCCOCCOC)CC2CCC(C(=O)NC3CCN(C)CC3)CC2C1 19386,c1(CC)nc(C(=O)NC(CNC(C2CCOC2)=O)C(C)C)c(N)s1 19387,c1(CC(=O)NCCCOCCN(C(C2(CCC=C)CC2)=O)C)csc(S)n1 19388,c1(CC)ncc(CNC2CCN(C(C3CC3(F)F)=O)C2)s1 19389,C1(C(=O)NCC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19390,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19391,c1(C(C)C)nnc(C=CC(=O)NC(C2CCCC2)CNC(C2CCN(C)C2)=O)o1 19392,Cc1cccc(C)c1NC(=O)C(N1CCCC(c2ccon2)C1)C1CCCOC1 19393,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(C(=O)OC)CC2)=O)C2C1C2)=O 19394,c1(C(=O)Nc2cn(CC(C)C#N)nn2)cccc(-c2conc2C)c1 19395,C(C)(CC(=O)N1CC(NC(c2cnc(Cl)s2)=O)C1)(C(F)(F)F)N(C)C 19396,C(=O)(C#CC1CCCCO1)NCC(C1CCN(C(=O)Cc2cn(C)nn2)CC1)C 19397,C1C(c2ccccc2)C(=O)N1.C1(CN(C)C)CCN1C(c1cnsn1)=O 19398,N1(C(=O)Nc2c(C)cc(Cl)cn2)CCCc2ncccc2C1C 19399,S(=O)(=O)(CCC(=O)N1CCC(CC(=O)NC2CC(N3CCCC3)C2)CC1)NC 19400,c1(OC)ncc(C)cc1-c1ccc(C2(NC(c3c(Cl)cnn3C)=O)CCC2)cc1 19401,N1(C(=O)OC(C)(C)C)CCc2nc(C(=O)NC3CCOCC34CCC4)ncc2C1 19402,C1(C2N(C(c3conc3C(C)(C)C)=O)CCC2)CCCN(C(=O)CC2CSC2)C1 19403,C1CC2(C1)CC(O)C2.C(=O)(CC(c1cccnc1)NC(N(CC)CC)=O)O 19404,c1(CC)ccnc(C(N2CCN(C3CN(C(=O)C(F)CC4CC4)C3)CC2)=O)c1F 19405,N1(C(Cc2n(C)cnc2)=O)CCN(CC(C2CCC2)NC(=O)CC2(O)CC2)CC1 19406,c1(C(=O)NCc2c(CCNC(C=CSC)=O)ocn2)cccc2c1OCCN2 19407,C1(C2CN(C(c3ccnc(Cl)c3O)=O)C2)(NC(CCC(=C)C)=O)CC1 19408,c1(CC)nn(C)c(Cl)c1C(N1CCC(C)(CNC(C2CC23CCC3)=O)C1)=O 19409,c1(OC)ccn2ncc(C(=O)N(C3CCN(C(c4ccc(Cl)cc4)=O)C3)C)c2c1 19410,C(C(=O)NC(C)C(=O)N(c1ccnc(O)c1)C)(C(C)C)NC(=O)OC 19411,C12(Nc3cc(NCc4ccn(C)c4)ncn3)CCC(CO)(CC1)C2 19412,CCC(CC(=O)N1CCC(C(C)(C)NC(c2ncc[nH]c2=O)=O)C1)C1CCC1 19413,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19414,N1(S(CC(=O)Nc2c(C#C)nccn2)(=O)=O)Cc2ccccc2C1C(=O)OC 19415,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(CCC(CC)OC)=O 19416,S(=O)(=O)(c1ccc2ccccc2c1)N1CC2N(C(=O)C(F)Cl)C(COC2)C1 19417,N1(C(CC(C)OC)=O)CCC(NC(=O)CC23COCC(C2)C3)C1C 19418,C12(CC(=O)NCCCCCN(C(C3CC(SC)C3)=O)C)COCC(C1)C2 19419,C1(CNC(CC(CNC(=O)CCN2CCOC2=O)OC)=O)CCCCC1(C)C 19420,c1(C(N(C(CNC(C2(C)C(C(=O)OC)C2)=O)C)C)=O)cc(-c2ccncc2)on1 19421,C(=O)(C(C)CC(C)(F)F)NCC1(C(C)(C)O)CN(C(C=CSC)=O)C1 19422,C1(CNC(CN(CC)CC)=O)C=CCN1C(=O)CC1CCC(C)O1 19423,Cc1cc(C(=O)OC2(C(F)(F)F)CC(CF)C2)cc(Cl)c1Br.C1(=O)CO1 19424,c1(NC)ccc(C)c(C(=O)NCC2COCC2NC(C2(N(C)C)CC2)=O)c1 19425,C12(C(N3CC(O)(C(C)NC(C4CCC(C)O4)=O)C3)=O)CC3CC1C2C3 19426,C1(C(=O)Nc2n[nH]c(-c3ccc(Cl)c(Cl)c3)n2)CCn2c(O)nnc2C1 19427,C1(NC(C(C)NC(N)=O)=O)CCCCN(C(C2CN3CCN2CC3)=O)C1 19428,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(CCNC(c2c(C)sc(Br)n2)=O)C1 19429,C(=O)(C(F)(F)CO)NC1CC(n2cc(C(CCC)=O)nn2)C1 19430,N1(C(C2CN(C(C3C(C#C)C3)=O)CC2C)=O)CCOC2C(O)CC12 19431,N1(C(c2cc(CC)ncc2)=O)CC(C)(C)CC1CNC(C1CCCSC1)=O 19432,c1(C(CCO)NC(=O)NCCc2ncon2)ccc([N+](=O)[O-])cc1F 19433,N1(C(CS(=O)(=O)N(CC)CC)=O)CC2CC1CCC2NC(C1CCN1CC)=O 19434,C1(OCCNCC2(NC(C(=O)OC)=O)CC2)CC2CCC1C2 19435,C(CCC(=O)NC(C)(CNC(=O)CCNC(=O)CO)CC)OCCOC 19436,c1(C2C(C(N(C)CCN(C)C(C3CC3Cl)=O)=O)C2)cccc(F)c1 19437,Cc1ccoc1C(c1nnnn1C1CCCC1)NC(C1CCOCC1)C 19438,C1(C)(C(c2ccco2)NC(C(C)(F)F)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 19439,N1(C(c2cn3c(n2)CCC3)=O)CCCCC2(CCN(C(c3ns[nH]c3=O)=O)C2)C1 19440,c1(C(=O)NCC2CN(C(c3c(C)ncn3C)=O)CC2(F)F)cc(Cl)cc(Cl)c1O 19441,Cc1ccc(C(=O)NCC2CN(C(C3CCCC3C(=O)O)=O)CC2O)cc1C 19442,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3C=CC=CC=C3)=O)CC12 19443,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)NC(c1nc[nH]n1)C1CC1 19444,O=C(CCCCCCCCC(=O)OC(F)F)NCCCn1ccnc1 19445,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19446,c1(C(=O)NC2(CCCNC(C(N)=O)=O)CC2)ccc(C(F)(F)F)cc1 19447,C(=O)(CCC(CC)OC)NC1CCN(C(C(CC)c2ccccc2)=O)C1CC 19448,C1(C(C)C)CN(c2ncc(CO)cn2)CCN1C(c1ccccc1-c1nn[nH]n1)=O 19449,Cc1cc(C(=O)NCCNC(C2(N(C)C)CC2)=O)c2ncccc2c1.C1CN1 19450,C=CCC(CC)N=c1[nH]c(N2CCC(OCCO)C2)nc2ncn(C)c12 19451,C1(CN(C(=O)CCC)CC)CCN(C(=O)C(O)C2CCC2)CC1 19452,C(=O)(C(F)(F)C(O)C(C)C)N1CCCCC(OC2CN(C(CS(=O)(=O)NC)=O)C2)C1 19453,C1(CNC(CN(C)CC)=O)CCOC1C(=O)NC1CC(O)C1 19454,N1(C(C(=O)NCC(F)F)=O)CCCC2(C=CCO2)CC1 19455,N1(C(CCC#C)=O)CCN(C(C(c2ccc(Cl)c(Cl)c2)CO)=O)CC(O)C1 19456,c1(C(=O)NC2CCCC(N(C(CC3C(OC)C3)=O)C)C2)ccc(F)c(C#N)c1 19457,C1(C(N2CC(O)(CCC)C2)=O)CCCCCCN1C(C1CN(C)CCN1C)=O 19458,C1(NC(=O)COc2ccncc2)CCC2CN(C(C3CC(CC4CC4)C3)=O)CC12 19459,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19460,c1(N2CCN(C(c3cncc(Br)c3)C(=O)NC)CC2)cc(C#N)ccc1F 19461,C1(N(C(c2c(CCC)n[nH]c2)=O)C)CN(C(C2C(C)(C)C2(C)C)=O)CCC1O 19462,CC1(CC(=O)NCCOCCN2CCOCC2)OCCc2sccc21 19463,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19464,c1(NC(CC#C)CSC)ccc(C(F)(F)F)cc1I 19465,c1(C(=O)OCC)ccc(N(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)nc1 19466,C12CN(C(=O)CC(OC)OC)CCN1C2.c1(SC)cc(Br)ccc1C(=O)OC 19467,C(=O)(CN1C(=O)CSc2ccccc21)N1CCC(NC(C2C(C)CCC2)=O)C1 19468,c1(C(=O)NCCCNC(C2CC(OCC)C2)=O)cccc(OC)c1 19469,N1(C(C2(CC)CCC2)=O)CCC(C(C)C(=O)N(C)C(C2(C)CC2)C)C1 19470,O=C1CCC(C(N2CCN(C(c3cn(C4CC4)cn3)=O)C(CCO)C2)=O)CCO1 19471,c1(CC)cc(C#N)nc(N(C2CCCN(C(c3cnc(C)[nH]c3=N)=O)C2)C)n1 19472,C1(CC)(CNC(c2ccc(C(F)(F)F)cn2)C)CCOCC1 19473,c1(C(=O)NC(C2CCCN(C(=O)COC3CCOC3)C2)C)ccc(C2CC2)nn1 19474,C#CC1CC2(CC2)CN1C(C1CC(C)(C)CN1C(C1CCCC2(CC2)C1)=O)=O 19475,C1(N(C(=O)CC#N)CCOC)CCCN(C(=O)C(c2cc(C)[nH]n2)N(C)C)C1 19476,c1(NC(C(C)NC(C(C)OC)=O)=O)cnc(F)nc1 19477,C1(CNC(CC(C)C)=O)C(O)C(O)CN1C(=O)CCC#N 19478,C12CCC(CC1)C(=O)N2C.N1(CC)CCCC(CC(C)CO)C1 19479,N#Cc1ccc(C=CC(N2CC3(CCN(c4cc5ncnn5cn4)C3)C2)=O)cc1 19480,c1(C(=O)NC(CC)CN(C(=O)C(O)CC)C)ccc(C(F)F)c(F)c1 19481,CC1(F)CCN(C(=O)CN(C2CC(C#N)C2)C(=O)CC2CCCC(=O)C2)CC1 19482,c1(C(N(C)CCNC(=O)CC2CCC(F)(F)CO2)=O)cc2ccc(O)cc2n1C 19483,N1(C(CSC2CC2)=O)CCC(NC(c2c(C)n[nH]c2C)=O)CC1C.C1(=O)CN1 19484,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19485,C1(NC(CCCCCSC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(F)F 19486,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)C(C1(O)CCCC1)F 19487,CN1C(=O)CC(NC(N2CC(CC(F)C(=O)O)C2)=O)C1Cc1ccccc1 19488,Cc1c(Br)cc(C(N2CC3CC3(CNC(c3cnc(Cl)cn3)=O)C2)=O)cc1Br 19489,C(=O)(C(O)CC(N)=O)N1CC2C(C(N(C(CC)C(=O)OC)C)=O)C2C1 19490,c1(N2CC(NC(c3ccc(OC)nc3)=O)C(F)CC2)ncnc2c(Br)cccc12 19491,N#CC1(C(=O)NC(CC(=O)NCC2CCCOCC2)C2CC2)CCCC1 19492,C1(NC(c2ccc(Cl)cn2)=O)CC12CCC(NC(=O)CCn1cncn1)CC2 19493,N#Cc1ccccc1-n1nnnc1C(c1cnno1)NCCCCc1cccs1 19494,N1(C(C(COC)C)=O)CCN(C)C(CNC(c2ccc(C(N)=O)c(Cl)c2)=O)C1 19495,CC1CN(C)CCC1NC(C1(NC(=O)Cc2ccc(O)nc2)CC(F)(F)C1)=O 19496,CCCCC(CC)CC(=O)NCC1(F)CC2CCC(C1)N2C(C1CC2(CC2)C1)=O 19497,C1(NC(C=CCC)=O)CCCC1C(=O)NCCn1cc(C)cn1 19498,c1(NC(c2cc(CNC(C(n3c(C)ccn3)C)=O)nn2C)=O)cccc(Cl)c1O 19499,C1(CNC(C2C(C(=O)OC)CCC2)=O)COCCN1C(C1(C#N)CCC1)=O 19500,C(=O)(C(CC(N)=O)NC(=O)C(COC)OC)N(CC(CC)O)C 19501,c1(C(N(CCN(C(=O)CC2CC(O)C2(C)C)C)C)=O)cc(C(C)(F)F)ccn1 19502,N1(C(CCC(=O)Nc2nccs2)=O)CC2CCC1CN2C(c1cc(O)ncn1)=O 19503,C1(C)(CNC(c2n(C)ncc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19504,C1(CCNC(=O)C(O)C2CC2)CCCN(C(C2(CO)CCCCO2)=O)C1 19505,c1(CC(N2CC3CC2CN3C(=O)C(F)(F)C(F)F)=O)sc2ccccc2c1C 19506,C1(C(N(CC(CNC(C(C)=C(C)C)=O)(C)C)C)=O)CCCCC(F)(F)C1 19507,CC1C(NC(c2ccc(O)c(F)c2)=O)CCCN1C(c1coc(C(F)F)c1)=O 19508,N1(C(CC(CCC)O)=O)CC2CCCC(NC(c3ccc(F)nc3F)=O)C2C1 19509,Cc1c(C(=O)NCCNC(C2CCC(O)(C(F)(F)F)CC2)=O)cnc2ncnn12 19510,C(CCN=c1cc(C)c(S(=O)(=O)NC2CCCC(O)C2)c[nH]1)(C1CCC1)OCC 19511,c1(N2C(CNC(C3(C(N(C)C)=O)CC3)=O)CC3COCC32)ncc2scc(Br)c2n1 19512,CC1CC(NC(=O)C(CO)NC(=O)C=CC2CCCCC2)CCO1 19513,c1(CC)ncc(C(=O)NCC2CCN(C(=O)C(C)C3(CO)CCC3)C2)s1 19514,N1(C(c2cc(C)nn2C)NC(=O)C(C)c2ccco2)CC(C)(C)CCC1CO 19515,c1(C(N2C3CN(C(C4OCC(C)C4)=O)CC2CC3)=O)coc(=O)c2ccccc12 19516,C1(CCC(=O)NC(C2CCCCO2)C2CCC2)CCCCC1 19517,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19518,N12CCOC(C1)C2=O.C1(OC)(CNC(=O)COc2cnn(C)c2)CCSC1 19519,c1(C(CC)C)nc(C)cc(=NCC2(O)CN(C(=O)C(CO)N(C)C)C2)[nH]1 19520,c1(C(N2CCC(NS(=O)(=O)Cc3ccccn3)CC2)=O)cnccc1Cl 19521,c1(CC(CC2=CCN(C(C3CC(CN(C)C)C3)=O)CC2)=O)ccc2[nH]ccc2c1 19522,CC(C)(C)C(O)C(=O)Nc1cnc(Cl)cn1.c1(C(N2C3CC3C2)=O)ccccc1F 19523,C(CC(C(=O)O)NC(N1CCCC1C(=O)Nn1cc(C2(C)CSC2)nn1)=O)SC 19524,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C)C(C3CC(O)CN3C(C)=O)=O)C2C1 19525,C1(NC(c2c[nH]cc2Br)=O)CC2C1CCN2C(=O)C=C1CCCCC1 19526,N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC(C)C(N)=O 19527,c1(CC2(NC(C=CCN(C(C=CC(=O)OC)=O)C)=O)CC2)ncccc1F 19528,C1(C(F)(F)F)(C(=O)NC(C)CNC(=O)CCCNC(=O)C2CC2)CC2C=CC1CC2 19529,Cc1cc(C(N2CC(C(C)NC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19530,c1(-c2c(CN(C(C(=O)OC)C)Cc3ccccc3)scc2)ccc(C)c(C)c1F 19531,CCC(CC)CCCCC(=O)NC1CC(C(=O)N(C)Cc2cnc(C)s2)C1(C)C 19532,c1(C(=O)OCC)ccc(OC(CN(C(=O)OC(C)(C)C)C(C)C)(C)C)cc1CO 19533,C1(CNC(C=C(CC)CC)=O)CCC(C(=O)N(CCO)CC2CC2)O1 19534,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2cc[nH]c12)=O 19535,C1(C)(NC(C(C)OCC(C)C)=O)CCCCC1C(=O)N(C)CC1CCN(C)CC1 19536,CC1(CNC(C2(C)C=CCC2)=O)CCN(C(=O)C(c2csc(=N)[nH]2)=O)C1 19537,C(=O)(C1=CCOCC1)N1CCC(CCOC)(NC(C2C(C#C)C2(C)C)=O)C1 19538,CN1CC(C(=O)NCC2(C(=O)NCc3ccccc3F)CC2)NC1=O 19539,N1(C(C(C)OCC=C)=O)CCN(C(=O)C(C(=O)OC)OC)C(C)C1 19540,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19541,CN(CCCC(=O)N1CCN(C)CC1CNC(=O)CC1CC(O)C1(C)C)N=O 19542,c1(C(=O)NC2(C)CCN(C(C3(CCO)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19543,c1(CNC(C2(CNC(CCc3onc(C)n3)=O)CC2)=O)cc(O)ccc1F 19544,c1(C(N2CC(CNC(CCCCOCC)=O)(CO)C2)=O)ccc(N(C)C)cn1 19545,N1(C(CCCC#CC)=O)CC(CNC(=O)C(O)CC(C)C)CC(C)(C)C1 19546,N1(C(C(C)SC)=O)CCC2(C1)CN(C(c1c(Cl)nnc(Cl)c1Cl)=O)C2 19547,N1(C(CC2C(C(=O)OC)C2(C)C)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19548,c1(C(C(=O)NC2(CC(=O)OC)CC2)N(CCCOC)C)csc2c(Br)cccc12 19549,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19550,N1(C(c2occ(C)c2)=O)CC(C)(C)CC1C(=O)NCc1ccc(Cl)o1 19551,CC1=NOC(C)(C(=O)N(CC(O)CN(C(=O)CC2CCN(C)C2=O)C)C)C1 19552,c1(CC(=O)NC(CNC(C2CC(C#C)(O)C2)=O)C(C)C)noc(C)c1C#N 19553,C=CCC(C(=O)NCCN(CC(C)O)C(C12CCC(OC)(CC1)C2)=O)C(C)(C)C 19554,CCC(CC(=O)NC1CC(CNC(c2cc(Cl)c(F)cc2F)=O)C1)C(C)C 19555,N1(C(C(C(C)C)SC)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19556,C1(NC(C2CCCC(N(C)C)C2)=O)CN2CCC1(F)CC2.C12CC(C1)CC(=O)N2 19557,Cn1nc(C(N2CCC(F)(CNC(=O)C(O)CN3CCCC3)C2)=O)cc1F 19558,C(=O)(C(F)C1=CCCCC1)N(CCCNC(c1ccc(C(=O)OC)[nH]1)=O)CCC 19559,C(=O)(CCC(F)(F)F)NC1CCCC(CC(=O)Nc2c(C(C)C)nn(C)c2)C1 19560,c1(C(N2CC(C(C)O)C2)=O)ccc(CN2CCCCC2)o1.C1(C(=O)NCC)CC1 19561,c1(CS(N2CC(COC(C)C)C3(C2)CC3)(=O)=O)c[nH]c2nccc-2c1 19562,N1(C(C(C)(C)Br)=O)CC2(CCCN(C(c3cccc4nscc34)=O)C2)C1 19563,C(=O)(C1=CNC2=NCCCN12)N1C(C(C)NC(C23CCC(CC2=O)C3)=O)CCC1 19564,N1(C(CC(CC)C2CC2)=O)CC2CCC(CNC(=O)C(C3CCCCC3)O)(C2)C1 19565,c1(CNC(c2ccc(F)cc2)CN(C)C)cc(N)cc([N+](=O)[O-])c1 19566,c1(C(N2CC(N(C)C(c3cscc3Cl)=O)C2)=O)ccnc2c(F)cccc12 19567,c1(C(=O)NCC2C(C(=O)NC3C(C)CN(C)CC3)CCC2)nccc2[nH]ccc12 19568,C1(NC(CC(=O)NCC)=O)CN(C(c2ccnn2CC)=O)CC12CCC2 19569,N1(C(c2c(C)scn2)=O)CCCC(N(C(=O)Cc2cc(Cl)cs2)C)CC1 19570,n1(CC)ccc(C(=O)N(CC(C)N(C)C(c2cc(C)n(CC)n2)=O)C)cc1=O 19571,N1(C(c2scc(C)c2C)=O)CCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)(C)C)C1 19572,N1(C(=O)OC(C)(C)C)Cc2nccnc2CC1C(=O)NC(C1CCOC1)CO 19573,C12CN(CC1C)CC=CC=CC(=O)NC2.n1(C2CC2)ccnn1.CC=C 19574,CC(N=c1ccc(C#N)n[nH]1)C1CN(C(c2ccc(CC3CCC3)cc2)=O)C1 19575,C1(NC(CN(S(CC)(=O)=O)C)=O)CCCCC1NC(=O)C=Cc1ncco1 19576,Cc1ccccc1N(C(CNC(=O)C(=O)NC1CC1(c1ccccc1)C)C)C 19577,c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)CC)nc(C)c(C)nc1C 19578,CCC(CC(C)C)C(=O)NCC(C)C(=O)N1CC(OC)C1 19579,c1(C(N2C(CNC(C(C(COC)C)C)=O)CCCC2)=O)cc2cn[nH]c2cn1 19580,N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 19581,C1(C)(C(=O)NCC(CNC(c2occ3c2CCC3)=O)OC)CCCNC1=O 19582,N12CC(CC(F)(F)C1)C2=O.n1(CC)ccnc1CNc1ncc(F)s1 19583,C(CCCCC(=O)NC(C)CCN(C(=O)Cc1cc(C2CC2)no1)C)OCC 19584,N1(C(COCC=C)=O)CCC(N(C(=O)CCN2CCCS2(=O)=O)C)C(C)C1 19585,C#Cc1ccc(CNC(N2CC(CC(=O)NC3CC3(C)C)C2)=O)c(F)c1Cl 19586,c1(C(CN(C(C(=O)NC2C(OC)CCC2)=O)C)OC)ccncc1F 19587,N1(C(C(C)N(C(CSC(C)C)=O)C)=O)CCCC(C)(O)C1 19588,c1(C(c2n(CCC)nnn2)NCCC2(OCC)CC2)c(OC)cccc1Br 19589,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19590,CC1CC(CNC(=O)C(=O)NCCc2cccs2)CC(C)C1.C1C(=O)N1 19591,c1(CNC(CCN)C2CCOC2)cc2ccccc2[nH]1 19592,N1(C(c2nccc(C(F)(F)F)n2)C(=O)N(CC)CC)CCC(CO)C(CO)C1 19593,c1(C(=O)NCC(CNC(c2nc(C(C)=O)sc2)=O)CO)nnc(C)cc1O 19594,Cc1noc(C)c1S(=O)(=O)N1CC2CN(Cc3cc(Cl)cnc3F)C2C1 19595,c1(OC)cc(C(=O)NCC2CN(C(C3CC34CC4)=O)CCO2)cc2cn(C)nc12 19596,N1(C(C2(CC)COC2)=O)CCC(O)(C(C)CNC(c2nnn(C)c2C)=O)C1 19597,C(=O)(N=c1ccn(C2CCC2)[nH]1)CCNC(CNC(CC1(C(=O)OC)CCC1)=O)=O 19598,c1(C(=O)NCC2(O)CCCN(C(C3ON=C(CC)C3)=O)C2)cccn2nccc12 19599,N1(CCCOC)CCS(=O)(=O)C(CCNC(C2CCCCC23CC3)=O)C1 19600,CC(C)C(C)CC(=O)NCC1CCC(C(N2CC(OCF)C2)=O)CC1 19601,N1(C(Cn2c(C)ccn2)=O)CC(C)C(NC(c2cccc(N)c2N)=O)C(C)C1 19602,N1(C(CCc2c(C)ncs2)=O)CC(O)(C2(CNC(C3(C)CCC(=O)N3)=O)CC2)C1 19603,c1(NC2(C)CC(CNC(CCc3cncc(C)c3)=O)C2)nc(Cl)ncc1Cl 19604,N1(C(C2C(OC)(OC)CC2)=O)CCC2C(NC(=O)Cc3cn4ccsc4n3)C2C1 19605,c1(C(=O)NCC2CCN(C(C3(C)CC3)=O)C23CCC3)coc2ccc(O)cc12 19606,C1(OC)CN(C(=O)COc2cc(C)on2)CC1C(=O)NC1(CN(C)C)CCC1 19607,c1(C(=O)NC2C3CN(C(C(C(C)C)N=[N+]=[N-])=O)CC2C3)cnnc2ccccc12 19608,c1(C(=O)OC)ccccc1C(N1CC(NC(c2nc(C)c(C)s2)=O)CC1CO)=O 19609,N=c1[nH]c(=NCC2CC(NC(=O)CC3CCCCC3O)C2)[nH]cc1[N+](=O)[O-] 19610,c1(C(=O)NC2(CC=C)CCCN(C(=O)C(C)CC)C2)ncn2c1COCC2 19611,CCC(CN(C)C)CC(=O)NCC1(O)CN(C(=O)CCC(C)N(C)C)C1 19612,c1(OCC(N2C(C(C)C)CC(C(F)(F)F)CC2)=O)ccc(CO)c([N+](=O)[O-])c1 19613,N1(C(CC(CC)SC)=O)CCN(C)C(CNC(C2CN3CCC2CC3)=O)C1 19614,C12(C(N3C(CN(C(CCCC(C)C)=O)C)CCC3)=O)CC=CCN1CCC2 19615,C1(NC(c2c(C)csc2)=O)COCCN(C(c2cn(C(C)C)cc2C)=O)C1 19616,Cc1cc(CNC(c2ccc(Cl)s2)=O)oc1C(=O)NCC1(F)CCCCC1 19617,C(C1CN(C(=O)CN2CC=CC2)CC1C(=O)NC(c1cnn(C)c1C)C)=CC 19618,C1(NC(CC2CCN(C)C2=O)=O)CC2(C1)CC(NC(c1ccc(CO)cn1)=O)C2 19619,C1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2COC)=O)CCc2nn[nH]c2C1 19620,C(C)(C(=O)NOCCC1CC1)(C1CCC1)NC(c1cccc(CC)n1)=O 19621,c1(CC)nccnc1C(=O)NC(CN(C)C(C1CCC1(F)F)=O)CC 19622,C1(CN(CC(O)COc2ccc(F)cc2F)C2CC2)CCOC2(CCC2)C1 19623,Cc1cc(F)cc(C(=O)NCC2CN(C(C3CC4(CC4)CO3)=O)CC2(C)C)c1N 19624,n1(CCC)c(C)cc(C=CC(=O)NC(=O)C(C)CC(N)=O)c1C.C12CCC1C(=O)N2 19625,N1(C(C2CCOC2C2CC2)=O)CCCCCCC1C(N1CCC(O)(CCO)C1)=O 19626,Cc1cn(C)nc1C(=O)NC(CO)C(=O)N(C)Cc1ccnn1C 19627,C(=O)(CCCCC#N)N(CCCNC(C1C(C)CC1C)=O)C 19628,N1(C(c2ccc(OC)o2)=O)CCn2cc(C(N3CCC(F)(F)C(O)C3)=O)nc2C1 19629,C1(CC2N(C(C=C(COC)C)=O)CCC2)COCCN1C(C1CCC1)=O 19630,C#CCC(CC#C)C(=O)N1CC(C)C(NC(c2nscc2C)=O)C(C)C1 19631,C(=O)(C1CCCc2nncn21)NC1C(NC(Cc2c(C3CC3)ccc(C)c2)=O)C1 19632,N1(C(COC)=O)CC2CC1CCC2NC(c1ccc(C(=O)NC2CCC2)o1)=O 19633,c1(C(=O)NC2CC(C)(NC(C(CC)CN(C)C)=O)C2)cc(O)cc(F)c1 19634,N1(CC(c2c(C)ccnc2)=O)CCC(C#N)(C2CCCC2)CC1 19635,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(=O)CC(C)NC(N)=O)CCC12CCC2 19636,C1(OC)CCC2(C(=O)NCC3CCN3C(=O)CSc3cnn(C)c3)CCC12 19637,N#CC1(C(=O)NCCNC(=O)CCN2CCCS2(=O)=O)CC2CCC1C2 19638,C=CC(C)(O)CC(=O)N(C(CCNC(=O)C(O)CCc1ccccc1)C(C)C)CC 19639,CCC(CC1CCCCC1)C(=O)NCC1CC(F)CN1C(=O)Cc1[nH]cnc1C 19640,N1(C(Cc2cc(C)on2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NCC2CC2)C1 19641,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC2CNC(=O)C2)on1 19642,C1(C(C)=O)CNC(=O)CN1CC(=O)Nc1ccc(CO)c(C)c1 19643,C1(F)(CNC(Cc2c(C)nn(C)c2)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC1 19644,C12(C(N)=O)CC(c3nc(CC4CC4)no3)(C1)C2 19645,Cc1cccc(CN(Cc2ccccc2)CC2(c3cscc3Br)CC2)c1C 19646,C=CC1(C(=O)NCCC2CCCN(C(C3CCC3)=O)CC2)CCCCC1 19647,Cn1c(NC(c2ccccc2-n2cncn2)=O)ccc1C=O 19648,c1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)ccc2c(c1)CCCC2=O 19649,C1(CC)CN(C(C23CC(C(F)(F)F)(CO2)C3)=O)CCC1NC(c1cncs1)=O 19650,C1(CC(=O)NCCCCCN(C(=O)CCC2CCCC(O)C2)C)OCCC1(C)C 19651,C(CCCCC(=O)N(C1CCN(C(c2cc(C)co2)=O)C1)C)OCC 19652,c1(C(N(CC(=O)Nc2ccc(C(C)F)nc2)CC#C)=O)[nH]ccc(=O)c1C 19653,C1(C(=O)Nc2ccc(N3C(C(C)C)CCC3)nn2)CC2CCC1CC2.CO 19654,C(=O)(CC(C)(C)C(F)F)NCCCC(C)NC(=O)CC1CCS(=O)(=O)C1 19655,c1(Cn2cc(CCN(CC)CC)nn2)cccc(Br)c1F.c12cccc(c1)CS2 19656,c1(OCC)ncc(C(N2CCC2COC)=O)cc1-c1cccc(C(F)(F)F)c1 19657,C1(C(NOCC(C)C)=O)CCC(C)(C)N(C(=O)C=CC2CCCN2C)C1 19658,C(=O)(CC(C)(C)NC(=O)C(C(C)C)C1CCC1)NC(CC)CSC 19659,C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)COC2(C)CCC2)CCO1 19660,n1(CC(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)CC2)ncn2cccc2c1=O 19661,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19662,Cc1cc(-n2cc(C(C)N(C(=O)C(CO)NC(N)=O)C)nn2)cc(C)c1 19663,c1(OC(C)C)nccc(C(=O)NCC(CO)NC(C2(CO)CCC2)=O)c1F 19664,C1(CNC(c2nnc(CC)s2)=O)CC2COCC2N1C(=O)C=C(C)C1CC1 19665,N1(C(CCOC(C)=O)=O)CCC2(CC(NC(=O)C=C(C)Cl)CO2)C1 19666,C1(NC(CN2CCC(C)C2)=O)CCCCN(C(c2cccc(OC(F)F)c2)=O)C1 19667,C(CNC(C1CC2CC2C1)=O)(CC(F)(F)F)NC(c1cncc(C)n1)=O 19668,C1(NC(c2c(CC)ocn2)=O)CCCN(C(c2cnoc2C)=O)C1 19669,N1(C(COCC(=C)C)=O)CC(C)CN(C(C2CCCCN2CC)=O)C(C)C1 19670,C1(NC(c2cnc(C3CC3)s2)=O)CC2CN(C(c3ccn(O)c(=O)c3)=O)CC12 19671,C1(CC)CN(C(c2cncc(Br)c2)=O)CCN1C(=O)C(F)n1cccn1 19672,c1(C(N2CCC(O)(C(C)NC(C3(C(=O)OCC)CC3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 19673,N1(C(c2cc(Br)ncc2Br)=O)CCC2CN(C(c3cc(O)cc(Br)c3)=O)CC2C1 19674,C1(NC(C(C)C(C)(F)F)=O)CCOC2(CCN(C(C3(n4cccn4)CC3)=O)CC2)C1 19675,C1(C(=O)OC)CCCC12CCNCC2.C(=O)(C(C)NC)N(CC(C)C)C1CC1F 19676,c1(C(=O)NC(COC)CCS(C)(=O)=O)ccc2n1CCNC2 19677,N1(C(C2(NC(c3csnn3)=O)CCN(C)C2)=O)CCC(O)C(O)C1 19678,C1(C(=O)NCC23OCC(NC(c4cn(C)nc4)=O)(C2)C3)CCC(=O)CC1(C)C 19679,C(=O)(C(F)(F)CCC(=O)N(CCCNC(c1cncc(N(C)C)c1)=O)C)OC 19680,c1(C(=O)NC2CC(NC(C(C)CC3CCCC3)=O)C2)ccc2ccc(O)nc2c1 19681,CC1CCCN(C(c2ccc(CO)cc2)=O)C1CNC(c1cc(F)ccc1O)=O 19682,N1(C(C(C)OCC#C)=O)CCCC(C)(CNC(=O)CC2(C)CCCO2)C1 19683,N#Cc1ccc(C(N2CCC(CO)(CNC(C34CCC(CO3)C4)=O)CC2)=O)nc1 19684,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(C)CC2)=O)cc1C 19685,N1(C(CC=CC=C)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1NCCC(C)C 19686,C1(C(N2CCC(OC)C2)=O)CCCC(NC(C2COCC2(C)C)=O)C1 19687,N1(C(C(C)Cc2cnc[nH]2)=O)CCN(C(=O)COC2(C)CCC2)C2COCC12 19688,N1(C(Cn2c(C(C)C)nnn2)=O)CCC2CCC(C1)N2C(=O)CC1CCC2CC12 19689,C(C(C)C(F)C(=O)NCC(n1ccnn1)C)NC(c1scc(CC)c1)=O 19690,CC1C(C(=O)NCCCOC2CN(C(C3OC(C)(C)OC3C)=O)C2)C(O)C(=O)N1C 19691,c1(NC(C2CCCCN2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO 19692,CCC1=C(C(=O)NC2(C)CCN(C(c3cncc4c3CCC4)=O)C2)SCCO1 19693,c1(CC)ncnc(N2CCCC23CC3)c1F.C12CCN(C1)C(=O)N2 19694,C1(C(=O)NCC(CC)NC(c2cc(C(F)F)no2)=O)C2CC2C2CC12 19695,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1ns[nH]c1=O)=O 19696,N1(C(=O)CCC2CC3CCC(C2)N3)CCC2CCN(C(C3(O)CCCC3)=O)CC12 19697,N1(C(c2ncc(C)cc2F)=O)CCC2C(CCCN2C(=O)CC(C)(F)F)C1 19698,C1(C(=O)NCCC2CN(C(c3c(OC)n(C)nc3C)=O)C2)CCCC1S(C)(=O)=O 19699,CCS(=O)CC(=O)NCC(c1ccc(F)cc1)NC(C1(OC)CC1)=O 19700,Cn1nc(C2CCC2)cc1C(=O)NCCCCCCNC(C12CCC1C2)=O 19701,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1cnn(C)c1CC)=O)C2 19702,CC1(C)CCOC(CC(=O)NC2CN(C(C3CN4CCN3CC4)=O)C2)C1 19703,c1(C(=O)NCC(CC=C)NC(c2cscc2C)=O)cc(N(C)C)ccn1 19704,c1(OCC(CC2C(C)C2)(C)C)nc(C2Cc3ccccc32)nn1C1CCCCCC1 19705,c1(OCCC(=O)NC2CC(F)(CNC(=O)NC3CC3Cl)C2)ccccc1F 19706,N#CC1(C(=O)NCC2CCN2C(=O)CCCCCNC(N)=O)CC2CCC1CC2 19707,C(=O)(C(CC(N)=O)NC(=O)COC1CCCOC1)N(C(C=C)C1CC1)C 19708,C(CCN(C(=O)CC1(COC)CC1)C)(C(C)(C)C)NC(CC1CC(OC)C1)=O 19709,CC(CN(C(=O)CN(C)C1CC1)C)N(C)C(C1CC1C(=O)NCCO)=O 19710,c1(C(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)CCC2)cccc2c1CCCCC2 19711,N1(C(C2CCCC(C)C2)=O)CCC(Nc2ncc3c(ncn3C)n2)CC(C)(C)C1 19712,c1(NCCCC=CC)cc(S(=O)(=O)NC(c2ccoc2)C)ccc1C#N 19713,N1(C(C=C)=O)CCN(C2CCC(NC(C3(C)CCC3)=O)C2)CC1 19714,C1(NC(c2cn(C)nc2C(F)F)=O)CCCCN(C(=O)CO)CC1 19715,N1(C(C(CC)OCC)=O)CCc2nc(CNC(c3cn(C)nc3C)=O)sc2C1 19716,C(N=c1ccnc(NC2CCCn3ccnc32)[nH]1)C1CCC(C(F)(F)F)(OC)CC1 19717,C(=O)(C(CC)NC(=O)OC(C)(C)C)NCC(CC)NC(=O)CC1CCC(=O)N1 19718,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19719,C12(CNC(c3c(C)coc3N)=O)CCCC1CCN2C(=O)CN1CC=CC1 19720,N1(C(CCc2cc(C)on2)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19721,C(=O)(C(C(C)CC)N(C(=O)CCN1CCCCC1)C)N(CC#C)C1CC1 19722,C1(NC(c2nnc(CC)s2)=O)CN(C(=O)Cc2ccn(CC)n2)CC1C1CC1 19723,c1(C(=O)OCC)ccc(CNC(C2(C)N(C(C3(C)COC3)=O)CCC2)=O)cc1F 19724,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(c3cc[nH]n3)=O)CC2)CC1 19725,N1(C(CSCCCC)=O)CCC2(CC1)CCN(C(C1CCC3CC3C1)=O)C2 19726,c1(NC(C(C)NC(CCNC(=O)OC)=O)=O)ccccc1NC(=O)NCCO 19727,c1(C(=O)NCC2C(NC(c3c(CC)noc3)=O)C2)c[nH]c2ccc(Cl)cc2c1=O 19728,c1(C(=O)NCC=CCOC)ccc(N2CCCC2CC(=O)Nc2cnccn2)nc1 19729,c1(NC(=O)CC2CC(NCc3cncs3)C2)c[nH]nc1Br 19730,c1(N(C)C)ccncc1CNC(=O)C(O)C1CCC1.c12conc1CNC2=O 19731,C(=O)(C(CCF)NC(=O)COCC1CCOC1)NCc1cc(CC)on1 19732,c1(N(C(=O)C(C2CCC2)NC(=O)C(COC)N(C)C)CC)ccnc(C)n1 19733,Cc1cccc(-c2cncc(C(=O)NCC(O)CCNC(C3CCCS3)=O)c2)c1 19734,CCCC(O)CC(=O)NC1CCC1NC(=O)CNC(=O)C(C)(C)C 19735,CC(C)(C)C(O)C(=O)N1CCCC(O)(CNC(=O)CCC2CCCC(=O)N2)C1 19736,C1(NC(C(CN(CC)CC)F)=O)C2CCCN(CC)C2C1(C)C 19737,c1(C(=O)NC(c2ccc(OC)cc2)CC(N)=O)cccc([N+](=O)[O-])c1N 19738,Cc1cc(CC(=O)N(C(C)CCNC(c2[nH]nnc2C)=O)C2CC2)cs1 19739,C1(CC)CN(C(=O)Cc2cncn2C)CCC1CNC(=O)Cc1ccnn1C 19740,C1(CCC(=O)NCC(C)NC(c2ccoc2C(F)(F)F)=O)CC(C)(C)CO1 19741,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19742,C(=O)(CS(=O)(=O)N(C)C)N(CC(C)C(=O)NCC(CO)NC1CC1)C 19743,c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCC3)CC2)cccn2nncc12 19744,N1(CC(C)C)CC(C(=O)NC2CCCCC2CNC(C2CCOCC2)=O)CC1=O 19745,c1(C(=O)NC2CC(NC(=O)C(F)(F)c3ncccn3)C2)cc2c(Cl)cncc2o1 19746,c1(C(N(CC(C)NC(C(CCC)NC(C)=O)=O)CC)=O)c(Cl)ccc(Cl)c1O 19747,c1(C(N2CC3CC3C2)=O)cnc2ccc(-c3cccc4c3OCO4)cn12 19748,CC1CC(O)CN(C(c2cccc(-c3cccnc3)c2)C(=O)NCC(F)F)C1 19749,C1(CNC(C(C2CCOCC2)OCC)=O)C(C2CC2)CCN1C(=O)C#CC1CCC1 19750,Cc1cccc(Cl)c1N1CC(CC(=O)O)CC1=O.CS(=O)(=O)NC1CC1C 19751,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nnn(O)c2c1 19752,CC(C)CC(C(=O)NC1CCCCC1CO)ONC(=O)C1CCSC1 19753,N1(C(C(=O)NC(C)C)c2ncco2)CCc2ncncc2C1 19754,C1(C(=O)NCCC2CCCN(C(c3scc(C)c3)=O)C2)COC2(CCC2)C1 19755,c1(NC(C(=O)OCC)=O)ccc(NC(=O)CCCCCBr)cc1C 19756,c1(CC)ccc(CC(=O)OC)c(OCCOc2nc(S)n[nH]2)c1 19757,C(=O)(C(CC(C)C)NC(=O)Cc1ccccc1C)N1CC(CC)(OC)C1 19758,c1(C(N2C(C)CC(CNC(C(C)NC(CC)=O)=O)C2)=O)ccc(C(C)=O)cc1Cl 19759,c1(NC2CC(CNC(c3ccc(CN(C)C)o3)=O)C2)ncc([N+](=O)[O-])cn1 19760,C12(C(N(C(C)CNC(C3CCC(C4CC4)CC3)=O)C)=O)C3CCC(CC13)C2(F)F 19761,Cc1sc(O)nc1C(=O)N(C)CC1CCN(C(=O)CCCOC(C)C)C1 19762,c1(C(F)(F)F)c(F)cc(OC2CN(C(c3ccccc3F)=O)C2)cc1F 19763,C1(C(=O)NCCSCC=C)CCC(C2CC2)N1C(c1cc(C#N)c[nH]1)=O 19764,C1(CN(C)C)CCN(C(=O)CC2(Cn3cncn3)CC2)C1.C1(C)(C)CNC(=O)CO1 19765,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19766,C1(CNC(C(C)(C2CC2)OC)=O)CCC2(CN(C(c3ccc(F)cc3)=O)C2)O1 19767,C1(CCC)CN(C(=O)CC(F)(F)F)CC1C(=O)NOC1CCN(CCOC)C1 19768,O=C(C1=CCCC1)NCc1ccc(C(=O)NCC(N2CC=CC2)=O)nc1 19769,c1(N(CCC2CN(C(CNC(COC)=O)=O)C2)C)ccn(CCO)c(=O)c1 19770,c1(C(=O)NCC2CN(C(c3n(C(C)C)ccc3)=O)C2)cc2n(c1)CCC2 19771,c1(OC)cc(CNC(=O)CCOCCCNC(=O)C(c2ccccn2)C)on1 19772,N1(C(CCCSC)=O)CCCC(CNC(c2ccc(F)nc2)=O)CC1 19773,Cc1ccn(CC(=O)N(CCNC(c2coc(CN(C)C)n2)=O)C(C)C)c(=O)c1 19774,c1(C(N2C3C(NC(c4ccc(C)nn4)=O)C(C3)C2)=O)n[nH]cc1[N+](=O)[O-] 19775,C1(CC)CC(O)CN1C(=O)C(CC1CCC1)NC(=O)C=CC(=O)OC(C)(C)C 19776,N1(C(c2c(C)cc(N)cn2)=O)CCCC2(CCCCC2NC(c2cn[nH]c2)=O)C1 19777,CC1CCCN(C(c2cnns2)=O)C1CCNC(c1cnc(S)[nH]1)=O 19778,CCC(CCOC)C(=O)NCC1CC(OC)CN1C(=O)CCSC(F)(F)F 19779,S(=O)(=O)(CCCCCl)N1CC2C(C(N3CCC(CC#C)CC3)=O)(C2)C1 19780,C=CCCCCC(=O)NC(CO)C(C)NC(c1ccnc(OCCOC)c1)=O 19781,N1(C(=O)C=C2CCCC2)CC2C3CCC(C2C1)N(Cc1c(F)cccc1F)C3 19782,CON1CCC(NC(C2CCCCN2C(c2c[nH]c(=N)c(C)c2)=O)=O)CC1 19783,N1(C(c2c(CC)ocn2)=O)CCC(NC(C23CCC(C2)C3(C)C)=O)C(C(N)=O)C1 19784,c1(C(N2CC(NC(=O)C=C(Cl)Cl)C(CO)CC2)=O)ccn2nccc2n1 19785,c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ccc(O)c2)=O)cc2sccc2n1C 19786,c1(-c2n(C(C)COC)nc(C3CC3)n2)ccc2c(c1)NC(=O)C2=O.CC(C)OC(C)(C)C 19787,c1(C(=O)NCC(C(C)C)NC(C2CC(OC)C2)=O)ccc2ccsc2c1 19788,CC1CCN(C(C2CCCN2C(c2ccc(CNC(C3C4COCC34)=O)s2)=O)=O)C1 19789,c1(CSCCC(=O)NCc2ccccc2)ccoc1CN(C)C 19790,S(=O)(=O)(C=Cc1ccccc1)N(CCC(N1CC2(CCS2)C1)=O)C 19791,N1(C(C(COCC)C)=O)CC(O)CC1CC(=O)NCC1(c2ccon2)CC1 19792,C1(NC(C2C(C(C)(C)C)C2)=O)CCCC(C(=O)NCCC2CCCCO2)C1 19793,CCC(C)(CNC(=O)C=Cc1ccncc1)C(=O)N(C)CC1(C)CCCC1 19794,N1(C(C(CCC)C)=O)CC2(CCC2)CC1CNC(C1(NC(C)=O)CCCC1)=O 19795,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19796,N1(C(c2ccc(C)cn2)=O)CCC2CCN(C(=O)CN3CCC(N(C)C)C3)CC12 19797,C1(NC(C2C(C(C)C)OCC2)=O)CC=C(C(=O)NCc2ccncc2)C1 19798,CC(C(=O)NCC1CC2(C1)CN(C(=O)CCc1cccc(C#N)c1)C2)C(C)(F)F 19799,C1(C(=O)NC2CC2)(OC)CCN(C(=O)C(n2cc(-c3csc(SC)n3)nn2)C)C1 19800,Oc1cc(Cl)ccc1CNC(=NCCN1CCCC1)NCC(c1cc[nH]n1)OC 19801,C(=O)(CCC(N)=O)NCC(N1CCC(O)C1)=O.C(C(OC)OC)SC 19802,C1(C(=O)NC2C=CC(C(=O)NCCCc3n[nH]c(C)n3)C2)(OC)CCSC1 19803,c1(OC)ccc(C(=O)N(C)Cc2cc(Cl)ccc2C)c(Br)c1 19804,c1(C(C(=O)OC)NC(CC=C=C)=O)ccccc1C#N 19805,C(C1=Cc2ccccc2OC1)=CC(=O)NC1CCN(C(CC(C)(C)O)=O)C12CC2 19806,C(=O)(C1=CCCCCC1)NCC(=O)NCC1CC[Si](C)(C)C1 19807,c1(C(N2CCCCC(CNC(=O)CC3CC4(CC4)C3)C2)=O)ccc2nsnc2c1 19808,Cc1cc(C)n(CCC(=O)NCC2CCCN2C(=O)CCCN2CCCC2)n1 19809,C(=O)(C(C)CC(C)(F)F)N(C(C)CNC(c1cccc(F)n1)=O)C 19810,C1(C(C(C)C)NC(C2CCCC(NC)C2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)CC1 19811,c1(OC)cc(C(=O)N(C2CCCCC2)CCNC(=O)C(C)C(F)F)ncn1 19812,c1(C(N2CC(CNC(C3CC(OC(F)F)C3)=O)C3(CC3)C2)=O)cccc(F)c1Cl 19813,c1(C(N2CC(O)CC(NC(C3CC(C)C3)=O)C2)=O)cc2nc[nH]c2cn1 19814,Cc1sc(=O)n(CC(N2CCCCC2CCNC(c2ccc(O)nn2)=O)=O)c1C 19815,C1(NC(c2c(C)cn(C)n2)=O)C2COCC1CN(C(=O)C=Cc1ccccc1)C2 19816,C1(C)(C)C(=O)N1.C(Cc1ccco1)(C(=O)OCC)NCC 19817,N1(C(c2cccc(N=[N+]=[N-])c2)=O)CC2CCCCC2(NC(C2CC(CF)C2)=O)C1 19818,N1(C(C(C)CC2CCC2)=O)CCN(c2ncnc(Cl)c2F)C(C)C1 19819,O=C(C1=CC2(CCN(C(=O)C(F)n3ccnc3)C2)C1)NCC1(CC2CC2)CC1 19820,N1(C(c2ccc(-c3ccccc3)cc2)=O)CCN(C(=O)C2=CCOC2)C(CF)C1 19821,C(=O)(C(C)(C)C1=CCN(C(=O)C=CCCC)C1)N(C(C#C)C1CCC1)C 19822,N1(C(C(C2CC2)OC)=O)CCCC(N(C)C(c2cccc(F)c2C(C)C)=O)CC1 19823,c1(CNC(N(C)Cc2c(OC)n[nH]c2)=O)cncc(F)c1 19824,N1(C(c2c(CC)csc2)=O)CCCC(C)(C(N2CCC(CC(=O)OC)C2)=O)C1 19825,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(c1cccc(NC(N)=O)c1)=O 19826,c1(C(N2CC3C(NC(c4cc(C(F)(F)F)c[nH]4)=O)(C3)C2)=O)ccc2ocnc2n1 19827,C1(Nc2c(NC(N3CC(N(C)C)C3)=O)cccc2)CCc2c[nH]nc2C1 19828,N1(C(Cc2c(C)ncs2)=O)CC2CC(N(C(=O)COCCOCCO)C)C1C2 19829,N1(C(C=CC)=O)CCN(C(c2cc(COC)n(C)n2)=O)C(CO)C1 19830,CC1ON=C(C(=O)N2CC(CNC(=O)CN3CCS(=O)CC3)C(C)(C)C2)C1C 19831,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3(O)CCCC3)CC12 19832,c1(C(N2CC(CCOC)N(C(=O)CCOC(C)C)CC2)=O)cc2oc(C)cc2[nH]1 19833,C(c1c(C)cccc1Cl)=CC(=O)N(C1CCN(C(c2cnnc(C)c2)=O)C1)CC 19834,c1(C(N(CC(C)O)CCNC(=O)C=CC(=O)NC2CC2)=O)cccn2c(O)nnc12 19835,N1(C(c2cn(CO)nn2)(C)C)CC(c2ccccc2)C(c2ccccc2)C1.C(CO)C=O 19836,Cn1cc[nH]c(=NCC2(CC3CCCCC3)COC2)c1=O 19837,C12(C(C)NC(c3n(C(C)C)cnc3)=O)CCCCC1C2 19838,O=C1CCOCCN1CCOC.C12COCCN1c1cc(ncn1)Cn1cc2nn1 19839,C(CC(C)C(=O)NCC(O)C(=O)NCc1ccncc1Cl)=CCC 19840,C1(COC)(NC(c2ccc(Br)o2)=O)CCN(C(c2ccc(Br)o2)=O)C1 19841,c1(C(=O)NC2CN(C(C3CN(C(=O)NC)C3)=O)C3C2C3)cccc2ccn(C)c12 19842,n1(CC)cncc1C(N1CCCC1Cc1cn(C(c2nnc(C)o2)C)nn1)=O 19843,CC1(C)CC(NC(C2(CCF)CC2)=O)CN(C(=O)CCc2cscc2Br)C1 19844,Cc1c(Cl)nc[nH]c1=NCC(O)CNC(C1CCCCC12CCC2)=O 19845,N1(C(COCCOC)=O)CC(NC(=O)CC2CCCNC2=O)C(C(F)F)C1 19846,C(=O)(CC1=CCOCC1)N1CC(CC)N(C(C2CCC(C(N)=O)C2)=O)CC1 19847,c1(C(N(CC(C2CC2)NC(CCNC(=O)OC)=O)C)=O)cc(C)n(C(C)C)n1.C1CC1 19848,c1(N2CCN(c3cncc(N4CCC(OC)CC4)n3)CC2)ccc2ncnn2c1 19849,O=C(CCC(F)(F)F)NCC(C1CC1)NC(c1cnn[nH]1)=O 19850,c1(C(=O)NCC2(NC(C(c3ccc(F)cc3)C)=O)CCC2)nc(CN)cc(O)n1 19851,C1(NC(c2cccc(CC#N)c2)=O)CCC2CN(c3cncc(Cl)n3)CC12 19852,C1(c2cn(CCC)nn2)CC2(CCC2)C1.C(C)(C)(C(=O)N(C)CC)OC 19853,N1(C(=O)C=CC=C(Cl)Cl)CCC(F)(CNC(=O)C(N2CCCC2)C2CC2)CC1 19854,c1(C(N2CCC3(NC(CCC)=O)C(CC2)C3)=O)cc2c(O)ncnc2cn1 19855,C(C)(CNC(=O)CCOCC(C)C)(CNC(c1cnc(SC)s1)=O)OC 19856,C1(C(N2CC(NC(c3n(C)c(Cl)nc3)=O)C2)=O)CC1C1CCCC1 19857,C#CCC(CC(F)F)C(=O)NC1CCN(C(c2cc(O)nn2C)=O)C(C)C1 19858,CCCC(CCC)C(=O)NC1CCN(C(c2cccc(O)c2C)=O)CC1CC 19859,C(=O)(CN1C(=O)CCc2ccccc21)NC1C(C)CCN(C(C2CC2(Cl)Cl)=O)C1 19860,C(c1cccc(F)c1)=C(C(N1C(CNC(C(N2CCCC(O)C2)C)=O)CC1)=O)F 19861,C1(CNC(C(=Cc2cncs2)C)=O)CN(C(=O)C(F)C(C)(F)F)CC1(C)C 19862,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(=O)Cc2ncccc2F)C1 19863,C1(C(=O)N)CNC(=O)CC1C.C(=O)(CNC(N1CCC1)=O)NCCOC 19864,C1(C(=O)NCCN(C)C2CC2)CC2CCC1N2C(=O)CCCOC(C)(C)C 19865,C1(NC(c2cc(C)oc2C)=O)CC2(CCCN(C(C3(CC(F)F)CCC3)=O)C2)C1 19866,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)CCO3)=O)C2C1 19867,C1(NC(C2CN(C(C)=O)C2)=O)CCC2CN(C(c3c(C(C)=O)coc3C)=O)CC12 19868,C(C(N=[N+]=[N-])C(=O)NCCCCNC(c1csc(C(C)=O)n1)=O)OCC 19869,CC1(C)C(C)(C)C1(F)C(=O)NCCCNC(=O)Cc1cccc(N)c1 19870,C(=O)(CC(C)(C)C)NCCC(C)NC(C1C(CCC)C1)=O 19871,c1(NCCCC)ccccc1C(=O)N(CCCN=[N+]=[N-])C 19872,c1(C(=O)NC2CCCCN(C(C(COC)OC)=O)C2)cccc2c1CNC2=O 19873,CC1(CNC(=O)CC2CCCO2)CN(C(c2ccsc2C(F)(F)F)=O)CCO1 19874,CN=c1[nH]c(=NCC(C)F)[nH]c(=NCCc2ccc3c(c2)CC(C)O3)[nH]1 19875,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2C=CCC2)=O)CC1 19876,c1(OC(N2C(CC(=O)OC(C)C)CCCC2)=O)ccc(C#N)cc1C(F)(F)F 19877,C1(C(=O)NCc2cccc(OC)n2)CC(C)(C)CN1C(=O)C=Cc1ccc(C)o1 19878,C1(n2cc(C(CN(CC)CC)C)nn2)CN(C(c2conc2C)=O)CC1C 19879,c1(C(N2CCC(N(C(=O)CCS(C)(=O)=O)C)C2)=O)ccc2c(c1)OCO2 19880,N1(C(C2(CNC(C3CC3(Cl)Cl)=O)CCCCC2)=O)CCC(F)(F)C(O)C1 19881,c1(C(N(CCCNC(c2c(CC)nns2)=O)C)=O)ccc(-c2cccs2)cc1F 19882,C1(NC(CC(C)O)=O)CC12CCN(C(c1cc(F)c(C#N)c(F)c1)=O)CC2 19883,N1(CCC)CCC(CNC(=O)NCC(C2CCCC2)N(C)C)C1 19884,O=C(C1=COCCO1)NCC1(NC(C2CC3C=CC2C3)=O)CCCCC1 19885,CC(=O)C(C)(C)CC(=O)NC(CCF)C(=O)NC1CC1(C)C(F)F 19886,c1(C(=O)NCCN(C(C(CCSC)O)=O)CC(C)O)cc(OC)cc(C)c1 19887,S1(=O)(=O)c2ccc(C)c(c2)N1.c1(CC)cnc(C(C)=O)s1 19888,C1(CNC(=O)CC(F)(F)F)CC2(C1)CN(C(=O)COCC(F)(F)F)C2 19889,c1(-n2cc(C3C(C(C)O)C3)nn2)ccncc1Br 19890,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 19891,C1(NC(CC(CC)C)=O)CCN(C(=O)CCSCCOC)CC1F 19892,N1(C(C)=O)CC2(CC(S(=O)(=O)N3CC(N4CCOCC4)C3)C2)C1 19893,c1(C(=O)NCC2CC(CCNC(C(C(=O)OCC)F)=O)C2)cc2nc(C)sc2[nH]1 19894,N1(C(C2(C#N)CCC2)C(=O)NCC(F)F)CCN(Cc2ccc(F)cc2)CC1 19895,C=CCCCCCN=c1nc(N2CCC(CO)C(C)(C)C2)c2c([nH]1)CCC2 19896,C(O)(C(=O)O)(C(F)(F)F)Cc1n(-c2c(C)cccn2)nc(-c2cnn(CCO)c2)n1 19897,N1(C(COC)=O)CC2CCC2(CNC(=O)C(C2CCCCCC2)O)C1 19898,C1(C)(CNC(COc2ccc(C)cc2)=O)CN(C(=O)CCCCCF)C(C)(C)C1 19899,C(=O)(C1SCCc2sccc21)NC1CN(C(C(C)(C)c2cc[nH]n2)=O)C1 19900,c1(C(N2CC(CNC(C(C)n3ccnc3)=O)N(C)CC2)=O)cnc2occc2c1 19901,C1(N(C(c2cc(SC)oc2C)=O)C)CN(C(C2(C)C=CCC2)=O)CCC1O 19902,N1(CC)CCCN(C(C2OCCC2NC(=O)C(C2CCCCC2)O)=O)CC1 19903,N1(C(c2cn(CC)nn2)=O)CCCC1C1CCCN1C(=O)C=Cc1nc(C)co1 19904,C(CCC(C)(C)NC(c1sc(C(C)C)nc1C)=O)NC(C(COC)OC)=O 19905,C1(C(N2CC(NC(COC)=O)C2)=O)CCC(O)CN1C(C12CC(C#N)(C1)C2)=O 19906,n1(CC(c2cncn2C2CC2)=O)cnnc1O.c12cn(nn1)C1CN(C1)C2=O 19907,C(=O)(CC(C(=C)C)OCC)NCC(C(N1CCC(C#C)C1)=O)C 19908,CC1CN(C(c2ncccc2C(F)(F)F)=O)CC1(C)CNC(=O)Cn1cncn1 19909,CC1=C(C)CC(C(=O)NCCC(O)CNC(=O)Cn2cc(C3CC3)cn2)CC1 19910,c1(C(N2CCC3(C(CNC(CCC(=C)Cl)=O)C3)CC2)=O)coc2c(OC)cccc12 19911,CC(C)CC(C)(CNC(=O)COC1CCCC(C)C1)NC(C1CC(F)(CO)C1)=O 19912,CCCCC(C(=O)N1C2CCC1CN(C(=O)C(F)(F)COC)C2)C(C)C 19913,CC(C)CC(CC(=O)O)NC(c1cnc(CC2CCC2)s1)=O 19914,c1(CNC(C2C(CNC(C3CCC(CC)O3)=O)CCC2)=O)nnc2n1CCC2 19915,C(CCCC(=O)NC1CC1CNC(=O)C=Cc1ccsc1)NCCC=C 19916,C1(NC(c2ccc(C)s2)=O)COCCC1NC(C1(F)CC=CCC1)=O 19917,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(N(C(=O)Cc2cnco2)C)C1 19918,c1(C(=O)NC2CC(C)(NC(C(C)SCCCC)=O)C2)cc2c(C)[nH]nc2s1 19919,N1(C(C(n2cc(Cl)cn2)C)=O)CCN(CCc2cccc(F)c2)CC(C)(F)C1 19920,c1(C(=O)NC2CCN(C(=O)C=Cc3cccs3)CC2F)ccnc2cc[nH]c12 19921,c1(C(=O)NC2CCN(C(CC(C=C)C)=O)CC2)cc(Cl)ncc1O 19922,C1(C(N2CCC(O)(CNC(c3cc(Cl)no3)=O)C2)=O)CC2CC(C1)CS(=O)(=O)C2 19923,O=C(CC1=CCN(C(=O)CC2CCCCO2)CC1)N1CCCN(C2CC2)CC1 19924,c12ccc-1s2.C(C(=O)NC)OC(=O)N.C1(C(=O)NNC=O)CC1C1CCC1.CO 19925,N1(C(c2cccc(C)c2)=O)CCN(C(C2CCC(C(C)C)CC2)=O)CC1C1CC1 19926,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CC2)C(C(C)C)C1 19927,N1(C(C(CC)C#N)=O)CCC(C2CC2)(NC(=O)C=CBr)C1 19928,C1(C)(NC(C=Cc2nc(C)sc2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 19929,Cn1c(Nc2ccccc2CN2Cc3ccccc3C2=O)nc2cc(Br)ccc12 19930,N1(C(CCC=C)=O)CCC(C(=O)NC2CCC(CCO)CC2)C1CC 19931,C(=O)(CCC(=O)NCC1CC1)N(CCCCNC(C(C)OCC)=O)C 19932,Cn1cc(C(=O)NCc2cn(Cc3ncoc3CNCCO)nn2)c(C(F)F)n1 19933,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 19934,C1(CC)CCC(CNC(=O)CC2CCN2C(=O)Cn2nnc(C)n2)CC1 19935,C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(C1CSC1)=O)C2 19936,C(=O)(C(O)C1=CCCCC1)N1CC(NC(CC(C)O)=O)C(C)C1 19937,c1(C(N2CCC(C(F)(F)F)(OC)C2)C(=O)NCC)ccc(OC)cc1Cl 19938,C1(n2c(-c3ccc(Cc4ccccc4)[nH]3)nc(CCSC)n2)CCOC(C)(C)C1 19939,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(C(F)F)n2)C1 19940,C(=O)(C1=CCCCCC1)N(CCCNC(c1c(C)nc(CCC)o1)=O)CC 19941,c1(CSCC(=O)N(C)CC2CN(C(=O)C(C3CCCCC3)O)C2)ccccc1 19942,N1(C(=O)OC(C)(C)C)CC2CCCCC2(CNC(=O)C(C)n2cnnn2)C1 19943,C=C(C)CC(C(=O)NCC1CSCCO1)NC(=O)C=C1CCOCC1 19944,N1(C(C(=O)NCCC(C)NC(=O)C(C)(C)c2cccs2)C)CCP(C)(=O)CC1 19945,CCCCC(O)C(=O)NC1C2CC(NC(=O)C=Cc3cn[nH]c3)CC12 19946,C1(C(=O)NCC2CC(OC)C2)(NC(c2cnncc2C)=O)CCN(C)C1 19947,Cc1ccc(C(=O)NCC(CNC(c2cn(C)nc2C)=O)C(F)(F)F)cc1CO 19948,N1(C(CC)=O)CCCCC1C(N1CC(CNC(=O)C2=CCCC2)C(C)C1)=O 19949,C(=O)(CCC(F)(F)C(F)F)NC1CCC(CCNC(c2c(C)cnnc2O)=O)C1 19950,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(C1(C(C)C)CCC1)=O)C2 19951,c1(C(C)OC)cn(CC2C=CCN2C(c2cc(C(C)=O)on2)=O)nn1 19952,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(C3(O)CCCC3)=O)C2)CC1 19953,c1(OC)c(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CO)ccnc1Cl 19954,c1(C(=O)NC(CNC(C(C(=O)OCC)(C)F)=O)C)cc2n(c1)CCOC2 19955,c1(C(N2CCC(N)C2)=O)cnc(C)c(CC)c1.CCC(C(=O)NCC)NC(N)=O 19956,c1(CC(=O)N(C2CC2)Cc2cccc(OC)c2)cccc2ccncc12 19957,C(c1ccc2c(c1)OCO2)=CC(=O)OC1COC2CCCC12 19958,C1(CNC(C2COC3(CCC3)C2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 19959,c1(C(=O)NC(C2(O)CN(C(=O)C(C)(F)F)C2)C)ccn2nncc2c1 19960,Cc1nnc2ccc(C(=O)NCC3(CNC(=O)C4CC4)CC3)cc2c1C 19961,CC1CC(CNC(=O)Cc2cscn2)CN1C(=O)CCN1CCCCC1 19962,CCCC(C(=O)N1CCCN(C(c2oc(SC)cc2C)=O)C(C)C1)S(N)(=O)=O 19963,C1(C)(C(=O)NCCCCC(C)C)CCCN(C(=O)CC2(O)CCCCC2)C1 19964,C#Cc1c(Br)cc(N(C2CCCC2)Cc2ccc(F)cc2C)cc1OC 19965,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CC(CC)C(F)C1)C 19966,C(CC(=O)N(CCNC(=O)CC1(C)CCC1)C(C)C)N(CCC)C 19967,CCC(COC)C(=O)NCC(C)(C)C(=O)NCC(C)C(=O)OCC 19968,N1(C(CC=CCC)=O)CC(C)(C)CC1C(=O)NCCC1COCCO1 19969,C1(C(N2CC(O)(CCNC(C3CC=C(C)CC3)=O)C2)=O)CCC(=O)C(C)C1 19970,C1(CCC(C)(C)C)C(=O)N1.C(CCCCNC(C)(C)C)N.C1CCC(=O)C(CC)N1C 19971,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)N(C)C(C1(C)CC2(CCC2)C1)=O)C 19972,CC1CCC(C(=O)NC2CC3(CCC3)C2O)N(C(=O)Cn2cc(CO)nn2)C1 19973,N1(CCC(=O)NC2CCCC(NC(c3ccnc(S)c3)=O)C2)CCNC(=O)C1 19974,c1(C(=O)NC2C(C(=O)NCCN(CCO)CC)CC2)cccc(C)c1O 19975,c1(OC)cncc(C(=O)NCC(C)(CO)NC(=O)Cc2nc(C3CC3)cs2)n1 19976,c1(C(=O)NCCCN(C(=O)CC(C)(C)O)C)c(COC2(C)CCCC2)cnn1C 19977,C1(F)(CNC(C(CC)=CCCC)=O)CCC(NC(=O)CC2(COC)CCCC2)C1 19978,Cc1ccc(OCCC(=O)NC2CCCC2NC(c2cc[n+]([O-])cc2)=O)cc1 19979,c1(CC(=O)NC(CC)CNC(C2(CC3CC3)CC2)=O)c(C)cccc1C 19980,c1(C(=O)NC(C2CCN(C(C3C4CN(C)CC34)=O)CC2)C)c[nH]nc1[N+](=O)[O-] 19981,C1(C(=O)Nc2ccc(CCO)cc2)(NC(C(C)C)=O)CCN(C)C1 19982,c1(C(C(=O)NCC(CCOC)NC(=O)C(C)C)(F)F)ccc(OC)c(OC)c1OC 19983,CC(=O)CCCC(C)C(=O)N(C1CN(C(C2CC(=O)NC(=O)N2)=O)CCC1O)C 19984,C1(C(=O)NCC23OCC(NC(c4ccnc(C)n4)=O)(C2)C3)COCC(C)(C)O1 19985,c1(C(N(CC)CC)=O)ccc(-c2nc(C(=O)NCCC3CC3(Br)Br)cs2)cc1.CC 19986,N1(C(Cc2c(OC)cc(Cl)cc2)=O)CCN(C(=O)C(C)CF)CC1C 19987,Cc1ccc(C(N2CCC(CO)(NC(=O)C(F)n3cccn3)CC2)=O)cc1F 19988,CC(CNC(c1[nH]nnc1C1CC1)=O)C(F)C(=O)N1CCC(F)(F)CC1 19989,C1(NC(C2(O)COC2)=O)CS(=O)(=O)CC1NC(C1CC(O)C1)=O 19990,c1(CCOCCCCCN(C)Cc2cn(CC3CCCO3)nn2)csc(=O)n1C 19991,C#Cc1cn(C)nc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(C1CC1C)C 19992,N1(C(c2n(C(C)C)ccc2)=O)CCCC(NC(=O)C(C)(F)c2ccccc2)CC1 19993,N#Cc1cnc(NC(=O)CC2CCN2C(=O)C=CC2CCCC2)cn1 19994,c1(CC#N)ccccc1C(=O)NCC1CCN(C(=O)CC2CC3C=CC2C3)CC1 19995,c1(OC(C)C(=O)Nc2ccc(Cl)cc2)ccc(O)cc1 19996,CC1(NC(c2ccnc(CNC(c3cncc(C#N)c3)=O)c2)=O)CCCC1(F)F 19997,c1(OC)nc(CCNC(C2CCC(NC(CN(CC)CC)=O)CC2)=O)[nH]c(=N)n1 19998,N1(C(C(C)NC(=O)NC)=O)CCC(F)(F)C(CNC(c2cnnc(O)c2)=O)C1 19999,N1(C(c2c(CCC)cccc2)=O)CCC(N(C(=O)CCC(C)OC)C)C(CC)C1 20000,C(=O)(N=c1ccc(C(N)=O)c[nH]1)C1N(Cc2ccc(C#N)c(F)c2)C2C(C1)C2 20001,C1(C(=O)OC)CCC(C(=O)Nc2cnn(C3CCNCC3)c2)CC1 20002,C1(F)(CNC(c2ccc(COC)[nH]2)=O)CCCN(C(c2nccnc2OC)=O)C1 20003,C(=O)(C1=CCN(C(c2coc(CO)c2)=O)CC1)N1C(C(C)O)COCC1 20004,N1(C(C2C(COC)CC2)=O)CCC2CN(C(C3CC(=O)C34CCC4)=O)C2C1 20005,C(=O)(C(C)(C)C(C)C)N(C1CC1)CC1CCN(C(C=Cc2n(CC)ccn2)=O)C1 20006,C(C(CCC)CCC)ONC(CC1(C=C)CN(C(=O)C(F)C(C)(C)O)C1)=O 20007,N1(C(C(C)OCC2CCS2)=O)CC(NS(=O)(=O)CCOc2ccccc2)C(F)C1 20008,C(=O)(C(C)(C)C1=CCN(C(c2sccc2N(C)C)=O)C1)NC1C(O)CCC(C)C1 20009,N1(C(c2cnc(Cl)n2C)C(=O)Nc2c(C)cc(F)cc2)CCCC2(CCC2)C1C 20010,c1(C(=O)NC2C(NC(Cc3c(CC)con3)=O)CCC2)cc2sc(Cl)cc2[nH]1 20011,c1(C(=O)NC2CC(CNC(CCC(C)SC)=O)C2)cnc2cnccc2c1 20012,C(C(COC)C(=O)NCCCCCN(C(=O)Cn1nccn1)C(C)C)OC 20013,CC1CC2CN1C(=O)C2.C(=O)(CCCn1cncn1)NC1CC(CO)(CO)C1 20014,c1(CC)nc(C(C)NC(=O)CCOC2CN(C(=O)CC=C(C)C)C2)n[nH]1 20015,Cc1cc(F)c(C(=O)NNC(=O)NCc2cn3ccsc3n2)cc1F 20016,CC#CCC(C(=O)N(C(C)CCC(C)C)C)NC(=O)CN1CCCCC1C 20017,C1(NC(C2CC(NC(C3CCC(F)(F)C3)=O)C2)=O)CCCC(F)(F)C1 20018,CC(C)CC(CNC(C1C2(CC2)C12CC2)=O)C(=O)NC(C)(C)CCO 20019,C(c1ccc(OC)c(Cl)c1)=CC(=O)NC(CNC(c1scc(OC)c1)=O)C(C)C 20020,CON(C(=O)c1[nH]ccc1C(=O)NC1(C2CCCCO2)CC1)C(C)C 20021,C1(C(=O)NCCC(C)NC(c2cn(C)c3ccsc23)=O)Cc2ccccc2O1 20022,c1(C(=O)Nc2cccc(NC(C34CC(C(C)(C)C)(C3)C4)=O)c2)ccc(N)c(F)c1 20023,c1(C(=O)NC2CC3(C2)CC3C(=O)NCC23CCCN2CCC3)ccc2cc[nH]c2n1 20024,C(=O)(C1CCc2ccccc21)NC1CN(C(COCCOC)=O)CC12CC2 20025,Cc1cc(-c2ncc(Cl)cc2C(=O)NCCN2CCOCC2)cc2c1NC(=O)CC2 20026,c1(NC(C)=O)cc(F)c(S(=O)(=O)NC(c2ccc(F)cc2)CCO)c(F)c1 20027,CC(N=c1ccnc(Cl)[nH]1)C1CCCN1C(=O)Cc1cnn(-c2ccccc2)c1 20028,C(C(COC)CC(=O)N1CC(F)(C(=O)NCC2CCOC2C)C1)OC 20029,c1(CC(C(=O)NC(CNC(COCCCCC)=O)CC)O)ccc(Cl)cc1 20030,CC1C(NC(=O)CN(C)C)CC2CCC1N2c1ccnc(-c2cccc(Cl)c2)n1 20031,C1(C(=O)NC(CCNC(Cn2nc(C)oc2=O)=O)(C)C)Cc2cc(F)ccc2O1 20032,c1(CNC(c2n[nH]c(C)c2Cl)=O)ccc2nccc(-c3ccc(N(C)C)nc3)c2c1 20033,N1(C(C2N(C(C(CC#C)C3CC3)=O)CCC(CC)C2)=O)CCCCN(C)CC1 20034,CCCC(CCC)CC(=O)N1CC(NC(=O)CCCc2cccc(Cl)c2)C(C)C1 20035,N1(C(CC(CC)C)=O)CCC(F)(F)C(CNC(=O)C2=CCCCC2)C1 20036,C12(CNC(C3C(C)C3C)=O)CCCCC1N(C(=O)COc1ccsn1)CC2 20037,C1(C(=O)NCCCN(C(C2CN(C(C)(C)C)C(=O)C2)=O)C)C2CCCCCC12 20038,c1(NC)cnc(Cl)cc1C(=O)NC1CC1CNC(C1CC1[N+](=O)[O-])=O 20039,c1(C(=O)NCC2(F)CC(Nc3nnc(C)c(C)n3)C2)n[nH]c2ccc(Cl)cc12 20040,C=CC(C)CC(=O)NCC1CCCCN1C(=O)CNC(N)=O 20041,N1(C(C(CC)CC2CCC2)=O)CCC2CCC(C1)N2C(=O)COC(F)(F)F 20042,c1(CC(=O)NC(C(C)NC(CC(=O)OC)=O)CO)cc(F)cc([N+](=O)[O-])c1 20043,CC1C(=O)N(CC(N2CCCCC2C2(NC(c3ccns3)=O)CC2)=O)C(=O)C1C 20044,C1(C(C)C)N(C(=O)C(C2CCCN(C(C3CNC(=O)N3)=O)C2)C)CC1(C)C 20045,n1(CCCOCC)c(N(C)CCOCCCO)nnc1-c1ccon1 20046,Cc1[nH]nc(C(=O)NC(C)(CNc2cc(O)ncn2)C2CC2)c1C 20047,C=CC1(CC(=O)NCC(O)(CO)CO)CN(C(=O)C(C)c2ccco2)C1 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20083,N1(C(N2CCCN(CC(=O)O)CC2)=O)CCC2(CCS(=O)(=O)CC2)C1 20084,c1(CC(=O)NC2C(C)COC2)ccc(S(=O)(=O)N2CCC(O)CC2)cc1 20085,C(=O)(C(C)(O)Cn1cc(Br)cn1)N(C(c1ccccc1)C)C1CC1 20086,c1(C(=O)NC(c2cccc(-c3ccc(O)nc3)c2)C)ccc(CN(C)C)cc1 20087,C(C(C)(CC(C)C)NC(C1CCC(C)(F)CC1)=O)NC(C(COC)NC(N)=O)=O 20088,C1(NC(c2c(C)c(F)ccc2)=O)CN(C(c2nnn(C)c2C)=O)CC(C)(C)C1 20089,C1(C(N2CC(F)(F)C2C2CC2)=O)CC2CCN(c3ncccc3F)CC12 20090,C=C=CCCC(=O)N1CCC(N(C(c2cc(-c3ccc(Cl)cc3)c[nH]2)=O)C2CC2)C1 20091,C(=O)(C1=CCCSC1)NC1CN(C(C2(C)CCCO2)=O)CC1C(F)(F)F 20092,N1(C(C=C(CC)C)=O)CCN(C2CCCN(C(=O)CNc3cccnn3)C2)CC1 20093,N1(CC(=O)NC(C)CNC(=O)CC2(C(F)(F)F)CC2)C(C)CCCC1C 20094,N1(C(C2N(C)C(=O)CC2)=O)CC2(CCCC(CNC(C3CC(F)C3)=O)O2)C1 20095,c1(C(N2CCC(OCC#C)C2)=O)cc(Br)c(C)c([N+](=O)[O-])c1 20096,CCCC(C)CC(=O)N1CCC(C(=O)NCCCN(C)C(C)C)(OC)C1 20097,C#CC1(O)CCCN(C(C2C3CN(C(=O)Cc4ccccc4F)CC23)=O)C1 20098,C1(C(C)(C)C)(CNC(COCC(=C)C)=O)CCN(C(C2CCN(C)C2C)=O)C1 20099,c1(NC(C2CC23CNCC3)=O)cccc2c1CCS2(=O)=O 20100,c1(SC)ncc(Cl)c(C(=O)NC2CN(C(=O)CCCC(C)C)CCC2C(F)F)n1 20101,Cc1noc(C)c1NC(c1c(CNC(C2CCC(CO)O2)=O)nnn1C)=O 20102,C1(N(CC(=O)N(CC(=O)NC2(CCOC)CC2)C)C)CCCC1 20103,C1(COC)CSCCN1C(=O)C(=O)NCC1(CO)CCCCC1 20104,c1(CC(CC)C)nc(-c2ccc(Cl)s2)n(CCC(C)(C)C)n1 20105,S(=O)(=O)(c1ccc2c(c1)COC2)NC1CC2(CNC2)C1.NC1CC2N(C1)C2=O 20106,n1(CC)ccc(C(=O)NCC(C(C)C)NC(=O)CCn2ncn(C)c2=O)cc1=O 20107,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)CC2)=O)ccc2sccc2c1 20108,C1(C(=O)NC2C(C(=O)NCCCn3ncc(C)c3)C2(C)C)CCCCCN1C 20109,C1(OC)CC(NC(C2CCCCN2CC(F)F)=O)CN(C(c2ccc(C)o2)=O)C1 20110,C#CC1(C(N2CCC(C(C)(C)C)(CNC(c3ocnc3C)=O)C2)=O)CCCC1 20111,N1(C(CC2CCN(S(C)(=O)=O)CC2)=O)C2CC(F)C(C2)C1C(=O)NCC(F)F 20112,CC1CCC(n2nc(-c3ccoc3)nc2C2CCCCN2)CC1 20113,CCCCC(C)CCC(=O)Nc1cnc2ncc(C(=O)NOCC(C)(C)OC)n2c1 20114,N1(C(C(C)SCC)=O)CC2(CCCN(C(=O)C=C3CCC(c4cccs4)C3)C2)C1 20115,N1(C(CC=CC)=O)CCC2C(CCN2C(c2cnccc2OC2CCCC2)C)C1 20116,C1(NC(C(C)(C)C2CCCCO2)=O)CN(C(=O)CC2CSC2)CC12CCOCC2 20117,C#CC1(O)CN(C(c2cc(CNC(=O)Cn3ncnn3)sn2)=O)C1 20118,c1(-c2c(C#C)cccc2)cnc2ncc(C(=O)Nc3cc4ccccc4[nH]3)n2c1 20119,C(=O)(C1=C(Cl)CCOC1)N(C)CC1CCCN(C(C2CCC3CC23)=O)C1 20120,C(CC(CC)C(=O)N1CCC(O)(CNC(=O)CSc2nncn2C(C)C)C1)=CC 20121,c1(C(=O)NC2C(CO)CCN(C(C3C(C)CCCC3)=O)C2)cncc(N=[N+]=[N-])c1 20122,c1(C(=O)NC(CC)CNC(c2cc(C(=O)OC)c[nH]2)=O)cccc2c1CCC2=O 20123,C(=O)(C#CC1CCCO1)N(C1CN(C(c2ccc[nH]2)=O)CC12CC2)C 20124,c1(C(=O)NC2CC(C(=O)Nc3ccc(OC)cc3C)C2)cc2cccc(O)c2[nH]1 20125,c1(C(=O)NC)cccc(C(=O)NCC2CN(C(=O)CNC(N)=O)CC2C)n1 20126,c1(CNC(C(N2CCC(CC)CC2)CC)=O)cnc(C)[nH]c1=N 20127,C1(NC(c2nccc(C)c2N)=O)COC2(CCN(C(C3CC(Cl)(Cl)C3)=O)C2)C1 20128,C(=O)(C(C)(CNC(=O)CNC(=O)CC)CC)NC1C(C#C)CCC1 20129,Cc1nc(C)c(C(=O)NC2CCCC2CNC(=O)CSc2ccccn2)o1 20130,CC1CCc2nc(Cl)[nH]c(=NC3CC(CNC(C4CC5(C4)CC(O)C5)=O)C3)c2C1 20131,Cn1cc(Cl)cc1C(=O)NC(C1CCOCC1)C(N1CCCCC1C(F)F)=O 20132,CCC1=C(C(=O)NC23CCC(C2)N(C(=O)C=NOC)C3)SCCO1 20133,C1(NC(c2c(C)onc2)=O)CCN(C(=O)Cn2c(C)ccc2C)CC1C 20134,N1(C(CC2(C=C)CC2)=O)CCC(CN(C)C(C2CCCN2S(=O)(=O)CC)=O)CC1 20135,CCC(O)(C(=O)NCCCOCCNC(=O)C(C1CC1)OC)c1ccccc1 20136,C1(C(=O)NC(c2ncc[nH]2)C)CN(C)CCN1C(=O)C(c1ccccc1)F 20137,C(=O)(C#CC1CCOCC1)NC1(C(N2CCC(C)CC2C)=O)CSC1 20138,C(CC1=CCN(C(C2(C3CCOCC3)CC2)=O)CC1)NC(C(C)(C)C(N)=O)=O 20139,c1(C(=O)NCCC2CN(C(C=CSC)=O)C2)ccccc1[N+](=O)[O-] 20140,c1(CC)onc(C(=O)NCC2CN(C(C3CCN(C)C3=O)=O)CC2C)c1C 20141,c1(C(=O)NC(C(=O)CC2CC2)=O)n[nH]c2c1CS(=O)(=O)CC2 20142,CCCC(CNC(=O)CCn1cccn1)NC(=O)COCCc1ccccc1 20143,C(=O)(C1CSc2ccccc21)N1CC(COC)(CNC(=O)C(C)CSC)C1 20144,CN1CC(CN2CCCC(c3cccc(Cl)n3)C2)C(F)(F)C1 20145,C1(OC)CC2(C1)CC(C(=O)NCCC(C)NC(=O)CC(F)(F)Cl)C2 20146,C(=O)(CC(F)(F)F)NC(CNC(c1ccn(CCC)n1)=O)(C)C 20147,C1(CC)CN(C(=O)CC(C)C(F)F)CCN1C(C1CC2CC1C2)=O 20148,c1(NCC(CC)NS(C)(=O)=O)ccc(S(=O)(=O)NC2COC(C)(C)C2)cc1Br 20149,Cc1cccc(CNC(=O)CC(C(C)C)NC(c2cncn2C(C)C)=O)c1C 20150,C12(CNC(CC3CCC(C)C3)=O)CC(NC(c3sccc3F)=O)(CO1)C2 20151,c1(C(C(=O)NC2CC(CNC(c3cn(CC=C)nc3)=O)C2)(F)F)cccc(C)n1 20152,S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)Nc1cncnc1Cl.C12CC1CNC2=O 20153,C1(COC)(CNC(=O)C(F)OC)CCN(C(=O)C(c2ccccc2)OC)CC1 20154,CN1CCN(C(=O)C(F)n2cccn2)C(CNC(c2cnc(C(F)(F)F)s2)=O)C1 20155,Cc1nc2c(NC(c3ncccc3NC(C3C4COCC34)=O)=O)cccn2n1 20156,Cc1ccccc1SC1(CNC(CNS(C)(=O)=O)=O)CC1.C12CC1NC2=O 20157,N1(C(CC2N(CC)CCOC2)=O)CCN(C(=O)CC(F)(F)F)C(C)C1 20158,C1(CC)CC(C)N(C(=O)NCCCN2CCCC2=O)C1 20159,C(C(C)(C)CC(=O)NC1(C(=O)NOCCC2CC2)CCCCC1)OCC 20160,C(C(=O)NCC)(C(C(C)CC)OC)N(CC(=O)OC)CC=C 20161,c1(C(=O)NC2CC(C(N(C(C(N)=O)C3CC3)C)=O)C2)csc(Cl)n1 20162,C1(NC(=O)CCc2cc(F)ccn2)CN(C(C2C=CCCC2)=O)CCC1(F)F 20163,O=C(C1=CN=C2N=CNN2C1)NCC=CCNC(c1cc(F)c(Cl)cc1F)=O 20164,CCC(CC(=O)N(CC(C)O)C)NC(C1(Cl)CC1)=O 20165,C1(CC(=O)NCC(C(C)C)NC(c2c[nH]c(=N)s2)=O)C2CC3CC(C2)CC1C3 20166,c1(CNC(N)=O)ccc(C#N)cc1O.C1(=O)C(CO)ONC(=O)OC(C)(C)CN1 20167,c1(CN(CC(=O)NC2(COC)CC2)C)ccco1 20168,c1(NC(CCC(F)(F)F)c2c(Cl)cccc2)nc(N2CC3CC3C2)nc2sccc12 20169,c1(OC)cc(C#N)ccc1C(N1CCC(C)(NC(C2C(Cl)(Cl)C23CC3)=O)C1)=O 20170,Cc1cc2n(n1)CCN(C(=O)CC1CN(C(=O)CSC(F)(F)F)CCC1C)C2 20171,c1(C(N(CCNC(CC2CN(C)C2)=O)Cc2cccc(Cl)c2)=O)cnc2[nH]cnc2c1 20172,c1(C(CN(C(=O)NC(CC)C(=O)N2CCCC2)C)C)cccc(C)c1 20173,c1(C(c2n(CCC)nnn2)NCc2nc(C)n(C)n2)ccc2c(c1)OCC(=O)N2 20174,c1(CNC(CC)CNC(C2(c3ccnn3C)CC2)=O)ccccc1-n1cccc1 20175,c1(C(=O)NC2CCC(CNC(c3cnc(C(C)=O)s3)=O)C2)cc(C)c(Cl)cc1C 20176,C(C(O)CS(C)(=O)=O)NC(C)CC1OCCC1C 20177,CCCCC(O)C(=O)N1CCCC(CC)C1C(=O)NCCC(COCC)OC 20178,Cc1cccc(C(N2CCC(F)CC2C(=O)NC2CCC(C(N)=O)C2)=O)c1O 20179,N(C1CCC(NC2CCC2)c2ccccc21)C(=O)Cc1ccccc1OC(F)F 20180,c1(C(=O)NC2C=CCN(C(Cc3c(C)occ3)=O)C2)cccc(Cl)c1C 20181,Cc1nc[nH]c1CC(=O)N(C1CCC(NC(=O)Cc2cnc[nH]2)C1)C 20182,CON(CCC(=O)NC1(C(C2CCCO2)=O)CC1)C(=O)c1cnn[nH]1 20183,C(CNC(c1cnn[nH]1)=O)(CCCC)NC(C(COCC)C)=O 20184,C12(C(=O)NCCN(C(CC(CC)C(C)C)=O)C3CC3)CC3CC(C1)CC(O)(C3)C2 20185,C#CC1(C(=O)NC(CC)CCCCC)CCN(C(C2C3CCC(C3)C2C)=O)CC1 20186,C1(NC(c2c(C)coc2C2CC2)=O)CC(F)CN(C(C2CCCOC2)=O)C1 20187,Cc1nc2nccc(NC3CC(F)(F)CC3NC(c3cnc4ccsc4c3)=O)n2n1 20188,Cc1[nH]c(=N)sc1C(=O)NCC1CCCN(C(C2(c3ccccc3)CCC2)=O)C1 20189,C1(NC(c2cnn3ccccc23)=O)COC2(CCN(C(C3CCOC3)=O)CC2)C1 20190,C1(CNC(C2CCC(C)(CC)O2)=O)CN(C(=O)N(C)C)CCN1C.c12cc-1n[nH]2 20191,c1(C(=O)NC2C(CO)CCN(C(c3c(CC)ccs3)=O)C2)cc(S(C)(=O)=O)co1 20192,Cc1cccc2c1CCCC2NCCC1(C)CCC(=O)N1 20193,N1(C(C(C)NC(=O)OC)=O)CCCCC1CNC(c1cnc(O)o1)=O 20194,CCC(CC)CC(=O)NC(CNC(C1CCCN1C)=O)C(C)C 20195,N1(C(c2c(CNC(c3c(C)[nH]c(C)c3C)=O)n[nH]c2)=O)CC2(C1)NC(=O)NC2=O 20196,N1(C(=O)CN2CCCC2)CC2(C(=O)O)CC1(CC1CCCC1)C2 20197,CC1(CNC(=O)CCOCC(F)(F)F)CCN(C(C2CCCC(F)C2)=O)C1 20198,Cc1cc(C(=O)NC2CC(CCNC(=O)CN3CCOCC3=O)C2)ccc1Cl 20199,N1(C(c2n(C)ccc2)=O)CC2(CCCC(CNC(=O)Cc3ccon3)O2)C1 20200,C=CCCC(C(=O)NCC1(C)CCCO1)NC(c1ccccc1Cl)=O 20201,c1(CC)ccc(C(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)cn1 20202,C1(C(c2cn(C)nc2)C(=O)NC2CC(CO)(CO)C2)CCC(F)(F)C1.C(N)(=O)N 20203,CS(C)(=O)=NC(=O)C(=O)NC12CC(CNC(=O)CCc3cn[nH]c3)(C1)C2 20204,C1(CNC(c2cnn(CCC3CC3)c2)=O)CC(F)(F)CN1C(=O)Cc1ccno1 20205,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(=O)CC2OCCCO2)C2CCCCC12 20206,CCCCC(C(=O)NCC(C1CCCCC1)NC(=O)C(F)F)NC(N)=O 20207,c1(C(=O)NCC(C)NC(C2CC(C(C)C)C2)=O)ccc2cc(O)ccc2c1 20208,C(C(C(C)C(C)C)NC(C1(C#N)CC2(CC2)C1)=O)NC(c1c(C)noc1)=O 20209,CC1(CN2CC(C(F)Cn3cc(CC(=O)O)nn3)C2)CCCCC1(F)F 20210,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)C(C)C)(COC)C2)=O)o1 20211,N1(C(c2cc(F)cc(Br)c2)C(=O)NC)CCC2CCCCC12 20212,c1(C(N(CCNC(C2(C)CC=C(C)CC2)=O)C)=O)cc(Cl)c(F)cc1Cl 20213,c1(-c2n(CC=C)c(N(CC(C)C)CC)nn2)ccc(S(C)(=O)=O)cc1 20214,C(=O)(C#Cc1ccccc1)N1C(CNC(C2CCN(C(=O)OC)CC2)=O)CC1 20215,c1(C(C)C)ccccc1C(=O)NC1CC1CNC(=O)C=C1CC1 20216,C1(NC(C(CSC)(C)NC(=O)Cn2cnnc2)=O)CCN(OC)CC1 20217,N1(C(CC(C)SC)=O)CCCC(C(=O)NCC2(n3ccnn3)CC2)C1 20218,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20219,CN=c1nc(N2CCC(C)(CO)C2)[nH]c(=NCC2(c3cccc(F)c3)CC2)[nH]1 20220,c1(C(N2CC(C)C(CCNC(=O)CCS(C)=O)C2)=O)cc(F)c(F)c(C#N)c1 20221,c1(C(C(C)C)NCC(Cc2ccc(OC)cc2)C)cc(Cl)cc(Cl)c1 20222,C1(C(=O)NCC(=O)N(CC)CC)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20223,C(=O)(CC1=CCOCC1)NC1CCCC(NC(C(CCC)OC)=O)C1 20224,n1(CC)cnc2c(N3CCC(CC(C)C)C3)nc(NC(C)(C)CF)nc12 20225,C1(N(C(CCC2CC(NC(c3cc(CC)[nH]n3)=O)C2)=O)C)CCCCC1CO 20226,CN1CC(CC(=O)NCCOCCNC(=O)CC=C(Cl)Cl)C(O)C1 20227,c1(C(=O)NC(C(C)C)CNC(C2(C)C=CCC2)=O)cc(F)c2c(c1)CCC2 20228,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2Cl)C1 20229,C1(CSC)CCCN1C(=O)C(C1CCCC1)NC(=O)CC1CC(=O)C1 20230,c1(CC)cc(N2CCCC(NC(C3CCC(=O)N3)=O)C2C)nc(CC)n1 20231,CCC(CC)CC(=O)N1CCC(NC(c2cc(SC)oc2C)=O)C(C)C1 20232,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20233,C(CN=c1nc(N2CCCn3cc(Br)cc3C2)c2c([nH]1)CCC2)(C(C)C)OCC 20234,Cc1nc[nH]c(=NCC2C(C)CCCN2C(c2ccc(Cl)nc2)=O)c1Br 20235,CCCCCCCCCCCC(=O)NC1CCCCC1NC(=O)CO 20236,C1(NC(c2cc(SC)ncc2)=O)C2CC(CN(C(C3(SC)CCC3)=O)C2)C1CO 20237,Cc1cccc2c(CC(=O)NC3COCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20238,C1(OCCCC)CCCN1C(=O)CCn1cc(NC(C)=O)nn1 20239,C12(CC3(CC(F)C3)C1)CNC(=O)C(=O)N2.C#CC1CCCC(COC)C1 20240,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20241,C1(CC(=O)NC(c2nc(C)cs2)CC)CN(Cc2ccc(C(=O)O)s2)CCO1 20242,Cc1cc(CC(=O)NC23CC2CN(C(=O)CSc2cn[nH]c2)C3)nn1C 20243,N1(Cc2ccc(-n3cnnc3)cc2)CC2CCOC2(C(=O)O)C1 20244,C1(N2CCC(C#N)C2)CCN(C(=NCC2CC2)NCc2cc(Cl)ccc2F)CC1 20245,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(=O)C(O)CC1CCCC1 20246,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20247,c1(-c2n(CCC)ccn2)cc(Br)c(NC(c2cc(C)[nH]c2C)=O)nc1C 20248,C=CCCCC(C(=O)NC(c1nnc(O)o1)C)NC(=O)CCN1CCCCC1 20249,O=C1NCCCCC1NC(c1ccc(I)cc1)c1nnnn1CCCF 20250,N1(C(C(CC=C)OC)=O)CCC(N=[N+]=[N-])(C(=O)NCCc2cccc(O)c2)C1 20251,Cc1cc(NCC2(F)CC(CO)C2)ncc1S(=O)(=O)NC1CCC2C(CC1)C2(F)F 20252,O=C(CC1=CSC2=NCCN12)N1CCC(F)(CF)C1 20253,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(O)Cn3cncn3)C2)=O)o1 20254,CCC(C(=O)N1CC2CC1(C(=O)NCC1(COC)CCCO1)C2)C(F)(F)F 20255,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(C)CCCC2)=O)C1 20256,c1(C(N(C)CC=CC(=O)NCc2cnccn2)=O)cn2cnnc2cn1 20257,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CCCCC1C(F)(F)F)=O 20258,C(CCCN=c1[nH]c2ccc(N)cc2s1)N(S(C)(=O)=O)CCN(CC)CC 20259,C1(NC(c2c(C)n[nH]c2)=O)C2CCN(C(=O)C=CC(=O)NC3CC3)CC12 20260,Cc1ccnc(CN(C)CCNC(c2cc(CNC(=O)OC(C)(C)C)n(C)n2)=O)c1 20261,Cc1cccc(CNC(=O)CC2CCCCN2C(=O)CCc2ccc(C)nc2)c1 20262,c1(C(CNC(c2ccc(C)cc2)Cc2ccccn2)=O)ccc(F)c(C)c1Cl 20263,N1(C(C2(C(=O)OC)CC2)=O)CC2(C(N3CCOC(C(F)(F)F)C3)=O)CC1(CO)C2 20264,CC1CN(C(C2(CO)CCCC2)=O)CC(C)C1NC(c1cc(C(F)(F)F)cs1)=O 20265,N1(C(c2c(CC)c[nH]c2)=O)CC2CCC(NC(C3C(C)(C)C3(C)C)=O)CC2C1 20266,c1(C(N2CCC(NC(Cc3c(C)nc(S)s3)=O)CC2C)=O)noc2ccccc12 20267,C1(N(C(CC)=O)C)CCCC(N(C)C(c2cn(CCOC)nc2C)=O)C1 20268,c1(C(C)C)ncc(Br)c(N2CC(CO)(NC(C3CC4CCCC34)=O)C2)n1 20269,c1(C(N2C(CNC(=O)COC3CCCOC3)CCC2)=O)c(F)ccc2occc12 20270,C1(OC)CCN(C(=O)CC2C3CN(C(c4ccc(CO)s4)=O)CC23)CC1C 20271,S(=O)(=O)(C1CCCCC1)N1CCN(C(C2(C)CCN(C(=O)OC(C)(C)C)C2)=O)CC1 20272,C1(C(N(C)CCOCCCNC(C2CCCCCC2)=O)=O)CC2(C1)CC(O)C2 20273,C1(C(=O)NCCCC(=O)OC)C(C2CC2)CCN1C(=O)CC1CCSC1 20274,C1(CNC(C(C)(C)O)=O)CC2(CCN(C(c3cnc(C#N)s3)=O)CC2)C1 20275,C1(C(=O)NC2CCN(C(C)=O)C2)CC(N=[N+]=[N-])CN1C(=O)Cc1cn[nH]c1 20276,C1(NC(c2ccon2)=O)CN(C(c2cnc3ccnn3c2)=O)C2(CCOC2)C1 20277,c1(C(C(=O)NCC(C)(C)CNC(c2cc(Cl)ccn2)=O)O)ccc(F)c(F)c1 20278,N1(C(c2c(CC)nc[nH]2)=O)CCC2(C1)CN(C(=O)CCc1ccncn1)C2 20279,N#Cc1ccc(C(=O)NC2CCN(C(=O)CC3CCS(=O)(=O)C3)C2)o1 20280,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20281,c1(C(=O)NC(CN(C(c2nccc(OC)c2N)=O)CC)C)cnn2c1CCC2 20282,C#CCCCC(C)C(=O)NC(c1ccc(CNC(=O)C(C)(C)OC(F)(F)F)cc1)C 20283,c1(C(=O)NCc2cc(C(=O)NC(C(CCC)C)C)n(C)n2)cc2occc2[nH]1 20284,N1(C(CN2CC(C)C2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20285,N1(C(C)=O)CCC(CNC(c2cn(Cc3ccc(Cl)nc3)nn2)=O)C12CC2 20286,C#Cc1ccc(C(=O)NC2CCCC2(C)CNC(C2CNC(=O)C2)=O)cn1 20287,c1(C(=O)Nc2cccc(C(c3csc(CO)n3)C)c2)cc2cc[nH]c(=O)c2s1 20288,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20289,C1(NC(c2scc(CNC(C(C(CC)C)N(C)C)=O)c2)=O)CCN(C)CC1(C)C 20290,c1(CC(=O)NCCOCCN(C(C(C)Cc2cnn(C)c2)=O)C)cccnc1Cl 20291,N(C1CN(C(C23CCN(CC2)C3)=O)Cc2ccccc21)C(=O)CCc1nccs1 20292,N1(CC(C)C)CC(NS(=O)(=O)CC2(C)CC2(F)F)CC1=O 20293,N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NCC23CC(C2)C(C)O3)C1 20294,C=CCC(C)(C)CC(=O)N(C)Cc1ccccc1CNC(C1NC(=O)CC1C)=O 20295,N1(CC=CCNC(C2C(=C)C2C(N)=O)=O)CCC(CO)C(O)C1.C1C(=O)N1 20296,O=C(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1CN(C(=O)CCC2CCC2)CCO1 20297,C1(NC(C(N2CCC(C)C2)=O)=O)CN(C(c2cc(O)cc(O)n2)=O)C(C)(C)C1 20298,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20299,Cc1cc(C(N2CCC(O)(C(C)NC(C3(O)CCC3)=O)CC2)=O)nc(C)n1 20300,N1(C(Cc2onc(CC)n2)=O)CC2(CC(NC(C3(C)CNC(=O)C3)=O)CO2)C1 20301,Cc1cc(F)c(CNC(=O)NC(CO)C(=O)N(C)C)nc1Br 20302,c1(OC)cnc(Cl)nc1N1CCCOC(CNC(=O)CC2CC=CCN2C)C1 20303,c1(CCC)[nH]ccc1C(=O)NCC1CCC1C(=O)NCC.C12CCCN1C2=O 20304,Cc1ccc(N2CCCOC2=O)cc1NC(c1cn(CC(C)N)nn1)=O 20305,C1(NC(=O)NCc2scc(C)n2)(C)CCCCC1.C(CO)(CC(C)C)N 20306,c1(CC)nc(N(CCNC(=O)N(c2ccccc2Cl)CC)CC)c(C)s1 20307,CC(C)C(C(=O)NCCCNCCCCNC(=O)CC1CCCC(=O)C1)NC=O 20308,N1(C(C2(OC)CCN(C=O)C2)=O)CC(C)(C2CCC2)C1.c1scnc1C 20309,c1(N2C(NC(c3nc(-c4cn(C)nc4)sc3)=O)CCC2)cc(C(C)(C)C)ncn1 20310,C1(O)(CN(C)C(c2ccc(C(C)(C)O)cc2)=O)CCN(C(C2CC2F)=O)C1 20311,N1(C(c2c(=N)[nH]cnc2)=O)C2CCC1CN(C(=O)CCc1cncs1)C2 20312,c1(COC)cccc(OC(c2nn[nH]n2)C)c1.c12nc(cs1)C(=O)OC2C 20313,N1(C(CCC)=O)CC(NC(=O)CCc2ccc(O)cc2)CC1(C)C 20314,C1(NC(c2csc(CC(F)F)n2)=O)CN(C(c2coc(Cl)c2)=O)CC1F 20315,c1(OC)ccc(-n2nc(C3CCOC3)nc2C(=O)Nc2cnn(CCF)c2)cc1 20316,c1(C(=O)NC2CC(C)N(C(c3cnc(C4CC4)[nH]3)=O)C2)cc2n(n1)CC1(CC1)C2 20317,c1(C(=O)NC(CC(C)NC(C2=CC(C)(C)C=C2OC)=O)C)ccc2nncn2c1 20318,CCCC(O)C(=O)N(C)CCOCCN(C(=O)CCOC1CCCC1)C 20319,C1(N(C(=O)CCCc2sccc2C)CC)CCCN(C(C2CCCCC2)=O)C1 20320,C#Cc1cccc(C(=O)NC2(C(=O)NC3CC(CC)(CC)C3)CCN(C)C2)c1 20321,C1(CNC(C(CC)C(C)C)=O)CC2(CCCN(C(=O)COCCCF)CC2)C1 20322,N1(C(CCSc2n(C)nnn2)=O)C2CCC1CC(CNC(=O)CCC1(C)N=N1)C2 20323,c1(C(=O)NC(C(=O)NC(COC)C2CC2)C2CCCO2)cnc(O)c(F)c1 20324,O=C1CC(C(=O)N2CCCOC(CNC(=O)C(c3ccccn3)O)C2)=NN1 20325,C1(C(C)C)CCN(C(=O)C(=O)Cc2ccccc2)C(CNC(=O)CCC(C)C)C1 20326,c1(C(N2CC(CCNC(CN3CC(C)C3)=O)C2)=O)ccc2cnoc2c1 20327,c1(CC)cc(F)ccc1C(=O)NCC(=C)CCNC(=O)C(C)(C)F 20328,c1(OCC(=O)N(CC(=O)NCC(C)Cc2cccs2)C)ccc(C#N)cc1Cl 20329,C1(CC(N2C(CN(C(C3CC(C(F)(F)F)C3)=O)C3CC3)CCC2)=O)CC(O)C1(C)C 20330,NS(=O)(=O)CCC(=O)NCCC1(O)CN(C(C23CCC(CF)(C2)OC3)=O)C1 20331,CCCC(CC(C)C)C(=O)N1CCC(O)(C(C)NC(=O)C#CCCCC)C1 20332,c1(C(=O)C(F)(F)F)ccccc1NC1CC(c2ccc(Cl)cc2)C1 20333,N1(C(C)C)C2CCC1CC(NC(=O)CCOCCO)C2.C(C(F)(F)F)CC(C)O 20334,N1(C(CN(C(C2(C(C)C)CC2)=O)CC2CC2)=O)CCCNC(=O)C1 20335,c1(OC)ccc(C(=O)NC2CC2C2CC2C)cn1.C12(CF)CCN(C1)C2=O 20336,C=C=C(C)CC(=O)NCCC(C)NC(=O)C(c1ccc(OC)cc1)(C)C 20337,c1(C(=O)NCC2CN(C(C3C4CCCC34)=O)CC2(F)F)scc2c1CCCC2 20338,c1(OC)cc(C)c(NC(N2C3CC2CN(Cc2ccccc2)C3)=O)cc1F 20339,C1(C(N2CCC(C(C)(C)C)(CNC(C3CN(C)C3)=O)C2)=O)CCCC(C)(C)O1 20340,C(=O)(C1=CCc2ccccc21)NS(c1c(C(=O)NC2CC2)scc1)(=O)=O 20341,C1(NC(c2onc(CC)c2C)=O)CCN(C(=O)CCCCCNC(C)=O)CC1F 20342,c1(C(=O)NC2CCC(N3CCN(C(C4CN(C)C4)=O)CC3)C2)cncc2nc[nH]c12 20343,Nc1c(C(=O)NCC2CC2NC(=O)CCF)cccc1C(F)(F)F 20344,C1(NC(C2(C)CCN(C)C2)=O)CC2CC(NC(c3occc3C3CC3)=O)C2C1 20345,c1(C(=O)NCC2(O)CCCN(C(C(C(C)O)(C)C)=O)C2)cccn2nccc12 20346,C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CNC(CCCCCC)=O)CCOC1 20347,C1(NC(COC(C)C)C)CC(Nc2cccc(-c3cnc[nH]3)c2)C1(C)C 20348,CC(C)=C=CC(=O)NCC(C1CCCC1)NC(=O)Cc1cnn(C(C)C)c1 20349,c1(CCCC2(C(=O)OCC)CCOCC2)ccc(OC)c(Cl)c1OCC 20350,c1(C(=O)NC(C2CCCC2)CNC(C=CC)=O)cnc(C)nc1C1CC1 20351,C12(CNC(C(C)CC(F)F)=O)CCC(CN(C(=O)CS(=O)(=O)C3CC3)C1)C2 20352,c1(C(N2CC(NC(c3onc4ccccc34)=O)C(F)C2)=O)ccc([N+](=O)[O-])cn1 20353,c1(C(=O)NCC(C(C)C)NC(Cn2c(C)nnn2)=O)ccc(N=S(C)(C)=O)s1 20354,C(CNC(=O)C(=O)NCC(C)CN)(CSC)OC 20355,C1(C(N(CCC#C)CCOC)=O)CCN(C(c2c(C)ncnc2C)=O)C1(C)C 20356,C1(NC(C(CC)SC)=O)CC2CCC1N2C(C1(NC(C)=O)CCC(C)CC1)=O 20357,C(=O)(C(O)C(F)(F)F)N(CCC(=O)NCC1CCC(=C)CC1)C1CC1 20358,c1(C(N(C2CCN(C(CCCC#C)=O)CC2C)C)=O)ccc2cccnc2c1 20359,c1(C(=O)NCC2(O)CCCN(C(C3C(C)C3)=O)C2)cc2ncccc2o1 20360,Cc1c([N+](=O)[O-])c(C(=O)N(C(C)Cn2cccn2)C)nn1C 20361,CCCC(C(O)C(=O)N1CCOC(C)(C)CC1)NC(c1ccc(CO)cc1)=O 20362,C(C)(CO)(C(=O)NC1CCOC(C(=O)NCC(C)CC2CCCC2)C1)OC 20363,c1(C(=O)NCC(C)N(C(=O)CC2CCOC2=O)C)ccc(C#N)nc1 20364,CCCC(O)C(=O)N1CCC(OC2CN(C(C3C4CNC(=O)C34)=O)C2)CC1 20365,C12(C(N3CCC(O)(CCC)C3)=O)CC(CO)(CN1C(=O)OC(C)(C)C)C2 20366,C1(C(=O)NCC2CC(F)(CNC(=O)C(O)CSC)C2)(OC)CCOCC1 20367,Nc1nccnc1C(=O)NC1CC(F)(F)C1.N12CC(C(c3ccccc3)C1)C2 20368,CN1C(=O)CN(CC(=O)NC(CNC(=O)CCc2cc(Cl)no2)C2CC2)C1=O 20369,N1(C(C)C)CC2CC2(Cc2ccn(C(=O)NCc3nnc(C)s3)n2)C1 20370,N1(C(C(C)OCCC=C)=O)CC(COC)(NC(=O)C(C)OC2CCCC2)C1 20371,n1(CCCC(=O)NC2CC(F)(CNC(COCCCC#C)=O)C2)c(C)csc1=O 20372,N1(C(CC(CC)(F)F)=O)CC2(CCN(C(C3CCC(=O)C3)=O)CC2)C1C(C)C 20373,C(CCc1ccc(Cl)cc1)(C(=O)NCCC#N)OC.C1C(C)CN1C 20374,n1(CCCC(=O)N)cnc2ccccc12.C1(CCCN(C(C2CC23CC3)=O)C)CCCC1 20375,Cc1c(NCCc2c(F)cccc2F)ncnc1NC1CCC(NC)C1 20376,N1(C(C2CC=C(C)CC2)=O)CCC(F)(C(N2CC(CO)C(CO)C2)=O)CC1 20377,CC1CC(C(N2CCC(CN(C(=O)Cc3cn(C)nn3)C)CC2)=O)CCO1 20378,C1(NC(c2coc(Cl)n2)=O)CCN(C(=O)C(O)Cc2ccccc2Cl)CC1F 20379,N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(C1)CN(C(=O)CC1CC(C)C1)CCO2 20380,c1(C(NOCC(=O)N(C)CC2CCCOC2)=O)ccc(=O)n(C)n1 20381,C1(OCC=C)C(NC(=O)C(N2CCC(OC)C2)c2ccsc2)CC1O 20382,C(=O)(CC1CCCc2ccnn21)N(C1CN(C(C=CCC)=O)C(CO)C1)C1CC1 20383,c1(C)cn(C)nc1C(C)(C)C.c1(C(c2cccs2)NC(C)CC(N)=O)nnn[nH]1 20384,CCC(C(=O)NCC(C)CCNC(c1ccc(C2CC2)s1)=O)c1nccn1C 20385,N1(C(C2(CC#C)CCC2)=O)CCC(NC(=O)CNS(N)(=O)=O)C2(CCC2)C1 20386,CC(C)CCCCC(=O)NC1C2CC3C(C2)C13C(N1CC2(C=CCO2)C1)=O 20387,c1(CNC(C(C(C)C)O)=O)cnn2c1CN(C(=O)Cn1cncn1)CC2 20388,C1(C(N2C(CN(C(C3CC(=C)C3)=O)C)COCC2)=O)OCCCC1(C)C 20389,C=C=C(C)C(=O)NC1CCCC1NC(=O)C=CCCC(C)C 20390,C1(C(C)(C)C)C(=O)N1.C1(CC(=O)OC)CCCN(C(c2n[nH]cc2N(C)C)=O)C1 20391,C1(C)(CNC(C2(CC3CC3)CCOCC2)=O)CCC(NC(c2c(CC)ncs2)=O)C1 20392,N1(C(C(N(C(c2ccn(CC)n2)=O)C)C2CC2)=O)CC(N(C)C)C(F)C1 20393,Cc1nc(O)nc(C)c1C(=O)NCC(CC(F)(F)F)NC(C1CC1C(N)=O)=O 20394,N1(C(C2CCCN(C(C)C)C2)=O)CCN(C(c2cnc[nH]2)=O)CC1C(F)F 20395,C1(CNC(=O)CCn2cccn2)CCCC12CCN(C(=O)Cc1ccccc1)C2 20396,CC1(C)CN(C(=O)C2=COCC2)CC1NC(C1C2CCCC12)=O 20397,N1(C(C(C(C)NC2(C(=O)OC)CCC2)C)=O)CCC2(CC1)CC(C(=O)OC)C2 20398,C=CCC(F)(F)C(=O)N1CCC(F)(C(=O)N(CC)Cc2noc(C)n2)CC1 20399,C(=O)(C(C)(F)C(F)(F)F)NCc1cccc(CNC(CCCC)=O)c1 20400,Cc1ccc(NC(=O)CCCN2CC3COCC23)c(C)c1 20401,c1(C(N2CCC(COC)(NC(=O)C=Cc3ccncn3)C2)=O)ccc(Cl)cc1O 20402,CCC(CC(=O)NC(CCO)C(F)F)N(C)C(C1CC(C)(CC)C1)=O 20403,C1(C(=O)NCC2(CNC(CNC(CC(C)C)=O)=O)CCC2)COCC(C)O1 20404,c1(C(=O)NC(C)CNC(=O)C(=Cc2cscn2)F)ccc(Br)cc1N 20405,C(=O)(C(O)CC(F)(F)F)NC(C(=O)N(C(C)C)CCN(C)C)CCN(C)C 20406,c1(OCCCC(=O)NC(C)CCCNC(=O)CC2CCC(=O)N2)ccc(F)cc1 20407,C1(C(N(CC(=O)NC(CC)CC)C(C)C)=O)CNC(=O)O1 20408,c1(CCNC(C(CC2CC2)NC(C(COC)C)=O)=O)ccccc1F 20409,c1(C(N2CCC(N(C(C3CNC(=O)N3)=O)CC)C2)=O)cc2cccnn2c1 20410,C1(C(N(C2CCC(NC(C3(CO)CCCO3)=O)CC2)C)=O)C2CC3C(C2=O)C13 20411,C(C(C)(C)CS(=O)(=O)NC(c1nnnn1C(C)C)C1CC(F)(F)C1)OC(C)C 20412,C1(NC(c2ccc(C)c(C)c2O)=O)COC2(CCN(C(C3CCCO3)=O)CC2)C1 20413,N1(C(C2(CNC(C(C)OCC#C)=O)CCC2)=O)CC2CC=CCC2C1 20414,c1(C(=O)OC(C)C(=O)Sc2cccc(C#N)c2)ccc(C(F)(F)F)c(Cl)c1Cl 20415,CC1CN(C(c2csc(-c3ccsc3)n2)=O)CC1CNC(C1(CO)CCC1)=O 20416,C(CNC(=O)Cc1nccn1C)(CC(=O)NC(C1CCOC1)(C)C)OC 20417,C1(C(N2CC(C3(C)CC3)OCC2)=O)CC12CCN(CC13CCC(CC1)CC3)CC2 20418,c1(NC(C=CC)=O)ccc(C2(C(=O)NCCC3(OC4CC4)CCC3)CCC2)cc1 20419,c1(C(=O)NCC(CC)NC(C)=O)cc(C)ccc1NC(=O)C(C1CCOCC1)F 20420,CCC(C)CC(CO)N=c1cc(C)[nH]c(=NCc2cccc(N)n2)[nH]1 20421,N1(C(c2sc3ccn(C)c3c2)=O)CCC2(CCN(C(C3(c4cnc[nH]4)CC3)=O)C2)C1 20422,C1(CNC(C(CN(C)C)N(C)C)=O)CCC(NC(C2(C)CCCS2)=O)CC1 20423,C12(C)CCCN(C1)C2=O.C1(C(=O)OCC)CCN(C(=O)C(C)CO)CC1 20424,CCCC(CCC)NC(=O)C(O)C1CN(C(=O)CCCC2CC2C)C1 20425,C12(c3cn(CCCC)nn3)CCC(C(F)F)(CC1)C2.C12CCN(CC1)OC2=O 20426,N1(C(CCCNC(C)=O)=O)CCC(N=[N+]=[N-])(C(N2CC(c3nncs3)C2)=O)C1 20427,c1(CC(N2CC3C(NC(c4cnc(SC)s4)=O)(C3)C2)=O)c(C)nc(O)nc1C 20428,C1(CNC(C2CC(C)(O)C2)=O)CC2(CO1)CN(c1cc(O)nc(O)n1)C2 20429,CC1CN(C(c2cc3sccc3s2)=O)CC2(CCN(C(=O)CCCC3CC3)C2)O1 20430,c1(C(=O)NCC(CNC(C(C)OCC=C)=O)O)sc(Cl)c(Cl)c1OC 20431,C=CCC(CC(C)C)C(=O)NC(C)CCN(C)C(c1ccc2oncc2c1)=O 20432,S(=O)(=O)(c1ccc(C(=O)NCC2CCC2NC(C2(C)COCCO2)=O)cn1)NC 20433,C1(CNC(=O)CCCc2ccsc2)CC2COCC2N1C(=O)CCCCCO 20434,C(=O)(CCC1=CCCCC1)NC1CCN(C(c2n(C(C)C)ccc2)=O)C1C1CC1 20435,N1(C(=O)CCN2CCCC2=O)CCCC2CN(c3cc4nncn4cn3)CCC12 20436,C1(C(=O)NC2(c3onc(C)n3)CC2)CC2CC1CC2OC(C)(C)C 20437,C1(CCC(=O)NCCN)CCCCN1CCC(C1CCOCC1)O 20438,C1(C(=O)NC2(CO)CCN(C(C(C(C)C)OCC)=O)CC2)COCC2(CCC2)O1 20439,C1(C(N2CC(CNC(COC)=O)C(C)C2)=O)CCCCC1C1CC1 20440,C1(NC(=O)Cn2cncn2)CCSC12CN(C(=O)CCc1cncc(F)c1)C2 20441,c1(C(N2CCC(NC(C)=O)C2)=O)ccc(C(N2CCCC2)=O)cc1C(F)(F)F 20442,c1(OCC)nc(N2CCC(CNC(=O)C(C)n3cncn3)C(C)C2)ncc1Cl 20443,Cn1nc(C(F)(F)F)cc1CC(=O)NC(CN(C(=O)CC1CCC2CC12)CC)(C)C 20444,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(c1nccnc1C(N)=O)=O 20445,C1(CCOC)(NC(=O)C(F)=CC2CC2)CCN(C(c2cnc(C)n2C)=O)C1 20446,c1(COC)noc(CNC(=O)Cn2cc(CCCn3cncn3)nn2)n1 20447,CC(C(=O)N=c1cc2n([nH]1)CCCC2)NC(c1ccon1)=O 20448,C1(C(=O)NCCCC(C)NC(=O)C(c2ccc(F)cc2)=O)CC(=O)NC(=O)N1 20449,O=C(CC1CC12CC2)Nn1cnnc1 20450,N1(C(c2ccn(CCOC)n2)=O)CC(CNC(=O)C=Cc2nnn(C)n2)C(C)C1 20451,C1(N(C(=O)NCC2(OCC)CCC2)C2CC2)CCC1C(F)(F)F.c1nnnn1C 20452,N1(C(C(=O)NC(C)CC2CCC2)=O)CCC(O)(c2cccc(Br)c2)C1 20453,c1(C(C)C)nc(CC(=O)NCCN(C2CC2)CC2CC2)cs1 20454,C1(C#CC(=O)N2CCC(F)(CNC(c3n[nH]c(C)n3)=O)CC2)(CC)CC1 20455,N1(C(C2CCC(n3cc(C4(O)CCC4)nn3)C2)=O)CCc2nccn2CC1 20456,C(=O)(C(CNC(C1CCCCO1)=O)CC1CC1)N(CC(CCC)O)C 20457,N1(C(C(CC)NC(N)=O)=O)CCC(C(F)(F)F)CC1CNC(=O)CN1CCCC1 20458,C1(NC(c2[nH]cc(CC(C)C)c2)=O)CC2(C1)CN(Cc1ccc(CO)cc1)C2 20459,c1(C(=O)NCC(CNC(C(c2scc(C)n2)C)=O)O)c(F)ccc(O)c1O 20460,N1(C(CC2(C)CC2(Cl)Cl)=O)CCCCC(C2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1 20461,c1(CSC(C(=O)NC(CC)CN2CCC2)C)ccccc1.C1(=O)COCC(C)N1 20462,C(C(O)CCNC(c1cc(F)c[nH]1)=O)NC(c1cc(-c2ccccc2)cs1)=O 20463,N1(C(C2(CC#C)CCC2)=O)CC2CCC(CNC(C3C4CCCOC34)=O)(C2)C1 20464,C(CC(=O)NC(CC(=O)NC1(C)CCSCC1)C1CC1)(C(C)C)OCC 20465,C(=O)(C1=C(C#N)CCC1)N1C(CC)C(C(=O)N(C)Cc2cccc(C)n2)CC1 20466,C1(NC(C(C2CC2)OC)=O)CCCC(NC(=O)Cc2cc(-c3cccs3)on2)C1 20467,Cc1cc(N(C)C(c2cccc(F)c2)C)n2ncc(Br)c2n1.c12ncc([nH]1)[nH]c2=O 20468,C1(C(=O)NCC2(CN(C(C(C)=CC)=O)C)CC2)CC(S(C)(=O)=O)C1 20469,C(C(CCNC(=O)NC1(CO)CCOC1)OC(C)(C)C)OC 20470,c1(C(=O)NCC2N(C)CCN(C(C3(C#C)CCC3)=O)C2)cc2cccc(C)c2s1 20471,c1(CC(=O)N(C)CC2OCCN(C(CCC#C)=O)C2)ccc(C#N)cn1 20472,C1(CC(=O)OC(C=CCOC2CC3CC3C2)CC2CCCC2)CC(=O)N(O)C1 20473,c1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CC2)c[nH]c2cnccc12 20474,c1(C(=O)NCC2(C)CCCN(c3nccc(C)n3)C2)cccc2ccncc12 20475,N1(C(C2(F)C(C)OCC2)=O)CC2(CCC(CNC(=O)CCC(F)F)O2)C1 20476,n1(CC)cnc2c(N3CC4CC4(CO)C3)nc(N3CCC(SC)CC3)nc12 20477,CCC(C(=O)NC1(C)CC(N(C)C)C1)C(CC)NC(=O)C(N=[N+]=[N-])C(C)C 20478,C1(CNC(CCC2CC(OC)C2)=O)CN(c2ccn3nccc3n2)CCC1(C)C 20479,Cc1ccc(C2CCC2)cc1NC1(CO)CCCC(C)C1 20480,c1(COC)cccc(C(=O)NC(CCNC(C2(C)CC(F)(F)C2)=O)C(C)C)c1C 20481,C(=O)(C=C1SCC(=O)N1C)NC(C(=O)OC)Cc1ccsc1 20482,CC1CC(CNC(=NCc2ncccc2Cl)NC2CCS(=O)(=O)C2)CCO1 20483,S(=O)(=O)(c1cccc(O)c1)NCC1N(C(C2CCC(C(=O)OC)C2)=O)CCOC1 20484,C(C(C)S(C)(=O)=O)NC(C=CCN(C(C(C1CCCC1)OC)=O)C)=O 20485,c1(C(CNC(C(=O)N(CC)Cc2cccs2)=O)O)cc(Cl)cc(Cl)c1 20486,Cc1cc(CCNC(C2CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)cc(=O)n1C 20487,N1(C(C2C(C)CCCC2)=O)CCC12CN(C(c1nc[nH]n1)=O)C2 20488,C1(N(C)C(C2(C(F)F)CCC2)=O)CN(C(=O)C=CCO)CC12CC2 20489,c1(C(=O)NCC2CCCN(C(c3cnc(O)o3)=O)CC2)cc2n(c1)CCOC2 20490,CN1CCC2CCN(C(c3ccc(CNC(c4ccncc4)=O)s3)=O)C2C1 20491,c1(C(N2CCN(C(CC=C=C)=O)CC2c2cccnc2)=O)cncc2sccc12 20492,N1(C(c2c(C)cccc2)=O)CC2(CC(CNC(C3(CO)COC3)=O)C2)C1 20493,O=C1CCc2cc(NC(C34CCC3CN(C(c3cnc(O)[nH]3)=O)C4)=O)cnc2N1 20494,CC1CN(C(=O)CCOC)CC1(C(=O)O)CNC(c1cccc(Cl)c1)CCCCO 20495,CC(C)CCC(=O)NCCOCC(=O)NC1CCCC(C)O1 20496,CC(CC(F)F)C(=O)NCC1(NC(=O)Cc2cc(F)ncc2Br)CCC1 20497,n1(C(C)C)cccc1C(c1nnnn1CC1CCCO1)NCCn1ncnn1 20498,C(=O)(C(C)(O)C1CC1)NCCC(C)NC(C1(C2CC2)CC1)=O 20499,N1(C(C(CC)F)=O)CCN(C(C2CC3CCCC23)=O)C2(CCC2)C1 20500,c1(C(=O)NC2CC(C)N(C(=O)CC34COCC(C3)C4)C2)cc(C(F)F)cc(F)c1 20501,N1(C(C(COC)OC)=O)CCN(C(=O)C(c2cccc(C)c2)(F)F)CC1COC 20502,c1(CC(N2C(Cn3cc(CCC)nn3)C(C)CCC2)=O)ccc2occc2c1 20503,Cc1c[nH]c2ncc(C(N3CC4CCC3C(NC(=O)Cc3ccno3)C4)=O)cc12 20504,CC(C)CCC(=O)C(=O)NCC1(C)CCCN(C(C2CCCN(C)C2)=O)C1 20505,N1(C)C(=O)C(C)(OCC)C1CCCCCC 20506,CC(C)CC(C)(C(N)=O)NC(=O)CCCCNC(=O)C=CC1CCCCC1 20507,CC1CC(NC(C2(C)CC2c2ccccc2)=O)CN(C(=O)C(C2CC2)C2CC2)C1 20508,N1(C(CCOCCSC)=O)CC2(CO)CC1(CNC(=O)C(C)SC)C2 20509,C(CC(CC)C(=O)NCCCCC1CCN(C(C2CCOCC2)=O)CC1)=CC 20510,c1(C(N2C(C)CCC(CNC(C3C(OCC)CC3)=O)C2)=O)cc2ccncc2[nH]1 20511,CC1CN(C(c2cccc(Cl)c2F)=O)CC2(CCN(C(=O)C#CC3CC3)C2)O1 20512,c1(SC)ccc(-c2cnnn2C)cc1.c12cscc1C(=O)NC(C)CCNC2=O 20513,C1(NC(CCCN(C(C)=O)C)=O)CCCCN(C(c2ccc(C)[nH]2)=O)C1 20514,C12(C(=O)NCCc3c(CNC(CN(C(C)=O)C)=O)nco3)CCC(C1)C(C)O2 20515,c1(CC2CCN(C(C3(COC)CN(S(=O)(=O)C(C)C)C3)=O)C2)ccc(C)cc1 20516,c1(SC)nc(=NC2CN(C(=O)CC(O)c3ccccc3)CC2CC(C)(C)C)s[nH]1 20517,C1(NC(C2CC(C)(N(C)C)C2)=O)COCCN(C(=O)CCC(=O)OC(C)(C)C)C1 20518,O=C(CS(=O)(=O)C1CC1)N1CCC2(NC(=O)CCC3CC(F)(F)C3)CC2C1 20519,CCCC(C)C(=O)NCc1cccc(NC(c2nnnn2C(C)C(=O)OC)C)c1 20520,N1(C(COCC)=O)CCC(O)(C2(NC(=O)C(C3CCOC3)NC(C)=O)CC2)CC1 20521,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCCC(O)(CNC(c2ncoc2C)=O)C1 20522,C1(NC(C(C)O)=O)CCC2(CC1)CN(C(c1ccc(Br)c(Cl)c1)=O)CCO2 20523,C1(Cl)(C(N2CCOCC(CNC(=O)C=C3CCOCC3)C2)=O)CC12CCOCC2 20524,c1(CNC2CC(C(=O)NCCc3nccn3C(F)(F)F)C2)csc2ccccc12 20525,C12(C(=O)OC)CC(CO)(C1)OC21CN(C(=O)NC2CS(=O)(=O)CC23CC3)C1 20526,C1(O)(CNC(c2c(OCC)cccc2)CC)CCc2ccccc2C1 20527,C(N=c1cc(F)nc[nH]1)C1N(C(C2=CCCN(Cc3nccc(C#C)c3)C2)=O)CCC1 20528,C123CCC(CC1n1cc(nn1)CCC(=O)N2)C3.C1(C(C)(C)SC)CCC(C)O1 20529,Cc1cn2c(n1)C(C)CC(C(=O)NC1CC(F)CN(C(c3cnco3)=O)C1)C2 20530,n1(CC)cc(CC(=O)NCCC(C)NC(c2c(C)coc2C(C)C)=O)c(C)n1 20531,NC12CC(C1)C2c1nc(-c2cc(-c3cnccn3)[nH]n2)no1 20532,C(=O)(CCC(CF)CF)N1CCC(NC(c2c(C(C)C)ncnc2)=O)C(C)C1 20533,CC(F)(F)C(C)(C)C(=O)NCC(=O)NCCC1=CCOCC1 20534,Cc1cc(C(=O)NCCC2CCCN2C(=O)CC23CCCC2C3)c(C)o1 20535,c1(C(=O)NCCCNC(COCC(=O)OC)=O)csc(CCc2ccccc2)n1 20536,C#Cc1cc(COC(C2CC2C2CCC2)=O)ccc1Cl 20537,n1(CC(=O)NCCC(CNC(c2coc(CC)c2C)=O)O)c(C)cc(O)cc1=O 20538,C(N=c1nc2c(ncn2C)c(N(C)C)[nH]1)C1CC(CN(CCC(C)CO)C)C1 20539,c1(C(N(CCCC(=O)NCCC(CC)O)C)=O)cnnc(C)c1 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20557,c1(NCc2cn(C)[nH]c2=N)[nH]c(=NC2CCS(=O)C2)nc2ncn(C)c12 20558,C(=O)(C(C#N)C(C)(C)C)N1C(CCNc2c(C)ccc(C(=O)NC)c2)CCC1 20559,Cc1c(C(=O)NC2(C)CC(NC(=O)CCC3CCCC(O)C3)C2)nnn1C(C)C 20560,N1(CCC(=O)NCCONC(=O)C2(CC3CC3)CC2)CCCCCC1 20561,C(=O)(CC(C)C(C)(C)NC(c1scnc1Cl)=O)NCCn1c(C)ncc1 20562,N1(C(C(C)C2CCC2)=O)CCCOC(CNC(=O)CC2CCCOCC2)C1 20563,CC1OC2CCC1(C(=O)NC1CCC(CCC(=O)NC3CCCC(CO)C3)C1)C2 20564,CC(C)CC(=O)NCC1CC1CNC(=O)C(N1CCNC1=O)C 20565,C1(C(=O)NCc2c(C)ocn2)CCN(C(C2(c3cccnc3)CC2)=O)CC1 20566,c1(NC(C2CCC(C)CN2C(C2CNC(=O)O2)=O)=O)ccc2ccncc2c1 20567,N1(C(C)C)CCCC(C(N2CC(CC(C)NC(=O)C(C)(C)CF)C2)=O)C1 20568,Cn1nc2n(c1=O)CCN(C(=O)NC1(C)CSC1)C2 20569,N1(C(C(C(=O)OC)C)=O)CC2(CCC(C(=O)Nc3oc(C4CC4)cc3C)O2)C1 20570,CC(C)CC(C)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 20571,N1(C(C(c2ccccc2F)OC)=O)CCC(CNC(=O)CCCC(N)=O)C1(C)C 20572,c1(C(C)C)ncc(C(=O)NC2CC(F)CC2NC(=O)Cn2cnnn2)cn1 20573,N12CCC(C(O)C1)C1C(=C)C1C2=O.c1(CNC(=O)C(C2CC2)SC)ccccc1 20574,c1(CNC(CSCCCC)=O)nc(CNC(c2csc(C)c2)=O)cs1 20575,c1(OCC)cccnc1C(=O)NC(CCNC(c1cnc(OC)s1)=O)(C)C 20576,N1(C(C(Cn2ccc(C)n2)C)=O)CCC(O)(CNC(c2ccnc(O)c2)=O)C1 20577,c1(SC)cc(C)nc(N2CCCC2CCC(N2CC(CO)C(F)C2)=O)n1 20578,C(=O)(CCC(C)(C)C)N1C(CNC(C2N(C)C(=O)CC2)=O)CCC1 20579,Cc1ccc(N(C(=O)CNC(C)C)Cc2cccnc2)cc1F 20580,c1(CC(=O)NC2CCCCC2CNC(c2c[nH]c(Br)c2)=O)noc2ccccc12 20581,C1(NC(C(COC)O)=O)CCCCC12CCN(c1ncnc3[nH]cnc13)CC2 20582,Cn1cccc(CNc2ncnc(Cl)c2C#N)c1=O 20583,CC(Cc1cnn(C)c1)C(=O)NCCCNC(=O)C=CBr 20584,C1(CC(=O)NC(CC)C(C)C)CN(C(c2c(C)noc2N)=O)CCO1 20585,c1(C(=O)NCC2CCC(NC(CN(C3CCC3)C)=O)C2)nnn(C)c1C(F)F 20586,C#CCC(C)(CC)C(=O)NCC1CCCCN1C(c1nccc(OC)c1N)=O 20587,N1(C(=O)OC)CC2C(C)C2C1.C1(N(C(CNC(=O)CNC(=O)OC)=O)C)CSCCO1 20588,N1(C(c2c(CC)csc2)=O)CC2CCC1C(CNC(=O)C1=C(Cl)CCCC1)C2 20589,c1(NC(C2N(C(C3(OC)CCSC3)=O)CCCC2)C)c(C)c(C)nc2ncnn12 20590,Cc1cc(C)c(NC(C2(CCn3cc(C(C)N(C)C)nn3)CCC2)=O)cc1Cl 20591,N1(C(CN(C(COC)=O)C)=O)CCN(C(c2coc(C(C)C)n2)=O)CC1C1CC1 20592,N1(C(c2cc(C)oc2)=O)CC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 20593,C(=O)(C(C)CC(F)F)NC(C1CN(C(=O)Nc2ccc(-c3nc[nH]n3)cc2)C1)C 20594,c1(C(=O)NCCn2cnnn2)cn(CCNC(C2CC2C(F)(F)F)=O)cn1 20595,c1(C(N2CC(CN(C(=O)C3=CCCC3)C)C3(C2)CC3)=O)cnc2[nH]ccc2n1 20596,C1(CC)CN(C(c2ccsn2)=O)CCC1NC(c1nc(CC)sc1N)=O 20597,CC(C)CC(C(=O)NCC1CCCC1NC(c1cnnn1C)=O)C(C)C 20598,C1(NC(=O)Cn2ccnn2)CC(F)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 20599,CCC(C)C(C(=O)NCCC1CN(C(c2sccc2SC)=O)C1)OC 20600,c1(NC(C(C)=C(C)C)=O)cccc(CNC(C2CCC(N3CCCC3)CC2)=O)c1 20601,C1(C(=O)NCC2(CC(=O)NCC3(SC)CC3)CC2)CC(O)C(F)C1 20602,CCC(C)(CNC(C)=O)C(=O)Nc1csc(C(=O)NCc2ccc(C)c(C)c2)n1 20603,c1(CCC(=O)NCC(C)N(C)C)ccc(OCC(=O)NC(F)CCOC)cc1 20604,C1(N(C(N)=O)CCO)CCN(C(=O)NC2CC(Cl)(Cl)C2)C1.O=C1CN1 20605,N1(C2C(=O)NC2)CCN2C(=O)OCC2(C)C1.C(C1=CCCOC1)OC 20606,CCC(CC(=O)N1CCC(N(C(=O)CCc2cccc(O)n2)CCO)C1)C(C)C 20607,C1(C)(C(=O)NCc2cc(COC)on2)CCN(C(C2CC(=O)CS2)=O)C1 20608,C1(CCC)(NC(=O)COC2CCCCC2)CCCN(C(C2CCCN2N=O)=O)C1 20609,C1(NC(C(CNC(C)=O)O)=O)CCN(C2CC2)C1=O.C1C(C)(C)OCC(=O)N1 20610,N1(C(c2c(NC(C(OCC)OCC)=O)occ2)=O)CCCC12CCNC2 20611,Cc1cc(F)ccc1C(O)C(=O)NCC12CCC(CN1C(=O)C(N)=O)C2 20612,c1(OCC)cc2ccccc2cc1C(N1CC(NC(c2nc(Cl)cs2)=O)C1)=O 20613,C1(C(=O)OC)CCC2CC1C2(C)C.C12CCN(CC1C)CC1(CC1)CC(=O)N2C 20614,Cc1n[nH]c(C)c1CCC(=O)Nc1cccc(C(N)=O)c1 20615,N1(C(Cc2ccc(C)nc2)=O)CCC2CN(C(=O)CN3CCCCC3=O)C2C1 20616,Cc1ccc(C)c(NC(CCCNC(=O)CCS(C)=O)c2ccccc2)c1 20617,Cc1cc(OC(C)C(=O)N(C2CCCC2)CCSc2cc(Cl)ccn2)cc(C)c1 20618,c1(OCCNC(=O)Nc2noc(C3CC3(F)F)n2)cc(C(F)(F)F)ccc1O 20619,C(=O)(C(C)CCC(C)(C)C)NC(CC)CC(=O)NCC1(CC(=O)OC)CC1 20620,c1(OC)cccc(Cl)c1N(C)C.N12CC(C3(CC3)C1)NC(=O)C2C1CC1(C)C 20621,CCC(C)(COC)C(=O)N(C)CCOCCC(=O)NC1(C#N)CCOCC1 20622,C1(C(=O)NCC(C)CN(C(=O)CC2CS(=O)(=O)C2)C)C2CCC(C2)C1(C)C 20623,N1(C(=O)OC(C(C(C)C)c2ccccc2)=O)CCC(C)C(C(=O)OCCC(C)(C)C)C1 20624,c1(CC)nc(Cl)n[nH]c1=NCC1C(NC(=O)Cc2cccc(Cl)c2F)C2CCC12 20625,C1(N(C(C(c2ccoc2)NC(C(C)c2ccco2)=O)=O)C)CCOC(C)(C)C1 20626,CCCCCC(=O)NCC(=O)NCCC1(C)CCN(C(=O)CN(C)C(=O)C2CC2)C1 20627,c1(C(N(C)CC=CC(=O)N(C2CCN(C)CC2)C)=O)cccc(O)c1F 20628,C(CCC(C)C(c1nnnn1C1CC(F)(F)C1)NCC1(C)CS(=O)(=O)C1)OC 20629,C1(C(=O)NC(c2nc(C(=O)NCC3CCC4CC4C3)co2)C)C2CC3C(C2=O)C13 20630,c1(OC)nccc(C(=O)NCC(O)CN(C(=O)CC2CC3CCC2C3)C)n1 20631,CCCC(O)(CCC)CC(=O)NC1CCC1NC(=O)CSCc1cccnc1 20632,c1(C(=O)NC2C(C)CCN(C(C3N=C(C)SC3)=O)C2C)c[nH]c2cc(F)ccc12 20633,c1(CNC(C2CN(C(C)=O)C2)=O)nc2c(s1)CCN(C(=O)CC1COC(=O)C1)C2 20634,c1(C(=O)NCCCCNC(C(CC=C)OC)=O)ccc2c(c1)CC(C)(C)C2 20635,CP(C)(=O)c1ccc(NC(c2ccccc2)COc2ccc(OC(F)F)cc2)o1 20636,c1(CN2CCC(C(=O)Nc3c(OC)cccc3O)C2)c[nH]c2ncccc12 20637,C1(c2cn(C3CC(C(=O)NCC4N(C(C)C)CC4)C3)nn2)CCN(C)C1=O 20638,C12(C(N(CC#C)CC#C)=O)CCC(CC1)N(C(c1cn[nH]c1)=O)C2 20639,c1(CNC(CC2C(CNC(C(CC)SC)=O)C2)=O)ccc(C)cn1 20640,c1(NC)ccc(NC(=O)C(=O)NC(C)CC(c2ccccc2C(F)(F)F)O)cc1 20641,n1(CC(=O)NC(CNC(C(C)C2(O)CCC2)=O)(C)C2CC2)ncc2cccnc12 20642,C1(C(=O)NCC2CCCCC2)(CNC(c2ccc[nH]2)=O)CC12CCC2 20643,N1(C(C(CC=CCC)C)=O)CCC(CNC(C2CC=CCC2)=O)C1(C)C 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20662,N1(CC=C)CC(C2CCCN(C(=O)Nc3cc(C)nc(N4CCCC4)n3)C2)C1 20663,N1(C(CC2C(C)C2)=O)Cc2ccccc2C(NC(c2cc(CO)n(C)n2)=O)C1 20664,C1(NC(c2ccc(C)cn2)=O)CC(O)CN(C(C2(C)C(C)(C)C2(C)C)=O)C1 20665,c1(CCC)[nH]ccc1C(=O)NC(C1CC=CCC1)C(=O)NCc1ccco1 20666,c1(CCC(=O)NCCC2(NC(C3CC(=C)C3)=O)CC2)cccc(F)c1 20667,N1(C(c2cn(CCC)nc2)=O)CC(CNC(C23CC(COC)(CO2)C3)=O)C(O)C1 20668,c1(OC)ccc(CC(=O)NCC2CC2NC(=O)CCn2cncn2)cc1 20669,CC1CCN(CC(=O)NCC=CCNC(=O)COC2CCCCCC2)CC1 20670,c1(C(c2ccccc2)OC)nc(-c2nc(Cl)oc2C)n(Cc2ccc(Cl)cc2)n1 20671,C1(CNC(C(CC)(C)C)=O)CN(C(C2CCN(C(C)=O)CC2)=O)C2CCN1C2 20672,N1(C(C(C)=C2CC2)=O)CCC(CO)(CNC(C2CCC2(F)F)=O)C1 20673,c1(C(=O)NCC(=O)N(c2ccccc2C(F)(F)F)C)ccc(S(C)=O)cc1 20674,Cn1cc(C(=O)NCC2CC2NC(c2ccccc2Cn2ccnn2)=O)ccc1=O 20675,c1(C(N2CC(CNC(c3c(C)cns3)=O)C3(C2)CC3)=O)cc2c(C)cccc2o1 20676,C1(CC)CCN(C(c2cccc(O)c2)=O)C1C(=O)N(CC(C1CC1)OC)C 20677,C(=O)(CCS(N)(=O)=O)N1CC(CC)C(C(=O)N(CC(O)COC)C)C1 20678,C1(CNC(c2c(OCC)n[nH]c2)=O)CCCN(C(=O)CN2CCS(=O)(=O)CC2)CC1 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20696,CCC(C)(CCC(=O)N)C(N)=O.n1(CC(=C)Br)c(-c2ccc(OCOC)cc2)csc1=N 20697,c1(C(N2CCN(C)CC2)CCNC(N2C(CC)CCC2)=O)ccc(C(F)(F)F)cc1 20698,c1(C(N2CCCC(CNC(c3c(C)ccn3C)=O)C2)=O)ccc2[nH]ccc2n1 20699,c1(CC)noc(CC)c1CC(=O)NC1(CNC(c2cncnc2)=O)CCC1 20700,C1(OC)CCC(CNC(=O)CCN(C(=O)CC2CCCC2)CCO)C1 20701,C1(O)(C(C(=O)Nc2cn(COC)nc2)=O)CCOCC1 20702,c1(SC)ccccc1C(=O)N(C)CCN(C(=O)CC1CC(C)(C)CO1)C 20703,C1(C(=O)NC2(C)CCN(C(C3C(OC)CCCC3)=O)CC2)CNC(=O)C(C)(C)C1 20704,c1(CC)c(C(=O)NCCC(C)NC(c2cn(C)nc2CC)=O)oc2ccccc12 20705,c1(CC(N2CC(NC(C(CCC)C)=O)C3(C2)CCC3)=O)cn2cc(F)ccc2n1 20706,C1(CNC(C(CC)O)=O)CN(C(c2cnn(C(C)C)c2)=O)CCCO1 20707,N1(C(C2CN(C(C)C)C2)=O)CCC(C(O)CNC(C2CCSC2)=O)CC1 20708,c1(CNC(=O)CCCC2CCS(=O)(=O)C2)ccc2ncsc2c1 20709,C(=O)(C(Cc1ccccc1)C1CC1)N(CC(CN(C)C(C1COC(=O)O1)=O)O)C 20710,c1(C(N2CC(CN(C(=O)CC3CC(N(C)C)C3)C)C2)=O)coc(CN)n1 20711,C1(CC(C)(C)N(C(=O)CC2(O)CCCOC2)CC)CCCCN1C(=O)C#CC1CC1 20712,c12cccc(c1)O2.C1(C(=O)NC(C)CCCNC(=O)C(=O)NCC)(OC)CCOC1 20713,CN1CCC(C(c2nncs2)NC2CC2)C1 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20784,c1(CCC(=O)NC(CNC(c2nc(C(C)=O)sc2)=O)CO)ccc(CO)cc1 20785,C1(NC(c2nc(OC)oc2)=O)CCCN(C(=O)Cc2c(N)nc(C)nc2O)CC1 20786,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20787,c1(C(=O)NCC(C(C)C)NC(=O)CCCCN2CCCC2)nnc2n1CCOC2 20788,c1(CC(=O)NC(C(=O)N(CC#C)C)CC2CCC2)ccccc1C 20789,C(=O)(C(C)(C)C(C)O)N1CC2C(C(N(C)CCC3CCCCO3)=O)C21 20790,C12(CNC(CCC#C)=O)CC(CN1C(=O)C(C1CCCCC1)F)C2 20791,c1(OC)c(OC)cccc1C1=CCN(CC(C2CCC3C2C3(F)F)=O)CC1 20792,c1(OC)ncc(C)cc1C(N1CC(NC(c2c(C)ncn2C)=O)CC(O)C1)=O 20793,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20794,c1(OC)ncc(C)cc1NC(=O)CCC(C)NC(C1CCC(C2CC2)C1)=O 20795,N1(C(c2n(CCC)ccc2)=O)CCC(C)C1CNC(=O)CCSCC(C)C 20796,c1(C(=O)NC(C2CCN(C(C34CC(C(F)(F)F)(CO3)C4)=O)C2)C)cnccc1Cl 20797,c1(C(=O)NC2(CNC(C(C)C(C)O)=O)CC2)c(F)cc(F)cc1Br 20798,C1(C(N2CCN(C(=O)CNC(=O)C(C)N(C)C)CC2)=O)(NC(C)=O)CCC(C)CC1 20799,C(=O)(CCCCNC(N)=O)N1C(C(C)NC(c2ccc(OC)s2)=O)CCC1 20800,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20801,n1(CC2CCN(C(C(n3cc(CC4CC4)nn3)C)=O)CC2)nc(C2CC2)ccc1=O 20802,CC1(CNC(C2C(NC(=O)Cc3ccnc(O)c3)CC2)=O)CC2CC2C1 20803,C(C(C)(C)CN(C)C(C12CCC1C2)=O)NC(CC1(SC)CC1)=O 20804,C(c1ccccn1)=CC(=O)NC(C1(O)CN(C(=O)CCN2CCOC2=O)C1)C 20805,N1(C(c2cnn(CC)n2)=O)CCC(C)C(NC(C2CCC(C)(C)O2)=O)C1 20806,C(=O)(C1=C(C)C(C)(C)OC1=O)NC1(CNC(C23OCC(COC)(C2)C3)=O)CCC1 20807,n1(CC(=O)NC2C3CC(NC(C4(C)CCC4)=O)CC32)cccc(O)c1=O 20808,C1(NC(c2nc(CC)sc2)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 20809,c1(C(N2CC3(C(C(=O)Nc4cn(C)nn4)C3)C2)=O)cnc(Cl)c(F)c1 20810,c1(CC)ccc(C(=O)NCC2OCCC2C(=O)NCC(C)(C)OCCO)cn1 20811,c1(NC(=O)Cn2cc(-c3ccc(C(=O)O)o3)nn2)cccc([N+](=O)[O-])c1Cl 20812,C(CCCCCC(=O)N1CC(NC(=O)CCc2ccsc2)CC(C)(C)C1)SC 20813,CC1CN2CCN1CC2C(N1CCN(C(=O)Cn2ccc(O)nc2=O)C(C)C1)=O 20814,N1(C(C2CC2F)=O)CCC(NC(C2(c3ccc(F)cc3)CCC2)=O)CC1 20815,N1(C(Cc2c(C)n[nH]c2C)=O)CCN(C(=O)CCOC2CC2)C(CO)C1 20816,C(N=c1nc(C#N)cc(C)[nH]1)C1(C)CCC(NC(C(=C(C)C2CC2)F)=O)CC1 20817,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20818,c1(OC)cccc(Cl)c1CC(=O)NC(C)CCNC(c1ccnn1CC#N)=O 20819,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(=O)C=Cc1nc(C)c(C)[nH]1)C2 20820,C1(NC(C)=O)CC(C)N(C(=O)CCC(=O)c2ccc(OCC(C)C)cc2)C1 20821,C1(=O)C(CC(F)F)N1.n1(CC)cc(CN(C(=O)C=CC(=O)N(C)C)C)cn1 20822,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1(CF)CCC1)=O 20823,c1(OC)c(C)ccc(C(=O)NCCC2CC(NC(c3cc(C)[nH]n3)=O)C2)c1F 20824,C=CC(C)(CC)C(=O)NC1CC(C(=O)N(CC(O)CN(C)C)C)C12CCC2 20825,C(=O)(C(C)CCC(C)(C)C)N1CCCC(C(C)NC(c2cnc[nH]2)=O)C1 20826,c1(-c2cn(-c3ccc(C(=O)NC(C(=O)NCCC)C)cc3)nn2)ncc(F)cn1 20827,c1(CCC(N2CCC(F)(C(=O)NOCCCO)C2)=O)c(Cl)cncc1Cl 20828,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20829,Cc1ccc(C(=O)NC2CCN(Cc3n[nH]c4c3CCC4)C2)c2ccccc12 20830,c1(NC)ncc(C(N2CCCC(CN(C(=O)C(F)CC3CCCC3)C)C2)=O)cn1 20831,CC(C(=O)NC(Cc1cn[nH]c1)CC(=O)NCCc1cn(C)nn1)C(F)F 20832,C(C(C(=O)N(CCCF)C)NC(c1cc(C(F)F)[nH]n1)=O)N(C)C 20833,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(=O)C(C)n1ccnc1)CC2 20834,C1(N(C(=O)CN2CCOCC2)C)CCC(NC(=O)CC(C)(C)C)CC1 20835,N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)Cc2cn[nH]c2)C2(CC2)C1 20836,c1(-c2scc(C)n2)ccc(OC(F)(F)F)cc1.C(C=C(C)Cl)O 20837,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)C)nc3)C2)=O)nn1C 20838,Cc1cc(CNC(=O)NCc2cnn(C(C)(C)C)c2)on1 20839,C1(CCC(=O)OCC)CCN(C(c2csc(C3CCCNC3)n2)=O)CC1 20840,c1(CC(C)C(=O)NC2CN(C(=O)CNC(N)=O)CC2O)ccc(Br)cc1F 20841,N1(C(=O)CSC(F)(F)F)CCC2(CCCCN(C(c3ccc(F)o3)=O)C2)C1 20842,C1(C(=O)NCCC(C(C)C)NC(C2(C)CC(C#N)C2)=O)CCC2(CCOCC2)O1 20843,C1(C)(NC(C(C)OCC2CC2)=O)CCN(Cc2nc[nH]n2)C1 20844,C1(NC(C2(CC)CCCC2)=O)CCC2CN(C(c3cc(C)cnc3C)=O)CC2C1 20845,c1(NC(C)=O)ccccc1C(=O)NCC1CC1NC(=O)CCc1ccon1 20846,C=C1CC2CCC(C1)N2C(=O)C(CCCC)NC(c1[nH]ccc1CC)=O 20847,CCCCCCCCC(=O)N1CCN(C)C(CNC(C2C3CCC(=O)C23)=O)C1 20848,C1(C(=O)NC2(CC#C)CC2)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 20849,Cc1cc(Cl)c2ccc(C(N3CCC(C#N)(NC(=O)CO)C3)=O)cc2n1 20850,C(=O)(CCC1CCc2ccccc21)N1CC(C)(CNC(=O)COc2ccsc2)C1 20851,C(=O)(C1CC(=O)c2ccccc21)N1CCC(CCNC(C2CCCCC2)=O)C1 20852,c1(N2CCCC3(NC(Cc4ccn(CC)n4)=O)C(C2)C3)nc(O)c2c[nH]nc2n1 20853,C(=O)(CC(C1CC1)NC(=O)CCCN(C(=O)Cc1cncs1)C(C)C)OC 20854,C=C(C)CCC(=O)NCC12CC(NC(c3cn(C4CC4)nc3C)=O)(C1)C2 20855,CCC(C(=O)NCC1CN(C(c2nn[nH]c2C(F)(F)F)=O)C(C)(C)C1)C(C)(F)F 20856,C(CC(C)C(F)(F)F)NC(c1n(CC(C)=S=C)nnn1)(C)CCC1=NC=CS1=CC 20857,C1(C(N(CC(CC)NC(C2CCCN(C(=O)CO)C2)=O)CC)=O)CC(=O)NCOC1 20858,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(NC(=O)CC2CCOC2=O)C1C1CC1 20859,N1(C(Cc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 20860,c1(C(=O)NCC2CCNCC2F)ccn2c(O)nnc2c1 20861,c1(CC(=O)NCC2(O)CN(C(C3CC34CCOC4)=O)C2)cc(F)ccc1Cl 20862,C(=O)(C(O)C(CCC)NC(=O)CC(C)OC)N(C1CCOCC1)CC#C 20863,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 20864,N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CC(C)N(C(=O)CCS(C)(=O)=O)C2 20865,c1(COC)ncc(C(N2CCC(CNC(c3ccc[nH]3)=O)C2)=O)c(=N)[nH]1 20866,c1(CC(=O)NC2(C)CCN(C(C(CC)F)=O)C2)nn(C)c(=O)c2ccccc12 20867,c1(C(=O)NCCN)cn(CCC)nn1.C(=O)(C(C)S)NCC(=C)C 20868,C1(C2(NC(c3cnn(C)c3Cl)=O)CC2)CCCCCN1C(C1CC(=O)OC1(C)C)=O 20869,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 20870,c1(NC(C)CCNC(=O)C(C2CCCCCC2)O)snc(Cl)c1C#N 20871,Cc1nncc(C(N2CC3CCC3(C(=O)NCCCc3nc[nH]n3)C2)=O)c1C 20872,c1(C(=O)NCCN(CC(C)O)C(C2CC23CC3)=O)cn2ccnc2s1 20873,C(=O)(CC1=CCN(C)CC1)NCC(C(N1CCC(C(=O)NCC)C1)=O)OC 20874,C#CC1(O)CC(C(=O)NCCCNC(=O)C(C)Sc2ccccc2C)C1 20875,CCCCCC(C(=O)NC1CC1NC(=O)CN1CCCCC1=O)C(C)C 20876,c1(CC(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)ccc(F)cc1F 20877,c1(C(F)(F)F)ccc(F)c(-c2cnc(C3OCCC3F)[nH]2)c1C(F)(F)F 20878,c1(CNC(C(c2nc(C)[nH]n2)N(C(C)Cc2nccs2)C)=O)ccccc1C 20879,C1(NC(C(C)n2cncn2)=O)CCC2(CC1)CN(CCc1cn3c(n1)SCC3)C2 20880,N1(C(c2cc(C(F)(F)F)cs2)=O)CC2CCC1CN2C(C1CC1Br)=O 20881,c1(C(c2nnnn2C(C)C)OCCOCCOCC(=O)OC)ccc(Cl)cc1F 20882,C(CCOCCO)(C(=O)N1CC(OCC)C1)NC(CCC=C)=O 20883,c1(NC2(CN(C)C(C3CCCCN3C)=O)CC2)nc(C2CC2)nc(=N)[nH]1 20884,C1(C(N2CCN(C(c3cc(C(N)=O)oc3)=O)CC2)=O)CCc2ccnn2C1 20885,Cc1ccc2c(c1)nc(COC(C1CCCC(C)(C)CC1)=O)n2C.C1CC(=O)N1 20886,C(=O)(C1CCc2c[nH]nc21)N1CCC2C(NC(c3c(O)ccc(CC)c3)=O)C2C1 20887,C(CS(=O)(=O)c1ccc(C(=O)OC)cc1)N(C(C(C=CCCC)O)=O)c1ccccc1 20888,C1(CC(=O)NC(C#C)CC)C=CC(NC(=O)CNC(=O)CCCC)C1 20889,c1(C(=O)NCCCN(CC(F)(F)F)C)cnc2ccnn2c1O 20890,FC1CCCCCC1Nc1ccc(OC)cc1 20891,N1(C(=O)OC(C)(C)C)CCC(CC(=O)NC(CNC(=O)CCCF)C(C)C)C1.O 20892,C1(NC(CN(C(COC)=O)C)=O)C(C)CN1C(=O)CN(C)C(C)C 20893,C=CCN=C(NCCc1cc(O)c(O)c(O)c1)N1CCC2OCCCC2C1 20894,N1(C(C(CC)c2cccnc2)=O)CCC(NC(c2cn(C)cn2)=O)C1C(C)(C)C 20895,CC1Cc2cc(C(N3CCCC(CNC(C4(C(N)=O)CC4)=O)C3)=O)ccc2O1 20896,C1(CN2CCCC2)CC2CCC(C1)N2C(=O)CC1(NC(CC2(OC)CCC2)=O)CC1 20897,Cc1nn(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C(C)(C)C(=O)N(C)C)c1Br 20898,C1(NC(c2occ(C)c2)=O)CCCCC1NC(C1CCC(C(N)=O)O1)=O 20899,c1(OC)ccc2nc(C(C(=O)NC(C)(C)C)N(c3ncc[nH]3)C)ccc2c1.C1CO1 20900,C1(C(N(CC(CC)NC(c2c[nH]nc2-c2ccco2)=O)C)=O)C(C)C1(F)F 20901,N1(C(Cc2ccc(C)s2)=O)CC2(CC(NCc3cccc(F)c3O)C2)C1 20902,CCCCC(CCCC)NC(C1CC(F)CCN1C(C1CCCC(C#N)C1)=O)=O 20903,CC1(C)CCCC1C1CCN(C(=O)C(N2CCCC3CC(O)CCC23)=O)C1 20904,C1(CNC(C2(NC(C)C)CC2)=O)CCCCC1NC(c1n[nH]cc1Cl)=O 20905,c1(C(N2C(CNC(CC(C)O)=O)COCC2)=O)cc(Cl)cnc1Br 20906,c1(OCC)ccc(C(=O)NC(C)(C)C(C)NC(c2nccc(C(F)F)n2)=O)cn1 20907,C1(NC(c2n(CCC)ncc2)=O)CCCCN(C(=O)Cc2cnccc2C)C1 20908,CC1(F)CC(N=c2[nH]c(N3CCC(C4CC4)CC3)nc3c(F)cccc23)C1 20909,C(N=c1nc(N2CC(=O)NC3(COC3)C2)c2c([nH]1)CCCC2)C1(C)C(C)(C)C1 20910,C1(C(=O)NC2CC(CC)OCC2)CCN(C(c2cn(C)nn2)=O)C12CC2 20911,c1(C(C(C)C)OC)nc(-c2cccnc2)nn1C1CCCCC1 20912,CC1(C)NC(=O)CCC1OC(c1cc(C2CCCO2)on1)=O 20913,c1(OC)cc(F)c(C(=O)NCC2COCCN2C(C2CCC2C(F)F)=O)c(Cl)c1 20914,c1(C(=O)O)nc2ccccc2nc1SC1CCNCCC1(F)F 20915,c1(C(C(=O)N(C2CCCC2)C)NC(C)=O)cc(F)ccc1C 20916,C1(C2CCN(C(=O)C3=CCCSC3)CC2)(NC(C(C2CCCOC2)OC)=O)CC1 20917,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 20918,c1(C2C(NC(CSC)=O)C2)ccccc1C(=O)NOCC(=O)OC(C)(C)C 20919,c1(OCC)cccc(C(=O)NC(C2CCN(C(=O)Cc3conc3C)CC2)C)c1 20920,c1(C(=O)NCC2(C(N)=O)CN(C(=O)Cc3n[nH]c(=N)s3)C2)cnc2c[nH]nc2c1 20921,CC(CC(=O)N(C1CC(N(CC(N2CCCC2)=O)C)C1)C)C(F)F 20922,Cn1cncc(C(=O)NC2CCCC2NC(=O)CSCCN(C)C)c1=O 20923,c1(C(N2Cc3c(C(N)=O)n[nH]c3C2)=O)ccc2c(c1)CN(C(C1CC1F)=O)C2 20924,N#Cc1ccc(C(N2CCCC2C2CCN(C(c3cnc(Cl)cn3)=O)C2)=O)cn1 20925,N1(C(CCCc2c(C)ccs2)=O)CC(CO)OCC1CNC(=O)COC1CC1 20926,C(CCCCCCCO)=CC(N1CC(CCNC(CCCC#C)=O)C1)=O 20927,N1(C(CCN2CCN(CC)CC2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 20928,C1(C(=O)NC2(CCCNC(c3c(SC)ccs3)=O)CC2)CN2CCN1CC2C 20929,CCC(C)(COC)C(=O)N1CCC(CCNC(c2cnsc2)=O)(OC)CC1 20930,C(=O)(CC(O)c1ccccc1)NC1C(NC(C(F)=CCC)=O)CC1 20931,CC1CCC(=O)N1NC(=O)C(C)OC(c1cncn1-c1ccccc1)=O 20932,Cc1cc(OCCCN2CCCCC2)ccc1N1CCCCC1=O 20933,C=CCC(C)(C)CCNC(C1CCOC1CNC(=O)C(C)(C)CC1CC1)=O 20934,N1(C(c2c(CCC)nns2)=O)CCN(C(=O)COc2ccc(CC)cc2)CC1C 20935,C(=O)(C1CCCn2cncc21)NC(CNC(c1sc(C)c(O)n1)=O)C 20936,C(=O)(C(O)CC(C)C)NC1CCC(N(C(CCOCCOC)=O)C)CC1 20937,S(=O)(=O)(c1cccc(N2CCSCC2)n1)N1CC(C)C(F)C1 20938,N1(C(C2OCCN(C(c3c(C)nc(O)s3)=O)C2)=O)CCOC(C)(C)C1C 20939,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCN(C(=O)CC#N)C(C)C1.C(=O)C(F)F 20940,C(=O)(C(C)(C)C(=O)NCCc1ocnc1CNC(=O)C1=C(Cl)CCC1)OCC 20941,C1(C(N2CC=CC(NC(=O)C(F)(F)CO)C2)=O)CCCCC1 20942,c1(N(C)CC2CN(C(C3(CC)CCCCO3)=O)C2)cc(C)nc2ncnn12 20943,n1(CCC)ncnc1C(C)Oc1cnn(-c2ccccc2OC)c1 20944,N1(C(CS(CC)=O)=O)CC2CCCC2(C(=O)NC(CC2CC2)C(=O)OC)C1 20945,CC1CCN(C(c2c(Cl)n[nH]c2C2CC2)=O)CC1NC(=O)CC12CCC(CC1)C2 20946,CC(C)C(C(=O)NC1CC(OCC(=O)NC2CCCN3CCCC23)C1)C(C)C 20947,CC(C(=O)N1CC2(CC2)CC1CNC(=O)Cc1cncn1C)C(C)(F)F 20948,C1(=O)C(C)(CC)C(=O)NCC(=O)N(C)C1CCNC(C(CCSC)C(C)C(=O)OC)=O 20949,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(c2ccnn2C2CCC2)=O)CCN1C 20950,C(=O)(CCCCCCS(N)(=O)=O)NCCn1cc(CNC(C(C(C)C)SC)=O)nn1 20951,C1(C(N2CC(OC)C(C(N3CCC(N(C)C)C3)=O)C2)=O)CCC2(CC1)CC2 20952,c1(C(N(C2CCN(C(=O)CC=C(C)C)C2)CC)=O)n[nH]c2c1CCC2 20953,C#CCC(O)C(=O)NCC1(C)CC1C1CCCCN1C(=O)CC1CCCCC1 20954,S(=O)(=O)(CC(=O)N1CCC(CCNC(C2CC(C)(F)C2)=O)CC1)NCC 20955,c1(C(=O)NCCOCCC=C)c(OC)cc(OCC(C)C(=O)OC)cc1OC 20956,N(C1CCSc2ccc(Cl)cc21)c1ccc(-c2nc(=N)[nH]cc2)c(F)c1 20957,C(CC(N)=O)(C(=O)NCCNC(c1cc(C(C)C)on1)=O)NC(CC(C)C)=O 20958,C1(NC(CNC(CC2(C)CN(C(C(C)OC)=O)C2)=O)=O)CCCN(C(C)=O)C1 20959,c1(CC)ncccc1NC(=O)C(C1CCN(C(c2[nH]c(C)nc2C)=O)C1)C 20960,C1(CNC(Cn2cc(C)c(C(F)(F)F)n2)=O)CCCN(C(=O)C(O)C(C)C)CC1 20961,C1(CN(C(C=COCC)=O)C)CN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)CCO1 20962,c1(NC(CC2(C#N)CN(C(C3CCSCC3)=O)C2)=O)nc2ccccc2s1 20963,N1(C(C2(C(C)C)CC2)=O)CCC1C(=O)NCc1cnn[nH]1 20964,c1(C(=O)NC2(CNC(c3cn(CCC)nn3)=O)CC2)ccc(F)cc1F 20965,C12CN(CCC1NC(c1cnc(C(C)O)s1)=O)C2=O.C1(C)(CC)CCC(=O)C1 20966,c1(C(N(CC(C)(C)NC(C2(F)CCS(=O)(=O)C2)=O)C)=O)cc2n(n1)CCCN2 20967,Cn1nc(CNC(C2CC(O)C(F)C2)=O)cc1C(=O)NCC1(C)CCCO1 20968,c1(-c2cc(OCCC)ncc2)cc(C(=O)Nc2ncncc2Cl)c2[nH]ccc2c1 20969,N1(C(CCSCC)=O)CCC(C2CCC2)(CNC(c2cc(=O)n(C)o2)=O)CC1 20970,CC(C)C(C(=O)N1CCCCC1CCN(C(=O)CCN(C)C)C)n1cnnn1 20971,CN1CCCC(O)(CC(=O)NC(C)(CNC(c2cc(Cl)ncc2O)=O)C2CC2)C1 20972,c1(CC(=O)N(C2CC(NC(C3COC(=O)N3C)=O)C2)C)ncncc1Cl 20973,C(CS(=O)(=O)N1CCC(F)(F)C1)(C1CCOCC1)OC 20974,CC(C)C(C(=O)N1CC(CNC(=O)NCc2cccc(Cl)c2)C1)c1ccn(C)n1 20975,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 20976,C1(CNC(c2c[nH]cc(F)c2=O)=O)CC2COCC2N1C(c1ccc(C2CC2)s1)=O 20977,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CC(=O)C2)=O)CC1 20978,C1(COC)C=CCCN1C(=O)CC=CCNC(=O)C(CC)N(C)C 20979,N1(C(C2CCCN(CCC)C2)=O)CC(NC(=O)C(=O)NCC(F)F)CC12CCC2 20980,C1(NC2CC(c3nnnn3C)(NC)C2)CNC2(CCC2)C1 20981,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(c2cc(N(C)C)no2)=O)CC1C 20982,Cn1c(CC(N2CC3CC3(NC(=O)C3=C(C#N)CCC3)C2)=O)cc2ccccc12 20983,N1(C(C(C2CCC2)OCC)=O)CCC(C)(CCNC(c2c(Cl)nsc2Cl)=O)C1 20984,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 20985,C1(O)(CCNC(C(C=C)(F)F)=O)CCCN(C(C2(CSC)CCC2)=O)C1 20986,c1(C(=O)Nc2ocnc2-c2cn(CC3CCCOC3)nn2)ncc(Br)cc1F 20987,CC1CCN(C)C(C)C1.c12nnnn1CCNC2C1C2COCC12.C1CC1 20988,C(=O)(C(C)(F)C(C)(C)F)N(c1cn(Cc2ccc(OC)c(C)c2)nc1)C 20989,N1(C(C(C)NC(CC)=O)=O)CCC(O)(CNC(=O)C=CC(=O)OC(C)(C)C)C1 20990,C(CNC(=O)C(F)F)(CC(F)(F)F)NC(c1cc(-c2ccc(F)cc2)no1)=O 20991,Cc1sc(O)nc1C(=O)NCC(C12CCC(CC1)C2)NC(C1CCC(O)C1)=O 20992,c1(C(N(CCCCCNC(C2CC2(F)Cl)=O)C)=O)cccc([N+](=O)[O-])c1Cl 20993,CCCCCCCC(=O)NCC1(F)CCN(C(c2sccc2COC)=O)CC1 20994,C(c1ccn2ccccc12)=CC(=O)NCC1COCCN(C(C2(C)CSC2)=O)C1 20995,c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)F)csc2c(F)cccc12 20996,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 20997,N1(C(C(n2c(C)ccn2)C)=O)CCC(CCNC(=O)Cc2ccsc2)CC1 20998,CCS(=O)(=O)CC(=O)NC1CCN(C(=O)CSc2ccc(OC)cc2)CC1C 20999,C1(C(=O)NCC(C)NC(=O)COCC2CCOCC2)Cc2ccccc2S1 21000,c1(NC(C2CCCCO2)=O)ncsc1Cn1cc(CCc2ccccn2)nn1 21001,C(=O)(C1CCCc2scnc21)NCC(C)N(C(c1ncc(C)cc1F)=O)C 21002,C(=O)(CC(O)CC(C)C)N1CC(N(C(c2c(OC)ccs2)=O)C)C(O)C1 21003,N1(C(c2ccc(C(C)=O)o2)=O)CCCC(C(=O)NC2(N3CCOCC3)CC2)C1 21004,CC1(C)NC(=O)OC12CCN(CC1CC1c1ccc(Cl)cc1Cl)C2 21005,N1(C(c2cncc(C)n2)=O)CCC2CN(C(=O)CC3CCCOC3)CC12 21006,c1(NC(=O)NCC2(c3cccn4ccnc34)CC2)ccc2[nH]c(=O)ccc2c1 21007,C1(C(=O)NCCN(CCC)C(c2cnn(C3CC3(F)F)c2)=O)CC2CCC1CC2 21008,N1(C(c2nc(-c3ccc(C)o3)oc2)=O)CCOCC1CNC(=O)C(C)C#N 21009,CCC(CC(=O)N1CCC(NC(=O)Cc2ccon2)C(O)C1)C(C)C 21010,C12(CNC(C(C)OCC)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21011,N1(C(C2C(C(C)=O)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21012,C1(CNC(=O)CC2(O)CC2)CCN(C(C2(Cc3ccc(Cl)cc3)CCC2)=O)CC1 21013,c1(C(N2CC(C)(CNC(c3cccc(OC)c3N)=O)C2)=O)ccn2cnnc2c1 21014,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21015,N1(C(=O)CCCC(F)F)CCCN(C(C2(CCc3ccc(Cl)cc3)CC2)=O)CC1 21016,C1(CNC(C2(C)CC2)=O)CN(C(=O)COc2ccc(CO)cc2)C2(CCC2)C1 21017,c1(C(N2C(C)CCC(CNC(CC(C(=O)OC)C)=O)C2)=O)ccn2cncc2c1 21018,CN1CCOC2CN(C(=O)C3=CCN(C(C4CCOCC4(C)C)=O)C3)CC12 21019,C=CC1CCC1C(=O)NC1CCCC1C(=O)Nc1cnn(C)c1 21020,c1(C(=O)NCCN(C(c2oc3ccccc3c2Br)=O)CC)ccc2nncn2c1 21021,Cc1noc(Cl)c1CCC(=O)N(C)CC1(NC(C23CC(C#N)(C2)C3)=O)CC1 21022,c1(C(N2C(C)CC(NC(=O)CC3CCOC3)C2)=O)ccc([N+](=O)[O-])cc1O 21023,c1(C(C(=O)NC2CCCC2)N(CC(COC)C)C)ccncc1F 21024,N1(CC(=O)NC(C)C(=O)NCCCN(C)C(C23CC(C)(C2)C3)=O)CCN(C)CC1 21025,c1(CN2C(C(N(c3cn[nH]c3)C)=O)CCCC2)ccc(NCc2cc(I)c[nH]2)cc1 21026,C(=O)(CCCC(=O)NCC(CO)NC(c1cccc(C2CCC2)c1)=O)N(C)C 21027,N1(C(CCSC)=O)CC2CCC(CNC(=O)C(C)(C)c3ccno3)C2C1 21028,C1(CNC(c2cscn2)=O)CN(C(c2ccc(F)cc2F)=O)C2CCN1C2 21029,Cn1cnnc1CCCC(=O)NCC1C=CCN1C(c1cnc(C(F)F)s1)=O 21030,C(C(=O)Nn1cccn1)C1C(C)=NO1.C12(CCCCC1)C(=O)N2 21031,C1(COC)(NC(=O)C(c2ccc(F)c(Cl)c2)C)CCN(C(=O)C2=COCC2)CC1 21032,c1(CC)n[nH]cc1CNC(=O)C=CC(C)(C)NC(=O)C(F)=C(C)C 21033,C1(O)(CNC(C2CC3CC3C2)=O)CCN(C(C2COCCN2C2CC2)=O)CC1 21034,C(CC(C)C(F)(F)F)NC(C(C1(O)CN(C(C2(COC)CCCO2)=O)C1)F)=O 21035,C1(C(N(CCC(C(C)(C)C)NC(=O)C(F)F)C)=O)CC1C1(C)CCOCC1 21036,C(C(CC(C)C)C(=O)NC1(C(=O)NCC#CC(F)(F)F)CC1C)OC 21037,c1(C(=O)NC2CC3(C(NC(c4c(C)occ4)=O)C3)C2)cc2c(o1)CCCC2 21038,C1(NC(C(CNC(=O)OC)(C)C)=O)CCC2(CC1)CC2C#N 21039,C1(COC)(CNC(C2CCC2F)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21040,C(CC(F)F)(C(=O)N=c1ccn(CCO)[nH]1)NC(C1C(C(=O)OCC)CC1)=O 21041,c1(CCC(=O)OCc2ccc(N)cc2)cccc(Br)c1F 21042,c1(CC(=O)NC2C(NC(CC3CC(=C)C3)=O)CC2)cc(OC)c(O)cc1Cl 21043,C1(NC(C=Cc2cc(OC)ns2)=O)CN(C(c2cccs2)=O)C2(CCOCC2)C1 21044,C1(NC(C(=O)N(C)C)=O)CCCC1C(C)(C)C.C12CC1(C)C(=O)N2 21045,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21046,Cc1ccnc(N(C)CCOCCNC(=O)Cn2cc(Cl)cn2)c1 21047,N1(C(c2cnc(C)o2)=O)C(C)CC2CN(C(=O)C=C(Cl)Cl)CC12 21048,C1(C(=O)NCC2(NC(C(C=CC)O)=O)CCC2)(Cc2ccccc2)CCCCC1 21049,c1(C(N2CCC3(CC3(C)C)C2)C(=O)NC(CC)C)ccc(C)c2c1CCC2 21050,N1(C(CCC(CC)C)=O)CC2CCC(C(=O)NC(CC)C3CC3)(C2)C1 21051,CS(=O)(=O)c1cc(C(=O)OC2CCCS(=O)(=O)C2)oc1Cl 21052,N1(C(CC(C(F)F)NC(C(C)OCCOCC)=O)=O)CCC2(CCCO2)CC1 21053,C(=O)(CCC(C)(C)C(=O)NOCC1CCOC1)NC(CCOC)COC 21054,c1(CC(=O)NCC2(O)CC(C(NOC)=O)C2)ccc(F)cc1 21055,c1(CC)cnccc1C(=O)NCCCCCNC(=O)CN1CCC(C(N)=O)CC1 21056,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21057,C1(CNC(C23OCC(C)(C2)C3)=O)CN(C(c2cnsc2)=O)CCC1(F)F 21058,C12CCN(CC1)C2=O.C=CC1(C(=O)N(C)CC2CC(F)C2)CCC1 21059,N1(C(CCSC)=O)CCC(C)(C(=O)Nc2cnn(CCF)c2)C1 21060,CC12CC(NC(C3CCCS3)=O)(C1)C1(CCN(c3ncnc(Cl)c3CO)CC1)O2 21061,c1(C(=O)NC(C)CN(C(=O)CCC2CCCO2)C)cnc(N)cn1 21062,N1(C(c2cccc(CC(C)C)c2)=O)CC(C)C(NC(=O)COC(F)F)C(C)C1 21063,CCC(C)(CCCNC(C)CCC1CC1)n1ccnc1 21064,C1(O)(CC(=O)NCc2ccc[nH]2)CN(C(c2ccsc2)=O)C1 21065,N1(C(C2COCCN(C(c3cc(C)c(O)nc3)=O)C2)=O)CC(C)CCC12CC2 21066,C(=O)(C1=CC2(CN(C(=O)C(F)=CC3CC3)C2)OC1)NCC(N(OC)C)=O 21067,CCCCC(C(=O)NCC1CC(NC(=O)C(c2cnn(C)c2)OC)C1)C(C)C 21068,C1(NC(C(C)(C)F)=O)CS(=O)(=O)CC1NC(c1ccc(C(C)C)c(Br)c1)=O 21069,C1(CC)CN(C(C2CC(C)(N)C2)=O)CC(C)S1=O 21070,N1(C(C2C(CC)CCN2C(c2ccnc(C)n2)=O)=O)CCc2ccsc2C1 21071,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21072,C12(C(=O)OC)CC(C1)C(C(F)F)N2CC12CCOCC1C2 21073,CCCC(CC)CCC(=O)NC1C(C)(C)C(NC(c2cc(OC)cs2)=O)C1(C)C 21074,Cc1ccc2c(c1)CC(C(N1CC(NC(=O)C=Cc3ccc[nH]3)C(C)(C)C1)=O)S2 21075,C(CC(C)CCS(=O)(=O)NC1(c2ccccc2)CC(O)C1)OC 21076,N1(C(CNC(C)=O)=O)CCOC2CCN(C(=O)Cn3cncn3)CC12 21077,N1(C(c2c(COC)nn[nH]2)=O)CC2CC1CN2C(=O)C=CCN(CC)CC 21078,C(C(=O)NCC1CCCCN1C(=O)CC1CCC(=O)N1C)(C(C)(C)C)SC 21079,C1(CC(=O)N(C(C)C(=O)NC2CC(=O)N(CC)C2)CCC)CCC(C)(C)C1 21080,N1(CC(=O)NCc2c(C)occ2)CC(NC(c2coc(O)n2)=O)CCC1C 21081,N1(C(C(CN(C)C)(C)C)=O)CC2(CCC(CNC(=O)CSCc3cscn3)O2)C1 21082,c1(C(N2C(CCC(=O)NC(CCSCC)C)CCC2)=O)cn(C)nc1OC 21083,C(CC(C)(C)C(=O)NC1COCCC1NC(c1cn(C2COC2)nn1)=O)OC 21084,c1(C(N2CCN(C(c3ccc(CC)s3)=O)CC2CF)=O)ccc2cccnc2c1 21085,c1(C(N2CC(C)(NC(C3C(SC)CCC3)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl 21086,C1(C(N(C2CN(C(c3csnc3Br)=O)C2)C)=O)CCCN(c2ccccc2)C1=O 21087,C1(C(N(CC)CC2CC2)=O)CN(C(=O)CCCN(C)C)CC1C 21088,n1(C(C)C)cc(C(C(=O)NCc2cn(C)nn2)N(CCC(O)CO)C)cn1 21089,C(N=c1ccnc(NCC2CCCC3(CCC3)C2)[nH]1)c1cccc(C(F)F)n1 21090,C(=O)(CC(C)(C)N(C)C(C1CCC=CCC1)=O)N(C)CC1CCCCO1 21091,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(C)C2)=O)cnn2c1OCCC2 21092,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(=O)C(CO)OC 21093,N1(C(C(C)SC)=O)CCC(C)C(CNC(c2nccc(Cl)c2C)=O)C1 21094,c1(CC(CO)NC(=O)NC(CC=C)C2CC2)ccc(F)cn1 21095,C1(OC)CC(CCNC(c2nc(C)sc2C)=O)N(C(C2CCSCC2)=O)C1 21096,C=CC1(NC(C23CC2CCN3C(c2sccc2Br)=O)=O)CCCC1 21097,Cc1cccc2oc(C(=O)NC3(CF)CCN(C(=O)CC4CCCCO4)C3)cc12 21098,C#Cc1ccc(F)c(C(N2CCC(CNC(C3CCC(C)(C)OC3)=O)CC2)=O)c1 21099,c1(C(CN(C(=O)OCCn2c(C)ncc2)C)=O)ccc(S(C)=O)cc1 21100,N1(C(C(C)Cc2ccccc2)=O)CC2CN(C(c3coc(O)n3)=O)CC2C1 21101,C(CCCC(=O)NCC(C)(C1CC1)NC(C1CC1(C)C(C)C)=O)N(C(C)C)C 21102,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21103,c1(OC)ccc(C(=O)NC2CN(Cc3cc(C)c[nH]3)CC2F)c(C#N)c1 21104,C(CCN(C)C)(C(=O)NCc1cn(C)cn1)NC(COCC)=O 21105,C=CCC(C)(CC)C(=O)N1CC(CCNC(=O)CC2(C)CCOCC2)C1 21106,C(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(c1[nH]cc(C)c1C)=O 21107,C(=O)(C(CC(F)F)NC(c1cccn1C)=O)NC(c1ncccn1)CC 21108,CCC(C)C(O)C(C)C(=O)NC1C2CCC(C2)C1C(=O)NC1CC(=O)N(O)C1 21109,C1(CNC(CC(C)OCCC)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21110,C1(C(=O)NCCCNC(C2CC(O)(C(=O)OC)C2)=O)CC2CC(C1)CC(F)(F)C2 21111,CCCC(C)(C)CNC(=O)CC1(OC)CN(C(C2CCCCC2C)=O)C1 21112,c1(C(N2C3CCC(NC(=O)C=Cc4cc[nH]n4)(C3)C2)=O)ccc2[nH]ccc2c1F 21113,c1(CN2CCCC(N(C)C(c3ncccc3C(F)(F)F)=O)C2)ccc(Cl)nc1Cl 21114,C(c1ccc(C2CC2)cc1)=CC(=O)NC1CC(NC(=O)CC2CCCS(=O)(=O)C2)C1 21115,C#CCC(O)C(=O)NCCn1cnc(C(=O)NC(CCOC)C(C)C)c1 21116,CC1CN(C(c2cn(-c3ccccc3)cn2)=O)CC(C)CN1C(C1CC1(F)F)=O 21117,C(C1Cc2ccccc21)NC(C(CCC=C)NC(=O)Cn1ccnc1)=O 21118,Cc1c(NC(=O)CC2CCN(C(=O)Cc3cccnc3)CC2)cnn1C1CC1 21119,c1(C(N2CCC(COC)(NC(c3cncs3)=O)C2)=O)c(C)oc2nc(Cl)ccc12 21120,C(=O)(CC1=CCCC1)NC(C(=O)NCc1snc(C)n1)CC1CCCC1 21121,C1(C)(C(=O)NC(C)CN(C)C(C2(NC(N)=O)CCC2)=O)CCc2ccccc2C1 21122,C1(CNC(c2c(C)nc(CO)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21123,C1(C(=O)NC2CCCCC2NC(C)=O)(NC(CCCCOC)=O)CCC(C)(C)C1 21124,C1(NC(CC(C)OC)=O)CCC(C)N(C(=O)C=CC2CC2)C1 21125,c1(C(=O)NC2CCN(C(CCc3ccc(C)cc3C)=O)C2)ccc2snnc2c1 21126,c1(OCC)ccc(Br)c(NNC(=O)C2Cc3c(F)cccc32)c1 21127,C(O)(CCNCC(CC(C)C)N(C)C)(C(F)(F)F)n1cc(C(CCC)=O)nn1 21128,c1(-c2nc(CNC(c3ccno3)C)sc2)cccc(Br)c1 21129,C1(NC(C(CC)C)=O)CC(NC(c2sccc2CO)=O)C(O)C1 21130,N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21131,CCCCC(C)CCC(=O)N(C)CC1(CNC(=O)CC#N)CC1 21132,c1(CCN(CCNC(CCCCC)=O)C(c2ccccc2)=O)cc(F)cc(Cl)c1 21133,Cc1cncc(-c2cccc(CNC(=O)C(C3(O)CCCC3)Br)c2)n1 21134,N1(CCC)CCCCC1C(=O)NCC1CC1C(=O)NC(c1nnnn1C)C 21135,CC1CN(c2nnc(CC(=O)N(C3CCC3C)C3CCCC3)n2C2CC2)CCS1 21136,CC(C)(O)C(F)C(=O)N1CCOC(C(=O)NCCC2CCCCO2)C1 21137,C(=O)(CCO)N(CC(=O)N)CCOC1CC1.c1(C(C)N(C)C)ccsn1 21138,c1(OC)cccc(-c2cc(C(=O)NC3(CNC(C4CCN(C)C4)=O)CC3)n[nH]2)c1 21139,c1(C(=O)NCC2(C(N(CC(O)CO)C(C)C)=O)CC2)csnc1Cl 21140,C1(C(=O)OCC)CCCCCC1n1cc(C(C2CCCNC2)C)nn1 21141,S(=O)(=O)(c1cnn(C)c1)N1C(C(=O)NCC2CCN(C(COC)=O)C2)COCC1 21142,C1(NC(COC2(C)CCCC2)=O)CC2C(NC(c3nocc3Cl)=O)C2C1 21143,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CCCC2)C1 21144,c1(C(=O)NC2C(NC(COCCCCC)=O)CCC2)c2ccccc2nn1C 21145,c1(OCCC(=O)NCC(C)NC(C2(n3ccnn3)CC2)=O)ccc(Cl)nc1 21146,CC(CNC(C1(Cc2ccccc2)CC1)=O)(CO)NC(=O)CC(F)F 21147,c1(CC(C)C(=O)NCCCCCCNC(C2(C#N)CC2C)=O)c(Cl)cccc1Cl 21148,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C1C=CCC1)=O)(C)C 21149,C(CC(=O)NC(Cc1cn[nH]c1)C(=O)N(C1CC(C(=O)OC)C1)C)(C(C)C)OCC 21150,c1(C(=O)NC2(CCOC)CCN(C(C3(C)CCC(=O)N3)=O)C2)ccnc(Cl)c1O 21151,C1(NC(C2(CNC(=O)CC3CCCC3)CCCO2)=O)CCCCCC1F 21152,c1(-c2onc(C3(C)CC3)n2)nc2ccccn2c1F 21153,c1(CC)cc(C(=O)NCCSCC(=O)NCC2(C#N)CC2)no1 21154,c1(C(N2CCN(C(C(CC=C)CC)=O)C(C)CC2)=O)cc(Cl)cc2cccnc12 21155,N1(c2snc(CC)n2)CC(C2CCCCN(C(=O)CC3(C)CCCO3)C2)C1 21156,S(=O)(=O)(c1[nH]c(=NC2CCCC(C(C)(C)C)C2)ccc1Br)NCCCOC(C)C 21157,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21158,CCC(CC)CCCC(=O)N(CCCNC(C1COCCN1C)=O)C 21159,N1(C(COCC)=O)CC2CCCCC2(CNC(c2cccc(C(F)F)n2)=O)C1 21160,C#CCC(O)C(=O)NCCCN(C(=O)C(O)(c1ccccc1)C1CCCC1)C 21161,N1(C(C(CCCC)C)=O)CCCCCC(NC(=O)CN2CC(C)C2)C1 21162,Cc1cncnc1N1CCC(C(=O)NCC(C2CCCCO2)(C)C)CC1 21163,C1(NC(C(c2ccccc2)N(C)C)=O)CCCC1NC(=O)C(C)(C)c1cc[nH]n1 21164,C1(CNC(C2CC(CCC)C2)=O)CC(C)CN(C(c2cn(CCO)nc2C)=O)C1 21165,NS(=O)(=O)C1(C(=O)NCC2(O)CCN(C(=O)Cn3ccc(C4CC4)n3)CC2)CCC1 21166,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21167,N1(C(C(C)n2cncn2)=O)CCN(C(c2cc(Cl)ncc2N)=O)C2COCC12 21168,O(NC(=O)C(C)CNC(C1CCCC(OC)CC1)=O)CCOC 21169,C1(SCC(C23CC(CO2)C3)N2CC(n3cc(C(C)(C)C)nn3)C2)CCCCC1O 21170,C1(O)(CC=C)CCN(C(=O)C(CO)N(C(=O)CSCC)Cc2cscn2)CC1 21171,c1(C(N2C(C)C(NC(c3coc(Br)n3)=O)CCC2)=O)nc2ccccc2o1 21172,c1(OC)cc2nc(n1)N1CCC(C1)CC(=O)N2.c1(C(=O)OC)nnn(C)c1C 21173,Cn1nc(C(F)(F)F)c(Br)c1CN1CCCCC1c1ccc(Br)cn1 21174,C1(NC(=O)CCN(C(=O)Cc2c[nH]ccc2=O)CC2CC2)CC(=O)N(C2CC2)C1 21175,C1(C)(CNC(C(C)OC)=O)CCC(NC(C2(F)CCCC2)=O)C1 21176,C1(C(N(C2CCCCC2)CCC)=O)CCOC1CNC(=O)C(C1CC1)OC 21177,C1(C(N2C(C(=O)NCCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21178,C1(NC(=O)CCn2ccnc2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21179,c1(OC)cccc2scc(C(N3CCC3CNC(C3CC34CC4)=O)=O)c12 21180,c1(C(N(CCOC)C)C)[nH]c(=N)ccc1-c1ccc(-n2cnnn2)s1 21181,C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(C(CC)C(C)C)=O)CCC1 21182,C(CSC)(C(F)(F)F)NC(C(C1CCCC1)OCc1c(C(=O)OCC)occ1)=O 21183,c1(OC)ccc(C(N2CCC(O)C(C(N3CCC(C)CC3)=O)C2)=O)cc1Cl 21184,C1(NC(c2c[nH]nc2C2CC2)=O)CC(NC(c2ccc[nH]2)=O)C12CCOCC2 21185,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CCC1F 21186,CC(C(=O)NCC1CCN1C(c1cncc(C(F)(F)F)n1)=O)C(C)(F)F 21187,c1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCC2)=O)cccc(C#CCO)c1 21188,C1(C(=O)NC(C2CCCN2C(C2CC(F)C2)=O)(C)C)CCC2(CC1)OCCO2 21189,C1(CNC(C=C(CC)CC)=O)(COC)CCCN1C(C1(CCF)CC1)=O 21190,C1(C)(C(=O)NC(C)CN(C)C(C2CCN(C)S2(=O)=O)=O)CCC(F)(F)CC1 21191,C(=O)(CC(=O)N(CC(C)CNC(c1cocc1C)=O)C)OCC 21192,N1(C(C)Cn2nccn2)CCN(C)CC(O)C1.C12(CCOCC1)C(=O)N2 21193,N1(C(C(C)(C)CF)=O)CCCC(O)(CNC(C2CC23CCC3)=O)CC1 21194,c1(C(N2C(CNC(C3N(CC)CCCC3)=O)CC(O)C2)=O)cc2cccnc2s1 21195,c1(NC(c2ccccc2)CCC)nccc(NCCC2(COC)CC2)n1 21196,O=C1CC2(CCOC2)C(C(N2CCCC23CCN(C(c2ccoc2)=O)C3)=O)CN1 21197,c1(C(N2CC(C)N(C(=O)CC3COCCOC3)CC2)=O)cc2c(cn1)CCCC2 21198,c1(CCNC(C2CCCN(C3CCNC3=O)C2)=O)ccc(I)c(F)c1 21199,C1(OC)CN(C(=O)C(C)C(=O)OC(C)(C)C)CCC1NC(=O)C(O)C(C)(C)C 21200,C(=O)(CC(C)(C)CCOC)NCC(CC(=O)N(N1CC(C(=O)NC)C1)CC)C1CC1 21201,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)COC(F)F)CC1O 21202,C(=O)(C1CCCc2cncn21)NCC1C2CN(C(c3c(C)cc(N)cc3)=O)CC21 21203,c1(C(N2CCC(C(=O)NCC3C(C(C)=O)C3)CC2)=O)ccc2c(C)nn(C)c2n1 21204,c1(-c2cc(C(N3CCC(C)(O)C3)=O)c(Cl)nc2)ccc(S(=O)(=O)NC2CC2)cc1 21205,C1(NC(CCCN(C(C)=O)C)=O)CN(C(=O)C#CC(C)C)C(C)(CC)C1 21206,Nc1ccc2c(C(N3CCCC3CNC(c3nccnc3Cl)=O)=O)c[nH]c2c1 21207,C1(C(N(CCCC(=O)NC2CCC2)C)=O)CCC=CCCC1.C(CCO)N 21208,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(CO)CCC2)=O)cc1Cl 21209,C1(C(=O)OCC)N(c2ccc(C(F)(F)F)nn2)CC12CCCC2 21210,N1(C(c2c(C)nc(CC)o2)=O)CCOC(C)(CNC(=O)CCOC2CC2)C1 21211,N1(C(C(C=C=C)C)=O)CC2CC(NC(c3n[nH]c(C)c3O)=O)C(C2)C1 21212,N1(C(CS(CC)=O)=O)CC(S(=O)(=O)N2CCCC2CNc2ccoc2)C1 21213,C(=O)(CCC(N)=O)N.N1(C(CC2(C(C)(F)F)CC2)=O)CCC(c2cn(CC)nn2)C1 21214,C1(c2c(Cl)ncc(CC)c2)NC(=O)N(CCC(C)C)C2=C1C(=O)NC(C)C2 21215,C(=O)(CCc1ncc[nH]1)NCCN(C(CNC(=O)NC)=O)C1CC1 21216,C1(C(=O)NCCCN(C(=O)CC2CCCCC2)CC)CCCN(C(C)=O)C1 21217,C1(NC(C(CO)NC(c2c(C)nc(C)o2)=O)=O)CC2(CCCC2)C1.CC1=CCSC1 21218,C1(CN(C(=O)Cn2ncccc2=O)C)CCCCN1C(=O)Cc1cncs1 21219,c1(C(=O)NCCCCN(C(=O)C(c2ccccc2)O)C)cc(C(N)=O)oc1C 21220,N1(Cc2occc2C(N2C(C(C)C)CN(C(C)C)CC2)=O)CCc2nc[nH]c2C1 21221,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21222,N1(C(CCCOCCC)=O)CCN(C(C2CC3COCC3C2)=O)CC1C1CCC1 21223,CCC(CCC(=O)N1CCCCC(C(N)=O)C1)SC.c12cn(C)nc1NC2=O 21224,C1(NC(C(CC(C)C)(C)O)=O)CCC2CN(C(=O)CCC(C)(C)F)CCC2C1 21225,n1(CC)nnnc1C(C1CCC1C1CC1)NC(C12CC(CO1)C2)C.CCO 21226,CC(C)(C)C(C#N)C(=O)NC1CCC(CNC(C2(C)CC3(CC3)C2)=O)C1 21227,c1(CC(=O)N(C)CCNC(C2CC(CF)C2)=O)cnn(C(C)(C)C)c1 21228,N1(C(C2N(C(C)C)CCC2)=O)CCC2CN(C(C3NC(=O)OC3C)=O)CC12 21229,CCC(C)(C)CC(=O)NC1CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 21230,N1(C(CCc2cc(C)no2)=O)CC(N(C(=O)COC(F)F)C)C(O)C1 21231,C1(F)(CNC(c2cc(CN)[nH]n2)=O)CCN(C(=O)CC2C=CCC2)C1 21232,Cn1nc(C(F)F)cc1NC(C1(C(C)(F)F)CC1)=O 21233,c1(OC)cccc(F)c1C1CCN(Cc2ccnc(Cl)n2)C1 21234,CC(C)CCCCC(CO)NC(=O)N(CCN1CCCCS1(=O)=O)C(C)C 21235,Cc1cc(C(C)NC(=O)N(C2CC=CCC2)CCO)no1 21236,CN1CCN(C)C(C(N2CCOCC2C(=O)NC2CCCC2O)=O)C1 21237,n12cc(nn1)C1(CC1)OCC(=O)NCC1CC1C2.CC(C)(C)C(=O)NC1CCC1 21238,C=C=CC(C)C(=O)N1CC2C(C(C(=O)NCc3cccc(Cl)c3)(C)OC)C2C1 21239,Cc1csc2c(CC(N3CC(NC(=O)C(F)=CCCF)C(O)C3)=O)cccc12 21240,N1(C(CCC(CC)C)=O)CC2(CCC(NC(=O)C(O)CSC)CC2)C1 21241,C12(CCNC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1cncn(C)c1=O)=O)C2 21242,C(=O)(NNc1ccc(C(=O)N(C)C)cn1)c1c(CC(C)(C)C)[nH]cc1 21243,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCc2ncccc2F)cn1 21244,CCC(C)(C)C(O)C(=O)N1CCCC(N(CCF)C(c2ccc(F)c(F)c2N)=O)C1 21245,c1(CC(=O)NC2(C)CC(NC(c3cccc(N)c3)=O)C2)ccc(S(=O)C2CC2)cc1 21246,Cc1ccc(C)c(C(N2CCCCC2CNc2ccc(F)cc2)=O)c1 21247,C1(OC)CCN(C(=O)CC2CC(C)N(C(=O)COc3ccccc3Cl)C2)CC1 21248,c1(CCC)cc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)ccn1 21249,C1(C(N(C)CC2(F)CCOC2)=O)CCN(C(c2c[nH]nc2C(F)F)=O)CC1 21250,c1(NC(=O)N(CCOC)CC2CCCC2)cc2c(cc1Cl)COC2 21251,C1(NC(c2cnc(C)[nH]2)=O)CCCN(C(=O)C=Cc2cncc(C(F)(F)F)c2)C1C 21252,CN1CCCC(NC(N2CCN(CCN(C)C)CC2)=O)C1 21253,c1(C(N(CC(C)N(C(c2nc(COC)sc2)=O)C)C)=O)ccn2ccnc2n1 21254,C1(C(=O)NCCCN(CCCNC(C2(CC)CCCO2)=O)C)CCCN1N=O 21255,C1(NC(c2ccc(OC)nc2)=O)C2CCN(C(=O)CCn3cnnn3)C2C1(C)C 21256,c1(C(=O)NC2(CN(C(Cc3c(OC)nccc3)=O)C)CC2)ccc(F)cc1C#N 21257,C(CCC(C)(C)C(=O)NC(c1nccn1C)C)NC(C(CCCC)O)=O 21258,C1(C(=O)NCCOCCN(C)C(C2SCCS2)=O)CCC1C(F)(F)F 21259,c1(C(=O)NCC2(c3ccc(Br)cc3)CCCC2)ccc(Cl)c(Br)c1Cl 21260,N1(C(COCC=C)=O)C2CCC1CN(C(=O)C(C)SCc1ccccn1)C2 21261,C1(C(=O)NC(C)CN2CCN(C(C3CC4(CSC4)C3)=O)CC2)CCC(=O)C(C)C1 21262,N#CC1CCN(C(C2(NC(C3CCOC3)=O)CC2)=O)C1 21263,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21264,CC1CC(NC(=O)Cc2ccon2)CN1C(=O)CCc1nc[nH]n1 21265,O(N1C(=O)c2ccccc2C1=O)CC(N1CCC(F)(NC(=O)COCCF)C1)=O 21266,c1(CC)nc(CC(=O)N(C)CCN(C)C(C2CC2(C)C)=O)cs1 21267,N1(C(C2N(N=O)CCCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21268,N1(C(CCCC(C)C)=O)CCC(C(=O)N(CCCF)CCO)=C(F)C1 21269,c1(OC)cc(C(=O)NC2CN(C(C3CC3C(F)(F)F)=O)CC2F)nn1C 21270,C1(NC(C(C=CC)O)=O)CC2(C1)CC(NC(C1CCC(C(C)(C)O)CC1)=O)C2 21271,C1(NC(Cc2cccc(OC)c2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 21272,N1(C(C(=O)NCCCOCC2CC2)CC2CCCCO2)CCCC(F)CC1 21273,C(=O)(C(C)(F)C(C)(C)F)NC(CNc1c(F)ccc(C(C)=O)c1)C 21274,CC1=CC(NC(=O)CCC2CC(NC(=O)CCc3cncs3)C2)CCC1 21275,N1(C(c2ccc(NC)cc2)=O)CCOCC(C(=O)NCC2CCC(=O)O2)C1 21276,C1(C(=O)N)CCCN(C(c2nc(=N)cc[nH]2)=O)C1.C1(C(N(C)C)=O)(C(N)=O)CC1 21277,CC(CCNC(=O)CCC1CCCCN1C(=O)C=CCC1CCCC1)CCCO 21278,c1(C(N(CC(CNC(C(CC=C)CC=C)=O)C)C)=O)cccc2oc(O)nc12 21279,c1(OCC)cc(OCCCOC)cc(NC(=O)C(N2CCCS2(=O)=O)C)c1 21280,C(C(CO)C(C)(C)C)NC(C(C1CCCC1)NC(c1nn(C)c(CO)c1)=O)=O 21281,c1(N(C)CC2CC(=C)C2)ccc(S(=O)(=O)NCC2(SC)CCC2)cc1Cl 21282,c1(CNC(c2ccccc2F)(c2n(CC(=C)C)nnn2)C)noc2c1CCC2 21283,N1(C(C(CC=C)(C)C)=O)CC(NC(C2(CF)CCC2)=O)CC(C)(C)C1 21284,c1(C(=O)NCCCNC(C(C(CC)(C)C)OC)=O)c(C)cnc2ccccc12 21285,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(N(C)C)c2C1.N12CCCC1CC2=O 21286,C(=O)(CCCC(=O)NOC(C)C)NCC(C)N(C(CC=CCC)=O)C 21287,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21288,c1(C(=O)NC2CN(C(CSc3nc(C)[nH]n3)=O)CC2C)cc([N+](=O)[O-])cnc1O 21289,N1(C(C(C)(F)c2ccccc2)=O)CCC2C(O)CC2C1 21290,N1(C(CSCC(=O)N(C)C)=O)CCCC2CN(C(=O)C(F)=C3CCC3)CCCC12 21291,C(C(F)(C(=O)N1CCCCC1C(C)C)C(C)C)NC(Cn1ccc(C)n1)=O 21292,N1(CC(=O)N(C(C(=O)NCCC(C)CO)(C)C2CC2)C)CCCCC1C 21293,N1(C(C(CNC(C)=O)(C)C)=O)CC2(CCCCN2C(=O)CN2CCC(=O)NC2=O)C1 21294,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCN(C)C 21295,C1(NC(Cc2cnc(C)s2)=O)CN(C(C2CC3CCC2O3)=O)CC1C 21296,C1(C(N(C(C)C)CCN(C)C(C23CC=CC(C2)OC3)=O)=O)CN2CCN1C(C)C2 21297,N1(C(c2ccn(CCN(C)C)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1 21298,c1(CCC2CCS(=O)(=O)C2)nc(N2CCN(N3CC4CC4C3)CC2)nc2cc[nH]c12 21299,C=CCC(CNC(=O)CC(C)(C)CC)C(=O)N1CC(=O)NC(C)C1 21300,c1(C(N(CCCCNC(=O)CC(C)C2CC2)C)=O)nccc2cccnc12 21301,C1(NC(C2(CC)CC2)=O)CN(C(=O)COc2ncccc2O)CC2(CC2)C1 21302,C1(NC(COCC(C)(C)C)=O)CN(C(=O)Cc2cnco2)CC2CC12 21303,O1NC(=O)C(CC#CC)NC(=O)C1.C=C1CC(NC(C)=O)C1 21304,c1(C(N(CCCC)C(c2cccc(N)c2C)=O)=O)cccc2[nH]cc(Cl)c12.C 21305,c1(C(=O)NC2CCC(C)N(C(c3nc(Cl)ccc3N)=O)C2)c(F)cc(O)cc1F 21306,c1(CC)noc(CCC(=O)NCC(CO)NC(=O)C(F)(F)c2nccs2)n1 21307,c1(CN2C3CN(C(C(C)NC(CC)=O)=O)C(C3)C2)cnc2cc[nH]c2c1 21308,N1(C(CCN(C(CCC=C(C)C)=O)C2CC2)=O)CCN(C)C(=O)C1 21309,c1(C(=O)NC2CCN(C(C3C(c4n(C)ncc4)C3)=O)C2)cc2ncccc2o1 21310,C(=O)(C(CC(C)C)N(C(=O)CN)C)NC.C1(NC(=O)O)CCN(c2ccccc2)C1 21311,c1(C(N(C(C)CCNC(c2cn(C3CCC3)nn2)=O)C)=O)cccc(=O)n1C 21312,c1(CC(=O)NC(CCNC(Cc2c(F)ccc(C)c2)=O)C)ccn2cncc2c1 21313,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21314,C1(CNC(CN(CCC)C)=O)CC(NC(=O)C=CC(=O)NC)C(O)C1 21315,c1(OCCC)cccc(C(=O)C(=O)NCCC2(C(=O)OCC3CC3)CCC2)c1 21316,C1(CSCC(=O)NC(C)CCC)CCCCO1.c12cc(ns1)NC2=O 21317,C(=O)(C1=CCCCC1)NCC1C(C)CCN1C(=O)CCc1cnc(O)[nH]1 21318,C(C)(C)(CCC(=O)N1CCC(c2cn(CC(O)COC)nn2)C12CC2)OC 21319,C1(C(=O)NC2C(NC(=O)CCF)C2)COc2ccccc2C1 21320,C1(O)(C(C)NC(c2csnc2Cl)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 21321,N=c1cc(C(N2CCCC2C2NC(=O)NC2=O)=O)c(Br)c[nH]1 21322,C1(C)(CNC(C(CC)(C)F)=O)CN(C(C23CCCC2CCC3)=O)CC1C 21323,c1(C(N2C3CN(C(C4CCC(OC)CC4)=O)C(C3)C2)=O)cccc2[nH]nc(O)c12 21324,N(C1CCCc2sc(Cl)cc21)C(N(CC)Cc1cncn1C)=O 21325,c1(C(N2CCC(CN=c3[nH]cncc3Cl)C2)=O)cccc2c(I)n[nH]c12 21326,C1(NC(CCc2c(C)ncs2)=O)CN(C(c2ncc(F)cc2F)=O)CCC1C 21327,c1(C(=O)NCC2CCN(C(C(C(C)C)N(C)C)=O)C2)cccc2nc(O)oc12 21328,C1(CN(c2cc(C(F)(F)F)c[nH]2)C(C=CCC)=O)CCCN1C(c1ccco1)=O 21329,C1(C(N(C)CC2CN(C(C3CN(C(C)=O)C3)=O)C2)=O)CC(C)(C)O1 21330,C(CC(F)(F)C(=O)O)NC(C1C(SC(C)C)NCC1)=O 21331,C1(NC(CC2OCC(C)(C)C2)=O)CC2CC1CC2C(=O)NCC1(c2ccon2)CC1 21332,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21333,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CC 21334,Cc1cc(Cl)ccc1OCCCNC12CC(C)(C1)OC2C 21335,N1(C(C2(C(C)C)CCC2)=O)CC(C(N)=O)(CNC(=O)Cc2cn[nH]c2)C1 21336,c1(CC(=O)NCCN(C(C)C)C(=O)Nc2nccs2)n[nH]c2ccccc12 21337,c1(OC)cccc(S(=O)(=O)NNS(=O)(=O)CC2(C(F)(F)F)CCC2)c1Cl 21338,C1(C(=O)NC2(C)CNC(=O)C2)CCC2(CCN(C(=O)C(=O)C3CCCC3)CC2)O1 21339,N1(C(COCCC(C)C)=O)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2CC1 21340,c1(C(=O)NC2C(CNC(C3CCC(C#N)CC3)=O)COC2)ccnc2[nH]nnc12 21341,CC1(C)NC(=O)CC1C(=O)NC12CC(C1)N(C(=O)Cn1cc(C3CC3)nn1)C2 21342,c1(OC)ccc2c(c1)OCC(C=CC=Cc1ccc(Cl)cc1N)=C2 21343,C12(C(N(C(C)CNC(c3ccc(O)c(Br)c3)=O)C)=O)C3C4C1C1C2C3C41C 21344,C1(C(=O)NCC(CC(=O)NC)C)CCN(C(c2occc2C)=O)CCO1 21345,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21346,C1(CC#C)(C(=O)NCC(C)(C)NC(c2csc(C(F)(F)F)c2)=O)CCCO1 21347,N1(c2snc(CCC)n2)CCC2(CCCCC2NC(=O)Cc2nnc(C)s2)C1 21348,CCC1=C(C(=O)N2CCC(C(C)NC(c3cc(C)ccc3C)=O)C2)CCCO1 21349,C=CCC(CC)C(=O)N(CC(C)(C)CNC(=O)C(c1cncn1C)O)C 21350,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CCC2)=O)C)ccc(F)c(Cl)c1F 21351,N1(C(CN(C(C2(C)CC(=C)C2)=O)C)=O)CC(C)C(C)C1C 21352,C(C(C)(C)CCNC(=O)C(C1CCCCC1)C)NC(C1C(C(=O)OC)COC1)=O 21353,c1(N(C(C(C)C(F)F)C(=O)Nc2ccccc2)C)cnn2ccccc12 21354,N1(CCCCN(C(c2cc(-c3ccccc3)sn2)=O)CC)CCN(C2CC2)CC1 21355,Brc1c[nH]c2ncc(CNc3cc(-c4nnnn4C4CC4)c4c(c3)CCC4)cc12 21356,C(C(COC)CC(=O)NCCCn1cc(CCS(C)(=O)=O)nn1)OC 21357,C1(NC(C2CC(C)(C)OC2)=O)CCN(c2ccc(C#N)nn2)CC1O 21358,C1(C(=O)NC2CC(C(=O)NCCSCC=C)C2(C)C)CC(=O)CC(=O)N1 21359,C1(NC(C(c2cccc([N+](=O)[O-])c2)C)=O)C2CCC1CN(C(=O)C1CC1)C2 21360,O=C(C1=COCCO1)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 21361,Cn1ncc(Cl)c1C(N1CCCC(NC(C23CC(C4CC4)(CO2)C3)=O)C1)=O 21362,C(=O)(C1CCCc2nn[nH]c21)N1CCCC(C2C(OCC)CCCO2)C1.C1CN1 21363,C1(C(N2CCC(N(C(c3ccc(C4CC4)o3)=O)CC)C2)=O)C(Cl)(Cl)C12CC2 21364,C1(C2CC2)(NC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN(C)C(C)=O)C1 21365,N1(C(C2CCN(C(C3C(OC)C3)=O)C2)=O)CCC(C2CCC2)C1 21366,c1(C(C)C)cc(NC2CN(C(=O)CCc3cncs3)CC2(C)C)nc(C(C)C)n1 21367,Cc1cccc2c1CCCN2C(=O)NCC1COC(C)(C)OC1 21368,c1(CC(N(C(CC)C)CC(=O)NCC(O)CF)C)ccc(C)nc1 21369,c1(C(N(C(C2CCCO2)=O)Cc2nc(C)oc2)C)ccc(-c2ccccc2)cc1 21370,C1(C(N2CCCC2(CCNC(c2nc(OCC)oc2)=O)CC)=O)CC2CCC1CC2 21371,c1(C(N2CCC(NC(C(S(C)(=O)=O)C3CC3)=O)C(F)C2)=O)c[nH]c2cccnc12 21372,N1(C(CC(=O)N(C)C)=O)CCCC2C(NC(c3[nH]nnc3C3CC3)=O)C(C)(C)C12 21373,N#Cc1ccc2c(c1)C(=CC(N1CCC(O)C(CO)C1C(=O)O)=O)C2 21374,C=CCC(O)(CN(CCSC)CC=Cc1c(CCCC)coc1C)CC=C 21375,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC=C)C1 21376,C(=O)(CCC(=O)C1CC1)N(CCC(C)NC(=O)CCN1CCC1)C 21377,C1(OCC#C)CCN(C(=O)C(CSC)NC(C23CC(OC)C2C3)=O)CC1 21378,N1(C(CCNC(C2(C)C(C)C2)=O)=O)CC=CC(NC(c2c[nH]ccc2=O)=O)C1 21379,CC(C)C(CNC(C1CCC2(CCC2)O1)=O)C(=O)NCc1cccc(Cl)c1 21380,C1(O)(CNC(CC(CNC(C=C=C(C)C)=O)OC)=O)CC2C=CC1C2 21381,c1(-c2nnc(C(C3CCN(Cc4ccc(I)cc4)CC3)C)o2)ccccc1F 21382,C1(C)(CC)CN(C(=O)C(C)(C)CNC(C2CC2(C)C)=O)CCO1 21383,N1(C(CC2(OC)CN(C(=O)C(O)C3CCCC3)C2)=O)CCCCCCC1C 21384,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnc(C)nc1CC)=O 21385,c1(SCC2CC(NC(C(=O)NCC(=O)NC3CC3)=O)C2)ccccc1F 21386,CCCCCCC(C)C(=O)N1CC(CN(CCC)CCO)C(C(=O)NC)C1 21387,c1(C(=O)NC(C)CCN(C(=O)C=CSc2ccccc2)C)ncc[nH]c1=O 21388,c1(-c2c(C(N(CC(C)N(C(CC=C=C)=O)C)C)=O)scc2)cccc(OC)c1 21389,C1(CNC(CC(CC)OC)=O)CN(C(=O)CCc2nc(C)no2)CCC1(F)F 21390,N1(C(c2ccc(CN(CC)CC)o2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 21391,c1(OC)c(C(N2CCOCC2)=O)cc(Cl)cc1Br.C1C(=O)O1 21392,c1(C(N2CCC3CCC(NC(=O)C(F)F)C2C3)=O)cc2c(c([N+](=O)[O-])c1)OCO2 21393,n1(CC)nc(C)cc1C(=O)NC1(C(=O)NC2CC(OCC)C2)CCC1 21394,N1(CC)CC(NCc2cnc(Cl)c(F)c2)CC(C)C1 21395,N#Cc1ccnc(N2CCCC(CNC(c3scnc3C(F)(F)F)=O)C2)n1 21396,C1(C(=O)NCCC2CCC(C)CC2)CN(C(C2CC(C)(O)C2)=O)CCN1C 21397,C=CCC(C)(C)CC(=O)NC1CC1NC(=O)C(c1ccc(OCC)cc1)C1CC1 21398,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21399,C1(C2CCN(C(=O)CCCCC(F)F)C2)(NC(C2C(CC)CCO2)=O)CC1 21400,N1(C(C2C(SC)CCC2)=O)CCC2(CC1)CCN(C(=O)CNC(N1CCCC1)=O)C2 21401,c1(CC(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)CO)C)ccccc1F 21402,c1(C(=O)NC2C(C)N(C(c3cc(Cl)c[nH]3)=O)CCC2)cnc2nccn2c1 21403,CC1C(C)N(C(=O)C2=CCCO2)CCN1C(=O)CCc1ccncc1Br 21404,c1(-c2c(C)oc(CNC(=O)NCCC3CC3C)c2)cccc([N+](=O)[O-])c1 21405,CC(C)C(C(=O)NC(C)Cn1cc(-c2cccc(C(F)(F)F)c2)nn1)C(C)C 21406,S(=O)(=O)(c1ccc(Cl)nc1C)NC1(C#N)CCN(C(c2c(OC)ccs2)=O)C1 21407,N1(C(COC2CN(C(c3snc(C)c3N)=O)C2)=O)CC2CC(C)(C)C2C1 21408,C(C(CC(C)C)C(=O)NCCc1c(C)noc1C)OC(C(=O)NCC)OCC 21409,c1(OC)ccc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)c(C)c1 21410,CC1(C)COCCC1C(=O)OC.C12CCC(C1)N(C[N+](=O)[O-])C(CC1CC1)C(=O)N2 21411,c1(CCC)ccc(F)c(-c2ccc(C(=O)NC(C)(C)C3CC3)c(OC)n2)c1 21412,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(C2CCO2)=O)C1 21413,c1(C(N(C)CC2COCCN2C(c2cn[nH]c2)=O)=O)noc2c1CCCCC2 21414,C1(C=O)C2CC3C(C2=O)C13.c1(CN2ONC(=O)C2)cccnc1OC.CC 21415,Cc1scnc1C(=O)NCC(C)CN(C(=O)CNC(C1CCC1)=O)C 21416,C=C(Br)CC(=O)NC(C1CCN(C(C2CCCC2C(C)C)=O)C1)(C)C 21417,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N2C(=O)COc1cccnc1 21418,OC1(CNC(c2ccc(-c3nnco3)nc2)=O)CC(O)C12CCC2 21419,Cc1cc(C(=O)NC2(CN(C(=O)CC3CCOC3=O)C)CC2)c2ccccc2n1 21420,CCC(CC(=O)NC1C(NC(=O)CCCOCCOC)CC1O)C(C)C 21421,CC1=CC(NC(=O)COC2CN(C(=O)CC3(C)CCOCC3)C2)CCC1 21422,CN1CCN(C(=O)CC2COCCN2C(=O)C=Cc2cccnc2)CC1=O 21423,c1(C(=O)NCC2C(NC(c3ncc(C)cc3F)=O)C2)cn2c(n1)CCCC2C 21424,N1(Cc2ccc(OC)c(OCc3ccc(F)cc3)c2)CCn2ncc(Cl)c2C1 21425,C(CCC(=O)NC(c1ccccc1)CNC(=O)Cc1ncccn1)=CC(C)C 21426,Cc1[nH]c(C)c(C(N2CCC(CC(N3CCC(CO)(CO)C3)=O)C2)=O)c1C 21427,CN1CCc2ccc(OCC(=O)Oc3ccc(-c4nncn4C)cc3)cc21 21428,C1(NC(C(C)=C)=O)CCOCC1NC(=O)CCC(=O)N1CCCCC1C.N(C)C 21429,CC1(C(=O)NC2CC(CNC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21430,CC1CN(C(C2(CCNC(=O)Cc3ccccc3O)CC2)=O)CC(C)(C)O1 21431,c1(OC)nn(C)cc1C(N1CCC(C(=O)Nc2cc(SC)ncn2)CC1)=O 21432,C(CCC(CO)NC(=O)CC1CC(O)C1(C)C)NC(C1(C(=O)NC)CCC1)=O 21433,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21434,C(=O)(C1=CCCSC1)NC1(C)CN(C(C2CCN(C3CC3)CC2)=O)C1 21435,C1(C(N(C2(C)CCCC2)C)=O)COCC1NC(c1cnn(C2CC2)c1)=O 21436,c1(SCC(=O)NCC(CC)NC(c2cn(-c3ccn(C)n3)cn2)=O)nnnn1C 21437,Nc1cc(C(N2CC=C(CNC(=O)COC3CCCCC3)CC2)=O)cc(F)c1 21438,CC(C(=O)NCCNC(c1ccns1)=O)C(F)F 21439,c1(-c2ccc(C(=O)NC(CNC(C=CCCC)=O)C(C)C)[nH]2)ccc(Cl)cc1 21440,N1(Cc2ccc(COC)s2)CCOCC(C(=O)OC)C1 21441,N1(C(c2cccc(CC)n2)=O)CCCC(C)(CNC(=O)CC2CC=CCC2)C1 21442,c1(C(N2CCC(NC(CCS(C)=O)=O)(CO)CC2)=O)ccc2c(c1)CC(=O)N2 21443,C1(CC)CCC(NC(=O)CC2(CCNC(C34CCCC3C4)=O)CC2)C1 21444,CCC1=C(C(=O)NC2CCC(NC(c3cc(OCC)ccn3)=O)C2)CCCO1 21445,C(CNC(=O)C(F)C1CC(NC(C2CC=CC2)=O)C1)(C(F)(F)F)OC 21446,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CC(O)C3)C1)=O 21447,C1(C(C)NC(c2cocn2)=O)CCN(C(=O)Cc2cn(C3CCOCC3)nn2)C1 21448,C(C(CC(F)(F)F)NC(C1(C)CC1(Cl)Cl)=O)NC(c1c(CC)oc(C)c1)=O 21449,CN1CC(C)(C(N2CCC3C(NC(C4CC(C)(C)CCO4)=O)C23)=O)CC1=O 21450,Cn1ncc2cc(C(N3CC(NC(=O)CC4CCCOC4)C(F)C3)=O)cnc12 21451,N1(C(c2cnc(C)o2)=O)CCC2CCCC12C(=O)N(C1CCCC(C)(C)C1)C 21452,C1(NC(CCCC(=O)N(CC)CC)=O)CCN(C(C2CC2C)=O)CCC1(F)F 21453,N12CCOC3(CCN(CC3)c3ncc(cn3)C1=O)C2.CCCC(CCO)OC 21454,c1(C(=O)NC(CNC(c2cc(C)no2)=O)C)ccn2ncc(Br)c2c1 21455,c1(C(=O)NCC23C(CN(C(CC)=O)C2)C3)ccc(S(=O)(=O)CC)cc1 21456,C(CCC)(C(=O)N(C(CC)CC(=O)NCc1ncc(CC)[nH]1)C)=CCC 21457,N1(C(c2cc(C)sc2)=O)CCC(C2CCCN2C(=O)C=CCO)CC1 21458,N1(C(C(c2nc(C)sc2)=O)=O)CC2CCC2(CC(=O)NCc2cc(C)nn2C)C1 21459,c1(C(=O)Nc2cccnc2N2CCCC2C(=O)O)ccc2c(c1)S(=O)(=O)CCC2 21460,c1(CCC(C)NC(C2CCN(c3nnn(C)n3)CC2F)=O)cccc2cccn12 21461,c1(N2C(CNC(c3c(C)ncnc3)=O)CC(C)(C)C2)nc2ccc(F)cc2s1 21462,c1(-c2nc(CCOC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21463,C1(C(N(CC(CC)NC(c2cc(O)ncc2F)=O)CC)=O)C2C3CCC(C3)C12 21464,C1(C)(C(N2CC(CNC(C3(CC#C)CCC3)=O)(OCC)C2)=O)CCCOC1 21465,N1(C(CS(N)(=O)=O)=O)CCC2(CCC(CNC(C3(F)CCOCC3)=O)OC2)CC1 21466,O=C(CC1CCOc2ccccc21)NC1C=CCN(C(c2c[nH]nc2F)=O)C1 21467,c1(COC)ccc(CNC2CN(C)CC2C(=O)O)cc1Cl 21468,N1(C(c2ccc(SC)o2)=O)CCCCC(CNC(=O)CC2COCCN2C)C1 21469,c1(CC(=O)NCC(C)(C)NC(c2nonc2N)=O)csc2nc(C3CC3)cn12 21470,c1(C(C)C)c[nH]nc1C(=O)NCCN(C(=O)CCc1cccnc1)C 21471,C1(C(N2CC3C(CNC(c4c(C)scn4)=O)C3C2)=O)CNC(=O)CC12CCC2 21472,C1(C)(C(=O)NC2CC(CCNC(C(C)OCCOC)=O)C2)CNC(=O)C1 21473,N(C1CCc2cc(Cl)ccc21)S(c1ccc(OCC)c(CC)c1)(=O)=O 21474,N1(C(CC(CC)C)=O)CCC2(CC2)CC1C(=O)NC(C)COC 21475,CC(C)CCNC(=O)CC1(NCC(=O)N(CCO)CC2CC2)CC1 21476,c1(C(=O)NCc2ccc(Cn3ccnc3)o2)ncccc1Cn1ccnn1 21477,c1(OC)cc(Cl)c(CN2CCC2(C)C(=O)Nc2ncc(C#N)cc2F)cc1Cl 21478,C1(C)(C(=O)NCCN(C)C(N2CC(C(N)=O)C2)=O)CCC(=O)N(C)C1 21479,C1(NC(c2scc(COC)c2)=O)(CO)CCN(C(c2cc(CO)c(C)o2)=O)CC1 21480,NCCCCN=c1[nH]ccc(=NCC(=O)NC(c2ccc(F)cc2)C)[nH]1 21481,c1(C(=O)NCC(C2CCCOC2)OCC)cnc2ccccn12 21482,C1(NC(CCC(=O)NCC)=O)CN(C(C2CCCOCC2)=O)CC12CCC2 21483,C1(N2CCCC2)CCCC1S(=O)(=O)N1CCCC(O)(N(C(C)(C)C)C)C1 21484,c1(NC(N2CCCC2c2cnco2)=O)cc(CCO)on1.C12CCN(C1)C2 21485,C(CN=S(C)(C)=O)NC1(c2n(CCC3(C)CC3)nnn2)CS(=O)(=O)C1 21486,n1(-c2ccn(CC)n2)nc(CC(C)(C)C)nc1-c1ccnn1C1CCCC1 21487,C(c1ccccc1F)=CC(N1CCN(C2CN(C(C(C)NC(N)=O)=O)C2)CC1)=O 21488,c1(CC(=O)NCC(CCOC)NC(C2CCC(COC)CC2)=O)sc(C)nc1C 21489,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21490,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21491,N1(C(CN(CC)CC)=O)CCOC(c2cn(CC3CCOC3)nn2)C1 21492,c1(COC(CC2CCCC(=O)N2)=O)cc(F)cc(F)c1 21493,N1(C(c2c(Cl)n[nH]c2C)CC)CCC(n2cc(C3CCCC3CO)nn2)CC1 21494,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CCN(C)C2)ccc2n[nH]c(C)c2c1Cl 21495,C(=O)(CC(C)CC(=O)NC(C(=O)N(C)Cc1cc(C)no1)C(C)C)OC 21496,C1(CC(N2CC(O)(CC(N3CCCCC3)=O)C2)=O)C=CCCC1 21497,CC1=NOC(CC(=O)NCc2ccsc2C(=O)N(CC(C)C)CCN(C)C)C1 21498,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21499,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21500,N1(C(c2n(C(C)C)nnc2)=O)CCC(O)(CN(C(=O)CCc2ncco2)C)C1 21501,O=C(C1CCCc2scnc21)NCCCCCNC(c1ccc2nonc2c1)=O 21502,CC1CCN(C(C2C(C(=O)O)C2C)=O)CCN1C(=O)CSc1ccccc1Cl 21503,C(=O)(C(F)(F)CCC(=O)NCCCN1CCS(=O)(=O)C(C)(C)C1)OC 21504,C1(C(=O)NC2(CC)CN(C(=O)Cc3csc(Br)n3)C2)CC=C(C)CC1 21505,C(=O)(C1=CCCC1P(C)(C)=O)OCC.CCCCC(C(=O)O)OC(C)=O 21506,c12ccc(Br)cc1CO2.CC(C)C(=O)C(=O)NC1CC(=O)N(Cc2ccccc2)C1 21507,CC1C2CC(C2NC(=O)CNC(c2ccccc2F)=O)N1C(C1CC12CCC2)=O 21508,C(=O)(CS(=O)(=O)CC(F)(F)F)N(CC(C)O)CCNC(c1c(OC)nn(C)c1)=O 21509,Nc1cnc(Br)c(C(N2CCC(NC(=O)CCN3CCCC3)C2)=O)c1 21510,c1(CNC(C2(C)CCS(=O)(=O)C2)=O)nc(CNC(=O)C2=COCCC2)cc(O)n1 21511,C1(CNC(C2(CC#C)CCOC2)=O)CN(C(C2COCOC2)=O)CC12CCC2 21512,N(C1c2ccccc2OCC1C)C(c1ncnc2cccc(Br)c12)C 21513,C(=O)(C(C)(CO)NC(C)=O)NCC1(COC)CN(C(=O)CCC2CCC(C)O2)C1 21514,C12(C)C=C(C(=O)NC3CC4(C3)CN(C4)C1=O)C2.c12nn(C)cc1C(=O)O2.CC.OC 21515,CCC(C)(COC)NC(c1cn(CCNC(=O)C(C)Cn2ccnc2)nn1)=O 21516,CC1CC(C(=O)N(C2CCCN(C(=O)CCNS(=O)(=O)C(F)F)C2)C)CCS1 21517,N1(CCOC)CCCC(OC2(c3n(C(CC)C)nnn3)CC(C)(C)C2)C1C(F)(F)F 21518,C1(C(=O)NC(C(C)C)c2nc[nH]n2)CC(=O)CN1C(C1CC1C(F)F)=O 21519,C1(NC(C(CCSC)OC)=O)CCC2CN(C(=O)C(C)N(C)C)CC12 21520,c12cccc(c1)C(C)O2.C(=O)(CP(C)(C)=O)NC(CNC(c1cc(C)oc1)=O)C 21521,N1(S(=O)(=O)Cc2nnc(Cn3cc(Br)cn3)o2)CCCC(CN=[N+]=[N-])C1 21522,c1(C(N2C(C)CC(CNC(C3(F)CCCC3)=O)C2)=O)cc(Cl)ccc1OC(F)F 21523,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21524,Cc1nn(C2CC2)cc1C(=O)NC(CO)CCCNC(C1CC1F)=O 21525,O=C1CCCC(n2cc(CNC(=O)C(c3ccc(Cl)cc3)O)nn2)O1 21526,Cc1cc(C(C)C)nc(N2CCCOC(CNC(=O)CC(O)CN(C)C)C2)n1 21527,CC1(C)CC(C(=O)NC2CCCCC2CNC(C2CCCN2C2CC2)=O)=NO1 21528,N1(C(C(c2cnn(C)c2)NC(C=CCC)=O)=O)CCC(C)(O)C(O)C1 21529,c1(N(CCCCC)C(=O)C(O)C2CN(C(=O)C(CC)C(C)C)C2)cnn2cccnc12 21530,C1(CNC(C=C(C)c2cccs2)=O)CCC2CN(C(c3cnc(C)s3)=O)CC12 21531,N#CC12CC(C(=O)NC3CC(NC(=O)CC4CCCCO4)C3)(C1)C2 21532,c1(N)cc(S(=O)(=O)N2CCCC(CCNC(C)CCCCO)C2)ccc1C#N 21533,Cc1ncc([N+](=O)[O-])cc1-c1cn(C2CCC(C(C(C)CC3CC3)=O)C2)nn1 21534,N1(C(COCC(C)C)=O)CCSCC1C(=O)NC(C)CC1CCCC1 21535,C1(C)(C(=O)NCC(CO)N(C(=O)Cc2ccsc2C)C(C)(C)C)CC(C(=O)OC)C1 21536,N1(C(Cc2n(CC)ccc2)=O)CCC(NC(=O)C(C)C2CCCC2)C1C(C)(C)C 21537,n1(CC)nc(C(=O)NCC2CCC(NC(c3nccnc3CC)=O)C2)ccc1=O 21538,C=CCC(CNC(C1CC2(C1)CC(O)C2)=O)C(=O)NC(CO)C(=O)OCC 21539,C1(C(=O)NC2CC3(C(NC(c4cc(SC)oc4)=O)C3)C2)CCCC1S(C)(=O)=O 21540,C1(CCC(=O)N(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)C)CCCCN1C 21541,N1(C(C2(C)CC2)=O)CC(CNC(=O)CCCNc2ccccn2)OC2COCC12 21542,c1(C(c2n(CCCOC)nnn2)OC)cccc(Cl)c1Br.O1NC(=O)CSCC1 21543,n1(C(C)C)cnc2c(N3CCC(F)(C#N)C3)[nH]c(=NCC3(C)CC3(F)F)nc12 21544,c1(C(N2CCN(C(C(C)SCCO)=O)C(CO)C2)=O)nc(O)nc(O)c1N 21545,c1(OC)ccc(Cl)c(C(=O)NCC2CN(C(c3cnc(-c4ccoc4)s3)=O)C2)c1 21546,N1(C(n2cc(-c3cncc(Cl)c3)nn2)CCC)CCN(C)C(=O)C1(C)C 21547,C(c1ccccc1)=CCC(=O)NC(C)(C)CNC(=O)Cc1csnn1 21548,Cc1cc(CN2CCC(CCNC(=O)CCOc3ccccc3F)C2)ccc1Br 21549,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21550,N1(C(c2ccncc2)=O)CC2CCN(C(c3nc(Cl)ccc3F)=O)C2C1 21551,C1(C(=O)NC(CC)(C)CNC(=O)Cc2cn[nH]c2)CC(C)CCO1 21552,Cc1nc(Br)sc1C(=O)NC1CCCC(NC(C2(C(C)(C)O)CC2)=O)C1 21553,N1(CC)CC2(CN(C(=O)C(C)(C)C3CCCN3C(=O)C(O)C(F)(F)F)C2)C1 21554,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21555,C1(NC(C(C=C)OC)=O)CCCCC1CNC(c1conc1COCC)=O 21556,Cc1ccnc(C(=O)NC2CC2CNC(c2snc(O)c2Cl)=O)c1N 21557,C(=O)(CC1OCCc2ccsc21)N(C1CCN(C(C(C2CC2)OC)=O)CC1)C 21558,c1(C(=O)NCC2C(NC(C(COC)OC)=O)CC2)cc(=O)n(C)cc1Br 21559,CCC(C(=O)NCC1CCN(C(c2cnn(C(C)C)c2)=O)C1)C(C)(C)CC 21560,N1(C(CC(=C)I)=O)CCOCC(Cn2cc(C3(N(C)C)CCOC3)nn2)C1 21561,C(=O)(C(C)(F)C(C)(C)F)NCC1(N(c2cnc(CC)nc2)CC)CC(COC)C1 21562,C1(C(=O)NCC2CCCN(C(c3ccoc3Br)=O)CC2)Cc2n[nH]cc2C(=O)N1 21563,CCC(CNC(=O)CCS(N)(=O)=O)(CC)C(=O)NCC1CCOC(C)(C)C1 21564,Cc1ccc(C(=O)NC(C)CN(C(=O)CCC2CNC(=O)N2)C)c2c1CCC2 21565,c1(NC(C2NCCN(C(C(C)O)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 21566,c1(C(C(=O)NC(CC)C)N(C2(C(=O)OC)CCC2)C)cc(=O)n(C)c(=O)n1C 21567,CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCC2CC2)C1 21568,C=C(C)CCC(C)N(C(N1CCC(c2ncc(Br)cn2)CC1)=O)CC 21569,c1(C(=O)NC2C(C)(C)C(CNC(C34CC(C3)C4)=O)C2)ccc2c(c1)OCCO2 21570,N1(C(CCN(C(C)=O)C)=O)CC2CC(C1)CN(S(=O)(=O)c1ccc(F)cc1)C2 21571,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CC=CC1)OC 21572,c1(C(=O)OCC)c[nH]c(=NCC2(F)CCN(C(C3CC3(C)C)=O)CC2)cc1C 21573,c1(-c2nc(-c3n[nH]c4ccccc43)nn2C2CCOC2)[nH]c2ccccc2c1Cl 21574,CCC(C)C(C(=O)N1CCC(C(F)(F)F)C(NC(c2ccnn2C)=O)C1)OC 21575,Cc1ccc(C(C)NC(C2CSCCN2C(c2ccc(F)s2)=O)=O)nc1 21576,Cc1csc(=O)n1CC(=O)NCC(C1CCCC1)NC(=O)C(C)N=[N+]=[N-] 21577,C1(C2CCOCC2)(C(=O)NCC2(NC(C34CCCC3C4Br)=O)CCC2)CC1 21578,c1(C(=O)NC(CC(C)NC(C2CCC(=O)N2)=O)C)ncccc1OC(F)F 21579,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21580,C1(N(C(=O)CC2CC(C)(C)C2)CC)CCCN(C(=O)CC2CCCCCO2)C1 21581,S1(=O)(=O)c2ccc(cc2)C(=O)N2C3CN1CCC23.C(C(O)CO)NC.CN 21582,C(CCC(C)(C)C)NC(C(Cc1cn[nH]c1)NC(CN1C(C)CCC1)=O)=O 21583,C1(NC(CSCCC)=O)CCN(C(=O)Cc2ccno2)CC1C(N)=O 21584,n1(CC(C)NC(c2csc(C(N)=O)n2)=O)cc(CNC(C2CC23CC3)=O)nn1 21585,n1(CC(=O)NC2C(CNC(Cn3c(C)ccc3C)=O)CCC2)cnc2c1CCCC2 21586,N1(C(c2c(=N)cc[nH]c2)=O)CCCC(NC(c2ccsc2Br)=O)C(F)C1 21587,c1(C(=O)NC(C)(CO)CCF)csc2c1CCNC2 21588,CC(CC(F)(F)F)N=c1[nH]c(N(C)Cc2ccc(S(N)(=O)=O)s2)nc2ccsc12 21589,c1(C(=O)NCC2CC(O)CN2C(=O)Cc2ccc(Cl)nc2)cc2ncccn2n1 21590,c1(C(N2CC3(C(CNC(C(C)CO)=O)CC3)C2)=O)ccc2c(c1)CN(C)C2 21591,C=CCCCC(=O)NCC1(OC)CN(C(=O)C(C)NC(C2CCC2)=O)C1 21592,C1(NC(CC=C)=O)CCC2CN(C(C3(c4ccc(C)cc4)CC3)=O)CC2C1 21593,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21594,c1(CC)ccc(C(N2CC3C(NC(c4ccsc4SC)=O)C3C2)=O)c(C)n1 21595,N1(C(C2CCC3(CCC3)O2)=O)CCC(F)(CNC(C23CC(F)(C2)C3)=O)CC1 21596,N1(C(C2(c3cc(C)no3)CC2)=O)CC(C)C(N=c2[nH]nc(C(=O)OC(C)C)s2)C(C)C1 21597,c1(CC(CNC(=O)C(F)=CCCF)NC(c2ccsc2Br)=O)ccccc1 21598,C(=O)(CC(C(=O)OC)C(C)C)N1CC2(C1)NC(=O)CCCC(=O)NC2.CC(CCC)OC 21599,S(=O)(=O)(c1cccs1)NC(C)C(=O)NC1CC(F)(CNC(c2ccc(C)o2)=O)C1 21600,c1(C(=O)NCC2CN(C(C3C(=C)CC3)=O)CC23CCC3)nc2ccccn2c1F 21601,c1(C(=O)OC)nnc2c(CSc3cc(Br)c4c(c3)OCCO4)cccn12 21602,C1(NC(C(F)=CCC)=O)CC2CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 21603,C(=O)(CC(CC1CC1)NC(C1C2CN(C)CC12)=O)NCCC(=C)C 21604,N1(C(C(C)(Cl)Cl)=O)CCC2(CNC(=O)C(c3ccc(Cl)cc3)(F)F)CCCCC12 21605,c1(SC)nc(-c2nc(-c3ccsc3)nn2CCN2CC(C)OC(C)C2)ccc1Br 21606,C(C)(C(=O)N(C)CCN(C1CCCC1)C(=O)CN(C)C)OCC 21607,CN1CC(C)(C)CC1C(N1CC2CC(C1)C2NC(=O)C(O)Cc1cnc[nH]1)=O 21608,C1(NC(CC=CC)=O)CCN(C(=O)C(COC)N(C)C)CC1(C)C 21609,c1(CSCC(=O)NC2C(NC(C(C)C)=O)CCC2)ccc(O)cc1 21610,Cc1c(C(=O)NCC2CCCC(NC(C34CC(CO3)C4)=O)C2)cnc2ccnn12 21611,C1(C(C)NC(C2CC(=O)C2)=O)CCCN(C(=O)C(c2ccn(C)c2)C)C1 21612,N1(C(C)C)C(=O)COCC1C(=O)NCC12CNC(C(=O)O)(C1)C2 21613,N1(C(C2C(C(C)C)(CC)C2)=O)CCC(CNc2cncc(Cl)n2)C(O)C1 21614,c1(NC(C2CN(Cc3c(Br)c(OC)n(C)n3)CC(F)C2)=O)cc(I)c(F)cc1Cl 21615,CC1CC(NC(C2CC3(CSC3)C2)=O)CN(C(c2ccc(CO)c(F)c2)=O)C1 21616,CCC(CC)C(C)C(=O)NCC1(F)CC(CNC(=O)CC2=CCOCC2)C1 21617,c1(C(=O)NC2CCN(C(C3CC3C3CC3)=O)C2C)ccc(NCC(F)(F)F)cc1.CN 21618,Cc1nc(C2CCCOC2)sc1C(=O)NCC1CN(C(=O)C(=O)N(C)C)CCO1 21619,CC(C(O)C(=O)NC1CC(CCNC(=O)Cn2cnnn2)C1)c1ccccc1F 21620,CC1CC(NC(=O)C=C2CCSCC2)CCN1C(C1CC(C)(C)O1)=O 21621,Cc1cc(C)n(-c2ccc(CN(c3cccc(C(O)C(F)(F)F)n3)C)cn2)n1 21622,C1(CCOC)(NC(=O)CC2CCCC(C)C2)CCN(C(c2ncnn2C)=O)CC1 21623,C(C)(CC(C)C(F)F)(c1n(CC)nnn1)NCc1ccc(OC)cc1.C12(N)CC(F)(C1)C2 21624,N1(C(C2=CCC(NC(c3ccnc(CC)n3)=O)C2)=O)CCCC(C)(C#N)C1 21625,C(C(C)CN=C(NCC1CCN1C1CC1)NCCOc1cccc(F)c1)OC 21626,N1(C(CCN(C(=O)C(C(C)O)N(C)C)CC)=O)CCCC(C)C1CO 21627,c1(C(=O)OCC)cc2cc(NCCCC3CCCC3O)ccc2s1 21628,c1(C(=O)Nc2cccc(CC)c2)nccc2cc(-c3cccnc3C#N)ccc12 21629,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21630,N1(C(C(C=C)C)=O)CCOCC1CC(=O)N(C1CCNC1=O)C 21631,Cc1cc(N)c(C(N2CCC(O)(CCNC(C3CCCC3C)=O)CC2)=O)cc1C 21632,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2csc(COC)c2)=O)CC1 21633,CC1CN(C(c2ccc(C3CCC3)nc2)=O)CC1NC(C1(F)CCOC1)=O 21634,C=CC1(C(N2CC(N(C)C(c3cc(C)ccc3F)=O)C2)=O)CCCCC1 21635,C(C(CC(F)(F)F)NC(=O)C(F)F)NC(CC(N1C(=O)CCC1=O)C)=O 21636,c1(C(=O)NCC2C(NC(Cn3c(CCC)nnc3S)=O)C2)cc2scc(Cl)c2[nH]1 21637,c1(COCC(=O)NC(CC(C)NC(C2CCCC2)=O)C)cnc2cc[nH]c2c1 21638,S(=O)(=O)(c1cccnc1NCC1CSCCO1)N(C1C(C)CCCC1)C 21639,C=CCCCCC(=O)N(C(C)CNC(=O)C(N1C(=O)CCC1=O)CC)C.CCS 21640,C1(C)(CNC(Cc2c(C)nc[nH]2)=O)CCCC1NC(c1cnc(C(F)F)cn1)=O 21641,C=CCC(C(=O)NCC(C1CC1)NC(=O)CN1CCCC1=O)NC(C)=O 21642,c1(-n2ncc(C(N3CC(C)(NC(CCOC)=O)C3)=O)c2)ccc(F)cc1 21643,c1(SC2CC(NCC(=O)NCCc3cccc(OC)c3)C2)nc2ccccc2s1 21644,CCC(C)(C)C(=O)C(=O)NCC1(C)CCN(C(C2(C(F)F)CCC2)=O)C1 21645,Cc1ncc(N)cc1C(N1CC(CCNC(c2ccc(Cl)cn2)=O)C(C)C1)=O 21646,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCCCCNC(=O)CC1(CO)CC1 21647,CCCCC(CNC(=O)CSc1cccnc1)NC(c1nccn1CC)=O 21648,c1(CCCC(=O)OC)ccc(CO)cc1.c12cn(nn1)C1CCC1C2NCC1CC1 21649,c1(C(=O)NCCN(C2CCCCC2)C(C2CSC2)=O)cccc(-n2cccc2)n1 21650,CC(C)S(=O)(=O)CC(=O)N1CC(CNC(=O)C(C(C)(C)C)N(C)C)C2(CC2)C1 21651,c1(C(N2CCC(CCNC(C3(N=[N+]=[N-])CC3)=O)C2)=O)cc(C(F)(F)F)ccn1 21652,C(=O)(C(CN(C)C)CC)NC1(C)CN(C(C2(C(=O)OC)CC(C(F)F)C2)=O)C1 21653,N1(C(C=C(CC)CC)=O)CCN(C)CC1CC.c12nnn(C)c1C(=O)NC2 21654,c1(CC(=O)NCC(C)N(C(=O)CC2CCC3CC23)C)cnc2cccnn12 21655,CC1CC(NC(=O)C(=O)NC2CCCCC2n2cccc2)CC(C)O1 21656,C(=O)(CC(C)(C)CC(F)(F)F)NCCCNC(c1cnc(OC)nc1)=O 21657,C1(NC(CCC)=O)(CC)CCCN(C(c2cnn(-c3ccc(Cl)c(Cl)c3)c2)=O)C1 21658,N1(C(C(C)OC2CCOC2)=O)CCCC1CNC(c1ccc(F)s1)=O 21659,c1(CCC(=O)NCCCN(C(C(CCC)NC(C)=O)=O)CC)ccc(C)cc1C 21660,C1(CNC(C(C)(C)OC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21661,c1(C(N2C(C)(CNC(=O)COC3CCOC3)CCC2)=O)ccn2nccc2c1 21662,C=CCCC(CO)NC(=O)CC(CNC(c1ncccc1N)=O)OC 21663,C1(C(N(C(C)CN(C)C)C)=O)CC2(C1)CC(O)C2.C12(CCCO1)CC2 21664,c1(OC)ccc(NC(=O)CCOCC2CC2)c(Br)c1 21665,CCC(C(=O)NCCOCC(=O)NC1C2COCC12)N(C)C 21666,C1(CNC(C2C=CCCC2)=O)C2CN(C(=O)COCC(F)F)CC12 21667,C1(CNC(C2Cc3ccncc3N2)=O)CC2(CCC2)CN1C(C1(C2CC2)CC1)=O 21668,C(=O)(C#CC1CCCOC1)NC1CN(C(COCC=C)=O)CC1c1ccccc1 21669,C1(NC(c2c(CCC)occ2)=O)CC2CC1N(C(c1cc(Cl)nn1C)=O)C2 21670,C1(C(N2CC(C#C)OCC2)=O)N(C(=O)CC2(N(C)C)CC2)CCCC1(C)C 21671,C1(C(N2C(C(=O)NC)CC2C)=O)CC(=O)N(Cc2ccc(F)cc2)C1 21672,c1(C(N2CCC(CNC(C(C)OCC(C)C)=O)C2)=O)c2c(c[nH]c1=N)CCC2 21673,N1(C(c2ccn(CC)n2)=O)CC2CN(C(=O)CC(c3cccc(F)c3)C)CC2C1 21674,C(c1cc2c(cc1OC(c1cnc(S)s1)=O)CC(C)O2)=CC(=O)N(C)CC 21675,c1(C(N(CCCNC(=O)CC(C)C(F)F)CC)=O)cn2cc(C)c(C)cc2n1 21676,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21677,C1(NC(c2ccc[nH]2)=O)CC(F)CN(C(=O)CN2CCN(C3CC3)C2=O)C1 21678,C1(C(=O)NC2(CCCC(=O)NC3CC4CCC3C4)CCC2)OC2CCC1C2 21679,C12(CNC(C(C)=CC)=O)CCCC1N(C(c1cnn(C)c1-c1ccccc1)=O)CC2 21680,N1(C(C2(CCC=C)CN(C(C3CCOCC3)=O)C2)=O)CCC(F)(C#N)C1 21681,c1(C(N2CCC(CNC(C(C)C(F)F)=O)C2(C)C)=O)ccc(N=[N+]=[N-])cc1 21682,CCCCC(O)CC(=O)NC1CCC(CNC(c2ccc3c(c2)C(C)CO3)=O)C1 21683,N1(C(C(CC(C)C)=O)=O)CCC2(CCCN2C(=O)CCC(C)N(C)C)C1 21684,C1(C(N2CC(CNC(c3c(C)ncs3)=O)C2)=O)CC(=O)N(C)C1c1cccnc1 21685,C1(C(=O)NCc2c(C)cccc2)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21686,n1(CC(N2CC=CC(NC(=O)C(F)(F)CO)C2)=O)c(S)nc2ccccc2c1=O 21687,N1(C(C2(CCNC(c3c(C)snn3)=O)CCC2)=O)CCCC(C)CC1 21688,c1(C(N2CCC(c3nc(C)c(C)s3)CC2)C(=O)NCC)cn2cc(C)ccc2n1 21689,c1(C(=O)NCCCN(C(C(C2CCOCC2)OC)=O)C(C)C)cn(C)[nH]c1=N 21690,c1(OC)cc(F)c(CC2(C(=O)O)CC2)c(F)c1F.c1(S)cccc2ccncc12 21691,C1(C(=O)OC)CC2CSCC(C1)C2C(=O)Nc1cc2ccc(C)nc2[nH]1.C1CS1 21692,C(=O)(CCN=c1[nH]c(=NC(C)c2cccc(O)n2)[nH]c2c1CC(C)CC2)NC 21693,C(=O)(C1CCCn2nccc21)N1C2C(NC(=O)CC3CCCCC34CC4)C(C2)C1 21694,N1(C(CN(c2ccccc2)CC=C)=O)CCN(C(c2cc(Cl)no2)=O)C2CC12 21695,CCCC(C(=O)N(CC(C)CNC(c1ocnc1C)=O)C)C(C)C 21696,N1(C(C2CCC(O)C2)=O)CCC(C(=O)NCc2ncn(C3CC3)n2)CC1 21697,O=C(C(F)(F)F)N(N1CC(CNCCO)(Cc2ccccc2)C1)CCCO 21698,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)ncn1)=O)C2 21699,c1(C(=O)NCCc2cn(-c3c(C)c(I)ccc3)nn2)ccc(C#N)nc1O 21700,c1(C(N2CCC(N(C(C)=O)CC)C2)=O)cc(C)cc([N+](=O)[O-])c1Br 21701,Cc1nn(C)cc1C(C)NC(C1CSCCN1C(=O)CC(C)(C)C1CC1)=O 21702,N1(C(CN2C(C)CCC2C)=O)CCC(CNC(=O)CC2CCCC2)C(CO)C1 21703,C1(C(N(C)CC2(C)CCCO2)=O)C2CC1N(C(C1CCOCC1)=O)C2 21704,c1(NC(C2C(CNC(COCC(N3CCCC3)C)=O)CC2)=O)cc2c(nn1)CCC2 21705,C1(n2cc(N(C)CC3CC3)nn2)CCN(C(c2cc(CO)[nH]n2)=O)CC1 21706,C(CCC(C)(C)NC(=O)CCSc1nccn1C)NC(C(CC)OC)=O 21707,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21708,c1(SC)nc(Cl)c(CC2(C)CCN(C(=O)CN3CCS(=O)(=O)CC3)C2)c(Cl)n1 21709,N1(C(CCN(CC)CC)=O)CCCC(Cc2nnc(N(C)C)o2)C1 21710,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21711,c1(C(=O)NC(C)Cn2cc(-c3ccsc3C(=O)O)nn2)ccc2c(c1)C(=O)C(=O)N2 21712,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(=O)CC1OCCCO1)C 21713,C(C(CNC(=O)C=C1CCC1)C(F)(F)F)NC(C(CC)(C)OC)=O 21714,N1(C(C(c2ccn(C)n2)C)=O)CCCCCC1C(=O)N(C)Cc1nccs1 21715,CCCCC(O)C(=O)N1CCCC(C(C)C(=O)NCCC(CC)CO)C1 21716,C(=O)(C(C)(O)CC(C)C)NCC(CNC(c1c(C)nc(Br)s1)=O)F 21717,N1(C(C2CC(NCc3c(C)nn(C)c3OC)C2)C(=O)NC)CCS(=O)(=O)CC(C)C1 21718,c1(C(N(C2CCN(C(c3ccc(C)c(Cl)c3)=O)C2)CC)=O)ccc([N+](=O)[O-])s1 21719,N1(C(C(C)CC2CCN(C(=O)COc3ccccc3)C2)=O)CCCC(O)C1 21720,C(=O)(CCC(=O)NCC1(C)CCN(C(=O)Cc2ccoc2C)C1)NCCCOC 21721,c12nnc3n1CCN(C3)C2=O.C(CCC(=O)NCc1cnc(C2CC2)nc1)SC 21722,c1(COC(CCC(N2C(C(=O)NCC)CC3CC32)=O)=O)oc(C)nc1C 21723,c1(CCC(=O)NC2C=CCN(C(c3ccc(Br)cc3)=O)C2)ccccc1CO 21724,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21725,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cnc(C(C)(C)C)[nH]1 21726,C=CCCCCCCCC(=O)NC1CC1CNC(=O)C(c1c(C)n[nH]c1C)OC 21727,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C=CC)C1 21728,CCCCCCN(C(=O)CCOCCOC)CC.C1(C(=O)N)CCCCS1 21729,c1(C(N2CC(CNC(c3cc(Br)no3)=O)C3C2C3)=O)ncc2ccccn12 21730,N1(C(C2CC(N(C)CC)C2)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21731,C12(CC(F)(F)C1)C(=O)N2.C1(C(=O)N(C2CCC2)CC2CC2)CC12CCOC2 21732,O=C(O)CC1CCN(C(=O)CCSc2ccccc2)c2ccccc21 21733,C(CCCC(=O)NC1(CO)CCN(C(=O)Cn2cc(C(C)O)nn2)C1)NC(=O)OC 21734,CC1=C(C(=O)O)CN(C(=O)NCc2nc3cc(F)ccc3s2)CC1 21735,c1(C2CCN(C(c3scnc3Cl)C(=O)NC(C)C)C2)cccc(F)c1 21736,c1(CCC(=O)NCCN(C(C2(O)CC(F)(F)C2)=O)CC)ccc(Br)cc1F 21737,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21738,N1(C(C2CCC(=C)CC2)=O)CC2(CC2)CC1C(=O)Nc1ccnn1C(C)C 21739,c1(C(N2CCNC(C(=O)Nc3cnc(Cl)cc3I)C2)=O)c(F)ccc(Cl)c1Cl 21740,c1(C(=O)NC23CC(NC(Cc4nc(C)[nH]n4)=O)(C2)C3)cc(Br)c(C)cc1F 21741,C(=O)(CCCN=[N+]=[N-])NCCC(C(C)C)NC(C1(C)CC1)=O 21742,Cc1cc(NCC2CCCC(NC(=O)OC(C)(C)C)C2)n2nc(C)nc2n1 21743,N1(C(C2(O)CCC2)=O)CCCC2C1CCN2C(c1cn(CC(F)(F)F)cn1)=O 21744,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21745,c1(OC(C)C)ccc(C(=O)NCCNC(C23CCCN2CCC3)=O)c(O)c1 21746,C(N=c1[nH]c(C)cc(=NC(C)Cc2c(C)noc2C)[nH]1)c1cnn(CCC)n1 21747,c1(OCC(N2CCC=C(Br)C2)=O)ccc(-c2ccncc2)cn1 21748,CCS(=O)(=O)c1ncc(CN2CCN(C(=O)NC3CCN(C)CC3)CC2)cc1Br 21749,N1(C(C2(C)CC(OC)(OC)C2)=O)CC(C)N(C(C2C3CC4C(C3)C24)=O)CC1C 21750,CCC(C)C(C)C(=O)c1ccccc1CC(=O)NCCC1OCCC1C 21751,c1(CC)nc(C(=O)NC2CN(C(c3noc(C4CC4)c3C)=O)CC2F)c(N)s1 21752,c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccn2ncccc12 21753,C(CCC(C)(C)C(=O)N1CCOCC(CC2CC2)C1)NC(c1ncc(C)nc1)=O 21754,c1(C(N2C(C(C)NC(C(C3CCC3)OCC)=O)CCCC2)=O)c[nH]nc1[N+](=O)[O-] 21755,CS(=O)(=NC(=O)c1ccc2n[nH]c(Br)c2c1)c1ccccc1[N+](=O)[O-] 21756,C(CS(C)(=N)=O)NC(C(n1cc(CC2(O)CCC2)nn1)C)=O 21757,O=C(C1=CCCOC1)NC1CC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C12CCC2 21758,C1(CNC(C23CCC(OC)C2C3)=O)CC(C(=O)NCC(O)C2CC2)=NO1 21759,c1(C(=O)NC2C(NC(C3N(CC)CC3)=O)CC2)oc2ccccc2c1COC 21760,c1(CSC)c(F)ccc(F)c1C.c12n[nH]c(c1C#N)NC1C(C1)C(=O)N2 21761,Cc1cc(C(N2CCC(C(C)(C)NC(=O)CSCC(N)=O)C2)=O)cc(C)c1F 21762,c1(NC(=O)COC2CC(OCC)C2)c(Cl)cccc1Cl.C12CCOC(C1)C(=O)N2 21763,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21764,CON(C)C(=O)C1CN(C(C2(N(C(=O)CCc3nncn3C)C3CC3)CCC2)=O)C1 21765,C12(CNC(C3(CCC=C)CC3)=O)CCCC1N(C(c1ccc(F)cn1)=O)CCC2 21766,Cc1ccnc(C(=O)NC2CCN(C(=O)CN3CCCC3(C)C)CC2CO)c1O 21767,CC1CCN(C(=O)C(N2CCC3CCOC3C2)=O)CCN1 21768,N1(C(C2CC(O)(CC#C)C2)=O)CCOC(CCNC(=O)CC2COCC2O)C1 21769,C1(F)(CNC(C2(C(=O)N)CCC2)=O)CCCN(C(=O)CCOC2CCOC2)C1 21770,N1(C(CCC(C)C#N)=O)CCC(S(C)(=N)=O)C1 21771,N1(C(=O)CC2CCC2)CCC(CCn2cc(C3(NCC4CC4)CCCC3)nn2)CC1 21772,CP(C)(=O)CC(=O)N1CCOC(CNC(=O)CC2CCC(=O)O2)C1 21773,c1(C(=O)NCC2C(C(=O)NCc3c(C)occ3)OCC2)cnc(S)nc1 21774,N1(C(CCN2C(=O)CCCC2)=O)C2CCCC1CN(C(c1ccc(CO)o1)=O)C2 21775,c1(C(N2CCOCC(NC(C(C(C)(C)C)=O)=O)C2)=O)ncn2cccnc12 21776,N1(C(C(Cc2ccco2)NC(CC2C(C)(C)C2)=O)=O)CCCC2(CCCC2)C1 21777,c1(CC(N2CC(CC(C(N3C(CNC(C)=O)CCC3)=O)F)C2)=O)cncc(C)c1 21778,c1(SC)cc(C(=O)NC(C)CNC(=O)C(C2CCCCCC2)O)ccn1 21779,c1(OC)cc(F)c(C(=O)N(C(C)C(=O)NC2CCS(=O)(=O)C2)CCO)cc1Br 21780,C12(NC(=O)Cc3cnccn3)CCCN(C(C3CC3(Cl)Cl)=O)CC1C2 21781,c1(CN2CCC(O)(CNC(COCCOC)=O)C2)cccc2sccc12 21782,c1(CC)occc1C(=O)NC1(CCNC(c2coc(N(C)C)n2)=O)CC1 21783,CCC(C)CCCCC(=O)N1CCC(C2(NCc3cnc(C#N)cn3)COC2)CC1 21784,C1(CNC(=O)COCC(F)F)CN(C(c2ccc(Cl)cn2)=O)C2CCN1C2 21785,c1(CC)cc(N2CCSC(CNC(=O)C(C#N)CC)C2)nc(CC)n1 21786,N1(CC)CCN(CC(N2CCC(OC(=O)Nc3ccc(F)cc3)C2)=O)C(=O)C1=O 21787,CC1CC(C(=O)NCC2(F)CN(C(c3c(F)cccc3Br)=O)C2)=NO1 21788,C(=O)(CC(C)C(F)F)NCC(CNC(=O)CSc1nncn1C1CC1)OC 21789,C1(CC(=O)NC(C(C)NC(COCC(=O)OC)=O)C)CCC(=O)N1C 21790,C(C(=O)N(OC)C1CCC1)N(CC#C)C(C12CCC(C1)C2)=O 21791,C1(C2CCN(C(=O)CCCCC(N)=O)C2)(NC(c2n[nH]c(CC)c2Br)=O)CC1 21792,N1(C(c2n(COC)ncc2)=O)CC2CC2(CNC(c2ccc(F)o2)=O)C1 21793,C(C)(C(CC(=O)N1CCC(CO)C1(C)C)NC(=O)CC1CC=CC1)OC 21794,c1(C(N2CCC(NC(C)C)C(C)C2)=O)ccc2c(c1)CCC(C)(C)O2 21795,N1(C(CC2(CSC)CC2)=O)Cc2[nH]nc(C(=O)NCC=CC3CCOCC3)c2C1 21796,c1(C(=O)NCCCC(C)NC(c2cc(F)cnc2O)=O)cc2n(n1)C(C)CCC2 21797,C1(C(=O)NCCNC(=O)OC)CC(F)(F)CN1C(=O)Cc1ocnc1C 21798,C(=O)(CC(C)(C)COC)NCc1cn(CCNC(C(CC)(C)C)=O)nn1 21799,c1(C(=O)N)cccc(CC(c2coc(C3CC3)n2)=O)c1.N(CCOC)(CC)CC 21800,N1(C(c2c[nH]c3ncc(C(N)=O)cc32)=O)CCc2cc(C#N)ccc2C1 21801,N1(C(c2cc(C)sc2C)=O)CC(NC(c2cn(C3COC3)nn2)=O)CC(C)C1 21802,c1(N(C)C)cccc(CC(N2CCCCC2CCNC(C2CCCCO2)=O)=O)c1 21803,C(=O)(NNc1nc(C)ns1)C1(O)CCN(c2c(-c3c(C)nc(C)o3)cccc2)CC1 21804,c1(C(=O)NC(C#C)C)n[nH]c2c1CCN(C(c1cccc(F)c1C)=O)C2 21805,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CCC2)CC1 21806,c1(C(=O)OCCOCC2(OC)CCN(CC(C)(C)C)C2)c(C)ccc(F)c1N 21807,C1(C(N2CC(NC(c3c(C)oc(-c4ccccc4)n3)=O)C2)=O)CCCC(=O)N1C 21808,c1(C(=O)NC2CC(C)(NC(C(c3cncnc3)C)=O)C2)ccc2nn[nH]c2c1 21809,C(=O)(CC(Cl)Cl)NC1(NC(C=CC=N)=O)CC1 21810,N1(C(C2CCC(C(F)(F)F)CC2)=O)CC2CCC1(CN(C(C1CC1F)=O)CO)CC2 21811,c1(C(=O)NCC=CCNC(C(CO)OC)=O)cccc(NS(C)(=O)=O)c1 21812,CCCCC(C)CCC(=O)N1CC2CC(C(=O)NCCCCCCO)(C2)C1 21813,N1(C(C2(COC)CCOC2)=O)CCC(F)(CNC(=O)Cc2ccon2)C1 21814,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21815,N1(C(C(P(C)(C)=O)O)=O)CCN(C(c2ccc(C(N)=O)s2)=O)CC(CO)C1 21816,Cc1c(Cl)ccc2c(CC(=O)NC3CCC(C)(c4ccccc4)C3OC)c[nH]c12 21817,CC1CC(CN(c2ccc(C(=O)NC3CC3)cc2)C)CN(C(=O)C(F)Cl)C1 21818,c1(C(C(=O)O)NCc2cnc(C3CCC3)s2)ccc(Br)cc1 21819,C1(C(C)(C)C)(CNC(c2cn(C)nn2)=O)CCN(C(=O)CC2CNC(=O)C2)C1 21820,CN1CCN(c2nccc(N(CCCN(C)C)C(=O)Nc3cccnc3)n2)CC1 21821,N1(C(C2C(C)C2)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21822,C1(CC)(NOC(c2scnc2COC)=O)CCN(C(C2CC23CCOC3)=O)CC1 21823,C(=O)(n1nccc1C(=O)NC(CNC(c1cccnc1)=O)CC)OC(C)(C)C 21824,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CC2(C)CC2(F)F)C1 21825,c1(C2(C)CC2NC(N2CCC(Cc3ccco3)CC2)=O)cccc(Cl)c1 21826,C(=O)(C(=O)CCC(C)C)NC(CCN(C(c1c(C)coc1)=O)C)C(C)(C)C 21827,C1(NC(c2cn(CC)c(=O)nc2O)=O)CN(Cc2c(O)cccc2O)CC1(C)C 21828,C1(C(=O)NCCC2(OCC)CN(C(=O)COc3cnn(C)c3)C2)CCC(C)(C)O1 21829,C(CC(C(C)(C)C)NC(c1coc(Cl)c1)=O)N(C(=O)CC1CCOCC1)C 21830,C(=O)(C1=CC2(CCOCC2)C1)N1C(C2(NC(CCNS(C)(=O)=O)=O)CC2)CCC1 21831,N1(C(c2cc(OC)no2)=O)CC2CC(C1)N2C(c1ccsn1)=O 21832,CC1C(C(N2CCC(C3OCCCC3NC(=O)C#CC3CC3)CC2)=O)CCN1C 21833,N1(C(c2cnc(SC)s2)=O)CCCOC(CCNC(C2CC2C)=O)C1 21834,c1(C(=O)NCC(C)(C)OCC(=O)NC2(C(C)C)CCOC2)cnn2ccn(C)c12 21835,C(=O)(C1=CC2C=CC(C1)C2)NC1COCC1N=[N+]=[N-].C(CCCC(=O)N)OCC 21836,CC1(C)CCCC(C(=O)NCc2ccc(C(=O)NCCc3cccnc3F)s2)C1 21837,C(=O)CC(C(C)C)SC.O(NC(=O)CNC(=O)C)CCCC=C 21838,C1(NC(CNC=O)=O)CCCCC1NC(=O)Cn1cc(CSC)nn1.C1(C)CC1 21839,c1(CCCC(=O)NC(C)CNC(C2CCC2(F)F)=O)ccc(F)cc1 21840,CN1C(=O)C2CN(C(C34CC(NC(=O)Cc5cncs5)(C3)C4)=O)CC2C1=O 21841,c1(NC(C(C)N(C(c2ccco2)=O)C2CC2)=O)ccc2c(c1)OCC2 21842,c1(CCC(=O)NCC(C)NC(C2CC(C(C)(C)C)C2)=O)ccccc1OC(F)F 21843,C1(CC=C)(NC(=O)CC(C)OC)CCN(C(=O)CSC(F)(F)F)C1 21844,Cc1cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]c(=NCC2CNC(=O)CO2)[nH]1 21845,c1(SC)ccc(NC(C2CC(=O)NC(c3ccccc3)C2)=O)cc1Cl 21846,N1(C(=O)CCCc2cnn[nH]2)CCC2(CC1)CCN(C(C13CC(F)(C1)C3)=O)C2 21847,C(=O)(N(CCC(=O)NCC1CC(=C)C1)OC)c1n[nH]c(C)c1C 21848,N1(C(N(CC(c2ccc(F)cc2)C)C)=O)CCS(=O)CC1C 21849,C(=O)(CC(C)C(F)(F)F)NC(CC)CCC(=O)NCC1CC12CCCCC2 21850,Cn1cnc(N2C3CCC2C(CNC(c2cc(=O)cc[nH]2)=O)C3)c(Br)c1=O 21851,c1(CC(N2CC(NC(C3C(C)C3C)=O)(CO)C2)=O)ccc(C#N)cc1 21852,C(C(C)C)(C(O)C(=O)NC(C)(CNC(c1cccc(C)n1)=O)CC(C)C)OC 21853,C1(C=C)(C(=O)NC2CN(C(C(CC#C)OC)=O)C2)CCN(C(=O)OCC)CC1 21854,N1(C(C=C(C)C(C)(C)C)=O)CCC(CCNC(c2ccnn2C)=O)C(F)(F)CC1 21855,C(=O)(C(CCNC(=O)C(C)c1ccsc1)OC)NCC(C#C)CC 21856,C1(C(=O)NC(CNC(C(C)SC)=O)(C)C2CCC2)CCNC(=O)C1 21857,CN=c1nc(C(N2CCN(C(=O)CCCC3CCC3)C(C3CC3)C2)=O)cc(C)[nH]1 21858,c1(C(=O)NCC(C)NC(c2nn[nH]c2C(F)(F)F)=O)n[nH]c(C2CC2)c1Br 21859,c1(OC)ccc(CNC(c2cnccc2OC(F)F)=O)c(C(F)F)c1 21860,C1(NC(C2(C)CCCC2)=O)CCOC(C(=O)NC(C2CCCCC2)CO)C1 21861,C1(OC)CCC(C)N(C(=O)C(=O)NC2CC3(C2)CC(CO)C3)C1 21862,Cc1cc(C(=O)NC(C)CCNC(c2c(C)noc2N)=O)nc(O)c1 21863,C1(NC(CCNC(=O)NC)=O)CN(C(c2cccnn2)=O)C2(CCC2)C1 21864,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 21865,c1(C(=O)NCCC(C)N(C(C2C(CC)OCC2)=O)C)c[nH]cc(Cl)c1=O 21866,Fc1cc(NC2CC2)cc(Cl)c1.c12c(ccnc1Cl)CS2 21867,N1(Cc2c(C(C)C)cccc2)CCC2(CCN(c3ncc4sccc4n3)C2)C1 21868,c1(OC(C)=O)cc(CNCC2CCCN(C(=O)CCC(C)N(C)C)C2)ccc1C 21869,c1(-c2ccc(SCC)s2)c(C(=O)NC)nc2ccccn12 21870,c1(C(N2CC(F)CC2CO)=O)cc2ccc(-c3ccc4n[nH]cc4c3)cn2c1 21871,N1(C(c2c(CC)nco2)=O)CC2CCC(N(C(=O)C(C)CC(F)(F)F)C)C2C1 21872,c1(C(N2C(CN(C(=O)C3=C(Cl)CC3)C)COCC2)=O)noc2c1COCC2 21873,C1(O)(C(C)NC(C2(CC=C)CCC2)=O)CCN(C(c2ccc(CC)s2)=O)C1 21874,C1(C(=O)Sc2cccc(Nc3cncc(C(=O)OC)c3)c2)CCc2ccccc2C1 21875,C1(NC(C(COC)NC)=O)CC2CCC1N2C(c1ccc(OC)c(O)c1)=O 21876,c1(CN(CCNC(c2coc(Cl)n2)=O)C(C2CC(F)(F)C2)=O)ccccc1 21877,c1(C(=O)NCC2(C(C)NC(C3CC3C(C)(F)F)=O)CC2)ccnc(Cl)c1F 21878,C1(C(=O)Nc2n(CC)ccn2)CCCN(Cc2nc(-c3ccccc3)no2)C1 21879,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 21880,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 21881,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(CCO)C1 21882,CCC(CCC(=O)NC1(C(=O)OC)CCC1)NC(c1ccc(CSC)c(O)c1)=O 21883,N1(C(=O)OC)CCCC(c2nc(C(C)C)no2)C1.c1(CC2CC2)cnccc1C 21884,N1(CCNC(=O)NC(c2ccc(Cl)cc2)C(N)=O)CCCCCC1 21885,N1(C(C2C(C(=O)O)C23CC3(F)F)=O)CCc2c(I)n[nH]c2C1 21886,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 21887,CCC(C)C(C(=O)N(CC(F)F)CCOC)NC(=O)C(=O)N(C)C 21888,C1(C(=O)OCC)CCN(C(=O)C2CCCN2C(=O)CC2(C(=O)OC)CC2)O1 21889,c1(C(=O)NCc2ccc(C(=O)NC(c3cccnc3O)C)s2)cn(C)ccc1=O 21890,C(C(C)N=c1[nH]c(=NCC2CC(C)(C)NC2=O)c2sccc2[nH]1)N(C1CC1)CC 21891,CC(C)C(C)(CNC(=O)C(CNC(C1C=CC=CC=C1)=O)N(C)C)C(C)C 21892,CN1CCC2(CCN2C(=O)CCC2CCCCN2C(=O)CSC(C)(C)C)C1 21893,c1(C(=O)NCCC(C)N(C)C(c2cc(-c3cccs3)on2)=O)csc(O)n1 21894,c1(OCC(=O)NCCNC(=O)C2=CCSC2)ccc(I)cc1Br 21895,c1(OC)cc(Br)cc(C(N2CCN(C(=O)C(C3CC3)N(C)C)C(CF)C2)=O)c1OC 21896,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 21897,c1ncc(Cl)cc1[N+](=O)[O-].C1C(C(C)C(C)C)NC2(CCCCC2)C(=O)N1.CC 21898,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOCC2CNC(c2cccnc2)=O)cc1 21899,N1(C(c2ccc(CC)s2)=O)CCC(C2CN(C(c3c[nH]c(C#N)c3)=O)C2)CC1 21900,CCN=C(NCC(C)Oc1cccc(C)c1)N1CCn2c(NC(C)=O)nnc2C1 21901,N1(C(C(C)OCCC(C)C)=O)CCC(C2(NC(=O)CNC(N)=O)CC2)C1 21902,c12cnn3c1CN(CC3)C2.c1(-c2nnc(C(C)C)s2)cnc(C(C)(C)C)nc1 21903,C1(C(=O)NC(C(OC)OC)C)CC(=O)N(C2CN(C(=O)CCN3CCC3)C2)C1 21904,c1(C(=O)NC(CNC(C#CC2(C)CC2)=O)C2CC2)ccc2cc[nH]c2c1F 21905,c1(C(=O)NC2C(OC)CN(C(C3(CC)CC3)=O)C2)c(C)nc2sccn12 21906,C1(C(=O)NCCCN(C(c2c(C)cc(C)cc2C)=O)CC)CCCCC12CCC2 21907,C1(C(N(CCCCO)C)=O)CC(=O)CN1C(c1ccccc1)=O 21908,C(CCCCC(=O)N(C1CCC(NC(C2CCCC(C#N)C2)=O)CC1)C)OCC 21909,c1(CCNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 21910,C(=O)(C(F)CCC(C)C)N1CCCC(C(NOC)=O)(CO)C1.C1CNC(=O)O1 21911,Cc1ccc(C(CNC(=O)N(CCCC(F)(F)F)CCC#N)O)cc1 21912,c1(C(=O)NC(CNC(C(c2cc(F)cc(F)c2)C)=O)(C)CO)cnc2[nH]cncc1-2 21913,C1(NC(C)CC(N)=O)CCCN(C(=O)C(N2CCN(CCF)CC2)=O)C1 21914,C(=O)(CC(C)(C)C(C)(F)F)NCCC1N(C(C2CCN(C(C)C)CC2)=O)CCC1 21915,c1(C(N2CCC(NC(c3c(C)nn(C)c3C)=O)C2)=O)cc(Br)c2ccccc2c1 21916,c1(CNC(C(C2CCCCC2C(F)(F)F)CC)=O)ccc(Cl)c(Cl)c1C 21917,Cc1cc(C)c(C(=O)NCCCC2CCCCN2C(=O)Cn2cnnc2)c(C)c1 21918,N1(C(C2C(C(=O)OCC)C=C2)=O)CCC2CCC(NC(=O)COCCC(C)C)C1C2 21919,CCCC(C)(C)C(=O)NCCNCc1ccc(C(=O)N(C)C)cc1 21920,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)CC2)C1 21921,N#CC1CCC(CC(=O)NC2CC(C(=O)NC3C=CCCC3)CC2O)C1 21922,N1(C(COCCC)=O)CC2CC2(CN(C)C(C2CC(c3cccc(F)c3)C2)=O)C1 21923,N1(C(CCc2cc(C)[nH]n2)=O)CCCCC1C(=O)NCCc1csnn1 21924,Cc1cnccc1C(=O)NCCC1CCCN1C(C1COC1)=O 21925,c1(C(=O)NCC23C(CN(C(C(CSC)C)=O)C2)C3)cccc(=O)n1C 21926,C1(CNC(C23CC(CO2)C3)=O)CC(F)(F)CN1C(C1CCC1(F)F)=O 21927,Cc1cc(C(=O)NC2CCC2NC(=O)C2=CCC2)nn1C1CCCCC1 21928,CCC1=NOC(C(=O)NC(CCC2CCC2)C(=O)Nc2ccccc2OC)C1 21929,C1(CNC(C(C)c2cccs2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C 21930,Cc1ccc2c(N3CCOC(CN(C)C)C3)nc(=NC3CCCCCC3C)[nH]c2c1 21931,C1(C(=O)NC2(CC(=O)N(C)Cc3c(C)cco3)CC2)CCCCN1C 21932,CC(C)(C)C(=O)C(CCN)=O.C1(NC(C2CC(F)(CO)C2)=O)CCC(C(N)=O)C1 21933,C#CCC(C(=O)NC(C)(C)C1CC1c1cccnc1)NC(=O)C=CC(C)C 21934,C1(C(N(CC(O)C2CC2)C)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1(C)C 21935,C1(C)(C(=O)NCC2CC3N(C(C(=O)NCC)=O)C(CC3)C2)CC(C(C)(C)C)=NO1 21936,Cc1cccc(CNC(=O)C(Cc2ccccc2I)NC(=O)OC(C)(C)C)n1 21937,N1(C(C23CCCC(C(=O)OC)(C2)C3)=O)CCCC2(CCCC2)CC1 21938,C(=O)(C1=CNS(=O)(=O)N=C1C)N1C2CC(NC(C(CC)F)=O)C(C)C1CC2 21939,Cc1ccc(C(=O)NC(C2CN(C(=O)C(C)c3cccs3)C2)C)nc1C 21940,C1(NC(c2cn(CCC)nn2)=O)CCN(C(C2CC(O)C2)=O)CC1F 21941,Cc1cncc(C)c1C(=O)NC1CC(C(F)C(N2CC3CC3(CO)C2)=O)C1 21942,C(=O)(C(F)(F)C1=CCOCC1)NC(C)C(C)NC(C1(CO)CCCC1)=O 21943,N1(C(C(COC)NC(=O)C(C)Cn2cccn2)=O)CC(C)OC(C)(C)C1C 21944,c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCCCC2C(C)CO)cn1 21945,N1(C(CSC(C)C)=O)CC2CC(NC(=O)C=CCc3ccccc3)C1C2.C(N)(=O)N 21946,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(=O)Cc1ccno1 21947,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(c4ccnc(Cl)c4)=O)C3)c2c1 21948,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 21949,CCC(C)(CNC(c1ccnc(C)n1)=O)C(=O)NCC1C=CCOC1 21950,N12CCN(CC1)C(=O)OC2=O.C1(NCCC(=O)OC)CC(OC(C)(C)C)CN1C 21951,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC#N 21952,Cc1cnn(C(C)C(=O)NC2(CCNC(c3ccn(CCF)n3)=O)CC2)c1 21953,C1(CN(C(c2ccc(-c3ccco3)[nH]2)=O)CC)CCN(C(c2ccc[nH]2)=O)C1 21954,c1(CN2CC3C(C(=O)Nc4cc(O)ncc4Br)(C3)C2)ccc([N+](=O)[O-])cc1O 21955,n1(C(C)C)cnc(C(=O)NC(C(=O)NCC2(C)CC2(C)C)C2(O)CCC2)n1 21956,c1(C(N2CC(O)(CCNC(C3CCOC3)=O)C2)=O)coc2c1CCCC2 21957,C1(C(C)C(=O)NCCCc2ccsc2)CCN(C(c2scnc2Cl)=O)CC1 21958,CN1CCN(C(c2ccsc2)=O)CC1C(=O)NCC1CCCC(F)C1 21959,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CC2)C1)N(C)C 21960,C12COCCC1C(=O)NCCn1cc2nn1.n1(CC(C)C)ccc(C(F)F)n1 21961,c1(CSCCC)ccc(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)o1 21962,c1(C(CC(=O)NC(CC=C)CNC(c2csc(C(N)=O)n2)=O)C)ccc(F)cc1 21963,Cc1oc(-c2ccc(F)cc2)nc1C(=O)NCC1CCC=CO1 21964,c12c(Cl)cc(cc1Cl)NC(=O)NC(C)CO2.C1(OC2(OC)CC2)CCN(C)CC1 21965,C1(OC)COCCN(C)CCNC1=O.c1(OC)ccccc1.C1(=O)CN1 21966,C(=O)(CCS(N)(=O)=O)NC(CC(C)C)CNC(=O)CCC(=O)NC1CCCC1 21967,C1(=O)CC(C)N1.C(=O)(C(C)(C)OCC)N(CCC)CCC.C1CC1 21968,c1(C(=O)NC2CCC(C)N(C(c3cccnn3)=O)C2)cccc2c1CCCCC2 21969,C(c1c(C)coc1C)=CC(N1CCC(CNC(C(C)=CC)=O)C1)=O 21970,Cc1ncccc1C=CC(=O)NC1(CN(C)C(c2nccn2C)=O)CC1 21971,c1(NC(c2nncn2C)C)[nH]c(=NCCc2ccncc2Br)nc2scnc12 21972,N1(C(=O)CC(F)(F)F)CC2CCC1C1CN(CC3CC3(Cl)Cl)CC21 21973,C(C(C(=O)NCCCF)N1CCC2CCC12)(C1CC1)OCC 21974,c1(OC)c(C(=O)N(C2C3CN(C(c4ccc(C)cc4O)=O)CC23)C)cccc1F 21975,C1(NC(COCC(C)(C)C)=O)CCN(C(C2CCC(N(C)C)CC2)=O)CC1CO 21976,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)N(C)CCF 21977,c1(CN2CCC(CC(N3CC4CC4C3)=O)CC2)cccc2ccncc12 21978,C1(CNC(=O)CCN2CCC2)CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1 21979,CN1CCOC(C(=O)NCC(C)(C)OCC(=O)NC2CC2(C)C)C1=O 21980,Cc1cccc(C)c1C(N1CCC(F)(CNC(C2CCC2CC(C)C)=O)CC1)=O 21981,c1(CC)nc(C(N2CCCC2CC(=O)NC(C)C2CC2)C)cs1 21982,C(C(C)(C)CC(=O)N(C1CC(C(N2CC3CCC3(C)C2)=O)C1)C)OC 21983,C1(CC=C)(NC(c2cnc(C(F)F)o2)=O)CN(C(c2cc(C(C)C)cs2)=O)C1 21984,Cc1cc(C)c(CN2CCC(N(C(=O)C(C)C)C)C2)cc1C 21985,c1(CC)ncc(C(=O)NCC2CCN2C(=O)CC2CS(=O)(=O)C2)c(C)n1 21986,c1(C(N2C(CNC(CC=CC)=O)CC2)=O)onc(Cl)c1C 21987,C1(N(C)C(C2CCCO2)=O)CC2CCC(C1)N2C(=O)Cc1ccc2ccoc2c1 21988,Cc1cccc2cc(C(=O)NC34CCC(CC3NC(C35CCC3C5)=O)C4)[nH]c12 21989,N1(C(CC2C(C)(C)OCC2)=O)CC2CCC(C1)N2C(C12CCCN1CCC2)=O 21990,CCCCC(C(=O)NC1(CC(N)=O)CCCN(C(c2cnc(N)cn2)=O)C1)C(C)C 21991,Cc1cc(C(=O)N(C)Cc2ccn(C)n2)nn1C(C)(C)C 21992,c1(C(N2CC(CNC(C3CN(CC(C)C)C3)=O)C2)=O)ccc2c(O)ncnc2c1 21993,c1(C(=O)NCC2CC(NC(c3occ4c3CCCC4)=O)C2)ccnc2[nH]cnc12 21994,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 21995,c1(CNC(C(C)OCCOC)=O)ncoc1C1CN(C(C2CCCS2)=O)C1 21996,N1(C(C2CCC(NC(C)=O)CC2)=O)CCC2(CCN(C(C3CCCS3(=O)=O)=O)C2)C1 21997,C=C(Cl)CCC(=O)NC(c1ccccc1)C(=O)Nc1ccnn1COC 21998,C(=O)(C1CCc2nccn21)NC(C)C(=O)NOC1CCCCCC1 21999,C(N=c1ccnc[nH]1)CC1OCCN(C(C2CCCN2C2CC2)=O)C1 22000,C1(C(=O)NCC2C(C)CN(C(=O)Cc3ccco3)C2)CCc2ncncc2C1 22001,C12(NC(C=Cc3c(C)ccs3)=O)CCC1CN(C(=O)C(C)c1cc[nH]n1)C2 22002,Cc1cc(N2CCCC(NC(C3CC4CCC(C3)S4)=O)CC2)n2nc(C)nc2n1 22003,C1(=O)CS(=O)Cc2nc(cs2)N1.CC(C)CC1CC1C1CC1 22004,c1(N2CCCC(OC)CC2)ncc2[nH]ncc2n1 22005,c1(C(C)N(C)C(=O)Nc2cnn(C3CCOC3)c2)ccc(Cl)cc1 22006,CC1CCC(NC(c2ccc(O)nc2Cl)=O)CN1C(c1cnccc1Br)=O 22007,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22008,C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1cccc3nncn13)=O)C2 22009,N1(C(C=CCOC)=O)CCC(NC(=O)COc2cccc(C)c2)C(C(C)C)C1 22010,C1(CNC(Cc2nc(C)sc2)=O)CCCCCN1C(C1CCCC1(F)F)=O 22011,c1(CNC2CCC(C(=O)NCc3ccn(C)n3)CC2)c(Br)ccc(Cl)c1F 22012,N1(Cc2cc(Cl)c(Br)nc2)CCC2(CCSCC2)C1 22013,c1(C(=O)NCC2CC(COC)CN2C(c2cnsc2)=O)cc(Br)ccc1Cl 22014,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CC=C)=O)CCC1CC2 22015,c1(C2C(C(=O)NCC(C)(C)C(C)(C)C)C2)c(F)cccc1F.C(=O)(CCC(=O)O)N 22016,N1(C(C(CCCC)=O)=O)CCC2CCCC12C(=O)NCC1CC2(CCC2)C1 22017,c1(C(N(C(CCNC(C(C=C)(C)O)=O)C)C)=O)cnc2onc(C)c2c1 22018,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22019,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22020,c1(CNC(=O)CC2CCCN2NC(CC2CN(C)C2)=O)ccc(C(N)=O)cc1 22021,C(C)(C(=O)N1CCC(N(C(=O)CC(F)F)CC(C)C)CC1)(C(C)C)NC(C)=O 22022,C(CCN=c1cccc(S(=O)(=O)NC(c2cccc(F)c2F)C)[nH]1)N(CCCC)C 22023,C(=O)(CCCCC(F)F)N1CC(C2(NC(=O)CC3CCCOC3)CC2)OCC1 22024,C(=O)(C1=CCCOCC1)NC1CCC(CNC(C(C)N(CC)CC)=O)CC1 22025,Cc1cc(C)c(C(=O)NCC2CCCC2NC(c2cccc(O)n2)=O)cn1 22026,c1(C(=O)NC(CNC(c2ccc(SC)o2)=O)C2CCC2)c(C)nnn1CC 22027,C1(CNC(C(C2CCC2)OC)=O)CC2CCC(C1)N2C(=O)Cc1csnn1 22028,N1(C(CCS(CC)=O)=O)CCC(=O)NC2CN(C(=O)C(C)=CC3CC3)CCC12 22029,C1(C(=O)NCC(C)N(C(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22030,N1(C(COC)=O)CCC(NCC(C(C)C)c2ccnn2C)C(F)(F)CC1 22031,C1(CC)CCCCC1C(=O)NCC(C)(C)Nc1cc(C(=O)OC)no1.C(=O)OC 22032,c1(C(N2C(C)CCC2)=O)cc(C(=O)N(C)NS(CCCC)(=O)=O)ccc1C.NC 22033,C#Cc1ccc(CC(N2CC(NC(c3cnccn3)=O)CC2CO)=O)cc1 22034,c1(C(C)C)conc1C(N1CCC1CC(N1CCCC1CN(C)C)=O)=O 22035,N1(C(c2c(CNC(CCC(C)OCC)=O)cnn2C)=O)CCCC12CCCC2 22036,Cc1ccc(C(C(=O)NCC(C)(C)OC(C)C)SC2CC2)cc1.C1(=O)CCCN1 22037,c1(C(N2CC(N3CCC(NCC(C)C(F)F)CC3)C2)=O)ccc2nonc2c1 22038,N1(C(C2C(COC)(COC)C2)=O)CC(F)CC1CNC(c1cc(C2CC2)cs1)=O 22039,C1(N(CCOC)C(c2ccncc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1 22040,N1(C(c2cc(CC)c(CC)o2)=O)CCC(CNC(C2CS(=O)(=O)C2)=O)C12CCC2 22041,C1(CNC(=O)C(=O)Nc2cccc(F)c2)CCC(NCC(F)(F)F)CC1 22042,C1(NC(C2(O)COC2)=O)CCC2CN(C(C3CCc4ccoc4C3)=O)CC12 22043,c1(CC(N2CCC(N(C(C3CC3[N+](=O)[O-])=O)CC)CC2)=O)ccc2c(c1)CC2 22044,c1(C(N2CC(O)(CC(=O)NCc3ccc(CC)cn3)C2)=O)cccc2c1CCC2 22045,c1(NC(C2(NC(C3CC(OC)(OC)C3)=O)CC(O)C2)=O)cnc(C)c(C#N)c1 22046,N1(C(CC2(C=C)CC2)=O)CC2CC2(NC(c2cc(C(F)F)cs2)=O)C1 22047,C(=O)(C(CNC(c1cnc(C)cc1C)=O)C(C)(C)C)NC1C(CCOC)C1 22048,C(=O)(C(C)CCCC(C)C)N1C(CNC(C=C(CC)C)=O)CC(OC)C1 22049,c1(C2(C)CCCO2)cc(=NC(=O)CCN(CCN)Cc2ccco2)[nH][nH]1 22050,C1(NC(c2ccnc(C)n2)=O)CN(C(C2CCN(C)C2)=O)C2(CCCCCC2)C1 22051,c1(C(N2CC(NC(CCCC#C)=O)C(C#N)C2)=O)ccc2nn(C)cc2c1 22052,N1(C(C(CC)OC)=O)CC2(C1)CN(C(C1(CCOCCO)CCCC1)=O)C2 22053,C1(C(=O)NCC(O)CNC(=O)Cn2ccnc2)(SC)CCOCC1 22054,c1(C(N2CCCC(c3cn(C4CCOC4)nn3)C2)=O)cc2scc(Cl)c2[nH]1 22055,C1(NC(COCC)=O)CCN(C(c2cc(C)n(-c3nccs3)c2C)=O)C(C)C1 22056,c1(C(=O)OC)cnc(C(N2CCC(CC(=O)NC(C3CCOCC3)C)C2)=O)cn1 22057,N1(C(C2CCN(C)C2=O)=O)C2CCC1CN(C(=O)CC(C)(C)c1ccccc1)C2 22058,C12(C(=O)NCc3ccc(C(=O)Nc4c(C)nc(Cl)nc4)o3)CC3CC(CC(C3)C1)C2 22059,CCCCCC(C)CC(=O)NCC1CCC2(CN(C(C3CC(C)(CC)C3)=O)C2)O1 22060,CN1CCOc2cc(C(N3CC4CN(S(=O)(=O)CC5CC5)C4C3)=O)ccc21 22061,N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC(NC(=O)CCc3ccn(C)n3)C2)C1 22062,CC1OCCCC1C(=O)NCC1CCC1NC(c1cccc(OCC(F)(F)F)c1)=O 22063,C1(O)(CNC(C=NOC)=O)CCN(C(c2csnc2C)=O)C1 22064,C1(C)(C(=O)NC2CCC(OC)C2)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 22065,N1(C(C(c2ccc(C)s2)C)=O)CC(CNC(C2(C)CCOCC2)=O)CC(C)(C)C1 22066,C(C(CNC(C1C(C)C1C)=O)CO)NC(CC1(OC)CC1)=O 22067,CC1c2cc(C(N3CC(C)(NC(c4ncncc4Cl)=O)C3)=O)ccc2OC1C 22068,C(=O)(C(CCCCO)C(C)(C)C)N1CCCC(NCC(C)C)C1 22069,C1(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CC(NC(c2cscn2)=O)C12CCOCC2 22070,c1(CN2C(C)(C(=O)NCc3ccc(OCCC)cc3)CC2)cc(F)cc(Br)c1Cl 22071,C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(C2(C)CCNC(=O)C2)=O)(CO)C1 22072,N1(C(c2c(CC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22073,N1(C(c2n(CC)nc(C)c2)=O)CCC(NC(=O)C=Cc2ccc(Cl)s2)C(C)C1 22074,Cc1cn(C2CCC2)nc1C(=O)NCC1CCC1NC(=O)CC1(O)CCCC1 22075,C(C(=O)NC1CCC(NC(=O)CN2CCCC2C)CC1)(C(C)(C)C)NC(=O)OC 22076,C1(CNC(C(CCC)(C)C)=O)CC2(CCOCC2)CN1C(=O)COC(C)C 22077,S(=O)(=O)(CC(=O)NC1(C)CC(C(=O)NC2CC23CCC3)C1)NCC 22078,N1(C(C(C)NC(=O)OC)=O)CCN(C(=O)CCC2CCCO2)CC1CS(C)(=O)=O 22079,Cc1cc(N2CCCS2(=O)=O)ccc1NC(=O)C1=NOCC1 22080,N1(C(c2ccc(Oc3ccccn3)cc2)=O)CC(CO)C2(CCOCC2)C1 22081,C(=O)(C(O)C(F)(F)F)N1C(CNC(=O)C=Cc2csc(Br)c2)CCCC1 22082,c1(C(N2CCN(C(=O)CC3CCN(CCO)C3)CC2)=O)c(F)ccnc1Cl 22083,C1(C(=O)NCC(CC)NC(C2CC2F)=O)CC2(CCC2O)C1 22084,c1(C(=O)NC2C(CNC(=O)CC3CCCCCO3)CC2)cnn2cnnc2c1 22085,Cc1nc(C(=O)NCc2cccnc2CO)c(C)o1 22086,c1(CC)c(C(N2CCN(CCOCCC(C)=O)CC2)=O)nnn1CC 22087,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22088,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)CC2=NC=CCCC2)CC)CCC1 22089,C1(NC(C2C(C)(C)C2)=O)CC(NC(=O)CNC(N)=O)C12CCC2 22090,N(C1CCCc2ccoc21)C(CC(C)(C)CNC(C1CC1F)=O)=O 22091,CC(C)C(CC(=O)NC1CCC(CCCF)C1)NC(C1CCC1C(=O)OC)=O 22092,C1(OCCC)CN(C(c2coc(COC=O)c2)C(=O)NCC)CCN1C.CCC 22093,c1(CNC(c2n(CC)nnn2)c2c[nH]nc2-c2ccccc2)ccc(F)c(Cl)c1 22094,C1(NC(=O)OC(C)(C)C)CCN(C(=O)NCC2CCCC2(F)F)CC12CCC2 22095,C1(NC(CCC(=C)C)=O)CC2CC(NC(c3ccc(N)cc3F)=O)CC2C1 22096,N1(C(CC2(CSC)CC2)=O)CC2CCN(C(c3cncc(O)c3)=O)CCC2C1 22097,C1(NC(C(=O)NCCC(N)=O)=O)CC2(CCN(C(=O)CC#N)CC2)C1 22098,c1(C(C(=O)N(CCCNC(=O)Cn2cc(C#N)cn2)C)(F)F)cc(F)ccc1F 22099,c1(NC(C2(c3ccccc3)CCOC2)=O)cncn1C1CCCC1 22100,N1(CC(=O)NC2CCCC2OC(C)=O)CCN(C2(NC(CCC)=O)CC2)C1=O 22101,CC#CC1CCN(C(=O)CC2CCCC2NC(=O)C(O)C(C)(C)C)CC1 22102,C1(C(CSC)(C)O)CCN(c2ccnc(NC(c3onc(SCC)n3)C)n2)CC1 22103,N1(C(CCOC(C)=O)=O)CCC(C)(CNC(=O)Cc2ccn(C)c2)C1 22104,c1(OC)cccc(F)c1C(=O)NCC1CN(C(c2c[nH]c(C)c2)=O)CCC1C 22105,C(=O)(C(O)CC(F)(F)F)N(CCC1N(C(CC2(OCC)CC2)=O)CCCC1)C 22106,C1(CCNC(c2c(C(C)C)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22107,c1(C(N2CCC(C(N3C(C#N)CC3)=O)C2)C2CC(=O)N2)nc2ncccn2n1 22108,C1(C(N2CCC(C3CCCO3)C2)=O)(OC)CCN(C(C2CC(F)CN2C)=O)C1 22109,Cc1c(C(N2CCOC(C(=O)NCC3OC(=O)NC3C)C2)=O)cnn1C 22110,C1(NC(C(C)n2cnnn2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22111,c1(OC)ccc(CN(C(=O)CC2CCCC3CC23)CC2OCCC2C(=O)O)cc1 22112,Cc1cc(NC(=O)NC2CC2F)cc(F)c1Br 22113,Clc1cc2c(cc1Br)N(Cc1cccc3nccn13)CCS2 22114,c1(CN(C(=O)CN2Cc3ncnc(N(C)C)c3C2)C)cccc2ccccc12 22115,c1(C2CC(=O)OC(=O)C(C)NCCNC2CC)ccnc(Br)c1 22116,N1(C(c2ccn(C)c2)=O)CC(CNC(c2c(C(N)=O)nccc2)=O)C(O)C1 22117,C1(CC=C)(NC(C2CCCN2C(C)C)=O)CCCN(C(c2cc(OC)cs2)=O)C1 22118,C12(CNC(C(C3CCCC3)OCC)=O)CC1CN(C(=O)COc1ccn(C)n1)C2 22119,Nc1cc(C(=O)NCCNC(=O)C(c2ccccc2)C2CC2)cc(F)c1Cl 22120,N1(C(C2N(C(C(C)OCCN(C)C)=O)CC=C2)=O)CCN(C)C(C)C1 22121,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22122,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22123,C1(NCC2CC3CCC2O3)CN(CC(=O)NC(=O)CC2CCCC2)CCCO1 22124,CCCCC(CNC(=O)C=C1CCCC1)NC(=O)CNC(=O)NC1CC1 22125,c1(OC)cc(C(N2CCN(C(c3ccncc3NC(C)=O)=O)CC2)=O)cnc1C 22126,c1(CN(C(C2CC(NC(CCOC(C)=O)=O)C2)=O)C)n[nH]cc1C 22127,N1(C(CCc2cc(OC)no2)=O)CCC(CO)(CNC(=O)C(C)C(F)F)C1 22128,c1(-c2c(F)cc(C)cc2F)ccc2c(C(=O)NC3(C)CC3)nn(C)c2c1 22129,c1(C(=O)NC(CN(C(c2ccc(COC)o2)=O)C)COC)occ2c1CCOC2 22130,COn1cnc(C)c1C(=O)NCC12CC(CN1C(=O)CC1CCCC3(CC3)C1)C2 22131,c1(C(N(CC(C)NC(CN(CCC)C)=O)C)=O)cn2cccc(Br)c2n1 22132,C12=CN=C(SC)NC1=NC1CCN(CC1)C2=O.c1(COCC)conc1C 22133,Cc1cc(CCNC(=O)C(=O)NC2CC(CO)C2(C)C)c(C)s1 22134,CC(CN(C)C)C(=O)NCCN(CCO)CCn1ccnn1.C(=O)O 22135,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)C(n2ccnc2C)C)CC#C)CC1 22136,c1(NC(C)NC2CCCCC2)[nH]c(=NC2CCc3occc3C2)nc2c1cnn2C 22137,N1(C(Cn2ccc(C(=O)OC)n2)=O)CCc2c(cc(C#N)n2CC)C1 22138,C1(CC(=O)NCC(C)(CO)NC(=O)C=CC2CCCO2)CCCCCCC1 22139,CC(C)C(C)(CNC(=O)CSCCNC(=O)CC1CCCC2CC12)C(C)C 22140,N1(C(C2OCC(C)C2)=O)CCCC2CN(C(c3cc(N)ccn3)=O)CCC12 22141,C(=O)(C1=CC2CCCC12)NCC1(F)CCC(CNC(CCCC#C)=O)CC1 22142,C1(C(N(CCOC)CCNC(=O)C(C)(C)n2cnnn2)=O)CCCC(F)C1 22143,CC1CC(C2CN(C(C3CCC3NC(c3ccnnc3)=O)=O)C2)=NO1 22144,C1(C(=O)NC(CCCNC(Cc2n(C(C)C)cnn2)=O)C)CCC(N=[N+]=[N-])CC1 22145,N1(C(c2cc(C)sc2C)=O)CCC2CN(S(=O)(=O)CCC(F)(F)F)CCC12 22146,CC1(SCC(=O)NCc2nc[nH]n2)CCC2(CC1)CC2.C12CN(CC13CC3)C2=O 22147,c1(OC)nc(C(N2CCCCC(NC(=O)CN3CCCCC3C)C2)=O)ncc1F 22148,c1(CCS(=O)(=O)NC(C)CCc2ccccc2F)c[nH]c2cc(Cl)ccc12 22149,N1(C(CCCC(C)NC(c2ccc(C)c(C)n2)=O)=O)CC2(C)CC1CCO2 22150,Cc1cnccc1C(C)C(N1CC(NC(=O)Cc2cncnc2)CC1C)=O 22151,CC1CCN(C(c2cc(C#N)c[nH]2)=O)C(C(N2CCC(F)(C(N)=O)C2)=O)C1 22152,c1(C(C(=O)NCCCOC)N(C)Cc2sccc2OC)ccc2c(c1)CCC2 22153,c1(C(=O)NCCC(C=C)C)n[nH]c2c1CN(C(c1cnc(Cl)s1)=O)C2 22154,N1(C(c2cnco2)=O)CCN(C(c2ccc(F)c(Cl)c2F)=O)C2COCC12 22155,CC1(C)CC(O)CCN(C(C2C3CC(O)C(C3)N2C(=O)CSC(F)(F)F)=O)C1 22156,c1(C(C(=O)NCCC(C)NC(C23CC(C2)C3)=O)OC(C)C)ccccc1 22157,c1(NC(C)=O)ccc(C(=O)NC2COCC2NC(=O)CCc2nncs2)cc1 22158,N1(C(C(CC2CCC2)OC)=O)CCC(NC(=O)C2=C(Cl)CCC2)C1(C)C 22159,N1(C(C(C)N(C(=O)CC2OCCO2)C2CC2)=O)CC(CO)C(O)C1 22160,C12CN(CCC13CCC3)C2=O.c1(N(CCCOC)C)nccc(OC)n1 22161,n1(CC)c(C(N2CC(C(=O)NCCC3CC4CCC3C4)C2)=O)cc2ccccc12 22162,Cc1c(CN2CC3(C2)CN(c2cc(C#N)ncn2)C3)cccc1O 22163,c1(C(N2CCCC(NC(c3c(C)ccnc3)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1C 22164,c1(OCC(c2n(CCC)nnn2)NC2CC(C(N)=O)C2)ccc(C)cc1SC 22165,N1(C(C2CC(CC)C2)=O)CCC=C(C(=O)NC2CC2(C)C(F)F)C1 22166,C1(C(=O)NCC(c2ccccc2)N(C)C(c2cscc2F)=O)(OC)CC(C)(C)C1 22167,c1(C(=O)NCCCn2nc(NC(N(C)C)=O)c(C#N)c2)cccc2c1C(=O)NC2 22168,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2cccnc2S)=O)C1 22169,c1(CC(=O)NCCC2N(C(C3COC(C)(C)O3)=O)CCCC2)ccc(Cl)cc1F 22170,Cc1ccc(C)c(C(=O)NCC(=O)NCC(=O)NC2CCCCC2)n1 22171,CC(C(C)CO)NC(=O)CCN(C(=O)CCc1cn[nH]c1)C1CC1 22172,Cc1cc(C(=O)NC(c2cn(C)nn2)C(=O)NC(C2(CO)CC2)C)ns1 22173,c1(CCN(S(=O)(=O)CC2COCC(C)(C)O2)C)nc2c([nH]1)CCCC2 22174,Cc1cc(NC(=O)C(C2CCOCC2)O)ccc1NC(=O)C(N1CCCC1)C1CC1 22175,C1(C(=O)N(CCNC(C(C)Cn2cccn2)=O)Cc2ccccc2)NC(=O)OC1C 22176,N1(C(c2ccn(COC)n2)=O)CC(NC(C2CCCOC2C)=O)C(O)C1 22177,C=CCC(CNC(=O)C(CC1CC1)OCC)C(=O)NC1(CO)CC2CCCC12 22178,N1(Cc2c(-c3ncn(C)c3)n[nH]c2)CCC2(CC1)CC(N1CCC(F)(F)C(O)C1)C2 22179,c1(C(C)=O)cc(C(=O)NCC(C)N(C(=O)COCc2scnc2C)C)c(C)o1 22180,C(C(F)(F)CNC(=O)CCCN(C(=O)C(O)Cc1ccco1)C)OC 22181,c1(C(=O)NC(C)CN(C(=O)C(=Cc2c[nH]cn2)F)C)cc2scc(Cl)c2[nH]1 22182,CC(C)C(C)C(CNC(N)=O)NC(c1cccc(-c2cscn2)c1)=O 22183,OC1(F)CCN(C(=NCCc2cncc(Br)c2)NCCF)CC1 22184,C1(OC)CN(C(C2(NC(=O)CC3CCOC3=O)CCC2)=O)CC1CC1CC1 22185,c1(OC)cc(C)c(CN2CC(O)(CNC(c3ccsc3Cl)=O)C2)cc1OC 22186,Cc1nn(C)c(C)c1CC(=O)NCCCCC(=O)N(C)CC1CCCC1O 22187,Cc1cc(C(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)CN(C)C)n[nH]1 22188,c1(N2CC(NC(CCCCC(C)C)=O)(CO)C2)nc2cc(Cl)cc(Cl)c2o1 22189,CC(C)(CO)C(=O)N1CCC(CCC(N2CCC(O)C2)=O)C1 22190,N1(C(C)C2CC2)CCN(c2nc(C(F)(F)F)cs2)CC1 22191,CC1CN(C(c2ccc(OCCF)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22192,C1(NC(C(CCCOCC)C)=O)CN(C(c2cc3ccccc3[nH]2)=O)CC(C)(C)C1 22193,c1(OC)cccc(NC(=O)C(=O)NC2CC(N(C)C)CCC2=O)c1F 22194,n1(C(=O)NCCOCCn2cc(-c3cccc(Cl)c3)nn2)cccnc1=O 22195,C12(C(=O)NCCc3cc(C)no3)CCCC1CCN2C(c1n[nH]c(=N)[nH]1)=O 22196,c1(C(=O)NCC2CC(NC(c3nnn(C)n3)=O)C2)ccc(O)c(Cl)n1 22197,C(=O)(C(C(C)C)C(C)C)N(C)CC1(C)C(NC(C(C(CC)O)C)=O)CCC1 22198,N1(C(C=CCOC)=O)CC2CC(NC(=O)C(c3ccccc3C(F)(F)F)O)C2C1 22199,c1(C(=O)NCC(C2CC2)NC(C(OC)OC)=O)ccc2cccnn12 22200,C1(C(=O)NC2CCN(C(=O)CCc3ccc[nH]3)C2)(OC)CCS(=O)(=O)C1 22201,N1(C(Cn2cc(CCCC(C)O)nn2)=O)CC(OCc2nccs2)CC2(CC2)C1 22202,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22203,Cc1ncnc(N2CCC(NC(=O)CCCCOC(C)C)C(C)C2)c1Br 22204,C(c1cncn1C)=CC(=O)NC1CCC(CCNC(c2n(COC)ncc2)=O)C1 22205,CC(CC(=O)N(CC(=O)NOCC(F)F)C1CC1)CC(C)(C)C 22206,c1(NC(CC)CO)ccc(S(=O)(=O)NCc2ccsc2Cl)cc1Br 22207,Cc1nn(C)c(C)c1CC(=O)NCCC(O)CNC(=O)C(=O)C(C)(C)C 22208,C1(NC(c2ncn(CC)c2)=O)CCCC(NC(=O)Cn2nnc(C3CC3)n2)CC1 22209,N1(C(CCC=C)=O)CCC2C(COC2CC(=O)NCc2ccsc2I)C1 22210,C1(O)(CNC(c2c(C(C)NC(C3CC3F)=O)nc[nH]2)=O)CCN(C(=O)OC)CC1 22211,CC1OCCC1(F)C(=O)NCC1(C(N)=O)CN(C(=O)CCC2CC3CCC2C3)C1 22212,c1(CC)nnc(NC(C)CNC(c2ccc3nonc3c2)=O)c(C#N)c1CC 22213,N1(C(C2C(C)C2)=O)CC2C(N(C(=O)CCSc3ccccn3)C)C2C1 22214,C=CC(C)(C)CC(=O)NC1COCCN(C(C2(c3ccccn3)CC2)=O)C1 22215,Cc1c(C(N2CC3CC2C3C(=O)NCCC2(O)CCC2)=O)cccc1F 22216,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(NC(c2ccnc(CO)c2)=O)C2CC2C1 22217,C=CCC(F)(F)C(=O)NC1(CNC(=O)CCCF)CC1 22218,C(=O)(CS(=O)(=O)NC)NCCN(C(=O)C(C1CCOC1)OC)CC 22219,N1(C(C(c2cn(C)nn2)NC(C2CC(C#C)(O)C2)=O)=O)CCC(O)C(F)(F)C1 22220,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22221,C12(CNC(COCCCCC)=O)CCC(C1)N(C(=O)C=Cc1ccsc1)C2 22222,n1(CCC)c(C)cc(C=CC(=O)NCC(O)CNC(=O)COC(F)(F)F)c1C 22223,N12CCC(C(O)C1)CN(C1C(C)COC1)CC2.C(c1ccccc1)=CCO 22224,c1(C(=O)NC2CC(NC(=O)CNC(c3ccsc3)=O)C2)ccc2c[nH]nc2c1 22225,N1(Cn2c(C3(OC)CC(OCC)C3)nnn2)CC2C(c3ccccc3)(C1)CS2(=O)=O 22226,CCCCCCC(F)C(=O)NCC1(NC(C2CCC2(C)C)=O)CCC1 22227,N1(C(CCCN(C)C)=O)CCC2(CC2C(=O)N(C)Cc2cn[nH]c2)C1 22228,c1(-n2cc(CSCCNC(Cn3c(C)ncc3)=O)nn2)ccc2c(c1)OCCO2 22229,C1(NC(CCC=C)=O)C=CCN(C(=O)CC(Cl)Cl)C1 22230,C1(=O)C(C(C)(C)O)CN1.c1(-n2cc(SCC)nn2)cccnc1C#N 22231,c1(C(=O)NCC2CN(C(C3CCCCC3O)=O)C2)nc2ncc(CCO)cn2n1 22232,N#Cc1cc(F)c(CN2CCSCC2C(=O)NCc2ccc(F)c(Cl)c2)c(Cl)c1 22233,Cc1ccc(SCC(N2CCCC(O)(CNC(=O)C(F)(F)CO)C2)=O)cc1C 22234,N1(C(CN(c2ccccc2)CC)=O)CCN(C(=O)C(C)(F)CCC)CC12CCC2 22235,C(=O)(CCC(CC)NC(=O)C1CC1)NC1C(C#C)CCC1 22236,n1(CC)cc(CC(=O)NC(C(=O)NCCC2CCOC2)C2CCCC2)cn1 22237,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)COC2CC=CC2)CC1O 22238,c1(C(=O)NC2CCC(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22239,C(C)(CNC(=O)Cc1ccc(O)c(C)c1)(CC(C)C)NC(C(=CC1CCCC1)C)=O 22240,n1(CC(=O)NC2C(NC(C(CC)OC)=O)CC2)nc(-c2cccs2)oc1=O 22241,c1(-n2cc(C(C)(C)N(C)C)nn2)ccc(C(=O)NCCC(O)CCO)cc1 22242,c1(C(=O)NC2CC(C(=O)NC3(CC)CCNC3=O)OCC2)ccc2n[nH]cc2c1 22243,N1(C(C(CC#C)(C)NC(=O)CCC#CC)=O)CC2(CNC(=O)C2)C1 22244,N1(C(CCC)=O)CCC(O)(CN(C(=O)COC(C)CC(C)C)CC)CC1 22245,C1(C(=O)NC(CC)C(C)(F)F)CN(C(=O)C(C)(C)CO)CC1C1CC1 22246,c1(C(=O)NCCN(C(=O)CC2COC3CC2C3)C2CC2)cc([N+](=O)[O-])ccc1Cl 22247,C(C(C)(C)C(=O)N1CCOC(C2CC2)C1)NC(C1C(C)(C(C)C)C1)=O 22248,CC1(C)CN(C(c2ccc[nH]2)=O)CC(CNC(C23CC(CN2C2CC2)C3)=O)O1 22249,Cc1ncc(Cl)c(C(N2CC3C(CN(C(=O)C(C)(C)O)C)C3C2)=O)n1 22250,N1(C(C2(F)CCN(C(C3(CCC=C)CC3)=O)CC2)=O)CC(C)N(C)CC1C 22251,c1(C(C(C)C)N(C(=O)N)CC)nnc2n1CCC2.c1(O)ccc(C2CCCC2)cn1 22252,c1(-c2cc(C)c(F)cc2)cc(S(=O)(=O)N2CCSCC2CCO)c(C)cc1C 22253,C(=O)(C1=CC2CCCC12)NC(CNC(c1n[nH]c(CC)c1Br)=O)(CC)CC 22254,C1(CNC(C(CC)(C)C)=O)C(O)C(O)CN1C(=O)CSc1nncn1C1CC1 22255,c1(CC)nn(C)c(C(=O)NC2C3CC2N(C(=O)CCS(=O)(=O)N(C)C)C3)c1Cl 22256,c1(CCC(=O)NC2C3CN(C(C4CCC4(F)F)=O)CC23)cccc2cnccc12 22257,C1(C2CC2)(C(=O)NC2C(C=C)COC2)CN(C(C2C3CN(C)CC23)=O)C1 22258,C1(NCc2c(C(F)(F)F)cccc2)CCc2nnc(CCn3cncn3)n2C1 22259,N1(C(CC(=O)OC)=O)CCC2CCCC12C(=O)NCC1(C(C)(F)F)CC1 22260,Cc1nsc(C)c1C(N1CCCC(CN(C)C(C2CCCN2N=O)=O)C1)=O 22261,C1(CCCNC(=O)CSc2cccnc2)CCCCN1C(c1cccnc1)=O 22262,c1(CC(N2CCC(N(C(CC(CC)OC)=O)C)C2)=O)c(F)cccc1Cl 22263,C1(COC)CCCN(C(=O)CN2CCNC2=O)C1.C1(=O)C#CCN1 22264,CC1CN(C(C2(c3ccccc3Br)CCC2)=O)CCN1C(C1C=CCCC1)=O 22265,C1(C)(CCC(=O)NC(C2(O)CCC2)C)CN(C(c2nocc2C2CC2)=O)C1 22266,C(CNC(=O)Cc1nccn1C)(CC(F)(F)F)NC(C1N(CC)CCOC1)=O 22267,N1(C(C(C)NC=O)=O)CCOC(C(=O)NCC2CC2(C)C)CC1 22268,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22269,c1(NC(=O)CNNC(=O)c2cccnc2OC(F)F)ncnc2[nH]cc(Cl)c12 22270,Cc1ccc2c(C(N3CC(CNC(c4ccc5nc[nH]c5c4)=O)C3)=O)n[nH]c2c1 22271,C1(COC)(CNC(=O)CC#N)CCN(C(=O)Cc2ncccc2C)C1 22272,c1(C(=O)NCC)cnc2n1CCN(C(=O)C(CC(C)C)N(C)C)C2 22273,S(=O)(=O)(c1ccc(-c2nc(C3CC3)no2)s1)N(c1ccc(Br)c(OCF)c1)C 22274,N1(C(CCC=C)=O)CCCC(NC(=O)CCc2ccc(C(C)C)cc2)C1 22275,C(=O)(C1=CNC2=NCCCC2=C1)NC1(CO)CCCN(C(C(C(=O)NC)(C)C)=O)C1 22276,c1(OCOC)cccc(NCCNC(=O)C(C(C)C)n2cnnc2)c1 22277,Cn1cc(C(=O)NCCCNC(C2CC2C2CC2)=O)nc1-c1ccccn1 22278,N1CCCC1C1(C(N2CCC(OCC=C(C)C)C2)=O)CC1.CC1(C)CC1CC(=O)OC 22279,c1(C(=O)NCC2(C(C)NC(=O)CCC3CCCO3)CC2)ccc2cccnc2n1 22280,C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(CC(=O)NC2(C(=O)NC)CC2)C1 22281,C1(NC(CC2CN(C)C2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 22282,c1(CCC)nc(=NCC(O)CNC(=O)Cc2cc3ccccc3[nH]2)s[nH]1 22283,CC(C(=O)NCC1CC1NC(c1cnc(N)c(-c2ccccc2)c1)=O)C(C)(F)F 22284,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2(CCC2NC(C2CCCOC2C)=O)C1 22285,Cc1ccc(C(C)C(=O)N(CC(C)NC(C2OCCC2C(C)C)=O)CCO)cc1 22286,C(=O)(C(CC(F)F)C1CCC1)NC1(CCNC(c2n(CCC)ncc2)=O)CCC1 22287,CC1=C(C(=O)NC2COCC2NC(C2NC(=O)OC2C)=O)C(=O)OC1(C)C 22288,CC1CC(NC(C2COCCN2CC(F)(F)F)=O)CCN1C(C12CC(F)(C1)C2)=O 22289,C1(C(=O)N(CCCO)CCO)CN(C(=O)C=CC2CCOC2)CC12CC2 22290,c1(CC)c(C(=O)NC(CN(C(=O)CC(C)C(F)F)C)CC)cccc1C 22291,c1(C(=O)NC2CC3CC(NC(CCCOC)=O)CC32)ccc2c(c1)ncn2C 22292,CC1OC2(C(=O)NCC3CN(C(=O)CCNC(N)=O)CC(C)(C)O3)CCC1CC2 22293,c1(CC)nnc(C)cc1NC(C1(CNC(=O)CS(=O)(=O)CC)CCCO1)=O 22294,N1(CC)CCC(NC(C2CCOCC2NC(C2CC2Cl)=O)=O)C1=O 22295,C12(NC(CC3(OC)CC3)=O)CCCC(NC(=O)CCc3nccn3C)(C1)C2 22296,C(C)(C(O)C(=O)NCC(C)(C)NC(=O)CNS(=O)(=O)C1CC1)OC 22297,C(=O)(C#CC(C)(C)C)NCCNC(CC(C)c1ccncc1)=O 22298,N1(C(=O)CSc2nc[nH]n2)CCC2(NC(=O)CC3CCSCC3)CCCC12 22299,N1(C(CC2(C)CC2F)=O)CCC(C2(O)CN(C(C3(n4cnnn4)CC3)=O)C2)CC1 22300,c1(CC)cc(F)ccc1CC(=O)NCC1CCN1C(=O)Cc1ncoc1C 22301,C1(NC(=O)NC2CCOC2c2cccnc2)CCC2(CCCN2)CC1 22302,c1(-c2ccc(NC3CCN(c4c(C)c(Cl)ncn4)C3)s2)nc2cccnc2s1 22303,C1(F)(C(NOC(C(=O)OCc2ncc(CC)s2)C)=O)CCCCC1 22304,c1(SCC)cn(C)nc1C(=O)NCCCNC(c1c(SC)scc1)=O 22305,c1(OC)cccc(CC(C)(C)NCc2c[nH]nc2C(F)(F)F)c1 22306,n1(CC)nc(C(N2CCN(C(C3CCS3(=O)=O)=O)CC2)=O)cc1C 22307,N1(C(CC=C=C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22308,C1(CCC(=O)NCC)C2CCC(C2)N1CC1(C)CC=CCC1 22309,N1(CCC)CCCCC1C(=O)NCC(CNC(c1cn(C2COC2)nn1)=O)CO 22310,Cc1[nH]ccc1C(=O)NCc1cn(CC(N2CCC2CN(C)C)=O)nn1 22311,c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)(C)CC)cc(Cl)c(C)cc1OC 22312,C1(OC)CCN(C(=O)CNC(=O)NC)C(C)C1.c12n[nH]cc1NC(=O)C2 22313,c1(CC)nnc(N(CCNC(C)=O)C(C2CCCNS2(=O)=O)=O)nc1CC 22314,Cc1cc(C)[nH]c(=NCC2(NC(c3cccn4c(O)nnc34)=O)CC2)n1 22315,C1(CC(=O)NC(C(C)(C)NC(c2cncc(COC)c2)=O)C)NC(=O)CNC1=O 22316,CC(N=c1cc(C(=O)Nc2ccc(Cl)c(Cl)c2)nc(Cl)[nH]1)C1CCCOC1 22317,CCCCC(O)CC(=O)NC1(c2nnnn2CC2CCCO2)CC(OC)C1OC 22318,n1(CC)cc(Cl)cc1C(=O)NC1(CNC(C23COCC(C2)C3)=O)CCCC1 22319,c1(CNC(C2C3CN(C(C4CCOC4)=O)CC23)=O)cc(Br)cc2cc[nH]c12 22320,c1(CCC(=O)OCc2ccccc2)cc(Cl)cs1.N1(CC2(C(=O)O)CC2)CCNC1=O 22321,CCS(=O)(=O)c1cccnc1C(=O)NCC(C)(N)Cc1ccccc1 22322,C(C)(C(CC(=O)NOCCF)C1CCC1)OCC.C1(=O)CCCN1 22323,N1(C(C)C)CCC(CC(=O)NC2CCC(NC(=O)COCCF)CC2)CC1 22324,Cc1ccc2[nH]c(C(=O)NC(C)CCNC(=O)C(C)CS(C)=O)cc2c1 22325,N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2=CCCCC2)C2(CCOCC2)C1 22326,c1(OC)ccc(NC(C(CCC)OC)c2nnnn2CC2CCCO2)cc1SC 22327,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22328,c1(C(=O)NCCCNC(c2c(C)nn(C3CC3)c2)=O)cnn2c(N)ccnc12 22329,C(=O)(C(=O)C(C)(C)C)N1CC(OC(C(C)C2CC2c2cccc(I)c2)=O)C1 22330,N1(C(C=C(C)CN2CCOCC2)=O)CCCC(CCC(=O)NC23CC(CO)(OC2)C3)C1 22331,c1(CC(C(N2CC(OC)(CNC(=O)C(C)CO)C2)=O)C)ccc(C#N)cc1 22332,C(C(CC(C)C)C(=O)NCc1ncoc1CCNC(c1cnc(Cl)n1C)=O)OC 22333,Cc1cc(N2CCC(C(C)NC(C3CCCC(O)C3)=O)C2)c(Br)cc1[N+](=O)[O-] 22334,c1(C(=O)NC2CCC(NC(=O)C3=CCSC3)C2)c(Cl)ccc(Br)c1F 22335,C12(NC(=O)C(c3ccccc3)F)CCCC(CN(C(=O)C3=COCC3)C1)C2 22336,Cc1cnn(C)c1C(=O)NCC1CN(C(=O)CCCF)C1 22337,C1(CCC#C)CCCN(C(=O)CCCNC(C2(CSCC)CC2)=O)C1 22338,CC1(C)CC(NC(=O)C(C2CCOCC2)F)CN(C(C2CCC2C(N)=O)=O)C1 22339,c1(OC)cc(CNCC(C#N)(CC)c2nnnn2C2CCCC2)cc(F)c1 22340,c1cccc2c1OCCO2.N1(c2c(C)c(Cl)ncn2)CCn2c(C)cnc2C1 22341,CC(C)(O)C#CC(=O)NCC(N1CC2(CCC1CO)CC2)=O 22342,Cc1cc2nc(C(=O)NCC3CCN3C(=O)C3=C(Cl)CCOC3)cn2cc1C 22343,N1(C(C(C2CCN(C(=O)C(c3cccn3C)=O)C2)C)=O)Cc2ccccc2C1 22344,C1(NC(c2ccon2)=O)CCCCC1N1CCN(C(=O)CC2CCCCC2)CC1 22345,N1(C(C2CC3(CC(NC(C(CC(C)(C)C)OC)=O)C3)C2)=O)CCC2(CCC(O)C2)C1 22346,C1(NC(C=CC(C)(C)C)=O)C2CC(CN(C(=O)Cc3ccc(F)cc3)C2)C1CO 22347,N1(C(c2ccc(OC)nc2)=O)CCCC(NC(c2cnnc(C3CC3)c2)=O)C1C 22348,C(=O)(C(F)C1=CCCCC1)N1CC(C)C(NC(c2c(Br)cnn2C)=O)C1 22349,C(=O)(C(C)CC(C)(F)F)NC(CCNC(C(c1ccc(OC)cc1)C)=O)C(C)C 22350,C(CCCC(C)C)NC(C1(C)CN(C(c2c(C)scn2)=O)C1)=O 22351,C1(n2cnnn2)(C(=O)NCCC2(NC(CC3N(C)CCC3)=O)CC2)CCCCC1 22352,c1(SCNC(Cn2cc(CC(C)(C)O)nn2)=O)nc2ccccc2s1 22353,N1(C(C2C(C)C2)=O)CC(NC(c2nccn3nccc23)=O)CC12CCCC2 22354,C1(CN(C)C)(NC(=O)CC(O)C2CCCC2)CN(C(C2(C(N)=O)CC2)=O)C1 22355,c1(C(=O)NCCC(C(C)C)NC(=O)C(=O)N(C)C)cc2occ(Br)c2[nH]1 22356,c12cccc(c1OC)S2.c1(CC)nnc(N(C)CC=C(C)C)n1CC1CCCO1 22357,N=c1[nH]cncc1C(=O)NCC1(c2cn(CC3CCC(=O)O3)nn2)CCCC1 22358,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22359,c1(N(C)CC2CCC3(COC3)OC2)ncnc2c1ncn2CCCn1nccn1 22360,CCC(CC)(CC)C(=O)NC(C)CN(C)C(c1ccc(O)c(F)c1)=O 22361,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22362,C12(C(N3CCC(C)(NC(C(c4cccnc4)C)=O)C3)=O)CCOC1CC(=O)NC2 22363,C(=O)(C(COC)OC)NC(C(=O)NC1(CC=C)CCC1)C1(O)CCC1 22364,C12=NC(=NC3CCCN1CC3)NC1=C(CSC1)N(CCC)CCCN2CC 22365,c1(C(C)C)ncncc1C(N1CC=CC(NC(=O)CC(C)NC(N)=O)C1)=O 22366,N1(C(C(COC(C)=O)C)=O)CCOCC(NC(c2cc(Br)nn2C)=O)C1 22367,c1(C(=O)NCC(C)NC(=O)CCC2CCOC2)cncc(F)n1 22368,C1(N(C(CC2C(C)C2)=O)C)CCCCN(C(=O)C(C)(C)C2CCCO2)C1 22369,C12CCCN(C1)C2=O.n1(CCC)cc(C(=O)NC2(C)CN(C(=O)CC)C2)nn1 22370,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC)[nH]2)=O)ccc(=O)n(C(C)C)c1 22371,c1(CCC(=O)NCC2(COC)CC2(F)F)cccc(F)c1Br 22372,C1(NC(C(=CC2CCCC2)C)=O)CN(c2nnc(C(F)F)o2)CCC12CCC2 22373,N1(C(C2(COC)CC2(F)F)=O)CCS(=O)(=O)C(CNC(=O)C=CC(=O)N(C)C)C1 22374,C(=O)(CC(C)(C)C(=O)N1CC2C(CNC(C3CCS(=O)CC3)=O)C2C1)OCC 22375,O(NC(=O)C(O)Cn1cncn1)C(C(=O)NCCSC)CC 22376,c1(NCC)ncc(C(=O)OC)cc1Cl.C1(=O)C(C)(OC)C(=O)N2CCC(C2)N1C 22377,c1(CC(=O)NCC23CC(NC(C(COC)N(C)C)=O)(C2)C3)c(O)ncnc1O 22378,c1(C(=O)NC2CN(C(CNC(=O)OCC)=O)CC(F)C2)csc2ccc(F)cc12 22379,CCCC(C)CC(=O)NC(C)C(C)NC(c1onc(OC)c1Br)=O 22380,c1(OCC)cccnc1C(=O)N(CCC(C)NC(=O)C=Cc1ccc[nH]1)C 22381,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22382,c1(C(N(C)CC2CCCC2NC(=O)Cn2cc(CO)nn2)=O)nsnc1O 22383,N1(C(c2cnc(OCC)nc2)=O)CC2(NC(=O)CC3CSCCS3)CCC1C2 22384,C1CN=C(NC2CCCC2)N2CC3C(C3C2)C(=O)N1CC(C)(C)C.C1(OC)CC1 22385,c1(C(=O)NCC(CO)NC(C(C2CCCC2)OC)=O)c[nH]c(=N)nc1C 22386,c1(C(N2CCN(C(C3CC(COCC)C(O)C3)=O)CC2)=O)cc2ccccn2c1 22387,CC(C)CC(O)C(=O)N(C1(C(=O)NC2CCCCCC2C)CC1)C 22388,CCCCC(C)(C)CNC(C1(C)CCCN1C(=O)CC(C)N(C)C)=O 22389,N=c1[nH]c2cccc(C(=O)NCC(O)CNC(c3csc4ccccc34)=O)c2o1 22390,C=C(Cl)CN=c1ccc(S(=O)(=O)NCCC(c2ccccc2Cl)O)c[nH]1 22391,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22392,c1(-c2cn(C(C)C(=O)NC3CCCC3n3cccn3)nn2)ccc(F)nc1F 22393,C(C)(C1COc2ccccc21)NC(c1c(C)ccc(F)n1)=O 22394,C1(NC(c2cncc(SC)c2)=O)(CNC(c2sccc2F)=O)CC2CCC1C2 22395,c1(-n2ncc(C)c2)cncc(N(C(c2cscc2SC)=O)CC2CNCCN2C)c1 22396,C1(C(=O)NCc2n(CC)nnn2)N(C(=O)C(C)n2cccn2)CCCC1(C)C 22397,c1(C(=O)OCCn2cc(C(C)NC)nn2)ccc2nc(Cl)nn2c1 22398,c1(C(=O)NCC(C)(C2CC2)NC(C(CC)COC)=O)ncnc2c1CCC2 22399,c1(-n2c(CCC#C)nc(C(C)CCC)n2)ccc(S(=O)(=O)N(C)CCC)cc1 22400,N1(C(CC(C)=C(C)C)=O)CCN(C2CCN(C(C3(C4CC4)CC3)=O)CC2)CC1 22401,N1(C(c2c(C)[nH]nc2C(C)C)=O)CCC(C2CC2)(CNC(C23CCN(CC2)C3)=O)C1 22402,C1(CCNC(C=COCC)=O)CC(F)(F)CN1C(=O)CCCn1ccnn1 22403,N1(C(c2cnc(-c3cccs3)nc2)=O)CC2COC(C1)C2O 22404,N1(C(C2CCC(C(=O)NC(CC#C)C(N)=O)C2)=O)CCCSCC1C 22405,c1(C(=O)NC(CN(C(=O)CC2CCCC2)CC)C)cccc(C(=O)NC)c1F 22406,c1(OCC)nc(N2CC(C)(NC(=O)Cc3sc(SCC(C)C)nc3C)C2)ncc1C 22407,C1(C)(C(=O)NC2C(CC(=O)OC)CCC2)CCCN(C(C2CCCC2(C)C)=O)C1 22408,N1(C(CC(C)(C)C)=O)CCC2CN(C(c3cc(F)cc(F)c3O)=O)CCC2C1 22409,C1(NC(=O)Nc2cnc(I)cn2)CCN(Cc2ccc(OC(F)F)cc2)CC1O 22410,C(C(C)(CCO)NC(=O)C(F)CC1CN(C(=O)Cn2ccnn2)C1)OC 22411,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22412,Cc1cc(C)n(CCC(=O)N(C)CC2CCN(C(=O)C(C)N(C)C)CC2)n1 22413,C(=O)(CS(=O)(=O)CC1CCCO1)NCCCN(C)C(C1CSCC(=O)N1)=O 22414,c1(C(N2CC(CNC(=O)Cc3ccoc3)C(O)C2)=O)cncc2sccc12 22415,C(CCC)(C(=O)NC1(CCOC)CCN(C(=O)Cc2cccc(C)c2)C1)=CCC 22416,c1(CC(=O)NCC2CCCN(C(CN(C(COC)=O)C)=O)C2)ccc(C)c(Cl)c1 22417,Cc1cc(C)n(CC(=O)NCCN(C)C(c2cccc(CS(C)(=O)=O)c2)=O)n1 22418,C12CN(CCC1O)C2=O.c1(NC(=O)NCC(=O)OCC)ccc(CC)s1 22419,c1(C(=O)NCC(CC=C)NC(c2coc(Br)n2)=O)ccc(OC2CCC2)cc1 22420,O=C(N=c1ccn(C2CC2)[nH]1)C1CCN(C(c2cc(Cl)c(Cl)cc2Cl)=O)C1 22421,N1(C(C2C(=C)CC2)=O)CCC(C)(CCNC(=O)CCc2ccc[nH]2)C1 22422,N1(C(C2(CCNC(c3ccn(CC)c3C)=O)CCC2)=O)CC(S(N)(=O)=O)C1 22423,CC1(C(=O)NC2CCC(CNC(=O)C(C3CCCCC3)O)CC2)COCCO1 22424,N1(C(CSCC)=O)CC2CCCC2(CNC(=O)C2=NOC(c3ccccc3)C2)C1 22425,c1(NC(=O)NC(c2cccc(C)c2)c2ccccn2)cc(F)c(I)c(F)c1 22426,N1(C(c2c(C)nsc2)=O)CC(NC(c2ncc(Cl)c(N)c2Cl)=O)CC2(CCC2)C1 22427,C(CN=c1[nH]c2c(c(=NCc3nc4ccccc4o3)[nH]1)CSC2)=CCCC 22428,N1(C(C2N(CC)CCOC2)=O)CCCC(C2CN(C(C3(C#N)CCC3)=O)C2)C1 22429,C1(N(C)C(c2cc(Cl)c[nH]2)=O)CN(C(C2COC(=O)N2)=O)CCC1O 22430,C1(OCC(N2CC(C(C(=O)N(C3CCCC3F)C)O)C2)=O)CCCCC1 22431,CC(C)CCCC(C)CCOC(C(c1ccc(Cl)cc1)C(=O)OC(C)(C)C)=O 22432,c1(C(N2CC(C(C)NC(C3CCC(O)C3)=O)C2)=O)cnc2ncccn12 22433,C(=O)(C(C)(O)COc1ccccc1)NCCN(C(C1CC(SC)C1)=O)C 22434,c1(C(C(=O)NCC(=C)C)N(C2CCC2C)C)cc2c(cc1OC)CCC2 22435,C1(C(=O)NCC(O)C2(Cl)CC2)CCC(NC(=O)C(C2(O)CCCC2)F)C1 22436,Cc1cc(NC(=O)NC(c2ccccc2)Cc2cnccn2)c(C)c(C)c1 22437,N1(C(C2(C)CCCO2)=O)CCOC2(CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)C1 22438,C1(C(=O)NC(C2CCCCC2)CO)(NC(C(c2ccnn2C)C)=O)CC(O)C1 22439,O=C(CC(F)(F)F)N1CCC(C2OCCC2NC(=O)CC2(O)CCOCC2)CC1 22440,c1(C(=O)OC)c(C)[nH]c(C(=O)NCC(C(C)(C)C)NC(=O)CC#N)c1C 22441,c1(C(N(CC(C)CNC(C23CCCC(CO2)C3)=O)C)=O)cc(O)c(O)c(O)c1 22442,C1(C(N(C(CCNC(c2nc(C)oc2)=O)C)C)=O)CCC(C)CC1 22443,c1(C(=O)NC2(CCNC(c3csc(-c4cccs4)n3)=O)CC2)ncc[nH]c1=O 22444,C1(C(=O)NC(c2ccc(F)cc2)C2CCN(C3CCC3)C2)CC2CC1CC2O 22445,c1(C(N(C)Cc2nccn2C)=O)ccc(=O)n(CCc2cn[nH]c2)c1 22446,C=CCC(CNC(=O)CC1(C#N)CC1)C(=O)NC(c1nnnn1C)C 22447,C(=O)(C1=CC2(CCOCC2)C1)NCCC(C)CNC(=O)C(CO)C(C)(C)C 22448,C(C(C)(C(=O)NC(C1CCCC1O)C)NC(C1(F)CC=CCC1)=O)OC 22449,N1(C(C(C(C)C)CNC(=O)CC2COCC(C)O2)=O)CCC(C)C(F)(F)C1 22450,N1(S(=O)(=O)c2cnccc2N2C3CCCC2CC3)Cc2ccccc2CC1CO 22451,N1(C(Cc2c(OC)cc(O)cc2)=O)C2CCC1CN(C(=O)CC#N)C2 22452,C1(NC(COC(C)=O)=O)CC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C12CCC2 22453,CN1CCCC1(C)C(=O)NCc1ccc(C(=O)NC2COCCOC2)cc1 22454,N1(C(c2ncc(NCC)nc2)=O)CC(C)C(C)(CNC(=O)CNC=O)C1 22455,Cc1ccc(C(N2CCC(C(=O)NCC(Cl)Cl)CC2CO)=O)c(C2CC2)n1 22456,Cc1cc(C(N2CCCCC2CNC(=O)CNC(=O)C(C)C)=O)cc(C(F)F)c1 22457,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C(=Cc1cscn1)F 22458,C(=O)(C1=C(C)S(=O)(=O)CC1)N(CCC1CCN(C(=O)OCC(=O)N)CC1)CC 22459,C1(C)(C(=O)NC2CCN(N(c3nc(C4CC4)cs3)C(C)=O)C2)CCCCCCC1 22460,c1(CC)ccc(O)c(OC)c1.C12(C(=O)NCC3C4CN(C4)CC(=O)N3)CCC(CC1)O2 22461,N1(C(Cn2nc(C)c(Br)c2)=O)CCOC2CN(C(=O)Cn3cnnc3)CC12 22462,c1(NC(C2N(C(c3c(C)nn[nH]3)=O)CC(O)C2)=O)ncc(Br)cc1F 22463,Cc1cc(C(N2CCN(C)CC2CNC(c2c(Cl)nsc2Cl)=O)=O)cc(=O)n1C 22464,c1(C(=O)NC2CC(NC(CCCOC)=O)C2)cc(C)c(N)cc1Cl 22465,N1(C(c2nc(C(C)OC)sc2)=O)CCN(C(c2cc(C)cc(C)c2)=O)CC1CO 22466,C#CCC(C(=O)NC(C1(CNC(=O)C(=Cc2cccnc2)F)CC1)C)C1CC1 22467,C1(NC(=O)NC2C(C)OCC2)CCC2(CCC2)C1Nc1ccc(Cl)cc1 22468,CCC(CC)(CC)C(=O)N(C)CCN(C(=O)CS(=O)(=O)CC)C1CC1 22469,C1(S(C)=O)(CNC(C(C2CCC2)NC(C(C)NC(COC)=O)=O)=O)CC1 22470,Cc1cn2c(C)c(C(=O)NCCN(C3CCCC3)C(C3CCOC(C)C3)=O)nc2s1 22471,C1(C(=O)NCCC(=O)NCC#C)CCC(O)CN1C(c1ncc(F)cc1F)=O 22472,S(=O)(=O)(c1ccccc1OC(F)(F)F)NC(C1C(C#C)C1(C)C)=O 22473,c1(N(C(=O)COCC2CC3CC3C2)C(C)C)ccccc1 22474,CC1COC(C(=O)NCC(C)NC(=O)Cc2ccn(C3CCCC3)n2)CO1 22475,C1(NC(C(C)N(C(C)=O)C)=O)CC1C1CCCN(C(=O)COCC2CCCC2)C1 22476,N1(C(=O)CCCN2CCCCC2)CCc2nc[nH]c2C12CCN(C(C1CC1F)=O)C2 22477,C1(CNC(C2C(CNC(=O)CNC(C3CCC3)=O)C2)=O)CCCO1 22478,Cc1nc(NC23CCCC2CN(C(c2nc(C)c(C)nc2C)=O)C3)c(C)c(O)n1 22479,C1(O)(CC(=O)NCC(C#C)NC(=O)C(C)(C)OC2CCCC2)CCCCC1 22480,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 22481,CC(C)CC(=O)N(CCC(=O)NCCCOC1CCC1)Cc1ccccc1 22482,C1(F)(C(=O)Nc2cn(CC=C)nc2)CCN(C(C2(C)CCN(C)C2)=O)C1 22483,N1(C(C2(CCC)CC2)=O)CCC(F)(F)C(CNC(C2(N(C)C)CC2)=O)C1 22484,CC1=CC(C)CN(c2cc(NCc3cc(C)c(O)nn3)ncn2)C1 22485,c1(C(N2C3C(NC(Cc4c(OC)ccnc4)=O)C(C3)C2)=O)cncc2nc[nH]c12 22486,C(C1=NOC2COCC12)CNCC(C)(C)NC(N)=O 22487,C1(CNC(C2CCCCO2)=O)CCCCN(C(C2CC3C=CC2C3)=O)C1 22488,c1(C(N(C)CC2N(C(C(C=C)C)=O)CCCC2)=O)cc(C(C)C)ccc1F 22489,CCC(C)(C)CCCC(=O)NCCC1(CNC(=O)CCc2ncccn2)CC1 22490,c1(N(C(c2cc(OCC)ns2)C(=O)NC(C)CC)C)cc(F)c2ncccc2c1 22491,C1(C(=O)NCC(C)CN(C)C(c2nccnc2O)=O)CS(=O)(=O)CC12CC2 22492,C1(C(N(C(=O)Cn2ncccc2=O)C)=O)CCN(C(C2(N(C)C)CC(F)C2)=O)CC1 22493,C(C(C)C(C)(C)C)NC(C1CCCN(Cc2ccccc2Cl)C1)C 22494,C1(NC(CC2(NC(c3ccc(C)c(F)c3)=O)CCC2)=O)CCCOC12CCC2 22495,c1(C(=O)NCCCCN(C)C(C2CC(=O)N(O)C2)=O)coc2c(F)cccc12 22496,C1(C(=O)NCC(c2ccc(F)cc2F)NC(CCCSC)=O)CC(S(C)(=O)=O)C1 22497,CCC(CO)CCNC(=O)C(C)CN(C(=O)CCC1CC(C)C1)C 22498,C=CCC(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)CN(C)C(C)=O)C1 22499,c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CCCC2)nocc1Cl 22500,c1(-c2cn(CCCC(=O)N3CCC3C3CN4CCC3CC4)nn2)ccc(Br)c(Cl)c1 22501,c1(CCC)c(NC(C2CC(NCc3cnc(C)[nH]3)C2)=O)cnn1C 22502,c1(OC)ccc(C(=O)NC2(C)CC(NC(=O)C(C)N(C)C)C2)cc1[N+](=O)[O-] 22503,c1(C(N2C3C(NC(C(c4ccccc4)OC)=O)C(C3)C2)=O)ccc(=O)n(C)c1 22504,c1(CC(N2C(C)CC(NC(=O)CSC(=N)N)CC2)=O)ccccc1S(C)(=O)=O 22505,C1(O)(SC)CCN(C(=O)NCC2(c3cccnc3)CCCCC2)CC1 22506,c1(C(=O)NC2CCC(NC(C(c3ccccc3)C)=O)CC2)ccnc(Cl)c1O 22507,CC1=C(C(=O)NC(C2CCN(C(c3ncccc3N(C)C)=O)C2)C)CCO1 22508,Cc1cccc(C(N2CC(CC(=O)N(CC(C)CO)C)C(C)C2)=O)c1O 22509,c1(C(=O)NCCC(C)(C)NC(c2cc(C(C)(F)F)n[nH]2)=O)ccnc(F)c1O 22510,N1(C(C(C)=C2CC2)=O)CCC2(COC(CNC(C3CC3C3CC3C)=O)C2)C1 22511,C(CN=C(NC1CCS(=O)(=O)C1)NCCCC=C)NC(C1CCCCN1C(C)C)=O 22512,N(C(=S)N1CC(=CBr)C2(CCC2)C1)C(C=C)CO 22513,C(C)(C(C(=O)NC(C)(C)CCN(C)C)C(C)C)NC(C(CC=CCC)C)=O.OC 22514,c1(CC(C)C(=O)N(C)CCOCCNC(C2(F)CC2C)=O)ccccc1F 22515,C(CNC(C1CCCC1F)=O)(CC(C)C)NC(c1n(COC)ncc1)=O 22516,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22517,c1(OC)cccc(C(=O)NC2(OCc3ccccc3)CC2)c1.C12CC(C1)CC2=O 22518,N1(C(CC(=C)Br)=O)CCC(NC(=O)COCCCC)C(F)C1 22519,c1(CCF)ccccc1OCNC(=S)NC1(C)CC1 22520,N1(C(c2cncc(C)c2)=O)CC2CC1CN2Cc1ccc(CO)s1 22521,C1(NC(C(N(C(=O)CCC2CCCC2)C)C2CC2)=O)CCCC1CNC(N)=O 22522,C(CCC(CO)NC(=O)CC(O)C1CCCC1)NC(c1cn(C(C)C)nc1)=O 22523,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22524,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(C(OC)OC)=O)CCC1 22525,c1(C(=O)NC2CC(C)(NC(COC(C)(C)C)=O)C2)cc(F)c2c(c1)CCC2 22526,C(C(=O)NCC1CC(O)CN1C(C1(C(C)(F)F)CCOCC1)=O)(C(C)C)OC 22527,c1(C(=O)NCC2(F)CCC(NC(CCCC(N)=O)=O)C2)ccc(F)c(F)c1F 22528,C(CO)(C(=O)NCCCN(C(=O)CC(=O)OC)C)OC 22529,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)CCOC2 22530,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOCC3)CO2)C1 22531,c1(CNC23CCN(C(=O)OC(C)(C)C)C2CCC3)nc2cc(F)ccc2s1 22532,c1(NC(=NC)NCC(N2CCCC(C)C2)C)ccc(Br)cc1OC(C)C 22533,N1(C(=O)CCCC2CC2)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22534,c1(SC)ccc(C(N2CCCC(NC(c3ncsc3C)=O)CC2)=O)cc1[N+](=O)[O-] 22535,C1(C(=O)NCCC2CCN(C(=O)CCc3ncc[nH]3)C2)CCCC(CF)C1 22536,C(CCCC(CO)NC(c1cc(C)nnc1O)=O)NC(c1cccc(CC)c1)=O 22537,C1(C(=O)OC)(COC)COCCN1C(=O)CCCN1CCC(N)C1 22538,C1(OC)CCC2(C(N3CCN(C(c4ccc(Cl)cn4)=O)CC3)=O)CCC12 22539,N1(C(CCP(C)(C)=O)=O)CCOC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 22540,N1(C(=O)COCCc2ccccc2)CCC2(CCCN2C(C2CCCO2)=O)C1 22541,Cc1cnsc1C(=O)N(C(CC)C(=O)NC1CC1C)C 22542,C1(CNC(C2C(F)(C(=O)OC)C2)=O)CCN(C(=O)C(C2CC2)OC)CC1 22543,N1(C(C=CCN(C)CC)=O)CC(O)CC1C(=O)N(CCN=[N+]=[N-])C 22544,c1(OC)ccc(CNC(CCN(C(=O)C(O)C(C)C)C)C(C)C)cc1.C1C(=O)N1 22545,c1(C(=O)NC(C2CCN(C(C=CC)=O)C2)C)cc2c(c(S(N)(=O)=O)c1)CCC2 22546,C1(CNC(NC(C=C)C)=NCCC=CCl)CCC2(CCC(C)(C)CC2)O1 22547,c1(C(N2CC(C(C)NC(c3nc(C)no3)=O)C2)=O)nc(-c2cccs2)oc1C 22548,N1(CC)CCC(C(N2CC(C(O)C(=O)NC(CC3CCCC3)CO)C2)=O)C1 22549,C1(CCN(C(c2n(CC)ccc2)=O)C)CCCCN1C(c1cnc(Cl)[nH]1)=O 22550,c1(C(=O)NCCN(CCC)C(C2CCC(=O)C(C)C2)=O)cnc(CC2CC2)nc1O 22551,C1(C(N(CCN(CC=C)C)CC)=O)C(C)CCN1C(=O)C(F)C1CCC1 22552,C1(N(C(CC(CC)OC)=O)C)CCN(C(=O)CCN2CCOCC2=O)CC12CC2 22553,CC(CS(=O)CCN=c1[nH]c(=NCc2cc(Cl)cc(Br)c2)c2sccc2[nH]1)N(C)C 22554,c1(CC)cc(-c2ccc(CO)nc2)n2ncc(C#N)c2n1 22555,C(=O)(CCC(CF)CF)NC(C(C(=O)NC(C)CC1CC1)(C)C)C 22556,Cc1cc(=NC(=O)C(C)(C2CC2)N(C(=O)CC(O)CN(C)C)C)[nH]n1C1CC1 22557,c1(NC(C2(NC(C(CC)(C)O)=O)CC(O)C2)=O)cc(OC)ccc1C 22558,C12(C(=O)NCCCCCCNC(=O)COC3CCCC3)CCCCC1C2(F)F 22559,c1(C(=O)NCCN(C(c2cc(CCC)c(C)s2)=O)CC)c(F)cc(C)cc1Cl 22560,Cc1nnc2n1CC(N=c1nc(N(C)CC3CCSC3)c3c([nH]1)CCOC3)CC2 22561,Cc1oc(C)c(C(=O)NC2CC2CNC(=O)CSc2ccc(Br)cc2)c1C 22562,C1(CNC(CCN(S(C)(=O)=O)C)=O)COCC1NC(C1CCCO1)=O 22563,c1(NC(=O)NCCOC(CNS(CC)(=O)=O)(C)C)cncc(-c2cncnc2)c1 22564,N1(C(c2nc(SC)sc2)=O)CCN(C(=O)CC2CCC(C)C2)CC1C1CCC1 22565,C1(c2cn(C(=O)Cc3sccc3Br)nn2)CCN(N(C(=O)C)C)CC1.C1CCC1 22566,c1(OC)ccc2c(C(=O)NC3CC(C)CN(C(c4[nH]ccc4C)=O)C3)cnn2c1 22567,C1(CC(N2CC(COC)(CNC(C3CNC(=O)N3)=O)C2)=O)CC2CCC1CC2 22568,N1(C(CC)=O)CCC(C)(C)C(C(=O)NCc2cc(C3(C)CC(C)(C)C3)no2)C1 22569,c1(N(CC(c2cccc(C(F)(F)F)c2)O)C(C)C)ccc(F)cc1F 22570,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(C2CC(O)C2)=O)CC1 22571,C(=O)(C1c2ccccc2CCN1CC(c1cc(Cl)ccc1I)=O)OC 22572,C=C(C)CC(C(=O)N1CCC(C)(N(C)C)C1)OC.C1CC(=O)ON1C 22573,CC1CN2CCN1C(C(N1CCCC1C1CCN(C(=O)CC3CC3(Cl)Cl)C1)=O)C2 22574,N1(C(COCCCCC)=O)CC(O)CCC1C(=O)N(C1CC1)Cc1ncnn1C 22575,Cc1cc(C#N)nc(=NCC(C)CNC(c2c(C3CC3)cnn2C)=O)[nH]1 22576,N1(C(c2cc(C)nc(O)n2)=O)CCCC2CCN(C(c3ncc[nH]c3=O)=O)CC12 22577,c1(OCC)ccc(C)nc1C(=O)NC(C1CCCN(C(C2C=CCC2)=O)C1)C 22578,N1(C(CSCC#C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ncccc12 22579,CCCC(CC)CCN1CC(=O)N(CCc2ccnc(C(N)=O)c2)C1=O 22580,c1(C(N2CCC(NC(CCn3c(C)ncc3)=O)C2)=O)cc2scc(C)c2[nH]1 22581,C=CC1(C(=O)NCCN(CC)CC)CCN(C(=O)CCCC2CC2)C1 22582,c1(C(=O)NCC2(F)CCC(NC(C3CN(C)C3)=O)C2)ccnc2ncccc12 22583,C12(C(=O)NC(C3CCN(C(c4ncc(CC)cn4)=O)CC3)C)CC1CCC2(F)F 22584,N1(C(C2=C(C)CC2)=O)CC2COCC2(C(=O)NCC(=C2CCCCC2)F)C1 22585,O=C1CCC2(CCCN(CC(C34CC(Br)(C3)C4)(F)F)C2)N1 22586,c1(CSC)cccc(C(=O)NC2CC2CNC(=O)C(C)C2CCCO2)c1 22587,c1(CC)nc[nH]c1C(=O)NCC(C1CC1)NC(C1(C(F)(F)F)CC1)=O 22588,c1(C(N2CC(CCCC)(C(=O)N(CC(C)(C)C3CC3)CC)C2)=O)ccc2cccnn12 22589,Cc1coc(C(=O)NCC(C2CC2)NC(=O)C(c2ccc(Cl)cc2)O)c1C 22590,C#Cc1ccc(C(N2CCC(C)(NC(c3cc(O)ncc3Br)=O)C2)=O)nc1 22591,CC1CCn2c(C(=O)N(C)Cc3ccncc3C(F)(F)F)cnc2C1 22592,Cc1ccc2occ(CC(=O)N(C(C)CNC(C3CCC(C)(C)OC3)=O)C)c2c1 22593,C1(NC(CC(C)C2CCCCC2)=O)CC2(CCCN(C(C3CC(=O)C3)=O)C2)C1 22594,c1(C(C)C)ccccc1CC(=O)NCC(C)(CO)NC(=O)C(C)NS(C)(=O)=O 22595,C1(CC(=O)NCC2(C)CCN(C(C34CCC3CC4)=O)C2)CN2CCN1CC2 22596,c1(C(N(CCNC(C2(CC)COC2)=O)CC)=O)noc2cc(F)ccc12 22597,C(=O)(C1=C(C)CCN(CCCNC(=O)NCCSC)C1)OC 22598,N1(C(c2c3ccc(C)cc3sc2)=O)CC2CCCC(C1)N(C(=O)C#CC(C)C)C2 22599,CCCCCC(O)C(=O)N1CC2CC1C2C(N1CCC2CC12)=O 22600,N1(C(C2(NC(c3c(CC)cno3)=O)CC2C)=O)CC(C)SC(C)C1 22601,C1(C(=O)NC(COC)C)CCN(C(c2c[nH]cc2OCC(F)(F)F)=O)CC1F 22602,N1(C(N2CCCC(N(OC)C)C2)=O)CCOC2(CCC(F)(F)CC2)C1 22603,N1(CC(=O)N(CCC(C)NC(c2scc(OC)c2)=O)C)CC2CCC1C2 22604,c1(C(C)=O)ccc(C(=O)NC(C)(C)CCNC(=O)CCS(C)=O)cc1 22605,CCCC(C(=O)NCC1(c2nn[nH]n2)CCCCC1)OCC 22606,c1(CCC(=O)N(C)CC2(NC(C3N(CC)CC3)=O)CC2)ccccc1C#N 22607,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22608,O=C(CC1=CCN(C(C2(O)CCOC2)=O)CC1)Nc1cncc(CO)c1 22609,c1(C(=O)Nc2cc(OCCO)n[nH]2)ncc(F)cc1F.c12occc1C(=O)NC2 22610,c1(C(N2C(C(C)NC(C3CC34CCCCC4)=O)CCC2)=O)ccc2snnc2c1 22611,C1(C(N(C)CC2(NC(c3ccc(CO)cc3F)=O)CC2)=O)CC(C)(C)OC1(C)C 22612,CC1=C(C)CC(C(=O)NCCC2(CNC(C3(O)CCC(C)CC3)=O)CC2)CC1 22613,c1(OC)cc(C(=O)N(C(CNC(c2nsnc2O)=O)C2CC2)C)ncn1 22614,C1(C2CCN(C(C#CC)=O)C2)CCCN(Cc2nccc(OC)n2)C1 22615,CCC(CC(=O)NC1CN(C(=O)C(C)(CC)OC)C1)C1CCC1 22616,Cc1ccn2cnc(C(=O)NCC3(F)CCN(C(=O)C=CCF)CC3)c2c1 22617,C(=O)(CC(C)(O)CCC)NC(CCCC)CNC(c1ccc([N+](=O)[O-])cn1)=O 22618,N1(C(C(CCC)OCC)=O)CCC(C(=O)NCCC2(CSC)CC2)=C(F)C1 22619,C1(CNC(CSCC(C)C)=O)CC2(CCC2)CN1C(=O)CC(C)n1cccn1 22620,O=C(C(F)C(F)(F)F)NC1CCC(C(=O)NCC2CC2c2ccco2)CC1 22621,C1(C(N2CCC(CF)C2)=O)(CC)CCCC1O.C(C(C)(C)SC)=CC(=O)N 22622,C1(NC(C2CC(CCC)C2)=O)CCN(C(c2ccnn2CC)=O)C(C)C1 22623,c1(C(=O)NCCN(C(C(C=C)O)=O)C)nc2ncccc2cc1C 22624,CCCC(O)CC(=O)N(C1CCCN(C(c2nccn2C(C)C)=O)C1)C 22625,C1(CC)CCC(COC)CC1.c12nc(n[nH]1)COC2 22626,C1(C(=O)NCC(CN(C)C(c2ccc(CO)cc2F)=O)O)CC2(COCCO2)C1 22627,N1(C(CCCCC(=O)OC)=O)CCC2(C1)CN(C(=O)C(F)C1CC1)CCO2 22628,N1(C2CN(C(C(C)OC(Cc3noc(C)c3C)=O)=O)C2)CCSC(C)(C)C1 22629,S(=O)(=O)(c1ccc(=NCC2CNC(=O)C(C)(C)C2)[nH]c1)NCC(c1n(C)ncc1)O 22630,CCC(CNC(c1cc(SC)cnc1C)=O)(CC)NC(=O)CN(C)C(C)C 22631,Cc1cc(C(N2CC3CC2CN3C(=O)C2=CCC(C)CC2)=O)cc(C)c1O 22632,c1(OCCC(=O)NCC(C)N(C(=O)C(C)(F)F)C)ccc(F)cc1 22633,C1(CC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22634,c12ccccc1CC(=O)NC(=O)CCCNC(C)(C(=O)OC)CS2.CC 22635,C(C(C(=O)NC1CC(C(C)O)C1)NC(C1OCCO1)=O)OC 22636,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22637,C1(NC(CC=CC)=O)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1CO 22638,N1(C(C=CCNC(C2(C(F)(F)F)CC2)=O)=O)CC2CCC=CC12 22639,C1(CC(=O)N(c2cccc(OC(F)F)c2)C)NC(=O)NC1=O.C1CCCC(=O)O1 22640,C1(C(N(c2ncncc2-c2ccccn2)C)=O)CNCC(F)(F)C1 22641,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22642,c1(CN(C)C(c2cnn[nH]2)=O)cnn2c1CN(C(C1(CO)CC1)=O)CC2 22643,c1(OC)cccc(NC(C2CCC(NC(C3CC(O)C3)=O)C2)=O)c1C 22644,C1(C(=O)NCC=C)CCC2(CN(C(=O)C(=O)NCc3ccc(Cl)c(F)c3)C2)O1 22645,C1(C(=O)NC(C#C)C(C)OC)CCCCCCN1C(=O)C(F)CCC 22646,c1(C(=O)Nc2c(C(=O)OC)oc(C)c2)cc(OC)ncc1C1=COCC1 22647,C1(OC)CC(NC(C2CC=CC2)=O)CN(C(c2cn(CCC(C)C)nn2)=O)C1 22648,C(=O)(C(CCF)NC(=O)C1CC1)NCC(C1CCC1)NC(CC=C)=O.C(C)(C)(C)C 22649,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22650,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22651,c1(CC)onc(C(F)(F)F)c1C(=O)N(CCNC(=O)CSC)Cc1nncn1C 22652,O=C(CC(Cc1cn(C2CCCCC2O)nn1)NC1CCCCC1)N1CCCC1 22653,c1(N2CC(CC=C)(NC(C3COCCN3C)=O)C2)ncc(C)c(C)n1 22654,c1(OC)cncc(C(=O)NC2CN(C(c3cn(C4CC4)nc3C)=O)C2)c1C 22655,CCCC(C(=O)NCC1CCC(C(=O)NOCC2CCCO2)CC1)NC(N)=O 22656,N1(C(C(C)(C)CO)=O)CC2CC1CCC2NC(c1cn(-c2cccnc2)cn1)=O 22657,c1(OCC)ccc(-c2ccc(NC(=O)Nc3cc(C)cc(C)c3)nc2)c(C)c1 22658,N1(C(C2C(c3n(C)cnn3)CCC2)=O)CCNc2cc(Br)ccc2C1 22659,N1(C(c2cn(CCOC)nc2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22660,C1(NC(C=C(CC)C)=O)CCN(C(=O)COc2ccc(C)cc2)CC1C 22661,Cc1c(N2CCN(C(=O)NCCCc3ccoc3)CC2)cccc1Cl 22662,CC1CC=C(C(=O)NC(CC2CC2)C(=O)NCCCn2cnnc2)CC1 22663,C1(C)(CC(C2CC2c2cccnc2)N(CCCCOCC)C)CCCO1 22664,c1(C(=O)NCC#CCNC(C(COC)COC)=O)sc(C)c(Br)c1OC 22665,C1(CC(=O)NC)CCCN(C(C2(OC)CN(C(C3CC3(C)C)=O)C2)=O)C1.C(C)(C)C 22666,c1(C(C)C)cccc(C(F)F)c1F.c12cccc(c1)CCCCC(=O)N2 22667,Cc1c(C(=O)NC(C)(C)CNC(C2(C)CC2)=O)nc(O)c2ccccc12 22668,N1(Cc2cn(C)nn2)CC2(C1)CC2(F)F 22669,c1(OCC=C)ccccc1C(N1CCCC1(C)C(=O)N(C)Cc1ccccn1)=O 22670,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22671,C1(NC(C2CC(N(C(C(C)Oc3cncnc3O)=O)C)C2)=O)CN2CCC1CC2 22672,C1(CNC(=O)C(F)=CCCF)C2CN(C(=O)Cc3ccsn3)CC12 22673,C1(CCC(=O)NCCNC(C2CC3CC3C2)=O)CCN(C(=O)C2CC2)C1 22674,N#Cc1c(Cl)nsc1NCC(=O)NC1CCCC1CO 22675,C1(NC(C=CC=CCC)=O)CCC(O)CN(C(=O)CCC2CCN(C)C2)C1 22676,c1(C(=O)NCCNC(c2c(C)n3c(n2)scc3)=O)ccc(S(N)(=O)=O)nc1 22677,CC(CC(C)(C)C)C(=O)N1CC(N(C)C(c2ncc(Cl)c(OC(C)(C)C)n2)=O)C1 22678,C(CNC(=O)Cc1c(C)noc1C)(CC(=O)NCC(F)(F)C(F)F)OC 22679,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2cccc(C)c2Cl)=O)CC1 22680,C1(CC)CN(C(=O)CCc2c(C)cnn2C)CCC1NC(=O)C(C)(C)COC 22681,c1(C(=O)NCC(CC)NC(C=CC=CC)=O)cnn2cccc(Br)c12 22682,N1(NC)CCOCC1.C1(C(CN(C(C(C)NC=O)=O)C)O)CCCCC1 22683,C1(CC(N2CC(CCC)C(C(=O)NCC(C)(F)C(C)C)C2)=O)CN2CCC1CC2 22684,CC1CCc2sc(CNC(=O)Nc3nc4ccccc4nc3C3CC3)cc2C1 22685,c1(NC(CC(COC)NC(c2cc(CC)ncc2)=O)=O)ccc(F)cc1C 22686,C(=O)(CC(O)C(C)C)NCC(CC)NC(=O)C=Cc1cocn1 22687,C1(CN(C)Cc2cnn(C)c2)CCN(C(=O)C(C2CCOCC2)=O)CC1 22688,C(=O)(C1CCc2cccnc21)NC1CCN(C(c2cc(C)on2)=O)CC1O 22689,C1(c2cn(NC(COC)=O)nn2)CN(C(=O)Cn2cccn2)CCC1(C)C 22690,c1(C(N2CCC(C(NOCC#CC)=O)CC2)=O)cc(C#N)[nH]c1C 22691,C1(C(=O)NCC2(C#N)CC2)CC2(CCN(C(C3CCCCO3)=O)C2)C1 22692,C(=O)(C(C)CC(=O)NC(c1cncc(C(=O)OC)c1)C)NC 22693,c1(NC(C(=O)NC(c2c(OC(F)F)cccc2Cl)C)=O)cccc2c1CCC2 22694,c1(C(C)C)nc(=NCC2CCCCN2C(c2cn(C)cn2)=O)s[nH]1 22695,C1(NC(c2cc(C)ncc2)=O)CCN(C(=O)CCc2ccoc2)CC1F 22696,c1(C(C)=O)c(Cl)cc(OC(=O)CSCC(=O)Nc2nnc(C)o2)cc1Cl 22697,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(C1CCCC(C)CC1)=O 22698,c1(CN2C3CC(C(=O)O)(C3)C2)cnc(N2CCOCC2)c(Cl)c1 22699,Cc1cc(N2CCC(NCCC3CCNC3=O)CC2)ccn1 22700,n1(CC)ncc(C(=O)NC(CO)C(C)NC(=O)C(C2CCCCC2)F)c1C1CC1 22701,Cc1cc(Cl)c(C(=O)NC2CC3CC(NC(C4C5COCC45)=O)CC3C2)cc1C 22702,Cc1ccc(OCC(=O)N(CCCCCNC(c2c(C)[nH][nH]c2=N)=O)C)cc1 22703,c1(C(N2CC(CCCCNC(CC(=C)Br)=O)C2)=O)ccc(C(C)C)nc1C 22704,Cc1ccc(OCC(=O)NC2CC(CCNC(=O)C(c3ccccc3)F)C2)cc1 22705,N1(C(=O)C2=C(Cl)CCCC2)CCC2(CCCN2C(C2(n3cnnn3)CC2)=O)C1 22706,c1(C(=O)NC(c2ccc(C)nc2)CO)cccc2cc([N+](=O)[O-])ccc12 22707,Cc1ccncc1C=CC(=O)NC1CC(NC(=O)CC2CNC(=O)C2)CC1O 22708,CC(CCCCNC(C1CCOC1C1CC1)=O)NC(c1ccc(F)nc1)=O 22709,C(=O)(C1=C(C)CN(C(c2ccc(N3CCCC(O)C3)nc2)=O)CC1)OCC 22710,C1(C)(COCC)COCCN1C(=O)Cc1ccc(Nc2ccc(Cl)c(Br)c2)cc1 22711,C1(NC(C2(C(C)C)CCN(C(CC3ON=C(C)C3)=O)C2)=O)CCN2CCCC12 22712,N1(C(c2cnn(CCC)c2C)=O)CCC2CN(C(c3coc(C)n3)=O)CC2C1 22713,C1(C(=O)NCC(C)NC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22714,CCCC(CC(C)C)C(=O)N1CCN(C(=O)C(O)COCC)CC1C 22715,c1(NC(C(C)C)CNC(=O)CP(C)(C)=O)ccc(S(=O)(=O)N(C)C)cn1 22716,C1(C(=O)NCC(CC)C#N)(CNC(=O)CC2COCC(C)O2)CC(C)(C)C1 22717,Cc1nc2cncc(C(=O)NCC3CN(C(C4C(Cl)(Cl)C45CC5)=O)CCO3)c2[nH]1 22718,C(CC(F)(F)Cn1cc(-c2cnn(C)c2F)nn1)COC(CC(C)F)=O 22719,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)C1CC1)C 22720,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccncc2O)=O)CC1 22721,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC(C)N(C(C3C4COCC34)=O)C2)c1)NC 22722,CC1CCN(C(=O)CCC2CC(NC(=O)CCc3cn(C)cn3)C2)C(C)C1 22723,N1(C(CC2ON=C(C)C2)=O)CCCC(C)(CNC(=O)CCCc2ccc(C)s2)C1 22724,c1(C(=O)NC2C3CCN(C(CN(CCOC)C)=O)C3C2)nccn2nccc12 22725,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)NC(=O)C(N1CCCCC1=O)C)C 22726,c1(OC)ccc(N(C(c2nc(-c3ccoc3C)n(C)n2)C(=O)NC2CCC2)C)cc1 22727,c1(CC(N2C(C(C)C)CN(C(C3(CO)CCC3)=O)CC2)=O)ccc2c(c1)OCO2 22728,c1(OC)cc(O)cc(O)c1C(N1C2CN(C(=O)CC34CCCN3CCC4)CC12)=O 22729,c1(OC)cc(C(N2CCN(CC(=O)OC)CC2)C(=O)NCCC#N)ccc1I 22730,c1(C(=O)NCCCN(C(C2(CC=C)CCCC2)=O)C)cnc2[nH]cnc2c1 22731,C(CNC(C1(C(F)F)CC1)=O)(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O 22732,N1(C(C2(C)CCC(C)CC2)=O)CC=C(CCNC(=O)C(C)(C)c2ccns2)CC1 22733,C1(C(=O)NC(C(=O)NCC(C(C)O)(C)C)C)CC(=O)NC1(C)C 22734,N1(C(COCC(=O)OC)=O)CCC(C)(C)C1C(N1CC(C)(C#N)C1)=O 22735,S(=O)(=O)(c1cccc(-c2nnc(CC(C)C)o2)c1)NC(CC=C)C1CC1 22736,C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CC2CCCOC2)CC2(CC2)C1 22737,C(C1C(C(=O)N(CCNC(c2sc(COC)nc2C)=O)C(C)C)C1(C)C)=C(C)C 22738,O=S(c1ccc(NC(=S)NCCc2cccs2)cc1)C(F)(F)F 22739,c1(CC(N2CC3(CN(C(c4cc(C(C)C)on4)=O)C3)C2)=O)cc2nc[nH]c2cn1 22740,CCC(CC)CC(=O)NC(c1nn(C)cc1O)C 22741,C1(C(=O)NC(C)C(=O)N(C)CC2CC(NC(N)=O)C2)CCCCC1 22742,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(=O)CCn3ccnc3)C2)c1C 22743,CCC(CC)CCCC(=O)NC(C1(O)CCN(C(c2noc(CC)c2C)=O)C1)C 22744,C1(NC(CCN2CCN(C(C)C)CC2)=O)CC(O)CN(C(c2csc(Cl)n2)=O)C1 22745,C12(C(=O)NCC(CC)NC(=O)C=Cc3cn(C)cn3)COCC(C1)C2 22746,N1(C(CN(C2CCC2Oc2ccccc2)C)=O)CC(=O)NC2(CC2)C1 22747,C1(NC(C2(N=[N+]=[N-])CC2)=O)CCCN(C(c2cc(C(F)(F)F)cs2)=O)C1 22748,C=CCC(C(=O)NC1CC2CCC1CN(C(=O)C1CC1)C2)C(C)(C)C 22749,C1(NC(c2nc(C)sc2)=O)CN(C(C2CNC(=O)C2)=O)CC12CCS(=O)(=O)CC2 22750,C(=O)(C1CCCn2cnnc21)NCC1(O)CN(C(c2n(CC)ncn2)=O)C1 22751,C1(C(C)(C)NC(=O)Cc2cn[nH]c2)CCN(C(c2cnnn2C2CC2)=O)CC1 22752,N1(C(c2c(C)ccnc2)=O)CCC2(CC1)CC(NC(C1CCN(C)C1C)=O)C2 22753,c1(CCC)nc(-c2cncc(Cl)c2)n(CCC(C)(C)C)n1 22754,C(CCN(C)C(=O)Nc1ccc(Cl)o1)(C(C)C)NC(Cc1cn(CC)nc1)=O 22755,c1(C(=O)NCC2(OC)CN(C(C(C3CCOC3)OC)=O)C2)ccc(O)c(CO)c1 22756,C(C)(N=c1cc(C)nc(N(C)C(C2CCOCC2)C)[nH]1)c1cccc(NC)c1 22757,N1(C(CC2(COC)CCC2)=O)CCC(C(C)(C)C)(CNC(C2CCCCC2)=O)C1 22758,c1(CC)cc(CNC(=O)C(C)=CCNC(c2cc(OC)n[nH]2)=O)on1 22759,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22760,C=CC1OCCC1C(=O)NCCC1CC(NC(=O)CCC2CC2C)C1 22761,c1(OC)cc(Cl)ccc1NC(=O)CCC(=O)NCC(C)(O)c1cccs1 22762,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22763,C(=O)(C1COc2ccccc21)NC1CCN(CC(=O)NC2CC2(Cl)Cl)CC1 22764,CC(C)C(O)C(C(=O)Nc1ccccc1CN(C)C)NC(c1ccco1)=O 22765,N1(C(C(C)NC(N)=O)=O)CCC2CN(C(c3ncc(Cl)s3)=O)C2C1 22766,C(=O)(CC(O)CC(C)C)N1CCC(CCNC(c2c(C)[nH]c(C)c2C)=O)C1 22767,c1(NC)c(C(=O)NC2CN(C(=O)OC(C)(C)C)CC2c2ccccc2)cccc1F 22768,c12ccc3c(c1)CN(C3)C2=O.C1(NC(C(C)C)=O)C2COCC12 22769,C1(C(NOCCC=C)=O)CCCCCC1NC(c1ncc(COC)cn1)=O 22770,c1(C(=O)NC2C3(CCN(C(C(C(=O)OC)C)=O)C3)C2)ccc2nc(COC)[nH]c2c1 22771,C1(NC(c2n(C(C)C)ncc2Br)=O)CCCCCN(C(=O)C(C)C2CC2)C1 22772,c1(C(=O)NCCC(C(CO)NC(=O)OC(C)(C)C)C)ccc(C#N)c(O)c1 22773,C=CC1(C(=O)NCCN2CCC(CO)C2)CCN(C(=O)C(C)C(C)(C)C)C1 22774,c1(C(N2CC3C(C(N4CC5CCC4C5)=O)C3C2)=O)ccc2ncnc(O)c2c1 22775,CCCCCCCCCCCCCCCOC(C1CC(=O)NC2(CCC2)C1)=O 22776,c1(C(N2C(C)(CC(=O)N(C3CC4(CC4)C3)C)CC2)=O)ncc(Cl)cc1Cl 22777,c1(CC(=O)NC(C)CNC(c2ccnn2CC#N)=O)ncccc1F 22778,N1(C(CSC(C)=O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)c(O)c(Cl)c3)c2C1 22779,c1(C(=O)OC)cc(C(=O)NCCNC(=O)COCC2CCCCO2)on1 22780,Cc1oc(C(F)(F)F)nc1C(=O)NCC1(NC(C2CN(C)C2)=O)CC1 22781,c1(C(=O)NCC2(CN(C)C)CCC2)ccccc1-n1cc(CCS(N)(=O)=O)nn1 22782,C12(CNC(C3(CSC)CC3)=O)CC(NC(=O)CCC=CC(C)C)(CO1)C2 22783,N12CC(O)CC1CNC(=O)NCC2=O.C1(C[Si](C)(C)C)(C(F)(F)F)CC=CC1.N 22784,C12(COC)CC(C(=O)NCC3CCC(F)(CNC(=O)CC(C)(C)C)C3)(CO1)C2 22785,C1(CC(=O)NC2CCC2)CCCN1C(c1cnsn1)=O 22786,c1(OCC)cc(CNCCc2noc(C3CCOCC3)n2)cc(F)c1 22787,Cc1nnn(CC(=O)NCCCCN(C(=O)Cc2ccn(C3CCCC3)n2)C)n1 22788,N1(C(C(C)(C)OCC)=O)CCC2(CC1)CC2NC(c1cnn(C2CC2(F)F)c1)=O 22789,c1(CC)nc[nH]c1C(=O)NCC1(Cn2cc(C(C)OC)nn2)CC1 22790,Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)CC(c2cccc(F)c2)O)CC1C 22791,c1(NC2(C(N3C(CC(=O)N(CC)CC)CCC3)=O)CC2)cc2ccccn2n1 22792,c1(C(C(C)(C)OC(=O)C(CCC#N)Nc2ccccc2)=O)nnc2n1CCCCC2 22793,c1(N(C(=O)NC(c2nnc(N(C)C)o2)C)C)nn(C)c2ccc(Br)cc12 22794,CC(C)CC(C(=O)N1CCC(C2CCCN2C(c2ncccc2Cl)=O)C1)C(N)=O 22795,N1(C(c2occ(C)c2C)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22796,N1(CCOC)CCc2c(NC(c3cc(CC(F)(F)F)ccc3F)=O)cccc2C1 22797,N1(C(CCCCC)=O)CC2(C1)CN(C(=O)CCC1CCCC(O)C1)CC2CO 22798,C(=O)(C(CCCC)C(C)C)N1CCN(C(CCC=CC)=O)C(C)CC1 22799,C1(CNC(c2c(C3(C)CC3)ocn2)=O)CCCCN1C(=O)C=CC(F)(F)F 22800,Cc1cn2c(C(=O)NCCCCC3CN(C(=O)C=C4CCOCC4)C3)c(C)nc2s1 22801,CC1(C)C(NC(=O)CCSc2ccc(Cl)cc2)CCN1C(=O)C(O)CC1CC1 22802,N1(C(CCC(C)C)=O)CC(C)CN(C(=O)C(c2cccc(Cl)c2)=O)C(C)C1 22803,c1(C(=O)NC2CN(C(C(C(=C)C)(C)C)=O)CC2F)cc2ccc(C)cc2[nH]1 22804,N#Cc1ccc(NC(C2CN(Cc3cc(Br)c[nH]3)CC2(F)F)=O)cc1Cl 22805,N1(C(C2(SC)CCC2)=O)CCC(N(C(=O)C(C)n2cncn2)C)C2(CC2)C1 22806,C(=O)(C(CCC(C)C)NC(=O)CCOCC(F)F)N1CC(NC(=O)NC)C1 22807,CC(O)CCC(=O)NC1CCC(NC(=O)C(c2cccc(Cl)c2)C2CC2)CC1 22808,C1(C(=O)NC2CCC2NC(C2CN(S(=O)(=O)CC)C2)=O)(COC)CCCCO1 22809,C1(C)(CC)CC(NC(c2cc(N)ccc2Cl)=O)CN1C(=O)CCC(C)SC 22810,c1(C(C(=O)NC2C(NC(c3occ(C(=O)OC)c3)=O)CC2)O)ccc(F)cc1C 22811,CC(C)CC(C(=O)NCC1CC(C)N(C(=O)COC(C)C)C1)C(N)=O 22812,C(=O)(CC(C)c1ccncc1)N(C(C)C)CCNC(=O)CCSC(F)(F)F 22813,Cc1ccc(C(=O)NC2CN(C(C3CC(CC4CC4)C3)=O)C2)cc1Cl 22814,c1(C(=O)NC2CN(C(C(CCC)C)=O)C2)c(NC(=O)NC(C)(C)C)sc(C)c1C 22815,c1(C(=O)NC(C2CCOC2)CNC(CNC(CCC)=O)=O)scc(C)c1Cl 22816,CCCCC(F)C(=O)NC1CCN(C(=O)C(O)C(C)C)C(C)C1 22817,c1(C(N)=O)cc(C(F)(F)F)ccc1Br.C12CCCN1C(C)CC2 22818,CC1=C(C(=O)NCCN(C)C(c2cscc2Cl)=O)CCCC(C)(C)C1 22819,N1(C(C2C(C)C2)=O)CC(CNC(=O)CCc2ccnc(Br)c2)C2(CC2)C1 22820,c1(OC)cc(C(=O)Nc2cnc(F)c(C)c2)c(=O)n(C)c1 22821,c1(C(c2n(CC)nnn2)NCC(c2cccs2)C2CCC2)nc(C)c(C)[nH]1 22822,CC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C(C)C1NC(=O)C(O)CN(C)C 22823,c1(CN(c2c(C(=O)OCC)nccc2)C)oc2ccccc2c1C 22824,C(c1ccc2ccccc2n1)=CC(=O)NCC(C1CC1)NC(=O)CC1COCCO1 22825,N12CCC3CC(C3C1)C(=O)N1CCC2C1.N1(Cc2ccc(C)o2)CCCCCC1 22826,C1(C2CCC2)(C(N2CCC(CNC(c3cnns3)=O)(CO)C2)=O)CC1 22827,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22828,c1(C(=O)NCC(C)NC(=O)CCCCO)ccc2c(c1)CCN2S(C)(=O)=O 22829,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22830,C1(NC(C(C)N(C)C)=O)CCN(C(=O)CCC(C)(C)c2ccccc2)CC1O 22831,N#CC1(C(=O)NCC2(CCNC(C3CCCCO3)=O)CC2)CC2(CCC2)C1 22832,C(C)(C)(CCC(=O)N1CCCC(O)(CNC(=O)Cc2ccc(Cl)nc2)C1)OC 22833,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22834,c1(CC(=O)NCCCN(CCCNC(C2C(C)C2C)=O)C)csc(Cl)c1 22835,N1(C(c2scc(C)c2C)=O)CCCC2CN(Cc3noc4c3COCC4)CCC12 22836,C(C(CO)(CO)NC(c1ccc(-c2ccccc2)n1C)=O)NC(C(COC)C)=O 22837,CC(C(=O)N1CCC(C(C)C(=O)N(C2(CCN(C)C)CC2)C)C1)C(F)F 22838,C(C1c2ccccc2CCN1C(C1CCCN1CC)=O)NC(COCCCC)=O 22839,Cc1ccc(F)cc1Cc1nccc(C(NC2C3CCC2CNC3)=O)c1.C(CCO)N 22840,C(=O)(C(C)(O)CCN(C)C)N1C2C(CNC(Cn3c(C)ccn3)=O)C(C2)C1 22841,C1(C(N2C(CN(C(c3c(CC)non3)=O)C)CCCC2)=O)Cc2ccncc2C1 22842,c1(NC(C)=O)cc(C(F)(F)F)cc(C(C)(C)C)c1O.N12CCC(C(O)C1)C2 22843,S(=O)(=O)(c1ccc(F)c(F)c1)N1C(C(=O)NCc2ccc(C(F)F)cn2)CC2CC21 22844,Cc1cc(O)cc(C)c1CNc1c[nH]nc1C(=O)NCC1CCCCC1(F)F 22845,CC1(C#N)CCN(C(=NC2CCC2)NCCN2CC34CCCCC3(COC4)C2)CC1 22846,CCC(C)C(O)C(C)C(=O)NCC(N1CCC(CCOC)(CC)C1)=O 22847,c1(C(N2CC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)ccc2ncccc2n1 22848,c1(OCC=C)ccc(Cl)nc1C(N1CC(C)(NC(C2CC2C(C)C)=O)C1)=O 22849,N1(C(c2c(CC)cno2)=O)CC(NC(=O)C(C)NC(C)=O)C2(CC2)C1 22850,N1(C(c2ccc(CSCC)o2)=O)CC2(CNC2)C1 22851,c1(CC(N2CC(CNC(C(C)C)=O)OCC2)=O)ccc2ccncc2c1 22852,CCCC(C)(O)CNC(C1(CO)CCN(C(=O)C=CCN2CCCC2)C1)=O 22853,C1(CNC(Cc2ccn(C)n2)=O)CC2C=CC1C2.c12cn(nn1)C1CN(C1)C2CO 22854,C1(NC(c2nccc(SC(C3CCCS3)=O)n2)=O)CCN(c2nncs2)CC1 22855,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCCCF)C2CC2)cc1 22856,C=C(CNC(=O)C(C)(C)C1CCCC1)CCNC(=O)CSCCOC 22857,C(C(=O)N(C1CCN(C(C2(OC)CCCC2)=O)C1)CC)(C(C)C)SCC 22858,C1(CNC(C(CC=CCC)C)=O)CN(C(c2cc(Cl)cnn2)=O)CC1(F)F 22859,c1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)coc2c1COC2 22860,N1(C(c2cn(CC=C)nc2)=O)CC(O)CC1CNC(=O)C(C)NC(=O)NC 22861,Cc1nc2[nH]c(C(N3CCN(C(C)CNC(=O)CN4CC=CC4)CC3)=O)cc2s1 22862,N1(C(COCCCOC)=O)CCC2(CC1)CC2CN1CCCC1C(N)=O 22863,Cc1cc(N2CCC3CC3C2)ncc1S(=O)(=O)NC(c1csc(C)n1)C 22864,C1(NC(C2C(NC(CCc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 22865,N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC(O)C1 22866,c1(CC(=O)NCC(CCOCC)NC(C2CC2C(=O)OC)=O)ccc(F)cc1 22867,C1(NC(c2ncc(NC)nc2)=O)CC2CCC1N(C(C1CC1(C)C(C)C)=O)C2 22868,N1(C(C(c2cn(C)nc2)O)=O)CC=C(CCNC(c2cnc(C(N)=O)s2)=O)CC1 22869,C1(O)(CNC(COC)=O)CN(C(c2ccnn2CC(F)F)=O)C1 22870,c1(CN)ccccc1CNC(=O)CCC(=O)NCc1cccc(C(F)(F)F)c1 22871,c1(COC)cnc(OC)cc1C(=O)Oc1cc(CC(=O)OC)n(C)c1 22872,c1(C(=O)NC2C(C)N(c3ccnc(Cl)n3)CCC2)nsc2ccccc12 22873,c1(OC)cncc(C(=O)NCC2(CNC(=O)C(C(C)C)SC)CC2(F)F)c1 22874,c1(C(=O)NC2(C)CC(NC(c3c(F)cccc3F)=O)C2)cc2c(s1)CCC2 22875,CC1CCC(C)N1CC(=O)NCCc1ccc(NC(N)=O)cc1 22876,c1(C(=O)NCC(CNC(c2ccsc2Br)=O)OC)cccc(F)c1F 22877,N1(CCC(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)CCCS1(=O)=O 22878,c1(C(=O)NC2CC3CC(NC(=O)CO)CC32)cc2ccccc2o1 22879,c1(OCCC)cccc(C(N2CCCCC2CCCNC(=O)C(C)(C)SC)=O)c1 22880,c1(C(=O)NCC2CC(NC(C(C)(C)NC(=O)OC)=O)C2)cc(OC)cc(Cl)c1F 22881,C1(C(N2C(CNC(c3[nH]nnc3C3CC3)=O)CC(F)C2)=O)CCC(F)(F)CC1 22882,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(C1CCN(C(=O)N(C)C)CC1)=O 22883,c1(OC)cc(F)cc(C=CC(=O)N(CCCNC(=O)C2=CCOC2)C)c1 22884,CCC(C)(CCNC(c1nocc1C)=O)NC(=O)COC1CCOCC1 22885,N1(C(C(N(C(C(C(CC)C)=O)=O)C)C2CC2)=O)CCCC(C2CC2)CC1 22886,c1(CN(C(=O)C(C2CCC2)NC(C2C=CCC2)=O)C)ncc[nH]1 22887,C(=O)(C(C(C)(C)F)NC(=O)OC(C)(C)C)N(C(C)C)C1CC1 22888,N1(C(c2c(C)nns2)=O)CCc2nc(CNC(C3CC(C)OC3=O)=O)sc2C1 22889,N1(C(CCC2CCC(=O)NC2)=O)CC2CC3CC2C1C3NC(C1CCNC1=O)=O 22890,CC(C)(O)C(C(=O)NOCC1CCCCC1)NC(c1cccnc1O)=O 22891,C(=O)(C(O)CCCC)NCC1OCCN(C(C2CC(O)(CC#C)C2)=O)C1 22892,N1(C(C(F)=CC)=O)CCC2CN(C(C3CCN(c4ccccc4)C3)=O)C2C1 22893,C1(CCNC(=O)C=CC=C(Cl)Cl)CCC(NC(=O)COc2csnc2C)C1 22894,c1(NC(C2CSCCN2C(c2ccc(O)c(O)c2O)=O)=O)cc2ccccn2c1 22895,N1(CCC(=O)NC(C(C)NC(c2cnn(C(F)(F)F)c2)=O)CO)CCNC(=O)C1 22896,C(CCCOC)(C(=O)NCC1CCCN(C(C)C)C1)NC(c1ccc(CC)o1)=O 22897,c1(CNc2ccc(C(C)(C)NC(CC(=O)OC)=O)cc2)ccc2c(c1)OCCO2 22898,C1(OC)CN2CCCC2(C(=O)NC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 22899,N1(C(C2(C(C)(F)F)CC2)=O)CC2CN(C(C3CCC(C)CC3)=O)CCC12 22900,C(CO)(C(=O)NCCOCCC(=O)NCC1CCOC1)OC 22901,N1(C(CCN(C(C2CCC2CCC(=O)N2CCCC2)=O)CCO)=O)CC(F)(F)C(F)(F)C1 22902,C#Cc1ccc(C(=O)NCC2CCN2C(C2CNC(=O)N2)=O)cc1F 22903,CC1CCC=C1C(=O)NCC1(C(=O)NC2CCCC(C=C)C2)CC12CCC2 22904,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2(C)C)=O)c1C 22905,C1(CC)(NC(c2ccnc(C(F)F)c2)=O)CCCN(C(C2(C)CCCCO2)=O)C1 22906,C1(O)(CC(N)=O)CCN(C(c2ccc(O)cc2)C(=O)Nc2ccccc2Cl)CC1 22907,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 22908,C1(CN(C(CC(=O)OCC)=O)C)CN(C(C2(C)CCN(C)C2)=O)CCO1 22909,c1(C(=O)NCc2cn(C3CCN(C(C(C)=CC4CC4)=O)C3)nn2)ccccc1C 22910,Cc1cc(OCCn2cc(CC(c3ccc(F)cc3)O)nn2)ncc1[N+](=O)[O-] 22911,S(=O)(=O)(c1ccccc1Cl)NCC(=O)NCCN(C)C(c1ccns1)=O 22912,c1(C(N2CCN(CC(C)OC)CC2)=O)csc2nccn12.N12CCCC(C1)C2=O 22913,S(=O)(=O)(c1cccc(=NCC(C)n2cccn2)[nH]1)NCC(COC)O 22914,N1(C(C2CCC(=C)CC2)=O)CCC(N=c2nc[nH]n3cc(Br)cc23)CC1C 22915,C1(OC)CC(C(=O)OC(C)(C)CCCNC(=O)Cc2ccccc2)CC1OCC 22916,C1(c2cccc(C)c2)CN(c2ccnc(N3CC(C(F)(F)F)C(F)C3)n2)CCN1C 22917,C1(CC)CCC(C(=O)OC)CC1.c12nc(sc1Br)NC2C 22918,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)C)c3)=O)CC2C1 22919,c1(C(=O)NCC2OCCCN(C(C(C)C)=O)C2)ccc2c(c1)C(=O)NCCO2 22920,C=CC(CCC)CC(=O)NC1CCC(C)N(C(c2cc(O)nc(O)c2)=O)C1 22921,C(=O)(CC(C)C(C)(C)C)NCCN(C(C(CC)CC)=O)CC1CC1 22922,C(CO)(C(F)(F)F)NC(C(Cc1cc[nH]n1)NC(=O)CCn1cncn1)=O 22923,N1(C(C=C(C)c2cccs2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 22924,C1(C(N2C(CCNC(c3nc(C4CC4)cs3)=O)CCC2)=O)CCC2(CCC2)C1 22925,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 22926,c1(N(C(=O)CNCCC#N)C)nc(Br)ccc1Cl 22927,N1(C(CC(C(C)C)O)=O)CC(C)(C(=O)NCCOCCN(C)C)CC1(C)C 22928,C#CCCCCC(=O)NCC(CC(=O)NCC(CC(=O)OC)CO)C1CCC1 22929,N1(C(CC)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)CC1CC1CC1 22930,Nc1ccc(OCC(=O)OCC(COC)=O)cc1Cl 22931,CN1CCCC1C=CC(=O)NCc1nc(C2CC2)n(C)n1 22932,C1(C(=O)NC(C2CCN(C(=O)C(F)CC3CCOCC3)C2)C)CC(F)C(=O)N1 22933,c1(C(=O)NCCCN(c2cnc(C3(C)CC3)s2)C2CC2)ccc(C2CC2)cc1F 22934,C1(C2CCC2)CCOCC1.c12nnc(o1)[nH]c2=O.CC1CN1 22935,c1(COC)cc(C(=O)NC2CN(C(C3(SC)CCCOC3)=O)CC2OC)n(C)c1 22936,C1(C(C)NC(c2cnsc2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)C1 22937,N1(C(C(CC)O)=O)CCN(C)CC1C(N1CC(CC)(CO)C1)=O 22938,CN1CC(NC(C2COCCC2NC(c2cccc(F)c2N)=O)=O)CC(O)C1 22939,c1(CNC(=O)NCC(CC#C)O)cccc(Br)c1CC 22940,c1(C(=O)NC(C(CO)NC(C(CC)NC(N)=O)=O)C)cc(F)c2nc(C)cn2c1 22941,c1(CC(=O)NC(C(C)NC(C2(c3ccncc3)CC2)=O)(C)C)ncc(F)cn1 22942,Cc1ccc(C(=O)NC2CC(C)N(C(=O)C=Cc3cnc[nH]3)C2)c(Cl)n1 22943,c1(C(N2CC3(OCC(NC(C4CC4(F)F)=O)C3)C2)=O)cc(Cl)cc2ccncc12 22944,N1(C(CCCOC(C)(C)C)=O)CC2(CC(NC(c3csc4cncn34)=O)C2)C1 22945,C1(N(C(C2C(OCC)C2)=O)CC)CCN(C(=O)Cc2cccc(F)c2)CC1 22946,N1(C(COC(C)C)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 22947,CN1CC2C(CCN2C(C2CCCN(C(C3CNC(=O)C3)=O)C2)=O)CC1=O 22948,C(CCC(=O)NCCC1CC(C(=O)NC(C)(CO)C2CCC2)C1)OC 22949,Cc1ccc(C(O)CNC2(c3cnn(C)c3)CCC2)nc1 22950,c1(C(=O)NCC(C)(C2CCC2)NC(C2=CCCC2C)=O)ccc2nn[nH]c2n1 22951,c1(Nc2scc(-c3c(C(=O)NCC(=C)C)cccc3)n2)ncc(F)nc1Cl 22952,n1(C(C)C)cc(N(CCCN(C(=O)Nc2ccsc2)C)C2CC2)nn1 22953,N1(C(c2n(CCOC)ncc2)=O)CCCN(C(=O)CCC=CC(C)C)C(C)C1 22954,C1(NC(c2c(CC)c[nH]n2)=O)CC2CCC1CN(C(=O)CC(C)C(C)C)C2 22955,c1(C(N2CC(CN(C(=O)C(c3ccc(O)cc3)=O)C)C2)=O)coc(S(C)(=O)=O)c1 22956,C1(C(=O)NCCN(C(Cc2c(C)non2)=O)CC2CC2)CCC2(CC2)C1 22957,C1(NC(COCCCC)=O)CC2(C1)CC2NC(C1C=CC=CC=C1)=O 22958,N1(C(C2COC(=O)O2)=O)C(CNC(C2(Br)CC2)=O)CC2COCC12 22959,C1(CNc2cccc(C(F)(F)F)c2)CCC2(CCCC2)CC1 22960,N1(C(c2cnc(C(C)(C)C)nc2)=O)CC(NC(C2CCCC2O)=O)CC(F)C1 22961,N1(C(c2c(C)ccnn2)=O)C2CCCC1CN(C(c1cnc(O)cc1O)=O)C2 22962,CCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)C=Cc1ccncn1 22963,c1(CCC)c(C(N2CCCC(CNC(C3CCCN3CC)=O)C2)=O)nnn1CC 22964,C(=O)(C(CNC(=O)Cc1ccsc1C)CC(C)C)NCc1cc(C)no1 22965,C(=O)(CCC(C)(C)C)N(CCOCCCN(C(C(C)N(CC#C)C)=O)C)C 22966,c1(C(N2CCc3nn(C)cc3C2)C(=O)NCCSCC)ccc2c(c1)n(C)c(=O)n2C 22967,c1(C(C)NC(c2occc2CNC(C2C=CCCC2)=O)=O)ccc2n[nH]cc2c1 22968,c12ncccc1C(=O)NC(C)CCN2.c1(CC(N2CCCC2)=O)csnn1 22969,n1(CC)c(C)cc(C(=O)N(C2CC(NC(=O)C(F)C(C)C)C2)C)c1C 22970,C1(CCNC(=O)NC(C)CN2CCOCC2)CCCS1(=O)=O 22971,c1(C(C)(C)C)nc(=NC2CCN(C(=O)C(c3ccc(Cl)cc3)(C)C)C2)s[nH]1 22972,CC(O)C(C)(C)C(=O)NCC1CN(C(C2(CC(C)=O)CCCC2)=O)CC12CC2 22973,C1(F)(C(=O)NC23CC(CNC(C(CC)COC)=O)(OC2)C3)CCC(F)(F)CC1 22974,c1(C(=O)NCC(CN(C(C(CC)SC)=O)C)O)[nH]c(=N)sc1C(F)(F)F 22975,C(=O)(C#CC1CCCCO1)N(CC(C)(C)NC(=O)COCC1CCOC1)C 22976,C1(C(C)CNC(=O)CC#N)CCN(C(c2c[nH]nc2-c2cccc(Cl)c2)=O)CC1 22977,C#CCC(C)(CC)C(=O)NCCN(CCOC)C(c1cc(C)[nH]n1)=O 22978,CCC(CCOC)C(=O)NC12CCC(C1)N(C(c1sc(F)cc1Cl)=O)C2 22979,c1(C(=O)NC(CNC(c2cn(CC)nc2C)=O)C)[nH]c2ccccc2c1COC 22980,N1(C(=O)NC(c2n(C)nc(Br)n2)C2CC2)CCNC(=O)C1c1ccccc1Cl 22981,N1(C(c2ncc(C)c(C)c2)=O)CC(NC(=O)CC2CCCCN2C)C2(CCC2)C1 22982,N1(C(c2cn(CCC)nn2)=O)CC2(NC(=O)C(c3ccc(F)cc3)F)CC1C2 22983,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 22984,C1(OCc2cn(CCCN(C(Cc3ncc(C)o3)=O)C3CC3)nn2)CCCCCC1 22985,Cc1cccc(C(N2CCOCC2CC(=O)NCC2(CO)CC23CCC3)=O)c1F 22986,C1(NC(C(=O)Nc2ccc(COC)s2)=O)CC2(CCC2)C1OC 22987,Cc1ccc(C(C)NC(=O)C(=O)N(C)C(c2ccccc2)C2CC2)cc1 22988,C1(C(=O)NCS(C)=O)C2CC1N(C(c1ccnc(C(=O)NC(C)(C)C)c1)=O)C2 22989,C1(NC(C=C(CC)C)=O)CN(C(=O)CNS(N)(=O)=O)CC1C 22990,C1(Cn2cc(C(C(C)C)O)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 22991,C1(C(=O)NCC2N(C(c3n(C)nc(O)c3)=O)CC=C2)CCC(C)(C)CC1 22992,C1(CC#N)CN(C(c2sccc2Cl)=O)CCN1Cc1ccc(Cl)nc1 22993,c1(C(N2CCC(O)(C(C)NC(C3CC3C)=O)C2)=O)cc2cc[nH]c(=O)c2s1 22994,c1(C(N2CCCC(NC(C3N(C)CCC3)=O)CCC2)=O)ccc2c(c1)CCCO2 22995,c1(C(C(=O)N(C(CNC(Cc2c(OC)cccc2)=O)C)C)C)cc(C)cc(F)c1 22996,c1(C(=O)NCC2C(C)CN(C(c3ccncn3)=O)CC2)ccc(Cl)c(F)c1N 22997,C1(CC)C(NC(c2cnn(C)c2Cl)=O)CCN1C(c1cnn(C2CCC2)c1C)=O 22998,C1(CC)(NC(=O)CCOCS(C)(=O)=O)CCN(C(=O)CC2CCOC2)CC1 22999,c1(NCc2ccc(C(=O)O)cc2)ccc2nn(C(c3nc(C)[nH]n3)C)cc2c1 23000,Cc1cc(C(=O)NC(C)CCN(C(=O)Cc2c(C)cccc2C)C)cc(C(F)F)c1 23001,C(C(=O)N1CCC(F)(NC(=O)CONC(=O)OC)C1)(C(C)C)SCC 23002,C(C(CCCC)NC(=O)C(C(C)C)SCC(CC)CC)NC(C(C#C)(C)C)=O 23003,CC(C)CCC(O)C(=O)NC1CCN(C(=O)CC2(O)CCCCC2)CC1F 23004,N1CC=C(C(C)(C)C=O)C1.N1(CC)CCOC(SCCCOCCC(C)C)C1 23005,c1(C(N2CC(C)(CC(=O)NCCSC(C)C#N)C2)=O)cc2c(cc1Br)OCCO2 23006,c1(C(N2CC3C(C(=O)NCc4cn(CCC)nc4)(C3)C2)=O)cc(I)ccc1O 23007,c12ccc(cc1)S(=O)(=O)N2.N1(C(=O)CCCF)CCCC(F)CC1 23008,C(CCC(CCC)NC(C1CC2(CC(=O)N2)C1)=O)NC(c1c(C#C)c[nH]n1)=O 23009,N1(C(C(c2cnn(C)c2)C)=O)CCOC(CNC(C2COCC2C(F)F)=O)C1 23010,C(=O)(C(F)(F)CC(C)C)N1C2CN(C(C(C(=O)OCC)CC)=O)C(C2)C1 23011,C1(C2CC2)(NC(c2c(C)cc(CC)o2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1 23012,CC1(CNC(S(=O)(=O)CC2CCC(C(F)(F)F)CC2)=O)CCCC1O 23013,c1(C(=O)NC2CN(C(C(c3c(C)cncc3)C)=O)CC2C)c(Cl)cccc1[N+](=O)[O-] 23014,c1(N(CC(Cl)Cl)C)nc(=NCC(C(F)F)N2CCOCC2)[nH]c2c1COCC2 23015,C1(CCNC(c2c[nH]nc2-c2cccc(Br)c2)=O)CCCCN1C(=O)C(F)F 23016,c1(C(N2C(CCCNC(C=CC=CC)=O)CCC2)=O)cnn(CC)c1N 23017,c1(NCC(=O)NCC(CC)NC(=O)CCC2CCCO2)cc(OC)ncn1 23018,C1(CNC(CCN(C(CCC)C)C)=O)CN(C(=O)CCCC(N)=O)CC1(C)C 23019,N1(C(C=C(C)C)=O)CCN(C(C2C3CCC2CC3)=O)CC1c1cccc(Cl)c1 23020,c1(C(=O)NCC2CCCN(C(CC(C)C3CC3)=O)CC2)nc2ccccn2c1F 23021,c1(C(=O)NCC2CCN(C(C3C(C)OCCC3)=O)C2)nccc2cccnc12 23022,C(CNC(=O)C=Cc1ncc[nH]1)(CCCC)NC(C1(CC#C)CCCO1)=O 23023,C1(CC(=O)N(C(c2ccccc2)C)CCSc2ccccc2)CCNCC1 23024,CC1CCCN(C(=O)Cc2cnc[nH]2)C1CCNC(=O)CCc1cncc(O)c1 23025,C#CCCCCC(=O)NC1CC2(C1)CC2NC(C1CC1c1ccc(Cl)cc1)=O 23026,CCCC(CC(C)C)C(=O)N1CCC(N(C(c2nocc2CC)=O)CC)CC1 23027,N12CC(C(=O)O)(CC1C)NC(=O)C2C(C1CC1)OCC.C1(S)CCOCC1 23028,CC1=C(C)C(C(=O)NCc2cnc(C(F)(F)F)s2)CCC1 23029,c1(CN(C)Cc2c(C)nsc2)nccc(C(C)(F)F)n1 23030,C12(C(N3CCC(N(C(c4c(C)cc(SC)o4)=O)C)C3)=O)CCC(CC1)C2(C)C 23031,C1(CC(=O)OC)(C(CNC(=O)C(O)CN2CCCCC2)OC)CCCCC1 23032,c1(COCC)c(C)ccc(C)c1C.C1C(C(=O)NC2CC2)n2cc(nn2)CN1C 23033,c1(CN(C)C)ccc(C(N2CCCC(CN(C)C(c3ccc(Cl)[nH]3)=O)C2)=O)cc1 23034,C(=O)(C1=CC2(CCN(C(=O)CC3(CSCC)CC3)C2)C1)NCC(CC)C 23035,N1(C(C23OC(C)C(CC2)C3)=O)CCN(C(c2csc(O)n2)=O)CC(CO)C1 23036,c1(OCC(=O)NCC2N(C(CCC(C)SC)=O)CC=C2)c(C(C)C)cccc1F 23037,Cc1ccc([N+](=O)[O-])c(C(=O)NC2(CNc3ncc(F)cn3)CCC2)c1 23038,C1(NC(C2CC(=C)C2)=O)CN(C(c2nc(C(C)(C)C)cs2)=O)CC1F 23039,C1(C)(C(=O)NC2CCCC(NC(c3c(C)occ3)=O)C2)CCN(C)C1=O 23040,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C#N)C2CC2)CC1 23041,C1(CC(=O)N(CCC(=O)N(C2CC2)CC2N(CC)CCC2)C)CCCC(=O)N1 23042,CCC(C)C(C(=O)N(C1(c2cccc(Cl)c2)CC1)CC)NC(=O)COC.C(C)(=O)OC 23043,C(C(F)(F)CCC(=O)N(C)C(C)C1CC1)n1cc(C(C)(C)OC)nn1 23044,c1(C(=O)NC2(CNC(C3(OC)CCOCC3)=O)CCOC2)cc2ncccc2o1 23045,C(=O)(CCC#Cc1ccccc1)N1C(C)C(NC(=O)CCc2nc[nH]n2)CCC1 23046,C1(CNC(C2CC(=O)NCC2)=O)CCCCN(C(=O)CCn2cnnn2)CC1 23047,C1(C(=O)NCC(F)CNC(c2sccc2C2CC2)=O)(COC)CC=CCC1 23048,CC1Oc2ccc(CNC3CCCC3OCc3csc4ccccc34)cc2NC1=O 23049,N1(CC(=O)NCC2C=CCCC2)CCN(C(=O)CCc2ccccc2)CC1 23050,Cc1c(C(=O)NC(Cc2ccco2)C(=O)NCCC(O)CCO)cccc1O 23051,CCCCCC(CC)C(=O)N1C2CCC(C2)C1C(=O)N(CCC(C)C)CCO 23052,C1(C)(C(=O)NC(c2cnccn2)C)CCCN1C(=O)CCN(C)C 23053,C#Cc1cccnc1NC(=O)C(=O)N(C)CCO 23054,c1(Cn2c(C3(NC(C(F)(F)C4C(C)C4)=O)CCSC3)nnn2)ccc(F)cc1 23055,C(=O)(C(O)CNC(=O)CC1CCCCC1)N1CC(CCOC)C1 23056,N1(C(CCSc2nc(C)sc2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23057,CCCCC(O)CCC(=O)N(CCCCN(C)C(c1ccc2nc[nH]c2c1)=O)C 23058,C1(C(=O)NC2(CCN)CCC2)CCN(C(=O)CN2CC(C)(C)C2)CC1.CSC 23059,N(C1CCc2c(Br)cccc21)C(=O)CC1CCCN1C(c1cccc2nc[nH]c12)=O 23060,C1(C(N2CCC(C(=O)Nc3ccc(CC)c(Br)c3)CC2)=O)Cc2ccccc2C1 23061,c1(CNC(C)=O)cccc(C(=O)N(C)C(c2cnn(Cc3nc(C)no3)c2)C)c1 23062,C1(c2[nH]c(NN3CCC4CCCCC4C3)nc(=N)n2)CC2(CCO1)CC(F)(F)C2 23063,c1(CN(C)Cc2ccncc2)ccc(F)cc1.c12nnc(o1)c(=O)[nH]2 23064,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23065,CC1CCCC(C(=O)NCCC2CCN(C(C3OCCC3C(F)(F)F)=O)CC2)C1 23066,N1(C(C(=O)NCC=C)CC2CCCCC2)CCC2(CC1)CC2c1ccc(F)cc1 23067,C1(CNC(=O)Cc2cncs2)CCC2(CCN(C(=O)CC3CCOC3)CC2)O1 23068,C1(NC(c2cnn(CC)c2Br)=O)CCC2(CC1)CC2NC(=O)CC(C)C 23069,c1(CCNC(c2n(C)nc(CC)c2C)=O)cnc2cccnn12 23070,S(=O)(=O)(c1c(C)sc(C)c1C(=O)OCC)N(CCCCC)C.C(COC)S 23071,C1(COC)CCCCN1C(C1CC2CC2N1C(C1CCCCCC1)=O)=O 23072,N1(CC)CCC(NC(=O)C(CC2CCC2)NC(C2CC2Cl)=O)C(C)C1 23073,O=C1CC(N2CCN(CC3CCN(C(=O)Cc4cccnc4F)C3)CC2)CCN1 23074,O(NC(=O)C(F)C1(O)CN(C(=O)CC2CCC(=O)CC2)C1)CC(=C)Cl 23075,CC(CC(=O)NCC1(F)CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23076,C1(NC(C(C2CCOC2)NC(Cc2n(C)ncc2)=O)=O)CC(O)C(O)C1 23077,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23078,C(=O)(C(CC)CCCCC)N1CC(NC(CC2(C(=C)F)CCC2)=O)C(C)CCC1 23079,Cc1c(C(N2CCC(=O)CC2)C(=O)NC(C)C)cccc1Br 23080,c1(C(=O)NCCC(=C)CNC(c2ccc(OC)cc2O)=O)cccc2nsnc12 23081,c1(CC(N2CCC(C)(CNCCC(C)(O)C3CC3)C2)=O)ccc([N+](=O)[O-])cc1 23082,c1(C(N2C(CNC(C(N3CCC(O)CC3)C)=O)CCC2)=O)cnn2ncccc12 23083,C(=O)(C1Cc2ccc(F)cc21)N1CC2(CN(C(CS(CC(=O)OC)(=O)=O)=O)C2)C1 23084,N1(CCC)C=C(C(=O)N=c2scc(Br)n2-c2cnn3c2OCC(O)C3O)SCC1 23085,Cc1cc(CNC(=O)NC(C2CC2c2ccccc2)C)cnc1Br 23086,c1(C(=O)NCC=CCNC(CC(C)c2ccccc2)=O)ccn2ncnc2c1 23087,C(=O)(C1=NOC(C2CN(C(C3CC=C(C)CC3)=O)C2)C1)NCC(NOC)=O 23088,N1(C(C2CC(SC)C2)=O)CCN(C)C(CNC(=O)C(F)F)C1 23089,c1(C(N2C(CNC(C(C)Cc3cnn(C)c3)=O)C=CC2)=O)c(Br)nnn1C 23090,C(=O)(C1=CC2C=CC1C2)N1CCCC(C2N(C(C3=CCCC3C)=O)CCCC2)C1 23091,CCCC(CCC)C(=O)NC(CCC1CC1)C(=O)NCC(CC)C(C)(F)F 23092,Cc1ncncc1C(N1CC(NC(C2CCCCC2)=O)C(C)C1)=O 23093,C1(C(C2(C)CC2)NC(CN2CCN(C(C(=O)OC)C)CC2)=O)CC2CCC1CC2 23094,c1(CN2CCCC(NC(C3N(C(N(C)C)=O)CSC3)=O)C2)ccc2cnccc2c1 23095,C1(NC(c2n(CCCOC)nnn2)CC2CCC2)CC(=O)N(C)C1=O 23096,Cc1ccc2ccc(C(=O)NC3CN(C(C4(C)CCCO4)=O)CC3C)nc2c1 23097,N1(C(=O)Nc2cccc3c([N+](=O)[O-])cccc23)CC=C(c2cccc3ccccc23)CC1 23098,C(CN=c1cc(C)nc(-c2ccccc2)[nH]1)N(C(C(=O)NCC)=O)CC 23099,c1(CC(=O)NC(Cn2cc(C3(C)CCCO3)nn2)CC2CC2)c(F)cccc1Br 23100,N1(C(CCSCCCC)=O)C(C(=O)NCCc2ccccc2C)CCC1C(C)C 23101,CC(C)C(C(=O)N1CCN(C)CC1)C(C)NC(c1ccn(C)n1)=O 23102,C(=O)(C(F)CC(C)C)NC(CC)(C)CCNC(=O)C(=O)NN(C)C 23103,c1(C(N2CCC3(CCCN3C(=O)C(F)C3CC3)C2)=O)ccc([N+](=O)[O-])cc1O 23104,C(C1=CCCNC1)CNC(c1cc(-c2ccc(CO)cc2)[nH]n1)=O 23105,C1(C(N2CC(NC(=O)NCC(C=C)O)C2)=O)CC(=O)N(c2ccccc2)C1 23106,CC1ON=C(C(=O)N2CC(NC(=O)Cc3nccn3C)C(O)C2)C1C 23107,C1(CN(C(c2cnn[nH]2)=O)CC)CCCN1C(=O)C(C#N)=CC1CC1 23108,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(C)N(c2nc(C)nc(Cl)c2C)CC1C 23109,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23110,N1(C(C=CC(CC)NC(=O)C(C)CN2CCCCC2)=O)CC2(COC(C)C2)C1 23111,c1(C(=O)NC(C)CCNC(c2c[nH]nc2-c2ccc(Cl)s2)=O)nnc(S)n1C 23112,N1(C(c2c(C(C)C)scn2)=O)CCc2ccccc2C1CNC(C1CSC1)=O 23113,N1(C(c2ccc(CC)c(F)c2)=O)CC2CCCC2(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1 23114,c1(CC)ccccc1COc1nc(CCCOC)nn1-c1ccccc1C 23115,c1(NC(C(CC)(C)CNC(=O)C(C)NC=O)=O)cnc2ccnn2c1 23116,C(=O)(C1=CCCCCC1)NC1CC(C(=O)NCC(C(=O)OC)C)OCC1 23117,N1(C(c2c(C)cc(F)s2)=O)CCCC2(CCCN2C(c2cncs2)=O)C1 23118,N1(C(=O)NC2CCCN(SC(C)=NOCCc3ccccc3)C2)CC[Si](C)(C)CC1 23119,c1(CCCCOC(C)=O)c(-c2cncc(CC3CCCO3)c2)ncn1C 23120,Cc1ccccc1C(C)CC(=O)N1CCC(C(=O)NCCOCC(C)C)C1 23121,CC1=C(C(=O)NC2CC3(C2)CN(Cc2ccc(COC)cc2)C3)CCC1 23122,c1(C(N2CCC(N(C(C3CC3C)=O)CC)CC2)=O)ccc(S(C)(=O)=O)cn1 23123,C1(CNC(c2nccn3ccnc23)=O)CCN(C(=O)CSC2CCC2)CC1(F)F 23124,S(=O)(=O)(c1cccnc1NCC(CO)C(F)(F)F)NCCN1C(=O)NCC1 23125,N1(C(CN(C)Cc2ccc(C)cc2)=O)CC2CC(NC(C3(O)CCC3)=O)C1C2 23126,c1(CC(=O)NC(CNC(C(C)OCCOCC)=O)CO)cc(C)no1 23127,Cn1nc(CC(=O)Nc2ncccc2-c2noc(CCCO)n2)c2c1CCCC2 23128,c1(N2CC(NC(c3nc(Cl)ccc3F)=O)(CO)C2)ncc([N+](=O)[O-])cc1Br 23129,C(=O)(C1=C(C#N)CCC1)N(C1CCN(C(c2cc(C3CC3)sn2)=O)C1)C 23130,N1(C(C=CCOCCOC)=O)CCC2(NC(C3CN(C)C3)=O)CCCCCC12 23131,C(=O)(CC(C)CN(C=O)Cc1nc(C2CCOC2)n[nH]1)NC 23132,N1(C(C=C(C)Cl)=O)CCC2(CCCCC2NC(=O)CCCCCF)C1 23133,CCC(CC(F)(F)F)C(=O)N1CC2(CNC(C3CCC(C)CC3)=O)CC1CO2 23134,c1(C(=O)NCCN(C(=O)CC2CCCC23CC3)C(C)C)ccc(C(F)(F)F)cn1 23135,c1(C(N(CC(C)(C)CNC(=O)CCC2CCOC2)CC)=O)cc2sc(C)cc2[nH]1 23136,N1(C(CCCC(=O)N(C)C)=O)CC2CCC1CN2C(c1ncccc1Cl)=O 23137,CC1(C)CCC(C(=O)NC2CC(NC(=O)C(F)(F)c3ccncc3)C2)OC1 23138,N1(C(C(Cn2cncn2)NC(c2nc(COC)oc2)=O)=O)CCc2ncsc2C1 23139,c1(C(=O)NCC2CC2C(=O)Nc2cncc(Cl)c2)ccnc(O)c1 23140,O=C(C1CCCn2nccc21)N1CCCC(O)(C(=O)Nc2cc(Br)ccc2F)C1 23141,C1(OC)CC(NC(N2CC(CCOCc3ccoc3)C2)=O)C(C(F)(F)F)C1 23142,C(C(=O)N=S(C)(C)=O)N1CC(n2cc(CCN(C)C)nn2)C(c2cccnc2)C1 23143,C#CCCCC(C)C(=O)NC1CCC(NC(c2ncn(C)n2)=O)C1 23144,CCS(=O)(=O)CC(=O)N1CCC(N(CCNc2ccncc2)CC2CC2)C1 23145,N1(NC(C(c2cc(OC)on2)OCCC(C)C)=O)CCN(CC(=O)C(C)C)CC1 23146,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CC2)cc2nn[nH]c2cc1F 23147,C1(C(N2CCCC(NC(c3[nH]cc(C)c3)=O)C2C)=O)CCOC2(CCCC2)C1 23148,Cc1nnc2n1CC(C(N1CCCCC(NC(c3ccc(Cl)c(F)c3)=O)C1)=O)C2 23149,c1(C(Cn2cc(CC3CN(C)C3)nn2)O)ccc(F)cc1.N12CCCC1CC2=O 23150,C1(CN(C(=O)C=CI)C)COCCN1C(=O)Cn1cnnc1O 23151,N1(C(C2(C#C)CC2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23152,C(=O)(C(O)CC(N)=O)NCCCOCCC(N1CCC(=CC#C)CC1)=O 23153,C(=O)(CCC(C)NC(=O)CC1CC2(CC2)CO1)NCc1c(C)ncs1 23154,C(C(CNC(c1scnc1C)c1nnnn1C1COC1)C(C)C)OCC.C1(C)CC1 23155,c1(NCC2(C(=O)NCC(C)CN(C)C)CC2)cc(O)nc(=O)n1C 23156,N1(C(C(c2ccc(C)o2)C)=O)CC(NC(c2onc(C)c2C)=O)CC(F)C1 23157,C1(CC)(CO)CCCN(C(C2OCCC2NC(=O)CC2COCCN2C)=O)C1 23158,CC(C)CCC(C(=O)N(C1CCCCC1)CCCO)NC(c1csc(Cl)n1)=O 23159,N1(C(CC(C)C)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC2(C)CCCC12 23160,C1(NC(c2cccc(C(=O)NC)n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1(C)C 23161,C1(NC(CC=CCC)=O)CCN(C(c2cc(OC)cc(C)c2)=O)CC1C 23162,N1(C(C)=O)CCC(C)(C(=O)N(C(C)CO)CCN(C)C)C1 23163,CC1CCn2nc(C(=O)NC3(C)CCN(C(=O)C(c4cncn4C)O)C3)n2C1 23164,N1(C(C(N2CC(C)C2)C)=O)CC(CNC(=O)CC2CC(C)(C)CO2)C(F)C1 23165,c1(C(=O)NC(C)CNC(c2n[nH]c3c2COC3)=O)cn2c(Br)cnc2s1 23166,N1(C(C(CC)N(C)C)=O)CCCC(C)(CNC(=O)CCc2cnco2)C1 23167,N(C1CCCc2ccc(F)cc21)CC(CC)c1nn[nH]n1 23168,c1(CCN2CCS(=O)(=O)N3CC2C3)nccc(=NCC2CCCOC2)[nH]1.NN=O 23169,CC1OC2(C(N3CCC3CNC(C3CC(C#N)(N(C)C)C3)=O)=O)CCC1CC2 23170,N1(C(c2cc(C)c(F)cn2)=O)CC2CCCC2(C(=O)NCC2(F)CCOCC2)C1 23171,N#CC1CN(C(c2cocn2)=O)CCN1C(=O)Cc1c(F)cc(F)cc1F 23172,C1(CC)CN(C(C2CCCC2F)=O)CC1C(=O)NC1CCCC1COC 23173,C1(C(=O)NCCN(C(CC(C=C)(C)C)=O)CCC)CC12CCC1(CC1)CC2 23174,N1(c2nccc(-n3cc(C(N)=O)nn3)c2)CC(C2CC2)OCC12CCCCC2 23175,C(=O)(C1=C(c2ccccc2)CCC1)NC1CCC(NC(CC(CC)C)=O)C1 23176,C1(CC(=O)NC2CCOCC2NC(c2ccnc(C)c2)=O)(COC)C=CCCC1 23177,c1(C(N2C3CN(CCCOC)CC2C3)=O)ccc(C#N)cc1Cl 23178,CC1(C)NC(=O)CC1C(=O)NC1(CNC(=O)CC2CC3CCC2O3)CC1 23179,c1(OC)ccc(C(N2CC(CC(=O)NCc3sc(Br)nc3C)C2)=O)c(OC)c1 23180,C1(C(=O)NC(C2CN(C(c3cc(F)n(C)n3)=O)C2)C)CCCCN1N=O 23181,N1(C(C(C)OCC)=O)CC2CCC1C2NC(c1nn(C)c(Br)c1C)=O 23182,N1(CCc2cn(Cc3c(C(=O)NCCC(F)(F)F)con3)nn2)C(=O)CNC1=O 23183,Cc1nccc(C(=O)NCCC2(C(=O)N(C3(CCO)CC3)C)CC2)c1N 23184,C#CCCCCC(=O)NC1(CNC(=O)C=Cc2cc(Br)cs2)CCCC1 23185,C(=O)(C(F)C(=O)N1CC(F)CC1CNC(=O)COCCCN=[N+]=[N-])OCC 23186,C(=O)(C1=C(C)CCN(c2cc(N(CCCCO)C)nc(C(C)C)n2)C1)OC 23187,O=C(C#CC1CCCCC1)NCC1CN(C(=O)C=CCN2CCCC2)CC12CC2 23188,O=C(N=c1[nH]nc2ccccn12)N1CCC(Cc2cccnc2)C1 23189,CCCS(=O)(=O)CC(=O)N1CCN(CC2CCN(C(=O)CSC(F)F)CC2)CC1 23190,Cc1cc(=NCc2cc(C3CC3)on2)[nH]c(N2CCc3ncncc3C2)n1 23191,c1(C(=O)NC(CC=C)CNC(c2ccc(CO)cc2)=O)c(F)ccc2n[nH]cc12 23192,N1(C(=O)CC2OCCCO2)CCC(C2CCCN(C(=O)C3=CCCOCC3)C2)CC1 23193,N1(C(CC(CCC)C)=O)CC2CCC(N(C)C(c3ncc(F)cc3C)=O)C2C1 23194,N=C1NC(=O)C(CC(=O)NCCC2(O)CN(C(=O)Cc3cc(C4CC4)no3)C2)S1 23195,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23196,N1(C(C(CC)c2ccccc2)=O)CCN(C2CC(NC(=O)COC(C)=O)C2)CC1 23197,C(=O)(C#CC1CCOCC1)NC(C1CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O)C 23198,C1(C)(C(N(CCNC(C2C(=C)C2)=O)Cc2ccc(Cl)nc2)=O)CC(OC)CN1C 23199,c1(CC)cccc(C(N2CCCC2CN(C(=O)Cc2cc(O)ncn2)C)=O)c1C 23200,C1(NC(COc2ccc(C)c(C)c2)=O)CC2(CCN(C(=O)CCC(N)=O)C2)C1 23201,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23202,N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(NC(c2ncoc2C)=O)C1C 23203,C1(CNC(c2c(C)[nH]cc2)=O)CN2CCCCC2CN1C(c1ccoc1Cl)=O 23204,c1(C(=O)NCC(c2cccc(C)c2)NC(C2C3CC3C3CC23)=O)cc(O)nc(Cl)c1 23205,c1(CNC(COC)=O)cc2n(n1)CCN(C(=O)C(NS(=O)(=O)C1CC1)SC)C2 23206,N1(C(C(=O)NCC2C(C)C2)C2CCCO2)CCCC(C2CCC2)C1 23207,c1(C(=O)NC2CC(F)(CNC(=O)CCc3ccc[nH]3)C2)cccc(C(F)F)c1 23208,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23209,CCCC(CNC(=O)CC1CCN(C(=O)C(C2CC2)OC)C1(C)C)CCO 23210,C(=O)(CCCCC(C)(C)C)N(C1CCN(C(C23CC(C)(CCO2)C3)=O)C1)C 23211,C(CCC(=O)N1CC(O)(CN(C(=O)C(F)CC2CCCC2)CC)C1)=CCC=C 23212,N1(C(C(CCC#C)O)=O)CCC(CCNC(c2[nH]c(C)nc2C)=O)C(F)(F)C1 23213,CC1CCCN1CCCn1cc(CCC2C=CCC2)nn1 23214,C=CC1(CC(=O)NC2CCC2)CN(C(C(=O)OC)C(C)CCCC)C1 23215,N(C(=NCCc1ccccc1)NCc1cc(OC)ccn1)C1C(Cl)(Cl)C1 23216,n1(CC)cc2ccc(C(=O)NCCNC(c3cccc(C(=O)OC)n3)=O)cc2n1 23217,c1(NC2CCN(C(CC3CCC(C)(C)C3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 23218,C1(C(N2CCC(CCCO)C2)=O)CC2CC2N1C(=O)C(O)c1ccsc1 23219,c1(CO)c(O)ncc2c1CCC2.C12CN(CCS1(=O)=O)CCn1cc(nn1)CC2 23220,N1(C(c2cc(CC)ncc2)=O)CC2ON=C(CNC(=O)C=CBr)C2C1 23221,c1(N(CC=C)C)ncc(C)cc1S(=O)(=O)NC1COCC12OCCO2 23222,Cc1nscc1CC(=O)N(CC(O)CN(C)C(C1CCC(CC(F)(F)F)C1)=O)C 23223,c1(N2C(C)C(NC(=O)CC3(CO)CC3)CCC2)ncc2ccnc-2[nH]1 23224,N1(C(C(N2CCN(C)CC2)C)=O)CC2CN(C(C3OCCO3)=O)CC(C1)O2 23225,c1(CC(C)C)cccc(C(=O)NC2CCC(NC(C3CC3(C)Br)=O)C2)c1 23226,CC(C(O)C(F)F)NC(=O)CC1(C)CCN(C(=O)CCSCCC#N)C1 23227,C(CCCC(=O)Nc1ccccc1OCCN1CCOCC1)(OC)OC 23228,C1(OC)CCN(C(c2cncnc2C2CC2)=O)C(C(=O)O)C1 23229,N1(C(C(C)OCCN(C)C)=O)CCC(C)(C)C1CC(=O)NC(c1cccnc1)C 23230,N1(C(COC)=O)CC2CCCC(NC(C3CCC=CCCC3)=O)(C2)C1 23231,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)ns3)=O)CC2)CC1C 23232,N1(C(C(C=C)OC)=O)CC2CCN(C(=O)C(c3cc(C)ccc3F)CCC)CC2C1 23233,c1(C(=O)NC2CN(C(c3conc3C3CC3)=O)C2)cccc2c1OCC2 23234,C(CC(C)(C)CC(=O)NC(CCF)C(=O)N(C)CCc1cc[nH]n1)OC 23235,C1(NC(c2ccc(SCCO)cc2)=O)CCCOC12CCNCC2 23236,CC1(C)CC(C(N2CC(CC(F)C(=O)NCC(CO)C(F)(F)F)C2)=O)CCO1 23237,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(O)CF)CCO1 23238,CC(C)C(C)CC(=O)N1CC(C)CCC1CNC(=O)Cc1ccccc1O 23239,c1(N2C(COC)(CO)CCC2)nccc(=NCCc2c(F)ccc(Br)c2F)[nH]1 23240,N1(C(c2cc(C(=O)OC)sc2)=O)CCCC2(NC(=O)CC=C(Cl)Cl)CCCC12 23241,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23242,c1(C2(NC(C)Cc3ccccc3N(C)C)CCC2)[nH]c(=N)c(C#N)cc1C#N 23243,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CC1CCCN1C 23244,C(=O)(C1=NNC(=O)CC1)NCC1N(C(c2nc(COC)[nH]n2)=O)CCN(C)C1 23245,C1(O)(CC(=O)NC(c2ccc(Br)cc2)C)CCN(C(=O)Cn2cccc2)CC1 23246,C1(C(=O)N(C(C)CCNC(=O)C(C(C)O)N(C)C)C)(COC)CCCCO1 23247,CC1=C(C(=O)N2CCCC(NC(c3cc(F)ccc3Cl)=O)C2C)CCC1 23248,c1(C(C(=O)NCCCCCOC)NC(c2nncn2C)=O)cccc(C(F)(F)F)c1 23249,c1(OCC)ncccc1C(=O)NCC1CC(NC(c2cnn(C(F)(F)F)c2)=O)C1 23250,C(CO)(CCCCNC(=O)C(C1CCCC1)OC)NC(C1(OC)CCSCC1)=O 23251,C(C(CNC(C1CC1(F)F)=O)C(F)(F)F)NC(c1cn(C(C)(C)C)nn1)=O 23252,c1(C(N2CC3CN(C(C=CCN(C)CC)=O)C3CC2)=O)cc(F)c(F)c(O)c1F 23253,CC1(NC(=O)CSC2CCOCC2)CCCN(C(C2CC2c2ccccc2)=O)C1 23254,c1(C(=O)NC(C2(O)CN(C(COC(CC)(C)C)=O)C2)C)cc(Br)cn1C 23255,CC1CCCCN1CCC(=O)N(CC(C)NC(=O)Cn1nnc(C(C)(C)C)n1)C 23256,c1(CCC(=O)N(C2CN(C(CN(C)Cc3ccccc3)=O)C2)C)cnc(O)[nH]1 23257,c1(OCC)cccc(C(=O)NCC2(NC3CNC(=O)N3)CCOCC2)c1[N+](=O)[O-] 23258,C=C1CC2(C1)CC(C(N1CCCC1CNC(=O)C(C(C)O)N(C)C)=O)C2 23259,C(=O)(CCCNC(C1CCOC1CNC(=O)Cc1cn(C)cn1)=O)NC 23260,c1(C(=O)NCC(C)OCc2ccc(OC)cc2C)cnc2ccccn12 23261,N1(C(C(C(C)C)CNC(C2(C)CCC3CC3C2)=O)=O)CCCOC(C)(C)C1 23262,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1cnc(Cl)s1)=O)=O 23263,C1(N(C(=O)CCc2cn[nH]c2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23264,C1(O)(CC)CCC(NC(=O)CC(C)(C)CNC(C2CCCOC2)=O)CC1 23265,N1(C(C2CCCN(CCC)C2)=O)CCC(NC(=O)CN2CCCCCC2)C(F)C1 23266,CC1CCN(C(=O)CCc2cncc(F)c2)C1CNC(=O)CSCC(F)(F)F 23267,c1(C(=O)OC)cc(C(=O)NCCCNC(c2[nH]ccc2C2CC2)=O)cs1 23268,c1(C(=O)NC2C(C(N(C)C)=O)COC2)cncc(C(F)F)c1 23269,C1(C(=O)NCC(C)(C)OCCNC(=O)Cc2ccc(Cl)cc2)CCC2CC2CC1 23270,N1(C(C(C)NC(COC)=O)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O 23271,c1(-n2c(NC(c3ccc(C)nc3)C3=CCO3)nc(CCO)n2)ccc2nc[nH]c2c1 23272,c1(C(=O)NCC(CCCC)NC(=O)CCc2ncc[nH]2)ccc(O)c(C)c1C 23273,C1(NC(CC2CCCC(C)C2)=O)COc2ccccc2N(C)C1=O 23274,n1(CCN(C)C2CC2)cc(C)nn1.C1(O)(C(=O)NN2CCCC2)CN(C(=O)COC)C1 23275,C1(CC=C)(N(CCCO)C(C2CCC2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)C1 23276,CC1(C)C(CNC(=O)CN2CC3CCC2C3)CCN1C(c1ncccc1F)=O 23277,C1(CNC(N2CCC(C3N(C(C)C)C(=O)CCC3)C2)=O)COC2(CCCC2)O1 23278,C1(C(N(CCCC)CC)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23279,C12(C(=O)NC(C3CCCC3)CNC(C(CC)CCOC)=O)CCCCC1CCCC2 23280,c1(C(=O)NC2CCCN(C(CSCCC)=O)C2C)ccn2ccnc2c1 23281,C(=O)(C(O)(C(C)C)C(F)(F)F)N1C(c2n[nH]cc2CC(C=O)C)CC(OC)C1 23282,N1(C(CSCC(=O)Nc2ncco2)=O)CCN(C(=O)C(F)C2CCC2)CC1 23283,c1(C(C(=O)NCCOCCC#C)NC(=O)COCC(C)C)cccnc1 23284,C(=O)(C(CC(F)F)N(C)C(c1cc(C)cnn1)=O)N(CCC)CC 23285,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)CN3CCC(C)(O)C3)C2)CC1 23286,c1(CCC(=O)NCC(CCOC)NC(c2c[nH]c(=N)s2)=O)cccc([N+](=O)[O-])c1 23287,N1(C(CCC2CC(C)C2)=O)CCC(NC(c2cn(CCF)nn2)=O)C12CCC2 23288,C1(NC(C2N(S(CC)(=O)=O)CCC2)=O)CN(C(c2cc[nH]n2)=O)CC1C(F)F 23289,N1(C(C(C(C)O)C)=O)CCC(C2(NC(c3ccccc3)=O)CC2)C1 23290,C1(NC(C=CC(C)(C)NC(C2CC2C(N)=O)=O)=O)CC2(C1)CC(C#N)C2 23291,C(=O)(CC(F)(F)C(F)F)N1CCC(NC(c2cc(COC)oc2C)=O)C(F)C1 23292,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)NC(Cc1c(C)ccnc1)=O 23293,C1(C(C)OC)CN(C(C2(N(C(=O)C(O)C3CCC3)C)CC2)=O)C1 23294,CC1CC(NC(c2cccn2C)=O)CN1C(C1CC1C)=O 23295,C12CCC13CCN(CC3)C(=O)CN2.Cc1cccc(NC(C)=O)c1.C1CC(=O)N1 23296,c1(NC(C2CCCN2C(=O)CN2CCOC2=O)=O)cnc2ccccc2c1Cl 23297,Nc1cncc(CNC(c2cnn[nH]2)=O)n1 23298,C1(c2onc(-c3ccc(C4(C(C)=O)CC4)cc3)n2)CS(=O)(=O)CC12CC2 23299,Cc1c[nH]c(C(N2CC(C3CCCN3C(=O)C(C)(C)n3cc(Cl)cn3)C2)=O)c1 23300,C1(NCc2onc(C)n2)CN(C(C2CC(C(=O)NS(C)(=O)=O)C2)=O)CC1F 23301,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23302,Cc1cnc2cccc(C(N3CCCOC(CNC(=O)CN(C)C(N)=O)C3)=O)n12 23303,N1(C(CC)=O)CCC(n2nc(-c3cccc(N)n3)nc2-c2c[nH]nc2C(C)C)CC1 23304,c1(C(=O)NC2CN(C(C(c3cccc(C)c3)(C)C)=O)C2)ccc(F)c2[nH]ccc12 23305,c1(C(=O)NCC(C)NC(C2CCCO2)=O)cccnc1-n1cncn1 23306,C=CCC(Cc1ccccc1)NC(=O)C(=O)Nc1ncsc1-c1ccccc1 23307,C1(C2(CNCC(C)C3CN(C(=O)CC4CCC(=O)O4)C3)CCC2)CCCCO1 23308,c1(OC)cc(OC)nc(N2CC(NC(C3(C)CCCC3)=O)CCC2C)n1 23309,N1(C(CSCCC)=O)CCC2CC(CNC(c3cc(CC)no3)=O)CCC2CC1 23310,N1(C(C2(OC)CCSC2)=O)CCC(C)C(CNC(=O)C(c2cccs2)C2CC2)C1 23311,N1(C(c2cnn(C)c(=O)c2)=O)CC(C(N2C3C=CCC2CC3)=O)CCC1(C)C 23312,CCCCC(C(=O)NCC(C)(O)CNC(=O)COc1ccsn1)N1CCCS1(=O)=O 23313,CC(F)(F)CCCC(=O)NC(CNC(C1OCC1(C)C)=O)CO 23314,C1(CC=C)CCCN(C(=O)CC(C)(C)OC2(C(=O)NC)CCOC2)C1 23315,C(=O)(CCCCCNC(c1scnc1C)=O)N(CCC(=O)OC)CC 23316,NC(=O)CCC(C(=O)NCc1ccc2occc2c1)n1cc(-c2cccs2)nn1 23317,CC1(C)CCC(C(=O)NC2CC23CCOCC3)CN1C(=O)CC(=O)NC1CC1 23318,CC(C)CCC(O)C(=O)N1CCC2CN(C(c3cccnc3)=O)CC12 23319,CC(C)(F)CCC(=O)NCC1CC(F)CN1C(=O)Cc1cccc(Cl)c1F 23320,N#Cc1ccccc1C=CC(=O)NC1(CO)CCN(C(C2(n3ccnn3)CC2)=O)C1 23321,Cc1cc(C#N)nc(NCC2CCC(NC(=O)CC3(O)CCC3)C2)n1 23322,C1(N(C(=O)C(=O)NCCC(N)=O)CC)CCN(C(=O)CCC(=O)OC)CC1 23323,CCC(CC(F)F)C(=O)NCCCCCN(C(=O)C(C(C)C)C1CCC1)C 23324,C1(NC(=O)CC2CC3CC3C2)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCCCC12 23325,c1(N(CCC)CCNC(=O)CCc2ccc(C)cc2)cc(F)cc2c1CCC2 23326,Cc1ccc(Cl)c(C(N2CC3(CCC3)CC2CNC(C2(CF)CC2)=O)=O)c1N 23327,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCCC(=O)N2C)=O)C1 23328,C(=O)(C(C)(C)c1cccnc1)NCC1C(NC(C(=O)NCCOC)=O)C1 23329,N1(C(COCCSC)=O)CCOCC(NC(=O)C(n2cnc(C#N)n2)C)C1 23330,c1(C(=O)NC(c2cccnc2)CNC(C=CC(=O)OCC)=O)nc(O)sc1C 23331,C1(N(C(C=CCC)=O)C)CCC(CNC(=O)CSc2ccncc2)CC1 23332,c1(N2CC3N(C(=O)CC4CCC5CC5C4)C(CC3)CC2)nc2ccc(F)cc2s1 23333,C1(CC(=O)N(c2cn[nH]c2)OCC)CCCN(C(=O)NC)C1 23334,CC(CC#N)C(=O)NCC1(C(NCP(C)(C)=O)=O)CCCCC1 23335,C(=O)(CC1=CCN(C)CC1)NCCC(C(N1C(C)CS(=O)(=O)CC1)=O)O 23336,N1(C2(CO)CC2)CCCN(Cc2cn(CC3CCCC3n3cccn3)nn2)CC1 23337,C1(CC)CN(C(c2ccc(-c3nnc(C)o3)cc2)C(=O)NC2CCCC2)CCO1 23338,c1(CN(C(C2CCCO2)=O)CC2CN(c3cncs3)C2)ccccc1.O=C1CN1 23339,C#CC1CN(C(=O)C(CC(=C)C)NC(C2(OC)CC2)=O)CCN1C 23340,Cc1nc2cncc(C(=O)N(C3CCN(c4cccc(Cl)c4)C3=O)C)c2[nH]1 23341,C=CC(C)(C)C(=O)Nc1cccc(CNC(=O)Cc2ccnn2C2CCCC2)c1 23342,c1(OC)c(C)cc(C(=O)NC2CCCC(N(C(=O)CSC3CC3)C)C2)cc1C 23343,N1(C(C(C)N(C)C)=O)C2CC=C(C(=O)NCCc3cccnc3)C1CC2 23344,c1(ONC(C2CC(N(C(C(C)OCCOC)=O)C)C2)=O)cc(C)ccc1C 23345,N1(C(c2cnn(C(CC)C)c2C)=O)C2CC1CN(C(c1cccnn1)=O)C2 23346,c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)cccc(Cl)c1O 23347,c1(C(N(C)CCNC(=O)CC2C=CS(=O)(=O)C2)=O)c[nH]c2ccc(Br)cc12 23348,c1(C(=O)NCC(CNC(c2cc(CC(C)C)on2)=O)OC)ccccc1C(N)=O 23349,c1(C(=O)O)cccn(O)c1=O.CC(C)COC(C)(C)C1(CO)CC1 23350,c1(C(=O)NC2C(CC)CN(C(=O)CCC3(C)CC3)C2)cc(S(N)(=O)=O)cnc1C 23351,N1(C(C(C(CC)C)OC)=O)C2CCC1CN(c1nccc(CCN(C)C)n1)CC2 23352,C(=O)(C(O)C(C)SC)N(CCNC(Cc1nnc(C)o1)=O)Cc1cccc(Cl)c1 23353,C(=O)(CC1OCCc2ccsc21)N(CCCN(C)C(C1CC2C(C1)C2(C)C)=O)C 23354,Cc1csc(C[SH]=CC(=O)NC(C)CN(C)C)n1 23355,c1(OC)cccc(C(N2CCCC(C)(C)C2)C(=O)NCc2nnn(C)n2)c1C 23356,N1(C(C(c2cccnc2)NC(c2n(C)nnc2)=O)=O)CC2CC2C2CC12 23357,n1(CC(=O)N(C(C)CN(C(=O)CCCNC(=O)OC(C)(C)C)C)C)ncn(C)c1=O 23358,C(=O)(CCC(CF)CF)N(C)CC1CCN(C(C2(C(F)F)CCCC2)=O)C1 23359,N1(C(c2occc2CN(C)C)=O)CC2C3CCC(C2C1)N(C(=O)CCF)C3 23360,N1(C(C2C(OC)CCC2)=O)CCC2(CCN(C(=O)CN3CCCCC3)CC2)C1 23361,c1(OC(C)C(N2CC(NC(C3(N(C)C)CC3)=O)CC(F)(F)C2)=O)ccc(F)cc1Cl 23362,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C3CC4(CCC4)C3)=O)C2)=O)c1C 23363,c1(C(C(=O)NCC)N(CCN(C)C)CC2CCC2)ccc(CC)s1 23364,C1(CNC(CCCc2c(C)ccc(C)c2)=O)(NC(=O)COC)CCC(F)(F)CC1 23365,N1(C(=O)OC(C)(C)C)CC2CS(=O)(=O)CC2(NC(=O)Cc2ccc(O)cc2)C1 23366,N1(C(C(CC#C)C)=O)CCOCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 23367,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23368,c12cncn1CCNC(=O)CNC(=O)C(=O)N2.C(CCOC(F)F)SC 23369,C(=O)(CC(F)(F)Br)N1CC(NC(COCCC#C)=O)C1 23370,C1(CN(C(=O)Cc2nc(=N)[nH][nH]2)C)CN(C(=O)CCC(F)F)CC12CC2 23371,C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1N(c1ncncc1C#N)C2 23372,C1(CC(=O)Nc2c(CC)noc2C)CN(C(=O)Cc2nc[nH]n2)CCC1C 23373,c1(C(N2CC(COC)(NC(c3ccc(CC)cc3)=O)C2)=O)ccc(C)cc1CC 23374,CCCC(C(C)(C)C)NC(=O)CC(C)(C)NC(=O)CCC1CC(OC)C1 23375,c1(CC)ccccc1OCC(N1CCCC1C(C)NC(=O)C(C)(C)C1CC1)=O 23376,CCCC(C(F)(F)F)NC(C1CCCC(NC(C2(Cl)CC2)=O)CC1)=O 23377,C1(OCCNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CCOC2C)CC1 23378,c1(C(=O)OCC)ccc(OCCc2ccc(NC(C)=O)cc2)cc1Cl 23379,N1(C(C(C(C)C)O)=O)CC2=C(C1)CN(C(c1cccnc1-c1nncn1C)=O)C2 23380,C1(CNC(CC(=C=C)C)=O)CC(NC(=O)C(C)=C2CCC2)C12CCC2 23381,c1(C(N(CC(C)NC(C2C(=C)C2)=O)C)=O)n[nH]c2cccc(OCC)c12 23382,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23383,O=C(CC1CCc2ccccc21)NC1CC(F)CN(C(C2(n3cnnn3)CC2)=O)C1 23384,CC1CCN(C(=O)C(F)CC2CCC2)CCN1C(=O)CCCC1NC(=O)NC1=O 23385,c1(C(N(C2CCCC(NC(C34CCC3CC4)=O)C2)C)=O)cc(F)cc(F)c1N 23386,c1(NC(c2ccc(CCC)s2)=O)cccc(NC(=O)Cc2cn(C)nn2)c1 23387,Cc1cccc(-n2cc(-c3c(C)noc3C)nn2)c1O 23388,c1(C(N(CC2N(C(C(CCC)F)=O)CCC2)CC)=O)cn2cc(C)ccc2n1 23389,CC1CN(C(=O)CC2CC(C)(C)C2)CC(C)C1NC(c1cccc(N)c1O)=O 23390,C=C1COCCN(C(=O)CC(CC)N(C(=O)Cn2cnnn2)C)C1 23391,C(=O)(C#CC1CCCOC1)N1CC(N(C(=O)C(N2CCCCCC2)C)C)C1 23392,CCCC(C(=O)N(C(CC)C(=O)Nc1ccc(OC)cc1)C)N(C)C 23393,N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)CCc2cnco2)C1 23394,c1(OC)ncc(Cl)cc1C(=O)NC1CC(NC(=O)CC2CCCC(OC)C2)C1 23395,C1(C(N(C2(CC(=O)N(C)CCc3ncccn3)CC2)C)=O)CCCC(C)(C)C1 23396,c1(NC(C(N2CCC(NC(C3CCOC3)=O)CC2C)CC)=O)c(C)cccc1C 23397,O=S(=O)(c1ccc(F)c(Br)c1)NC1C2CC1N(Cc1c(OC(F)F)cccc1Cl)C2 23398,N1(C(=O)Nc2cc(OCC)cc(F)c2)CCC2(COC(CSC3CC3)C2)C1 23399,c1(CNC(c2cc(CCNC(C3CC(C)OCC3)=O)on2)=O)cc(F)ccc1O 23400,c1(C(=O)NC(CC)CNC(=O)C(C)OCCC(C)C)cc2cccnc2[nH]1 23401,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(C(C)C)nn2)=O)C1 23402,CN1CCC(C)(C(=O)NC2CC(NC(=O)Cc3ccc(OC(F)F)cc3)C2)C1=O 23403,C1(N(CC(=O)OC)C(C2(N(C)C)CC2)=O)CCCC(CSc2ccccc2)C1 23404,Cc1oc(C2CC2)nc1C(=O)NC(CNC(=O)CCN(C)CCO)(C)C 23405,C(C)(C(C(C)C)NC(c1csc(Br)c1)=O)NC(c1ccn(C(C)C)c1)=O 23406,c1(NCCC(C(C)C)OCC)nc(N(C)C)nc2ncn(CC)c12 23407,S(=O)(=O)(c1cnc(NCc2conc2COC)cc1C)N(CC)CC 23408,c1(C(=O)NC(CN(C(=O)CNC(N)=O)C2CC2)C)cn[nH]c1 23409,O=C(NNC(=O)C(O)c1cn(CCO)nn1)c1cc(C2CC2)no1 23410,N1(C(CC2C(OC)COCC2)=O)CC(C2(NC(=O)C(C)=CC3CC3)CC2)C1 23411,c1(CNCc2ccc(C3(C(=O)OC)CCC3)cn2)ccc2occc2c1 23412,c1(OC)cc(C(=O)NC2CC3(C2)CN(C(C2C(C)C2C)=O)C3)cnc1OC 23413,N1(CC(=O)NCCN2CCCCC2)CCC(c2nc(-c3ccccc3)no2)CC1 23414,C(=O)(C#CC1CCOC1)N1CCN(C)C(CNC(N)=O)C1.C123CC4CC1C2C34 23415,C1(C(N2CC(N(C(=O)CC3(C)CC3)C)C2)=O)CCN(S(=O)(=O)N(C)C)C1 23416,CC(N=c1[nH]c(=NCC(F)(F)Br)[nH]c2c1CSC2)c1nc(C(F)(F)F)n[nH]1 23417,CC(C)(O)C(F)C(=O)N1CCOC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C1 23418,c1(N(C)Cc2nocc2Br)nc(=NCC(c2ccccc2)C2CC2)[nH]c2cc[nH]c12 23419,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCC(O)CF 23420,C(CCSC)(C(=O)NCC1(NC(=O)CC2CSCCS2)CC1)OC 23421,c1(-c2nnc(C(C)N(C)C)n2CC(=O)NC2CCSC(C)C2)ccc2c(n1)CCC2 23422,c1(OC)ccn2cc(C(=O)N(CC(CC)NC(=O)CC3CNC(=O)C3)C)nc2c1 23423,CC1(C)C(NC(c2cnn(CCCc3ccccc3)c2N)=O)CC1CN 23424,C1(C(N(C(C#C)C)CCCC)=O)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23425,C(=O)(C1=NOC(CNC(c2cccc(CC)c2)=O)C1)NC(C(=O)OCCC)C 23426,N1(C(CC2(COC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23427,N1(C(C(CSC)C)=O)CC2CCC(C1)N2C1CCN(C(=O)CC(F)F)CC1 23428,c1(N2CCCCC(NC(CSC)=O)C2)cc2nnc(-c3ccccc3)n2cn1 23429,C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1(CC#C)CCCOC1)=O 23430,c1(C(N2CCCC(C)(F)C2)=O)ccc2ncsc2c1.c12cccc(Cl)c1C(=O)N2 23431,C1(C(N2CCC(F)(CNC(c3nn(C)c(O)c3)=O)CC2)=O)CC2CCCCN2C1 23432,C(=O)(C(CCC(N)=O)n1cc(C(O)CC(C)C)nn1)OC.C12CN(C1)C2 23433,Cc1ccc(CC(=O)NCC2C3CN(C(=O)CC(F)(F)F)CC23)c(Br)c1 23434,c1(C(N(CCCCC)C)=O)ccc(-n2cc(CS(C)(=O)=O)nn2)cc1 23435,C1(C(N2C(C(C)(C)NC(C(C)OC(C)(C)C)=O)CCC2)=O)CCc2nncn2C1 23436,C(=O)(C(C(=O)N1CCC(C(=O)NC2CCCC2CN(C)C)CC1)OC)OC 23437,N1(C(COCCOCC)=O)CC2ON=C(CNC(c3cnn[nH]3)=O)C2C1 23438,c1(C(=O)NC2(C3N(C(CS(CC)=O)=O)CCC3)CC2)ccc(F)c2ccccc12 23439,Cc1nn(C)c(C)c1CC(=O)N(CCCCCCNC(=O)C(=O)N(C)C)C 23440,C(=O)(C(CC(C)C)NC(=O)C(N1CC(=O)NC1=O)C)NC(C#C)C 23441,CCC(C(=O)N1CC(C)(C)C1Cn1cc(C(C(C)C)N(C)C)nn1)C(C)(C)CC 23442,N(C1CC(C)(C)Oc2ccc(F)cc21)C1CC(S(=O)(=O)N)C1.CCC 23443,n1(C(CC)C)nnnc1C(C)(C1CC1)NC(C)CCC1CCC1 23444,CCC(C)(C)C(=O)C(=O)N1CCCCC(C(=O)N(CCCN=[N+]=[N-])C)C1 23445,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23446,S(=O)(=O)(c1c[nH]ccc1=NCCNC1CCCC(CC2CC2)C1)NCc1ccn(CC)n1 23447,CC(C)S(=O)(=O)c1ccc(NC(c2ccc(-c3ccco3)c(C)c2)=O)cc1 23448,C1(C(N2CCC(NC(C(N)=O)=O)C23CCCC3)=O)CC(c2ccccc2F)=NO1 23449,N1(S(c2c(C(C)(C)C)n[nH]c2)(=O)=O)CCN2C(=O)OCC2C1 23450,Cc1cnccc1C(=O)NCC1CCC(NC(=O)C#CC2CC2)C1 23451,C1(C(=O)NC(CC(C)NC(c2cn(CCC(C)C)nn2)=O)C)CCC(C(N)=O)CC1 23452,c1(C(C)C)ccc(N)c(C(=O)NC(CNC(C2(CO)CCCC2)=O)C2CC2)c1 23453,N1(C(Cc2c(C)occ2)=O)CCN(C)CC1C(=O)NCC1(O)CCCC1 23454,C1(C)(C(N2C(CCNC(C(CCOC)C)=O)COCC2)=O)CCC(C)(C)CC1 23455,N1(C(C(C)OCCC(C)C)=O)CCC(NC(=O)C(C2CCC(=O)N2)C)C1(C)C 23456,C(=O)(CC(C)(C)CC(=O)N1CC(NC(C2CCN(C3CCOCC3)C2=O)=O)C1)OC 23457,c1(NC(C)=O)c(C(=O)NCC2C=CC(NC(C3(F)CC3)=O)C2)cccc1C 23458,C1(NC(=O)CCn2ccnn2)CCC(NC(=O)C(C2CC(F)(F)C2)O)C1 23459,C1(NC(C2CCc3nncn3CC2)=O)C2CC3CN(C(=O)CCC4CC4)C1C3C2 23460,c1(C(N(C2CCN(C(=O)CSC(F)(F)F)C2)C)=O)cnn(C(F)(F)F)c1 23461,c1(C(=O)OCCC2CCCOC2)cc2ccccn2n1 23462,Cc1ccc(C(N2CCC2CNC(=O)C(n2ccnc2C)C)=O)c(N)c1 23463,N12CCC(C)(C)C1CC(=O)OC2=O.N1(C(CC2(OC)CC2)=O)C(C(=O)NC)CC1C 23464,CCCC(CC)CC(=O)N(C(C)CNC(c1ccoc1-c1ccccc1)=O)C 23465,CC(c1cccs1)=CC(N1CCC(C2CCCN2C(=O)C(C)OC2CC2)C1)=O 23466,N1(S(CC(=O)OC)(=O)=O)CCCC2(CCN(C(c3ncc(OC)cc3F)=O)C2)C1 23467,N1(CCCC(C=C)Nc2ccc(S)cc2OC)CCc2[nH]nc(C(F)(F)F)c2C1 23468,C#CCCC(C(=O)NCC1CCSCC1)NC(c1cc(CCC)[nH]n1)=O 23469,CCC(C)(CNC(C1CCN(C)C1=O)=O)C(=O)NCc1ncoc1C1CC1 23470,N1(C(C(C)CC(F)F)=O)CC(C)(C)OCC1CNC(=O)CC1CC2CC2C1 23471,Cc1cccc(CCC(=O)NCC(CNC(=O)CCC2CCC2)CO)c1Br 23472,N1(C(C(C)(C2CCC2)NC(CSC(C)(C)C)=O)=O)CCC(N=[N+]=[N-])C1 23473,C(C)(CNC(=O)COCC1CCCC1)(CO)NC(C(C)OCCOC)=O 23474,N1(C(C(Br)=C(C)C)=O)CCN(C(C2CCCCO2)=O)C(CO)C1 23475,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)ccn2nccc2n1 23476,S1(=O)(=O)c2cc(ccc2F)N1.c1(-c2cn(C)nc2)ncccc1C(F)(F)F 23477,C1(NC(c2cnsc2)=O)CCCC(NC(C2OCCO2)=O)CC1 23478,CCCC(C)CN=c1[nH]c2c(c(=NC3CCC4(CCC4)C3)[nH]1)CSC2 23479,N1(C(C2CC(CC)C2)=O)CCN(C(=O)C(N)=O)C(C2CC2)C1 23480,C1(C#CC(=O)N2CCN(C(c3cnn(-c4ccncc4)c3)=O)CC2)(CC)COC1 23481,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23482,O(C1CCOc2cc(Cl)ccc21)C(c1c(F)cc(OC(F)F)cc1F)=O 23483,Cc1cc(C(=O)NCC2C3CC2N(C(c2occ4c2CCC4)=O)C3)c(O)nn1 23484,c1(CC)ncccc1C(=O)NCc1cnnc(C)c1 23485,N1(C(C2C(OCC)CCC2)=O)CC(NC(=O)Cn2nc(C)cc2C)CC1(C)C 23486,C=CCC(CC(F)F)NC(=O)CC1CCCCC1NC(C1CCC(C)O1)=O 23487,c1(C(C2CCCCC2)NC(C(=O)NCC2(F)CCCC2)=O)cc(F)cc(F)c1 23488,C#Cc1cccc(C(N2CCN(CC(=O)NCC3CCC=CO3)CC2)=O)c1C 23489,C1(c2cn(C(CC)C)nn2)(C(=O)N(C2(C)CCCC2)CCN(C)C)CC(F)(F)C1 23490,C(=O)(CCCCCC(C)(C)C)NC1CCC(N(C(c2c(C)cc(N)cc2)=O)C)C1 23491,C12(CNC(c3c(SC)csc3)=O)CCCC1N(c1cc(C)nc(SC)n1)CCC2 23492,CC(C)C(C)CCNC(=O)C(C(C)O)NC(=O)CN1C(=O)CNC1=O 23493,Cc1ccc(Cl)c(O)c1C(N1CC(NC(c2ccc(F)s2)=O)CC(O)C1)=O 23494,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CN(Cc1ccc3scnc3c1)C2 23495,C1(CC)(NC(=O)CCC2CC(NC(=O)C(C)CN(C)C)C2)CCCCC1 23496,c1(C(N2C(C(C)(C)NC(C(F)=C(C)C)=O)CCC2)=O)cc2cc(Br)cn2cn1 23497,C(=O)(C(C)C(CC)CC)NC(CC)C.c12nc(nc(C)c1F)NC1CN2CN1 23498,Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)cnc1O 23499,C1(NC(C(C(=O)NC)C)=O)CC2(CCCN(C(=O)C(COC)C(F)(F)F)C2)C1 23500,c1(CC(=O)NC(CC(C)NC(C(CC)NC(N)=O)=O)C)ccccc1OC(F)F 23501,N1(C(CC2C(C)(C)CCCC2)=O)CC2CC(C1)CN(C(c1ccc(F)o1)=O)C2 23502,C1(NC(c2c(C(C)(C)F)cccc2)=O)COC2CNCC12 23503,C(C(C)(C)CC(=O)NCC(c1ccccc1)NC(=O)CC1CC1(Cl)Cl)OC 23504,Cc1cccc(Cl)c1CC(=O)NCC1CC1CNC(=O)CC1CCOC1 23505,N1(C(C2(CC=C)CC=CC2)=O)CCC(C)(CNC(=O)CC2CCCCC2C)CC1 23506,CC(C)C1=NOC(c2nnc(CCCN(C(=O)OC(C)(C)C)C(C)C)o2)C1 23507,C=CCC(F)(F)C(=O)N(CC(O)CNC(=O)CSc1nnnn1C)C 23508,C#Cc1ccc(C(C)Nc2cc(NC3COCC3OCC(F)(F)F)ncn2)cc1 23509,C1(NC(CCCN(C)C)=O)CC2CN(C(c3cccc4ccoc34)=O)CC12 23510,c1(OC)cccc(C(N2CCC(C(C)NC(=O)CNS(N)(=O)=O)C2)=O)c1 23511,Cc1nn(CCF)cc1NC(C1CC(C)CN1C(c1ccnc(CO)c1)=O)=O 23512,CN(C)NC(=O)CCC(=O)N1CC2(CCN(C(c3ccc(CO)cc3)=O)CC2)C1 23513,N1(C(C(C)S(N)(=O)=O)=O)CCCCC2(C1)CN(C(=O)CC1(O)CCCCCC1)C2 23514,C(=O)(C1CCc2c[nH]nc21)NC1(C2N(C(CCc3nnc(C)n3C)=O)CCC2)CC1 23515,c1(OC)ccccc1C(=O)NCC(=O)NC(C)CCN1CCOCC1 23516,CC(C(=O)NC1(CNc2nc3ccc(F)cc3o2)CCOCC1)C(C)S(C)(=O)=O 23517,c1(CC(=O)OC(C(=O)OCC)Cn2cccn2)cccc(OC)c1 23518,c1(C(=O)NCC2(C)CCN(C(C34CCC(F)(CC3)C4)=O)C2)noc2ncccc12 23519,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23520,Cc1c(C(=O)NC2CN(C(=O)COCCF)CC2O)oc(=O)c2ccccc12 23521,CC1CN(C(=O)C(C2CCCCCC2)F)CCN(C(c2ccc(O)c(F)c2)=O)C1 23522,CC(C(C)C)=CC(=O)NC(C)(CNC(c1ccc[nH]1)=O)C1CC1 23523,N1(C(c2c(C#C)c[nH]n2)=O)CCCC(O)(CNC(=O)COC2CCC2)CC1 23524,c1(C(c2nnnn2C2CCCC2)NC(C2CCCC2)C2(COC)CC2)cc(Cl)no1 23525,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23526,N1(C(CCNC(=O)NC)=O)CC2CCC1CN2C(=O)Cc1ccc(C#N)cc1 23527,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23528,C(C(C#C)CC(C)(C)C)NC(C1(F)CCCN(C(CCC#CC)=O)C1)=O 23529,C1(C(N2CCC(CNC(C(c3cncn3C)C)=O)CC2)=O)CCC2(CCC2)C1 23530,C12(CC(=O)NC(CCN(CC)CC)C)CCN(C(=O)CC(C)(C)C)CC1C2 23531,c1(OC)ncnc(C)c1C(=O)NCC1CCN1C(C1CC(F)(F)C1)=O 23532,c1(C(=O)NCCCN(C(C(C)(C)OCC)=O)C)ccc(C)c(C)c1O 23533,c1(C(=O)NCCN(C(C2CC(=C3CC3)C2)=O)CC)cc(-c2cccnc2)no1 23534,C1(C(=O)NCC2=CCN(C(=O)CC3CCCC3)CC2)CCC2(CCOC2)O1 23535,c1(C(C(=O)NC(C)C2CC2)N(CC(C)N(C)C)C)cc(C(F)(F)F)on1 23536,C(=O)(CCCCCC(C)(C)C)NC1C(NC(C(c2cnccn2)C)=O)CCCCC1 23537,Cc1oc(C)c(C(N2CC(C)(NC(=O)CC3CC4COCC34)C2)=O)c1C 23538,c1(C(C)(C)C)nnc(C(=O)NC2CC(n3ccnn3)C2)o1 23539,N1(C(c2ccc(C(F)(F)F)o2)=O)CCCC2(CCCN2C(C2CC23CCC3)=O)C1 23540,N1(C(c2cc(CC)on2)=O)CC(C)C(C(=O)NC)C1C.C1(CO)CC1NC=O 23541,N1(C(c2cnc(OC)s2)=O)CC2CCC1C(CNC(=O)CCCC(N)=O)C2 23542,Cc1cc(Br)ccc1C(=O)NC1CCCC(NC(=O)CC2(C)CCCO2)C1 23543,c1(CCC(=O)NCCOCCN(C(=O)CC(O)c2ccccc2)C)nocc1C 23544,C1(CC(N2CC(c3c(CNC(C4(C)CCCC4)=O)nco3)C2)=O)CCCC1(F)F 23545,C1(NC(C(C2CCN(C(Cc3c(C)occ3)=O)C2)(C)C)=O)CCC12CCCC2 23546,C1(NC(COCCC(C)C)=O)CCN(C(C2CC3CC2CC3O)=O)CCC1CO 23547,c1(C(N(c2cc(C)c(Cl)cc2)C)=O)ccc2c(c1)COC2 23548,N1(C(c2ccc(C)o2)C(=O)NCc2ccc(Br)cc2)CCCC(C)(C(F)(F)F)C1 23549,c1(N2CC3CC(NC(c4cccc(C(C)C)n4)=O)C3C2)ncnc2c1CCO2 23550,N1(C(C)=O)CCC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(CO)C1 23551,N1(C(C23CC(NC(C(CC)n4cncn4)=O)(C2)C3)=O)CCC(O)(COC)C1 23552,N1(C(c2c(C)nn(C)c2Cl)C(=O)NCC2CCOCC2)CCCc2ncccc2C1 23553,C(C(=O)N=c1ccc(Cl)n[nH]1)C1N(CC2(c3ccc(C)cc3Cl)CC2)CC(O)C1 23554,c1(OC)cc(F)c(S(=O)(=O)NC2CCCC2P(C)(C)=O)cc1OC 23555,c1(CC(=O)NC2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)cccc2nonc12 23556,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC2NC(=O)C(C)(C)Cc2cnn[nH]2)c1)NC 23557,N1(C(CC(c2ccccc2F)C)=O)CCCC(O)(CCNC(=O)C(C)(C)CF)C1 23558,C(=O)(C(O)CC(F)F)NC(C1CCN(C(Cn2nc(C)c(Cl)c2)=O)CC1)(C)C 23559,C(=O)(C1=CCC(NC(=O)CN2CCNC2=O)C1)N(C(C#C)C)C 23560,CC(C)(C)C(CNC(=O)CCC1CCCO1)NC(=O)CCC1(C)N=N1 23561,c1(C(=O)NCCCN(C(CCCOCC)=O)CC)ccc(N)c(N)n1 23562,c1(C(N2CC(COC)(CNC(=O)C=Cc3cn(C)cn3)C2)=O)cccc(Cl)c1N 23563,C1(NC2CCC(C(N(C)C)=O)C2)CCNC(C2CC2)C1 23564,N1(C(Cc2ccc(C)nc2)=O)CC(C)(C)C(NC(c2cccnc2O)=O)C(C)(C)C1 23565,C(CO)(CCCCNC(=O)CC1OCCCO1)NC(CCn1c(C)nc(C)n1)=O 23566,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23567,c1(C(=O)NCC23CCC(NC(C4CCC(C)O4)=O)(C2)CO3)[nH]c2ccccc2n1 23568,C(CN=c1nc2scnc2c(NCc2cn[nH]c2)[nH]1)N1CCC(O)CC1 23569,c1(C(=O)NC2C3CC(NC(C4C5COCC45)=O)CC23)ccc(F)cc1[N+](=O)[O-] 23570,C1(OCC)CCCN(C(=O)Cc2nc(CNC(=O)C(CC)n3cncn3)cs2)C1 23571,C(=O)(C(C)(C)CC(C)=O)NCC1N(C(C(C(CC)C)OC)=O)CC=C1 23572,C1(CC(=O)NCC2CN(C(C3(C)CCCOC3)=O)CC2O)CN2CCN1CC2 23573,CC1(C)CN(C(c2cc(CNC(C3CCC(O)C3)=O)[nH]n2)=O)CC1CO 23574,N1(C(C(C)SCCCC)=O)CCCCC(C(N2CC(CCC)C2)=O)C1 23575,C(=O)(C#CC1CCCCO1)NCC(C)(CC1CC1)NC(c1cccnn1)=O 23576,c1(C(=O)NC(C2CCCCN2C(C2CC(C#N)C2)=O)C)cc2cc(F)ccc2o1 23577,CCCCC(F)C(=O)N1CCCCC1CCCNC(=O)OC 23578,NS(=O)(=O)c1ccnc(C(=O)NC2CN(C(C3C(C4CC4)C3(F)F)=O)C2)c1 23579,Cc1ccc(C(F)F)cc1OC(C)C.C1C(C)(C(C)C)NC(=O)N1 23580,C1(C(=O)NCC2(OC)CCN(C(=O)C(C)c3ccsc3)C2)CCC(N=[N+]=[N-])CC1 23581,N1(C(COCCCC(C)C)=O)CCC2(C1)CN(C(C1CC1C#N)=O)C2 23582,CCC(O)CCN=c1[nH]c(N2CCN(CCCOC)CC2)nc2cccnc12 23583,c1(CC)nc(C(N2CCC(C(C)NC(c3cnccn3)=O)C2)=O)co1 23584,c1(C(=O)NC(C2CCCC2)CNC(C(C)C#N)=O)ccc(C2CC2)cc1 23585,N1(C(c2cc(C)n(CC)c2C)=O)CCC2C(C1)CN2C(=O)C(C)C(F)(F)F 23586,C(CC(C)C(=O)NCC1CC1NC(c1c(C)nsc1I)=O)OC 23587,C12(CNC(C=CC(=O)N(C)C)=O)CC1CN(Cc1cccc(CO)n1)C2 23588,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23589,C1(NC(CC2C(=O)NCC2)=O)CC2CC(C1)N(C(=O)Cc1cnsc1)C2 23590,C12(C(N3CC4C(NC(c5cc(O)ccc5Cl)=O)C4C3)=O)CC3CC1C2C3O 23591,N1(C(C2CCN(CC)C2)=O)CCCC(CCNC(=O)Cc2cnnn2C)C1 23592,c1(COCC)nnc(N2CCCC2c2ccn(C)n2)n1CC 23593,CC1CN(CC2(O)CCOCC2)CC1C(=O)NCc1ccccc1F 23594,C(=O)(C(F)NC(=O)COC(C)(C)C)N(C1(CC(C)C)CCC1)CCOC.CC 23595,C(=O)(CC(C)CNC(C1(CF)CCOCC1)=O)NC(c1ncccn1)C 23596,N1(C(CC2(C(=O)OC)COC2)=O)CCC(CNC(c2nccnc2SC)=O)CC1 23597,c1(NC(=O)COC2CCC2)ccc(CC(C2CC2)NC(C)C(C)(C)O)nc1 23598,C1(NC(c2cnc(OC)s2)=O)CN(C(c2ccc(C(F)(F)F)cc2)=O)CC1O 23599,c1(C(=O)NC(C(C)NC(C2C=C(C)CS2)=O)C)cn2cccnc2n1 23600,c1(C(=O)NCC(=C)CCNC(=O)C(C)CN(C)C)noc2ncccc12 23601,c1(C(N2CCC3(C2)CN(Cc2ccccc2)C3)=O)ccc(Cl)c2cccnc12 23602,c1(OC)cccc(C)c1C(C)N(C)C(=O)NC(CNC(C)=O)C1CC1 23603,CC(CC(C)(C)C)C(=O)NC12CCCN(C(=O)C3=COCCO3)CC1C2 23604,c1(C(N2C3(CN(C(=O)CS(=O)(=O)C4CC4)C3)CC2)=O)cnc2ncnc(O)c2c1 23605,Cc1ccc(SCC2CCCN2C(c2c[nH]c(C#N)c2)=O)cc1.C12(CC1)C(=O)N2 23606,C(C(C)(C)C(F)(F)F)C(=O)NC(C(N1CC(C(=O)NC)C1)=O)C1CCCC1 23607,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23608,N1CCC2(CC1)CC2c1cn(CC2CC(O)(CC=C)C2)nn1.C(=O)CC(O)CC 23609,C1(C(=O)NCC23N(C(C4(C)CCCCC4)=O)CC(C2)C3)CS(=O)(=O)CC(=O)N1 23610,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23611,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23612,CC1CC(C(=O)NCC#CCNC(C2CC2C(c2ccccc2)=O)=O)CC(C)C1 23613,N1(C(C2C(C(=O)OC)C2)=O)C2CCC(C(=O)NC3(CC(C)C)CC3)C1CC2 23614,C(CCCCC(=O)N1CC2CC2(CNC(=O)C2=CCCCC2)C1)SC 23615,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23616,C1(CNC(C2C(=O)OCC2)=O)CC2CC2N1C(=O)Cn1cnc(C(N)=O)n1 23617,n1(CC(=O)NCC(CNC(C2CC3CCC(C2)O3)=O)OC)nc(C)c(C)c1C 23618,C1(C(=O)NC(CNC(c2c(C)noc2)=O)(C)C2CC2)CCOC2(CCC2)C1 23619,C1(O)(CN(C)C(c2ccc(C(F)F)nc2)=O)CCN(C(=O)CCc2nncs2)C1 23620,c1(C(=O)NC2(CCNC(C3C(C)CCC3)=O)CCC2)cc2c(F)c(F)ccc2[nH]1 23621,c1(N(C)C)ccc(C(=O)NC(CNC2CCC(=O)N2)C2CC2)cc1[N+](=O)[O-] 23622,c1(CC(=O)NC2CCC(CNC(=O)CC3CCCCC3)C2)cc(C(F)(F)F)co1 23623,C1(F)(CNC(c2ncc(OC)cc2F)=O)CC2CCC(C1)N2C(c1cnns1)=O 23624,Cc1cc(C)n(-c2ccc(-c3nc(-c4cncnc4)nn3CC(C)CO)cc2)n1 23625,c1(C(=O)NC2C(O)CCN(C(CCCC3(C)N=N3)=O)C2)cnc2ccsc2c1 23626,C(=O)(C(O)CCNC(C1CCCC1F)=O)N(CCCC=C)C 23627,C1(CNC(C=CC)=O)COCCN1C(=O)C=CC(=O)NCC 23628,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(C)C)CC(F)C1 23629,c1(C2(n3cc(C(=O)NCCNC(Cn4c(C)nnn4)=O)nn3)CC2)ccc(C#N)cc1 23630,N1(C(C2N(CC)C(=O)CC2)=O)CC(NC(c2ccccc2O)=O)CCC1C 23631,CC(C)CC(F)C(=O)NCC1(C)CN(C(=O)CCCN2CCCCC2)CC1C 23632,N1(C(CCCCC#C)=O)CCCC2(CCC(NC(c3n[nH]cc3CC)=O)C2)C1 23633,C1(C(=O)NC(c2ccco2)C)(C(N)=O)CCN(C(C23CC4CC2C3C4)=O)C1 23634,N1(C(c2ccnc(C)n2)=O)CC2(CC(NC(c3n[nH]c(C)c3[N+](=O)[O-])=O)CO2)C1 23635,c1(C(=O)NCC2(F)CCN(C(CCCCC#C)=O)CC2)cc(N)cc(C)c1F 23636,N1(C(c2c(CCC)n(CC)nn2)=O)CC(NC(=O)C=C2CCCCC2)CCC1C 23637,c1(CC)cc(C(=O)NC2(C)CCN(C(c3coc(C4CCC4)n3)=O)C2)ccc1C 23638,c1(CC(=O)NCC(CNC(CC(=O)OC)=O)OC)ccc2ncsc2c1 23639,C1(C(=O)NC2C(C=C)OCC2)CN(C)CCN1C(c1cc(OC)cc(F)c1)=O 23640,C1(CNC(C(C2CCN(C(C3OC4CCC3C4)=O)CC2)C)=O)NC(=O)OC1(C)C 23641,N1(C(c2cc(NCc3ccc(OC)cc3O)ccn2)=O)CCC(C2CC2)C1CO 23642,c1(C(N2CC(CNC(C(CC)(C)O)=O)CC(C)(C)C2)=O)ccc([N+](=O)[O-])c(N)n1 23643,CCC(CC)CCCC(=O)NC(CC1CCC1)C(N1CC(O)CC1CO)=O 23644,CC(C(=O)NCC1CN(C(c2coc(Cl)n2)=O)CC1C)C(C)(C)C 23645,C1(OC)CC(CNC(c2csnc2C)=O)N(C(C2CC(N(C)C)C2)=O)C1 23646,C(=O)(C(C)S(N)(=O)=O)N1CC(c2cn(CC(COC)OC)nn2)(O)C1 23647,C(CCS(C)(=O)=O)SCCNCc1scc(C(C)=O)c1 23648,CCCC(C(O)C(=O)NCC(O)C1CC1)NC(=O)CCc1nncn1C 23649,N1(C(c2ccc(OC)cc2F)=O)C2CCC1CC(NC(=O)C(C)CS(C)(=O)=O)C2 23650,C=CCCCC(C(=O)Nc1cccc2c1CCO2)NC(=O)CC1C=CCCC1 23651,c1(C(=O)OC)cnc(SC)[nH]c1=NCCCCNC(c1cnnc(Cl)c1)=O 23652,C(CCCC(=O)N1CC(NC(c2sc(CCC(C)C)nc2C)=O)C(C)C1)OC 23653,C(C(C)(C(=O)NC(CCCNC(=O)CCC1(C)CC1)c1ccccc1)OC)OC 23654,c1(CC(N2CCC(N(C(CC(CC)SC)=O)CC)C2)=O)ccc(C)c(C)c1 23655,Cc1c(C(N2CCC3(CC3C(=O)Nc3cc(O)ccn3)C2)=O)ccc(Br)c1F 23656,C1(CC=C)(C(=O)NC2CC(C(C)NC(c3cscc3Cl)=O)C2)CCOC1 23657,N1(C(CC2(C)CCOC2)=O)CCC(C(C)(C)C)(CNC(c2ncc(F)cn2)=O)C1 23658,C(=O)(C(C)Cn1ccc(C)n1)NCCN(C(=O)C(C)c1ccon1)CCC 23659,C1(C(=O)NCC2(CO)CCN(C(c3c(C)cc(F)s3)=O)C2)SC2C=CC1CC2 23660,C#CC1(O)CCN(C(c2coc(C(C)NC(=O)C(C)(C)C=C)n2)=O)CC1 23661,c1(C(=O)NC(C(C)NC(C(C)NS(CC)(=O)=O)=O)CO)cccc(N)c1F 23662,c1(C(=O)OC(C=C)OC2CCCC2)cccc(C2CC2)n1 23663,N1(CC(=O)NCC2(CC(=O)N(CCOC)CC3CC3)CC2)C(=O)CCCC1=O 23664,Cc1cnccc1CN1CCCC(CNC(C2C3CN(C(C)C)CC23)=O)C1 23665,Cn1cnc2nc(N3CCC(C(N)=O)CC3)ncc12.c12ccc(cc1)NC(=O)C2 23666,Cc1nc2cccc(C(N3CC(NC(C4CCS4(=O)=O)=O)CC3(C)C)=O)c2s1 23667,C(=O)(C(C#N)=CC(C)C)NCC1(NC(C=CCOC)=O)CCC1 23668,N1(C(c2cnn(C)c2Cl)=O)CCCC(NC(=O)CC2CCCOCC2)CC1 23669,Cc1cc(C(=O)N(CCCCNC(=O)C2=CCCC2)C)ccc1Cn1ccnc1 23670,C(=O)(C(C)(CC1CCC1)OC)NCC1C(NC(CCNS(CC)(=O)=O)=O)CC1 23671,Cc1nnc2ccc(C(N3CCC(NC(=O)CC4(O)CCOC4)C3(C)C)=O)cn12 23672,c1(C(=O)NCC(C)(C)C(=O)NCC2(C)CC3CC3C2)cccc2c[nH]nc12 23673,C(=O)(CC(O)CC(C)C)N(CCCOC)C.C1(OC)CNC1=O.C(CO)N 23674,C1(CC(=O)N(CCOC)CC)CN(C(=O)CC2(COC)CCOCC2)CCO1 23675,Cc1nn(CC(=O)NC2CC3C(NC(=O)Cc4cnccn4)C3C2)c(=O)o1 23676,c1(C(C(N2C(CN(C(C(F)=CCC)=O)C)CCC2)=O)O)ccccc1F 23677,N1(C(C(C(C)O)(C)C)=O)CC2COCC2(C(=O)NCc2ccc(Cl)cc2)C1 23678,c1(C(C(=O)N(CC(C)O)CCNC(=O)C(C)(C)C)(F)F)c(F)cccc1F 23679,C1(C)(C(N2CCN(CCCNC(C(C(C)C)F)=O)CC2)=O)CCCCC1(F)F 23680,C1(C(=O)NCCOC2CCN(C(c3cnc(C)s3)=O)CC2)CC(C(C)C)=NO1 23681,C(C(CCC)C(=O)N1CCC1(C)CC)NC(C(C=C)(C)C)=O 23682,c1(OC)ccn2cc(C(N3CC(C(C)NC(=O)CC(C)C(C)C)C3)=O)nc2c1 23683,N1(C(CCCCSC)=O)CC2(C)CC1C2NC(c1ccc(=O)n(C(C)C)c1)=O 23684,C(C)(C)(C(=O)N1CCC(CCNC(=O)Cc2[nH]cnc2C)C1)OCC 23685,c1(C(=O)NCC2CC(C)N(C(=O)CC3C=CCC3)C2)ncc(Cl)cc1Cl 23686,c1(C2C(=O)N(C3CCOCC3)CC2)ccc(F)c2cccnc12 23687,c1(CC)ncsc1C(=O)NC1(CCNC(=O)CC(F)F)CC1 23688,CCCCC(Cc1ccccc1)NC(=O)CC1CC(c2ccccc2)C1 23689,C1(NC(CCC2C(C)C2)=O)CC(C)(CNC(=O)CC23CCCC2C3)C1 23690,N1(C(C2CC2C2CC2)=O)CCC2CN(Cc3ccccc3)CCN2C1 23691,C1(C(=O)NC(C)(C)CCNC(=O)CC2CC=CC2)CC2COCCN2C1 23692,Cc1c(NC(c2n[nH]cc2NC(c2ncccc2C(F)(F)F)=O)=O)ncnc1Cl 23693,CCC(C)C(O)C(=O)NCC1CN(C(=O)C(CC(=O)OCC(C)(C)C)C2CC2)C1 23694,c1(C(=O)NC(C(CO)NC(Cc2cccc(CC)c2)=O)C)onc2c1CCCC2 23695,N1(C(C2CCC(N(C(COC(C(C)C)=O)=O)C)CC2)=O)CCC(CO)C(F)(F)C1 23696,C=CC(C)CC(=O)NCC1(OCC)CN(C(c2ncn(C)n2)=O)C1 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23714,CCCC(CCCO)C(=O)N1CCCC(NC(c2cc(Cl)cs2)=O)C1C 23715,C1(C2CCOCC2)(NC(Cn2c(C)nnc2S)=O)CC1 23716,CCC(c1cccc(Cl)c1)=CC(=O)NCC=CCNC(C1CCC(C2CC2)C1)=O 23717,C(=O)(C(O)CCCC)NCC1(O)CCN(C(CSCCC)=O)C1 23718,N1(C(C(C2CCCC2)OCC)=O)CCC(CCNC(c2cnc(O)o2)=O)CC1C 23719,N1(C(C=CC=CC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(c2ncc[nH]2)C1 23720,Cc1cc(C(=O)NCC(C)(CC(C)C)NC(=O)C(C)Cn2ccnc2)c(C)cn1 23721,Cc1cc(CNC(=O)C(C)(C2CC2)N(C)C(C2CC(C)C2)=O)cc(F)c1 23722,N1(C(c2nc(C)n(C)c2C)=O)CC(C)OC2(CCN(C(=O)C(O)C(C)C)C2)C1 23723,N1(C(C(CNC(c2c(OC)ccnc2)=O)C)=O)CC=CC12CCCCC2 23724,C(=O)(CS(=O)C(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23725,c1(-c2c(C(N3CC(C)(NC(C4(C)C(C)C4)=O)C3)=O)c[nH]n2)cccc(Cl)c1 23726,c1(C(=O)NCCCNC(c2cncc(C)c2)=O)sc2nc(C)nc(C)c2c1C 23727,Cc1ccc(-n2ccnc2)c(C(=O)NC2C=CCN(C(C3CC3C)=O)C2)c1 23728,c1(CC(N2CCCC2C2CCN(C(C3(CO)CC3)=O)CC2)=O)cccc(O)c1 23729,Cc1cc(=N)[nH]cc1C(=O)NC1CC(C)N(C(c2cn(CCF)nn2)=O)C1 23730,N1(C(C(C(CC)O)C)=O)CC2(C)CN(C(c3cn(C)nn3)=O)CC2(C)C1 23731,CC#CCC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)NC(N)=O 23732,c1(C(N(CCN(C(C(CCCOC)C)=O)C)C)=O)cccc2c1C1CCC2CC1 23733,N1(C(c2ncn(CCNC(C(C(CC)C)N(C)C)=O)c2)=O)CC2C=CCC(C2)C1 23734,c1(OC)c(Cl)nc[nH]c1=NCC1CCCN1C(C1Cc2ccccc2CO1)=O 23735,C12(C(=O)NCc3ccc(C)c(Cl)c3)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23736,c1(NC(C(C)C)CNC(c2ccncn2)=O)cnc2ccccc2n1 23737,S(=O)(=O)(c1c(C)ccc2ccccc12)N(C(CC)Cc1ccc(F)cc1)C 23738,c1(ONC(C(c2n(C)nnn2)N(C)C)=O)ccc(Cl)c(C(N)=O)c1 23739,N1(C(=O)CCC2CC2)CC(O)(C2CCN(C(c3n[nH]c4c3NCCC4)=O)CC2)C1 23740,CCS(=O)(=O)CCNC(=O)NC(c1nc(-c2ncccn2)no1)C 23741,c1(NC(CC2N(C(CC(C)O)=O)CCCC2)=O)ncc(Cl)cc1O 23742,c1(N2CC(CC(C)NC(=O)CNS(=O)(=O)C3CC3)C2)ncc2c(ncn2C)n1 23743,c1(CNC(C=CCC)=O)cnn(C)c1CC1CCC1.C1(C=O)CCC(C)C1 23744,C1(NC(c2ccccc2CO)=O)CC2CC1N(C(c1ccc(O)c(Cl)n1)=O)C2 23745,C(C)(C(=O)N1CCCC(C)(CNC(=O)C(C2CCCCC2)F)C1)(C(C)C)OC 23746,N1(S(c2c(N3C(COC)C=CC3)nccc2)(=O)=O)CCc2cc(C)cc(C)c2C1 23747,C1(CNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 23748,C(=O)(C1=CCCOC1)NCC1CCCN(C(C(C)(C)Cc2ccccc2)=O)C1 23749,c1(C(N2C(CNCc3c(C)cccc3)CCCC2)=O)c2n(c(=O)n1C)CCCC2 23750,N1(C(C(C)(C)C(F)(F)F)=O)CCN(C(=O)CC(F)(F)C(F)(F)F)C2COCC12 23751,Cc1nccc(CCC(=O)NCC2CCCCN(C(C3(C)CCCCO3)=O)C2)n1 23752,CCCCC(C(=O)NC)NC(C12CC1CN(C(c1cc(C)ccc1N)=O)C2)=O 23753,c1(NC(c2nnc(S)n2CC(=O)NCC2C(CC)CCC2)=O)ncc(OC)cc1C 23754,n1(CCC(C)C)ccc(=NC(=O)c2ccc(C3CCNCC3)s2)[nH]1 23755,C1(CC(=O)NC2(C)CN(C(C(C)O)=O)C2)CN(C(N)=O)CCO1 23756,C(=O)(CCCCC(F)F)N(C(=O)C(C)OCC1CC(OC)C1)Cc1ccccc1 23757,C(=O)(C#CC(C)(C)C)N1C(C)(C(N2CC(CCCCC)C2)=O)C=CC1 23758,CC(CN=C(NCC1(C2CCCO2)CCCC1)NCC(F)F)CC(F)(F)F 23759,N1(C(C2CC(SC)C2)=O)CCC(N(C(=O)CC2CCN(C(C)=O)C2)C)C1C 23760,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23761,C1(C)(CNC(C(c2ccc(C)s2)C)=O)CCN(C(=O)CC2CC=CCC2)CC1 23762,c1(OC)cc(CN(C(=O)C(N)CCCC2CC2)c2ccccc2)ccc1I 23763,N1(C(COC(C)=O)=O)CC2CCC2(CC(=O)NC(C)(CO)C2CCC2)C1 23764,N1(C(CN(C(COC)=O)C)=O)CC(C)(CCC(=O)NCC(C)O)C1 23765,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23766,c1(OC(C(N2CC(O)(CNC(C(CC(C)C)OC)=O)C2)=O)C)ccccc1C 23767,N1(C(CCC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23768,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(=O)Cc2nnc(O)s2)CC2(CC2)C1 23769,C1(CNC(C(C)Sc2ccncc2)=O)C2CCCC1N(C(=O)C(C)(C)C1CC1)C2 23770,CCCCCCCC(F)C(=O)N1CC(Cn2cc(CCS(=O)(=O)NC)nn2)C1 23771,Cc1c(C(=O)NCC2CN(C(=O)Cc3csc(NC=O)n3)CC2O)cccc1F 23772,S(=O)(=O)(c1cccc(-c2nn[nH]n2)c1)N(C)C(C1CC(c2ccc(O)cc2)C1)=O 23773,N1(C(C(C)N(C)C)=O)CC(F)CC1C#N 23774,C1(OC)CN(C(=O)C=CCOCc2ccccc2)CC1NC(=O)C(F)C1CCC1 23775,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23776,C(c1ccc(F)cc1F)=CC(=O)NCC1(NC(C(CCSC)OC)=O)CCC1 23777,C1(=O)CCCCC(=O)O1.CC1CC(C(=O)NC2CCCC2CC(C)(C)C)CCO1 23778,C(=O)(C1=CC2C=CC(C1)C2)NC(COCC)C(=O)NC1CCCCN(C)C1=O 23779,C(CCC(O)C(=O)Nc1cccc(F)c1)NC(C1CCC2(CCC2)O1)=O 23780,C1(CC)CN(C(=O)CCc2nc(Cc3ccccc3)no2)CCN1 23781,C1(C(=O)NC2CC(CNC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23782,FC1(F)CC12CCC(CSc1ccc(-c3nnco3)cc1)C2 23783,c1(C(N2CC(C)C(NC(c3ccc(Cl)cn3)=O)C2)=O)c(N)sc2c1CCSC2 23784,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23785,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(C(C)(F)F)CC3)=O)CC2)C1 23786,N1(C(C(C2CC2)OC)=O)C2CCCC1CN(C(=O)C(C)N(C)C)C2 23787,N1(C(CCOCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23788,C=CC(CC)CC(=O)NC(CSCC)C(=O)Nc1cn(C(C)C)nc1C 23789,CCC(C)CCC(=O)N1CCC(CNC(c2cncnc2C)=O)C1(C)C 23790,C(C)(C(=O)N(CCC)CC=CC(=O)N(C)CCN1CCCC1)OCCC#C 23791,C#Cc1cc(NC(C2CC2CC(C)C)=O)ccc1C.C1C(N(C)C)C(=O)N1 23792,Cc1nsc(C(=O)NCC2CC2(C)Br)c1N 23793,C1(C(=O)NCCC(=O)OCC)CCCC(NC(=O)COCCCOC)CC1 23794,C1(NC(CCC#C)=O)CN(Cc2cccc(OC(F)(F)F)c2)CC1C#N 23795,c1(C(=O)NC(C)CCNC(CC2(OCC)CC2)=O)cnc2nc(C)ccc2c1O 23796,N1(C(C(CCCC)O)=O)CCOC2(C1)CN(C(=O)C(c1ccc(O)cc1)=O)C2 23797,c1(C(=O)NC(c2ccc(O)cc2)CC(=O)OC)cc(Br)cc2c1OCC2 23798,C1(OC)CC(C(=O)NCC23CCC(CC2)N3C(=O)CC2CCCOC2)C12CCC2 23799,c1(C(=O)OC)cc(Br)cc(C)c1NC(C1CN(C(=O)C(C)(C)F)CC12CC2)=O 23800,Cc1ncnc(C(N2CCCC(C)(NC(=O)C(C)Cc3ccco3)C2)=O)c1C 23801,Cc1noc(C)c1CC(=O)NC1CC2(C1)CC2C(=O)N(CCCF)CCO 23802,N1(C(c2cc(C)c(C)o2)=O)CCC(C)(CNC(=O)CCNC(C2CC2C)=O)CC1 23803,C1(CN(C)C(C2C3CNC(=O)C23)=O)COCCN1C(=O)CCN(S(C)(=O)=O)C 23804,C(N=c1[nH]c2ccc(Cl)cc2c(=N)[nH]1)C1(C(C)C)CC1 23805,CCC(C)(CNC(c1cc(C)c(C)nn1)=O)C(=O)Nc1cccc(C)c1C 23806,n1(CC(C)C)cc(C(=O)NCC2COCC2NC(=O)CC2CC2)c2ccccc12 23807,C(=O)(CCCCC(N)=O)N1CCC(C(C)NC(C2(C)CCNC(=O)C2)=O)C1 23808,c1(NC(C2(CNC(=O)CCc3ccsc3)CC(=C)C2)=O)ccc(CC)nc1 23809,C(=O)(NNC(=O)SC)C1(c2n(-c3n(C)ncc3)ccn2)CC1 23810,c1(CCC)cccc(C(=O)NC(C)CCCNC(=O)CC2CC3(CC3)C2)c1 23811,C1(COC)(NC(=O)CNC(N)=O)CCN(C(c2ncncc2Br)=O)CC1 23812,c1(C(=O)NCC2C(C)CCN(C(=O)CCc3cnc[nH]3)C2)cccc2nncn12 23813,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C)n[nH]1 23814,O=S(=O)(c1ccc(NCc2cc(F)ccc2F)cc1Br)NCCC1(CO)CCCC1 23815,C1(NC(C(CC=C)C)=O)CCC2(CC1)CC(NC(c1ccc(Br)cc1)=O)C2 23816,c1(CSCC(=O)NC2(CF)CCN(C(C(CC)SC)=O)C2)nc2ccccc2[nH]1 23817,c1(C(N2CCN(C(C3C(COC)C3)=O)C(C)C2)=O)sc2ccccc2c1Cl 23818,CC1(C)CCCC(CC(=O)NCC(C)(O)CNC(=O)CCc2nccs2)C1 23819,CC1CC(C(N2CCCN(C(C3CC(NS(C)(=O)=O)C3)=O)CC2)=O)CCC1C 23820,N1(C(CC(=O)NCCOc2cncc(Cl)n2)=O)CC(C(=O)NCC)C(F)C1 23821,c1(SCC(=O)N(C2CC3CC3C2)C)nnc(-c2ccccc2)n1CC(F)F 23822,C1(NC(COCCOC)=O)CC(NC(c2sccc2C#N)=O)C12CCC2 23823,C1(N(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2cccc(O)n2)=O)CC1(C)C 23824,C(c1cccc(F)c1)=CCC(=O)NC1CC1NC(=O)C(F)(F)CC1CCCCC1 23825,C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(C(C)C)F)=O)CCCC1 23826,CCS(=O)(=O)CC(=O)NC1CC1CNC(c1c(-c2cccc(C)c2)n[nH]c1C)=O 23827,c1(NS(C)=O)ccc(C2C(NC(=O)NCCOC)C2)cc1 23828,Cc1c(NC(=O)CC2CCN(C(c3ccc(N)cc3F)=O)CC2)cccc1C#N 23829,N1(C(C(F)=CCC)=O)CCC(NC(C23CC(C)C2C3)=O)C2(CCC2)C1 23830,N1(C(C2CCC(C(C)C)CC2)=O)CC2CC(CNC(=O)CCCCF)C2C1 23831,C1(N)(C(C)(C)C)CCN(C(C2CC(=O)CCO2)=O)C1 23832,N1(C(c2noc(CC)c2C)=O)CC2C(NC(=O)CCc3nc(C)c(C)o3)C2C1 23833,Cn1nnc2ccc(=NCc3ccc(Br)c(F)c3)[nH]c12 23834,Cn1cnc(C#N)c1C(=O)NCCCCNC(=O)C(CCO)C1CC1 23835,CCC(C)C(C(=O)N(CCCCN(C(=O)CC1CCCO1)C)C)NC(N)=O 23836,c1(C(=O)NCC2CCC(NC(CCC3N(C)CCC3)=O)C2)nccc2occc12 23837,C(Cc1ccccc1)(C(=O)NOC1CCC(N)C1)NC(C(CCOC)C)=O 23838,N1(C(C(CCC)C(C)C)=O)CCC2CN(C(c3conc3C)=O)C(C)C12 23839,c1(C(=O)NCC2N(C(CC#N)=O)CCOC2)cccc2c1OCC2 23840,C(C(=O)N1CC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C(O)C1)(C(C)(C)C)N(C)C 23841,c1(OC)cc(NCc2cc(O)nc(O)n2)nc(OC)n1.C1CO1 23842,c1(-c2cncc(OC)c2)ccc2c(c1)CN(Cc1cnc(O)nc1O)C2 23843,C1(C(N2C(C(=O)O)(CC)CCC2)=O)CN(C(c2cnc(C)s2)=O)CCC1O 23844,N1(C(C2(OC)CC2)=O)CCC(NC(=O)C=Cc2nc(C)cs2)C(CO)C1 23845,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2CC3C=CC2O3)=O)C1)OC 23846,N12CCS(=O)(=O)C(C1)CC1N(CC=CC1)C2=O.c1(OC(C)(C)C)ccccc1F 23847,c1(CCN(C)CC2(CC(=O)N(C)C)CCC2)cc(O)ccc1O 23848,c1(C(N(CCN(C(C2C(C(C)C)C2)=O)C)C(C)C)=O)c[nH]nc1-c1cccnc1 23849,c1(OC)ccc(C(=O)NC2CC(NC(=O)Cc3cscn3)C23CCC3)c(F)c1Cl 23850,O(NC(=O)C(CCC1CC1)NC1CC1C1CC1)CCCC(=O)OC 23851,C1(C(N2CC(CC)OCC2)=O)CCN(C(=O)OC(C)(C)C)C(C#N)C1 23852,c1(C(N2CC3C(CNC(C4=CC(C)(C)C4)=O)C3C2)=O)[nH]cc2c1CCC2 23853,C(=O)(C(F)C(F)(F)F)N1C(CN(C)C(c2ccc(C(F)(F)F)s2)=O)COCC1 23854,c1(CC(=O)NCc2cnn(CCOC)c2C)ccc(Br)cc1OC 23855,C1(CC(C)C)CCCCN1C(c1ccc(CNC(=O)Cc2ccnnc2)cc1)=O 23856,C1(C(=O)NCCCC(C=C)(C)C)CCCCCCN1C(=O)Cc1cccnc1C 23857,CCC(C)CCCCC(=O)N(C1CCCN(C(c2cnc(S)n2C)=O)C1)C 23858,Cn1ncc2c(C(=O)NCC3CC4CN(C(=O)CC5CC5)CC34)ncnc12 23859,C(=O)(CCCCNC(=O)CCc1ccn(C)n1)N(C)CC1CCC1 23860,CCC(C)CCCCC(=O)N(CCCN(C)C)CCNC(C1(C)CCC1)=O 23861,CS(C)(=O)=Nc1nccc(NC(C2CC3(CCC2=O)CC3)=O)n1 23862,C1(CC)(CC)CN(C(=O)CC2CC(F)CN2C(=O)C=NOC)CCO1 23863,c1(C(=O)NC(CNC(C(CC)=CC)=O)C)c(C)c[nH]c1CC(N)=O 23864,c1(C(C)N(C)Cc2noc(C(N)=O)n2)cc2c3c(c1)CCCN3CCC2 23865,C#Cc1cncc(C(=O)N(C(C)C(N2CCC(C3CC3)C2)=O)CCN(C)C)c1 23866,Nc1cnc(Br)cc1C(=O)N(C(c1cnc(Cl)cc1)=O)Cc1ccco1 23867,c1(OC)ccc(C(C(=O)NCCSC2CC2)N(C2CC3CCCC23)C)cn1 23868,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 23869,N=c1cc(C(=O)N(c2ccccc2)CCOC(F)F)c(Br)c[nH]1 23870,Cc1nc(-c2ccccc2)sc1C(=O)NCC1(NC(C2(C)CC2(F)Cl)=O)CC1 23871,C1(NC(C(c2ccc(F)cc2)C)=O)CN(C(=O)C=CC(=O)N(C)C)CCS1 23872,c1(CCC(=O)NC2C(NC(=O)CC3CC(F)(F)C3)CCC2)nnc(S)nc1O 23873,c1(NC(c2nnn(C)n2)(C)C2CC2)ncccc1OCn1cccc1 23874,c1(OCC)ccnc(C(N2CC(CNC(C3(OC)CCOC3)=O)C(C)C2)=O)c1 23875,C1(NC(CNC(C)=O)=O)CN(C(c2csc([N+](=O)[O-])c2)=O)C2(CCC2)C1 23876,CCCC(CCC)C(=O)NC12CC(C1)N(C(=O)CCCOCCOCC)C2 23877,C1(C(C(=O)N(C(COC)C)C)C)CCN(C(c2ccns2)=O)C1 23878,C1(NC(CC(C)SC)=O)CCCCC1NC(c1cc(C(C)=O)c(C)o1)=O 23879,c1(C2N(C(c3cnn(C)c3CN)=O)CCNC2=O)ccc(Cl)c(F)c1 23880,c1(C(=O)NC(CC)(CNC(C2(C)CSC2)=O)CC)ccc2occc2c1 23881,c1(OC)cnccc1CC(=O)NC1CCCC(CNC(C2(C)CNC(=O)C2)=O)C1 23882,N1(C(=O)Nc2cc(CO)ccc2F)CCN2C(c3ccccc3)CS(=O)(=O)C2C1 23883,C(=O)(C1=C(C)CCC1)NC1CCN(CCCNC(C(CC)O)=O)C1 23884,c1(C(N2CC(CC(=O)NCCC(CCC)C)(OC)C2)=O)ncc2ccccn12 23885,N1(C(c2ncn(C)c(=O)c2)=O)CCCC2(CCN(C(=O)CC=C(Cl)Cl)C2)C1 23886,CP(C)(=O)c1cncc(C(=O)NCC(C2CC2)NC(c2cnn[nH]2)=O)c1 23887,C#CCC(CC(=O)NCc1cnc(C)o1)NC(=O)CCNC(C)=O 23888,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1C1CC1)=O)C2 23889,C(CCCC(=O)NCc1sncc1Br)n1cc(-c2n(C)cnc2)nn1 23890,c1(C(N2CC3(CN(C(C4=C(C)OCCS4)=O)C3)C2)=O)ccc2c(c1)OC(C)(C)C2 23891,C1(C(=O)Sc2cn(CC3CC3)nn2)CCCN(C2CCCC2)C1.C12CC(=O)N(C1)C2 23892,c1(OC)c(F)ccc(F)c1C(=O)N(CCCCN(C)C(C1CC=CCO1)=O)C 23893,c1(C(=O)NCCn2cc(C(N(CCC(=O)NC)C)=O)nc2)cnc(S)nc1 23894,c1(C(=O)NCC(CC)NC(c2sc(NC(C)=O)nc2C)=O)ccc(Br)c(C)c1N 23895,N1(C(CC(C)SC)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 23896,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 23897,c1(C(N2CC(CNC(c3c(CC)noc3)=O)C(O)C2)=O)c(S(C)(=O)=O)cnn1C 23898,C1(CNC(C(=C2CCCCC2)C)=O)COC(C)(C)CN1C(c1ccc(O)c(F)c1)=O 23899,N1(C(C)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 23900,N1(C(C2(C(N(C)C)=O)CC2)=O)CC(O)(CNC(=O)Cc2cc[nH]c2)C1 23901,C1(CC(=O)NC(C#C)C(C)C)CCCCN1C(=O)C(C)NC(=O)CC 23902,C1(NC(CCc2cc(C)sc2C)=O)CC12CCN(C(c1nccnc1N)=O)C2 23903,N1(C(c2nccc(C)c2N)=O)CCC2CC(CNC(=O)C(N)=O)CCC2C1 23904,N1(C(C2(CC#C)CCCCC2)=O)CC2CC(NC(=O)C=Cc3cccs3)CC2C1 23905,C1(NC(=O)CC2CCCOCC2)CC2CCC1(NC(=O)C=CC1CC1)C2 23906,C(=O)(C(C)CC(F)(F)F)NC(CCCCNC(c1ccc(OC(C)C)nc1)=O)C 23907,c1(CC(=O)NCCC(CNC(C(CC)C)=O)O)cccc2cnccc12 23908,CCCCC(C)CCC(=O)NCC(CC)NC(C1CCN(C)C1CC)=O 23909,c1(OC)cc(O)c(C(=O)NC2CC2Nc2cnc(OC)c(F)c2)c(Br)c1 23910,CC1CN(C(=O)C#CC(=O)Nc2nccs2)C(C)CN1C(c1cc(N)cnc1Cl)=O 23911,Cc1c(C(=O)NC(c2nncn2C2CC2)C2CCCO2)cnn1CC(C)C 23912,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2(CCCCC2NC(=O)Cc2cnc[nH]2)C1 23913,CCC(CC(=O)NC1CCC(C)N(C(=O)Cc2nc(C)sc2Cl)C1)CC(C)C 23914,c1(C(=O)NCC(CNC(c2cc(C)ccc2N)=O)OC)coc2c(Cl)cccc12 23915,c1(C(C(F)(F)F)NC(C(C)C(F)(F)CN)=O)c(Cl)cc(Cl)cc1Cl 23916,N1(C(C2N(C(CC(CC)(C)C)=O)CC23CCCC3)=O)CC2CCC(C1)C(=O)N2 23917,C12(C(=O)NCC(CCOC)NC(c3ccsc3)=O)CCC(OC)C1C2 23918,C1(CNC(c2ccc(C(C)C)o2)=O)CN(C(C2(C3CCCCO3)CC2)=O)CC1C 23919,Cc1ccc2c(C(=O)N(C3C4CN(C(C5(CO)CCC5)=O)CC34)C)onc2c1 23920,C=CCCCCCNC(=O)N(c1ccccc1)C(CO)C1CC1 23921,c1(C(=O)NCC2C(NC(C3C(=C)C3)=O)CCCC2)cc(F)c2[nH]nnc2c1 23922,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 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23941,CC1C(NC(=O)Cc2c[nH]ccc2=O)CC2CCC1N2C(c1ccc(F)s1)=O 23942,c1(CN(C2CCC2)C(C)=O)ccc(NC(=O)N(C)CC2(C)CCCO2)cc1 23943,C(=O)C(C)CC(C)(C)C.C(CC(=O)NCC(O)CN(C)CCF)OCCOC 23944,C1(C(=O)NC2CC(CC#N)C2)CS(=O)(=O)C2CN(C(C3(C(F)(F)F)CC3)=O)CC12 23945,N1(C(CC=C=C)=O)CC2(C1)CN(C(c1cc(C)nc(C)n1)=O)C2 23946,c1(C(C(N2CC(N(c3cnc(Cl)[nH]3)C)C2)=O)O)ccc(OC(F)F)cc1 23947,C1(C(N2CCN(C(CC(c3c(C)noc3C)C)=O)CC2)=O)CC(C2CC2)=NO1 23948,C12(C(=O)NCc3cc(C)on3)CCCC1CCN2C(C1CCCC1)=O 23949,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)NC3CC(O)C3)C2)c1 23950,C1(CC(=O)NC2CC(C)OC2=O)CC(C)(C)CN1C(=O)CCC1CCCCC1 23951,c1(CNC2(c3nnnn3C3COC3)CC(CC)C2)ccc(C#N)c(C#N)c1 23952,C(=O)(C(C#N)C(C)C)NCC1(C(=O)NC(c2ncc[nH]2)CC)CC(=C)C1 23953,C1(CC=C)(NC(=O)C(O)C2CCC2)CN(C(=O)C(C)(C2CC2)OCC)C1 23954,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cccc3oncc23)=O)C1 23955,C1(C(=O)NC2(CCOC)CCC2)CN(C(C2CCN(C)C2=O)=O)CC1(F)F 23956,C(=O)(C1=CCCCC1C)N(C1CCCC1)CC(=O)OC(c1cc(C(C)=O)cn1C)=O 23957,C(CC(O)C(=O)NC1CC(NC(=O)CCN(c2ccccc2)C)C1)SC 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23976,n1(CC)nnc(C(=O)NCc2csc(CNC(c3cc[nH]n3)=O)n2)c1C 23977,c1(C(=O)OCCC(N2CC(C3CC(=O)NC3)(O)C2)=O)cccc2nccnc12 23978,Cc1nc(C2CC2)ncc1C(=O)NC(CNC(c1cnn(C)c1Cl)=O)C1CCC1 23979,CC(C)(C)CCCC(=O)NC1CCC(CCNC(c2cnn(C(C)(C)C)c2)=O)C1 23980,c1(C(c2nnnn2C2CC2)NCC(C)OC2CCOCC2)nc2c(s1)CCCCC2 23981,CC1CCCN(C(C2(C)CCCN2C(c2cocc2C(N)=O)=O)=O)C1CO 23982,N1(C(c2c(COC)cco2)=O)CCC2CNCC12 23983,Cc1cc(O)c(F)cc1NC(C1CCN(C(c2cscc2Cl)=O)C1C(C)C)=O 23984,N1(C(CCCC=C)=O)CC(C(N2CCCC2CSC)=O)C2(CC2)C1 23985,CC(CCC(=O)N1CCOC(CO)C1)NC(=O)C=C1CCC1 23986,N1(C(=O)OC(C)(C)C)CC(CCCF)(CCNC(C2(c3ccno3)CCC2)=O)C1 23987,Cc1coc(C)c1C=CC(N1CC(O)(CCNC(C2COC(C)C2)=O)C1)=O 23988,C1(=O)C(CC(C)C)N(C)CC(C)CC1=C.C(COCC)(CCCC)N 23989,c1(C(=O)NC(CN(C(c2nscc2C)=O)CC)C)cnn(C(C)(C)C)c1 23990,c1(CC)[nH]nc(C(=O)NC2(CCNC(C3CN(C)C(=O)N3)=O)CCCC2)c1C 23991,C1(C(N(C2CCN(C(C3CC(C)C3C)=O)CC2)CCO)=O)SC2C=CC1CC2 23992,CC(C)C(C)CC(=O)NCC1CCCC(CNC(=O)C=Cc2cc[nH]n2)C1 23993,C1(C(N2CC(NC(CC3(COC)CCC3)=O)CC2(C)C)=O)CC2(CC(C)=NO2)C1 23994,Cc1c(C(N2CCN(C(c3c(Cl)cnn3C)=O)C3CC23)=O)cccc1O 23995,c1(C(=O)OC)ccc(C(=O)NCC2CC2F)o1.C12CC(C1)CNC2=O 23996,N1(C(C(C)Sc2ccc(F)cc2)=O)CCCN(C(=O)Cc2ccsn2)CC1C 23997,c1(C(N2CC(C(Cn3cc(COCC)nn3)F)C2)=O)nnc(O)nc1O 23998,C(=O)(CC(c1ccccc1)N(C)Cc1ccccc1)NC(C1CCCC1)C 23999,S(=O)(=O)(c1cnc(NCCN2CCC(CO)C2)c(Cl)c1)NCCC1(N(C)C)CC1 24000,C1(C)(C(=O)NCC(CCNC(C2(C)CC(C(F)(F)F)C2)=O)O)CC2CC2C1 24001,C(=O)(C(O)CC(F)F)NCC1(C)CCN(C(=O)Cc2ccc(CO)cc2)C1 24002,C1(CC=C)CCCCC1NC(C1(CC=C)CN(C(=O)COCC2CCCO2)C1)=O 24003,C1(NC(COC2(C)CCC2)=O)CC2CCC1CC2NC(c1cc(F)cnc1Cl)=O 24004,N1(C(c2c[nH]c(=N)s2)=O)CC2(C1)CN(C(=O)Cc1cccnc1O)CC2CO 24005,c1(C(=O)NC(C)CCCNC(C2CC3CC3CC2C)=O)ccc(F)c2c1CCC2 24006,c1(C(=O)OC)c[nH]c(=NCC23CCN(C(c4nc(Cl)cs4)=O)CC2C3)cn1 24007,C1(C(=O)NCCC(C)NC(c2cc(Cl)cc(Cl)c2N)=O)OCC2COCCC12 24008,N1(C(COCCOCC#C)=O)CCCC12CCCN(C(=O)C=CC)C2 24009,CC1(C)C2CCC(C2)C1(C)C(=O)NCC(CO)NC(c1ccccc1CN(C)C)=O 24010,C1(C(=O)NCCn2cc(C(=O)NCC(N3CCCC3)C)nn2)C2CC3C(C2=O)C13 24011,c1(CNC(=O)NC(C)CC2CCCC2)ccc2c(c1)CC2 24012,c1(CNc2nccc(=NCc3ccc(OC)nc3Br)[nH]2)cc(C)ccc1S(N)(=O)=O 24013,c1(C(=O)NCC2(CCNC(C3(O)CCC3)=O)CC2)ccncc1OC1CCOC1 24014,c1(C(N2CCC(N(C)C(C3CN(C(N)=O)C3)=O)C2)=O)cccc(Cl)c1Cl 24015,N1(C(=O)C=CCO)CCC(C2CCCN(C(C3(CO)COC3)=O)C2)CC1 24016,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2CC2)C1CNC(C1CSCC(=O)N1)=O 24017,CC1CN(C(C2CCC(C)CC2)=O)CC(CCNC(c2cn3ccnc3s2)=O)O1 24018,c1(SC)ccc(C=CC(=O)NC23CCC2CN(C(=O)CC2CC(F)C2)C3)cc1 24019,Cc1nc2cnn(C)c2cc1C(=O)NC1CCCN(C(=O)CC(F)(F)F)CC1 24020,c1(C(N2CCC(C3N(C(c4nnn(C)n4)=O)CCC3)C2)=O)c2c(nn1C)CCSC2 24021,CC1CC(=O)NC1C(=O)N(CCCNC(C12CCC(CC1)C2)=O)C 24022,c1(-c2ncc(C(=O)NC3CCOC(C(=O)O)C3)s2)ccccc1F 24023,C1(O)(C(N(CCNC(COCC)=O)Cc2ccc(C)cc2)=O)CC2CCC1C2 24024,C(=O)(C1=C(C#N)CCC1)NC(CC(=C)Cl)C(=O)N1CCCC(F)(CO)C1 24025,c1(C(N2CCCC(CNC(C3C(CC)CCO3)=O)C2)=O)cc2cc[nH]c(=O)c2s1 24026,C1(C(=O)NC2(C(=O)NCC3(OC)CCCC3)CC2C)CCC(=O)N(C)C1 24027,c1(CC(=O)NCCCCCNC(C(CC)N(C)CC)=O)cc(C)ccc1F 24028,C1(C(=O)NCC(C)N(C(=O)Cc2ccnc(C(F)(F)F)c2)C)Cc2cscc2C1 24029,CCC(CC(=O)NC(C)(CO)C(=O)NCc1ncn(C2CC2)n1)SC 24030,c1(CC(=O)NC2CC(CNC(c3c(CC)con3)=O)C2)ccc(O)nc1 24031,C12(C(=O)NC3CC4C(NC(Cc5n(C)ccc5)=O)C4C3)CCC(C1)C(C)(C)O2 24032,C(=O)(CCCCCF)Nc1n(CC(N2CCC(OC)(CO)C2)=O)nc(C2CC2)c1 24033,C1(CNC(Cc2c(C)nccc2)=O)CC(F)(F)CN1C(=O)C1=CCCS1 24034,C1(C)(C(=O)NCCCOC(C)C)CCCN(C(=O)CC2CCOCC2)C1 24035,C1(NC(COCCC)=O)CCC2(CCN(C(c3cc(CC)ccc3F)=O)C2)C1 24036,CC1(C)CCCC1CCNC(=O)C(=O)NN1CCCCC1.C12=CC=C(C=C1)C2 24037,S(=O)(=O)(c1ccc(NCCCO)cc1Br)N1CCN(C)C2(C1)CC2 24038,O=S1CCC(CNCc2n[nH]c(=N)s2)C1 24039,C(=O)(CCS(N)(=O)=O)N(CCCCCNC(C(c1cccc(C)c1)OC)=O)C 24040,c1(C(=O)NC(c2ccc(F)cc2F)CCO)csc2ccncc12 24041,Cc1ccn2cc(C(N3CCC(C)CC3CNC(=O)CC3CCCO3)=O)nc2c1 24042,c1(N2CCC(CC)OCC2)[nH]c(=NCc2ccc(C)cc2Cl)nc2scnc12 24043,CCC(C)(CO)C(=O)NC(C)C(C)(C)NC(=O)COC1CCCCCC1 24044,N1(C(C(CC)OC)=O)CCN(C(C2CCC(C)(OC)CC2)=O)C2(CCC2)C1 24045,N1(C(CC(C)NC(N)=O)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24046,c1(CCC(=O)N(C(CCC)C)C)cccc(-n2cc(-c3cnccn3)nn2)c1 24047,N1(c2snc(COC)n2)CCCC(C2CC2)CC1 24048,c1(CC)cc(C(N2CCCC2C(C)NC(=O)CSCC2CCCO2)=O)n[nH]1 24049,C(=O)(CCCCC(F)F)NCC(CNC(C(C(C)C)F)=O)O 24050,c1(C(=O)NC23C(CN(C(CC#C)=O)C2)C3)ccc(N=Nc2ccc(C)cc2)cc1 24051,CC1CN(C(=O)CCc2ccc(Cl)s2)CCC1NC(c1ccc(CF)cc1)=O 24052,C1(C(=O)NCC(CNC(COCc2cccc(C)c2)=O)CO)OCC2CCCC12 24053,c1(NC(C2C3CC2N(C(C2CC4C=CC2C4)=O)C3)=O)ncc(Cl)nc1Cl 24054,N1(C(c2cc3cccnc3s2)=O)CCCC2C1CCCN2C(c1ccncc1)=O 24055,C1(C(=O)NC2C(O)CCN(C(c3n(CCC)ncc3)=O)C2)CCn2cnnc2C1 24056,c1(C(=O)NC2C(NC(C3CCC(C(=O)OC)CC3)=O)CC2)cc(SC)cc(F)c1 24057,C1(C)(CNC(CC2(COC)CC2)=O)CN(C(c2ccc(C(C)C)cc2)=O)CCO1 24058,c1(C(N(C)C)=O)cc(NCc2ccncc2Br)ccc1F 24059,N1(C(c2c(OC)nccc2)=O)CC2OCCN(C(C3CC34CCSCC4)=O)C2C1 24060,C1(CCCCNC(=O)CC2CC23CC3)CCN(C(=O)CC2OCCO2)CC1 24061,c1(CNC(C(COC)OC)=O)ccc(CCNC(c2c[nH]c(C#N)c2)=O)cc1 24062,C(=O)(C(O)C(C)(C)C)N1CCC(CCOC)(NC(=O)CCc2cncnc2)C1 24063,CCCS(=O)(=O)C(C)C(=O)NC1(CNC(C2(n3cnnn3)CC2)=O)CC(OC)C1 24064,CC1CCCCC1(CNC(=O)C(F)=C1CCCC1)NC(C1CCC(=O)N1)=O 24065,c1(C(=O)NC(CCOC)CNC(C2(C)CCCCC2)=O)cc(=O)n2nccc2[nH]1 24066,N1(C(=O)CN2CC(n3cc(Cl)cn3)C2)CCCC(F)(CO)C1 24067,C=CC(C)(C)CCN=C(NCc1ccco1)NC1CCN(C(=O)OCC)C1 24068,c1(C(N2CC(C(=O)OC)(Cc3cccc(CC)c3)C2)=O)cc2cccnc2s1 24069,C1(C(=O)NCC(C(=O)OC(=O)C2CC2)OC)CCCN(C(=O)OC(C)(C)C)C1 24070,Cc1ccccc1C(C)(C)CNC1CCOC(c2ccc(F)cc2)C1 24071,C(CC(O)CNC(C1(CO)CC1(F)F)=O)NC(c1cnc(-c2cccs2)s1)=O 24072,C1(CNC(c2n(CCC)ncc2)=O)CCC12CCN(C(C1CCO1)=O)CC2 24073,CCCCC(C)CCC(=O)NC1(COC)CN(C(=O)C(C)CN(C)C)C1 24074,c1(C(=O)NCC(C)CNC(c2ncncc2Cl)=O)ccc2cnsc2c1 24075,Cc1cc(C(=O)NCCC2(NC(=O)COC(C)(C)C)CCC2)c(O)c(C)n1 24076,c1(CC(N2CC(N=[N+]=[N-])C(NC(c3cocn3)=O)C2)=O)n[nH]c2c1CCCC2 24077,CS(=O)(=O)CCC(=O)NC1(NC(=O)CCNC(N)=O)CCOC1.C1C(=O)N1 24078,c1(C(=O)NC(C2CC(C(=O)NC(C)(C)C)C2)C)cncc(F)c1.C12CC1NC2=O 24079,C(=O)(CC1=CCN(C(=O)Cc2cccnc2)CC1)NC(CCCC)(C)C 24080,C1(NC(c2cccc(O)n2)=O)(CF)CCN(C(C2CN(C3CCOC3)C2)=O)C1 24081,O=C1NCCC2CCN(C(C3(F)CN(C(c4cc5cccnc5[nH]4)=O)C3)=O)C12 24082,c1(CN=C(NCC2CC2)NCC2(C(F)(F)F)CCCCO2)cccc2c1OCO2 24083,c1(OC)cc(F)c(C(=O)NC2CC2CNC(c2ccc(Cl)c(Cl)c2)=O)c(F)c1 24084,c1(NC(=O)C(F)CC2CCC2)ccc(S(=O)(=O)N2CCCC3COCC23)cc1Cl 24085,C1(C(=O)N(CCCC)CC2CCC2)CCCN(c2cnc(C(=O)O)cn2)C1 24086,Cc1c(C(=O)N(C)CC2CCCN2C(=O)Cn2cnnn2)ccn1C1CC1 24087,C1(COC)(CNC(=O)C(C)C#N)CCN(C(c2coc(C#N)c2)=O)CC1 24088,N1(CCN(C(=O)NC2C(C=C)C2)C)CCC(COC)C1 24089,n1(CC)ncn(NC(=O)Cn2cc(CC(C3(C(F)F)CCCO3)=O)nn2)c1=O 24090,C1(CNC(=O)C=CC2CC2)CC2CN(C(=O)C(c3ccccc3F)F)CC12 24091,c1(CC(=O)NC(C2CN(C(C3CC3C3CC3)=O)C2)C)csc(-c2ccccc2)n1 24092,C1(CNC(=O)C=CCO)CC(C(=O)NC(CO)C2CCC2)=NO1 24093,C1(NC(C(C)CS(C)(=O)=O)=O)COC2(CCN(C(C3C4(CC4)C34CC4)=O)CC2)C1 24094,C1(OCC(N2CC(CNC(C(C3CCC3)OC)=O)C2)=O)CCC(C)CC1 24095,C(=O)(CCCCC(=O)NCC1(CCNC(C2CCC(F)C2)=O)CC1)OC 24096,C(=O)(CCCCCNC(=O)Cn1nc(C)oc1=O)NCc1ccn(CC)n1 24097,c1(Oc2c(OC)cccc2)cc(F)cc(OCC2CCCCC2)n1 24098,C1(C(=O)NC2CC(OCC)C2)CCN(C(=O)C2CN(C(C)C)CCN2C)O1 24099,C1(CC)COC(C)CN1C(=O)COC1CC(ONC(c2ncon2)=O)C1 24100,N(C(=NCCCCl)NCCC(C)C)CC1CCOC(c2ccc(OCC)cc2)C1 24101,C1(C(N2CCCCC(NC(C34CCC3C4)=O)C2)=O)CN2CCC1CC2 24102,C(C(=O)OC(C)(C)C)(C(C)N(C)N1CCC(CC)C1)OCC 24103,c1(NC(CN(CC(=O)NCCN(S(=O)(=O)CC)CC)C)=O)nc(C)nn1C 24104,C1(c2nnnn2C2COC2)(NC2(C(C)C)CC2)CCN(CC2CCC2)CC1 24105,c1(NC(CCC(C(=O)OCC)O)C)c(Cl)nc(-c2ccccc2)nc1Cl 24106,C1(C(=O)NCCSCC=C)CCCCN(C(c2c[nH]c(=N)o2)=O)C1 24107,c1(C(N(C)CC2C(NC(CSC)=O)CCCC2)=O)cc(C)c(O)c(N)c1 24108,C(=O)(C(F)C(C)(F)F)N1C(CCC(=O)NCc2c(C)occ2)CCCC1 24109,C(C1=CCN(C(=O)C(c2cccnc2)N2CCCC2)CC1)NC(n1ccnn1)=O 24110,C(=O)(CC(C)C(=O)c1ccc(Cl)cc1)NCC1CN(C(C(C)c2ccco2)=O)C1 24111,c1(N2CCC(N(C(=O)C=Cc3ccccc3C)CCC)C2)ncnc(O)c1Br 24112,c1(CCNC(COC2CN(C(c3nc(CC)oc3)=O)C2)=O)nccc(OC)n1 24113,CC(C)C(C)(O)C(=O)NC(Cc1ccccc1Br)C(=O)NCCCC(=O)N(C)C 24114,c1(C2C(C(N3C(CC(N)=O)CCC3)=O)CCC2)ccc(O)c(Br)c1 24115,c1(CN2C(C(=O)Nc3cncc(Br)c3C)CC(=C)C2)c[nH]c2c(F)cccc12 24116,C(CC(C(C)C)(c1nnnn1CCCF)Nc1ccc(C(C)(C)C)cc1)OC 24117,C(CCC(=O)N1CC(c2nncs2)C1)(C(C)C)NC(c1c(C)cc[nH]1)=O 24118,c1(NC(c2cccnc2)C(=O)NCC2(C)CCC(=O)N2)ccn2ccnc2c1 24119,Cc1cc(C(=O)NCC2(CNC(=O)C=Cc3cn[nH]c3)CC2(F)F)ccc1O 24120,CC1C2CC(C2NC(C2CCC(F)(F)CC2)=O)N1C(c1c[nH]c(=O)cn1)=O 24121,C1(C(=O)NCC2(NC(c3n(CC#C)ccc3)=O)CCCC2)CCn2nnnc2C1 24122,N1(C(C(CSC)O)=O)CCN(CCCCCNC(=O)CNC(C2CCC2)=O)CC1 24123,C1(NC(N2CCC(Cc3ccncc3)C2)=O)CC(F)(F)C1 24124,c1(C(=O)NCC2(NC(C=Cc3nnc(C(C)C)o3)=O)CC2)ccc2cnnn2c1 24125,C1(C(=O)OC)CC2CC1CC2NC(=O)Nc1cc(C(F)(F)F)cc(F)c1 24126,CC1CCN(C(C2C(C)C2(F)F)=O)CC1NC(=O)Cc1c(F)cccc1Cl 24127,N1(CC(=O)NCc2cn(CCNC(=O)NC(C)C)nn2)CCCCCC1=O 24128,C1(NC(c2c(Cl)cn(CC)n2)=O)COCCN(C(=O)C(C)Cn2ccnc2)C1 24129,c1(C(N(CCN(C(C(CCC)OC)=O)C(C)C)C)=O)cc2c(cc1Cl)OCCO2 24130,C(C)(C(=O)NCCCCO)OCCC1CC(C(=O)N(C)CCSCC)C1.CCC.CC 24131,N1(C(CC2CC(=C)C2)=O)CCC(CO)(NC(c2cnc(C3CC3)s2)=O)C1 24132,c1(N2CC(C)(C)SCC2)nc(N(C2CCCNC2=O)CCF)nc2c1SCC2 24133,C1(CCc2n(-c3c(SC)cccc3)nc(-c3ccn(C)n3)n2)CCCC2(CC2)C1 24134,c1(CNC(C2CCC2CN(C)C)=O)ccc(CCNC(C2C(C)C2)=O)cc1 24135,Cc1c(CNC(=O)CC2(CNC(=O)CC3CCCC3C)CC2)ncn1C 24136,N1(C(COC(C)(C)C)=O)CC2COCCC2(NC(c2ccn(C3CC3)n2)=O)C1 24137,Cc1cccc(C(=O)N(C2CCC(NC(C3CN(C)C(=O)N3)=O)CC2)C)n1 24138,N1(OCc2c(CC)cccc2)CCC2(CCC(NC(C)(CO)CO)O2)CC1 24139,c1(NC(COC)CO)ccc(S(=O)(=O)NCC2CC23CC3)cc1Br 24140,C1(C(=O)NCCCOCCNC(C(C=C)O)=O)CCC2C(CC1)C2(F)F 24141,N1(C(CCc2c(C)nccc2)=O)CCC(NCc2ccc(F)cc2F)C(F)C1 24142,C=CC(CC(=O)N(CCC1(C)CCCCC1)Cc1ccccc1)c1ccccc1 24143,C(=O)(C1=C(Cl)CCC1)NCC(C1CCN(C(c2cncc(F)c2)=O)CC1)C 24144,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)(C)C 24145,c1(CC(=O)NC2CC2CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1F 24146,C(CN=C(NCc1ccco1)NCc1c(F)cncc1F)C1CC(OC)C1 24147,C1(C(=O)NCC2(C)CCN(C(c3cc(SC)oc3C)=O)C2)CCCCS1(=O)=O 24148,c1(C(=O)NCC2CC(C)N(C(=O)CC3(OC)CCC3)C2)cnc(N(C)C)nc1 24149,c1(C(C(N2CCC(O)(C(C)C)C2)=O)(F)F)ccc2c(c1)OCO2 24150,Cc1cncc(C(=O)NCC2CC2CNC(c2ccc(=N)[nH]c2Cl)=O)c1Cl 24151,N1(C(c2cc(C)nn2C)=O)CCN(C(c2c(C)coc2C)=O)CC12CC2 24152,c1(OC)c(C(=O)NCCCN(C(C23CC(OC)C2C3)=O)C2CC2)csc1Cl 24153,N1(C(CC2C(C)(C)C2)=O)CCCN(C(=O)CC2CC2(C)C)CCC1 24154,Cc1cc(C)nc(C2CN(C(C3CCN(C(C)(C)C)C3C)=O)C2)n1 24155,Cc1ccc(Br)c(F)c1CN1CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 24156,C(=O)(CC(O)C(C)C)NC(CCN(C(C1N(Cc2cc(C)no2)CC1)=O)C)C(C)C 24157,N1(C(CN(C(=O)C(O)C(C)CC)CCC)=O)CC2(COCC(=O)N2)C1 24158,c1(C(=O)NCCN(C(CC2CC(C)C2)=O)C2CC2)cnn(C(C)C)c1N 24159,N1(C(c2ccc(CC)o2)=O)CCc2cc(OC)ccc2C1C 24160,c1(COC)nc(NC2CC(O)(C(F)(F)F)C2)cc(CNC(=O)C(C)CO)n1 24161,c1(SCC(=O)NCC2CC2CNC(c2cccnc2C(F)F)=O)ccc(O)cc1 24162,C(C(=O)N1CC(NC(C2CN(C3CC3)C2)=O)C(c2cnn(C)c2)C1)(C(C)(C)C)SC 24163,c1(C(N2CCC(NC(=O)CSC3CCCS3(=O)=O)C2)=O)cccc2nsnc12 24164,C1(C(N(C(C)C(=O)OC)CCCNC(=O)C2CC2)=O)CCCC1n1ccnn1 24165,C(C(CC(C)C)C(=O)N(C)Cc1c(C)cnn1C)NC(CC(C=C)C)=O 24166,C1(NC(C(CC)NC(C)=O)=O)COCCC1C(=O)N(CC)Cc1cnco1 24167,N1(C(CCCNC(CCCC)=O)=O)CCN(C(=O)CNc2ccccc2C)CC1 24168,c1(CC)cccc(C(=O)N(C)CC2CCCN(C(=O)CN(C)C(N)=O)C2)c1N 24169,c1(OC)ccccc1C(C)=CC(=O)NCCCN(C)C(c1ccc(Cl)c(O)c1)=O 24170,C1(N(C(CC)C)C(C2CCOCC2)=O)CCC(C2CCC2)CC1 24171,c1(CCNC(c2ccc(C)o2)=O)ccc(C(=O)N(C)Cc2ncon2)cc1 24172,N1(C(c2c(OC)nsc2)=O)CC2CC(NC(=O)C#CC(C)C)C2C1 24173,c1(CNC(C2CC(C)CN2CC)=O)c(F)cc(Cl)cc1F.C12C=CC(C1)NC2=O 24174,N1(C(c2n(CC)ncc2)=O)CC2(CC2)CC1C(N1CCC(N2CCC2)C1)=O 24175,C(=O)(CCCCCN=[N+]=[N-])N1CC(C(C)C)N(C(=O)CC(C)c2cnn(C)c2)CC1 24176,CCC(C)C(O)CC(=O)NCCCCCN(C)C(C1(NC(C)=O)CCC1)=O 24177,c1(C(N(CCNC(C(C)SCCCC)=O)CC2CC2)=O)ccn(C(C)C)n1 24178,c1(CC)cccc(C(=O)NC2CC(NC(=O)CC3CCCO3)CC2O)c1 24179,c1(C(N(C2CCCN(C(C(CC(=C)C)C)=O)C2)C)=O)ccc(C#N)c(O)c1 24180,c1(C(=O)NCC(C2CC2)NC(C2C(COC)C2)=O)cc2cc(Cl)cnc2[nH]1 24181,CC1(C)CCCOC1CC(N1CCOC(C(=O)NCc2cncc(Cl)c2)CC1)=O 24182,N1(C(C(C2CCCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24183,Cc1cc(C(N2CCC(CNC(c3nc(O)sc3C)=O)C(C)C2)=O)[nH]c1C#N 24184,C1(C(N(C(c2ccccc2F)CNC(C2OCCCO2)=O)C)=O)C(C)(C)C1(F)F 24185,Nc1ccc(CCCC(=O)N(C)CCNC(C2CCOC(CF)C2)=O)cc1 24186,Cc1ccc(S(=O)(=O)N2CCN(C3CCCN(Cc4ccccc4)C3=O)CC2)nc1 24187,Cc1ncnc(C(N2CC3(CCN3C(C3CCC(=O)O3)=O)C2)=O)c1C 24188,C=CC1CCCCN1C(=O)CC(C)N(C(=O)C(C)S(C)(=O)=O)C 24189,c1(CN2CC3C(CNC(c4ccc(OC)nc4)=O)C3C2)ccc(C)c(F)c1F 24190,c1(CC(=O)NC2CCN(C(COCCCC#C)=O)C(C)C2)cnn2ccccc12 24191,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC(c2cn[nH]c2)C)C2(CC2)C1 24192,c1(N(C)CC2CCC(=O)N2)nc(NCc2ccc(F)c(Cl)c2)c2cnn(C)c2n1 24193,n1(CC)cc(C(=O)NCCC2(NC(=O)CC3CCNC3=O)CCC2)c(C)n1 24194,Cc1ccc2c(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)n[nH]c2c1 24195,c1(C(N2CC(O)(CCNC(C3(C(=O)OCC)CC3)=O)C2)=O)ccc(N(C)C)cc1 24196,c1(C(=O)NCCCNC(Cc2c(C)ccc(C)c2)=O)ccc2c(c1)B(O)OC2 24197,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24198,N1(C(C(C)(C(C)C)OCC)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24199,C1(CC)CCOC1CNC(=O)C=CC(C)NC(=O)CCC1(O)CCCC1 24200,N1(C(C2C(C(C)O)C2)=O)CCCCC1CN(C)C(C1(n2cccc2)CCCC1)=O 24201,C1(C(N2CCC(NC(CCc3cnc(C)s3)=O)C2C(C)C)=O)CCS(=O)(=O)CC1 24202,Cn1cc(C(=O)NC2CC3(C2)CC3C(=O)NCCC23CC(CCO2)C3)ncc1=O 24203,C(=O)(CC(F)(F)F)OC.c1(CCC)nsc(N2CCOCCO2)n1 24204,CC(N=c1[nH]c(N(C)CC2CN(C)C2)nc2c1CCC2)c1nnc2n1CCC2 24205,N1(C(Cc2nnc(SC)s2)=O)CCCC(CN(C(=O)C(c2ccc(C)o2)=O)C)C1 24206,C1(CSC)CCC(c2ccccc2)CC1.c12ccc([nH]1)C(=O)NC1CN(C1)C2=O 24207,C1(COC)CC2(CCO1)CCN(C(C1CN(c3ccccn3)CCC1O)=O)CC2 24208,C(=O)(C1CCc2c[nH]nc21)NC(C(NOCC=C(C)C)=O)Cc1cnc[nH]1 24209,C(C)(CCC(=O)NC1CC1CNC(c1cnc(-c2ccccc2Cl)nc1)=O)OC 24210,C1(CNC(COCC#C)=O)CC2(CCN(C(C3(COC)CC3)=O)CC2)CO1 24211,c1(OCCOCC)ccc(C(=O)NC(C(C)NC(CCOCC)=O)(C)C)cc1 24212,c1(C(c2n(CCC)nnn2)NC(C)CC(C)C)c(F)ccc(Br)c1C 24213,C1(NC(CN(C)CCO)=O)CC2CN(C(=O)C(c3ccccc3)N(C)C)CC2C1 24214,C#CC(C(C)(C)C)NC(=O)C(C)=CCNC(=O)C(C)SC 24215,c1(C(=O)NCCCC(C)NC(=O)C(F)(F)C(F)F)cc(N)c(O)c(F)c1 24216,n1(C(C)(C)C)ncc2c(NC3COC(C4CC4)C3)ncnc12 24217,C(C)(C)(CCCNC(=O)C(C)C(C)C)NC(C1C(=C)CC1)=O 24218,C1(C(=O)NC(C)C(=O)N(C)Cc2cncn2C)CCCC2(CC2)C1 24219,C1(C(=O)NC2(C#C)CC2)CC12CCN(C(C1C3CN(C)CC13)=O)CC2 24220,n1(C(CC)C)ccc(=NC(=O)CCNC(c2nncn2C2CC2)=O)[nH]1 24221,N1(C(C(C)Cc2cccnc2)=O)CCC(OCCNC(C2CC2CF)=O)CC1 24222,N1(C(c2c(COCC)cc[nH]2)=O)CC2CC(NC(c3ccncn3)=O)CC(C2)C1 24223,N1(CCCCNC(C(C)OC)=O)CCC(NC(=O)C(C)(F)F)C1 24224,C(=O)(C1CCCc2nncn21)NC(CCNC(CC1(NC(C)=O)CC1)=O)C(C)C 24225,C(C)(CN=c1cc(COC)nc[nH]1)(C(C)C)NC(c1ccc(CC)cc1)=O 24226,C(C)(CC1CCC1)(C(=O)NC1CN(C(=O)CN2CCCC2)C1)OC 24227,C1(NC(CC(=O)NCC)=O)CCC(F)(CNC(=O)CCc2cccnc2F)C1 24228,C(=O)(C(CCC(N)=O)NC(=O)CCOCCC1CC1)N(C)CCOCCCO 24229,C1(CN(CC(=O)N(CC#C)C)C(=O)OCc2ccccc2)CN(C)CC(C)O1 24230,C1(NC(CCN(C(c2ccc(OC)cn2)=O)C(C)C)=O)COC2(CCCC2)C1 24231,Nc1cccc(C(N2CCN(C(c3ccnc(-n4cccn4)c3)=O)CC2)=O)c1O 24232,C(=O)(CCS(=O)(=O)N(C)C)N(C(C)C)CCN(C)C(c1ccncc1Cl)=O 24233,N1(C(C2C(C)(C)C2(F)F)=O)CCC(C(=O)NCCc2ccnc(O)c2)C12CCC2 24234,N(C(=NCCF)NCCN1CCCCCC1)CC1(C(F)(F)F)CCC1 24235,C#CCCCCCCCNC(=O)C(CC(N)=O)NC(=O)CNC(=O)C(C)CC 24236,C12(OC(C=O)C3CC3)CC(C(=O)NCC3(C(F)(F)F)CCC3)(C1)C2.CCS 24237,C1(C(=O)NCC2C(C(NOC(C(C)C)CO)=O)CC2)COC(=O)N1C 24238,C1(NC(C(CC)(C)CC)=O)CC2CN(Cc3ncc(C(F)(F)F)s3)CC2C1 24239,N1(C(COCCSC)=O)CCC(NC(c2cccc(Cl)c2N)=O)C(C)(C)C1 24240,C12(NC(C3CCC(C)C3)=O)CC(CNC(=O)CCS(C)(=O)=O)(C1)OC2(C)C 24241,c1(C(=O)NCC2CN(C(Cc3scc(C)c3)=O)C2)ccc(Br)nc1C 24242,N1(C(c2n(CC)cnn2)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 24243,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24244,c1(C(=O)NCCC2N(C(C(N3CCOCC3)C)=O)CCC2)cc2ccccn2n1 24245,C1(C(=O)NCC(C2CCC2)OCC)CC(O)CN1C(c1ncccc1Cl)=O 24246,C(=O)(C(CO)C(C)(C)C)N1CC(COC)(NC(=O)Cn2ccc(O)nc2=O)C1 24247,N1(C(CCCC#C)=O)CCC(C(=O)NCC2(O)CCC(C)C2)C12CCC2 24248,c1(CC(=O)NCCC2CCCN2C(=O)CCc2cn[nH]c2)cn(C2CC2)cn1 24249,c1(CNC(C2N(CC(=O)NCC(C3CCC3)OC)CCC2)=O)cc(Cl)ccc1Cl 24250,N1(C(c2ccc(COC)s2)=O)CC(CNC(=O)C(C#N)C2CC2)CC1C 24251,Cn1cc(C(N2CC(O)CC2C(N)=O)=O)c(-c2ccc(Cl)cc2)n1 24252,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2CCC2C)=O)CC1 24253,c1(C(=O)NCC2C(CNC(C(C)(C)OC(C)C)=O)C2)cn2c(n1)CCCC2 24254,c1(C(=O)NC2C3(CC(NC(C(C)C4CCC4)=O)C3)C2)c(F)cc(N)cc1F 24255,c1(C(N2C3C(NC(C(C)O)=O)C(CC3O)C2)=O)ccc2ccnc(Cl)c2n1 24256,C(N=c1nc2c(ncn2C2CC2)c(NCCCCCF)[nH]1)c1c(C)cccc1N 24257,Fc1cc(CCNCc2nc(C3CC3)cs2)ccc1Cl 24258,N1(CC)CCOC(Nc2ccc(NC(c3cc(NC(=O)C4CC4)n[nH]3)=O)cc2)C1 24259,C1(CNC(c2ccc(OCC)cc2)=O)CCC(C)CN1C(c1ncccc1C)=O 24260,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24261,c1(CSC)cccc(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)c1 24262,C1(NC(C(c2cccnc2)C)=O)CC12CCN(C(C1CC(N=[N+]=[N-])C1)=O)C2 24263,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24264,C(C(=O)N1CCC(NC(=O)CCN2CCOCC2=O)C1C)(C(C)C)SC 24265,c1(C(=O)NC(C)CCCNC(c2cn(C3CC3)cn2)=O)cccc2nc[nH]c12 24266,N1(C(C)(C)C)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24267,Cc1ccc(CO)cc1C(=O)NCC1CCCC1NC(=O)CN1C(=O)CCC1=O 24268,N(C(=NCC(C)OC(C)(C)C)NCc1cccc(N2CCOCC2)c1)C(CC)C 24269,CCC(CC(=O)NC(CCOC)C(=O)N(C1(c2cc[nH]n2)CC1)C)C(F)F 24270,C1(C(=O)NC(C#C)C)(NC(=O)CC2CCOCC2)CCSC1 24271,c1(C(N2CCC(NC(C(C=C)O)=O)C(O)C2)=O)c(C)cc(O)cc1C 24272,Cc1cc(C(N2CC3(NC(c4nnc(S)n4C)=O)CCC2CC3)=O)cc(N)c1O 24273,C1(C(N2CC(NC(COCCC)=O)C(C)C2)=O)CCC2(CC1)CC(O)C2 24274,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(C)ccnc2O)=O)CCCC1 24275,CC1(C)CN(C(=O)C#CC2CC2)CC1C(=O)NCC(C1CCCCC1)O 24276,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24277,c1(CNC(C(N(C(C(C)OC)=O)C)C2CC2)=O)cncn1C 24278,C#Cc1ccc(NCC(C2CCN(Cc3ccc(=O)n(O)c3)CC2)F)nc1 24279,C(=O)(CC(C)C(C)(C)C)NCC1N(C(C(CC(=O)OCC)O)=O)CCC1 24280,c1(NC(N(C)CC2C(CC)C2)=O)cc(Br)cc(F)c1OC 24281,c1(C(=O)NCC2C(CNC(C(C)SCC)=O)C2)c[nH]c2c(C)c(C)ccc2c1=O 24282,c1(CC(=O)NC(CNC(CC2(CSC)CC2)=O)C)ccc2c(c1)CCO2 24283,c1(NC(C(OC)OC)=O)cccc(CNC(=O)Cc2sccc2Br)c1 24284,c1(OCC)nc(C2CC2)sc1C(=O)Nc1cc(CNC(C2CC2OC)=O)on1 24285,CC1COCC(C(=O)NCC2CCC2C(=O)NCCN2CC(CF)C2)O1 24286,c1(C(=O)NC2CN(C(C(C)OCC)=O)CC2C2CC2)c(C)[nH]cc([N+](=O)[O-])c1=O 24287,N1(C(CC2CCN(Cc3c(C)nc(Cl)cc3)C2)=O)CCc2cc(O)ccc2C1 24288,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(C)CN(C(=O)CC1CCSC1)C)C2 24289,c1(C(N(C2CCC(NC(C34COCC(C3)C4)=O)C2)C)=O)cccc2nsnc12 24290,c1(C(C)C)cncc(C(=O)NCC2(C)CCN(C(C34CCC3C4)=O)C2)c1 24291,C(=O)(N=S1(=O)CCNC(CNC(=O)OC(C)(C)C)C1)c1c(C)c(Br)c(Br)s1 24292,N1(C(C(=O)NCC)=O)CC=C(C(C)(C)C(=O)NCC2OCCC2(C)C)C1 24293,C1(CCNC(C(CC)O)=O)CCN(C(c2cc(C(C)=O)ccn2)=O)CC1(F)F 24294,C1(C(=O)NCCC2(CC3CC3)OCCO2)Cc2ccncc2C1 24295,C(CC(C(=O)NCCc1ccc(F)nc1)NC(C1OCCC1C)=O)=CC 24296,C12(NC(C3CCC(C)O3)=O)CC(CNC(C3(N(C)C)CCC3)=O)(C1)OC2C 24297,Cc1ccnc(C(N2CC(C)(OCC(=O)NC3CC(=O)NC(C)C3)C2)=O)c1F 24298,c1(-c2cc(C(=O)NCC3C(CNC(C=CCOC)=O)C3)n[nH]2)ccccc1Br 24299,c1(COC(=N)O)ccccc1Br.c1(CC(F)F)cccc(Cl)c1 24300,c1(C(N2CC(CNC(C)=O)C(C)C2)=O)ccc(Nc2[nH]cnc2C#N)cc1 24301,c1(N2CCN(C(CN(C(=O)C=CCF)C)C3CC3)CC2)ncnc2c1ncn2C 24302,c1(CCCCC)cn(CC(N2CC(F)(F)C2CC)=O)nn1 24303,CC1CC(c2nnnn2CCN(C)C)(NCC2CC2n2cc(Br)cn2)CS1 24304,N1(C(CC2(CSC)CCC2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CO)CC1 24305,N1(C(C(c2ccccc2F)C)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24306,N1(C(CCC2CCC(=O)C2)=O)CC2CCC1CN2C(C1C2COCC12)=O 24307,C1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)Cn2cccn2)CCC(O)CN1C 24308,Cc1nc2ccc(-c3cncnc3C(=O)NCc3cncs3)cc2[nH]1 24309,N1(CC(=O)N(C)CCNC(C2(F)C3CCCC23)=O)CCc2ccccc2C1 24310,C1(C(=O)NC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24311,Cc1csc2c(NC3CCC(NC(c4ccccc4CO)=O)CC3)ncnc12 24312,c1(C(=O)NC2(CNC(C3(CCCC)CCC3)=O)CCC2)cc(F)cc(Cl)c1O 24313,c1(OC)ccc(N(C(=O)C(c2ccoc2)NC(c2cn(CC)nc2C)=O)C)cc1 24314,C(=O)(CC(C)(C)C(F)F)N1CC(Cn2cc(CCN3CCC(OC)CC3)nn2)C1 24315,C(CC(CC)C(=O)N1CCCC(OC(C)C)C1)=CC.C1(C(=O)OC)CN1 24316,N=c1[nH]n(Cc2ccccc2-c2cncc(Cl)c2)cc1-c1c[nH]nn1 24317,c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)c(C)nc2sc(C)cn12 24318,C1(NC(c2sc(C)c(Br)c2C)=O)CCCC2CN(C(c3cncs3)=O)CC12 24319,C1(c2ccccc2)(C(=O)NCC(C)NC(c2cc(C(=O)C(C)C)c[nH]2)=O)CCCO1 24320,c1(C(N2CC(NC(COC)=O)C(F)CC2)=O)cnc2[nH]c(C)nc2c1 24321,CC(C)C(C(=O)NCC(C)NC(C1(F)CC1)=O)c1ccncc1 24322,CC1CCC(C(=O)N(c2ccccc2N(C)C)C2CCCNC2)CN1CC#N 24323,Cc1nc(NCC2CCCN(C)C2)cc(Cc2cccc(OC(F)F)c2C(F)F)n1 24324,n1(CC)nc(C)cc1C(=O)NCc1ocnc1C(=O)N(C12CC(C1)C2)C 24325,c1(C(=O)NC(C2CCCCN(CC3CCCO3)C2)C)cnc(N)c(Cl)c1 24326,Cc1ccc(-c2cc(-c3cn(C4C=CCCC4)nn3)n[nH]2)s1 24327,C1(CC(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)(C)C)COCCN1C 24328,CN=c1[nH]ccc(C(N2CCC(C)(C)C2CNC(C2CCC(C)CC2)=O)=O)c1N 24329,c1(CCC)ccc(C(=O)N(C2CN(C(C3CC(N4CCCCC4)C3)=O)C2)CC)s1 24330,CCCCC(CNC(C1CCN1CC)=O)NC(=O)Cn1cc(C(F)(F)F)nn1 24331,C#CC1CCCC(c2nnnn2C2CCCC2)(NC2CCN(C)CC2C=C)C1 24332,c1(CC)cccc(C(=O)N(C2CC(NC(c3cnc(O)[nH]3)=O)C2)C)c1O 24333,c1(C(N2CCCCC(NC(c3scc(OC)c3)=O)C2)=O)cnc2nncn2c1C 24334,N1(C(CCOCC(C)(C)C)=O)CC2(CCN(C(C3CN(CP(C)(C)=O)C3)=O)C2)C1 24335,N1(C(C(COC)(F)F)=O)CCC2(CCN(C(=O)CN(c3cccc(Cl)c3)C)C2)C1 24336,c1(CC)ccc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)cc1Br 24337,C1(NC(C=C(COC)C)=O)CN(C(C2CCC(OC(F)(F)F)C2)=O)CC1N=[N+]=[N-] 24338,c1(NC(c2cn(C3CC(O)C3)nn2)=O)ccc2c(O)ncnc2c1 24339,C(=O)(C(C)C(F)(F)C(F)F)NCC(C1CC1)NC(c1cc(SC)c(N)cc1)=O 24340,c1(C(=O)NCCC2CCN(C(C(n3cccn3)OC)=O)CC2)cc2n(c1)CCC2 24341,n1(-c2cc(C)cc(F)c2)nc(-c2cn(C3COCC3O)nn2)nc1C1=NOC(C)C1 24342,CC1CN(C)CC1NC(C1CCN(C(=O)Cn2cnnc2O)CC1)=O 24343,c1(C(N2C(N(C)C)C(C)(C)C2)=O)ccc2nnn(C(C)(C)C)c2c1 24344,CC1CCNC(=O)C1NC(C1CCC(CNC(=O)CC2CCCCC2)O1)=O 24345,C(CC)(CCCC(=O)NCc1ccc(O)cc1)NC(C1CC(OCC)C1)=O 24346,CCCCC(CO)NC(C1CC=CC(NC(c2cnnnn2)=O)C1)=O 24347,C1(C(=O)NCCCN(CC)CC)(NC(=O)CCC2CC2)CCOC1 24348,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24349,c1(CCC2(C)CC2)cc(N(CCC(F)(F)F)CCNC2CC2)ncn1 24350,c1(C(=O)OC)[nH]c(=NCC(C2CC2)NC(=O)C(c2ccccc2F)OC)sc1C 24351,CC1CCCC(N=c2nc(N3CC4C=CCC(C4)C3)c3c([nH]2)CCOC3)C1 24352,C1(COC)(NC(c2cocc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24353,c1(CC(=O)NC(CC(C)NC(CCOCC(C)C)=O)C)ccc(F)cn1 24354,c12csc(c1)C(=O)NC2.c1(NC(C2(C(F)F)CC2)=O)cnn(CC(F)F)c1 24355,CCC(C)C(C(=O)NC(C)CC(=O)O)OC.c12ccnc(c1)NC2=O 24356,C1(C(N2C(CNC(=O)CN3CSCC3=O)CCCC2)=O)CCC=CCCC1 24357,N1(c2n(-c3cccc(C(=O)OC)c3)nnn2)Cc2nccn2CC(NC(C)=O)C1 24358,C(=O)(CCC(CF)CF)NCC1(F)CC(CNC(=O)C(F)(F)C(F)F)C1 24359,C1(NC(Cc2c(C)scc2)=O)CN(C(=O)C(C2CCOCC2)C)C2(CCC2)C1 24360,C(CS(=O)(=O)c1ccc(F)cc1F)OC(CCC1(C(C)=O)CCC(=O)N1)=O 24361,C12(CCCNCC1)c1noc(n1)CC2.C(=O)(C1=CCOC1)OC 24362,c1(CNC(=O)C(=O)NC2(C(=O)OC)CCC2C2CC2)ccc(OC)cc1Cl 24363,Cc1c[nH]c(C#N)nc1=NC(=O)c1ccnnc1 24364,Cc1ncc2n1CC(C(N1CC3CC3(NC(C3CCN3S(C)(=O)=O)=O)C1)=O)CC2 24365,C1(NC(C(CCCCC)O)=O)CCN(C(c2c(OC)ccnc2O)=O)CC12CCC2 24366,c1(C(C(=O)N(CC(=O)NCC(C)N(C)C)C)C)cccc(O)c1 24367,C(C(CC(C)C)C(=O)N(C)Cc1ccncc1)NC(C(CCC)CC)=O 24368,N1(C(CCC=C)=O)CC2COCCC2(NC(=O)Cc2cccc3c2NC(=O)C3)C1 24369,N1(C(C2N(C(C3CCC(=O)OCC3)=O)CCCC2)=O)CCC2(CCC2)CC1 24370,c1(C(=O)NCC(=O)NC2C(CNC(=O)CCCN=[N+]=[N-])C2)ccccc1Cl 24371,C(=O)(C(F)(F)C(O)C1CC1)N1CCCC(N2CCN(C(c3cnc(S)[nH]3)=O)CC2)C1 24372,C(=O)(CCc1ccc[nH]1)NC(C1CC1C(=O)N(C)Cc1ncco1)C 24373,C1(CC(=O)OC)CC(N=c2[nH]c3c(c(=NCCCCCS(C)(=O)=O)[nH]2)CSC3)C1 24374,N1(C(C2CCC(NC(c3cncc(Cl)c3)=O)C2)=O)CCn2ncnc2C1 24375,c1(C(=O)NCC2C(CNC(CC3C(C)(C)C3)=O)C2)cocc1Br 24376,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24377,C(C1CN(C(c2cnn3c2OCC3)=O)CC1C(=O)NC(C)CCC(C)C)=CC 24378,n1(CC(C)CO)nc(-c2cccs2)nc1-c1cccc(-c2ccncc2)n1 24379,C(=O)(C(F)C(C)CNC(c1ccc(F)c(O)c1)=O)N1C(COC)COCC1 24380,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(CC)=O)C1 24381,Cc1ccc(F)cc1-n1cc(C2(O)CCCCCC2)nn1.C1(=O)CCCN1C 24382,C(=O)(C(F)C(F)(F)F)NC(C)(CCCl)n1cc(-c2cccc(S(C)(=O)=O)c2)nn1 24383,Cc1cncnc1C(N1CCCCC1CC(=O)NC(c1ccoc1)C)=O 24384,CC(C)CS(=O)(=O)CCC(=O)NC(C=CCCC=CCNC(=O)CNS(C)(=O)=O)=O 24385,CC1(C)CC2N(C1)CC1CN(CC1O)C(=O)C2.C1(C(=O)NC)CCS1(=O)=O 24386,C1(C(C)CNC(=O)CN(C)C(=O)C2CC2)CC(F)(F)CN1C(=O)CCc1cn[nH]c1 24387,CCCCCC(CC)C(=O)NC1C2CCC1N(C(=O)C=Cc1cccc(Cl)c1)C2 24388,c1(CC(=O)NC2CC2c2cc(Cl)ccc2Br)ncc([N+](=O)[O-])cn1 24389,N1(C(=O)CSCCNC(C2C=CCS2)=O)CC=CC12CCCCC2 24390,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(C1CN(C)C(=O)N1)=O)C2 24391,Cc1cc(C(F)(F)F)nn1CC(=O)NCCNC(=O)C(c1ccccc1F)(C)F 24392,N12CCCC(C1)N(C)C(=O)c1coc(c1)C2.C(C)(CC1CCC1)S.CCO 24393,N1(CCNc2ccc3ncc(C(=O)OC)n3n2)Cc2ccc(F)cc2CC1C 24394,C1(C(=O)NC2(CF)CCN(c3c(C)c(Cl)ncn3)C2)CCOC2(CCCCC2)C1 24395,c12cncc(c1)O2.N1(C(C(C)SC)=O)CC(NC(=O)COC2CCC2)C(CO)C1 24396,c1(NCC(C(C)C)OC)ccc(S(=O)(=O)NC(c2cccnc2)C)c(Cl)c1 24397,C1(NS(CC=C)(=O)=O)CC2(C1)CN(C(c1cc(I)ccc1O)=O)C2 24398,C1(CC(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24399,CC1(C)CN(C(=O)CC2CC(O)C(F)C2)CC(C)(C)C1NC(c1cccc[n+]1[O-])=O 24400,C1(NC(=O)C=CCN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24401,C(=O)(CC(O)CC(C)C)N1C(C(=O)NC2C(OC)C(C)(C)C2)CC(C)C1 24402,c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(C2C=CCCC2)=O)C3)=O)cc1F 24403,C1(CN(C)CC2(CC)CCCC2)NC(=S)N(C)C2=C1C(=O)N(C)C2C 24404,C(C(=O)N1OC2CCC1CC2)NC(C=CC(C)NC(=O)C(F)OC(F)(F)F)=O 24405,C1(c2c(C)nc(-c3ccncc3)n2C2CC2)CCC2(CC1)OCCO2 24406,C(C)(CCCNC(=O)CCSc1nncn1C)NC(C=CCOC)=O 24407,c1(C(C)C)ccc(C(c2nnnn2C2COC2)NCC2(CCO)CC2)cc1F 24408,Cc1cc(O)cc(=O)n1CC(N1CC(CNC(=O)CCC(C)(F)F)C2CC12)=O 24409,C1(CNC(CN(S(C)(=O)=O)C)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)C2CC12 24410,C=C=C(C)CC(=O)N1CCC(O)(C(C)NC(=O)Cc2cnn(C)c2C)C1 24411,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24412,N1(S(CC(C)N(C)C)(=O)=O)CCN(C(=O)CNC=O)C(C)(C)C1 24413,c1(C(=O)NC(C2N(C(CSCC)=O)CCC2)C)ccc(=O)oc1 24414,N12CCC(C(C)(C)C1)NC(=O)c1ccnc(c1)C2.n1(CCCNC)cc(Cl)cn1 24415,C(=O)(C(O)C(C)CC)NCC1(NC(C(F)(F)NS(CCCC)(=O)=O)=O)CCC1 24416,N1(C(CN(CC(C)C)C(c2c(C)con2)=O)=O)CC2CC2C2CC12 24417,c1(NC(CC(C)F)=O)sc2c(c1C(=O)Nc1cccnc1)CCCC2 24418,c1(OCC(=O)NCC(C)N(C(C(c2cccc(F)c2)C)=O)C)ccc(Cl)cc1 24419,N1(C(=O)C(N2CCC(N3CCCC3=O)C2)=O)CCc2c(Cl)ccc([N+](=O)[O-])c2C1 24420,N#Cc1c(N2CCC(F)(CNC(C34CC=CCN3CCC4)=O)CC2)cccc1F 24421,c1(C(N2CCC(O)(C(C)NC(=O)CS(N)(=O)=O)CC2)=O)nc(N(C)C)nc(=N)[nH]1 24422,Fc1cc(Cl)cnc1-c1nnc(N2CC3CCC(C2)O3)n1C 24423,C(=O)(C(C)(CNC(=O)CN1CCC(OC)CC1)CC)NC(CC)CC 24424,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24425,c1(C(=O)NCC2OCCCN(C(CSC(C)C)=O)C2)cccc2nc(O)[nH]c12 24426,N1(C(CC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccc(C3CCC3)cc1)=O)C2 24427,c1(C(=O)NC23CCN(C(=O)Cc4nc[nH]n4)CC2C3)ccc2ccsc2c1 24428,N1(C(CCCOC)=O)CC2CCCC(N(C(=O)CC3CCCC34CC4)C)C2C1 24429,CC#CCCCC(=O)NC1CN(C(c2cccc(C(=O)OC)n2)=O)CC1F 24430,C(=O)(C(CCC(C)C)NC(c1ccnn1-c1ccccc1)=O)OCCC 24431,CCC(O)C(C)C(=O)N1CCCCC(NC(c2ccc(F)nc2F)=O)C1 24432,c1(OC)ccc2nc(N3CC(CO)(NC(c4c[nH]nc4-c4ccco4)=O)C3)sc2c1 24433,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(C2(P(C)(C)=O)CC2)=O)CC1(C)C 24434,N1(C(C(CC)F)=O)CC2(C1)CN(C(c1ccc(C3CCOC3)cc1)=O)CC2CO 24435,CCC(C)(CO)C(=O)NCCC1CC(NC(=O)C(C(C)C)n2cnc(C)c2)C1 24436,C12CCC(CC1)C(=O)N2.c1(OC)cc(CC(=O)NC(C)CN(C)C)on1 24437,c1(OC)cccnc1C(=O)NC(CNC(=O)CCSc1nnnn1C)C1CC1 24438,N1(C(C2CCN(C)C2=O)=O)C(CC(=O)NC(c2ccsc2)(C)C)C2CCCC12 24439,C(C(C)(O)CC)NC(C1(CNC(C2CC(=C)C2)=O)CCC1)=O 24440,CC1CCSCCN1C(c1ccc(CN(C)C)s1)C(=O)NC1CC(F)(F)C1 24441,C(=O)(C(C)(C)C(C)(C)C)NCC(=O)NC1C(CNCc2cccc(C)c2)C1 24442,Cc1ncnc(C)c1CC(N1CCN(C(c2csc(CO)n2)=O)CC1CO)=O 24443,C1(CC)(CNC(=O)CC2CCOC2)CCN(C(=O)CNC(=O)C(F)(F)F)C1 24444,N1(C(C=CCOC)=O)CC2(CCC(NC(=O)Cc3ccsc3S(C)(=O)=O)CC2)C1 24445,c1(CN(c2cc3ncnn3cn2)C2(C#N)CCN(C3CC3)C2)[nH]nc2ncccc12 24446,c1(-c2c(CC)ccs2)ccc2c(c1OC(C)C)OCO2 24447,C1(NC(c2c(OC)scc2)=O)CC2CC(C1)CN(C(c1ccc(O)nc1)=O)C2 24448,CC(CC(N)=O)C(=O)NC1(CNC(c2cccc(O)c2)=O)COC1 24449,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24450,N1(C(CC=C)=O)CCOC2(CCCN(C(c3cc(Cl)n(C)n3)=O)C2)C1 24451,c1(C(=O)NC(C2CCN(C(=O)CC(C)(C)C3CC3)C2)C)cccnc1O 24452,N1(C(COCCCOC)=O)CCC(NC(c2cc3c[nH]nc3s2)=O)C(O)C1 24453,Cc1ccccc1C(N1CCC(NC(=O)CCSc2nccn2C)C2CC12)=O 24454,C(=O)(C1CCCc2nn[nH]c21)NCC(CC=C)NC(c1ccc(C)s1)=O 24455,N1(C(C=C(C)Cl)=O)CC(CNC(C23CCC(C)(CC2)CO3)=O)CC12CCOCC2 24456,CCC1(N=c2[nH]nc(SC)s2)CC(CC(C)C)C(=O)Nc2c(cccc2)C1.OC 24457,C1(C(N2CC(CCNC(=O)C=C3CC3)(OC)C2)=O)CC1C1CCCC1 24458,C(CCC(=O)N1CC2(CCC2(C)C)C1)(C(C)C)NC(c1cccc(CC)n1)=O 24459,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)CN(C)C)nc2n(c1Cl)CCCC2 24460,N1(CC(N2CCC(CNC(C(c3ccccn3)C)=O)C2)=O)CCC(=O)CC1 24461,CC1CC(CNC(=O)C(C)OC2CCCC2)CN(C(c2cncc(F)c2)=O)C1 24462,c1(CN2CCC(C(=O)NCc3cnccc3Cl)C(O)C2)cccc2c1OCCO2 24463,c1(CCNC(c2ccnn2C2CCC2)=O)cccc2c1OC(F)(F)O2 24464,N1(C(Cc2c(C)occ2)=O)CC2(CCCC2)C1C(=O)NCC12CC(CCO1)C2 24465,N1(C(CSCC#C)=O)CCn2ncc(N(C)C(c3ccc4nncn4c3)=O)c2C1 24466,C1(N(C(CSCCOC)=O)C)CCN(C(=O)Cn2nc(C)oc2=O)C1 24467,c1(CC(=O)NCCN(C)C(C2CC2[N+](=O)[O-])=O)cncc(F)c1 24468,Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCc2nccs2)nc(O)n1 24469,N1(CCCCCNC(C2CCC(OC)C2)=O)CCN(C(=O)COC(C)C)CC1 24470,N1(C(C(C)Oc2cncc(Cl)c2)=O)CCCC(F)(C(=O)NOC2CSCCO2)C1 24471,C1(C(=O)N(CC)CC)(OC)CCN(C(c2ccc(C)o2)C)CC1.CCO 24472,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24473,C1(NC(=O)C=Cc2cnc[nH]2)CC2CC(NC(=O)CCc3cscn3)CC2C1 24474,Cc1cc(C(=O)NCC2(C)CCN(C(c3nnn(C)c3N)=O)CC2)ncc1Cl 24475,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NC(C1CSC1)C 24476,C1(C(N2CCCC(CN(CCCCCC(=O)OC)C)C2)=O)CCC(N=[N+]=[N-])CC1 24477,Cc1nc(-c2ccn(C)n2)sc1C(N1CC(NC(=O)C(C)C(C)C)C1)=O 24478,C(=O)(CC(CC#N)c1ccccc1)NCCCN(C(=O)C(F)OC(F)(F)F)CC 24479,C1(CC(=O)NCCC2CCN(C(C3(O)CC(F)(F)C3)=O)C2)CCCOCC1 24480,c1(C(=O)NCC2CCC(NC(c3cc(C)on3)=O)C2)cc2c(C)cc(F)cc2[nH]1 24481,N1(CC)CCOC(C(N2CCOC(CN(C(=O)CC(F)(F)Br)C)C2)=O)C1 24482,CCN=C(NCC(C)SC)NCC(c1cccc(OC2CCOC2)c1)F 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24606,c1(C(N2C(CN(C)C(C3CC=CCO3)=O)CCC2)=O)cc(Br)ccc1O 24607,CCC(CO)C(=O)NCc1cccc(CN(C(=O)C(C(C)O)NC(C)=O)C)c1 24608,C(=O)(CCCCC(=O)NC(C1(CNC(c2cnc(N)cn2)=O)CC1)C)OC 24609,Cn1cc(N)c(C(N(C2CCN(C(c3ccc(Cl)s3)=O)C2)CCO)=O)n1 24610,S(=O)(=O)(c1ccnc(N2CCOCC2)n1)NC1(C)CC2C=CC1C2 24611,c1(C(N2CCC(C(C)C(=O)NC3CCCCC3C)CC2)=O)cc2ccccn2c1 24612,c1(C(C(=O)NCCC(C)Sc2ccccc2)C2CC2)ccccc1.C1(C(=O)N)CC1F 24613,C1(C(N(C)CC2CCCO2)=O)CCC=CC1NC(=O)C(=O)NC1CCC1 24614,Cc1ccc(F)c(OCC(N2CCC(CNC(=O)Cc3ccccc3F)C2)=O)c1 24615,C1(C#N)(C(=O)NCC(C2(O)CN(C(C(CCC)=CCC)=O)C2)(C)C)CC2CC2C1 24616,n1(CC(=O)NC(COC)OC)cc(C(C)N(C)C)nn1.C12CN(C1)C(=O)CS2 24617,Cc1cc(Br)cc(C(N2C3CCC2(CNC(=O)COC(C)C)CC3)=O)c1N 24618,c1(NCCN2CCN(CCNC(C3C(CC)C3)=O)CC2)cc2c([nH]1)CCCC2 24619,N1(C(COCC)=O)CCC2CCN(C(=O)Cc3c(C)nn(C(C)C)c3C)CC2C1 24620,c1(N2CC(C(=O)Nc3ccc(C#C)cc3)C(O)CC2)ncnc2sc(Br)cc12 24621,Cc1c(C(=O)NCCCOCCNC(=O)CC(C)c2ccco2)ccn1C(C)C 24622,CCCC(C(=O)Nc1ccc(CCO)cc1)NC(C1CCCS1)=O 24623,c1(OC)cc(C(=O)N(C(C)CN(C(=O)C(C)CC2CCC2)C)C)ccc1C(C)C 24624,CC1(C)C(CNC(C2(C(F)F)CCC2)=O)CCN1C(C1(CF)CC1)=O 24625,c1(CNC(N(C)Cc2nnnn2C)=O)cn(C)nc1C(C)(C)C 24626,N1(C(c2c(OC)csc2)=O)CC(C)(CNC(C2CC3CCC2CC3)=O)CC1(C)C 24627,C1(C(=O)NCC2CN(C(C(C)CC3CCCO3)=O)C2)C2CC3C(C2=O)C13 24628,N1(C(C(C(C)C)NC(=O)C2=CCCOC2)=O)CC(C)(C)CCC1C 24629,C1(C(N2CC(C(=O)OCC)C2)=O)CC(=O)CN1C(=O)CCOCC 24630,Cc1ncc(N)cc1C(=O)NC(C)CCNC(C1(c2ncco2)CCC1)=O 24631,CN1CCN(C(=O)C(C)(C)CC2CCC2)CC1C(=O)NCC1CC1CO 24632,c1(C(=O)NC)cccc(C(N(CC(=O)NC(C)CNC(C)(C)C)C)=O)c1 24633,C1(C(N2CCCC(O)(Cn3cc(CC(=O)O)nn3)C2)=O)CS(=O)(=O)CC12CC2 24634,C1(NC(CCCNC(C)=O)=O)CN(C(=O)Cc2cc(F)cc(F)c2)CCC1CO 24635,C1(C(=O)NC2CCCCN(C(c3ccco3)=O)C2)CCC2C(CC1)C2(F)F 24636,c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCC2(C)C)cnc2ccnn2c1C 24637,C(=O)(C1Cc2ccccc21)NCC1CCN(C(CC(C)C(F)F)=O)CC1 24638,N1(C(CC(C)OC)=O)CC(C)(C)OCC1CNC(=O)CC1CC2(CC2)C1 24639,C1(C(=O)NC(CNC(c2n(C)ncc2)=O)C(C)(C)C)CCCCN1N=O 24640,N1(C(COC2CN(C(CCc3onc(C)n3)=O)C2)=O)CC(O)CC(O)C1 24641,c1(OCC)cc(Cl)ccc1CNCCN1CC(=O)NC(C)C1 24642,N1(C(C(C)(C)C2CC2)=O)CCOCC(C(=O)NCC2(CC3CC3)CCC2)C1 24643,N1(C(CCOC)=O)CCOCC(CNC(c2cccnc2OCC(F)F)=O)C1 24644,C=CCCCC(C(=O)NCCC(C)CC(C)(C)C)NC(c1ccsc1C)=O 24645,Cc1cc(CC(=O)NC(C)CCNC(=O)CC2CCOC(C(C)C)C2)c(C)o1 24646,c1(C(N2CC3(C(NC(c4cc(C)[nH]c4C)=O)CC3)C2)=O)c(Cl)nc2sc(C)cn12 24647,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24648,C1(C(=O)NC(C2CCCC2)CNC(C2NC(=O)OC2)=O)CCS(=O)CC1 24649,CC1(C)CC2(CN1CC(=O)NC1CCC1)C(F)(F)C2(F)F.c12ccccc1CO2 24650,c1(CNC(COC(Cc2cncc(C)c2)=O)=O)cccc2ccccc12 24651,N1(C(c2n(CCCC)ncc2)=O)CC(NC(c2cc(O)ncn2)=O)CC(O)C1 24652,N1(C(C(c2ccccc2)NC(c2ccc(OC)nn2)=O)=O)CCC(O)C(O)C1 24653,CC1CCc2[nH]c(=NCC34CCCC3C4)[nH]c(=NCC3COC(C)(C)CO3)c2C1 24654,CCCC(CCC)CCCC(=O)NCCCNC(=O)CC(C)(CC)C(=O)OCC 24655,n1(CC(=O)NC2C(NC(C(C)C(F)(F)F)=O)CCCC2)ccc(=O)n(C)c1=O 24656,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1CNC(=O)N1)=O)CC2 24657,c1(C(N2CCC(CNC(CC3N(CC)CCC3)=O)CC2)=O)cc2c(ncn2C)s1 24658,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(c2ccsn2)=O)C1 24659,N1(C(=O)NC(CCC)C(=O)OC)CC(OC)CC(C)C1 24660,CC1CCN(C(=O)CSCC(F)(F)F)CC1NC(C1(CCF)CC1)=O 24661,C1(c2cc(C)no2)CCCCCN1C(=O)C(C1CCN(C(=O)OC(C)(C)C)C1)O 24662,CCC(CC)C(C)C(=O)NCC1C2CN(C(C3CCC(C)=C(C)C3)=O)CC12 24663,c1(CNC(C2(C)CCN(C(=O)C(=O)C3CCCC3)C2)=O)cnc(O)c(F)c1 24664,C1(C(C)NC(CC(C)SC)=O)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1 24665,N1(C(=O)C=CC2CCN(C(C3(F)CC=CCC3)=O)CC2)CCC2CCCC2CC1 24666,c1(-c2c(C)cnc(F)c2)cccc2c(C(=O)NCC(C)O)n[nH]c12 24667,C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)CO)CCOC(C)(C)C1 24668,c1(C(=O)NCC2N(C(CN(C(C)=O)C)=O)CCCC2)ncc(Cl)cc1Br 24669,C1(C(=O)NCC(C(C)C)NC(CCc2ccc(C(=O)OC)[nH]2)=O)CC(C)(C)CN1C 24670,C1(CNC(c2cncc(C)c2)=O)CN(C(c2cnn(C)c2C)=O)CCC12CCC2 24671,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(C1CCOC1)=O)C2 24672,O=C1CCCC(C(N2CC(F)(CNC(c3nc(Cl)cs3)=O)C2)=O)C1 24673,C12CCC3(CCN(CC3)C1)C2.C12(C(CC=CC(=O)NCC(F)(F)F)=O)CCCC1C2 24674,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24675,Cc1ccn2ncc(C(N3CC4CC(NC(=O)CCCOC(C)C)C3C4)=O)c2c1 24676,N1(C(C=Cc2c(C)ncs2)=O)CCN(C(c2occc2F)=O)C(C)CC1C 24677,C12(CC(=O)NCC(CNC(c3cc(COC)[nH]n3)=O)C)CCC(CC1)C2(C)C 24678,Cc1c[nH]c(=NC(=O)c2cnc(NC(c3snnc3C)=O)cn2)cn1 24679,c1(C(=O)NCC2(NC(C(C)OC3CCCCCC3)=O)CC2)ccc(P(C)(C)=O)o1 24680,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCC(C)SC)cc1Cl 24681,c1(C(=O)NCC(C)NC(=O)Cc2cc(F)ccc2O)cc(F)c2cn[nH]c2c1 24682,c1(C(N2C(CN(C(C(COC)C)=O)C)COCC2)=O)cccc2[nH]cc(Cl)c12 24683,C12CC(F)(C1)CNC(=O)C=CC(=O)C2=O.c1(C(=O)OCC)cc(Cl)no1 24684,c1(OC)nc(C(N2CCCC(C)(NC(C3CC3C(F)F)=O)C2)=O)cc(O)n1 24685,c1(SC)nc(N(C)CC2CCCN(C(c3cscc3Cl)=O)C2)cc(C)n1 24686,c1(OC)cc(C(=O)O)cc(C2CC2)c1N.c1(S)ccc(C)cc1 24687,Cc1cnncc1C(=O)NCC1CN(C(c2nc(CC3CC3)cs2)=O)CC1O 24688,C1(NC(C2CCCCCC2)=O)CN(Cc2ccncc2Br)CC(F)(F)C1 24689,C(=O)(CC(C)CCC)N1CCC(N(C(C(=Cc2ccco2)C)=O)C)C1 24690,c1(CNC(CCSCC)=O)ccc(CCNC(c2ccncc2F)=O)cc1 24691,CS(=O)(=O)C1(C(N2CC3CC(NC(=O)COc4ccsc4)C2C3)=O)CCC1 24692,CC1CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CCC1N(C(=O)CSc1cn[nH]c1)C 24693,c1(CN2CCC(NC(=O)CSc3nc[nH]n3)CC2)c(Br)ccnc1Cl 24694,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)C1CC1 24695,Cc1ncnc(C)c1CC(N1CC(O)(CNC(=O)Cc2c(O)ncnc2O)C1)=O 24696,C12(F)CCC(C1)CN2.c1(C(=O)OCC)sccc1OC(c1conc1CC)=O 24697,C1(CN(C)C)CCCN1C(=O)CCn1cc(CCC2CCOCC2)nn1 24698,C(=O)(CC(C)C(F)F)N1CCC(CN(C(c2ccnc(OC)c2)=O)CC)CC1 24699,CCC(C)(C#N)C(=O)NCc1ccc(C(=O)NC2(CC(N)=O)CC2)s1 24700,c1(C(=O)NC(CNC(=O)C(F)OC(F)(F)F)C2CC2)cc2c([nH]1)CCOC2 24701,S(=O)(=O)(c1ccc(C(=O)NCC#CCNC2CC(F)C2)cc1)N(C)C 24702,Cc1cnn(C)c1CNC(=O)Nc1nnc(N(C)C)s1 24703,CON=CC(=O)N1CCC(C(=O)NC2CCOCC2C)O1 24704,N1(Cc2c(C)cc(Cl)cc2)CC2C3CCC(C2C1)N(C(c1ccncn1)=O)C3 24705,c1(C(=O)NC2CC(C)CN(C(c3ccc[nH]3)=O)C2)ccc2c(c1)CCCC2 24706,CCCCC(O)CC(=O)NCCCC1CCCN1C(=O)CCSC(F)(F)F 24707,N1(C(C=C(C)C)=O)CC(NC(C2(N(C)C)CCCSC2)=O)CC2(CCC2)C1 24708,CCC(C)(CO)C(=O)N1C(C(=O)NCCCC2CCCCO2)CCC1C 24709,Cc1cccc(-n2cc(C(=O)NC(C)(CNC(C3CNC(=O)N3)=O)CO)nn2)c1 24710,c1(N2CCC3(CN(C)C3)C2)ccc(Br)c(S(=O)(=O)NC2C(CO)C2(C)C)n1 24711,CC(C)C(C)(C(N)=O)NC(C1CC2CC2N1C(C1CC2C=CC1O2)=O)=O 24712,c1(CCC(N2CCCC(c3ncn(-c4ccccc4)n3)C2)=O)ccc(Br)nc1 24713,c1(OCC=C)ccccc1C(=O)NCC(C)NC(C1CC(CCN(C)C)C1)=O 24714,c1(C(=O)NC(CNC(C2C(c3n(CC)cnn3)CC2)=O)(C)C)cc(N)ccn1 24715,c1(N2C(CC(=O)N(CC)CC)C(C)(C)CC2)ccc(F)cc1[N+](=O)[O-] 24716,c1(CC)nn(C)cc1C(=O)N(CC(CC)NC(=O)C(C)Cc1cccc(F)c1)C 24717,c1(C(=O)NCC2CN(C(C(C(CC)O)C)=O)CC2C)cncc2c[nH]nc12 24718,C(c1ccc2cc(OC)ccc2c1)=CC(=O)NCCNC(CCC(=C)C)=O 24719,c1(C(=O)NCc2c(C3CCN(C(C)=O)C3)n[nH]c2)cccn2c(C)nnc12 24720,Cc1csc(=NCC(=O)N2CCC3CCCC23CNC(=O)C(=O)NCC2CC2)[nH]1 24721,C(=O)(C1CCCc2nc[nH]c21)NC1CC(NC(c2csc3ncnc(O)c23)=O)C1 24722,C1(C(=O)NCC2C(NC(c3nc(OC)c(C)s3)=O)C2)CCc2ncnn2C1 24723,c1(OC)cc(N2CC3CN(C(c4ccco4)=O)C3C2)nc(C)n1 24724,C=CCC(CNC(=O)C(C1CCOCC1)F)C(=O)NCCC1CC=CCC1 24725,c1(C(=O)NCC2COCCN(C(=O)CCc3nc[nH]n3)C2)ccc2n[nH]cc2c1 24726,N1(C(c2c(C)[nH]nc2C(F)F)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24727,C(=O)(C(O)C(C)(C)C)NC1CCN(CCCNC(Cc2cnc(C)[nH]2)=O)C1 24728,C(CNC(=O)CCCN(C)C)(C(C)(C)C)N(C)CC1C(C)C1.C(CC=O)N 24729,C(=O)(CCCS(C)(=O)=O)N1C(CCNC(=O)C(C)n2cncn2)CC(OC)C1 24730,C(=O)(CS(=O)(=O)CCO)NCC(C1CC1)NC(C1(CC#C)CCOCC1)=O 24731,Cc1n[nH]c(C)c1C(C)C(=O)NCCC1CCCN1C(=O)CC1(N(C)C)CC1 24732,c1(N(C2C3CCC2CNC3)C(c2n(C)ccc2)=O)nc(Cl)c(Br)cc1O 24733,N1(C(C=COCC)=O)CCCC(N(C)C(c2ccc(OCCF)cc2)=O)CC1 24734,C(=O)(C(CNC)CC(C)C)NC1(CC)CCC1.C12(CCCCC1)CC(=O)N2 24735,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24736,Cc1cccnc1CC(=O)NC1CC(C(N2CC(N(C)CCO)C2)=O)C1(C)C 24737,c1(OC)cc(F)c(CN2CCOC(CNC(c3ccc(Cl)cc3)=O)C2)c(F)c1 24738,c1(CC(C(=O)NCC2(F)CN(C(CCNC(C3C(C)C3)=O)=O)C2)F)ccc(F)cc1 24739,c1(CONC(C2C(OCC)CCC2)=O)ccccc1Br 24740,c1(NC(C(C)NC2CC(C)(CC)C2)=O)cccc(OC(F)(F)F)c1 24741,c1(C(C(=O)NC)N(C(C)C)CC2(C#N)CC2)ccc(-c2ccc(C)o2)s1 24742,c1(OCC)cc(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2(O)CCC2)ccn1 24743,c1(SC)cc(C(=O)NC2CN(C(=O)COCC(F)(F)F)CC2C)c(C)o1 24744,O=C(C1=NOCC1)N1CC(C2CCCCN2C(=O)C(O)CC2CCCCC2)C1 24745,C(CCCCCN=C(N)NC1CC(c2ccccc2F)C1)C1C=CCC1 24746,C1(NC(CN(CC#C)C(c2cc(OC)ns2)=O)=O)CCCOC12CCC2 24747,c1(CC)cc(C(=O)NC2(C)CN(C(C3(C)CNC(=O)C3)=O)C2)nn1CCO 24748,c1(C(=O)NCC(CNC(C2CN(C)C(=O)CC2)=O)F)c(F)ccc2[nH]ccc12 24749,c1(CNC(=O)C(c2ccccc2)=O)cccc(NC(C2CC(Cl)(Cl)C2)=O)c1 24750,c1(C(=O)NCC(CC)NC(C2C3CC(=O)CC23)=O)nc(C)oc1C 24751,C(C(=O)N(CC(=O)NCc1nonc1C)CC(C)C)(C(C)C)SCC 24752,c1(OC)ccccc1OC(C)C(=O)NCCC(C)NC(c1c[nH]c(C#N)c1)=O 24753,C1(C(=O)OCC)CCN(C(C2CN(C(c3ocnc3C(C)C)=O)CCS2)=O)CC1 24754,C12(C(N3CC(=CC=CCC)C3)=O)CCCC1CCN2C(c1cnnc(C)c1C)=O 24755,CN1CCC(CC(=O)NC(C)(CNC(=O)CN(C2CCC2)C)C2CCC2)CC1 24756,N1(C(C2CC23CCCC3)=O)CC2CCC1C(CNc1ncc(O)cn1)C2 24757,C1(NC(c2cc(CC)nn2C)=O)CC2CC1N(C(c1cnn(C)c1C)=O)C2 24758,CCC(C(=O)N1CC(CO)(NC(C2COCCN2CC2CCCC2)=O)C1)C(C)C 24759,Cc1cc(C(N2C3CC2CN(C(c2c(O)cccc2Br)=O)C3)=O)cc(Br)c1 24760,Cc1ccc2cc(C(=O)NC3CCCC3(C)CNC(=O)C(=O)N(C)C)cnc2c1 24761,c1(-c2occ(C(=O)NC3CCC(C(=O)OC)CN3)n2)ccc2c(c1)CCC2 24762,Cc1ccc(NNC(=O)c2csc3cc(Br)ccc23)cn1 24763,c1(OC)cc(C=CC(N2CCC(C(C)NC(=O)C=C3CCC3)C2)=O)sn1 24764,c1(C(=O)NCCC2(O)CCCN(C(C3CC3F)=O)C2)ccc2cccc(Cl)c2n1 24765,N#Cc1ccc(Cl)c(C(=O)NC2CC2NC(C2CCOC2c2ccccc2)=O)c1 24766,c1(C(N2C(C(=O)NCc3n(C)cnc3)CC3CC32)=O)n[nH]c2c(F)cccc12 24767,O=C(C(Cc1ccccc1)CC(F)(F)F)NCC1CCN(C(c2nncs2)=O)C1 24768,C1(NC(CCCOC)=O)CCC2CCN(C(=O)C=Cc3cncn3C)C1C2 24769,c1(CNC(N2CC(C(=O)OC)OC(C)C2)=O)ccc2sc(C)nc2c1 24770,C12CCC(C1)CC(=O)N2C.c1(C(=O)NCC(O)C2CC2)ccc(CO)o1 24771,Cn1nc(C(=O)NC2CCC2NC(c2cn(C(C)(C)C)nn2)=O)cc1Cl 24772,CC1CC2(C(N3CCCC3C3CCN(C(=O)C=CCF)C3)=O)CC12 24773,C1(C(=O)NCCC2(CNC(COCC#C)=O)CC2)CC=CCO1 24774,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24775,N1(C(c2ccc(C(C)C)cc2)=O)CCC(NCCN2C(=O)COCC2=O)C1(C)C 24776,CC(CC(=O)NC1CCC(NC(c2ccc(OCCO)nc2)=O)CC1)C(F)(F)F 24777,C=CC(CC)CC(=O)NCC(C(=O)NCc1ccc(N(C)C)o1)C(C)C 24778,c1(CNC(C(=O)NCCCC(=C)C)=O)nc(Cl)ccc1Cl 24779,c1(OC)ccc(C(C(=O)NCc2cccs2)N(C2CCC2(F)F)C)c(C)c1 24780,N1(Cc2nnc(-c3ccc(OC)c(OC)c3)o2)CCCC(C2CCC2)CC1 24781,c1(CN2CCC(NC(C(c3ccnn3C)C)=O)C(O)C2)ccc(F)c(C#N)c1 24782,C12(CC(=O)NC3CCCC(NC(c4conc4C4CCC4)=O)C3)CCC(CC1)C2 24783,C(C(=O)NCCCC(C)NC(=O)CCNC(c1ccco1)=O)(C(C)(C)C)SC 24784,Nc1nc(C(=O)NCCNC(c2csc(C(F)F)n2)=O)ccc1Br 24785,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)N(C2CCCC2O)C)C1 24786,N1(C(Cc2c(C)non2)=O)CCC(C)(C(N2CCC(OC(C)C)C2)=O)C1 24787,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24788,N1(C(C2N(CCC)C(=O)CC2)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 24789,C(=O)(CCCCC#N)NCC1CN(C(COCCC=C)=O)C(C)C1 24790,C1(NC(CCN(C)CC)=O)CC2CC(C1)N(C(=O)Cc1ccccc1Cl)C2 24791,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCC(C)(C)CO2)=O)C1)=O 24792,C(=O)(C1=CCC(C)CC1)NC1(CO)CCN(C(C(CCC)NC(N)=O)=O)C1 24793,C(=O)(CCCC(N)=O)N1CCC(NC(C2C(C)C2(F)F)=O)C1C1CC1 24794,CCN=c1[nH]cc(C(=O)NCCCN(C)C(c2cnoc2C)=O)s1 24795,CCC1(C)CNC1=O.C1(C(N(C)CCF)=O)C=CCC(C(=O)O)C1 24796,C1(C)(C(=O)NCC(CCNC(C(C(C)C)n2cnnn2)=O)O)CC2CCC(C1)S2 24797,N1(C(c2nc(Cl)c(Cl)s2)=O)CCc2sccc2C1c1ccccc1 24798,c1(N2CCCC(NC(C3(C)CCC(O)CC3)=O)CC2)ncnc2cccc-2n1 24799,Cc1cnc(C(N2CC3CC2C3C(=O)N(C)Cc2cnn(C)c2C)=O)c(F)c1 24800,c1(OC)ccc(C)cc1C1(C(=O)NC(C)CNC(C2C3CCC2CC3)=O)CCCC1 24801,c1(C(N2CCSCC2C2CCC2)C(=O)N(CCCCCC)CC)ccccc1F 24802,N1(C(c2ccc(C#C)cn2)=O)CCC(C)(C)C(NC(=O)C=CC=CC)C1 24803,c1(CC(=O)NC(CN2CCN(C(C(F)=CC)=O)CC2)(C)C)ccc(OC)c(OC)c1 24804,Cc1cccc(CNC(=O)CCOCCCC2CC2)c1NC(=O)C(F)C(C)C 24805,N1(C(c2n[nH]c(C)c2C)=O)CC(C)(CNC(=O)C(c2ccccc2)O)CC1(C)C 24806,C1(C(N2CC(C3N(C(CCC(=C)Cl)=O)CCC3)(O)C2)=O)CCc2cnc(C)n2C1 24807,C=C=CC(C)C(=O)NC1(CO)CC(C(=O)NOC(=O)CCCOCCOC)C1 24808,N1(C(c2ccc(C3CC3)s2)=O)CC2CCCC(N=c3ccn(CCO)[nH]3)C2C1 24809,CCC(CCCC(=O)N1CC2COCC2O1)NC(C1(C)CCCCC1C)=O 24810,N1(C(CCC(C)OCC)=O)CCN(C(c2cnc(C)s2)=O)CC1CC(F)(F)F 24811,CC1CCN(C(c2ccc(Cl)o2)=O)CC1NC(=O)Cn1cccnc1=O 24812,N1(CC(C(=O)OC)NC(c2ccc(C)o2)=O)CC(c2cccc(Cl)c2)OCC1C 24813,CCCCC(C)C(=O)NCCn1cc(CNC(=O)CSc2ccc(Cl)cc2)nn1 24814,c1(C(N(C(CCNC(C=NOC)=O)C)C)=O)cccc2c(C)coc12 24815,C=CC(CCC)CC(=O)NCc1ccoc1C(=O)NC1(C)CC1(C)C 24816,C1(NC(C2(CCC=C)CC2)=O)CC2CCC1CN(C(c1cn(C3CC3)cn1)=O)C2 24817,C(=O)(CCC(C)(C)O)NC(C(C)C)CNC(=O)Cc1ccc(C(N)=O)cc1 24818,C1(C(=O)OCC)(CO)CCN(C(C2CC3(CSC3)C2)=O)C1.C12CN(C1)C2=O 24819,N1(CCC2CCC(C)O2)CCN(C(C2CCCC2)=O)CC1 24820,c1(C(=O)NCC2C(NC(c3ccc(CN(C)C)cc3)=O)C2)cnn2c1CCCC2 24821,C1(NC(C(C(=O)OCC)F)=O)Cc2ccccc2C1.C1(CCC2CCC2)C(=O)N1 24822,c1(CCC(=O)N(C2CCNCC23CC3)C2CC2(F)F)ccc(F)c2c1CCCC2 24823,O=C(CC1CCOc2ccccc21)NC1CN(C(c2nccc(Br)c2)=O)C1 24824,Cc1cc(-c2cncnc2C(N(C(CO)CC(C)C)c2ccccc2)=O)c(C)cc1O 24825,C1(C(C)C)CCCCC1N(C(=O)O)C.C(C)(O)(CCO)C1CN(CC)C1 24826,CCC(C)(C)C(=O)N(CCNC(=O)Cn1nccc1C)C1CC1 24827,C1(CC)CN(C)CCCN1C(=O)C(CC(N)=O)NC(=O)C(C(C)OC)N(C)C 24828,c1(Oc2cc(C)c(N3C(=O)CCC3=O)cc2)ccc2c(c1)CNC(=O)N2 24829,c1(OC)ccc(N(CCCCC2CN(C(=O)C(CC)NC(C)=O)C2)CC)cc1 24830,C1(OC)CC(COC(C2CC3CNC(C2)O3)=O)CCC1O 24831,Cc1cc(CNCC(C(=O)C(Cc2cn[nH]c2)NNC2CC2CC(C)C)=O)no1 24832,c1(C(C)NC2CCCC=C2Br)ccc(Cl)c(Br)c1 24833,CC1(CNC(c2cncc(N)n2)=O)CCCN1C(=O)CSC(=N)N 24834,C=CC1(C(=O)NCC(C(C)C)NC(c2cncc(OCC(F)F)c2)=O)CCOCC1 24835,c1(C(=O)NC(C)CN(C(=O)CCCn2ccccc2=O)C)cc(Cl)ccc1N 24836,CCCC(C)C(=O)N1CC(CNC(=O)C(=O)NC2CC(F)(c3ccccc3)C2)C1 24837,C1(Oc2ccccc2)CCC(NC(C)=O)CC1.N1(C(C2C(=C)C2)=O)CC2(C1)C(=O)N2 24838,N1(C(C(C)C2CCCO2)=O)CCC2(CCCN(C(=O)Cc3ccon3)C2)CC1 24839,N1(CCC(C)C)CC(C(=O)NC(C)(C)C(C)NC(c2ccc(F)cc2)=O)CC1=O 24840,C1(NC(CCCCCOC)=O)CC2(CCN(C(c3cc4n(c3)CCC4)=O)CC2)C1 24841,c1(CC)ccc(N)c(C(=O)NC(CNC(=O)C=Cc2nc(C)co2)C2CC2)c1 24842,C1(CC(=O)N(CCNC(C(C)NC(c2cccs2)=O)=O)C)CNC(=O)C1 24843,N1(C(C(CC)C(C)C)=O)CC2CN(C(C34CC(C)(C3)OC4C)=O)CCC12 24844,C=CCC(CC)C(=O)N1CC(O)(C(C)NC(=O)CSS(C)(=O)=O)C1 24845,C1(C(=O)NCC(CC)n2cccn2)CN(C(c2cc(C)[nH]n2)=O)CC12CCC2 24846,C(CC(C)CNC(C1C(NC(C2CC(Cl)(Cl)C2)=O)C1(C)C)=O)OC 24847,C=CCCCCC(=O)NC1CCCN(C(c2cc(OC)ncc2F)=O)C1C 24848,N1(C(C2(C)CC2(F)F)=O)CC(CNC(c2cscc2F)=O)C2(CCC2)C1 24849,N1(C(C(COCC)N=[N+]=[N-])=O)CC2CC(NC(c3ccc(F)c(CC)c3)=O)C1C2 24850,c1(C(=O)NN2CCCC(O)C2)ccccc1O.C1(C)CC1C(=O)N 24851,N1(C(CC2=NNC(=O)C2)=O)CCC2CCN(C(C3CC(n4ccnc4)C3)=O)C2C1 24852,C1(C(=O)Oc2ccnn2C2CCC2)CS(=O)(=O)CCN1C(=O)N 24853,c1(C(N2CCC(NC(C3CC4(CC4)CO3)=O)C23CC3)=O)noc2c(F)cccc12 24854,C(=O)(C(C)(C)CN1CCOCC1)NC(C)CC1CN(C(=O)CCN2CCC2)C1 24855,Cc1ccnc2sc(C(=O)NCC3CC3NC(=O)Cc3ccc(O)c(F)c3)c(C)c12 24856,CC1CN(C(=O)CC2(CO)CCCC2)CCC1CNC(C1CCCCC(=O)C1)=O 24857,C(=O)(CCNC(=O)N(C(=O)C=CC(C)C)C1CC1)NCC=C 24858,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 24859,CC(C)CC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1ccccc1N=[N+]=[N-] 24860,c1(C(=O)NCCN(C(=O)C(O)CCN(C)C)CC)onc(CC)c1C 24861,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2noc3c2CCCC3)=O)CCC1(C)C 24862,C(C(O)CC(=O)N(C)CCN(C(=O)CCC1CCCC1)CC(=O)N(C)C)NC(N)=O 24863,CN1CCC(N=c2[nH]c(=NCc3ccc4ncsc4c3)c3sccc3[nH]2)CC1=O 24864,C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1CC(NC(CC(C)N(C)C)=O)C1 24865,C1(OCCOC)CCN(C(c2cn(CCO)nn2)=O)C1C1CC1.C(C(=O)OC)=C 24866,C(C(c1nnnn1C)Sc1ncccc1C)(C(C)C)NCCNc1scc(C)n1.C1CC1 24867,C(CO)(C(=O)NC(c1cscn1)CO)NC(=O)COCC1CCCO1 24868,C1(NC(=O)CCOCCF)C2CC3CC(C2)CC1(CNC(=O)Cc1cccs1)C3 24869,c1(S(Oc2ccc(C3(N)CC3)c(OC)c2)=O)ncnc2c1ccn2C.CO 24870,C(=O)(C1=COc2ccccc2O1)N(C(CNC(C1ON=C(C)C1C)=O)C)C 24871,c1(CC(=O)NC(CC(C)C)CNC(=O)C(O)C2CC2)c(F)c(F)cc(F)c1F 24872,c1(OC)ccc(C2CC2C(=O)NCCCCNC(=O)C(F)(F)c2cscn2)cc1 24873,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 24874,C1(NC(C(c2ccccc2)(C)O)=O)CCCCN(C(C2CCC(N(C)C)CC2)=O)C1 24875,C1(C(=O)NCC2(C)CCC(NC(CCC=C(C)C)=O)C2)CC12CC(C)(C)C2 24876,C(=O)(C(C)CS(=O)(=O)NC1CCC(SC)C1)OC 24877,CCC(c1ccccc1)=CC(N1CCC(C(C)(C)NC(=O)C(O)COC)CC1)=O 24878,C1(C(=O)NCCCN(C(C2CC(C)CO2)=O)CC)CCCOCC1 24879,c1(C(N2CCCCC2(C)C2CC2)C(=O)NCC=C)cc(C)c(Br)cc1F 24880,N1(C(C2C(OC)CCC2)=O)CCCCC(C(=O)NCCC2(CO)CCC2)C1 24881,N1(C(C#CC(=O)O)=O)CCC2(CCN(C(c3cc(Cl)c4n[nH]cc4c3)=O)C2)C1 24882,C1(CC(=O)NCC(C)N(C)C(c2n[nH]cc2C2CCC2)=O)CCn2cncc2C1 24883,C(N=c1cc(C(N)=O)nc[nH]1)C1CN(Cc2cc(Cl)nc(=N)[nH]2)CC1C(F)(F)F 24884,C=CC(O)C(=O)N1CCC(n2cc(CNC(=O)C(=O)NCC(F)(F)F)nn2)C1 24885,C1(NC(c2ccsn2)=O)COCCN(C(=O)CCc2ccsc2)C1 24886,c1(NC(C(=O)N(CC(C)(C)NC(C(CC=CC)C)=O)C)=O)cc(F)cc(F)c1 24887,C(=O)(C1SCc2cccnc21)N(CCCNC(c1cc(COC)[nH]n1)=O)C 24888,C(=O)(C1CCc2c(F)cccc21)NCc1cc(OC)ns1 24889,C1(c2nc(C3C(c4nnc(C(C)=O)o4)OCC3)on2)CCOC(C)C1 24890,C(=O)(C(C)(C)CNC(=O)CCCOC(C)C)NCC(C1CC1)OCC 24891,c1(CC)cccc(CC(=O)NCC2CC(C)N(C(=O)CCn3cccc3C)C2)n1 24892,c1(OC)cc(I)c(C(N2C3CCC2CC(c2cnn(C)c2)C3)=O)cc1OC 24893,c1(NCC(=O)NCCCN(C(=O)CCc2cnco2)C2CC2)nncs1 24894,N1(C(c2cnn(CC)c2C)=O)CCC(CNC(=O)CCCC2CCCC2)C(O)C1 24895,N1(C(C(N2CC(N(C(c3cc(C)[nH]n3)=O)C)C2)=O)=O)CCCC(C)C1 24896,c1(C(N2CC(NC(C(C)CF)=O)C2)=O)nc(-c2ccccc2)[nH]c1C(F)(F)F 24897,C=CCC(C(=O)NCC(CCOC)NC(c1[nH]nc2ncccc12)=O)C(C)C 24898,c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc2cc(F)ccc12 24899,C1(NC(CN(C(=O)CN2CCCC2C)C(C)C)=O)COCCOC1 24900,C(C(=O)Nc1cn(C)nc1C1CCCN(C(=O)COC2CC2)C1)(C(C)C)SCC 24901,C1(CCC(=O)NC(CCCNC(C(C)NC(CC)(C)C)=O)C)CCCC(O)C1 24902,c1(CC(=O)NC2CC(C)(NC(c3ncccc3F)=O)C2)ccc2ncccc2c1 24903,C1(OC)CC(NC(c2cn(C)c(=O)n2C)=O)CN(C(=O)Cn2cccn2)C1 24904,CC1(CNC(C2CCC(N(C)C)C2)=O)CCCN1C(=O)C(O)C1CCCC1 24905,C1(C(=O)N(C2CN(C(C)C)C2)C)(CC)CCN(C(=O)C(C)(CO)NC(C)=O)C1 24906,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 24907,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 24908,C1(CNC(C(C)CCO)=O)COCCN(C(c2cnc3n2CCC3)=O)C1 24909,S(=O)(=O)(c1cc(C)ccc1C)N(CC(CC)CC(C)C)C1CC2CC1CN2 24910,c1(C(=O)NCC(CO)C2CCC2)ncc(C2CC2)s1 24911,c1(OC)cc(OC)cc(C(N2CCNC(C(=O)OC(C(=O)NC(C)C)C)C2)=O)c1 24912,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)C)coc(S(N)(=O)=O)c1 24913,CCCCC(CC)C(=O)N1CCCC(C)(CNC(=O)Cc2ccc(Br)cc2)C1 24914,C1(OCC)CN(C(c2cn(C)nc2C(F)F)=O)CC1CNC(=O)CCC(F)F 24915,c1(C(=O)NC2CCCN(C(C3CC3F)=O)C2)c(OCF)cccc1Br 24916,c1(C(N2C(CNC(c3scc(OCC)c3)=O)CC2)=O)n[nH]c2ccccc12 24917,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 24918,c1(C(=O)NC(Cn2cc(-c3c(C)csc3Cl)nn2)C)ccc2c(c1)CCNC2=O 24919,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC23)CC1)N1CCOC1=O 24920,Cc1cccn(CC(N2CCN(C(=O)CCCCCN(C)C)CC2C)=O)c1=O 24921,N1(C(CC(C)C2CC2)=O)CCC2CCCC12CNC(=O)CCOC1CCOCC1 24922,c1ccc2ccccc2c1O.c1(C(=O)NO)cccc(OC(F)(F)F)c1 24923,c1(CC)cc(C(=O)NCCCN2CCN(C(=O)C=CC(C)C)CC2)cn(C)c1=O 24924,N1(C(C(C2CCN(C(CCCOCCC)=O)C2)(C)C)=O)CCCC2C(O)CC12 24925,N1(C(C2CC(CCNC(C(C)n3ccnn3)=O)C2)=O)CC(C)(C)C12CCC2 24926,c1(C(=O)NC(CC)C(N2CC(O)CC(C)(C)C2)=O)ccc(C#N)c(C)c1 24927,C1(NC(C(C)C(C)O)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 24928,C(CCCC(C)(C)C(=O)NNC(=O)C1CSC1)NC(c1cc(C)c(C)nn1)=O 24929,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2cccn2C2CC2)=O)C(C)C1)=O 24930,c1(C(=O)NC2C(NC(C3(C(C)(F)F)CCCC3)=O)C2)cccc(CCO)c1 24931,C(=O)(CC(C)C(F)(F)F)N1CC(CC(=O)N(C)CC2COCCO2)(OC)C1 24932,C1(F)(CNC(C(C)NC=O)=O)CCN(C(C2SCCC2C)=O)CC1 24933,N1(C(C2CCCC(C(C)=O)C2)=O)CCCC(C)(CNC(c2cn(CCF)nn2)=O)C1 24934,N1(C(c2c(C)snc2)=O)CCCCC(CNC(c2c(C#N)cnn2C)=O)C1 24935,NS(=O)(=O)CC(=O)NC1CN(C(C2C3CNC(=O)C23)=O)CC1O 24936,c1(C(=O)NCC(CC)NC(=O)C(c2ccccc2OC)=O)cn(C)nc1C(C)C 24937,N1(C(=O)C(F)(F)C2CCC2)CC(C2CCCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 24938,Cc1ccc(C)c(CC2CCN(C(c3cc(C4CC4)[nH]c3C3CC3)=O)C2)c1 24939,c1(C(=O)NCC(C(C)C)NC(C2CCc3c[nH]nc3C2)=O)cncc2ccsc12 24940,C1(NC(c2cnn(-c3ccncc3)c2)=O)CN(C(=O)C=C(Cl)Cl)C2(CCC2)C1 24941,C(=O)(CC(C)(C)CC(=O)NC1(C2CC2)CCN(C(=O)C(C)(F)F)C1)OCC 24942,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2occc2C2CC2)=O)CC(O)C1 24943,C(=O)(CC(F)(F)CC(=O)NC(C)CN(C(=O)COCC1CCCOC1)C)OC 24944,N1(C(C(c2n(C)cnc2)O)=O)CCCC(C(C)(C)O)C1.C1=CCNC1=O 24945,C(=O)(C1CCCCc2ccccc21)N1CC(O)(CCNC(CCCOC)=O)C1 24946,c12cc(ccn1)C(=O)NC2.N1(NC(COCC(=C)C)=O)CCC1CC 24947,NS(=O)(=O)CC(=O)NCCN1CCC(NC(=O)CC(F)(F)F)C1 24948,c1(C(N2C(CNC(C(C(CC)C)O)=O)CC2)=O)ccc2nc(COC)[nH]c2c1 24949,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NCCc2cnc(C)s2)c1C 24950,N1(C(C2C(C)C2)=O)CC2OCC(CNC(=O)CCSCc3ccccc3)C2C1 24951,CC(c1cccnc1)=CC(=O)NCC1CC2CCC1N2C(c1ccc(F)s1)=O 24952,c1(C(C(=O)NC(c2ncc[nH]2)COC)NC(=O)C(=O)NOC)ccnc(OC)c1 24953,c1(C(=O)NCCC(C)CCNC(=O)CCn2cnccc2=O)cc(O)nc(O)n1 24954,CC(CC(=O)NCC1C(C(=O)NC(CC(N)=O)C2CC2)C1(C)C)C(F)F 24955,CCCC(CC1CCCC1)C(=O)N(CC(C)(C)NC(=O)Cc1ccncc1Cl)C 24956,c1(OC)cc(F)c(F)cc1S(=O)(=O)N(C1CCCNC1=O)C 24957,c1(OC)ccc(C(=O)O)cc1S(=O)(=O)CN(C(C1C(NC(=O)C(C)S)C1)=O)C 24958,C(=O)(C(C(C)(C)C)NC(=O)C(C)C)NCCC1(NC(CCC(C)OC)=O)CCC1 24959,C(CNC(=O)CC1(n2ccnc2)CC1)(CC(F)(F)F)NC(c1c(C(C)C)ocn1)=O 24960,c1(C(=O)NC2CC(NC(c3cc4ccccn4n3)=O)C2)ccc([N+](=O)[O-])cc1Cl 24961,C1(CNC(C(C#C)(C)C)=O)CCCN(C(c2ccnc(NC3CC3)c2)=O)CC1 24962,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(CC)c2)=O)C1C)C(C)C 24963,Cc1nn(CCO)c(C)c1C(=O)NCC(C)(C)OCCNC(=O)CCC1(C)CC1 24964,CC1CCC(NC(C23CC(C2)C3)=O)CN1C(=O)Cc1cccc(O)c1F 24965,C1(CNC(CC(C)CN(C)C)=O)CC2(CCN(C(=O)Cc3ccno3)CC2)C1 24966,N1(C(C(C)(C)CO)=O)CCCC(CO)(NC(c2cnn[nH]2)=O)C1 24967,c1(OC)ccnc(C(=O)NC2(CC(N3CCCC4(CC4)C3)=O)CC2)c1 24968,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 24969,c1(C(C2(CCCC)CC2)NCC2(C3OCCO3)CC2)nnnn1CCC1CC1 24970,CC1CN(C(=O)CC(O)c2ccccc2)CC(c2ccc(Br)cc2)O1 24971,C1(NC(C(CC)NC(C)=O)=O)CC2CN(C(=O)CNC(C3CCCC3)=O)CC2C1 24972,c1(C(=O)NC(CCCNC(C(CC)SC)=O)c2ccccc2)cc(C)cc(Cl)c1N 24973,C1=C(CSC2CC2)CCN(CC2CC2)CC1 24974,C1(NC(=O)COCC2CCCC2)Cc2ccccc2N(C(=O)C(O)C2CC2)C1 24975,c1(OC)ccc(COCCC(=O)NCC2C=CCN2C(C2C3COCC23)=O)cc1 24976,c1(C(N2C(CC(=O)NCc3ccc(Cl)o3)CCC2)=O)csc(-c2ccsc2)n1 24977,c1(-c2ccc(CNC(=O)CSc3ccncc3)o2)c(F)cccc1Cl 24978,c1(OC)cnc(F)c(C(=O)N(C(C)CNC(c2cncc(C(=O)NC)c2)=O)C)c1 24979,S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NCC1N(C(CC=CC=C)=O)CC1)C(C)O 24980,CCC(C)CC(=O)C(=O)NC(CSCC)C(=O)NC(C)CCN1CCCC1 24981,CC1(C)CCCOC1CC(=O)NC1(C)CN(C(=O)C(c2ccccc2F)(C)F)C1 24982,N12CCCCC(C1)N(C(C1CC(OC)C1)=O)C(=O)C2.N1(CCC)CCN(C)CC1 24983,C12(C(N3CC(CC(=O)OC)C3)=O)CCN(C(C3(C)C=CCC3)=O)CCC1C2 24984,C1(CCNC(CCCOCCOC)=O)CCCN(C(=O)Cn2cnnn2)CC1 24985,CC(C(=O)N1CCC(N(C)C(C2CCCN2CC(F)(F)F)=O)CC1)C(F)(F)F 24986,N1(C(CC(C)O)=O)CC23CCCC2(C1)CN(C(c1cc(C(F)(F)F)no1)=O)C3 24987,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(F)cc2)C1C 24988,CC1CCN(C(c2cscc2Cl)=O)CCN1C(C1CCc2nc[nH]c2C1)=O 24989,c1(CN(CC(C)NC(C23CCC(OC)C2C3)=O)C)cc(C)ccc1F 24990,c1(OC)ccc(SCC)cc1.n12nnnc1C(c1cc(C3CCC3)[nH]n1)NCC2 24991,N1(C(CN(C(=O)CCC2CC(C)C2)CC)=O)CC(CC)OCC1C 24992,C1(CNC(CC=C(C)C)=O)CN(C(=O)CC2CCCCCC2)CC12CCC2 24993,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(c2c(NC(C)=O)cccn2)=O)CC1 24994,C(CC)(C(=O)NC1(C)CC(NC(=O)CCn2ccnc2C(C)C)C1)=CC 24995,Cc1noc(C(C)C)c1C(=O)N.c1(S)ccccc1F.C(=O)(CO)N1CC1 24996,N1(C(C(C)O)=O)CCCC(C(=O)N(C(C)CC(F)(F)F)C)CC1 24997,c1(C(=O)NCC(c2ccccc2)N(C(C(COC)OCC)=O)C)ccncc1F 24998,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 24999,c1(C(=O)NC2CCCN(C(C3(C)C(C)(C)CCC3)=O)C2)n[nH]c2c1CCCC2 25000,c1(SCC(C2CCN(c3ccnc(N4CCC4)n3)CC2)C)ccc(Cl)cc1 25001,C1(=CC(=O)NC(CNC(C23CSCC2C3)=O)C2CC2)CN2CCC1CC2 25002,CC1CCN(C(c2conc2C(C)(C)C)=O)CC1NC(=O)CC1CCC(=O)N1 25003,C#CCCC(O)C(=O)NCC(c1ccccc1)NC(c1sc(C)nc1C)=O 25004,CC1CCC(C(=O)NC(CN(C)C(c2cnc(C3CC3)[nH]2)=O)(CO)CO)CC1 25005,c1(OC)ncc(C(=O)N(C(C)CNC(=O)C(O)C2CC2)C)c(C)n1 25006,O=S(=O)(c1cnn2ccc(=NCCN3CC4CC4C3)[nH]c12)NC1CC(CF)C1 25007,C(=O)(N=S1(=O)CCc2ccccc21)Nc1c(C)oc(S(C)(=O)=O)c1 25008,c1(CNC(c2nc(C)oc2)=O)cc2n(n1)CCN(C(=O)C(C)CC1CCC1)C2 25009,CCCC(C(=O)N1CC(O)(CCNC(=O)C(=O)N=S(C)(C)=O)C1)S(N)(=O)=O 25010,CC(CC#N)C(=O)NC(C(N1CCC(C(F)F)CC1)=O)c1ccco1 25011,CC1CC(CO)CCN1C(=O)N(c1ccccc1C(=O)NNC(=O)c1ccccc1)C 25012,CCC(C(=O)N1CC(CNC(=O)CC2CCOC2=O)C1)N(C)C 25013,N1(C(C(c2cc(C)c(NC(=O)NC(C)C)o2)C2CC2)=O)CC(COC)OC(C)(C)C1 25014,N1(C(C2(OC)CCCC2)=O)C2CCCC1CC(NC(=O)C(C1CC1)SC)C2 25015,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CC(=O)N(OC)C3)=O)=O)ccc12 25016,C1(C2CC2)(C(N2C(C(C)C)CCCC2)=O)CN(C(C2C(C)(C)C2(C)C)=O)C1 25017,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25018,C1(C)(NC(c2c(C(C)NC(c3cn(CCC)nn3)=O)noc2)=O)CC(F)(F)C1 25019,CCCC(O)CC(=O)NCC1CCN(C(c2ccc(COC)o2)=O)C1(C)C 25020,N1(C(=O)C=Cc2cocn2)CCCC(C2CN(C(=O)Cc3cc[nH]c3)C2)C1 25021,C1(CC(=O)NC2CN(C(c3ccc(C)o3)=O)C2)COCCOC1 25022,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)NCCCc2nccs2)(CC)C1 25023,c1(COC)ccc(CC(C)NC(C2(C)C=CCC2)=O)cc1.C1C(=O)N1 25024,C(=O)(CC(C)C(F)F)NC(C)C(=O)NC1CCCCC1Nc1ccc(F)c(F)c1 25025,C(CC(C)(C)CC(=O)NC1COCCC1NC(c1cc(C(C)=O)cn1C)=O)OC 25026,Cn1c(C(N2CC3CCN(C(=O)COCC4CC4)C3C2)=O)cnc1[N+](=O)[O-] 25027,N#Cc1cc(NCCc2cccc(F)n2)cc([N+](=O)[O-])c1Cl 25028,Cc1nc(C(=O)NCC(C)(C)NC(=O)C(C)(C)CF)ccc1[N+](=O)[O-] 25029,N1(C(CC(C)c2ccncc2)=O)CCSCC1C 25030,Cn1ncc(Cl)c1C(c1nnnn1-c1ccon1)NC1(CCNC(N)=O)CCC1 25031,c1(C(N2CC(NC)C2)=O)cccc(Cl)c1Cl.CC(Cc1ccco1)C(=O)C(C=C)=O 25032,C(=O)(CCCCNC(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25033,Cc1cc(O)cc(C)c1OCCCNC(=O)CN1CCC(OC2CCCC2O)CC1 25034,C1(CNC(CSC)=O)CN(C)CCN1C(c1cn(C(C)(C)C)nn1)=O 25035,C1(=O)C(CCCC)NC(=O)C(C)CC(C)(C)C(C=C)(CCC)N1CC 25036,Cn1ncc(Cl)c1NC(C1(C2CCCN2C(=O)CCOC2CCOCC2)CC1)=O 25037,C1(C)(CC)CCN(C(C2CCCCCN2C(=O)C(C)NC(N)=O)=O)CC1 25038,N1(C(CNS(N)(=O)=O)=O)CC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 25039,CN1CC(F)CC1C(N1CCC(F)(CNC(=O)COc2ccsn2)C1)=O 25040,CC1CC(CNC(c2ccc(=N)[nH]c2)=O)CN1C(c1ccc[nH]1)=O 25041,C(CCN(C)C)(C(=O)NOC1CCOCC1)NC(c1c(C)cc(F)s1)=O 25042,C1(OC)(CNC(C23CCN(CC2)C3)=O)CCN(C(=O)CN2CC(C)(C)C2)C1 25043,C(C)(C(=O)NC(C1CN(C(c2conc2C2CCCC2)=O)C1)C)(C(C)C)OC 25044,C(=O)(C(C(C)(C)C)C1CCC1)NC(C(=O)NC(C(C)C)(C)CO)(C)C 25045,C(C(CC(=O)NC1(CCO)CCC1)NC(=O)CC1CCC(=O)N1)OC 25046,CC(=O)CCC(=O)NCc1ccoc1C(=O)NC1CCNC1=O 25047,c1(NC(=O)OC(C)(C)C)ccc(=NCCCNCCC(C)N2CCCC2)[nH]c1 25048,c1(C(=O)NC(CC=C)CNC(c2cn(CCC)nn2)=O)cc(OC)nn1C 25049,CCC1=C(C(=O)N2CCN(C(C3(CF)CC3(F)F)=O)CC2C)CCCO1 25050,CON(CCO)C(=O)CC(C(F)F)NC(=O)CC1CCOCC1 25051,C1(C(N(CC(CN(C(C(N2CCC(O)CC2)C)=O)C)O)C)=O)CCCCC1(F)F 25052,c1(C(=O)NCC#CCNC(c2c(CC)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25053,CCCCCCCC(=O)N1CC(C)C(NC(=O)C(O)Cc2cnc[nH]2)C(C)C1 25054,C(c1cc(C)c(C)cc1C)=CC(=O)NCC1CCCN(C(C2(C)CC(=C)C2)=O)C1 25055,C1(NC(CC2C(C)=NOC2=O)=O)CC2CCC1N(C(=O)COC1(C)CCCC1)C2 25056,C1(NCc2cnn(C)c2C2CCC2)CC(O)C12CC(F)(F)C2 25057,Cc1ncccc1CC(=O)NC(C(CN(C(=O)Cn1c(C)ccc1C)C)(C)C)=O 25058,c1(C(N2CCC(N(CCC)C(C3CCC3C(F)F)=O)C2)=O)c(F)ccc(F)c1Cl 25059,c1(C(=O)NCC2(F)CCC(NC(C(C(C)C)O)=O)C2)c[nH]nc1[N+](=O)[O-] 25060,N1(C(c2ccsc2Cl)=O)CCC2C(C1)CN2C(c1cnnc(O)c1)=O 25061,c1(CC)ccc(C(N2CCC(CNC(c3cn(C(C)(C)C)nn3)=O)C2)=O)c(O)c1 25062,CCC(CC)CCC(=O)N(c1cn(C2CCCN(C(=O)C(C)CC(N)=O)C2)nn1)C 25063,C(=O)(CN=S(C)(C)=O)NCC(NC(CCNC(COC)=O)=O)Sc1ccccc1 25064,c1(-c2n(CC)c(N3CCC(Cc4cncc(Cl)c4)CC3)nn2)c(C)cc(C)cc1C 25065,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25066,O=C1NC(C(N2CCC(CNC(=O)CCCc3cc[nH]n3)CC2)=O)C2CCC12 25067,c1(C(=O)NCC2N(C(C(n3ccc(C)n3)C)=O)CCC2)ccc(C)cc1[N+](=O)[O-] 25068,c1(C(=O)NCC(CCC)NC(=O)CCCCSC)cc(O)n(CC)n1 25069,C1(C(=O)OCC)(CNC(=O)NC(CCO)c2cncs2)CCCCO1 25070,N1(C(c2cnn(CC3CC3)c2)=O)CC2(CCN(C(c3c(=N)cc[nH]c3)=O)C2)C1 25071,C1(CN(C(=O)CC2(COC)CC2)C)CCCN1C(=O)CCCN1CCOCC1 25072,N1(S(C(C)(C)c2ccc(F)cc2)(=O)=O)CCC2(CCC2)CC1 25073,C#Cc1cccc(OCCC(N2CCC(C(=O)NCc3cccc(O)c3)C2)=O)c1 25074,C1(NC(C2N(C)CC(C)(C)C2)=O)CCC2(CC1)CC2NC(=O)CSS(C)(=O)=O 25075,C(=O)(C(CC(C)C)C(N)=O)N(CCCN(C(c1ccc(CC)cc1F)=O)C)C 25076,c1(C(=O)NC(C)CCCNC(C2(C(F)(F)F)CC2)=O)conc1CSC 25077,N1(C(c2ccc(C#C)cc2)C(=O)NCCSC)CCC(O)(C#N)CC1 25078,C1(NC(COc2cc(C)on2)=O)CC2(C1)CC2NC(=O)CN1CCCCC1 25079,CC1(C)CCCC(O)(C(=O)NC2COCCN(C(c3nscc3N)=O)C2)C1 25080,C(C)(CCC(=O)NCCc1nnc(O)o1)NC(CCCOC)=O 25081,N1(CC(=O)N(CCC(C(C)C)NC(=O)C=C2CCOCC2)C)CCCCS1(=O)=O 25082,CC1CCN(C(C2CC(C#N)C2)=O)C1c1ccccc1.c12cccc(c1)NC2 25083,C1(O)(C(C)NC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25084,C(N=c1nc2sccc2c(N2CCCC(OCCF)C2)[nH]1)c1c(Cl)cc(Br)cc1 25085,CCC(CC)C(C)C(=O)N1CC(OCC(=O)Nc2ccc(N)c(SC)c2)C1 25086,C1(C(=O)NCCOC2CCN(C(=O)C(F)C3CCCC3)C2)CC2(C1)CC21CC1 25087,Nc1cc(C(=O)NC2CC2CNC(=O)Cc2cc(C(F)(F)F)cc(F)c2)cc(N)c1 25088,N1(C(c2c(C)n(C)n(-c3ccccc3)c2=O)=O)CC2(CCCC2)CCC1CO 25089,C1(CCNC(c2nnnn2CCCF)(COC)C)CCC(C)CC1 25090,C#Cc1cnn(C)c1C(N1CC(CO)(NC(C2CC(O)C2(C)C)=O)C1)=O 25091,n1(CC(=O)NC2CCC(F)(CNC(C=CCCC)=O)C2)cnc2ccccc12 25092,C(C)(CN=c1nn[nH]n1C(C)C)NC(=O)NC.C1(C)C(=O)N1 25093,C12(NC(C(SC)SC)=O)CC(CN(C(=O)CC(C)n3ccnc3)C1)C2 25094,C1(C(=O)OC(C)(C)C)(NC(C(=O)CNC(=O)COC2CC2(F)F)=O)CCC1 25095,c1(NC(=O)OC)scnc1C(=O)NC1CC1CNC(C1OCCC1C)=O 25096,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25097,CCC(CNC(C1CC2(CC2)CO1)=O)(CC)NC(C1CC2CCC2C1)=O 25098,N1(C(CCCNC(=O)OC)=O)CC2(CCC(NC(=O)C(C)C(C)(F)F)CC2)C1 25099,Cc1nn(C)c(N)c1C(=O)NC(C(=O)NC(C)C(O)C(C)C)C(C)C.C(C)(C)(C)O 25100,C(=O)(CC(C)(C)C(C)(F)F)N(CC(C)NC(c1ccc(NC(N)=O)cc1)=O)CC 25101,c1(NC(CN2C(C)CCC2)=O)ccc(C(=O)NC2CC(C)(NC(N)=O)C2)nc1 25102,CCCC(CC(C)C)C(=O)N1C(C(=O)N(CCC(=O)OC)CC)C2CC(O)C1C2 25103,C1(CNC(C(C)SC)=O)CN(C(=O)CC#N)CC1O 25104,N1(C2CN(Cc3c(C)ncs3)C2)CC(NC(c2ccnc(S)c2)=O)CC1=O 25105,CCCCC(O)C(=O)NC1(CCC(=O)NCC(N2CCOCC2)C)CCCC1 25106,Cn1ncc(Br)c1C(N1CCC(NC(C2CCC(n3cccc3)CC2)=O)C1)=O 25107,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(CC(CC)C)CC 25108,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CCn2nnnc2C1 25109,C1(C(=O)NC2CC(CNC(C34CCC(CC3)CC4)=O)C2)CCCC2(CCCCC2)C1 25110,c1(C(=O)NC(C)CC2CN(C(=O)COC3CC3)C2)c[nH]c2cccc(Cl)c12 25111,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25112,C1(=CCC)CCN(C(=O)CN(CC(C)C)C(=O)CC2CCC(=O)C2C)CC1 25113,c1(C(C)(C)C)[nH]cnc1C(N1CC(CNC(c2cn(CC(F)F)cn2)=O)C1)=O 25114,CC(C)C(C)(CNC(C1CCOC1)=O)NC(=O)Cc1csc(-c2ccoc2)n1 25115,c1(C(=O)NCCOCC(=C)C)c[nH]cc1CC.C(=O)C(=O)N(C)C(C)C 25116,C1(NC(C2CC23CCC3)=O)CCC(O)CN(Cc2ccc(-c3ccsc3)cc2)C1 25117,N1(C(c2c(C)c[nH]c2)=O)CC2CCCC(C1)N2C(=O)Cc1cc(Cl)ccc1F 25118,C1(CNC(C2CCCN(C(C(C)C)=O)C2)=O)CCCN(CCC2CCC2)C1C 25119,c1(C(=O)NCCCNCCCCNC(=O)Cc2cnns2)cccc(C2CC2)c1 25120,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25121,C1(CCC(CNC(=O)CCC=CC(C)C)C(C)C)(C(=O)N)CCN(C)CC1.CCS 25122,c1(CCC)cc(C(=O)NC2CN(C(=O)CCC(=O)OCC)CC2C)ccn1 25123,C1(CC(=O)NCC2CC2CNC(C23CC4CC2C3C4O)=O)CCC(F)(F)CC1 25124,N1(C(CNC(=O)C(F)(F)F)=O)CCC(C(C)C(c2cccs2)c2ccoc2)CC1 25125,C1(C2CC2)(C(=O)NCC(CC)OC)CN(C(C2CCC(C)C2)=O)C1 25126,Cn1ncnc1CNC(c1ocnc1C(F)F)c1nnnn1C1CC1 25127,c1(CC)c(C(N2CC(N(C)C(c3ccnc(OC)c3)=O)C2)=O)cnn1C 25128,c1(C(N(C)CC2CCN(C(C34CC(COC)(C3)C4)=O)C2)=O)cn(C)[nH]c1=N 25129,C1(NC(CN2CCSCC2)=O)CC(N)C12CCC2.c1(CCC(=O)SC)nnc(S)n1C 25130,N1(CC)CC2CC1CN2C(C1(CC)CN(C(C2CN(C3COC3)C2)=O)C1)=O 25131,C1(NC(CC(C)c2ccco2)=O)COC2(C1)CN(C(=O)CC1CC(F)C1)C2 25132,C(C)(CO)(C(=O)NCc1ccc(CN(C)C(c2ccc(F)cn2)=O)cc1)OC 25133,Cn1ccc2cccc(CC(=O)NC3(C)CCN(C(=O)Cc4sc(O)nc4O)C3)c12 25134,C(CCN(C)C(c1c(C)noc1C)=O)(C(C)(C)C)NC(c1cncc(C)n1)=O 25135,C(=O)(CCCCCCNC(=O)CN(C)C)NCc1c(C)ncnc1 25136,CCCCC(C)CCC(=O)NC(CNC(=O)COC1(C)CCC1)CC 25137,N1(C(C2N(CCC)CCC2)=O)CC(C)(C)C(NC(c2cnc(Cl)[nH]2)=O)C(C)(C)C1 25138,N1(C(C23CCC(OC)C2C3)=O)CCC2(CC1)CCN(C(=O)COC(C)=O)C2 25139,c1(NC(C2C(NC(C(CC=C)C)=O)CCC2)=O)ccc(Cl)nc1NC(C)=O 25140,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25141,C1(C(=O)NCC(=O)NCC(=O)NCC)(CO)CCN1C(C1CC(C)=NO1)=O 25142,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)C 25143,C1(CC)C(C(=O)NC2CCN(C(=O)CCCn3nc(C)nc3C)C2C)CCN1C 25144,C12(C(=O)NS(=O)(=O)c3cc(OCCO)ncn3)CC3CC(CC(C3)C1)C2 25145,C(=O)(C(C)C(O)C(C)C)N(CC(COC)C)C.C(=O)C(C)(C)C1CCCC1 25146,N1(C(C)=O)CCC(c2nc(-c3ccccc3C)nn2Cc2cccs2)CC1 25147,c1(C(=O)NCC(C)CNC(C2(F)CCOC2)=O)nc(Br)c2c(F)cccn12 25148,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25149,S(=O)(=O)(c1cccc(Cl)c1F)NC1CC(C(=O)NCc2ccc(O)c([N+](=O)[O-])c2)C1 25150,c1(C(C(=O)O)NC2CC(C)(CC)C2)ccc(F)cc1F 25151,N1(S(CC)(=O)=O)CCC(NC(=NCC2CCCCO2)NC2CC23CCC3)CC1 25152,C(CC(=O)N(CC(C)CN(C)CCNC(C)C)C)N(C1C(C)C1)C.C(CCO)N 25153,C1(F)(CNC(=O)Cc2c[nH]nc2O)CCCN(C(C2(C3CC3)CCCO2)=O)C1 25154,c1(C(N2C3CN(C(CC4CC(=C)C4)=O)C(C3)C2)=O)cc2ccc(OC)cc2s1 25155,C(CCCCC(=O)NCCC1CCCCN1C(c1ccnn1C(F)F)=O)N(C)C 25156,CC1(C)CN(C(=O)CC2(O)CCCC2)C(NC(=O)CNS(=O)(=O)N(C)C)CO1 25157,C(=O)(C1=C(C#N)CCC1)N(C)CC1CCCN(C(c2c(C)nc(N(C)C)s2)=O)C1 25158,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25159,C1(NC(CCCN(C(C)C)C)=O)CC2CC(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 25160,O=C1CC2CN(C(=O)C(=O)NCc3cnn(CC4CC4)c3)CC2N1 25161,C=C=CCCC(=O)N1CC(CNC(c2cncc(NC)c2)=O)C(C(F)(F)F)C1 25162,c1(C(=O)NC2CC(N(C)C(c3c(C4CC4)cnn3C)=O)C2)ccn2c1CSCC2 25163,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25164,C1(CC)CCN(C(=O)CC2CCN2C(=O)CCCCNC(N)=O)C1C 25165,c1(C(=O)NC2CCCN(C(c3cnc[nH]3)=O)C2)cc(S(=O)(=O)N2CCCC2)c[nH]1 25166,C1(C(=O)NC2(CNC(C=C(C)C)=O)CC2)CCC(OC2CCOC2)CC1 25167,N1(C(c2c(CC)c[nH]c2)=O)CCC(C)C(NC(C2OCCN(C)C2=O)=O)C1C 25168,N(C(=NCCc1cn(C)nc1C)NCCc1cccnc1F)CC(COC)OC 25169,c1(C(N2CC(C)C(NC(=O)COCC(F)F)C2)=O)cccc2ccnn12 25170,C#Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)cc1 25171,C1(C(=O)NC(C(C)NC(C2N(C(C)=O)CC(O)C2)=O)CO)CC2(C1)CC(F)(F)C2 25172,C1(CCN)(NC(C(C(C)=CC)O)=O)CCCN(C(c2ccnc(CO)c2)=O)C1 25173,Cc1nc(NC2CCC2)sc1C(N1CC(O)(CC2(C)CCC(C(=O)NC)O2)C1)=O 25174,C=Cc1cnn(C)c1C(N1CCC(O)(C(C)NC(=O)C=C(C)C(F)F)C1)=O 25175,C1(NC(C(C)N(C(C)=O)C)=O)CC(C(=O)N(CC(c2nn[nH]n2)C)C)C1(C)C 25176,C1(C(N2CC(NC(CN(CCC)C)=O)(CO)C2)=O)CC(=O)N(CC(C)C)C1 25177,CCCCCC(O)CC(=O)N1CCOC(CCNC(=O)CC2CC=CCC2)C1 25178,c1(OC)cccc(OCCN2N3CCC(C3)C2=O)c1.C1(CC)CCOC1.CO 25179,C(=O)(C(Cn1cccn1)NC(C1(O)CCC1)=O)NCCOC(=N)O 25180,C1(Nc2nc(C)nc(C#N)c2)CC2CN(C(C3CC=CC3)=O)CCN2C1=O 25181,c1(NC(C2CC2Cc2ccccc2)=O)cnn(-c2nccs2)c1 25182,c1(CC)nc(C(N2CCC(CCNC(C3(C4CCCCO4)CC3)=O)C2)=O)co1 25183,N1(C(C2N(CCC)CCC2)=O)CCCC(C(=O)NCCN2CC(OC)C2)C1 25184,Cc1nn(CCOC2CCC2)cc1CC(c1nnnn1C(C)(C)C)N1CCCC1 25185,c1(N2CC(C(=O)Nc3cc(C(=O)OC)ncc3)SCC2)ncnc2cnccc12 25186,c1(C(N2CCC(NC(CN(C)C3CC3)=O)C23CCC3)=O)ccc2ncn(C)c2n1 25187,N1(C(C(c2cccnc2)NC(c2cnn(C)n2)=O)=O)CCC(O)(CO)CC1 25188,c1(N2C(CC)CN(C(C)C)CC2)nc(S(C)(=O)=O)ncc1Br 25189,N1(C(CC(C)C2CC2)=O)CC(C(=O)NCC2(n3ccnn3)CC2)CC12CCC2 25190,c1(C(=O)NC(CC)CNC(C2CC(F)C2)=O)nc(C)n(C(C)C)c1C 25191,C1(CNC(CCCC(=C)C)=O)CCC2CN(C(c3n[nH]c(C)c3O)=O)CCC2C1 25192,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)N(C)CC1(N(C)C)CCC1 25193,S(=O)(=O)(c1ccc(NCC(c2cccs2)O)nc1)NC(c1ccc(Cl)cc1)CC 25194,c1(C(=O)NCC2C(NC(=O)Cc3cc(F)ccc3F)C2)cc2ccc(F)cc2o1 25195,C(=O)(C1OCCc2c(C)cccc21)NC(CCN(C(c1c(CC)scc1)=O)C)C 25196,c1(N(C)C)c(C(=O)N(C2CCCCNC2=O)Cc2ccccc2)c(=O)c1=O 25197,C1(C(=O)NC2CN(C(CSC(C)=O)=O)C2)COCCN1CC(F)(F)F 25198,C(=O)(C1CC(O)c2ccccc21)N1C(CN(C(CC(CC)(C)C)=O)C)CCC1 25199,C1(C(=O)NCC23CC(CNC(C4C(CC)OCC4)=O)(OC2)C3)CCCNS1(=O)=O 25200,Cc1ccc2c(c1)C(C(=O)NC(C)CNC(c1ccc(CO)cc1F)=O)C2 25201,CC1(C(N2CCC(C)(CNC(c3cc(F)cnc3O)=O)C2)=O)CCCCC1(F)F 25202,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)nc3O)=O)c12 25203,C1(NC(C2CC(O)(CC#C)C2)=O)CCC2(CCN(C(=O)CC(C)CC)C2)C1 25204,c12ccc(cc1)[nH]c2=O.C(CCC(N)=O)NC(C(=O)N(C)C)=O 25205,Cc1cc(C(N2CCCC(CN(C)C(c3cnccc3N(C)C)=O)C2)=O)sc1C 25206,c1(-c2ccc(C(N3C(CCCNC(C=C(C)C)=O)CCC3)=O)s2)cccc(F)c1 25207,Cc1cccc(OCCC(=O)NCC(C)(C)CNC(=O)C2=CCCS2)c1C 25208,C1(O)(CNC(CCC)=O)CCCN(C(C2COCCN2CC(F)F)=O)CC1 25209,C1(NC(C(CC=C)NC(N)=O)=O)CC(NC(C2(CO)CCCC2)=O)C12CCC2 25210,C1(C(C(N2CC(=CCC)C2)=O)C)CCN(C(c2ncn(CC3CC3)n2)=O)CC1 25211,c1(C(N(CCc2cn(CCS(C)(=O)=O)nn2)C2CC2)=O)cc2n(n1)CCCCO2 25212,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25213,C1(C2=CCN(C(c3c(C)nc4sc(C)cn34)=O)CC2)(OC)CCC1 25214,O(NC(=O)C(CC(N)=O)NC(c1ccc(C)s1)=O)CC=C(C)C 25215,C1(C)(CC)NC(=O)N(CC(N2CC(F)CC2CNC(=O)C(C)(C)C2CC2)=O)C1=O 25216,c1(C(N(CCNC(C(CC)F)=O)CC)=O)cccc(N(C)C)c1 25217,c1(C(=O)NC2CCN(c3ccc(C(=O)OC)cc3)CC2)cc(C)c(F)cc1Cl 25218,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25219,CC1(C(N2CCN(C3CN(C(c4cnc(O)o4)=O)C3)CC2)=O)CC(F)(F)C1 25220,c1(C(=O)N)ccn(CCC2(O)COC2)n1.c1(CC2(O)CCSC2)c[nH]nn1 25221,N1(C(=O)N(c2cc(CC(C)C)on2)C2CCCC2)CCC(C)C1c1ccc(Br)cc1 25222,C12(CCCCO1)C(=O)N(CCOC)CCOC2.C(CC(=O)NC(C)C)NC(C)=O 25223,C12C3CN(CC13)C(=O)c1cn(cn1)C2.c1(SC(C)C(=O)N2CCCC2)ccccc1 25224,C(CCC(C(=O)NCCC1CCOC1(C)C)NC(=O)C(C)=CC1CC1)OC 25225,C#CC1CN(C(C2(CC#CC)CC2)=O)CCN1C(=O)CC1CCC(C)(C)CO1 25226,N1(C(C2CN(C(N)=O)C2)=O)CCC(CNC(C2C(F)(F)C23CC3)=O)CC1 25227,N1(C(CCSCC)=O)CCOC2(CCN(C(=O)CN3C(=O)CNC3=O)C2)C1 25228,c1(C2CCN(C(C=C)=O)C2)nc(N2C3CCC2COC3)ncc1F 25229,C(C(CC(=O)OC)NC1CC(=O)N(c2ccc(O)cc2)C1)OC 25230,C1(CNC(c2c(C)nns2)=O)CC(F)CN1C(c1sccc1C(F)F)=O 25231,C1(O)(CNC(C2CC2c2ccncc2)=O)CCCN(C(C2(F)CCC2)=O)C1 25232,N1(C(C2C(=C)C2)=O)CCC(C2CCCN(C(=O)C(C)(C)CO)C2)CC1 25233,c1(C(=O)NC(COCC)C(=O)NC(Cn2cncn2)CC)cnn2ccccc12 25234,C(=O)(CC1=CCOCC1)NCC(CC(N1CCN(C)CC1C)=O)OC 25235,c1(C(=O)NCCCCN(C)C(C2CCN2C)=O)ccc(CO)cc1F 25236,CC1(C(=O)NCC(C2CCN(C(=O)CCC3CCC3)CC2)F)CCNC1=O 25237,c1(C(=O)NC(C(C)NC(CCCCCC)=O)C)sc2cc(C(C)C)ccc2c1Cl 25238,Cc1cc(C(=O)NCC2OCCC2C(=O)NCC(O)CNC(N)=O)sn1 25239,C(=O)(CCCCC(C)(C)C)NC(C(C)C)CCNC(=O)C=Cc1ccc(F)cc1 25240,N1(C(c2ccc(C)nc2C2CC2)=O)CC(C)N(C(=O)CN(C)C2CC2)CC1C 25241,CC(C(=O)NCC1CN(C(=O)CCn2cccnc2=O)CC1O)C(F)(F)F 25242,C1(C(N2C(c3cn(CC4CCC(=O)O4)nn3)CCC2)=O)CC2CCCC2C1 25243,CC(CC(C)NC(=O)CCCNC(=O)OCCCC1CCC1)NC(N)=O 25244,C1(C(C)C)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)CCO 25245,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)N1)=O 25246,CCCCS(=O)(=O)CC(=O)N1CCC(C)C(N(C)C(c2cc(COC)on2)=O)C1 25247,C(=O)(CC(C(F)(F)F)NC(C1CC(N(C)C)C1)=O)NC(c1onc(C)n1)C 25248,C=CCC(CC1CC1)N=c1nc2sccc2c(N2CCC(N(CCCNC)C)C2)[nH]1 25249,C1(CNC(CSC)=O)CN(C(C2(n3cccn3)CC2)=O)CC1C 25250,S(=O)(=O)(c1cn(C)cn1)NCC(=O)NC1(CCNC(C(C)OCC)=O)CC1 25251,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25252,c1(C(=O)NC(C2CCCC2)CC)cn(CCNC(c2cc[nH]n2)=O)cn1 25253,N1(C(CCNC(=O)CO)=O)CCC(C2CCN(C(c3ncc(Cl)cc3F)=O)C2)C1 25254,N1(C(c2n(CCC)ccc2)=O)CC(CNC(C2(C)CCCCC2)=O)CC12CCC2 25255,N1(C(=O)NC2CCC(C)CC2)CCN(CC(C)NC(CC=CCC)=O)CC1 25256,n1(CC(N2CC(N(C(=O)CCC(C)(C)C)C)C2)=O)c(O)nc2ccccc12 25257,c1(C(=O)NCCC2OCCCN(C(CC(CC)(F)F)=O)C2)cc(S(N)(=O)=O)c[nH]1 25258,c1(CN(C(=O)NC(c2cccc(F)n2)C)C)cccc(Cl)c1Cl 25259,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25260,c1(C(N2CC3CC(NC(c4n(C)ccc4)=O)C3C2)=O)cccc2[nH]cc(C#N)c12 25261,Cc1cnc(C(N2CCC(C)C(Nc3cc(C)nc(C)n3)C2)=O)c(F)c1 25262,C(=O)(C(C(C)O)N(C)C)NCC(CC)NC(C1(CC2CC2)CCC1)=O 25263,C1(C(N2C(C(=O)N(C)C)CC3CC23)C(=O)NC)CCC(=O)N(C(C)C)C1 25264,C1(C(N(CCN(C(=O)CCCCc2ccccc2)C)C)=O)CCC(C)(F)CC1 25265,Cc1nsc(C(N2CCCCC2CCC(=O)NCC=C(Cl)Cl)=O)c1N 25266,N1(C(CCC=C(C)C)=O)CCCC(CCNC(=O)CCC2CCCN2C)C1 25267,Cc1nc(NCCCN2CCC(O)C2)cc(=NCc2c(F)cccc2Br)[nH]1 25268,CCC(C(C)(C)C)NC(=O)C(c1cccnc1)NC(c1cccs1)=O 25269,C(CO)(C(C)(C)CO)NC(C1(CCC=C)CN(C(C2CCC(=O)CC2)=O)C1)=O 25270,CON(C)C1CCN(C(C2C3CCN(C(C45COCC4C5)=O)CC23)=O)CC1 25271,C1(CC(=O)NC(C(C)(C)C)CNC(=O)C=Cc2cnccn2)CCCC2(CC2)C1 25272,N1(C(C2C(C)(C)N(C(=O)COc3cccnc3)CC2)=O)CCc2nc(O)[nH]c2C1 25273,C1(O)(C2CN(C(C3CN(CC)C3)=O)C2)CCN(C(=O)OC(C)(C)C)CC1 25274,c1(C(=O)NC2C(C)(CNC(C3CCCOC3)=O)CCC2)nnc(O)cc1O 25275,C1(CNC(C(=O)Nc2ccc(CSC)cc2)=O)Cc2ccccc2O1 25276,c1(SC(CNC(=O)C(=O)N(C)C)=O)ccc2c(c1)OCCO2.C1C(=O)NC1C 25277,N1(C(c2c(OC)nsc2OC)=O)CCCC(CNC(c2csnc2Cl)=O)CC1 25278,C(=O)(CCCC(C)(c1nnnn1C1CCCC1)NCc1ncc(Cl)n1C)OC 25279,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25280,C(COC1CC1)(CC)OC(C1(F)CC1CC(=O)OCC)=O 25281,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1C(F)(F)C2 25282,N1(C(CC(=C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25283,C1(C(N(CCCNC(c2c(C)oc(Cl)n2)=O)C2CC2)=O)CCOC(=O)CC1 25284,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25285,C(=O)(CC1COc2ccccc21)NC(N(Cc1cn(CC)nn1)O)=O.c1ccccc1C 25286,C(C(C)CC(=O)N1CCCCC1C(C)(C)C(=O)Nc1cc(OC)ns1)OC 25287,N1(C(C2(CNC(CCc3ccc(C)o3)=O)CCCC2)=O)CCCC(C)CC1 25288,c1(SC)cncc(C(=O)NC2CC(NC(C3CC3(F)F)=O)CC2O)c1 25289,C1(OC)CCC2(C(N3CCCC(C(=O)NC4(c5cccnc5)CC4)C3)=O)CC12 25290,c1(C(C)(C)O)cc(C(=O)NCC(O)CCNC(=O)C(c2cccnc2)O)ccn1 25291,CC1c2cc(O)ccc2CCN1C(c1nc(-c2ccc(OC(F)F)cc2)cs1)=O 25292,c1(C(=O)NCCN(CC(C)O)C(C2(C)CC2(F)F)=O)cc(-c2ccccn2)ns1 25293,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25294,C1(CNC(C2(OC)CCCC2)=O)CN(C(C2(CO)CCOCC2)=O)CC(C)(C)O1 25295,C1(C(C(C)C)NC(C=CC)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 25296,C(=O)(NNC(=O)C1CCCN1C(=O)OC(C)(C)C)N(CCC)C(C)C1CC1 25297,Cc1cc(C(=O)NC(CNc2nccc(-c3cnccn3)n2)C2CC2)ncn1 25298,N1(C(=O)C=CCF)CCC2CN(C(C3CC3C3CCCCO3)=O)C2C1 25299,N1(C(c2c(CC)n[nH]c2)=O)CCC(F)(C(=O)NC2(COC)CC2)CC1 25300,CS(=O)(=O)C(CNC(=O)CC1CC2CCC2C1)CNC(c1cn(CCF)nn1)=O 25301,C12(CC(=O)NC3COCC3Nc3ccc(-n4cccn4)cc3)COCC(C1)C2 25302,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(c2cc(Cl)cn2C)=O)CC1C 25303,N#Cc1c(NCc2cccc3c2CCC3)sc2cccc(F)c12 25304,c1(OC)ccc(-c2cc(C(=O)N(CCNC(c3csnc3C)=O)C(C)C)[nH]n2)cc1 25305,C(=O)(C1SCCc2sccc21)OC(C)CNCC(C1CCCC1)OC 25306,C12(NC(c3cc(-c4cn(C)nn4)on3)=O)CCN(C(c3ccn(C)c3)=O)CC1C2 25307,Cn1ccc(C=CC(=O)NCC2(NC(=O)CC3(C4CC4)CC3)CC2)c1 25308,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25309,Cc1cc(-c2cnc(NS(=O)(=O)c3cccc(C4CC4)c3)s2)cc(C)c1C#N 25310,c1(C(=O)NC2CCN(C(c3c(C)ccc(OC)n3)=O)C2C)cn(C)c2ncccc12 25311,CCCCCC(O)C(=O)NCCNC(=O)Cc1ccc(=O)n(C)c1 25312,N1(C(c2cc(C)no2)=O)CC(C)CN(C(c2ccn(C)c2C)=O)C(C)C1 25313,C1(CC(=O)NC(C(=O)OC(C)(C)C)c2cscn2)(OC)CN(C(C)=O)C1 25314,c1(CC)c(C(=O)NC2C=CCN(C(C3CC3c3ccccc3)=O)C2)ccn1C 25315,c1(C(=O)NC2C(CNC(CCc3cc(C)no3)=O)C2)nc(C(C)C)oc1C 25316,Cn1c(NCC2CCCCN(C(c3scnc3C(F)F)=O)C2)cc(=O)n(C)c1=O 25317,c1(C(=O)NC(CN(C(=O)CCC2CCCN2C)CC)C)cc(CCO)on1 25318,N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 25319,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25320,c1(C(N2CCN(C)CC2)=O)ccc(SC(N2CC(CC)C2)=O)cc1 25321,N1(C(c2n(C)nc(Br)c2)=O)CCC(NC(=O)CCc2cnco2)C12CC2 25322,C1(C(C)O)CC(C(=O)N(C(C)CCNC(=O)C(C)C)C)C1 25323,N12CC(C(C(=O)O)C1)OCC2=O.c1(-c2cn(CCOC)nn2)ccc(C)cc1 25324,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ncc1C 25325,N1(C(CC=C)=O)CCC2CCCC12C(=O)NCc1ccnn1C 25326,S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(NC(C3C4CCCC34)=O)C2)cc1)NCC 25327,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25328,c1(C(N(C)CC2N(C(=O)CN(CCCSC)C)CC2(C)C)=O)cnc2ccoc2c1 25329,C1(C(N(C)CCc2cnn(C)c2)=O)CC12CCN(C(=O)C(F)C(C)(C)O)C2 25330,C=CC1(C(=O)NC2CCC(NC(=O)C(C#N)=CC(C)C)CC2)CCCCC1 25331,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)C(c2occc2C(=O)OC(C)(C)C)=O)CC1 25332,CN1CCN(C(=O)CC2CCCC(C)(C)C2)CC1CNC(c1ccnnc1O)=O 25333,C1(CNC(C(C)(C)CO)=O)C(O)C(O)CN1C(C1(C)CCCNC1=O)=O 25334,c1(C(N2CC(C)(NC(C3(C)N(C(C)=O)CCC3)=O)C2)=O)cnc2ncccc2c1 25335,N1(C(C=C(CCC)C)=O)CCC(CNC(C2CCCCN2CC)=O)C12CCC2 25336,C(=O)(CC(O)CCCC)NC1(CC(N2CC(CC#C)OCCC2)=O)CCCCC1 25337,N1(C(C)C)C(=O)CCC1C(=O)NCCCNC(=O)CC1CC2(COC2)C1 25338,C1(C)(C(N2CCC(C(=O)NC)CC2)=O)Cc2ccc(Br)cc2C(=O)C1 25339,Cc1ncnc(C)c1NC(C1CCCC1CNC(c1cc(F)n(C)n1)=O)=O 25340,N1(C(C(C)OC2CCCC2)=O)CCN(C(=O)CCOCCNC(C)=O)CC1 25341,C1(C(=O)NC(CO)C(C)NC(=O)Cc2csc(NC(C)=O)n2)(CC)CNC(=O)C1 25342,Cc1cc(CCC(=O)N(CCNC(=O)CC2(C)CC2(F)F)C(C)C)on1 25343,C1(NC(C=C(C)c2cccs2)=O)CC2CCC1CN(C(c1coc(CO)c1)=O)C2 25344,c1(NC(=O)NCCN(C)Cc2ccc(C)c(C)c2)cc2ccncc2s1 25345,N1(C(c2c(C)cn(C)c2)=O)CCC(F)C(NC(=O)CC(C)(C)c2ccccc2)C1 25346,c1(CC)cc(C(=O)NCCN(C(=O)CNC(C2CCSC2)=O)C2CC2)sc1C 25347,Cc1nn(C)c(C)c1CN1CC(C(N(NC)C(C)C)=O)C1.C1(NCC)CCCOC1C 25348,c1(OCC)cc(NC(c2cc(Br)nc(CNCCO)n2)=O)ccc1OCC 25349,N1(C(Cn2ccc(C)cc2=O)=O)C2CCCC1CNC2.C12CCCN1C2 25350,C1(C(N(C2CC(C)OCC2)C)=O)CN(C(C2CCC(C)(C)CC2)=O)CC1(F)F 25351,N1(C(C(c2ccc(C)cc2)=O)=O)CC2(C1)CN(C(=O)CS(C)=O)CCO2 25352,C1(C(N2C3C(NC(COCCC)=O)C(C3)C2)=O)CCCC2CCCN12 25353,c1(CN2CC(CCNC(C(CC#C)O)=O)C2)ccc(OC)c(C)c1 25354,c1(C(=O)NC2CC23CCN(Cc2cncc(Br)c2)CC3)ccc(I)c([N+](=O)[O-])c1 25355,N1(CCN(C(=O)C(C)CC(F)F)C(CCCCC)=O)CCN(CC)C(=O)C1 25356,c1(NC(CS(=O)(=O)NC)=O)cc(N)cnc1Cl.C12CN(CC1C)C2 25357,C1(C(N2CC(C)(NC(=O)C(O)C3CCCC3)C2)=O)(NC(C)=O)CCC(C)(C)C1 25358,c1(N2CC(N(C(c3ccn(COC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25359,c1(C(=O)NC2C(NC(C3C(C)(C)C3(C)C)=O)C2)cc2n(n1)CCCCO2 25360,Cc1ncc(Cl)cc1NC(C1CN(Cc2ccc(C3CCCCC3)o2)C1)=O 25361,c1(-n2cc(CONC(c3ccc(C(=O)OC)cc3)=O)nn2)ccc(Cl)c(C)c1 25362,C(=O)(CC(CC1CC1)NC(c1cc(NC)n(C)n1)=O)NCCOCCCC 25363,C1(C#N)(C(N(CCCCNC(c2c(C)n[nH]c2)=O)C)=O)C(C#N)C1(C)C 25364,C1(c2onc(-c3ccc(C4CCCC(N(C)C)C4)cc3)n2)CCCC12CCC2 25365,N12CCCC(C3CN(C3)C(=O)c3c(cnn3C)C1=O)C2.C12(CC(=O)OC)CCC1C2 25366,C=CCC(CNC(=O)C(C#N)CCC)C(=O)N1CCC(OC(C)=O)C1 25367,c1(NC(c2cccs2)C#C)cc(OCC2CC2)ncn1 25368,c1(NC(C(C(C)(C)C)SC)=O)ccc2nc(NC(c3ccccn3)=O)sc2c1 25369,C1(CNC(C2CCS(=O)(=O)C2)=O)CC(F)CN1C(=O)CN1CCCS1(=O)=O 25370,CN1CCC(=CC(=O)N(C2C3CN(C(=O)C(C)(C)n4ccnn4)CC23)C)CC1 25371,Cc1nc(C(F)(F)F)ccc1C(N1CCCC1c1ccccc1)=O 25372,CC1(CNC(c2cc(Cl)ccc2F)=O)CN(C(C2(O)CCCCCC2)=O)CCO1 25373,C=CCCC(C(=O)N1CCOC(C)(C)C1)NC(=O)CC=C(Cl)Cl 25374,c1(C(N2CC(CNC(c3cc(OC)ncn3)=O)C2)=O)ccc(F)c(F)c1F 25375,c1(CC(N2CC(F)CC(NC(C3CC4CCC3O4)=O)C2)=O)ccc2c(c1)COCC2 25376,N1(C(C(CNC(CC(CCC)C)=O)CC(C)C)=O)CCC2(CCC2)C(O)C1 25377,C(C)(CCC(=O)N(CCC(=O)N(C)CC1(C)CCCO1)C1CC1)OCC 25378,CC(C)(C)CCCC(=O)NC1CC2CCC1CN2C(=O)COc1cccnc1 25379,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25380,c1(C(c2nnnn2CC2CC2)Nc2ccc(C(CC)C)cc2)c(C)nn(Cl)c1C 25381,c1(C(N2C3CCC(NC(C=CC=CC)=O)C(C3)C2)=O)cc(C)cc([N+](=O)[O-])c1 25382,C(=O)(C1Cc2c(Cl)cccc21)NC1C(F)CCN(C(C2(C)CC2)=O)C1 25383,c1(C(=O)NCCCN(C(=O)CCn2ccnc2)CC)nc(Cl)ccc1F 25384,C(=O)(C1CCc2ccccc21)N1CCC(CC(=O)Nc2cc(C)nc(O)c2)C1 25385,c1(C(=O)NC2CN(C(CCC=C)=O)C(C)(COC)C2)cccc([N+](=O)[O-])c1 25386,C(=O)(C(C)(C(C)C)SC)NC(CC=C)CNC(C1(S(C)(=O)=O)CC1)=O 25387,c1(C(N(CC(C)CNC(c2cnsn2)=O)C)=O)cc2c(nc1O)CCCC2=O 25388,C1(COc2cnn(C)c2)CCN(C(C2N(C(CCn3ncc(C)c3)=O)CC2)=O)CC1 25389,c1(OC)cc(CSc2ccccc2)ccc1Cl.c12nc(cc(C)n1)S2 25390,C1(NC(=O)C=CI)CCCN(C(C2(O)CCSCC2)=O)CC1F 25391,C=CCC(CNC(=O)CC1OCCC1(C)C)C(=O)NCC1(CO)CC2CCCC2C1 25392,C1(N(C(=O)CCc2ccsc2)CC#C)CCCN(C(=O)CCCCCCC)C1 25393,c1(COC)nc(NCc2c[nH]nc2C)cc(=NC2CCCC(C)C2)[nH]1 25394,c1(C(C)C(=O)NC(C)CCNC(=O)COC2CCOC2)ccccc1 25395,C1(NC(c2cccc(CNC(CCSCC)=O)n2)=O)CC(CO)C2CC12 25396,c1(OC)nc(C(=O)NCC2CCC(NC(C3CCC4CC4C3)=O)CC2)cc(O)n1 25397,N1(CCN(C(C(C)OC)=O)C)CCc2sccc2C1.C1C(=O)NC2CC2C(=O)N1 25398,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25399,N1(C(C(C)(CO)OC)=O)CC2(CNC(=O)Cc3nc(C4CC4)cs3)CC1CO2 25400,N1(C(c2c(C)nc(Cc3ccncc3)s2)=O)CC(S)CC12CCOCC2 25401,C=CCCCCCC(=O)N1CCC2(C(=O)NCCn3nc(C)cc3CC)CC2C1 25402,CC1CCN(CC(C)(C)C(=O)O)CC1.c12ccc(cc1)NC(=O)C(=O)N2.C1C(=O)O1 25403,c1(C(N2C(C(N3CC(CC)OCC3)=O)CC2)=O)ccc(I)cc1Br 25404,C1(CN(C(=O)C(C)C(=O)OC(C)(C)C)c2cn(CC(C)C)nn2)CCCC(=O)CC1 25405,CC1(C)COc2c(C(=O)NCC3CCN(C(c4csc(C#N)c4)=O)C3)cccc21 25406,N1(C(c2ccc(C#C)cc2Cl)=O)CC2CCCCC2(NC(=O)CN2CCOC2=O)C1 25407,c1(C(C(=O)NC(CN(C(c2cccc(C(C)C)n2)=O)C)C)O)ccc(Cl)c(Cl)c1 25408,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25409,Cc1nc2cc(n1)CNC(=O)NC2.C1(C(=O)OC(C)(C)C)CCCC1C(F)F 25410,N1(C(c2c(CCC)cccc2)=O)CC2CCC2(CCNC(=O)C2=CCCCC2)C1 25411,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25412,C1(N(C(C=CC=CC)=O)C)CCN(C(=O)CNC(=O)NC)CC1C 25413,C12(CNC(C(c3c(C)noc3C)C)=O)CCC1CN(C(c1nnsc1N)=O)C2 25414,Cc1cc(C(=O)NCC(C)N(C)C(c2ccc(CC(F)(F)F)cc2)=O)ccc1O 25415,CCCC(O)CC(=O)NC1CN(C(=O)Cc2ccnn2C)CC1O 25416,c1(C(=O)OCC(c2n(C)nnc2)=O)cc2cc(Br)cn2cn1 25417,n1(CC)cc(C(=O)NC2CCCCC2NC(=O)CCS(N)(=O)=O)c(=O)cc1C 25418,c1(C(=O)NC23CC(CNC(C4(C)CCN(C)CC4)=O)(C2)C3)cnc2ncccn12 25419,C12(N(C(C)C(=O)OC)C(=O)C=Cc3cocn3)CCN(CC1)CC2 25420,c1(NCC(CCCC)NC(=O)Cn2ccnn2)ccc([N+](=O)[O-])cn1 25421,c1(SC)cc(C(N2CCCC(CNC(C3CC3F)=O)C2)=O)c(C)o1 25422,C1(OC)(Cn2cc(NC(=O)C(N3CCCCC3C(C)(C)O)=O)nn2)CCCSC1 25423,C1(NC(c2n[nH]cc2Br)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 25424,C1(C#N)(C(=O)NC2(O)CCOCC2)CC2CCC1C2.CCC1CN1 25425,CS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)Cc2ccns2)C1 25426,C(CCCCC(=O)NCC(C)(CO)NC(=O)CN1CCS(=O)(=O)CC1)OC 25427,c1(C(=O)NC2C3CN(C(c4cc(C#N)[nH]c4)=O)C2C3)ccc(C(F)F)cc1Cl 25428,C=CC1(C(=O)NCC2CC(OC)CCO2)CCN(C(=O)Cn2cc(C3CC3)cn2)C1 25429,c1(C(N2CC(C)CC(NC(COC(C)C)=O)C2)=O)cc2ccc(Br)cc2o1 25430,c1(C(=O)Nc2ccc(-c3ccc(C)cc3)cc2)cnc(N2CCCC2)cc1C 25431,c1(OCCN(CCOCCNC(C2C(C)(C(C)C)C2)=O)C)ccc(Cl)c(Cl)c1 25432,c1(C(N2CCCC(C(N3C(C(C)O)COCC3)=O)C2)=O)cnnc(Cl)c1Cl 25433,c1(CN(C(CC2CC(OCC)C2)=O)C)ccccc1CNC(c1ccc[nH]1)=O 25434,CCC(C(=O)NC1CN(C(c2ccc(C(C)O)cc2)=O)CC1C)C(C)C 25435,c1(CC(N2CC(C(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25436,c1(C(=O)NCCC(N)C(=O)NC2CCC(OC(F)(F)F)C2)cc(C(F)(F)F)c(O)nn1 25437,c1(C(=O)OC)c(C(=O)COC(=O)CC2CCC(=O)N2)c[nH]c1C 25438,C(C)(C)(C(O)C(F)F)NCC(=O)NC1(CNC(Cc2nccc(SC)n2)=O)CC1 25439,N1(C(c2c(C)scn2)=O)CC(C)CN(C(=O)Cc2ncncc2Cl)C(C)C1 25440,N#Cc1cc(C2(NC(N3CCCC3c3ccccn3)=O)CC2)ccc1F 25441,N1(C(CC(=O)NCC)=O)CCC(NC(=O)CCSc2ccccc2)C1C 25442,c1(C(N2C(C(=O)Nc3ccc(CC(=O)OC)nc3)CC2)=O)cccc2occc12 25443,Cc1cc(C(=O)NC(C2CCCN(c3nnc(CO)s3)C2)C)nn1C(F)F 25444,C1(NC(CC(C)c2ccccn2)=O)CCC(CNC(=O)CCCC2(C)N=N2)CC1 25445,N1(C(CCC=C)=O)CCC2(CC1)COC(CNC(C1(COC)CCOC1)=O)C2 25446,c1(C(N2CCCC(C(C)NC(=O)C(C)(CO)CO)C2)=O)cc2ncccc2[nH]1 25447,C1(CC(=O)NCc2c(C(N(C3(C)CCCC3)C3CC3)=O)cco2)CC(O)C1(C)C 25448,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25449,N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(=O)C(C)(C)CCC)CO2 25450,C1(NC(C2CC3CCC2C3)=O)CCCN(Cc2nnc(C3CC3)o2)CC1 25451,Cc1nc(N)c(CC(N2CCC(N(C(=O)CC(C)(O)CN(C)C)C)C2)=O)c(O)n1 25452,Cc1nc2cc(CC(=O)NCC(O)CN(C)C(c3c[nH]cc3C)=O)ccc2o1 25453,c1(C(=O)NC2C=CC(CC(=O)N(C(C)C)CCN(C)C)C2)cccc(C#N)c1F 25454,C(C)(CNC(C1(C2(C)OCCO2)CC1)=O)(CC)NC(C1C(=C)CC1)=O 25455,N1(C(C)C)CCCN(C(c2ccc(-c3cccc(C(F)F)c3F)nc2)=O)CC1 25456,Cc1cc(F)cc2[nH]c(C(=O)NCCNC(c3cnn4c3NCCC4)=O)cc12 25457,c1(OC)cccc2ccccc12.N12CC(C1)NC2=O.C1(C2CC2)CNC(=O)N1 25458,n1(CC)cnc2c(N(CC(C)(C)C)C)[nH]c(=NC3CCOC(C(C)(C)C)C3)nc12 25459,CC1(C#CC(=O)NC(C2CCCC2)CNC(C23CCCC(CO2)C3)=O)CC1 25460,N12CCN(CC1)C2=O.C(C)(CNC(=O)CCC(N)=O)(C(C)C)NC(C(CC)C)=O 25461,C1(NC(C2C(C3C(C)C3)C2)=O)CCN(C(=O)Cc2ccccc2Br)C1(C)C 25462,n1(C(CC)CC)cc(CCCCC#N)nn1.n12cc(nn1)C2 25463,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25464,c1(C(=O)NC2CC(N(C)C(C3CC34CCCC4)=O)C2)c[nH]c2ccc(Cl)cc12 25465,c1(C(C(=O)CC2CC2)=O)ccc(-n2nc(-c3cc[nH]n3)nc2CF)cc1 25466,C1(CC)CC(C(=O)N(CCCCN(C(=O)Cn2cccnc2=O)C)C)CCO1 25467,N1(C(C)=O)CC2CC1CN2C(C1C(CNC(C2C3CCC(=O)C23)=O)C1(C)C)=O 25468,C(=O)(CC(C)C(C)(C)NC(=O)C(CCC)C1CCC1)N(CC(CCC=C)O)C 25469,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CN(C)C(c1cnccn1)=O 25470,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25471,c1(CC=C)ccccc1NC.C1(N2CC(=O)OCC2)CC(C)OC1C 25472,N1(Cc2cn(CCCCCN)nn2)CCOc2ncccc21 25473,C1(CNC(C(c2ccccc2)SC)=O)CC(C)N(C(=O)CCn2ccnn2)C1 25474,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25475,c1(C(=O)OC)cc(C)cnc1NC(CNC(=O)C(=Cc1cccnc1)F)C(C)C 25476,c1(C(N(C)CC2CCC2O)=O)cnc(N(C)C)nc1 25477,C(CN=C(NCc1nnn(C)n1)NC(c1c(Br)nnn1C)C)OCCOC 25478,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25479,CN1CC(C)(C)CC1C(=O)NCC1CCC(C(=O)NCCC(F)(F)Cl)O1 25480,Cc1cc(O)c(C(=O)N(CCCNC(C2CC2CF)=O)CCO)cc1Br 25481,C(CC(C)C)(C(=O)N1CCC(CO)(CNC(=O)C(F)F)C1)OC 25482,C=CCN=C(NCC(c1ccc(F)cc1)O)NC1CCN(S(C)(=O)=O)CC1 25483,N1(C(=O)CSC(F)F)CC2CN(C(=O)C3=CCOCC3)CC2C(F)(F)C1 25484,N1(C(=O)CCOCC2CCCO2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25485,Cc1ncnc(C(N2CCC(C(C)NC(c3n[nH]cc3C3CC3)=O)C2)=O)c1C 25486,N1(C(=O)CSCC(F)F)CCC(C(=O)NCC2CCCS2)C12CCC2 25487,N1(C(C(C=CC)O)=O)CCC(C2N(C(c3ccnc(OC)c3)=O)CC2(C)C)CC1 25488,C(C(F)(F)F)(c1ccccc1)CC(=O)N(CCCn1ccnn1)CC 25489,N1(C(C(C)(C)C2CCOC2)=O)CC2C(CNC(=O)C(N)=O)C2C1 25490,Cc1ncc(CCNC(=O)C(CC2CCCC2)NC(=O)C(N2CCCCC2)C)s1 25491,c1(C(=O)NCCN(C(C=C(CCN(C)C)Cl)=O)CC2CC2)cnc(C2CC2)nc1 25492,C1(F)(CNC(c2ncccc2N2CCCC2)=O)CCN(C(C2CC2C2CCC2)=O)C1 25493,C(=O)(CCCCC#N)N(C(c1ccc(-c2cn(C(C)C(=O)O)nn2)cc1)=O)C 25494,CC(C)CC(CCO)N(C)C(C1(O)CCCN(C(C2CCS(=O)(=O)C2)=O)C1)=O 25495,C1(O)(CN(C)C(c2cnco2)=O)CCN(C(c2coc(Cl)n2)=O)C1 25496,CC1CN(C(=O)C(C2(O)CCC2)NC(c2cncc(CO)c2)=O)CCS1=O 25497,C(CNC(C1(F)CC=CC1)=O)(CC(=O)N1CCC1(CO)CO)OC 25498,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25499,C1(CC(=O)NC2CC(CCNC(=O)COC3CC3(F)F)C2)(N(C)C)CCC1 25500,C(=O)(C1=NNC(=O)CC1)NC(C1CCCN1C(=O)C(C)(C)NS(C)(=O)=O)C 25501,C1(NC(C(C)OCCC#C)=O)CN(C(=O)Cc2csc(C3CC3)n2)CCC1C 25502,C(C1CCCCCC1)=CC(=O)NC(CN(C(C1(C(=O)NC)CCC1)=O)C)C 25503,N1(Cc2ccc(C(=O)OC)cc2)CC2CCN(C(C3(C)CCOCC3)=O)CC2C1 25504,c1(OC)cccc(C(=O)NNC(=O)COC)c1CCO 25505,c1(C(=O)NCC2N(C(CCC)=O)CCCC2C)cc2ccccn2c1 25506,Cc1cc(C(N2CC3CC2CCN3C(c2csc(=N)[nH]2)=O)=O)c(S(N)(=O)=O)s1 25507,N1(C(C2C3CN(C(C(C)N(C)C)=O)C2C3)=O)CC2CCC1C(CO)C2 25508,c1(C(=O)NC2CCCN(C(C(C)NC(CC)=O)=O)C2)cccc(CC)c1O 25509,N1(C(=O)Oc2ccccc2)CC2C(CNC(c3cc(Cl)ncn3)=O)C2C1 25510,c1(C(=O)NC2CCC(N(C)C(C3CC(Cl)(Cl)C3)=O)CC2)ccc(C#N)cc1 25511,Cc1ccc(F)c(C(=O)NCc2occc2C(=O)NC(C)C(F)(F)F)n1 25512,C1(NC(=O)CN2CCS(=O)CC2)CN(C(=O)CCC2CCCCCC2)CC12CC2 25513,C=CCC(C(=O)NC1(COC)CN(C(=O)C(F)C2CCOC2)C1)OC 25514,c1(C(=O)NC(C2(O)CN(C(C3(S(N)(=O)=O)CC3)=O)C2)C)ccc(=O)n(CCO)c1 25515,S(=O)(=O)(c1cccc(N2CCC(CCO)C2)n1)NCC(=O)NC1CC1 25516,c1(N2CC(NC(CCOCCOC)=O)C(C)CC2)ncc([N+](=O)[O-])cn1 25517,C1(C(=O)NC(CCCC)CNC(=O)COC2(C)CCC2)Cc2nccn2C1 25518,Cc1nn(C)c(C)c1C(=O)NC(CNC(c1cc[nH]c1C1CCC1)=O)C(C)(C)C 25519,C1(C#CC(=O)NC2CCC(NC(c3nc(C)c(C)[nH]c3=O)=O)CC2)(CC)COC1 25520,CC(CCCO)N=c1cc[nH]cc1S(=O)(=O)NCCCc1cccc([N+](=O)[O-])c1 25521,Cc1cc(C(=O)NC2CC3CCC2N(C(C2(CCF)CCC2)=O)C3)cc(C)c1Cl 25522,c1(C(=O)NCCC2(NC(c3nc(Cl)cs3)=O)CCC2)cccc(F)c1O 25523,C1(CC(=O)NC2(CNC(CCC#C)=O)CCCC2)CCOC(C(C)C)C1 25524,C1(NC(c2c(C)sc(Br)n2)c2nnnn2C)C=C(c2ccc(Cl)cc2)CCC1 25525,CCCC(CCCNC(C1CC(C)OC1=O)=O)NC(c1ccnn1CCC)=O 25526,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)CCSC(F)(F)F)C1 25527,N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(C2CCC(c3ccccc3)O2)=O)C(C)C1 25528,c1(C(=O)NCCN(C(CCc2c(C)nn(C)c2C)=O)C)nc(=N)[nH]c2ccccc12 25529,C(C(=O)Nn1cnnc1C)C1CN(C(CCc2c(C)ncs2)=O)C(C)(C)C1 25530,C(C(CC(C)C)C(=O)N(C1CCCC1O)C)NC(c1cc(C)oc1)=O 25531,C(=O)(C1=CCCS1)NC1C(CNC(CCc2ccc(C)o2)=O)C1 25532,N1(C(C2(C#N)CC23CCC3)=O)CC2CC(C1)N(C(c1cnc3cc[nH]c3c1)=O)C2 25533,c1(C(=O)NCC2CCC(NC(=O)CCC3CCOC3)CC2)c[nH]c2ccncc12 25534,C(=O)(CCC(C)(C)N(C)C)NC1CC(CNC(c2ncc(OC)cn2)=O)C1(C)C 25535,N1(CCO)CC2(CCCCC2)CC1N(CC(F)F)C(C)C1CC1 25536,C1(CC)CC(O)CN1C(=O)CCCCN(C)C.c12cc(on1)CNC2=O 25537,c1(C(=O)NC(C2(O)CN(C(=O)CCC3CC3(Cl)Cl)C2)C)cn2ccccc2n1 25538,C1(CNC(CC(C)SC)=O)CN(C(C2CC=CCC2)=O)CCC1C 25539,CCCCC(CC(=O)NC1CC2OCCCC12)NC(c1cccc(CC)n1)=O 25540,CC1CCN(C(=O)C(=O)NC(c2cc(C(F)F)[nH]n2)=O)C(C)C1CC(N)=O 25541,C(c1cc2ccccc2o1)=CC(N1CC(CNC(CNC(N)=O)=O)OCC1)=O 25542,c1(C(N2CC(O)CC(NC(CC(=O)OC)=O)C2)=O)c(F)ccc(C)c1Cl 25543,N1(C(C2C(CC)OCC2)=O)CCC(C(C)NC(=O)C=CC(C)C)CC1 25544,c1(OC)cnc(CNC(=O)C(=O)NCC2CCCC(C)C2)cc1Br 25545,N1(CC(=O)NC2CCC(n3cc(CSCCOCCO)nn3)C2)C(=O)CCC1=O 25546,C=C(C(=O)N1CCCC1CNC(c1ccc(OC(F)(F)F)cc1)=O)C(F)(F)F 25547,c1(C(N(CC(C)O)CCNC(=O)C=Cc2cnccn2)=O)cc(O)cc(C#N)c1 25548,Cc1ccc(C)c(C(=O)NCC2CCC2)n1.N12CCCC(C1)CC1(CC1)CCC2=O.O.CCO.C(OC)C 25549,C1(NC(C2C(C)CC2)=O)CN(C(C2CN(C3CCCC4(CC4)C3)C2)=O)C2(CCC2)C1 25550,CC1CN(C(=O)CN2C(C)CC2(C)C)CCN1C(=O)CCCC(=O)C1CC1 25551,CCCC(CCC)=CC(=O)OCC(c1nc(C2CCCCC2)no1)C 25552,N1(C(C=CC)=O)CCC12CN(C(c1cncnc1)=O)C2 25553,CN1C(=O)OC2CN(C(C3(F)CN(Cc4ccncc4Cl)C3)=O)CC12 25554,N1(C(CCC#C)=O)CC(N(C(=O)CN(C)C)C)C2(CC2)C1 25555,N1(C(C(Br)=C(C)C)=O)CC(CNC(=O)C(C)C(C)(C)C)OC(C)(C)C1 25556,C1(C(N(CCNC(CCOCCOC)=O)C(C)C)=O)CCC(N=[N+]=[N-])CC1 25557,N1(C(c2ccc[nH]2)=O)CCC2CCCN(C(c3ncoc3Br)=O)C2C1 25558,C=CC1COCC1NC(=O)C(CCOC)NC(c1ccc(COC)cc1)=O 25559,CC(C)CC(C(=O)NCCSC1C2CCCOC12)NS(C)(=O)=O 25560,c1(NCC2(CCC)CC2)nc2ccccc2nc1NCc1cc(Br)ccc1N 25561,C123COC(CN1C(=O)C1(CC1)CCn1cc2nn1)C3.C1(OC)CC(O)CO1 25562,c12ccc([nH]1)C(=O)NOC2.C(CCCCC)NC(CC1(C=C)CC1)=O 25563,c1(C2(N)CC2)cccc(C)c1.C(c1ccsc1C(F)(F)F)=CC(=O)C(=O)COC 25564,C(CC(N)=O)(C(=O)N1CCCC1c1ccco1)NC(C(C)C1CCCC1)=O 25565,C1(NC(c2occ(C)c2C)=O)CCCCCCC1NC(c1cnn(C2CC2)c1)=O 25566,c1(C(C)(C)C)ncc(C(=O)NCC2CCC2N(C(=O)C2CC2)C2CC2)s1 25567,O(NC(=O)C(Cn1ccnn1)NC(=O)Cn1cccc1)CC#C 25568,C(C(CC)(CC)CO)NC(c1cc(CNC(C2C(CCC)CCC2)=O)nn1C)=O 25569,C1(CCC(=O)NCC(C)NC(=O)C(C)(C)C)CCc2ccccc2NC1=O 25570,N1(C(C=CSC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25571,CN1C(=O)NCC1C(=O)NC1CCCC1CNC(=O)C=Cc1cccnc1 25572,C#CCCC(O)C(=O)NC1(C)CN(C(=O)C2=CSCCO2)C1 25573,O(P(C)(=O)CNC(=O)CCOC1CN1C(=O)CCCC(C)O)CC 25574,Nc1nccnc1C(=O)NCC1CN(C(=O)Cc2cn[nH]c2)CC1C(F)(F)F 25575,CC1C(NC(c2ccsc2C(F)F)=O)CC2CCC1N2C(C1CN(C)C(=O)N1)=O 25576,c1(CN2C(C(=O)NCC3OCCO3)CC(F)(F)C2)ccc(F)c(F)c1O 25577,c1(C(=O)NCC(N2CCN(C(C(C)NC(C)=O)=O)CC2)C)ccn2ncccc12 25578,C12CC3CCC1(C3)CC1(CCCO1)C(=O)N2.C(F)(F)(C(=O)OC)c1ccccc1 25579,N1(C(C2(NC(C3CC(CC)C3)=O)CCCCC2)=O)CCCCC(CO)C1 25580,C(COC)(C(=O)N1CCCC1C(=O)N(C)C)NC(C(c1cncnc1)C)=O.C1(C)CC1 25581,N1(C(CNC(C(C)OCC2CC2)=O)=O)CCC(O)C(C)(C)C1 25582,c1(C(N2CCCC(F)(CNC(c3ccns3)=O)C2)=O)cccc2nn[nH]c12 25583,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=Cc2cnc[nH]2)c(C)s1 25584,N12CCOC(C)(C1)Cc1cn(nn1)CC2=O.c1(OC)ccc(OC(F)F)cc1 25585,N1(c2nccc(C#N)n2)CCCC(O)(CNC(C2CCCSS2)=O)CC1 25586,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25587,c1(-c2nc(C(CC)CC)nn2Cc2cccs2)cnc2n1CCCCC2 25588,C(CCC(=O)N1CCC(NC(=O)C(N2CC3CC3C2)C2CC2)C1)NC(COCC)=O 25589,C#CCCCCC(=O)N1CCC(C(F)(F)F)C(NC(c2cccnc2C)=O)C1 25590,C1(OC)CCN(C(c2nn(-c3cccc(C#N)c3)c3c2CCC3)=O)C2(CC2)C1 25591,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25592,C12CC(=NO1)C(=O)N(C(C)C)C2.C=CC(C)C(=O)NCC(F)F 25593,CCCC(CCC)CC(=O)N(C(C(=O)NCC1(C(F)(F)F)CC1)C1CC1)C 25594,c1(C(=O)NC(CCNC(C2N(CCC)C(=O)CC2)=O)C)cn2c(n1)CCC2 25595,c1(C(N2CCC(F)(CNC(CC=C=C)=O)C2)=O)cc2cccnc2cc1F 25596,N1(C(CCC(C)SC)=O)CC(NC(c2csc(C)c2C2CC2)=O)C(C2CC2)C1 25597,c1(C(=O)NCC2C(C)(C)C(NC(=O)CCc3cccnc3)C2)ccc2c(c1)CC2 25598,C1(C(=O)NCC(C(C)O)O)(CO)CCN(C(C2CC=CCO2)=O)CC1 25599,N1(C(CC2C(C)(C)C2)=O)CCC(OCCNC(c2cocc2Br)=O)C1 25600,C1(NC(C2CC(C)OC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25601,C1(C(=O)NOCCSC2CC2)CN(C(c2cnco2)=O)C2(CCC2)C1 25602,c1(C(=O)NC2C(NC(C3(Cl)C(C)(C)C3)=O)COC2)cccc(OCC(F)F)n1 25603,C(CCN=c1[nH]c(=NCC2COC(C)(C)C2)[nH]c2c1CSC2)NC(C(C)C(C)O)=O 25604,c1(C(=O)NC2CCN(C(C3CCc4nccn4C3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 25605,c1(N2CCCC(CCC(C)C)C2)nc(=NCc2ccc(C#N)o2)[nH]c2c1CSC2 25606,c1(C(N(C)CCNC(c2csc(S)n2)=O)=O)ccc(-c2ccncc2)s1 25607,c1(C(N2CCN(C(c3nc(Cl)sc3Cl)=O)C3C2C3)=O)cn2ncccc2n1 25608,C(=O)(C(CCC(=O)OCC)Nc1cc(C)ccc1Cl)OCC 25609,N1(CCN(CCC)CCNC(c2cnccc2C)=O)NC(=O)CCC1=O 25610,Cc1nc2c(NC(=O)NCC=Cc3sccc3Br)cccc2o1 25611,c1(OC)ncc(Br)cc1CN1CCC(CC(=O)NCCCC(F)(F)F)CC1 25612,c1(C(N(CC(CC)CS(C)(=O)=O)C)=O)ncc(C)cc1Cl 25613,Cc1cccc(OC(C(=O)Oc2ccccc2N(C)C)C2(C)CC2)c1 25614,C1(CNC(C(C)Nc2ccccn2)=O)CN(C(C23CC(C2)C3)=O)CC1(F)F 25615,N1(C(C2CCCC(=O)C2)=O)CC=C(C(=O)NCC(c2cccnc2)O)CC1 25616,CCCCC(COC)(c1nnnn1Cc1cccs1)NC(c1ccncc1)C 25617,CC1=C(C(=O)NC(CCN(C(=O)CC2CC(O)C23CCC3)C)C(C)(C)C)CCO1 25618,CC1CCN(C(c2cc(Cl)nnc2O)=O)CCN1C(C1C2CCC1CC2)=O 25619,N1(C(CSC(C)=O)=O)CCCC(C)(C(=O)NCCOC2CCC2)C1 25620,N1(C(C(CC)=CC)=O)CC(NC(=O)CN(C)CC)CCC1C 25621,C(=O)(C(O)CC(C)(C)C)NCC1CC(CNC(C(C(=O)OC(C)(C)C)OC)=O)C1 25622,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25623,CC1CC(CN(CC(c2cccs2)C)C)C1 25624,C(N=c1nc2scnc2c(NCC2CSCCO2)[nH]1)C1CCN(CC)C1 25625,c1(NC(CC2N(C(C(c3cnn(C)c3)C)=O)CC2)=O)ccc(O)cc1F 25626,S1(=O)(=O)c2ccc(nc2)N1.c1(NCC2(CC)CC2)cn(C)nc1C1CC1 25627,n1(O)cc(CNC(=O)C=CC=O)nn1.C(C)(CNC(C)=O)OCC#C 25628,N1(CC(=O)NC2(CF)CN(C(C34CC(C)(C3)C4)=O)C2)C(=O)CCC1=O 25629,Cc1nc2ccsc2c(=NCCNC(c2ccc(F)c(F)c2F)=O)[nH]1 25630,C1(C(=O)N(CC(O)CN)C)(COC)CCCCC1.C12CN(CC1OC)C2=O.C(C)(=O)O 25631,N1(Cc2cccc(C#N)c2)Cc2ccc(NC(c3cc(Cl)c(Cl)cn3)=O)cc2C1 25632,C1(NC(C(C(=C)C)(C)C)=O)CC2CCC(C1)N2C(=O)C1=CC2CCCC12 25633,CCC(CC)CCC(=O)N1CCC(N(C(=O)C#CC2CCC2)CC)C1 25634,N1(Cc2cnc(=N)[nH]c2)CCC2(CC1)CC2C(N1CCOCC1c1cccnc1)=O 25635,N1(C(CCN(CCC)C(c2cc[nH]n2)=O)=O)CC2C3CCC(O3)C2C1 25636,C1(NC(CC2CCC(C)(C)C2)=O)CCN(C(=O)CC23CCC(CC2)OC3)CC1F 25637,C1(C2CCC2)(NC(c2c(C)nn[nH]2)c2nnnn2C2COC2)CC1 25638,c1(C(=O)NCCCC(C)NC(=O)Cc2ccc(F)cc2)ccc2c(c1)CC(=O)N2 25639,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]c2=O)=O)CC(O)C1 25640,N1(C(CC(C)C#N)=O)C(C(N2CC(F)C2)=O)CCC12CC2 25641,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25642,C1(NC(C(CC)C)=O)(CNC(=O)C(C)(F)C(=O)OC)Cc2ccccc2C1 25643,CCCCCC(=O)NC1CCC(CNC(c2ccn(-c3cccc(O)c3)n2)=O)C1 25644,c1(C(=O)NC(CNC(c2c(C)cccn2)=O)C(C)(C)C)ccc(F)c2occc12 25645,c1(COC)cc(NC(C2CC(OC)(OC)C2)=O)ccn1 25646,c1(NC(C2(CCC=C)CN(C(C3CC3=C)=O)C2)=O)cncnc1OC 25647,C(CO)(CCCCNC(C1CC(F)C(=O)N1)=O)NC(=O)CCN1CCOCC1 25648,N1(C(C(C2CCOCC2)C)=O)CC(=O)CC1C(=O)NCCN1C(=O)CNC1=O 25649,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C)NC(c1ccoc1)=O 25650,CC1CN(C(C2CCCC2)=O)CCC1CNC(c1c(F)cccc1Cl)=O 25651,CN1CCN(C(c2c(CNC(=O)CCc3cn[nH]c3)cnn2C)=O)CC1CO 25652,c1(C(N2CC3C(CNC(c4c(C)ccnc4O)=O)(C3)C2)=O)cccc2[nH]ccc12 25653,C(c1ccc(F)c(F)c1)=CC(=O)NC1CC(C)CN(C(c2cnccn2)=O)C1 25654,C1(C(=O)NCCCN(C(CNS(CC)(=O)=O)=O)CC2CCCC2)CCN(C(C)C)N1 25655,Cc1cc(C(F)(F)F)cc(C(=O)NC2CCC2NC(C2(CF)CC2)=O)n1 25656,c1(C2(C(N(CCN(C(=O)CCc3nc[nH]n3)C)C3CC3)=O)CC2)ccccc1 25657,c1(CN(C(C(CCC)C)=O)CCOCC)cc2n(n1)CC(F)C2 25658,N1(C(C2CC(=O)N(Cc3ccccc3Cl)C2)=O)C2CCC1CC1(C2)CC1(F)F 25659,c1(C(=O)NC2C(NC(Cc3nnc(C)o3)=O)CCCC2)cccc(O)c1Cl 25660,CCC(F)(F)C(C)(C)C(=O)NCC1CC(NC(=O)CCS(C)=O)C1 25661,CCCCCO.C1(n2ccnc2)(CCN2CC2)CCC1 25662,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25663,C(=O)(CCCCCC#N)NC(C)CC(C)NC(c1cccc(OC(F)F)c1)=O 25664,C(=O)(C1=C(Cl)CCOC1)N(CC)CC.CCC(CN(C(C1CCCC1C)=O)CC)C(C)(F)F 25665,C(=O)(CC(C)(C)O)NCCOCC(=O)NCC(n1cncn1)C 25666,CC1(C)CC(NC(=O)CCC2CCOCC2)CN1C(=O)CN1CCCCCC1 25667,N1(C(c2nc(C)oc2)=O)CCN(C(c2cc(Br)sc2C)=O)C(C)C1 25668,C1(C(C(C)C)NC(=O)C(Cl)=CCl)CN(C(=O)C=Cc2cn(C)cn2)CCO1 25669,n1(CCC(=O)N2CCC2CNC(c2cnn[nH]2)=O)cnc([N+](=O)[O-])c1.C1(C)CCCCC1 25670,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25671,C=CCCC(C(=O)NC(C(N)=O)C1CCCC1)NC(c1cc(Cl)n[nH]1)=O 25672,Cc1cc(-c2cn(CC3C(C)CCN3C(C3CC(=CBr)C3)=O)nn2)c(Cl)cc1F 25673,c1(C(=O)NCC(C)(C(C)C)NC(C(CCCC)C)=O)nccn2cc(C)nc12 25674,N1(C(C(=O)NCC2(COC)CC2)Cc2nc(C)cs2)CC2C3C=CC(O3)C2C1 25675,C1(c2nnc(C)o2)CN(C(c2coc(C3CC3)n2)C(=O)NC(C)C)CCO1 25676,N12CC3(Br)CC3(C1)NC2=O.S(C)(=O)(=O)N(CCOC)C 25677,C1(C)(C(N(C)CC)=O)CC(NC(=O)CC2CCSCC2)C1 25678,C1(NC(C(C=C)(F)F)=O)CS(=O)(=O)CC1NC(c1cc(C)cs1)=O 25679,Nc1cccnc1C(=O)NC1CCC(C(=O)NCC2CC2c2ccsc2)C1 25680,C1(C(N(CC(CC)NC(c2nc(C)n(C)n2)=O)C)=O)CC2(C)CC1CO2 25681,CS(=O)(=O)CC(=O)NC1CCOC(C(=O)NOCC(=O)OC(C)(C)C)C1 25682,N1(C(CCOC)=O)Cc2nccn2CC(NC(=O)CC2CCCO2)C1 25683,c1(C(=O)NC2CCCCCN(C(CC=C)=O)C2)n[nH]c2cc(Br)ccc12 25684,Cn1cnc(I)c1C(N1CCC(c2nc(C3CC3)no2)CC1)C(=O)NC1CCC1 25685,C1(CNC(COc2ccc(C#C)cc2)=O)CN(C(C2(C)CC2(F)F)=O)CC12CCC2 25686,Cc1[nH]nc(C(=O)NCC2CN(C(c3ocnc3C(F)F)=O)CCO2)c1F 25687,C(=O)(CCCC(C)O)N(C(C)C)CCNC(=O)Cc1ccnc(Br)c1 25688,N1(C(c2c(C(F)(F)F)nc(C)o2)=O)CC2CN(C(=O)C(C)CS(C)=O)CC2C1 25689,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25690,Cc1c(C(N2CCC(NC(=O)CC(F)(F)CC(F)F)C2)=O)sc2[nH]cnc(=S)c12 25691,c1(C(=O)NC(CN(C(c2c[nH]nc2C(F)F)=O)CC)C)n[nH]c2cc(Cl)ccc12 25692,N1(C(CCOC)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C1c1ccccc1 25693,N1(C(COCC(=O)OC)=O)CC2CC1C2NC(=O)C(C)(C)n1ccc(C2CC2)n1 25694,CC1CCn2cc(C(=O)NC(C)(C)CNC(=O)Cc3c[nH]c(=N)nc3O)nc2C1 25695,N1(C(c2ccc(C(F)(F)F)nc2)=O)CC=CC(C(N2C(CO)CC2CO)=O)C1 25696,CCCCS(=O)(=O)CC(=O)NCCCN1CCN(C(=O)C2=CS(=O)CCC2)CC1 25697,C#Cc1ccc(C(=O)NC(C)CN(C)C(c2cscn2)=O)c(OC)c1 25698,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC1(F)F 25699,C1(C(=O)NC(CNC)(C)C)C2CC2CN1C(=O)C(C)OCC(F)(F)F 25700,C1(NC(c2nn(C)c(O)c2)=O)CN(C(C2CC(C(C)(C)C)=NO2)=O)CC2(CC2)C1 25701,N(C1COc2ccccc21)CCOC(C)C(=O)NC(CCC1CCC1)C(=O)NC.CO 25702,c1(C(C)(C)C)cccc(C(c2nnnn2C2CCCC2)NC(=O)CC2CCOC2)c1 25703,N1(CC)CCCC(C(N2CC(CN3CCN(C(C4SCCCS4)=O)CC3)C2)=O)C1 25704,N1(C(C(Cc2c(C)ncs2)NC(=O)OC(C)(C)C)=O)CCCC(N(C)C)C1 25705,C(C)(C)(C#Cc1cn(C2(C)CC2)nn1)NC(C(CC)OC1CCCCC1)=O 25706,C(C)(CCCC(=O)NCC1CNC(=O)CO1)NC(C1C(CCOC)C1)=O 25707,C1(COC)CN(C(=O)CCN2CCCC2)CCN1C(c1sncc1C)=O 25708,c1(NC(C2C(NC(c3ccc(C)s3)=O)CC2)=O)cc(F)c(O)cc1C 25709,Cc1ccc(C(N2CC(C(=O)NCCCn3cccn3)C(C)C2)=O)nc1 25710,C1(C(N2CC(CNC(CCOCC#C)=O)(OC)C2)=O)CCOC(CC)C1 25711,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(c1cnn(C(C)C)n1)=O)C2 25712,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25713,c1(OC)ccn2c(-c3c(C)cccc3F)nnc2c1 25714,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25715,c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc2c(c1)C(=O)NC2=O 25716,c1(OCCC(=O)NC2(CC)CCN(C(=O)CNC=O)C2)cc(Cl)ccc1Cl 25717,N1(C(CCN2C3CC(N)C2CC3)=O)CC(=O)Nc2ccccc21 25718,c1(COC)nn(C)cc1C(=O)NC(C1CN(C(C2(F)CC2)=O)CCO1)C 25719,c1(OC)ccc(F)c(C(=O)NC2CC3(C2)CC3NC(c2nccc(C)n2)=O)c1 25720,C1(NC(c2c(C)noc2)=O)CC(C)N(C(=O)Cc2ccc(C3CC3)s2)C1 25721,N1(C(CCC2N(C(C3C=CCCC3)=O)CCC2)=O)CC(O)C(O)C1CO 25722,S(=O)(=O)(c1ccccc1F)NCC(=O)NC(CNC(CCCCNC(C)=O)=O)C 25723,c1(C(N2CC(CN(C(=O)CC3C(C)C3(F)F)C)C2)=O)cc(-c2cnn(C)c2)on1 25724,c1(CN(CCCCCO)C(c2cc(C)cc(Cl)c2)=O)ccc(S(=O)(=O)N(C)C)cc1 25725,C1(C(=O)NCC(CC)(C)C)CN(C(c2ccc(O)nc2C)=O)CC1(C)C 25726,C1(NC(C2CCC(C(N)=O)CC2)=O)CCN(C(C2CC3CCC2O3)=O)CC1CO 25727,C(C(C)(C)CO)N(C(=O)C(Cn1ccnn1)NC(=O)CC1C=CCC1)C 25728,N1(C(c2nnn(C)n2)=O)C2CCC1CC(NC(=O)CCC1CC1)C2 25729,C(=O)(C1CCc2nccn21)N1CC=C(CC(=O)N)CC1.C(C)(C(=O)N(CCO)C)OC 25730,C12(CNC(c3cc4ccncc4[nH]3)=O)CCC(CN(C(c3ccns3)=O)C1)C2 25731,C1(C(=O)NC2CCCN(C(CC)=O)C2)CC(C)CN(C(=O)CSCCCC)C1 25732,c1(NC(c2ccccc2-c2cocn2)=O)c(O)ccnc1F 25733,c1(C(N2CC(C(C)NC(=O)C(C3(O)CCCC3)F)OCC2)=O)cc2occc2s1 25734,C(=O)(C(CO)C(C)(C)C)NCC1(C(=O)NC(C=C)C(F)(F)F)CC1 25735,c1(OC)ccc(C(=O)NC(CNC(=O)CCC2NC(=O)NC2=O)C2CC2)nn1 25736,C=CC(CCC)CC(=O)NC1C2CCN(C(c3sc(C(C)(C)C)nc3C)=O)C12 25737,C(C(O)CC(=O)NCc1ccccc1)NC(C1CN(C(C(C)CF)=O)C1)=O 25738,c1(C(N2CCC(C3N(C(C4CCC5(CC4)CC5)C)CCC3)C2)=O)nnc(O)nc1O 25739,c1(C(=O)OC)c[nH]c(=NC(CNC(c2cnnc([N+](=O)[O-])c2)=O)C(C)C)cn1 25740,C(=O)(C1CCCn2nccc21)N(CC(CN(C(CCC=C=C)=O)C)O)C 25741,N1(C(=O)CCOc2cc(F)ccn2)CCC2C1CCN2C(C1CCCCC1)=O 25742,c1(N(C)C(C)C)ccc(S(=O)(=O)NC(c2c(CC)cc(Br)cc2)=O)cc1 25743,CC(C)C(F)(CNC(=O)CC1CCC(C)(C)O1)C(=O)N(C1CCCC(O)C1)C 25744,Cc1ccc2[nH]c(=NC(C)C3CCN(C(C4CCCCC4O)=O)CC3)sc2n1 25745,c1(NC2(CNC(C(CCC)OCC)=O)CCCC2)cccc2c1CN(C(C)=O)C2 25746,N1(C(Cc2cc(C)cc(Cl)c2)=O)CCCc2c(O)cccc21 25747,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C)(CNC(=O)CC(C)(O)C2CC2)C1 25748,c1(SC)ccc(C)c(C(N2CCCCC2CCN(C)C(c2nnc(C)s2)=O)=O)c1 25749,N1(C(C(C)OCC)=O)CCN(C2CCN(C(=O)C(O)COC)CC2)C(=O)C1 25750,C1(NC(Cc2c(C)nn(C)c2Cl)=O)CC2CCC(C1)N2C(=O)CCc1cnn[nH]1 25751,c1(Cc2nn(-c3cc(C)ncc3)c(C3CCCC3C(C)C)n2)c(F)cccc1Br 25752,N1(C2(O)CN(C(C)CNCCc3ccccc3Cl)C2)C(=O)c2ccccc2C1=O 25753,c1(NC(c2csc(C(=O)NC3CCCC(CO)C3)n2)=O)cc(Cl)ncc1[N+](=O)[O-] 25754,c1(C(N2C(C)(C)C(CNC(c3nc(Cl)cs3)=O)CC2)=O)ncnc2c1CCC2 25755,CCCC(C)(C)CC(=O)NCCC1(O)CN(C(c2ccsc2-n2cnnn2)=O)C1 25756,Cc1ccc2cc(C(=O)N(C3CCCN(C(c4sccc4C)=O)C3)C)nn2c1 25757,C1(OC)CN(C(C2(F)CC2)=O)CC1NC(C1(O)CCOCC1)=O 25758,N1(C(C2(NC(C3(CCCC)CC3)=O)CC2)=O)CC2CC1CN2C(C)=O 25759,CN1CC2C3CCCN(CCC13)C2N1C2CCC1CC(n1cc(C3CC3)nn1)C2 25760,c1(C(=O)NC2C(OC)CN(C(C3(CC)C=CCC3)=O)C2)snc2ccccc12 25761,c1(C(N(CC(CN(C)C)O)C)=O)sccc1CNC(c1cnn(C2CC2)c1)=O 25762,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25763,c1(C(N2CCC(NC(c3ccc(C)nc3C)=O)C2(C)C)=O)ccc(C#N)c(C)n1 25764,c1(C(=O)NC(CCN(C(C(C)CC(N)=O)=O)C)C(C)(C)C)ccc2occc2c1 25765,CN1CC2CCC(NS(=O)(=O)Cc3ccc(-c4cccc(C(N)=O)c4)cc3)C2C1 25766,c1(CC(=O)NC(C=CC(=O)NCC(C)CC2CC2)C)cnn(C)c1 25767,c1(N(C)C)ncc(C(=O)NC2(C3CCCCN3C(=O)CCF)CC2)cc1Cl 25768,c1(C(=O)NCCN(CCCOC)C(C2CCC(C(N)=O)CC2)=O)cccc(C)c1 25769,N1(C(c2c(C)cc(SC)o2)=O)CC2CN(C(c3cc(C)c(Br)o3)=O)CC2(C)C1 25770,c1(CNC(C2CCN(C)C2)=O)c(C2CCCN(c3nnn(C)n3)C2)cnn1C 25771,CCCC(C(=O)NC(C(=O)N1CCC(CC(=O)OC)C1)C(C)OCC)OC 25772,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25773,Brc1cc(I)c(CNC2CC23CCC3)cc1Br 25774,n1(CCC(=O)NC(C2CN(C(=O)C(C)(C)CCl)C2)C)ccc2cc([N+](=O)[O-])ccc12 25775,N1(C(Cc2cc(C)ncc2)=O)CC(N(C(=O)C(F)=CC2CC2)CCO)C(C)(C)C1 25776,c1(SC)ccc(C(=O)NC(C)COCCC(F)(F)Cl)cc1 25777,Cc1nc(O)nc2ccc(NC(C)C)cc12.N12CCC(C1)CNC(=O)C=CC2=O 25778,c1(OC)ccc(C(N2CCOC(CN3CCCC3=O)C2)=O)cc1-n1cccc1 25779,Cc1nnc(CC(=O)NC2CC2NC(c2cn[nH]c2)=O)o1 25780,CC(Cc1cccs1)N=c1[nH]c(N(C)Cc2ccc(Br)cc2Cl)nc2ccsc12 25781,Cc1ccccc1C(=O)NCC1(CNC(=O)CC2COCCO2)CCCCC1 25782,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(C(N)=O)CC3)=O)CO2)C1 25783,c1(C(N2CC3CC3(C(N3CCc4sccc4C3)=O)C2)=O)cc2n(n1)CCCO2 25784,c12nc(nc3ccccc13)CC1(NC(C3C(=C)CC3)=O)CCCN2C1.OC 25785,c1(C(=O)NCC(CNC(C2CCC(N(C)C)C2)=O)F)ccccc1-n1ccnn1 25786,C(CC(C)(C)C)(C(=O)NCCCCC(=O)Nc1cc(C)c(F)c(C)c1)OC 25787,c1(OC(N2CCC(C(=O)O)C2)=O)ccccc1OCC1CCCO1 25788,C(C(C)(F)C(C)(C)F)N(c1n(CC=C)c(CC(=O)NCCCCO)nn1)CCO 25789,C1(CC=C)(NC(c2cocn2)=O)CC2CCC(C1)N2C(C1CCCO1)=O 25790,N1(Cc2ccc(C#C)s2)CCCN(C(c2ccnc(Cl)c2)=O)CC1 25791,N(C1CN(C(=O)Cc2cncn2C(C)C)Cc2ccccc21)C(CC=CCC)=O 25792,C(=O)(C(C(C)(C)C)NC(C1CN2CCN1CC2)=O)N(C)Cc1cocn1 25793,C(C(C)(C)CN(C(c1nnn(-c2ccccc2)n1)=O)CC)NC(C(F)OC)=O 25794,c1(OC)cncc(C=CC(N2C3CCC2C(CNC(c2ccsc2C)=O)C3)=O)c1 25795,Cc1cc(C(=O)N(C2CCN(C(c3ccnc(O)c3)=O)C2)C)nc(O)n1 25796,c1(C(N2CCC(n3ccnn3)C2)C(=O)NCC)ccc(Oc2ccccc2)nc1 25797,c1(CC)cc(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)ccc1OC 25798,c1(CN2CC(C(=O)Nc3cc(Br)cc(Br)c3)SCC2)cccc2c1CCC2 25799,CCC(CCC(=O)NCC(CC(=O)NCC(O)C(C)C)C1CCC1)OC 25800,C1(SC(C)C(=O)N=CC2CCCC2)CCCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 25801,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCCO1)=O 25802,C(=O)(CCCCCCCCNC(c1cc(COC)no1)=O)OCC 25803,c1(OC)cc(OC)c2c(c1)CCN(C(=O)C(C)(C)CN1CCOCC1)C2 25804,c1(C(=O)NCCN(C(C2N(CC)CCCC2)=O)CCOC)ncc(N)cc1Cl 25805,CCCCCCCCCCCCNCC(=O)Nc1ncc[nH]1.c1(=O)c(=O)n1C1CC1 25806,c1(C(N2C(C)(CNC(C3(C)C(C)CCC3)=O)CCC2)=O)cn2c(n1)CCCC2 25807,CC(C)(COC1CCCC1)C(=O)NCCCNC(C1(O)CCOC1)=O 25808,CC1(C)CC(C)(C)CC(O)(CNC(=O)NCc2cscc2Br)C1 25809,C1(CNC(Cc2ccc(CC)s2)=O)CN(C(=O)C=CS(C)=O)CC(C)(C)O1 25810,c1(C(N(CCC(=O)NCCSc2ccco2)CC2CC2)=O)cccc(=O)o1 25811,C1(C(=O)Nc2cccc(CNC(C3COCCC3(F)F)=O)c2)CC2(C1)OCCO2 25812,c1(C(N2C(CC)C(NC(=O)C(C)Sc3ccccc3)CC2)=O)cc(C)ccc1N 25813,C12(C(N(C3CCCN(C(C(CCSC)OC)=O)C3)C)=O)C3C4C1C1C2C3C41C(N)=O 25814,C1(NC(c2c(C)nc(O)s2)=O)C2CC3C(C2)C13C(=O)NCc1ccccc1F 25815,c1(C(N2C(C)CN(C(c3cncc(N)n3)=O)CC2)=O)cc2c(nc1O)CCCC2 25816,CCC(C)(C(=O)N1CCC(C)N(C(c2cc(N)c(F)cc2F)=O)CC1)C(F)F 25817,C(=O)(C(C)(C)C1=CCN(C(=O)CC(O)CC(C)C)C1)NCC(CC)C#N 25818,C(C(C)(C)C#CC(=O)N1CC(O)(C(C)=C)C1)NC(C(CC#C)C1CC1)=O 25819,CC1(C)CN(C(c2cccnn2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)O1 25820,N1(C(C2(C)CCNC2=O)=O)CC2CC(NC(=O)CN3CC=CC3)C(C2)C1 25821,Cn1cnc2c(N3CCCCC(NC(c4cncc(Cl)n4)=O)C3)nc(Cl)nc12 25822,C(=O)(C(C)(C)c1sccc1Cl)NCCN(C(=O)Cn1nnc(C2CC2)n1)C 25823,C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1C(F)(F)CCN(C(C(C)OCCOC)=O)C1 25824,c1(OCC#C)cc(OC)ccc1CN1CCC1CNC(c1scnc1C)=O 25825,Cc1nn2[nH]cnc(=O)c2c1S(=O)(=O)NC(c1ccccc1)C1CC1 25826,N1(C(c2cc(CC)sn2)=O)CC(OC)C(OC2CC2)C1.c12coc(n1)CNC2=O 25827,C(=O)(C(CNC(=O)CNC(C)=O)CC1CCCC1)N(CCC#C)CCO 25828,N1(C(c2ccc(N)c(O)c2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)CC12CCC2 25829,c1(OC)ccccc1NC(c1ccc(C#N)s1)=O.C1(CN(C)C)C(=O)N1 25830,C12(CNC(=O)C(C3CC3)C3CC3)CCCCC1N(C(=O)Cn1cnnn1)CCC2 25831,Cc1nc(N(C)CC2CCCN2C(C2CCC3CC3CC2)=O)c(C)c(Cl)n1 25832,C1(C(N)=O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 25833,c1(C(N(C)CC2CC(F)CN2C(=O)C(F)=C2CCCC2)=O)cc(N)ccc1O 25834,c1(C(=O)NCCC2(C(=O)NCC3C(C)OCC3)CCCC2)ccc(C#N)cc1 25835,c1(C(C(N2CCC(CN(C(c3c(CC)ccs3)=O)CC)C2)=O)F)ccc(F)cc1 25836,C1(C(N2CC(NC(C(c3ccccn3)C)=O)CC2(C)C)=O)CCCCC1C1CC1 25837,c12coc(n1)NC2=O.C(C(CO)C(=O)OC(C)(C)C)NC(C1(COC)CC1)=O 25838,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 25839,CC(C)S(=O)(=O)C1CCN(C(CCCCC(C)(C)C)c2nnnn2CCSC)CC1 25840,C1(CCNC(C2CCN2C2CCCC2)=O)CSCCN1C(C1CCC(F)(F)C1)=O 25841,C1(NC(C2(C#C)CCN(C(c3nccc(C)c3N)=O)C2)=O)CC2C(O)C(O)CC12 25842,c1(C(=O)NC(c2ccccc2)C(=O)NC2COCC2O)coc2c1COC2 25843,c1(C2(C(=O)NCCCCN(C(C(c3ccc(C)o3)C)=O)C)CCC2)cccc(F)c1 25844,N1(C(C(C)O)=O)CCC2(CCN(C(=O)Cc3ccc4nc[nH]c4c3)C2)C1 25845,N1(C(C)Cc2nncn2C)CCCC2(CN(C(c3cccc4ncsc34)=O)C2)C1 25846,N1(C(CC(C)F)=O)CCC2CN(C(=O)Cc3scnc3-c3ccccc3)CCC12 25847,C(C)(C(=O)Nn1ccccc1=O)NC(C(CN(C)CC)C)=O 25848,C=CCCCCCCCC(=O)N(CC(CC)NC(c1ncc(OC)cn1)=O)C 25849,c1(C(N2CCC3CN(C(C(F)=CCC)=O)CC3C2)=O)n[nH]c2c1CC(C)OC2C 25850,C1(NC(CCCOC)=O)CN(C(=O)CC(O)C2CC2)CC1S(C)(=O)=O 25851,C(=O)(C(C)(C)C(F)F)NCC(C(=O)N(C(C(C)C)C(N)=O)C)C 25852,c1(N(CCN(C(C)C)C2CC2)C(C)C)cc(=NCc2ccc(O)nc2)[nH]cn1 25853,C1(C#N)(C(N(C(C(=O)Nc2ccc(SC)nc2)C)C)=O)CC(F)(F)C1 25854,c1(C(CN(C2CCC2)C(C2CCCC2)=O)=O)cnn(C)c1 25855,c1(C(N(CCCNCc2ccccc2)C)=O)ccc2cnn(C)c2c1 25856,C12(N(N3CCN(c4nnn(C(C)(C)C)n4)CC3)C)CC(C=O)(C1)OC21COC1 25857,N1(C(c2c(OCC)scc2)=O)CCN(Cc2ccc(C(C)(C)C)cc2)CC1 25858,c1(C(=O)NC2CN(C(C3C(C=C)OCCC3)=O)CC2O)cc(F)cc2nn[nH]c12 25859,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(CC)c(C)cc1)=O 25860,C=CC(CC(=O)NCCCCN(C(=O)COCC1(F)CC1)C)c1ccccc1 25861,N1(C(c2c(NC)ccc(F)c2)=O)CCC(CNC(=O)CC(C)C(F)F)C12CCC2 25862,c1(OC)ccc(C(F)F)cc1C(=O)NC(C)CNC(c1csc(=N)[nH]1)=O 25863,C1(NC(c2cnc(CC)o2)=O)CCCN(C(C2(c3ccno3)CC2)=O)CC1F 25864,Cc1nc(NC(C2CCCN2Cc2ccncc2O)=O)cnc1Cl 25865,C1(CC(=O)NCCCN(C(=O)CC2CCCC23CC3)C)CCC(C)(C)CO1 25866,N1(C(C(CCNC(Cc2nc(COC)on2)=O)O)=O)CC(O)CC12CCOC2 25867,N1(C(CC2(C)OCCO2)=O)CC2CC1CC2CNC(=O)C(c1ccccc1)O 25868,C1(CNC(CN(C(COC)=O)C)=O)CN(C(=O)CO)CC2(CC2)C1 25869,O=C(C#Cc1ccccc1)N1CC(F)(C(=O)Nc2cccc(C(F)(F)F)c2)C1 25870,N1(C(c2cc(C)on2)=O)CC(NC(=O)CN2CSCCSC2)CC12CCOCC2 25871,c1(C(=O)NCCCC(C)(C)NC(=O)CC2CCOCC2)ccc2nonc2c1 25872,c1(N2CC(C)C=C(C)C2)nc(N(C)CCc2ccccc2F)c2ccsc2n1 25873,C1(=O)CC(NC(N)=O)CN1.C=C1CC(C)C1.C1(=O)C(C)N1C.OC 25874,C(=O)(C(C)C(F)(F)F)N1CCC(CNC(c2n(C=C)ncc2)=O)CC1 25875,C(CN=c1[nH]c(=NC2CC2C(C)(C)C)c2ccccc2[nH]1)c1c(C)nc(C)s1 25876,N1(C(CCCCCNC(C(C(C)C)OC)=O)=O)CC=C(CO)CC1 25877,C1(C(=O)NCc2cc(C)oc2)CN(C(=O)CCCc2ccco2)CC1F 25878,c1(NCC(CCC)(F)F)ccc(Cl)cc1N1CCNCC1 25879,CN1CCCCC(C(N2CC=CC(NC(c3csc(C(F)(F)F)c3)=O)C2)=O)C1=O 25880,CCCC(CC)C(=O)N1CC(N(C(=O)C(C)C(=O)OC(C)(C)C)C)C1 25881,CCC(C)C(=O)NNC(=O)c1nn(-c2cccc(C)c2)cc1I 25882,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 25883,c1(CC(C(=O)NC(C)CN(C(=O)C(O)Cc2ccccc2)C)O)ccccc1Cl 25884,N1(C(C(C)OC)=O)CC2CCC1C(NC(C1CCCN1Cc1ccccn1)=O)C2 25885,C=CC1CCCN1C(=O)CNC(=O)CNC(=O)CN1CCCC1 25886,C(=O)(CCC(C)(C)C#N)NCC(C)(CC(C)C)NC(C(C)CF)=O 25887,N1(C(=O)NCCNC(c2cncs2)=O)CC2C(C(=O)NC3(O)CCCCC3)C2C1 25888,c1(NCC(C)NC(=O)C(C)S(N)(=O)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] 25889,c1(C(=O)NC2CN(C(C(C(=O)OC)(C)C)=O)C3C2C3)cc2c(Cl)nccc2s1 25890,Cc1cccnc1C(=O)NC1CC(NC(c2cncc(-c3ccncc3)c2)=O)C1 25891,c1(CC(C)C(=O)N(C)CCN(C(c2cnccn2)=O)C(C)C)ccccc1F 25892,C(=O)(C(CC(C)C)ONC(C1CC2(C1)CC(C)C2)=O)NC(CC)C1CCC1 25893,C1(SCC(=O)N(C2CCN(C(=O)C=C=C(C)C)C2)CCC)CCCCN1CC 25894,[N-]=[N+]=NC1CCCCC1C(=O)NCC1CC(F)(F)CN1C(=O)CC1C=CS(=O)(=O)C1 25895,CCCCCC(O)CC(=O)NCC1CC(NC(=O)C2=CCCC2(C)C)C1 25896,C1(C(=O)NCC2(NC(=O)Cc3ccccc3F)CC2)CC2C=CCC(C1)C2 25897,c1(C(N2C(CNC(c3ccco3)=O)CC3CC32)=O)cc2ccc(Cl)cn2c1 25898,c1(N2CCCC(CC)C2)nc(N2CCCC(C)(F)C2)nc2ccc(Cl)cc12 25899,C1(C(=O)NC2C(CC(C)(C)C)C2)CCCC(NC(C2(F)CC=CC2)=O)CC1 25900,c1(CC)ccc(F)cc1NC(=O)CCN(C(C12CCC(C1)C2)=O)CC1CC1 25901,CN1CC2CCC(C1)N2C(=O)CCC1CCCN1C(=O)C1=COCC1 25902,CC1=C(C(=O)N2CCC(N(C)C(C3CCC(N(C)C)C3)=O)C2)CCCO1 25903,N1(C(c2nn(-n3c(C)cc(C)n3)c(C)c2)=O)CCOC2CN(C(=O)CC#N)CC12 25904,c1(CC(=O)NCC(CC)(C)NC(c2ncoc2C)=O)cc(Br)ccc1F 25905,c1(C(=O)NCC(c2ccccc2)N(C(CCC#C)=O)CC)[nH]c(COC)nc1C 25906,C(=O)(CC(C)(C)CC)N1CCC(N(C(C2(NC(C)=O)CCCCC2)=O)CCO)C1 25907,c1(C(N2CCC(F)(CNC(c3c(CC)cccc3)=O)C2)=O)ncc(N)cc1Cl 25908,N1(C(C(=O)Nc2c(C)cnc(Cl)c2)=O)CCCC(C2OCCO2)CC1 25909,C1(n2cccn2)(CNC(C(C)N(C)C)=O)CCN(C(=O)C(F)=CCCF)CC1 25910,Cc1cc(-c2nccn2C(c2ccccc2)COc2ccccc2Cl)cc(C)c1 25911,N1(CC)CCOC(C(=O)NC2CCCC2NC(c2sccc2OCC)=O)C1 25912,c1(NCc2cnc(OC(C)C)c(Cl)c2)c(Br)cccc1C#N 25913,N1(c2nnc(C(C=C)O)n2Cc2cccs2)CCN(C(C)=O)C(CCOC)C1 25914,c1(C(C)(C)C)cc(CNC(=O)CN2CCCC(N(C)C)C2)cc(Br)c1 25915,N1(C(c2cncc(C)c2C)=O)CCCC(C2CC2NC(C2(N(C)C)CCC2)=O)C1 25916,N1(C(C(n2cc(-c3cccc4nsnc34)nn2)C)=O)C2CNC(=O)CC1COC2 25917,N1(C(C2CC(NC(C3(C)CCNC3=O)=O)C2)=O)CC(O)C(C2CC2)C1 25918,N1(C(C(C)Cc2ccncc2)=O)CC2(CC(NC(c3cncs3)=O)C2)C1 25919,N1(C(C(C)=C2CCCC2)=O)CCCCC(C(=O)NC(CO)C(C)C)C1 25920,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 25921,c1(OC(C)=O)cc(C)ccc1C(=O)NCC1CCN(C(=O)CC=CC(C)(C)C)C1 25922,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2ncc[nH]2)C1 25923,C1(CNC(C2(C(C)C)CC2)=O)CCC2(CN(C(=O)Cn3ccnn3)C2)O1 25924,C(=O)(C1CCc2c[nH]nc21)NC(C)CC1(NC(=O)C(C2CCCCC2)C)CCC1 25925,N1(C(CCC#CC)=O)CCCC(C(=O)NCC2CCOC2)CC1 25926,c1(C(=O)NC2C(NC(C=CC(C)C)=O)COC2)cc(C#N)n(C)n1 25927,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 25928,C1(CCC)CN(C(=O)C(C)Cn2cccn2)CCN1C(=O)C(F)F 25929,c1(C(=O)NCCCCN(C)C(C2CC2c2cccs2)=O)c[nH]nc1C(C)(F)F 25930,N1(C(c2cnc(C)o2)=O)CCCC2(NC(=O)C(C)N3CCC3)CC2C1 25931,c1(OCC)nc(C(N2CC(C(O)C(=O)NCc3nonc3C)C2)=O)co1 25932,N1(Cc2c(C)ccnn2)CCCC(Nc2ccccc2CC(=O)NC(C)C)CC1 25933,c1(CC(=O)NC2CN(C(C(C)OCC3CC3)=O)C(CO)C2)ccc(F)c(Cl)c1 25934,c1(-c2ccc(CC)cc2C)ccc2oc(C(=O)NC(CC)C(C)C)cc2c1 25935,c1(N(C)C)noc(CNC(=O)CONC(=O)CC2CCSC2)n1 25936,c1(NCc2cncc(OC)c2)ccc(S(=O)(=O)NCC2(C)CC(C)=NO2)cn1 25937,c1(CC)[nH]nc(C(=O)NCCC(C)N(C(=O)C(C)(Cl)Cl)C)c1Cl 25938,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2CCNC2=O)CC(O)C1 25939,C1(CCNC(CCC(=O)C2CC2)=O)CCCN(C(=O)COc2cccnc2)CC1 25940,c1(C(=O)NC(C(C(C)C)C)CNC(=O)C2=CCOCC2)c(F)ccc2occc12 25941,O=S(=O)(c1ccc(CNCc2cn3ccccc3n2)cc1Br)N1CCCC1(F)F 25942,CC(C)(C#N)CCC(=O)NC1CCSC12CN(C(c1cc(O)nc(C3CC3)n1)=O)C2 25943,C1(CC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)C=C(C)C 25944,c1(C(N2CC(C(=O)NC(c3cc(C)on3)C)OCC2)=O)cc(Cl)cnc1Cl 25945,C#CCC(C)(C(=O)N1CCC(CN(C)C)C1(C)C)NC(c1ccc(F)c(C)c1)=O 25946,C(=O)(C1=COCCO1)N(C)CC1CCN(c2cc(COC)ncn2)CC1 25947,N1(C(C)=O)CCC(NC(C2CCC(NC(C3(C)CC3)=O)C2)=O)CC1 25948,C1(C(=O)N(C(C)CO)C)(NC(c2cn(CC=C)nc2)=O)CCOCC1 25949,c1(OCC)c(F)ccc(F)c1CN1CCC1C(=O)NC(c1ccc(Cl)cc1)CO 25950,C1(C(N(C)C)=O)CC(C)(C)CN1C(C1CCOC1)=O 25951,c1(N2CCCC(NC(c3c(C)nns3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 25952,C1(OC)COCCC1N(C(C1CCCOCC1)C(N1CCOCC1)=O)C1CC1 25953,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 25954,N1(C(C2(N(C(C(C)N(C(C)=O)C)=O)C)CC2)=O)CCC(CO)C1(C)C 25955,C1(CN(C)C(c2ccc(F)s2)=O)CCN(C(C2(O)CCC2)=O)C1 25956,S(=O)(=O)(c1ccc2ccccc2c1)N(CC(c1ccn(C)n1)(C)C)C(=O)CCCl 25957,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)CCCNS(C)(=O)=O)CC)(C)C 25958,CCCCCCC(CC)C(=O)NCC1COCCN(c2nccn3nnnc23)C1 25959,C(N=c1[nH]c(=NC(CCO)c2cccnc2)[nH]c2ccccc12)C1(C)CCC1 25960,C1(C(C(=O)NCc2cnn(Cc3ccc(Cl)o3)c2)N(C)C)CCC(F)(F)CC1 25961,N1(C(=O)Cc2cnc(C3CC3)[nH]2)CCC2C(CCCN2C(c2ccoc2)=O)C1 25962,C(=O)(C1CCCc2ncc(C)n21)NCC1C(NC(Cc2ccc(OC)nc2)=O)C1 25963,CCS(=O)CC(=O)N(CC(=O)N(C)CCc1nccs1)C.C(CO)N 25964,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 25965,c1(NCC(C)N(C(=O)Cc2ccccc2OC)CC)nc(Cl)nc2[nH]ccc12 25966,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 25967,C1(NC(COCC(=O)NC)=O)CCC(F)(C(=O)Nc2csc(Cl)c2)C1 25968,C1(C(N(C)CC2(C#N)CC2)=O)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C2(CCC2)C1 25969,C1(CC(=O)N(C(C)C(C)(C)O)C)N(C(c2ccncc2Cl)=O)CCC1(C)C 25970,c1(OCCC(=O)NCCC2CCCN(C(c3ccsn3)=O)C2)ccc(Cl)cc1 25971,C1(C(=O)NCC2N(C(CC3(CC)CCC3)=O)CC(F)C2)CC1C1CCCC1 25972,N1(C(c2cncc(C)c2C)=O)CC2CC(NC(=O)C(C)(C)CC(C)C)CC2C1 25973,N1(C(C(C)Cc2cnc[nH]2)=O)CCCCC1CCNC(=O)Cc1cnc[nH]1 25974,C(CC(CNC(C1(Br)CC1)=O)NC(=O)C(O)CN(C)C)OC 25975,N1(c2ccsn2)CCC(n2nc(C3CSC3)nc2C)CC1.CC(C)(C)O 25976,C1(C(=O)NC)CCCCN1C(c1ccc(-c2cnn(C)c2C)o1)C(=O)NC(C)C 25977,C12CC(=NO1)C(=O)NC2.N1(C(CCOCCOC)=O)CCC(C2(C)N=N2)C1 25978,C1(CC(=O)NC2CC2NC(c2cncc(CO)c2)=O)CN2CCN1CC2 25979,[N-]=[N+]=NC1(C(=O)NCCCc2ccsc2)CCN(C(C2CCOC2)=O)C1 25980,S(=O)(=O)(CCC(F)(F)F)N(C1CN(C(C2CC2(F)F)=O)CC1F)C 25981,c1(OC)ccccc1NC(=O)C(F)CC1CN(C(=O)CN2CCOCC2)C1 25982,C(CCCCCN=C(NCC(C1(O)CCOCC1)(F)F)N1CCCC(C)(C)C1)SC 25983,C1(OC)(OC)CCC(c2nnnn2N(C(C)CC(C)C)c2ccco2)C1.C1CO1 25984,N1(C(CC2(C)CCN2C(=O)CC2CC(F)(F)C2)=O)CCOC(C)(C(F)(F)F)C1 25985,C1(C(=O)NCc2cn(CC=C)nn2)C2CCC(C2)C1NC(C1(SC)CCC1)=O 25986,N#Cc1cc(NC(c2cc(Cl)cn2-c2ccccc2)=O)c(Br)cc1F 25987,N1(C(CC2C(CNC(c3ncc(CC)cn3)=O)C2)=O)CCNC(=O)C1C(C)C 25988,C1(NC(CCCOC2C(C)CCCC2)=O)CCN(C(=O)CCF)CC1O 25989,C1(NC(C(C(CC)C)C)=O)CCC2(CC1)CN(C(=O)C=CC1CCOC1)CCO2 25990,C(CC(C)NC(=O)CCn1cccn1)N(C(CN(S(C)(=O)=O)C)=O)C 25991,C(CC(C(=O)NCc1ncsc1C)NC(=O)C(COC)CC)=CC 25992,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 25993,c1(CCC(C)N(C2CS(=O)(=O)C2)C(=O)C(O)C2CCCC2)cccc(F)c1 25994,CC(N=c1cc(N(C)C)nc(CNc2cocn2)[nH]1)C(F)F 25995,C1(NC(CCOCCC)=O)CC2(CCN(C(c3nc(C)ccc3F)=O)C2)C1 25996,Cc1cccc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CCCC2)c1O 25997,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1C1CC1 25998,c1(C(=O)NCCC(C)N(C(c2nccc(C#C)c2)=O)C)ccc2nnc(O)n2c1 25999,C1(NC(C2CC(=C)C2)=O)CCCCC1CNC(=O)CCc1cn[nH]c1 26000,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26001,c1(CN(C(c2cscc2C)C(=O)NCCCC)C)cccc(OCC#N)c1 26002,C1(COC)CC(C(=O)OC)CN(C(=O)NCc2[nH]nnc2-c2ccccc2)C1 26003,CCC(C)CCC(=O)NCCOC1CN(C(=O)CCCc2ccc(C)s2)C1 26004,c1(CNC(C(CC2CN(C(c3c(C)ocn3)=O)C2)F)=O)cc2cc(Cl)cnc2[nH]1 26005,N1(C(Cc2n[nH]c(=NC)s2)=O)CC(NC(=O)C=CC=C(Cl)Cl)CC(C)(C)C1 26006,c1(C(=O)NC2CCCN(C(COc3cc(C)on3)=O)C2)c(Cl)c([N+](=O)[O-])nn1C 26007,CCC(CCC(=O)N(CC(C1CCC1)OC)C)NC(c1ccc(F)c(O)c1)=O 26008,C1(C)(C(NOCc2cn(C(C3CCCC3)CC)nn2)=O)CNC(=O)N1 26009,C1(NC(C(CC)(F)F)=O)(CNC(c2ccnn2COC)=O)CCCCC1C 26010,c1(CC)c(C(=O)NC(C2CCOC2)CNC(=O)CN2CCCC2=O)cccc1F 26011,c1(OC)cccc2nc(C(=O)Nc3cc(F)c(Cl)cc3Cl)n(C)c12 26012,N1(C(C2C(NC(c3ccccc3)=O)CCCC2)=O)C2CCC1CC(O)C2 26013,c1(N2C(CNC(C(c3ccc(OC)cc3)OC)=O)CC2)nc(Cl)c(C#N)s1 26014,C1(C(=O)NC(C(C)C)CO)CCN(C(c2ccc(=O)n(C)c2)=O)C1(C)C 26015,C1(C(=O)NCC(=O)NCCC(C)N(C)CC2CC2)CCN(C(=O)OC(C)(C)C)C1 26016,C1(NC(=O)COC)CCN(C(C2CCCO2)=O)C1.C1CC(n2ccnc2)C1 26017,c1(C(=O)NCC(CC)(CC)OC)ccc(C(C23COCC2C3(F)F)=O)nc1OC 26018,NS(=O)(=O)CCC(=O)NCCC1(CNC(=O)CC2CCC(O)C2)CC1 26019,C1(C)(CNC(c2ccc(C(C)(F)F)cc2)=O)CCC(NC(C2CCC3CC23)=O)CC1 26020,c1(C(=O)NCC2OCCN(C(c3c(C)ncnc3C)=O)C2)ccc(F)c(F)c1C 26021,CC1CCN(C(C2(F)CCN(C(=O)CCN3CCCC3)CC2)=O)CC1O 26022,C(C1CN(C(c2coc(C(F)F)c2)=O)CC1C(=O)N(C)CC1CCSC1)=CC 26023,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26024,C(=O)(C(CO)C(C)(C)C)N1CCC(CC=C)(NC(c2coc(CC)n2)=O)C1 26025,C(=O)(CS(=O)(=O)C1CC1)NCCCC1N(C(C2C(C)(Br)C2)=O)CCSC1 26026,c1(OC)ccc(C(=O)NC(CNC(C2(F)CCCOC2)=O)CO)cc1S(N)(=O)=O 26027,N1(C(C2CC(CC)C2)=O)CC2(C1)C(NC(=O)C(CC)C(C)C)CCS2(=O)=O 26028,Cc1nc2c(C(=O)NC3COCC3N3CCCC3)cccn2c1Br 26029,CON1CCC(C(N2CC(C(=O)NCCOCC(F)F)C(C=CO)C2)=O)CC1 26030,C12C=CC(C1)OC(=O)C2.C(=O)(CC(Cl)Cl)N.O=C1CCC2CC(C2)N1 26031,c1(OC)cc(OC)cc(C2CCC2c2nc(-c3cnccn3)nn2CCCO)c1 26032,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26033,Cc1sc(Cl)nc1C(=O)NCC1CC1CNC(C1CCN(C(C)C)CC1)=O 26034,N1(C(C(C)OCCC2CC2)=O)CCN(c2ccc([N+](=O)[O-])cc2F)CC(C)(F)C1 26035,C1(CCNC(c2c(CC)cc[nH]2)=O)CN(C(=O)CCCNC(=O)C2CC2)CCCO1 26036,C(=O)(CC1=NNC(=O)C1)NC1C(CCC)CN(C(c2ccn(C(F)(F)F)n2)=O)C1 26037,c1(C(N(CC(C)NC(=O)C(C)(O)Cn2ccccc2=O)C)=O)nnn2ccccc12 26038,N=c1ncc(C(=O)NCC2(COC)CCCN2C(=O)CCC2CCCCO2)c[nH]1 26039,C(CN(C1(OCC#C)CCOCC1)C(=O)CC(=O)NC)(C(C)C(C)C)N(C)C 26040,N1(C(c2c(C)noc2)=O)CC2(C=C(C(=O)NCCc3nnc(O)o3)CO2)C1 26041,Cc1cc(C)n(CC(=O)N(C)CC2CCN(C(=O)CC3CSC3)C2)n1 26042,C(C#N)(C(=O)C(C)(C)C)c1cccc(NC(N2CC(C3C(OC)C3)C2)=O)c1 26043,c1(OC)cc(C(=O)NC23CCC(CN(C(C4CC4(F)F)=O)C2)C3)sc1S(N)=O 26044,N1(C(C=CC(CC)=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26045,Cc1nsc(Cl)c1C(=O)NCCCCCNC(=O)C(C)(C)c1cscc1Cl 26046,N1(C(COC)=O)CC(C(F)(F)F)OCC1CNC(=O)CCSCCCC 26047,c1(N2CC(CCNC(=O)CC(O)C3CC3)(OCC)C2)ccnc(CC)n1 26048,S(=O)(=O)(c1cn(C)nn1)N(CC(=O)Nc1cccc(C)c1)C 26049,c1(C(=O)NCC(C)NC(=O)COc2ccc(F)cc2)cnc(Cl)cn1 26050,C(CO)(CCCCNC(c1ccncc1O)=O)NC(C1(O)C(C)(C)C1)=O 26051,c1(C(=O)NC2C(CO)CCN(C(CC=CCC)=O)C2)ccc2nccc(C)c2c1 26052,c1(CNc2c(CNC(=O)CC(O)c3ccccc3)nccc2)cc(Cl)ccc1Br 26053,C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CN(C(=O)CCN3CCOC3=O)CC12 26054,C(CC(C(C)C)NC(c1c(C(C)C)cnn1C)=O)N(C(C(C)=C1CCC1)=O)C 26055,c1(C(N2CC(CNC(c3c(CC)csc3)=O)OCC2)=O)cccc(C)c1N 26056,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26057,N=c1[nH]c(CCC(=O)NC2(C3CCCO3)CCC2)cs1.C1(=O)C(=O)NCCN1 26058,Cc1cc(CC(=O)NCC(n2cc(CCCCO)nn2)C)ccn1 26059,C1(C(=O)NCC2N(CC)CC2)C=CCN(C(=O)CN2CC(=O)NC2=O)C1 26060,CCCC(C(=O)N(C(C)C(=O)NCC(C)(CC)CC)C1CC1)N(C)C 26061,N12CCc3ccc(cc3C1)CNC(=O)C2.Cc1ncnc(C)c1Br 26062,n1(CC(=O)NC2CN(C(C(F)=CC)=O)C(C)CC2)ccc2ccc(F)cc12 26063,c1(COCC(=O)N(CCC)CCNC(C2CCCC(=O)O2)=O)cc(F)cc(F)c1 26064,N1(C(C2C(C)(C)CCC2)=O)CC(NC(=O)CCc2cccc(F)c2F)C(C)(C)C1 26065,C1(CCNC(C(C)(C)SC)=O)CN(C(=O)Cc2nnc(O)s2)CC(C)O1 26066,c1(CSCC(=O)NCC(C)N(C)C(C2COCCO2)=O)ccccn1 26067,CC(CC(N)=O)C(=O)NC1CC(NC(c2cc(C3CC3)nn2-c2ccccc2)=O)C1 26068,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26069,c1(CC(N2CC(NC(c3cccc(F)c3O)=O)(CO)C2)=O)nc2ncccn2n1 26070,N1(C(CCC#C)=O)CC(CCNC(C2CN(C3COC3)C2)=O)OC(C)C1 26071,Cc1cc2c(cc1C)C(C(=O)N1CCCC1CNC(c1cnc(N)s1)=O)CO2 26072,N1(C(C=C(C)c2ccco2)=O)CCN(C(=O)CCOCC2CCC2)CC1C1CC1 26073,Cc1cccc(C)c1-n1cc(CC(N2CC(CC3CC4(CCC4)CO3)C2)=O)nn1 26074,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26075,CC1(C)CC2(CC(C(N3CCN(C(C4CCCOCC4)=O)CC3)=O)C2)C1 26076,CC(C)C(CN(C)C)C(=O)N1CCOCC(NC(=O)CC(Cl)Cl)C1 26077,c1(C(N2CC3C(CNC(=O)CCC4CC4)(C3)C2)=O)cccc2cccc(O)c12 26078,c1(C(=O)NC2(C#N)CC(O)(C(F)F)C2)c(F)ccc2c1OCO2 26079,c1(NC(CC)CSC)ccccc1OC.c1(C2c3nnnn32)ccc(C)o1 26080,Cn1cc(C(=O)NCc2cocn2)c2cc(-c3ccc(O)c(CO)c3)ccc12 26081,C(=O)(CC(O)CC(C)(C)C)OC.C1(=O)CC(COC)COc2cccc(c2)N1CC 26082,c1(C(=O)NC(CCCNC(CSCC#C)=O)C)ccc(Cl)c(Cl)c1C 26083,C1(NC(C2(C)CC(=C)C2)=O)CCC(F)(CNC(=O)CNC(C2CCCC2)=O)C1 26084,CC(C)C(F)(F)CC(=O)N1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1 26085,c1(OC)cc(C=CC(N2CCCC2C(C)NC(c2cocc2C)=O)=O)ccc1N 26086,Cc1cc(C(=O)NC2CCN(c3nc(Cl)ncc3C3CC3)CC2F)c2[nH]cnc2c1 26087,C1(OCC(=O)NC2CCCC(NC(C3(C)CSC3)=O)C2)C#CCCCCC1 26088,C1(C(N(CCCNC(c2ccc(CC(C)C)s2)=O)C(C)C)=O)CCCCCCC1 26089,c1(CC(=O)NC(C(=O)OC)CC2(O)CCOCC2)cn(C)c2ccccc12 26090,N1(C(C2C(C(C)NC(C3CC3C3CCOCC3)=O)C2)=O)CC2CCCC(C1)N2C 26091,c1(NC(C2N(C(c3ncn(C)c3)=O)C3CCC2C3)=O)cncc([N+](=O)[O-])c1 26092,C1(C(N(CCCC=C)C)=O)CCC2(CCN(C(C3CCC4(CC3)CC4)=O)CC2)O1 26093,c1(OCCCNC(=O)CCNC2CCOCC2)cnn2cc(Br)ccc12 26094,N1(C(c2n(CCC)ccc2)=O)CC2C(CNC(c3ccc(Br)o3)=O)C2C1 26095,c1(OC)cc(C)c(C(=O)NCC2(F)CCN(C(C3COC(C)(C)C3)=O)C2)cn1 26096,C1(NC(c2c(CC)cccc2)=O)CN(C(=O)C(O)Cn2cncn2)CC12CCC2 26097,C1(NC(c2c(C)nc(C(C)C)s2)=O)(CNC(=O)COC(F)(F)F)CCCCC1C 26098,C=CCC(CC=C)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)CC2)CC1C 26099,Cn1nnc2cc(C(=O)NC3CN(C(C4CC4F)=O)CC3C(F)(F)F)ccc12 26100,C1(NCCC(N2CC(N(C)C(C3(C(F)F)CCC3)=O)C2)=O)CCCOC1 26101,c1(OC)ccc(C(C)NCC(=O)N(C)Cc2ccccn2)nn1 26102,c1(NC(C2CC(CNC(CCOCCC)=O)C2)=O)nccnc1CC 26103,c1(C(=O)NC2CCC23CCNCC3)nn(CCO)c(=O)c2ccccc12 26104,C(=O)(C1=C(Cl)CC1)N(C(C(N1CC(O)(CC=C)C1)=O)CC)C1CC1 26105,N1(C(CCn2ncc(C(=O)OC)c2)=O)CC(N(C(=O)CC2(C)CC2)C)C(O)C1 26106,C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(=O)COCCOC 26107,c1(CNCCCCC(=C)C)cnn2ccc(OC)cc12 26108,CC1(C)CN(C(=O)CC2(C(F)(F)F)CCC2)CC1NC(c1ccccc1F)=O 26109,N1(C(c2ccc(Cl)cc2Br)=O)CCC2(CCN(S(=O)(=O)c3cccc(F)c3)C2)C1 26110,c1(OC(c2nc(CF)nn2-c2c(C)noc2C)CC)cc(F)cc(F)c1 26111,c1(C(=O)NC2CN(C(C3(C#C)CC3)=O)CC2C(F)F)cnn2ccsc12 26112,C(=O)(CCCC1CCCCC1)NCC(CC)NC(COCCOCC#C)=O 26113,C(C1CCOCC1)=CC(=O)NC1CC(n2cc(C(C3CC3)OC)nn2)C1 26114,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)O)C)C1)=O 26115,c1(C(C(=O)NC2CCC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)O)cccc(Cl)c1 26116,C1(CNC(c2nncc(C)c2)=O)CCN(C(c2cc(CC(C)C)on2)=O)C(C)C1 26117,c1(CCNC(C2N(C(C#C)=O)CC2)=O)ccc(Cl)c(Cl)c1 26118,Cc1cc(N(C)C)cc(C)c1CC(=O)NC(=O)CC#N.N1(C(C)=O)CCC(=CCN)CC1 26119,N1(C(=O)COc2ccccc2)CC2(CC(NC(C3CC(n4ccnn4)C3)=O)C2)C1 26120,N1(C(CC(C=C)C)=O)CC(C2CCCN(C(=O)COc3cccc(OC)c3)C2)C1 26121,C1(C(=O)NC(CCOC)COC)CN(C(C2CCS2(=O)=O)=O)CC1(C)C 26122,Cc1ncnc(C)c1C(=O)NCc1cc(C(=O)NCCC2CCCC2)cs1 26123,O=C1Cc2c(C(N3CC4(CC4)CC3CNC(=O)C(O)C3CCC3)=O)cccc2N1 26124,C1(NC(CCOCC)=O)CCN(C(CC2CC(OCC(C)C)C2)=O)CC1C(N)=O 26125,c1(C(N(CCCNC(CC(CCC)C)=O)CCO)=O)csc(=NC2CC2)[nH]1 26126,c1(C(C)NC(=O)NCC(C)(C)CSCCO)ccc(Cl)cc1F 26127,C(=O)(N1CC(O)CCO1)C1CCCN(C(c2ccnn2C(F)F)=O)CC1 26128,C(C1(C)CCOCC1)=CC(=O)NCC(CNC(CCN(CC(C(C)C)C)C)=O)O 26129,c1(CC(=O)OC(N2CC(CC=CCNC(C(C)SC(F)(F)F)=O)C2)=O)cn(C)nn1 26130,CCC(CC)(CO)C(=O)NC1CC(CC(=O)NCc2ccccc2OC)C1(C)C 26131,n1(CCC)cc(C(=O)N(CCCNC(=O)CNC(=O)NC)C(C)C)cn1 26132,Cc1sc(C(=O)NC2CCC(C)(CNC(=O)Cc3cn(C)cn3)C2)nc1O 26133,N1(C(=O)Cc2ccc(Cl)s2)CC2CC(C1)CN(C(C1CCCC1)=O)C2 26134,c1(OCCOC(CCC(c2ccc(C)cc2)O)=O)cc(C)ccc1F 26135,C1(CNC(C=CC(C)(C)NC(c2cn(CC=C)nn2)=O)=O)CCCCCCC1 26136,N1(C(C2COCC2C(F)F)=O)CCN(C(c2ccco2)=O)C(CO)C1 26137,N1(C(C2(CC3CCC3)CC2)=O)CC2(C1)SCCC2NC(C1CCCO1)=O 26138,c1(C(=O)NC(CCC)CO)ccc(OC(=O)CCCN2CCOC2=O)cc1 26139,c1(C(N2CCC3CCN(C(=O)C(F)C4CCC4)CC23)=O)cc2cc(F)ccc2o1 26140,c1(C(=O)NC2C3(NC(c4cc(C)nn4C)=O)CCC(C2)C3)cccc2[nH]ncc12 26141,CCCCCC(O)CC(=O)N1CCN(C(c2sccc2F)=O)CC1CCC 26142,Cc1cnc(C(N2CCOC(CNC(=O)C=CC(C)C)C2)=O)nc1 26143,c1(CN=C(NCc2cc(C)on2)NC2CC2c2ccnn2C)cn(C)c(=O)nc1O 26144,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26145,c1(C(C)=O)ccc2nnn(CC(F)(F)F)c2c1.N1(C(C)=O)CCCC1c1cnn(C)c1 26146,c1(C(=O)NC2C(NC(c3c(C)cc(O)cc3)=O)C2)[nH]c2cc(F)cc(F)c2c1C 26147,C(C1=CCN(C(C2(C)CCN(C(=O)CCNC(C)=O)CC2)=O)CC1)OC 26148,C(=O)(CCC(C)SC(C)C)N(CC(CNC(CSCCC(C)C)=O)(C)C)C 26149,C1(NC(C2(C(C3CCNC3=O)=O)CC(COC)C2)=O)CC2(C1)CC(N)C2 26150,CCCCC(CC)CCCC(=O)N1CC(N(C(=O)CNC(c2cnoc2)=O)C)C1 26151,N1(c2nc(C#N)cc(C)n2)CCC(C2CCN(C(c3ccc(O)nn3)=O)CC2)C1 26152,C(=O)(CCC(=O)NCC)NCC1(NC(CC=CC)=O)CCC1 26153,N1(C(C(CSC)N(C)C)=O)CCCN(CCO)CC1.C(=O)C(C)OCC1CC1 26154,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(N2CC(c3nncn3C)C2)=O)C1 26155,C(C(C)(CNC(c1cnc(CC(C)C)[nH]1)=O)OC)NC(C(C)OCC)=O 26156,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26157,c1(C(N2C(CNC(=O)CCC3CCCCC3)C=CC2)=O)ccn2ccnc2n1 26158,N1(C(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C1 26159,N1(C(c2c(CC)n(C)nc2)=O)CCC2CCN(C(=O)C(n3cc(Cl)cn3)C)CC12 26160,CCCCC(C)C(=O)NCCCC(O)C(=O)NCCCC(=O)NO 26161,N1(C(C(C)(F)F)=O)CCC2CC(NC(=O)CC3(C(F)(F)F)CC3)CCC2C1 26162,c1(NC(N2CCC(O)(C(=O)Nc3ncc(C)s3)C2)=O)c(O)cccc1[N+](=O)[O-] 26163,n1(CCOC)ccc(C(N2CCC(N(CCOC)C(C3CCCC3C)=O)C2)=O)n1 26164,CNS(=O)(=O)NCCCNC(C1(CC2COCC2n2cc(OC)nn2)CCC1)=O 26165,C(CC(CC)C(=O)NC(COC)C(=O)NCCCN(C)C1CC1)=CC 26166,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C(C)C2CC2)CCC12CCOCC2 26167,C1(F)(C(=O)NCC(CC=C)NC(C2CC23CC(=C)C3)=O)CCCCCC1 26168,CC1(C)CCN(C(C2CCO2)=O)C1CC(=O)NCCCCCCO 26169,C1(NC(C(C)(C)N(C2CC3CC2C2CC32)C)=O)CC2CCC1N2C(=O)OC(C)(C)C 26170,c1(C(N(CCN(C(=O)CCc2ccnc(Br)c2)C)C)=O)ccccc1C#N 26171,C1(C)(C(=O)Nc2cccc(C(=O)OC)c2)CN(Cc2cc(C#N)n(C)n2)CCO1 26172,c1(C(=O)NCC(CN(C(COCCCC)=O)C)C)ccc(F)c(C(F)(F)F)c1 26173,CCC(C)(C)CC(=O)N1CCCC(C(C)(O)CNC(c2cc(CO)oc2C)=O)C1 26174,C1(C(=O)NC(C2(O)CN(C(C(CC)C(C)C)=O)C2)C)CCC2(CCCCC2)CC1 26175,Cc1c(CCC(=O)NC2CCCNOC2)cccc1Br 26176,C1(NC(C2CC(NC(C(NOC)=O)=O)C2)=O)CC2CCCC2C1 26177,C1(C(N2CCC(C)C2CNC(c2ccoc2)=O)=O)CCCNS1(=O)=O 26178,Cc1ccc(C)c(C(=O)NCC2OCCC2C(=O)NCc2nn(C)c(=O)o2)c1 26179,c1(C(=O)NC2C=CC(CNC(c3cn(C(C)C)nc3)=O)C2)ccc(C#N)cc1 26180,N=c1[nH]cc(C(=O)NCC2CC(F)(CNC(C3(C(F)F)CCC3)=O)C2)o1 26181,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC(O)CNC(C1(O)CCSC1)=O 26182,Cc1ccc(N)c(C)c1C(N1CC2CCCC2(NC(C2CCC(O)CC2)=O)C1)=O 26183,C1(C(=O)NC2(CNC(c3ccc(CC)cn3)=O)CCCC2)CCCC(N=[N+]=[N-])C1 26184,c1(C(=O)NCCC2CC(OC)CN2C(=O)CC(C)SC)ccc2ccsc2c1 26185,N1(C(C(CCC)O)=O)CC2(CCN(C(=O)CCc3cnoc3)CC2)CC1C 26186,c1(NC(c2cc(I)ccc2C(F)(F)F)=O)cc(F)c(Cl)cc1Cl 26187,C1(CC(N2CCC(NC(c3ccc(COC)cc3)=O)C2C)=O)CC(C)CC(C)(C)C1 26188,c1(CC(=O)NCC(C)(C2CCC2)NC(C(C)OCC)=O)ccc([N+](=O)[O-])c(N)c1 26189,C=CC(CC)CC(=O)NCC(C)(CO)NC(c1ccnc(C(F)F)c1)=O 26190,N1(C(C(=O)NC(CC)C(C2CC2)SCC)=O)CC2(C(=O)O)CC2(C(F)(F)F)C1 26191,CCCCC(O)C(=O)N1CC(NC(c2nccc(O)n2)=O)C(CO)C1 26192,N1(C(C(n2c(C)cc(C)n2)C)=O)CC2CCC(C1)N2Cc1cccc(O)c1O 26193,Cc1ccc(F)cc1C(=O)NCC(CNC(C1CC2(CSC2)C1)=O)CO 26194,N1(C(Cc2n(C)nnc2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C1(C)C 26195,C1(CNC(C=CCCC)=O)CC2CC(C1)N(C(=O)CCc1cccnc1)C2 26196,CC(C)(CCCNC(=O)CNC(C1CCC1)=O)NC(c1sccc1C(F)F)=O 26197,c1(C(N(CCC)CCNC(=O)CCSc2ccc(Cl)cc2)=O)cccc(F)c1 26198,Nc1c(C(=O)NC2CC(NC(C3(CN4CCCC4)CCCC3)=O)C2)ccc(Cl)c1Cl 26199,c1(C(N2CCc3c(F)cccc3C2)=O)cnc2ncnn2c1O 26200,C1(OC)CCC(C(=O)NC2CC2CNC(=O)CCc2cccs2)C1 26201,c1(CC)cc(C(=O)NCC(O)C(=O)NC(C(=O)OC)C2(C)CC2)no1 26202,C(=O)(CC1COCc2ccccc21)N1CCC(CNC(C(C)=C2CC2)=O)C1(C)C 26203,CCCCCCCC(=O)N1CCC(CCNC(c2ccncc2CC)=O)CC1 26204,c1(NC(=O)Nc2c(C)scn2)cccc(CNC(C2CCCS2)=O)c1 26205,c1(C(=O)NCC(CC)(C)NC(=O)C(C)C)cc(F)cc(Br)c1 26206,N1(C(C2C(C(N)=O)C2)=O)CC2(NC(C3CC4CCC(C3)C4F)=O)CCC1CC2 26207,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CN(Cc1cncn1C)CC2C(=O)O 26208,C1(N(C(C(C2CCCC2)OCC)=O)CC(=O)NCCOC)COCCO1 26209,c1(CC)nn[nH]c1C(=O)NCC(O)C(=O)N1CCC(c2ncc[nH]2)C1 26210,CC#CCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C)=C1CCCC1 26211,C1(c2n(CCCOC)nnn2)(NS(C)(=O)=O)CCN(Cc2c(C)cnn2C)C1 26212,C1(NC(CCN(CCC)C)=O)CCCN(C(=O)CCCSC)C1 26213,c1(C(C)C)ccc(C(N2CCC(F)(CNC(c3cnco3)=O)CC2)=O)c(O)c1 26214,c1(C(=O)NCC(CNC(CC2N(C)CC=CC2)=O)O)cc(=NS(C)(=O)=O)cc[nH]1 26215,c1(CN2CCC(F)(C(N(CCC(C)C)CCC#N)=O)C2)ccc2ncccc2c1 26216,C1(NC(CCC2(CCC#C)N=N2)=O)CCC12CN(C(C1(N3CCCC3)CCC1)=O)C2 26217,c1(C(=O)NCC23CCC(NC(C(C)CO)=O)(C2)CO3)cc(F)c(F)c(F)c1F 26218,C12(CNC(C(C=C)O)=O)CN(C(c3ccccc3)=O)CC1CCO2 26219,C1(NC(c2c(C)noc2)=O)CCN(C(=O)CCc2ccccn2)CCC1CO 26220,S(=O)(=O)(c1ccccc1N1CCN(C(c2cc(O)cc(=O)o2)=O)CC1)NC(=N)N 26221,C(=O)(C1CCCc2ccnn21)NC1CCN(C(C(C)CF)=O)C1C 26222,c1(OC)cc(C(=O)NC2CC(C)N(C(C3CCC3)=O)C2)sc1Cl 26223,C(=O)(C(CC)CCNC(=O)C1CC1)N1CC(C(C)N(C)C)C1.C12(CC1)C(=O)N2 26224,c1(C(N2C(C3(NC(C=CC=CC)=O)CC3)CCCC2)=O)cccc2ncc(C)n12 26225,Cc1onc(C(F)(F)F)c1C(N1CCC(CNC(=O)CN2CCCC2=O)C1)=O 26226,c1(C(N2CC(C3(NC(C(C)NC(COC)=O)=O)CC3)C2)=O)nc(N(C)C)nc(=N)[nH]1 26227,c1(OC)cc(F)c(C(=O)NC(C)(C)CNC(C2CNC(=O)C2)=O)c(F)c1 26228,c1(C(=O)NCC2N(C(C(C)Cc3ccnn3C)=O)CC2)cccnc1OCCO 26229,CC(C)C(F)(CNC(=O)CCS(C)(=O)=O)C(=O)N1CCOC(C2(C)CC2)C1 26230,c1(CCC)nc(CNC(=O)C(c2ccco2)NC(=O)CC2(C(=O)OC)CCC2)no1 26231,C#Cc1ccc(CC(N2CCN(C(c3cccnn3)=O)C(CO)C2)=O)cc1 26232,N1(CC)CCCC(C(N2C(C(N3CC(n4cnnc4)C3)=O)CC2C)=O)C1 26233,C1(NC(C2(N(C)C)CC2)=O)C2CC1N(C(c1ccc(OC(F)(F)F)cc1)=O)C2C 26234,Cc1csc2ncc(C(=O)N(CCC(C)NC(C3CCC(F)(F)C3)=O)C)c(=O)n12 26235,c1(NC=O)ncnc2[nH]cc(C)c12.c1(SCC)ccc(NC2(C)CC2)cc1F 26236,C1(C(=O)OC)CC(C)N1C(c1cnc(C2CC2)o1)=O.c12csnc1NC2=O 26237,c1(C(=O)OCC)ccc2c(c1)C(=O)NCC2NC(N1CCCCC12CCC2)=O 26238,c1(CC)cc(C(N2CCOCC2CCNC(=O)CC2C=CCCC2)=O)cc(O)n1 26239,c1(SC)ccccc1C(=O)NCC(O)CNC(=O)C(C)=O 26240,C1(NC(CNC=O)=O)CN(C(c2cncc(CO)c2)=O)CC1C(F)F 26241,C1(CC)CCN(C(C2CCC2C(N)=O)=O)C1C(=O)NCCCC1(C)CC1 26242,c1(CC(=O)NCC(CN(C(C2C(CC)CCC2)=O)C)C)ccc2ccccc2c1 26243,C(C(O)CC(=O)NCc1cccc(C)c1)NC(COCCC#C)=O 26244,C1(C(=O)NCC(CC)NC(C2CCCCCCC2)=O)OC2CCC1CC2 26245,C1(N(C(c2coc(Br)c2)=O)CC)CCN(C(c2sccc2CO)=O)CC1 26246,c1(C(=O)NCCC2CCC(NC(c3cc(OC)n(C)n3)=O)C2)cn2ccsc2n1 26247,C(=O)(C(C)(C)CC=C)N1CCC(N(C(CC=C)=O)C)CC1 26248,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26249,C12(CC(=O)NC(C)CNC(C3COC(=O)N3C)=O)CC3CC(C)(C1)CC(C)(C3)C2 26250,C1(NC(C(CC=C)C)=O)CCN(C(c2ncc[nH]2)=O)CC1C 26251,c1(OC)ccc(C(=O)N(CCOCCCNC(=O)C#CC(C)C)C2CC2)cc1N 26252,c1(CC(N2CCN(C(C(C(=O)OC)C)=O)C(CCO)C2)=O)c[nH]c2cnccc12 26253,c1(C(C)(C)NC(c2n(C)nnn2)c2cnoc2C(C)C)nn(C)cc1I 26254,c1(NC(c2cc(C(C)C)no2)=O)c(C)cc(NC(=O)C(C)(C)CCl)cc1C 26255,Cc1nn(C(C)C(=O)NC(c2nc(C(C)(C)C)no2)C)c(C)c1Br 26256,C1(NC(CC2(OC)CC2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CCC1(F)F 26257,C(CCS(=O)(=O)C1(NC(CNCC2C=CC(NC(=O)C=C(C)C)C2)=O)CC1)OC 26258,c1(CC(=O)OCC)ccccc1NC(=O)C(Cc1ccoc1)NC(=O)CC 26259,C1(OC)CCCC1CC(=O)NCc1ncoc1CNC(c1sccc1C1CC1)=O 26260,c1(OC(C(=O)N2CC(CCCCSCC)C2)(F)F)ccc(NC)cc1 26261,C(CCCCCC(=O)NCC(CC)N(C)C(C)=O)N(C(CC(C=C)(C)O)=O)C 26262,C1(NC(c2c(COC)noc2)=O)CCCCN(C(=O)C(C)CSC)C1 26263,CC1CC(NC(=O)C=Cc2ccc(Br)s2)CN(C(=O)C(CO)NC(N)=O)C1 26264,CCCCCC(O)CC(=O)NC1CC1CNC(=O)CCNc1cccnc1 26265,N1(C(C2C(C(=O)OC)C2)=O)CCC(C2CCN(C(=O)C(C)(C)SC)C2)CC1 26266,c1(N(C)C)ncc(S(=O)(=O)NC(c2cc(C#N)ccn2)=O)s1 26267,CCC(F)(F)C(=O)NC(C)CN1CCN(C(=O)CS(=O)(=O)NC)CC1 26268,N(C(=NCc1ccc(Cl)c(OC)c1)N1CCC2=C(COC2=O)C1)C(COC)C 26269,C=CCCCCCC(C(=O)N(CC(C)CC)Cc1ccccc1)NC(C)=O 26270,CCCC(C(O)C(=O)NC1(C)CC(F)C1)NC(C1CCCO1)=O 26271,c1(C(N(CC(C)CNC(=O)CC(C)P(C)(C)=O)C)=O)ccc(F)c2ncccc12 26272,C(=O)(CS(=O)(=O)CC(=O)NCCCC1CCCN1C(=O)C(C)CC(C)C)OC 26273,c1(OC)cccc(CC(N)C(=O)NCC(=O)OCc2cccs2)c1 26274,c1(CC)cc(C(N2CCCC2c2ccc(F)cc2)C(=O)NC(C)(C)C)ccc1Br 26275,N1(C(CC2CC(CC)C2)=O)CC2(CCOCC2)CC1CNC(C1OCCC1C)=O 26276,C12(C)CN(CCO1)CCNC2.C1(CC)OCCC1c1ccccc1 26277,C1(CNC(C(C(C)C)C#N)=O)C(C2CC2)CCN1C(=O)C=Cc1cocn1 26278,N1(C(C2(CC)CCCC2)=O)CC(NC(C2CN(C(C)=O)C2)=O)CC1(C)C 26279,N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26280,C1(C(C(=O)NCC(=C)C)N(CCF)CCOC)CCSC1(C)C 26281,CCCCCC(O)C(=O)NCC1CN(C(=O)C(=O)NCCOCCOC)CCO1 26282,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)CNC(=O)CCC3CCCC3)C1C2 26283,c1(C(=O)NCC2CCC(CC(n3cc(C=CC)nn3)C)CC2)cc(F)ccc1Cl 26284,C1(C)(C(=O)NCC(C(=O)NC)C)CCN(C(=O)CCOCC(F)F)C1 26285,C12(NC(c3cc(CC)ncn3)=O)CN(C(c3cnc4sccn34)=O)C(COC)(C1)C2 26286,CCCC(C#N)C(=O)NCC(=C1CN(C(C2OCCC2c2ccccc2)=O)C1)F 26287,N1(C(CC(CC)SC)=O)CCc2nc(CNC(=O)COCc3nc[nH]n3)sc2C1 26288,c1(-c2scc(C(=O)NC3CN(C(C4CC(F)C4)=O)C3)n2)cccc(Cl)c1 26289,CC(C)C(F)(F)CC(=O)NC1CC(F)(CNC(C2CCC(=O)N2)=O)C1 26290,c1(-c2cn(C)nc2)ccc2c(c1)CCN(CS(=O)(=O)CC1(C)CCN(CC#N)C1)C2 26291,N1(C(C=NOC)=O)CC2COCCC2(NC(=O)CCc2cccc([N+](=O)[O-])c2)C1 26292,C1(CCCN2CC(NC(C(CC)c3cccnc3)=O)C2)CCC(OC)CC1 26293,c1(C(c2scc(C(N)=O)n2)=O)cncc(N2CCN(C(=O)C3CC3)CC2)c1 26294,c1(N2CCN(c3nc(=N)[nH][nH]3)CC2)nc(=NC2CCCSC2)[nH]c2c1COC2 26295,N1(C(C2(CCCC)CC2)=O)CCC2(NC(c3ccc(-c4cccs4)[nH]3)=O)CC2C1 26296,c1(C(CNC(c2c(C)cncc2)=O)NC(c2ncccc2N)=O)cc(F)cc(Cl)c1 26297,C1(C(C)C(=O)NC2C3CN(C(=O)CCCCF)CC23)CCC(C)(C)CC1 26298,n1(CC(=O)N(CCCNC(C2C(C(=O)OCC)CC2)=O)C)cc2c(n1)CCCC2 26299,c1(C(N2CCC(NC(C3(CC(C)C)CCNC3=O)=O)C2)=O)cnc2sccc2c1 26300,C=CC1(C(N2CCC(C)C(NC(=O)CSCc3ccccn3)C2)=O)CCCCC1 26301,CC1(C)OC2(CN3CCCC3C(=O)NCCSCCC(=O)O)CCC1CC2 26302,C1(C(=O)OC)C(C)CCN1C(=O)CC1C(=O)NN=C1C.C12CC(C1)CCNC2=O 26303,C1(C(=O)NCC2(CNC(Cc3nnc(C)o3)=O)CC2)CCC(C)(C)O1 26304,C1(NC(C2N(N=O)CCC2)=O)(CNC(C2CC(O)C(=O)N2)=O)CCCCCC1 26305,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(C)n2)=O)(COC)CCOCC1 26306,N1(C(c2cnc(OCC)s2)C(=O)NC2CCOC2)CC(C(N)=O)C2(CC2)C1 26307,C12(CSC)CC(C(N3CCC(C)(CCNC(=O)CC=C(C)C)C3)=O)(CO1)C2 26308,c1(OCCC(=O)NC2CC(NC(=O)COC3CCC3)C2)ccccc1 26309,C1(NC(c2c(C)sc(O)n2)=O)C(CNC(c2cc(C#N)n(C)n2)=O)CCC12CCC2 26310,C1(CC)(NC(C2OCCC2CNC(=O)COCC(C)C)=O)CCCC1 26311,CC1CC(C(=O)NCCSCc2ccn(C)c2)CCS1 26312,C(=O)(CCCC(F)F)N(CCOc1ccc(C)cc1)C.N12CCCC1NC(=O)C2 26313,C1(F)(CNC(C2C(C)(C)C2)=O)CC(NC(c2cnsc2Br)=O)C1 26314,C1(CNC(C(=O)NCC(CO)OC)=O)CCCOCC1 26315,C=C(C)CCCC(=O)NCC=CCNC(=O)C(C)c1cncs1 26316,c1(NC(c2cn(CCOC(=O)NC3CCCCC3)nn2)=O)ccncc1C(F)F 26317,CC1CCN(CC(=O)NCCCN(CCCNC(C2CCSCC2)=O)C)C1 26318,C(CCCCCF)N(C(C)C1(CCCF)CC1)CCO 26319,c1(OC)cc(NC(=O)CC2C=CC(NC(c3ccsc3)=O)C2)ncn1 26320,c1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCCCO2)cncc(N=[N+]=[N-])c1 26321,CCC(C)(CC)C(=O)N(C1CN(C(C2CC(CC)=NO2)=O)C1)C 26322,N1(CC)CCCCC1C(=O)N(C)CC1CCCCN1C(C1(O)CCCCC1)=O 26323,CC(O)CCC(C)NC(=O)C(C)(C)CNC(c1cncs1)=O 26324,c1(C(C)(C)C(=O)NCC2(O)CC(NC(C3CCCO3)=O)C2)cccc(Cl)c1F 26325,c1(C(N(C2CC3CCC(C2)N3C(=O)CC2CSC2)C)=O)n[nH]c2ccccc12 26326,N1(c2cc(NCC(C3CCOCC3)OC)ncn2)CCC(O)(C(F)F)CC1 26327,C1(C(=O)NC)CN(C(=O)CN(C)C(=O)C2CC2)CC1(C)C 26328,C1(C(N(CC(F)F)C(C)C)=O)CN(C(c2cnccn2)=O)CC1(C)C 26329,c1(C(CNC(C2N(C(C)=O)CCC2)=O)O)c(F)cccc1Cl 26330,c1(C(=O)NC(C2(O)CN(C(=O)CC3CCC3(C)C)C2)C)cnccc1Cl 26331,C(=O)(C1SCc2cccnc21)N1CCN(C(CNC(CCC#C)=O)=O)CC1 26332,c1(CC(C(N2CCCSC2C)=O)CC(c2ccccc2F)C)ccc2c(c1)CCC2 26333,c1(OC)cccc(F)c1NC(=O)NC(C)C(C)C1CCC1 26334,c1(OC(C(=O)NC(c2cn(-c3c(C)cccc3)nn2)C)C)c(Cl)cc(Cl)cc1Cl 26335,CCC(CC)CCC(=O)N1CCC(N(C(=O)C(CC)OC2CCCCC2)CC)CC1 26336,C1(NC(C(=O)NCCOC)=O)CCC(CNC(=O)CC2CCOC2)C1 26337,c1(OC)cc(CNCC(c2ccc([N+](=O)[O-])cc2)O)cc(NOC)c1OC 26338,C1(NC(Cc2c(C)nn(C)c2)=O)CCS(=O)(=O)C12CN(C(=O)C(F)C1CCC1)C2 26339,c1(OC)cc(C=C2CN(c3ccn(C)c3)C2)ccc1OCC(C)C 26340,c12cc(ccn1)OC(=O)C(F)CC1CN(C1)C(=O)N2.C1(CN(C)C)CCOCC1 26341,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26342,c1(CC(=O)NC2CC(NC(C3CC(Cl)(Cl)C3)=O)C2)cnc2ncccn12 26343,c1(C(=O)NCC2CCN(C(C)C)C2c2cccnc2)c(F)cc(C#N)cc1F 26344,c1(C(N(CC(C)NC(C2CCCSC2)=O)CC)=O)cc(SC)ccc1Cl 26345,C1(C(=O)NC2CCCC2)(N(C)C)CCCCC1.C1(=O)CCOC(=O)CN1C 26346,CCCCC(CNC(C1C2CCC12)=O)NC(C1(O)CCC1)=O 26347,Cc1cccc(OCCC(N2CC(O)(C(C)NC(c3c(C)nsc3C)=O)C2)=O)c1 26348,N1(C(Cc2n(C)ccn2)=O)CCC(NC(c2ccnc(O)c2F)=O)C(CO)C1 26349,c1(N2CC3C(C)(CC3)C2)nc(=NCc2noc3c2COCC3)[nH]c2ccsc12 26350,c1(N2CCN(C)CC2CNC(c2cc3sccc3s2)=O)ncccc1[N+](=O)[O-] 26351,c1(NC)ncc(C(N2CC(CC(C)NC(=O)Cc3cccnc3)C2)=O)s1 26352,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26353,C1(CC)(NC(c2ccnc(C(C)(C)C)c2)=O)CCCN(C(c2snnc2C)=O)C1 26354,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CCC2)c(Br)ccc2c1CCC2 26355,C1(NC(=O)Cc2cccc(Cl)c2)CN(Cc2cccc(F)c2)C2CCCCC12 26356,C(CCN(C(=O)CCC=C(C)C)C)(C(C)C)NC(CCSCCC)=O 26357,c1(C(N2CC=CC(NC(C3CN(S(=O)(=O)C(F)F)C3)=O)C2)=O)sc([N+](=O)[O-])cc1Cl 26358,C(CN=c1cc(C)nc(O)[nH]1)(N(C(=O)Cn1cnc2ccc(C)cc12)C)C1CC1.CO 26359,C1(C(=O)NC2CC3(CN(C(C(n4cc(Cl)cn4)C)=O)C3)C2)CC2CCCC(C1)C2 26360,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26361,C1(C(N(CCOCCN(C(Cc2ccc(CC)cc2)=O)C)C)=O)CC2C(C1)C2(C)C 26362,S(=O)(=O)(c1ccc(NCC(C)Sc2cccs2)c(C#N)c1)NCCCCCCF 26363,c1(NC(c2ccc(F)nc2F)=O)nccc(C(=O)Nc2cccc(CO)c2)c1Cl 26364,C(=O)(CCCC(=O)OC)N(C)CC1OCCN(C(C(C(C)C)SC)=O)C1 26365,c1(CC)nc(N2CC3CC(NC(=O)C(C)C)CC3C2)c(C)c(Cl)n1 26366,C#CC1CCCN(C(C2(CNC(=O)C=Cc3ccoc3)CCC2)=O)C1 26367,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26368,c1(C(N2CCC(NC(CN3C(C)CC3)=O)CC2C)=O)cccc2[nH]ccc12 26369,Cc1ccnc2nc(C(=O)NC3CN(C(C4(C)CCCC4)=O)CC4(CC4)C3)nn12 26370,Cc1ccc(C(C)CN(C(N2CCCCC2)=O)CCN)cc1 26371,C(=O)(CC(C)C(C)(C)C)N1C(C(C)C)CN(C(=O)CCCc2ccsc2)CC1 26372,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2nc(C)cs2)C12CC2 26373,N1(C(COCCCCCC)=O)CC(NC(=O)C(CC)OC)CC1CO 26374,C(=O)(C#CC1(C)COC1)NCC1CC(F)(CNC(Cc2cc(CC)nn2C)=O)C1 26375,c1(NC(C2CC(NC(=O)NC(c3nncs3)C)C2)=O)cccc(C#N)c1 26376,c1(C(=O)NC2CCC(CC(=O)N(CC(O)C(F)(F)F)C)C2)cncc2[nH]ccc12 26377,CC(C)CC(C)CC(=O)NCC=CCNC(C1CCC(c2ccccc2)CC1)=O 26378,C(=O)(CC(O)C(F)(F)F)N1CCC(NC(=O)CCC2OCCO2)C(O)C1 26379,CCC(C)C(C(=O)N1CCC(n2cc(CCn3cncn3)nn2)C(O)C1)N(C)C 26380,N1(C(=O)Nc2c(C)nn(CC(C)C)c2C)CCN(C(=O)C(C)NC)CC(C)(C)C1 26381,C1(N(C)C)CCCN(C(C2C=CCN(C(=O)C=Cc3cncn3C)C2)=O)C1 26382,C1(NC(N(CC)CC2(c3ccc(C)cc3)CCC2)=O)CC2(COC(=O)N2)C1 26383,N1(CC(=O)NCc2scc(C(C)C)n2)CCN(C(c2cnc(Br)s2)=O)CC1 26384,c1(NC(C=CCN(C(=O)CC2C=CCC2)C)=O)ncn2ccccc12 26385,CP(C)(=O)CC(=O)N1CC2(N(C(C3CC(OC(F)F)C3)=O)C3CC3)CC1C2 26386,C1(C(c2cccnc2)CN2CC2)CCCC(C(F)(F)F)C1.CO 26387,c12cc(c(C)cc1C)NC1(CC1(F)F)C(=O)N2.c1(OC)ccc(C(F)(F)F)cc1 26388,C1(C(=O)Nc2c(Br)nn(C)c2C(F)(F)F)CCN(C(=O)C(F)(F)F)CC1(F)F 26389,CCC(C(=O)NC(C)(CNC(c1cc(C2CCCCC2)[nH]n1)=O)CO)C(C)C 26390,N1(C(C(=O)NCCC)CC2CC(F)(F)C2)CCC(C2CCCCC2)CC1 26391,c1(CC(=O)NC2(C)CC(NC(C(CC)(C)O)=O)C2)cccc(F)c1Cl 26392,C12CCN(CC1)C(c1occc1Br)C(=O)NCC2.c1(COC(C)=O)ccccc1 26393,c1(CC(=O)NCC(C)(C2CC2)NC(C(COCC)C)=O)cccc(S(C)(=O)=O)c1 26394,CC1CC(C)C1C(=O)NC1CCC(CNC(=O)C(C)n2cccn2)C1 26395,N1(C(CNC(=O)NC)=O)CCN(C(=O)C(O)CC(=O)OC(C)(C)C)C2(CCC2)C1 26396,CC1CC(NC(C2CC2C#N)=O)CCN1C(c1cnn(C2CC2)c1Cl)=O 26397,c1(C(=O)NCC(C)(O)CNC(c2cccnn2)=O)cc2c(nn1)CCC2 26398,n1(CCC(N2CC(CCC)N(C(=O)C(N)=O)CC2)=O)cnc2c(cnn2C)c1=O 26399,C1(CC(N2CCC(NC(=O)CCCC3CCCC3)CC2)=O)CC(O)C12CCC2 26400,c1(C(=O)NC(CC)CN(C(=O)C=CC2CC2)C)cccc(NC(N)=O)c1 26401,C1(C(N(CCOC)Cc2ccccc2)=O)CC(NC(C2OCCC2(C)C)=O)C(O)C1 26402,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26403,c1(CNC(c2ccc(OCC#C)cc2)=O)ccc2c(c1)C(CN)CCC2 26404,C1(OC)CC(N(C(=O)C(C)=C(C)C)C)C1.C1(=O)CC2CC2CN1 26405,C#CC1(C(=O)NCCN(C)CC)CCN(C(=O)CCNC2CCCN2CC)C1 26406,c1(OC)ccc(F)cc1CC(N1CC(C)C1CNC(c1cc(O)nn1C)=O)=O 26407,C1(C(N2CC(CC(C)(C)C)C2)=O)CCCC(NC(=O)C(C)(C)C(C)O)CC1 26408,c1(NCC2(NC(C(CO)NCC)=O)CCCC2)nc(C)nc2sc(C)c(C)c12 26409,c1(OCC)cccc(C(N2CC3(NC(=O)CC(=O)NCC(F)(F)F)CC2C3)=O)c1N 26410,C1(C(=O)NC(CCOC)CO)C=CCCN1C(=O)Cc1cc(C)cs1 26411,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 26412,N1(CCC)CCC(C(=O)NCC(CNC(C2CC2[N+](=O)[O-])=O)CO)CC1 26413,C1(C(=O)NCC2CC2CNC(C2(O)CCOCC2)=O)C2CCCCCC12 26414,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26415,C(=O)(CCC(C)(C)C(=O)N(CCO)CCNC(C1CCCCC1F)=O)OC 26416,N1(C(C2CC(=C)C2)=O)CCN(C2CCC(NC(=O)Cc3ncccc3C)C2)CC1 26417,c1(C(=O)NCC2N(C(CC(C)C(F)F)=O)CC(F)(F)C2)cc2ccccn2n1 26418,N1(C(N2CC(c3ccc(C#N)cc3)OCC2)=O)CCc2ccc(Br)cc2C1 26419,c1(C(=O)NC2(C)CN(C(C3C(CC)CCCC3)=O)C2)cc2c(C)ccc(F)c2[nH]1 26420,C(c1ccccc1NC(c1c(CC)cncc1)=O)=CC(=O)NCC1CC1CSC 26421,N1(C(C(CSC)O)=O)CC(C(=O)NCC2(C(C)C)CC2)CC1(C)C 26422,N#Cc1c(Cl)c(NC(C23CC2CN(Cc2cnco2)C3)=O)cc(F)c1Cl 26423,CC1(CNC(C2C3COCC23)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 26424,N1(Cc2cccc(C)c2)CCC(C)C(NC(c2cc(-c3ccco3)nn2C)=O)C1 26425,C1(NC(COCC=C)=O)CCCC(NC(c2cccc(CCN(C)C)c2)=O)C1 26426,CCC(C)(C#N)C(=O)NCCN(C(c1ccccc1NCCO)=O)CC1CC1 26427,c1(NCC2CN(C(CC(C)C(F)(F)F)=O)CC(C)(C)C2)ncc(Cl)cc1[N+](=O)[O-] 26428,c1(OC(=O)NCC2CC(O)CN2C(=O)NCC(O)CO)cccc([N+](=O)[O-])c1 26429,N=c1nc[nH]n1CC(=O)NCCC1CN(C(=O)Cc2cnsc2)C1 26430,N1(C(C(CC)NC(c2cc(C)cnn2)=O)=O)CC(C)N(CC)CC1C 26431,N1(C(c2c(C)nn(CCO)c2)=O)CCN(C(=O)CN2CC2C)CCC1C 26432,N1(CCC)CC(C(=O)NCC2CCN(C(c3cocc3C)=O)CC2)CC1=O 26433,N1(C(C=C(C)c2cccs2)=O)CC2CCC1C(CNC(C1(OC(C)C)CCC1)=O)C2 26434,c1(C(=O)NCC2N(C(C(CCOC)(C)C)=O)CCC2C)cccc2ccc(O)nc12 26435,C1(C(N)=O)(NC(c2ccc(F)o2)=O)CCN(C(C2OCCO2)=O)CC1 26436,S(=O)(=O)(CC(=O)NCC1(CSCCCC)CCCCC1)NC(C1(CCC)CC1)=O 26437,CCC(CCCC(=O)N1CC2(C1)CC2(F)F)NC(C1(O)CCSC1)=O 26438,c1(CN(CC(C)(C)CBr)C)csc(C(C)(C)C)c1 26439,c1(CC(=O)NCCC(C)(C)NC(C(C2CCCCCC2)C)=O)cn(C)nc1Cl.C1CC1 26440,C1(C(N(CCC)CC)=O)CCCCN1C(=O)CCc1cn(C)nn1 26441,C(=O)(C#CC(C)(C)C)NCC1(NC(c2ccc(OC)s2)=O)CCCCC1 26442,CCS(=O)(=O)C=CC(=O)NCC1CC12CCN(C(C1(C(N)=O)CC1)=O)CC2 26443,C1(c2cn(CCCOC)nn2)C(C)CCN1C(c1ccc(C(C)=O)s1)=O 26444,C(c1ccccc1)=[SH]CC(=O)NCCC1CC(NC(CCc2nc(=N)[nH][nH]2)=O)C1 26445,c1(OC)ccc(S(=O)(=O)N2CCOC(C)(C(F)F)C2)cc1-c1ccc(C)cc1C 26446,CCCCCC(F)C(=O)N1CC=CC1C(N1CCc2ncsc2C1)=O 26447,C1(NC(=O)Cn2cnnc2O)CCCN(C(C2(F)C3CCCC23)=O)CC1 26448,c1(NC(CSC(C)(C)C)=O)ccc(SC(F)F)cc1 26449,N1(C(c2cc(CO)ccn2)=O)CC2(C=C(C(=O)N3CC=C(CO)CC3)CO2)C1 26450,C1(C(=O)NC(CN(CCCC)C)C)CCN(C(=O)CC2CCCOC2)CC1(C)C 26451,C1(O)(C(=O)NCCOCCCNC(CC2C(C)(C)C2)=O)CCOC1 26452,c1(C(N2CCN(C(C(C)C3CCC3)=O)C(CO)C2)=O)ccc(N)c2ncccc12 26453,C1(C)(C(N(CCC)CCNC(=O)Cc2ccn(CC)n2)=O)CC(C#N)C1 26454,N1(C(Cn2cc(-c3ccc(NC(C)=O)nc3)nn2)=O)CC(C)C(C(=O)O)C(C)C1 26455,c1(C(N2CCCC(N(C(c3cc(OC)ccn3)=O)CC)C2)=O)cc(C)c(C)cn1 26456,c1(C(N2CCCCC(NC(C(COC)OC)=O)C2)=O)cc2cc(C)[nH]c2cc1Cl 26457,C(=O)(CC1=CCOCC1)NCC(CO)NC(CCC(c1ccccc1)N(C)C)=O 26458,C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(C)(NC(C2(CC)CC2)=O)C1 26459,c1(C(C)NC(c2nc(C)n(-c3ccccc3Cl)n2)=O)nnc2c(=O)[nH]ccn12 26460,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26461,C(=O)(C(CNC(C)=O)c1ccccc1)NCCCN(C(S(=O)(=O)C(C)C)=O)CC 26462,c1(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Cl)cnnc1Cl 26463,c1(NC(c2scc(-c3c(F)ncc(C)c3)n2)=O)cc(Br)c(F)cc1C 26464,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26465,c1(C(N2CCC(CNC(c3c(CC)scc3)=O)C2)=O)n[nH]c2c1COC2 26466,N1(C(C(C=CC)O)=O)CCC2CCCC12C(=O)NC1CCC2CCC12 26467,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26468,C(=O)(C(F)(F)C(C)(C)O)N1CCC(CN(C(=O)C(=Cc2c[nH]cn2)F)C)C1 26469,C1(F)(CNC(C2C=CC=CC=C2)=O)COCCN(C(=O)CC23CCC(CC2)C3)C1 26470,C#CCC(C)(CC)C(=O)NCCN(CCOC)C(c1cnc(C2CCC2)o1)=O 26471,C#Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)N(C(C(N)=O)C2CC2)C)cc1 26472,Cc1c(O)ccc(C(=O)NC2(C)CCN(C(c3ccc(F)c(N)c3)=O)CC2)c1C 26473,c1(C(=O)NC2C3N(C(c4c(CC)oc(C)c4)=O)C(CC3)C2)ccsc1S(C)(=O)=O 26474,c1(C(=O)NC(C(C)NC(=O)C(F)OC(F)(F)F)CO)ccn(C)c1-c1cccs1 26475,c1(NC(C2CN(C(c3ncccc3F)=O)CCN2)=O)cccc2nc(O)ccc12 26476,CC1(C)CCN(C(c2cnns2)=O)CC1NC(=O)CCc1cncnc1 26477,c1(C(N2CCC(N(C(=O)CCCCC#N)C)CC2)=O)cc2ccncc2cc1F 26478,c1(-c2nc(COCC)oc2)nc(C(c2cccc(Br)c2)C)nn1-c1ncnn1C 26479,c1(CCC(=O)NCCC(C)NC(C2(C)CSC2)=O)cncnc1O 26480,C1(C(=O)NCC(C)NC(=O)N(C)C)CCCCN1C(C1CN(C2CC2)C1)=O 26481,N1(C(c2c(C)noc2)C(=O)NC(c2ccccc2)C)CC(C)(C)C1C(C)C 26482,C1(C(=O)NC(c2ccsc2)C)CN(C(=O)C(=O)NC2CC2)CCC1(C)C 26483,c1(OCC)cc(C(C(=O)NC2(O)CCCCCC2)N(C2(C)CC2)C)cc(Br)c1OC 26484,C12(C(=O)NC3C(NC(CC=CC=C)=O)CCCC3)CCC(CC)(C1)OC2 26485,C(C(C)NC(=O)CCc1ccccc1C)(C(C)C)NC(C(C)=CC)=O 26486,C(=O)(CCC(C)NC(C1CC(O)CN1C)=O)NC(CCOC)(C)C 26487,C1(NC(CCC)=O)CCN(C(=O)CCNC(C2CCOC2COC)=O)C1 26488,N1(C(c2c(CC)nn(C)c2)=O)C2CCC1C(NC(C1CCOC1)=O)C2 26489,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCc2cccs2)C1 26490,CCCCC(C(=O)NC(CNC(c1cnn(C)c1)=O)CC(C)C)NC(N)=O 26491,C1(C)(CC)CC(C(N2CCC(OCCNC(c3sc(C)c(C)c3C)=O)C2)=O)CCO1 26492,c1(C(N(CCNC(=O)C(C)(C)SC)CC)=O)ccc2nc(C)cc(Br)c2c1 26493,S(=O)(=O)(c1ccc(Br)cc1N(CCCF)C)NC(C)CN(C)C 26494,N1(C(CCC(=O)NCC)=O)CC(NC(C2CC=CC2)=O)CC(F)C1 26495,c1(C(=O)NC23CC(CNC(C(C)=C(CC)C)=O)(C2)C3)cn(C)cc1C(F)(F)F 26496,C12(C(=O)NC(C3N(C(c4c(C)n[nH]c4C)=O)CCC3)C)CCC(CC1)C(C)O2 26497,N1(ONC(c2c(NC(Cn3ccc(C)n3)=O)occ2)=O)CC(C(N)=O)C2(CC2)C1 26498,c1(C(N(CC(CC)NC(=O)C(O)CC2CCCC2)C)=O)cc(F)n(C)n1 26499,N1(C(C(COCC)C)=O)CC2CC(NC(c3cccnc3N)=O)C(C2)C1 26500,C(C1=CCN(C(=O)C2=CCCOC2)CC1)NC(C(c1ccc(CC)cc1)C)=O 26501,N1(C(C(C2(O)CN(C(C(C(C)C)OC)=O)C2)F)=O)CC2CN(C)CC2C1 26502,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26503,N1(C(C(CC#C)(C)C)=O)C2CCC1CC(N(C)C(c1ccc([N+](=O)[O-])cn1)=O)C2 26504,C(CC(C)CC)(C(=O)N(CC(C)(C)CN(C)C)C)NC(c1c(C)nc(CC)o1)=O 26505,c1(C(N2CCC3CCC(C2)N3C(C23CC(F)(C2)C3)=O)=O)cnn2c1CC(F)(F)C2 26506,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26507,Cc1ccc(Br)c(CNC2COCCC2c2ccccc2)n1 26508,C1(CNC(c2c(C)nco2)=O)CN(C(=O)CSc2n[nH]c(O)n2)CC12CCC2 26509,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1CC#N 26510,C1(C2(O)CN(C(=O)CC3CNC(=O)O3)C2)(CNC(=O)CCc2cnco2)CC1 26511,CN1CCCC(C)(C(N2CC(N(C)C)C(C(=O)OC(C)(C)C)C2)=O)C1 26512,C1(OC)CC(CO)N(C(C2CN(C(=O)C(C)(C)C)C2)=O)C1.C1(=O)CN1 26513,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26514,c1(N(C)C)cccc(-c2cn(C3CCC(C(=O)NCCCO)CC3)nn2)c1 26515,C1(C(N2CC(CNC(C(c3n(C)cnn3)(C)C)=O)C2)=O)CCC(C)(C)CO1 26516,c1(N)cccnc1-c1ncsc1C.N1(CC(=O)NC2CCCC2)CCC1CNCC 26517,c1(C(=O)NC2CCC(CCNC(CC(=O)NCC)=O)C2)noc2ccc(Cl)cc12 26518,Cc1cnc2n1CC(C(N1CC(NC(C3SCCS3)=O)C3(CC3)C1)=O)CC2 26519,N1(C(=O)CC2(O)CCOC2)Cc2n[nH]cc2C1C(=O)N1CC2CCCC2C1 26520,c1(C(N2CCCC(C(=O)OC)C2)C(=O)NOCCF)c[nH]c(=S)cn1 26521,c1(OC)ccc(C=CC(=O)NC2CC(C)N(C(c3ccc[n+]([O-])c3)=O)C2)c(C)c1 26522,c1(OC)cc(C)c(C(N2CCCC(N(C)C(C3(C4CC4)CCCO3)=O)C2)=O)cn1 26523,N1(CC(=O)NC(C(=O)N(CCC(=O)OCC)C)C)CCCCC1=O 26524,c1(C(C)NC(=O)NC(C(=O)N(CCOC)C)C2(O)CCC2)ccc(F)cc1 26525,C1(NC(c2cncc(C)n2)=O)CCN(C(=O)COC2CC2)CC1(C)C 26526,Cc1nn(C)cc1C(=O)NCCCN(C(=O)C(C)NC(c1ccc(Cl)cc1)=O)C 26527,CC(C(O)C(=O)NC1CC(CCNC(c2cccnc2S)=O)C1)c1ccccc1 26528,c1(NC(C2C(NC(C(c3ccccc3)C)=O)CC2)=O)cncc(C#N)c1 26529,N1(C(=O)OC(C)(C)C)CC2C(C(=O)OC3CCC3O)C2C1 26530,C1(C(=O)NCC2N(C(CCc3cc(OC)no3)=O)CCC2)CC(C)OC(C)C1 26531,N1(C(CN(C(=O)NCC)C)=O)C2CCC1CC(NCC=Cc1cn(C)cn1)C2 26532,C1(C(=O)NC(CN(C(c2c(C)scn2)=O)C)(C)C)CCCC(F)C1 26533,N1(C(Cc2ccn(C)n2)=O)CCC(O)(CCCc2nc(-c3ncccn3)no2)C1 26534,C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(c2nnc(CCOC)s2)C1 26535,C1(CNC(C2C(C(C)(F)F)C2)=O)CCN(C(=O)CCC2OCCO2)CC1CO 26536,N1(C(C(COC)C)=O)CC2(C1)CN(C(c1c(F)ccc(C)c1F)=O)CC(C)(C)O2 26537,c1(C(=O)NC23CCCC(NC(C(CC)=CC)=O)(C2)C3)ccc(Cl)c(F)c1N 26538,c1(CN(C2CCN(C(c3nn[nH]c3Cl)=O)C2)C)cccc(F)c1[N+](=O)[O-] 26539,C1(C(=O)NC)(C2CC2)CC12CC2.C1(C(=O)NCC(=O)C(C)SC)(COC)CCCC1 26540,c1(C(=O)OCC)cc(C(=O)NCC(O)CNC(c2ccn(CCF)n2)=O)nn1C 26541,N1(C(c2nccc(C)c2)=O)C2CCC(C2)C1CNC(=O)COc1ccccc1F 26542,c1(C(=O)NCC(C)NC(=O)C(c2cc(Cl)ccc2F)(F)F)cncc([N+](=O)[O-])c1 26543,N1(CC(=O)NC2C=CCCC2CO)C(=O)CCC1=O.N12CCC(C1)CC2=O 26544,C(=O)(C1OCCc2ccccc21)N(CCNC(CC(C)OC)=O)C(C)C 26545,C=Cc1ccc(NC(C2CN(Cc3cccc(N(C)C)c3O)CCO2)=O)cc1 26546,C1(NC(C(COC)O)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CC12CCC2 26547,Cc1cc(C(N2CC(OCCNC(=O)C=CCF)C2)=O)c(C)cn1 26548,C12CN(CCO1)Cc1cn(nn1)C2.CCS(=O)(=O)NCC(=O)NCC(F)(F)F 26549,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26550,N1(C(CCCC(C)C)=O)CC2(CCN(C(c3cc(CO)ccn3)=O)C2)C1 26551,c1(CN(C(=O)CCN2CCC=C(F)C2)C)ccc(F)cc1Cl.C1(=O)CO1 26552,C12(NC(c3c(CC)cccc3)=O)CCN(C(=O)Cc3cc(C)on3)CCC1C2 26553,C1(CCN(C(COCc2onc(C)n2)=O)C)CCCCN1C(C1CC1F)=O 26554,CCC(C(=O)N1CCOC(CNC(=O)Cn2ncc(O)nc2=O)C1)C(C)(F)F 26555,CC1CC2(CCO1)CC2C(=O)NC(CNC(c1cc(C(F)F)on1)=O)C1CCC1 26556,S(=O)(=O)(c1cccnc1Cl)N1C(C(=O)NC(c2ccc(Br)cc2Cl)CO)CCCC1 26557,N1(C(C(CCC)(C)C)=O)CCC2(CC1)CC(CNC(=O)CC(C)CC)C2 26558,C1(C(N(CC(C)C(=O)NC2CCOC2)C)=O)CCC(O)CN1C 26559,C=CCCCCCCC(=O)NC(C1(O)CN(C(=O)C(C)=C(C)CC)C1)C 26560,CC(C)(C)CCC1CCN(C(c2ccncc2)C(=O)NC2CCC2)C1 26561,c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)nc2cccnc2s1 26562,N1(C(c2c(C)nc(CO)o2)=O)CCN(C(=O)C(C)O)CC(O)C1 26563,c1(C(N2CC3N(C(C(C)SC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26564,C(CN=c1cc[nH]cc1S(=O)(=O)N1CC(C)(C)C(O)C(C)(C)C1)C1N(C)CCC1 26565,C(CC(=O)NC1(CCC(=O)NCCc2cn[nH]c2)CCC1)=CC=C 26566,c1(C(=O)NC(C)CCNC(C2COCCN2C)=O)cccc2nc(O)[nH]c12 26567,c1(C(=O)NC2(C)CCN(C(C(C(C)(C)O)F)=O)CC2)cc(O)c2ccoc2c1 26568,c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCO)ccc(OC(F)F)cc1 26569,C1(NC(CC)=O)CN(C(=O)CCn2cnnn2)CC1NC(=O)CCN(C)C(C)=O 26570,N1(C(C2C(C)(C(C)C)C2)=O)CC2CC3CC2C1C3NC(c1ccccc1NC=O)=O 26571,C1(NC(C2C(C)=CCS2)=O)CCN(C(c2ncnn2C)=O)CC1O 26572,c1(C(C)NC(C)=O)nc(-c2cccc(Cl)n2)nn1CC(C)C 26573,C(=O)(CC(F)(F)C(F)F)N1C(C(=O)NCC(CCOC)(C)O)CCCC1 26574,C1(C(N(C2(CO)CCOC2)C)=O)CCCCC1(F)F.C12(CC1)N(C)C2=O 26575,C(CCCCC(=O)NCC(CC(F)(F)F)NC(=O)Cc1cccnn1)OCC 26576,Cc1cccc(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3CC23)=O)n1 26577,C=CCCCC(C(=O)NC1CC(C2CCC2)C1)NC(=O)CCCC 26578,Cc1cnccc1C(=O)NC(C)C(CO)NC(=O)C(c1ccc(Cl)cc1)(C)C 26579,c1(CCNC(=O)NC(c2ccccc2Cl)C)c[nH]c2ccc(O)cc12 26580,Cn1cnc2c(C(=O)Nc3cccc(Cc4ccc(C#N)cc4)c3)ccnc12 26581,CCC(CCOC)C(=O)N1CC(OC)C(C(=O)N(C)CCOCCO)C1 26582,C1(COC)(CNC(c2cnncc2C)=O)CCCN1C(=O)C(C)CC1CCCO1 26583,N1(Cc2ccc(OCC=C)cc2)CCN(C(=O)C(C)COC(C)=O)C(CC)C1 26584,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26585,c1(C(=O)NCC(CC)NC(=O)CCCF)ccc(S(=O)(=O)C(C)C)cc1 26586,N1(C(CC=C=C)=O)CCC(C2CCN(C(c3cc(C#N)c[nH]3)=O)CC2)C1 26587,Cn1cc(CCCNC(=O)C(C2(O)CCC2)NC(C2CCCC2)=O)nn1 26588,C(=O)(C1=C(C)CCC1)NCC(=CC(=O)N(CC)CC1CCCO1)C 26589,c1(SC)cc(C(=O)NCC(C)(C)CNC(c2cscc2SC)=O)n(C)n1 26590,C1(C2CC(=O)N2)CC2CCC1C2.C(CC(=O)NC1CCCC1)OCCN(C)C 26591,CCCC(C#N)C(=O)N1CC(C(=O)NCC2CC(OCC)C2(C)C)C(F)(F)C1 26592,N1(C(CC(=O)OC)=O)C2CCC1CC(CC(C)NC(C13CCC(C)(C1)OC3)=O)C2 26593,C1(CNC(CCS(C)=O)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)C12CCC2 26594,C(=O)(C1=CCCCC1C)NC(CN(C(c1c(OC)cc(O)nc1)=O)C)C 26595,C=CCC(C)C(=O)N1CCOC(CNC(=O)CCc2nncs2)C1 26596,c1(C(C(=O)N(CCNC(CC(C)CN(C)C)=O)C)O)ccc(Cl)c(Br)c1 26597,c1(C(=O)NCC(CC)NC(c2ccn(CCC)n2)=O)cccc2c1CCOC2 26598,c1(C(=O)NCCCN(C2CCCC2)C(C2C(SC)CCC2)=O)nc(SC)ncc1Cl 26599,C(C(=O)NNC(=O)OC)OCC(c1ccccc1)OC1C(OCC)OCCC1 26600,C1(C(=O)NCC=CC(=O)N(CCCCC=C)C)CC2(CC2)CO1 26601,N1(CC)C(=O)CCC1CC(=O)NC1CN(C(C2(CC3CCC3)CC2)=O)CC1O 26602,C(=O)(CCCC(=O)NC(C)C)NCC12CC(NC(C3N(C(C)C)CCC3)=O)(C1)C2 26603,N1(C(C2C(=C)CC2)=O)CCN(C(c2ccc(C(C)(C)C)cc2)=O)CC1CO 26604,c1(C(N2CCC(N(C(=O)COc3cccnc3)CC)C2)=O)ccc2cccnn12 26605,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26606,CC(C(C)CO)NCc1ncoc1C1CNC1 26607,c1(CC(C(N2CCC(CN(C)C(C3CC(CF)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26608,C(=O)(C(C(C)O)c1ccccc1)NC1(CCOC)CC1.C12(CCC1)C(=O)NC2 26609,c1(CC(N2C(C(C)NC(C(CC#C)(C)C)=O)CCCC2)=O)c[nH]c2ncccc12 26610,C1(C(=O)NC(C)CF)CCCCCC1NC(c1nc(Cl)ccc1N)=O 26611,Cc1snnc1C(=O)N(C(C)CNC(C1CCC1C(F)(F)F)=O)C 26612,N1(C(c2cc(C)[nH]c2C)=O)CC2(CCC(C(=O)Nc3cnn(C4CC4)c3)O2)C1 26613,c1(CC(=O)N(CCC(=O)NC(C=C)C2CCC2)C)cc(C)on1 26614,c1(CNC(CC)=O)ccc(CN(C(=O)CC=CC(C)(C)C)C)cc1 26615,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26616,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26617,c1(NC(C2CCN(C(C3CN(CCOC)C(=O)C3)=O)C2)=O)c(Cl)cc(Br)cc1Cl 26618,c1(CC(=O)NCCCN(C(=O)CNS(C)(=O)=O)C(C)C)nccc2ccccc12 26619,C1(C(=O)NC)CC12CCN(C(c1c[nH]c(C#N)c1C)=O)C2 26620,c1(C(C(=O)NCC2CC2)N(C)C)ccccc1.n12cc(nn1)C(=O)N1C(CC1)C2C 26621,C(CC(Br)C(=O)OC)(c1nnnn1CCOC)NCC=CC 26622,COn1cnc(C)c1C(=O)NC1CC(=O)N(C2CN(C(C3CC3C#N)=O)C2)C1 26623,n1(CC)ncc(Cl)c1C(=O)N(CC(O)CN(C)C(C1(C)CC1)=O)C 26624,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26625,c1(OC)cc(Br)c(NC(=O)NCC(C)(C)C(N)=O)cc1F 26626,C(=O)(C(C(C)(C)C)c1ccccc1)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26627,n1(CCC(N2C(CN(C)C(c3cnn(CCF)c3)=O)CCC2)=O)cnccc1=O 26628,c1(SCC(c2n(CCCC)nnn2)NC(CC)CC)cc(Cl)cc(Cl)c1Br 26629,O=S(=O)(c1ccc(C(F)F)cc1F)N(CCO)CC1(Br)CC1(F)F 26630,Cn1nnc2c1CCC(CNC(=O)OC(C)(C)C)C2.C1(C)(S)CC(C2CC2)=NO1 26631,CC1CN(C(=O)CCc2cccc(C#N)c2)C(C)CN1C(=O)CCc1nc[nH]n1 26632,c1(C(N(CC(CN(C(C(C)=C2CC2)=O)C)O)C)=O)cc(F)cc2nc[nH]c12 26633,C(=O)(CC(C)CF)N(CC(C)CNC(c1c[nH]nc1-c1cnn(C)c1)=O)C 26634,N1(C(C2(Cn3cc(-c4c(C)cccn4)nn3)CC2)=O)CC2OCCN(CO)C2C1 26635,C=CCC(C)(C)CNC(c1cnccc1OCC)=O.c12conc1CNC2=O 26636,CN=C(NCc1cnn(C(C)C)c1)N1CC2CC2(CC)C1 26637,CCCCC(C(=O)NCCCCCCNC(=O)C(F)=C1CCCC1)N(C)C 26638,C1(C(=O)NCC(=O)OCC=C)CC12CC(NC(c1ccoc1)=O)C2 26639,N1(C(c2c(C)sc(O)n2)=O)CC2COCC2(C(=O)NCC2CCOC2)C1 26640,Cc1cc(C(=O)N(CCC(=O)NCCc2ncc[nH]2)CCO)nc(O)c1 26641,c1(SC)ccc(F)c(-c2c(N(C)Cc3ccccc3N3CCCC3)ccnc2)c1 26642,Cc1nc(O)nc(C)c1C(=O)NC1CCCCC1CNC(c1ccc(N)c(Cl)n1)=O 26643,CC1CN2CCN1C(C(=O)NCCCCC1CN(C(=O)CC3C=CCC3)C1)C2 26644,C(=O)(CCC(=O)NCC1OCCC1C(=O)NC1(C)CC1(C)C)NCCC 26645,CC1CN(C(=O)CC2(c3ccccc3)CCC2)CCC1NC(c1cnnn1C)=O 26646,C1(F)(C(N2CC(=C(CC(=O)NCc3noc(CO)n3)F)C2)=O)C2CCCCC12 26647,N1(S(C)(=O)=O)CCCC(C(=O)NCC#CCNC(C2CCCC(O)C2)=O)C1 26648,c1(C(=O)OC)cc(C(F)F)cc(N=c2[nH]c(C3CNC3)ncc2OC)c1 26649,N1(C(C2CC(F)(F)C2)=O)CCCC(NC(C2(c3ccccc3)CC2(F)F)=O)C1 26650,N1(C(C2OCCC(C)(C)C2)=O)CCOC2(C1)CN(c1nccc(C(F)(F)F)n1)C2 26651,C=C(CNC(c1cnc(C2CC2)s1)=O)CCNC(c1cc(CC(C)C)c[nH]1)=O 26652,N1(C(c2c(CC)cc[nH]2)=O)CC2C(C(=O)N(C)Cc3nnc(C)o3)C2C1 26653,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cc(Br)nn1C)=O)C2 26654,c1(C(=O)NCC(CNC(=O)C(O)Cc2ccccc2)OC)ccnc2ccsc12 26655,C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(c2nc(COC)nc(C)c2)CC1)C 26656,c1(CNC2(c3nnnn3C(C)(C)C)C(CC)CC2)csc2cccc(F)c12 26657,c1(C(=O)N(CCC(C)N(C(=O)CC2CCCC2(F)F)C)C2CC2)cccc(=O)n1C 26658,c1(C(N2C(C(C)(C)NC(CS(CC)(=O)=O)=O)CCC2)=O)cn2nc(OC)ccc2n1 26659,CC1CC(C(=O)NCC2CCN(C(=O)COc3ccn(C)n3)CC2O)=NO1 26660,N1(C(c2c(C)nc(CO)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(C2CC2)n1 26661,C1(CC)CC(C(=O)NCC(C)(C)NC(c2ccc(CCOC)cc2)=O)CC(=O)N1 26662,C(CC1=CCN(C(=O)C=Cc2cnc[nH]2)CC1)NC(C1CC1C(F)F)=O 26663,c1(C(N2CCCC(N(C(C(CC)NC(C)=O)=O)C)C2)=O)cc2cccnc2[nH]1 26664,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2ccc(Br)o2)=O)C1 26665,Cc1ncc(C(=O)N(CCCN(C(=O)C(F)Cc2ccccc2)C)C)[nH]1 26666,N1(C(CC(CC)OC)=O)Cc2nccn2CC(NC(=O)CCc2cc(Cl)no2)C1 26667,c1(C(=O)NC(C)CCNC(C2CC2c2cc[nH]c2)=O)c(Cl)cccc1Br 26668,O=C(CN=c1cc[nH]cc1)NCC1CCCN1C(=O)COc1ccc(F)cc1F 26669,N1(C(C23CSC(C2)C3)=O)CCN(C(C2(CO)CC2)=O)CC1c1ccncc1 26670,S(=O)(=O)(c1ccc(N2CCN(c3cccc(C)c3)CC2)cc1Cl)NC(C=C)(C)C 26671,c1(NC(C2(F)CCN(C(c3cccc(C)c3)=O)C2)=O)cc(Br)c(Cl)cc1F 26672,C1(CC(=O)NC2(CC=CC(=O)NCCCOCC)CCC2)CCOC1(C)C 26673,C(=O)(C(C#N)C(C)(C)C)NC(C(C)C)CCN(C)C(C1CCCC1C(F)F)=O 26674,c1(C(N2CC3CCN(C(C(C)OCCCC)=O)C3C2)=O)oc2ccccc2c1C 26675,CCC(C)(CSC)C(=O)N1CCN(C(=O)CSC)CC1 26676,c1(C(c2cccnc2N)NC(N(CC(c2ccccc2)C)C)=O)ccccc1F 26677,N1(C(CCC(C#C)(C)C)=O)CCC2CCN(C(c3coc(COC)n3)=O)CC2C1 26678,C=CC(C)(O)CC(=O)N1CC(C)(OCC(=O)NC(C)CCN(C)C)C1 26679,C(=O)(C1=C(C#N)CCC1)N1CCC(C(N2CCC(CN(C)C)C2)=O)(CO)CC1 26680,c1(C(C)(C(=O)NC2CN(C(c3cncc(Cl)c3)=O)C2)N(C)C)ccc(F)c(F)c1 26681,c1(C(=O)NC(C(C)NC(c2nc(C)oc2)=O)C)cccc2c1COCCN2 26682,C1(C(=O)NCCn2cc(C(=O)NCC(=O)OCC#C)nc2)CCSC(C)C1 26683,C(c1cccnc1)=CC(=O)N(C)CC=CC(=O)NC1CC=CCC1 26684,C(CCCCC(=O)N1CC2(C)CC1(C(=O)NC1CCCC1CF)C2)OC 26685,C12(CNC(=O)CCn3ccnn3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26686,C(CN=c1[nH]c2c(c(=NCc3noc4c3CC(F)(F)CC4)[nH]1)SCC2)OC 26687,O=C(Nn1ccnn1)C1(c2ccccc2)CC1 26688,C(=O)(C(CC(C)C)CC(C)C)N1C2(CN(C(C(CC=C)(C)C)=O)CC)CCC1CC2 26689,C=CCC(CNC(=O)COC(C)(C)CNC(C1(c2ccno2)CC1)=O)CC(C)C 26690,C(CC1=CCN(c2ccnc(-c3nccs3)n2)CC1)NC1N(C(C)C)CCC1 26691,Cc1ccc(C(C)(C)C(=O)NC(C)CCCNC(=O)C=CCN(C)C)cc1 26692,Cc1onc(C(=O)NC2CCN(C(c3cnn(CC(F)F)c3C)=O)C2)c1[N+](=O)[O-] 26693,Cc1cc(C(=O)NCC2CN(C(c3ccc(F)nc3)=O)CCC2C)cc(C)c1O 26694,C#CCCCC(=O)N1CCN(C2CN(C(c3ocnc3C)=O)C2)CC1 26695,C(=O)(C(F)(F)C(O)C(C)C)NC1CCN(C(c2cccc(OC)c2N)=O)C1 26696,c1(C(N2C3(CNC(C(C(C)O)C)=O)CCC2CC3)=O)ccc(Cl)c2occc12 26697,N1(C(c2c(OCCCC)c(CC)ncn2)=O)CC(CN)OCC1C 26698,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2ccncc2)C(O)C1 26699,c1(NC(CC(COC)NC(c2cc(C)ccc2I)=O)=O)c(C)cccc1C 26700,C1(C)(C(=O)NC2CCC(NC(C=CC)=O)C2)COC(C)(C)CO1 26701,CCC(C)C(C)C(=O)NCCC1CN(C(=O)C(C#N)CCc2ccccc2)CC1C 26702,C(C1=NOC2CN(C(c3cc(C#N)c[nH]3)=O)CC12)NC(CSC(C)C)=O 26703,CON(Cc1ccccc1)C(=O)C1CCOC1CNC(C1(C#N)CC1(C)C)=O 26704,C(CCCC(=O)N1C2CCC(C2)C1CC(=O)Nc1cc(C2CC2)n(C)n1)(OC)OC 26705,CCC(C)C(C(=O)NC(C)CC(C)NC(c1ccc(COC)cc1)=O)OC 26706,N1(C(CCCCSC(C)(C)C)=O)CC2(C1)C(NC(=O)C(F)F)CCS2(=O)=O 26707,Cc1cccc(C(C)C)c1C(N1CCC(C(C)NC(=O)CC2C=CCC2)C1)=O 26708,CCC(C(=O)NC(CNC(=O)C(C)C[SH](c1ccccc1)(=O)OC)(CC)CC)C(C)C 26709,CCC(C)(C#N)C(=O)NCC1CCCC(C(=O)NCCOCC(C)C)C1 26710,C1(C(=O)NC(C)CN(C(=O)CC2(C)CC2)C)CCCCO1 26711,N1(C(C=C(CC)C)=O)CCN(C(C2C=CCC2)=O)C(c2cncn2C)C1 26712,Cc1cc2cc(C(=O)NCC(C)CNC(C34CC(CF)(CO3)C4)=O)c(Cl)cc2[nH]1 26713,C1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CCCC2)(CO)CC2CCC1CC2 26714,N1(CC)CC(C(=O)N(C)CC2CN(C(=O)CN3C(=O)CCC3=O)C2)CC1=O 26715,c1(C(N2CCN(C(=O)C=Cc3ccc[nH]3)CC2C(F)F)=O)cc2n(n1)CCCC2 26716,C1(C(=O)NCCCCN(C)C(c2coc(C(=O)OC)c2)=O)CC(C(F)(F)F)CO1 26717,CN=S(C)(=O)c1cccc(C(=O)NC2CC(C3CCNC3)C2)c1 26718,N1(C(C(C)N(C(CC2(OCC)CC2)=O)CC)=O)CC(Cl)(Cl)C1 26719,C(C(C)(C)CNC(=O)C(=O)NCC(=O)OC(C)C)NC(COCCC#C)=O 26720,C1(NC(N2CCC(c3n[nH]c(C4CC4)n3)CC2)=O)CNC(C2CC2)CO1 26721,C1(CC(=O)N(CC(C)O)CCNC(C2C(CC)CC2)=O)CC2CCC1N2C 26722,c1(C(C)=O)ccc(Cl)c(NC(C2COCCN2C(C2CC2c2cccs2)=O)=O)c1 26723,N1(C(CCCC#N)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26724,c1(OC2CCN(Cc3ccnc(N4CCOCC4)c3)C2)ccc(F)nc1 26725,c1(C(=O)NC(C)CC2CN(C(=O)CN3CCCC3=O)C2)ccc(CCF)cc1 26726,C#Cc1ccc(C(=O)NC(CNC(c2cccn2C)=O)CC)o1 26727,c1(C(N2CC(N(C(c3nc(CC)oc3C)=O)C)C2)=O)cc(C)nc(O)n1 26728,C1(CNC(Cc2c(C)nccc2)=O)CC2CCC1N2C(C1CC1C)=O 26729,N1(C(C(C=C)O)=O)CCC(C(C)NC(=O)CCn2ccc(C)n2)CC1 26730,S(=O)(=O)(c1cc(C(=O)NC2CC3CN(C(c4ccco4)=O)CC23)co1)NC 26731,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26732,c1(C(N2CC3C(NC(c4cc5n(c4)CCC5)=O)(C3)C2)=O)cc2ccc(Cl)cn2c1 26733,CCC(C)(COC)C(=O)N1CCCC(CNC(c2ccn(C)c2C)=O)CC1 26734,C(C(=O)NOCC(F)F)=C(C)C=C1N(C(=O)CN2CCCC2=O)CC1 26735,C1(C)(COC)CC(NC(c2ccc(N)cc2Cl)=O)CN1C(=O)C(F)=C(C)C 26736,c1(NC(c2c(C)cccn2)C)nc(N(C)CC2CCC(=O)N2)c2ccsc2n1 26737,N1(C(c2cc(C)cnc2OC)C(=O)NCC=C)CCc2n[nH]cc2C1 26738,N1(c2n(CC(=O)OCC)c(C3(C)CCCO3)nn2)CC=C(c2cccs2)CC1 26739,c1(CC2N(C(C(C(C)C)OC(CC)=O)=O)CCC2)cccc([N+](=O)[O-])c1 26740,C1(NC(c2c(CC)oc(C)c2)=O)(CO)CCCN(C(c2csnn2)=O)C1 26741,c1(CC)ncccc1NC(=O)C(C)C(C)NC(C1(COC)CCCCC1)=O 26742,c1(OC(C)(C)C)cc2c(s1)CN(N1CC=CC1)C(C(C)(C)C)C2 26743,c1(OCC(=O)NCC2CC2NC(=O)C(c2ccccc2)C)cccc(NCC)c1 26744,Cc1cc(F)ccc1COC(C1(C(F)F)CCCC1)=O 26745,CC1CCN(N2CCC(N(C(=O)CS(=O)(=O)N3CCN(C)CC3)CC=O)C2)CC1 26746,N1(C(C(CC(C)C)O)=O)CCCCC2C1CCCN2C(c1n[nH]c2c1CSCC2)=O 26747,C=CCC(C)(C)CC(=O)NC(Cc1cn[nH]c1)C(=O)NCCc1noc(=O)n1C 26748,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26749,C(CCC(C(=O)Nc1csc(C)c1)NC(c1cc(C)ccc1F)=O)OC 26750,CCCCCCN(CC(=O)NC1CCC(N(CC)CC)C1)C 26751,N12CC(=CC(C)OCC1=O)C2.CCCCC(=O)CN(C)CC 26752,c1(CNCC23C(CN(C(c4n(C)ccc4I)=O)C2)C3)c(Cl)ccc(Br)c1F 26753,c1(C(N2CC(CNC(Cc3cc(CC)on3)=O)C(C)C2)=O)ccc(N)c(Cl)n1 26754,C(=O)(C1=C(C)CCCC1(C)C)NC(CCNC(c1c(C(=O)OC)cccc1)=O)C 26755,Cc1ccc(C)n1CCNC(=O)CC1(C)CC1(F)F 26756,Cc1c(C(C(=O)NCC(F)F)N(CC(C)C#N)C)cccc1Br 26757,c1(CC)nccnc1C(=O)N(C(C)C(N1CCC(O)C1)=O)C1CC1 26758,C1(CC)CN(C(c2ccnn2C2CCC2)=O)CCC1NC(=O)CC(C)(F)F 26759,N1(C(CCN(C(Cn2ccc(C)n2)=O)CCO)=O)CC2(C)COCC2(C)C1 26760,c1(CN2C(CNC(C(C)C(F)(F)F)=O)CCC2)ccc2c(c1)NCCC2 26761,C#Cc1cncc(C(=O)NCc2csc(CNC(c3csc(C#N)c3)=O)n2)c1 26762,CCC(CC)(CC)C(=O)NCCNC(C)CC(C)C 26763,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26764,C1(NC(C2(CC=C)CCCC2)c2nnnn2C(C)(C)C)CCC2(CC1)CC(O)C2 26765,CCC(C(=O)NCCCN(C(=O)C(C)NC(N)=O)C(C)C)OC 26766,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26767,c1(C(=O)NCC2N(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2)ccccc1C#N 26768,Cc1ccc(CC(=O)N(CC(=O)N(C)C)C(C)C2CC2)o1 26769,c1(C(=O)N)ncsc1N.C1(OCC(=O)OCC)CC(C2CC(COC)C2)C1 26770,N1(C(Cc2ccc(C)nc2)=O)CC2CCN(C(=O)CCc3cnccn3)C2C1C 26771,C(CCCC(=O)NCC(CCF)C(=O)OC)NC(C=CCN(C)CC)=O 26772,N1(c2nnc(C)c(C)n2)CCC(C)C(NC(=O)CCN2CCN(C)CC2)C1C 26773,C1(CC(N2CCC(OC(C)=O)C2)=O)CCN(C(=O)Cc2cnnn2C)CC1 26774,c1(COC2CCCN(C(CNC=O)=O)C2)cccc2cncn12 26775,N1(C(C2C(=C)C2)=O)CC=C(C(=O)NCC2Cc3nccn3C2)CC1 26776,c1(C(=O)NC(C(=O)NC(C2CCOC2)CC)c2cccs2)cccc(CO)n1 26777,c1(CCCCC)cc(C(N2CCCC2C2CN(C(=O)C(F)C3CCC3)C2)=O)n[nH]1 26778,Cc1nc(C=CC(=O)NC2(CCCNC(C3(CS(N)(=O)=O)CCC3)=O)CC2)cs1 26779,C1(C)(C(=O)NCC(CN(C)C(c2csc(-c3ccco3)n2)=O)O)C(C)(C)C1(C)C 26780,C1(C(N(C2CCCNC2=O)C)=O)CCN(C(c2cccs2)=O)C12CC2 26781,C1(C)(CC(=O)NCC2(CC(C)C)CC2)CCN1C(C1(COC)CC1)=O 26782,C1(C(=O)OC)(C(=O)NC(c2ccc(Cl)nc2)(C)C)CC2CC1C2 26783,N1(C(c2cnc(SC)s2)=O)CC2CN(Cc3ccc(C)nc3)C2C1 26784,C1(NC(C=CCNC(c2nc(C)oc2)=O)=O)CCCC1(C)N(C)C 26785,C1(c2nnnn2CCCF)(Nc2ccc(N(C(C)=O)C)nn2)CCCC2(CC2)C1 26786,C1(NC(CN(CC)CC)=O)CCS(=O)(=O)C12CN(C(=O)C=Cc1ccsc1)C2 26787,N1(C(C2(C(=O)OCC)CCC2)=O)CCC(NC(=O)CC2(C)CC2)C(O)C1 26788,CCCCCCCC(=O)NC(CC)CCC(=O)N(C)CC1CCOCC1 26789,C1(C(N2CCC(CCC(=O)NCC(c3nccs3)C)C2)=O)CCCC1C1CC1 26790,CCCCC(CC)C(=O)NC1CCN(C(=O)C(C)(C)c2cccs2)CC1(C)C 26791,N1(C(C(C)NC(CC)=O)=O)CCC12CN(C(=O)C(C)(C)c1cc[nH]n1)C2 26792,O=C1Cc2c(NCC3CCCN3C(c3cc(Cl)c([N+](=O)[O-])[nH]3)=O)ncnc2N1 26793,C1(NC(CCCC)=O)CCN(C(c2ccc(C#N)s2)=O)CC1C 26794,C1(NC(C2C=CCC2)=O)CCC2CN(C(c3n[nH]cc3Cl)=O)CC2C1 26795,C1(NC(C=CCOC)=O)CCN(C(c2cc[nH]c(=N)n2)=O)C1C 26796,c1(C(N2CC(NC(C3CC3(C)C)=O)CC(C)(C)C2)=O)cccc2nc(CO)[nH]c12 26797,N1(C(CC2C(C)CCC2)=O)CCCC(C)(CNC(c2scnc2C(C)(C)C)=O)C1 26798,c1(C(=O)NC(CC)C(O)c2ccccc2)cccnc1NC(N1CCOCC1)=O 26799,N1(C(C2CCN2C2CCC2)=O)CC(F)(F)CC1CNC(C12CCCC(CO1)C2)=O 26800,c1(CN(C)C)cc(C(=O)NC2CC2CNC(=O)C2=COCC2)ccc1F 26801,N1(C(c2c(C(C)C)onc2)=O)CC2CCC1CN2C(c1cccc2nccn12)=O 26802,C1(NC(c2c(OC)csc2)=O)CN(C(C2CSCC(=O)N2)=O)C2CCCC12 26803,N1(C(c2cc(CS(C)(=O)=O)[nH]n2)=O)CC2(NC(=O)CCc3ncc[nH]3)CC1C2 26804,n1(Cc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26805,c1(OC)nc(NC2CC(C(=O)NCC3CCCC3C)C2)nc2[nH]cnc12 26806,C1(C(=O)N(C(C)C(=O)NCc2cc(O)ns2)C2CC2)(CC)CCCCO1 26807,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)Cn2nc(O)ccc2=O)C1 26808,C(N=C(NCc1cccc(C2OCCO2)c1)NCC1CCCO1)c1cnc(C)s1 26809,N1(C(CCC2CCC(=O)N2)=O)CCCC(F)(C(=O)N(C2CC2)CC2CC(CF)C2)C1 26810,N(C1CCOc2ccc(F)cc21)N(c1ccc(C)nc1)C1CC2CNC1C2 26811,NS(=O)(=O)c1ccc(C(N2CCC(CNC(=O)Cc3cc[nH]n3)C23CC3)=O)o1 26812,c1(C(=O)NC(CCN(C(CCCC(C)=O)=O)C)C(C)(C)C)cc2c([nH]1)CCCC2 26813,c1(C(C(=O)NC)N(CC(=O)NC2CC(F)(F)C2)CC)nc(Cl)cc(Cl)c1C 26814,c1(OCCOC)ncccc1C(=O)NC1CCC(NC(=O)C(C)(C)O)CC1 26815,N1(C(C2=NOC(C)C2C)=O)CCC2CC(NC(C3(O)CCOC3)=O)CCC2C1 26816,N1(C(c2c(SC)cn(C)n2)=O)CCC(CC(N)=O)C(CNC(C2OCCO2)=O)C1 26817,c1(OC)cc(Br)c2c(c1)CCN(C(=O)NCC1(OC(C)C)CCOCC1)C2 26818,N1(C(c2cccc(CC)c2)=O)CCC2(CCCN2C(c2ccc(OC)o2)=O)C1 26819,N1(C(c2c(CC)occ2)=O)CC(NC(C23CC(CC)(CO2)C3)=O)C(C(F)(F)F)C1 26820,CCCC(C)(CC)C(=O)NC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC1F 26821,Cc1cc(N)c(C(=O)NCC(C)N(C(=O)C(C)(O)c2ccccc2)C)cc1C 26822,C(CNC(=O)CCN1C(=O)CCC1=O)(CO)(CO)N(C(=O)C=Cc1cncs1)C 26823,N1(C(c2ccc(C(C)=O)cn2)=O)CCC(CNC(=O)C(C)C2CC2)C(F)(F)C1 26824,S(=O)(=O)(c1ccc(C(=O)N(C)C)cc1)NC1CCC(CC)CC1 26825,C1(N(C(C2C(OCC)C2C)=O)CCOC)CCN(C(=O)COC)CC1 26826,C=CCC(CC)C(=O)NC1CC(C)(NC(=O)C(c2ccc(Cl)c(Cl)c2)N(C)C)C1 26827,c1(NCC)ccccc1C(N1CCCC1CC(=O)NC1(C2CCCCO2)CC1)=O 26828,CCCCCCCN(C(=O)CCNC(c1cnc[nH]1)=O)C 26829,N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CC(=O)NCC23CCCC2C3)CC1 26830,c1(C(=O)NCC2CCN(C(Cc3n(C)cnc3)=O)CC2)cccc(C#N)n1 26831,C(C1=NOC2CN(C(=O)Cn3cc(Cl)cn3)CC12)NC(c1cscc1Cl)=O 26832,CC1CCC(=CC(=O)NC(C)(CNC(=O)CCc2ncc[nH]2)C2CCC2)CC1 26833,CCC(CC(=O)NC(C)C(C)(C)NC(C1CCN(C)C(=O)C1)=O)C(C)C 26834,C1(NC(c2c(C)nco2)=O)C2CCCN(C(c3cccc(F)c3C)=O)C2C1(C)C 26835,c1(NC(=O)NCC(C2CC(C)NC2)=O)ccc(N2CCCCC2)cc1 26836,N1(c2c(OC)nnc(-c3ccccc3)c2)CCC2CN(C(C3CC3F)=O)C2C1 26837,N1(C(c2cccc(OCC)c2)=O)CCn2c(C)nnc2C1.N12CCN(C)CC1C2=O 26838,C1(C)(NC(C2(C)N(C(C(C)SC(C)C)=O)CC=C2)=O)CCC(C)=C(C)C1 26839,C1(CNC(=O)COCCCF)CCC2(CCC2)C1.C12CN(CC1F)C2=O 26840,C(=O)(C1CSc2ccccc21)NC1C(C)CN(Cc2cccnc2)C1 26841,C(=O)(C(Cc1ccoc1)NC(=O)C(C)n1cccn1)N(CCN=[N+]=[N-])CC 26842,C(C)(C(N)CC(=O)N1CCCC1CSc1cccs1)OC 26843,N1(C(C(C2CC2)OCC)=O)CC2(CCC(NC(c3ccnn3C(C)C)=O)CC2)C1 26844,N1(C(C(=O)NCC(C)N(C(CSCC=C)=O)C)CC)C(=O)c2ccccc2C1=O 26845,c1(C(N(CCNC(=O)CC2CCC3CC23)C2CC2)=O)ccc(-c2cnccn2)cn1 26846,C(=O)(C1=NOC2(CCC2)C1)NCC(C(C)(C)C)NC(c1cc(O)ccc1Cl)=O 26847,CC(C)(C)C(O)C(=O)N1CCC(OC2CN(C(C3C(C(F)F)C3(C)C)=O)C2)CC1 26848,CC1(C)CC(CNC(=O)CC23COCC(C2)C3)N(C(C2CN(S(C)(=O)=O)C2)=O)C1 26849,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CNC3)CC2)cc1 26850,C1(C(N2CCC(CC(=O)OC)C2)=O)CN(C(=O)C(=O)NCC2CC2)CCO1 26851,c1(CNC(=O)NCC2CCN(c3ncccn3)CC2)coc2c(Cl)cccc12 26852,c1(CC)cc(OC)ccc1C(C(=O)OC)N(CC(C)(C)CNC(C)=O)C 26853,CC1(C)CC(CC(=O)NCCCO)(OC)C1.C(=O)O 26854,C(=O)(C1=C(Cl)CCCC1)NCC(CC)(CC)CO.C12CC(C)CN1C2=O 26855,c1(C(N2C(CNC(C(Br)=C(C)C)=O)CC2)=O)cnc2ncccn12 26856,N1(C(N2CCN(C)CC2)=O)CCc2cc(C(=O)NC3CC3)ccc2C1 26857,c1(C(N2CC(NC(CC(C=C)(C)C)=O)C(O)C2)=O)ccc(C)c(Br)c1N 26858,c1(C(=O)N(CC(C)NCCCOCc2ccncc2)C)cc2ncccn2n1 26859,c1(NC(C2OCCN(C)C2)=O)cc2c(cnn2C)nc1C(F)(F)F 26860,c1(C(=O)NN(C(=O)C=CCF)C)cccc(OCCCCC2CC(CF)C2)c1 26861,N1(C(C(CO)NC(C(C)C)=O)=O)CCCC(C)(NC(C2CCC(=O)NC2=O)=O)C1 26862,N1(C(CCN(C(CCC(C)OCC)=O)C2CC2)=O)CC2CCC2(OC)C1 26863,n1(CC(=O)NCC(C)CNC(c2cc(COC(C)(C)C)on2)=O)cc(Br)cn1 26864,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 26865,N1(C(Cc2c(C)cco2)=O)CC2CCC1C1CN(C(c3occc3F)=O)CC21 26866,c1(C(C(=O)N(CC(O)CNC(C23CCC(C2)C3)=O)C)(C)C)cccc(Cl)c1 26867,C1(C(=O)OC)C(CC(C#C)OC)CCN1C(c1csc(CC)n1)=O 26868,N1(C(c2nnc(C(C)C)o2)=O)CCCC(c2ncc(C(=O)O)[nH]2)C1 26869,N1(C(CCCOc2ccc(CC)cc2)=O)CCC(C2(CO)CC2)CC1 26870,C1(C(N(CCOCCN(C)C(=O)C2CC2)C)=O)CCC(Oc2ccsn2)C1 26871,Cn1c(C(N2CCC(CNC(C3(C)CCNC3=O)=O)C2)=O)nnc1S 26872,C1(C(C)NC(=O)C(F)CC2CCOC2)CCCN(C(=O)C=Cc2ccno2)C1 26873,N1(C(c2nc(C(C)C)sc2)=O)CCCC(NC(C2(CCN(C)C)CC2)=O)C1 26874,C1(C(N2CC3(C2)CN(C(C24CCC2CC4)=O)C3)=O)CC12CCC1(CC1)CC2 26875,c1(C(=O)NC(CC)CNC(=O)COCC2CCOC2)ccnc2c(Br)cccc12 26876,C1(NC(c2cncc(C)c2)=O)COC2(CCN(C(=O)CC34CCCC3C4)CC2)C1 26877,C1(CN(C)C(c2cnc(Cl)s2)=O)CCN(C(C2CCCN2C2CC2)=O)C1 26878,C(=O)(C1CCc2nccn21)NC1C2(OC(C3CCN(C(C)=O)C3)=O)CC2CC1 26879,c1(NC(C2CCC(=O)N2)C)cncc(N2CCCCC2)n1 26880,c1(C(N2CC(C(=O)Nc3ncncc3Cl)C3C2C3)=O)ccc2scnc2c1 26881,c1(C(=O)NC2(CCC(=O)NCCCCC(=O)NC)CCC2)cc(C)nc(C)c1 26882,C(=O)(C(C)C(=O)OC)NCCC(C)CO.C1C(C)=CC(=O)N1C(C)(C)C 26883,c1(C(=O)NCCNC(c2c(C)nc(SC)s2)=O)c(F)c(F)cc(F)c1F 26884,c1(C(=O)NCCC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)nnn(C)c1C 26885,N(C(=NCCF)NC1CCCCC1)C(=O)NCC(=O)NC1(O)CCS(=O)(=O)C1 26886,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2CC2C2CC2)=O)CC1(C)C 26887,C1(CC(=O)NCCCOC(C2C(C)(C)C2(C)C)=O)OC(C)(C)OC1=O.CN1CC1 26888,c1(C(N2CCN(C(COC)=O)CC(CO)C2)=O)ccc2nc(N(C)C)nnc2c1 26889,C(=O)(C1=CSCCO1)NCC1CC(C)N(C(=O)COCC(F)(F)F)C1 26890,C(=O)(C(=O)CC(C)CC)N1CC(c2c(C(=O)NC(CCC)C3CC3)nco2)C1 26891,Cc1c(C(N2CC3C(CNC(=O)CCCc4ccsc4)C3C2)=O)cnn1C(C)C 26892,N1(S(CC)(=O)=O)CCCC1C(=O)NCCCCNC(=O)C=CSc1ccccc1 26893,N1(C(C2CCOC3(CCC3)C2)=O)C2CCC1CC(NC(C1(C3CC3)CC1)=O)C2 26894,CC1CCC(CO)N(C(C2C3CC4C(C3NC(c3cc(O)nn3C)=O)C24)=O)C1 26895,N(C(=NCCc1ccc(Br)cc1)NC1CN(C2CC2)CC1C)C(C#C)CC 26896,CC1C2CCCCC2CN1C(=O)CCCCCN(C(=O)Cc1ccn(C)n1)C 26897,N=c1nc(O)c(C(N2CC(CNC(=O)C#CC(=O)O)C2)=O)c[nH]1 26898,CCCS(=O)(=O)C(C)C(=O)NCCCOCCNC(=O)CN(c1nccn1C)C 26899,C1(NC(c2coc(Sc3ncccn3)n2)=O)CC2CCC1N2C(C1CCSC1)=O 26900,CCC(C)CCC(=O)N(C)CCNC(=O)CC1CC=CCN1C 26901,c1(C(N(CCCNC(c2ccc(C3(O)COC3)cc2)=O)C)=O)cccc(F)c1F 26902,N1(C(C(c2cccc(F)c2)C)=O)CC(C(C)NC(c2n[nH]cc2F)=O)C(C)C1 26903,N1(C(c2c(OC(C)C)nccc2)=O)CCCN(C(c2ccc(=N)[nH]n2)=O)CC1CO 26904,C(=O)(C1=CC2(CCN(C(=O)CC(C)C3CC3)C2)C1)N1CCCC(OC)CC1 26905,C1(C(N2CCC(OCC)C2)=O)N(C(=O)CC2CC(C)(C)C(=O)N2)CCC1(C)C 26906,N1(CCNC2CCCN(C(c3ccc(C#N)cc3)C)C2)CCn2ccnc2C1 26907,C=CCCC(C(=O)NCC(CC)C(N)=O)NC(=O)CCSCC.C(=O)NC 26908,c1(C(N2CCC(C(C)NC(C3CCC(C)O3)=O)CC2)=O)cc(Cl)c2n[nH]cc2c1 26909,Cc1cc(C(=O)NCC2CC3CCC(C2)N3C(=O)C(C)C2CCC2)c(N)c(Cl)n1 26910,c1(NC(=O)C=CC2CC2)cccc(C(F)(F)F)c1.c12nc(cs1)CC(=O)N2CCO 26911,C1(CC)CCC(NC(C2(C)CC(NC(=O)C(C)C3CC3)C2)=O)CC1 26912,c12ccc(cc1)[nH]2.C(C(C)(CN(C)C)OCCNC(C1(OCC)CC1)=O)OC 26913,C1(CCC)CN(C(C2CC2OC)=O)CCN1C(c1ccc(C(O)CF)cc1)=O 26914,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 26915,C(C)(CCCC(=O)NCc1c[nH]nc1C1CC1)NC(COCCC=C)=O 26916,C1(NC(=O)CN2CCCC2)CN(C(c2ccc(C3CC3)nc2O)=O)CC1(F)F 26917,N1(C(c2cc(CCOC)on2)=O)CC2CCC2(CC(=O)NCCC(=O)N(C)C)C1 26918,c1(CCC)onc(C)c1C(=O)NCC1(C)CCN(C(C2(C#N)CCCO2)=O)C1 26919,C=CC1(C(=O)NC2CN(C)CCC2O)CCN(C(=O)C2=NOC(C)C2)CC1 26920,C1(CC)CN(C(=O)Cc2cnc(-c3cccc(C)c3)s2)CC(=O)N1 26921,CC1CC(C)CC2(C1)NC(=O)N(CC(=O)NC1CC3CC1C(O)C3O)C2=O 26922,Cn1cc(C(N2CC(OC)CC(NC(=O)CCNC(=O)CO)C2)=O)ccc1=O 26923,c1(C(N2CCC3CN(C(C4CCCS(=O)(=O)C4)=O)CC23)=O)cccc2c[nH]nc12 26924,CN=c1[nH]c(=NCCOCC(C)C)[nH]c(=NCCc2cn(C)c3ncccc23)[nH]1 26925,c1(-n2cc(C(C3CCOC3)OC)nn2)ccc(C)cc1NCCn1ccccc1=O 26926,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CCCC2C3)=O)CC1 26927,Cc1cccn2ncc(C(=O)NCC3CCC4(CO3)CC(NC(=O)C(C)C)C4)c12 26928,C1(C(=O)NCC2CC(NC(C(C)OC)=O)C2)CC2CCC1O2 26929,c1(CCC(=O)NCCSCc2nc(-c3ccns3)no2)cnc2n1CCCC2 26930,C1(CC(=O)NCC(=O)NCC#C)CCCN(C(=O)CC(=O)OCCC=C)CC1 26931,CN1CC(F)CC1C(=O)NCC1CCC(NC(=O)C=CC2CCC2)C1 26932,C1(C)(C(=O)NCc2n(C)cnc2)CCCN(Cc2cccc(Br)c2I)C1 26933,C1(CNC(COCCOCC#C)=O)CCCN1C(=O)CC1C=CCCC1 26934,c1(C(=O)NCC(CNC(C2(C#N)CCOCC2)=O)F)ccc2nnnn2c1 26935,C1(C(=O)NCC(CNC(C2(CC=C)CCCCC2)=O)OC)CCC(C)(C)CO1 26936,C1(C(=O)NCCC(CNC(c2csnn2)=O)O)CCCCC(=O)N1 26937,c1(COC(C2CCC(C(F)F)CC2)=O)nnn2c1COCC2 26938,C(=O)(C1=NOCC1)NC1CC(N(C(C(CC)OCc2ccccc2C)=O)C)C1 26939,C(C(CC1CC1)C(=O)NCC1CC1Cl)NC(C(CC)n1cncn1)=O 26940,c1(OCC)ccc(C(=O)NCc2cc(C(N3CC=CC3)=O)cs2)cc1 26941,C1(NC(C(N(C(=O)CCc2cnoc2)C)C2CC2)=O)CCc2nncn2C1 26942,C1(CC)(NC(=O)C(Cn2cncn2)NC(=O)CC2CC3(CC3)C2)CCCC1 26943,c1(OC)cc(C(=O)Nc2cccc(F)c2C(N)=O)cc(O)c1O.C12CC1C(=O)N2 26944,C(=O)(C(C1CCCC1)NC(=O)CCNC(=O)C=CCl)OCC 26945,Cn1nc(Br)cc1CC(=O)N(CC(F)F)C1CCC1 26946,N1(C(CC(CC)C)=O)CC(C)CN(C(c2sc(C)cc2Br)=O)CC1C 26947,C12(CNC(C(Cc3ccoc3)NC(=O)CC34CCCC3C4)=O)CCC(CC1)O2 26948,C(=O)(CCC(=O)c1ccc(Br)cc1)NC(C)CNC(=O)CC1COCCO1 26949,N1(C(C(C=C)CC)=O)CC2(C=C(C(=O)NCC3CC(OC)C3)CO2)C1 26950,N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCC2(CC3CC3)CC2)CCC1(C)C 26951,C(=O)(CC(CC)C(C)(C)C)NCC1(COC)CCCN1C(c1coc(Br)c1)=O 26952,C(CC(C)(C)C(=O)NCc1cnns1)N(CC(=O)NC(C(C)C)C1CCC1)C 26953,S(=O)(=O)(c1cc(F)cc(F)c1)NC1CN(C(=O)CCCCBr)CC1F 26954,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC#C)CC#C)=O)C(C)(C)C1 26955,C(C1=CCN(C(C2CCC3(CC2)CC3)=O)CC1)N(CC=C)C(C)=O 26956,c1(OC)cc(CN=c2cc(CC(N3CCSCC3)=O)nc[nH]2)c(F)c(F)c1F 26957,C1(Nc2ncc(Br)cn2)CC(O)CN1C(C1CCC(c2cn(CC)nn2)CC1)=O 26958,n1(CC(=O)N(CCCCN(C(=O)CCP(C)(C)=O)C)C)nc2c(n1)CCCC2 26959,C1(CNC(C2CC2F)=O)CN(C(C2CCN(C(C(C)(C)OC)=O)CC2)=O)CCCO1 26960,c1(N2C(C3(NC(C4C(C)CC(=O)N4)=O)CC3)CCC2)nc(Cl)ncc1C1CC1 26961,c1(C(N2C(C(=O)NCCn3c(O)nnc3O)C=CCC2)=O)n[nH]cc1[N+](=O)[O-] 26962,CN1CC2CCC(C1)N2C(=O)CC1CCN1C(=O)C(F)F 26963,CC1(Oc2ncccn2)CC(NC(=O)CN(C2CC2)CCF)C1 26964,N1(C(C(C)S)=O)CCN(Cc2sc(Br)nc2Br)CC1CC#N 26965,C1(C(=O)NCCCNC(c2ccc(C(CC)(C)C)cc2)=O)CN2CCN1CC2C 26966,N1(C(c2n[nH]c(C)c2O)=O)CCC2CN(C(=O)CCc3nc(C(C)C)no3)C2C1 26967,Cn1c(=O)n(C)c2cc(C(N)=O)ccc12.C12CC3(CCC(CC3)N1)C2 26968,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCCC(CF)C1)c1c(C)c(Cl)c(Cl)cc1 26969,c1(OCC(=O)NC(C2CCN(C(C(CC)F)=O)C2)C)ccc([N+](=O)[O-])cc1 26970,c1(C(=O)NC2CN(C(C3COCC(C)O3)=O)C2)cc(Br)cnc1N(C)C 26971,N1(C(CC2C(C)OCC2)=O)CCOCCC1C(=O)Nc1cnc(Cl)nc1 26972,CCC(F)(F)CC(=O)N1CCC(C)C(NC(=O)Cn2cnnn2)C1 26973,C(CNC(=O)CCn1cccnc1=O)(C(C)(C)C)NC(C(CSC)OC)=O 26974,c1(C(N(C2CCCCN(C(C3CC3C#N)=O)C2)C)=O)cc2cn[nH]c2cn1 26975,C1(NC(C2CCC(CC)O2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 26976,C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCc2nc[nH]n2)CC1O 26977,N1(C(C2CC(OC(C)(C)C)C2)=O)CCC(F)(CNC(=O)CN2CCCOC2=O)C1 26978,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 26979,C1(COC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)CSc1nncn1C 26980,N1(C(Cn2cc(C(C)O)nn2)=O)CCCC(CO)(NC(c2ccc(Cl)s2)=O)C1 26981,C1(C(N2CC(O)(CCC)C2)=O)CCN(C(=O)CCN=[N+]=[N-])C(C)(C)C1 26982,N1(CC#N)CCCC(C2CCN(C(C3CC34CCOC4)=O)CC2)C1 26983,N1(C(C(C(C)C)SCC)=O)CC2CC(NC(c3c(C)cnn3C)=O)C1C2 26984,N1(C(CCOCC)=O)CCOC(CCNC(c2cccc(Cl)c2)=O)C1 26985,Cc1nc(N)cnc1C(=O)NCCCNC(c1cn(C)c(C(F)F)n1)=O 26986,N1(C(CN(c2ccc(Cl)nn2)C)=O)CC2CC(NC(c3cn(C)nn3)=O)CC2C1 26987,C(CC(C)(C)C)(C(=O)NC1(CNC(c2ccc(F)c(C(F)(F)F)c2)=O)CC1)OC 26988,O=C1CCN(CC(O)COC2CC(O)CC2O)CC1 26989,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 26990,C(C(C)C(=O)NOCC1CCOCC1)NC(C(COC)(C)OC)=O 26991,CC(=O)CCCC(=O)NCCCN(C(C1CC(C)(C)CCO1)=O)C1CC1 26992,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 26993,N1(C(CCOCC#C)=O)CCC(O)(C(C)CNC(C2(NC(C)C)CCCC2)=O)C1 26994,c1(C(N2CC(CCNC(C3CC(C)OC3)=O)C2)=O)cc2cc(Cl)ccc2o1 26995,c1(NC(=O)NC2CN(C(C(C)O)=O)C2)c(F)cccc1C#N 26996,c1(C(N2CCC(CNC(C3CCC(C)(C)C3)=O)CC2)=O)cc(N)ccc1[N+](=O)[O-] 26997,C(=O)(C1=CC2(CCOC2)C1)N(C(=O)CC(O)C(Cl)(Cl)Cl)CCC1CN2CCC1CC2 26998,c1(C(N2C(CCCNC(c3ccno3)=O)CCC2)=O)cnc(C(F)(F)F)cn1 26999,Cc1c(-c2cccnc2C(N2CCC(C(N)=O)C2)=O)c(CO)nn1C 27000,N1(C(CCC(C)(F)F)=O)CC(NC(=O)CS(=O)(=O)C2CC2)CC12CCC2 27001,n1(CC(=O)NCCC2CCCN2C(=O)CCC2CC2)ccc(O)nc1=O 27002,N1(C(c2c(C)cc(C)o2)=O)CCC(CO)C(NC(=O)C(O)C2CCCC2)C1 27003,C1(C(=O)NC23CN(C(c4cnn(C)c4N)=O)C(CC2)C3)CCCCCC1(F)F 27004,c1(C(N(C2CCCN(C(c3ccccc3CO)=O)CC2)C)=O)cccn(C)c1=O 27005,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27006,N1(C(CC(CC)C)=O)CCC(CNC(=O)C#CC2(C(F)(F)F)CC2)C12CC2 27007,N#Cc1ccsc1C(N1CCC(NC(=O)C(O)c2ccsc2)C1)=O 27008,CCC(C(=O)NCC12CC(NC(=O)C(F)OC)(C1)C2)n1ccnc1 27009,c1(C(=O)NCC2N(C(C(C)(C)c3cnsc3)=O)CC2)cc(OC(F)F)nc(Cl)c1 27010,Cc1cc(C)c(CNC(=O)CC2COCCN2c2ncc3ccsc3n2)c(C)c1 27011,Cc1ccc(CNC2C(c3ccccc3)CCN2C(=O)OC(C)(C)C)c(O)c1C 27012,c1(CC)nc(NCCC(C)NC(C2CN(C)CC(C)O2)=O)c(C#N)cc1C 27013,C1(CNC(=O)CC2CCC(NC(c3cccc[n+]3[O-])=O)C2)CCCC2(CC2)C1 27014,C1(NC(CCSCCC)=O)CC2CCC1CC2NC(c1csc2nccn12)=O 27015,c1(C(=O)OC)oc2cccnc2c1NCc1cccc(C(C)(C)C)c1.C1(=O)CO1 27016,N1(CCNS(N)(=O)=O)CC2(CCCN2C(C23CC2CNC3=O)=O)C1 27017,C1(CNC(C2CCCC2)=O)CCCN1Cc1ccc(Cl)o1 27018,c1(CCC(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27019,C1(F)(C(=O)NCCc2onc(C)n2)CCCN(C(=O)C=C2CCC2)C1 27020,Cc1c(O)ccc(C(N2CCCC(CN(C)C(C3(C(C)C)CCC3)=O)C2)=O)c1C 27021,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1CC1C(F)(F)F)=O 27022,C(=O)(C1=CC2C=CC1C2)N1CCN(C(C2N(C(C)=O)CCC2)=O)C(CO)C1 27023,C(=O)(CC1OCc2ccccc21)N1C2CN(C(=O)CC(F)(F)C(F)(F)F)C(C2)C1 27024,C1(C(=O)NC2(C)CCN(N3CC4CCCC(C3)N4)C2)C2Cc3c(Cl)cccc3C12 27025,C1(C)(C(N2OCC(=C)C2)=O)CN(C(=O)CCC(C)OC)C(C)(C)C1 27026,CC1CN(C(=O)C(C)Cc2cccc(F)c2)CCC1CNC(=O)C1=C(Cl)CC1 27027,CC1CC(N(C)C(C2CSCCN2C(=O)CCN2CCOCC2)=O)CC(C)C1 27028,N1(C(C(COC(N(C)CCOCCN(C)CC)=O)C)=O)CCN2CC(F)CC2C1.CO 27029,c1(-c2cccc(OC)c2CO)cnc2c(C(=O)O)c[nH]c2c1 27030,CC1(C)CC(C(N2CCC(C3(C)CC3)C2)=O)CN(C(=O)CC2(C)CCCCC2)C1 27031,Cc1cccc(C(C)NC(C2CC2c2ccccc2-c2cncn2C)=O)n1 27032,c1(CN2CC3(C(C(=O)OCC)C3)C2)cc(Br)c(F)cc1Cl 27033,C(=O)(CCS(C)(=O)=O)NCC(C(=O)NC(C#C)C(C)OC)(C)C 27034,c1(C(N2CCC(CNC(CC(CC)C3CC3)=O)C2)=O)cc2ccccc2n1CC 27035,C(C(O)C(=O)N1CCC(N(C(=O)C(C)(C)O)CCO)C1)SC 27036,c1(C(CC)N)nnc(N2N3CCC(C3)N3CCC2C3)n1COC.c1(SC)cccs1 27037,C1(NC(c2scc(C)c2C)=O)CCCC12CN(C(C13CCC(C)(CC1)OC3)=O)C2 27038,C=CC1CCN(C(C2CCN(C(c3cc(C)nc(O)c3)=O)C2)=O)CC1 27039,N1(C(c2cc(SC)c(C)o2)=O)CCC2CN(C(C3CC(N(C)C)C3)=O)CCC2C1 27040,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27041,c1(C(=O)NCC(C(=O)N(C(C=C)C)C)(C)CC)cn2ccccc2n1 27042,C12(CC(=O)N(CC(CN(C)C)O)C)CCC1CN(C(c1csc(Cl)c1)=O)C2 27043,c1(CN2CCCC(C(C)NC(c3ccc(I)c(F)c3)=O)C2)cccc2ncsc12 27044,C1(CO)C2CCCC(F)(F)C12.CCC1(C)CNC(=O)NC1 27045,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27046,N1(C(C(CCNC(C(C)OCC)=O)O)=O)CCCCC(C)(F)C1 27047,c1(CN(C(c2cc[nH]n2)=O)C(C2CCN(C(C)C)C2)=O)cc(F)cc([N+](=O)[O-])c1 27048,C12(CNC(CCCNC(=O)OC)=O)CCC1CCN2C(=O)C(C)Cc1cnco1 27049,C1(N(C(CCN(C)CC)=O)C)CN(C(=O)C(N2CCN(C)CC2)C)CCC1C 27050,CC1COc2ccc(C(N3CCC(NC(c4ncc[nH]c4=O)=O)C3)=O)cc21 27051,CCC(CNC1CC(OCCN(C)C)(OC)C1)CCC1CCCC1 27052,N1(C(C2N(C(CC(=O)OC)=O)CCC2CC#C)=O)CC(C2CCCC2)C1 27053,C(C)(C)(CC(C)NC(=O)C=CCC1(NC(=O)C=Cc2cc[nH]n2)CCC1)OC 27054,c1(C(=O)NCC2(F)CC(NC(C(CCC)OC)=O)C2)ccc(C(C)C)nc1O 27055,c1(CNC(C2(C)C(C)(C)C2)=O)nnc2n1CCN(C(c1ccc(Cl)c(N)c1)=O)C2 27056,Cc1sc(C(=O)N(CCCCNC(=O)C(C23CCC(CC2)C3)N(C)C)C)nc1O 27057,c1(C(=O)NCC(C)CNC(C2CCCOCC2)=O)ccc2c(c1)CCCC(=O)N2 27058,C1(CS(=O)(=O)NCC(=O)OC)CCCOC1c1cn(-c2ncccc2Br)nn1 27059,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)c2)=O)CCC1 27060,Cc1cc(O)cc2c1CN(C(C1CC1C(=O)Nc1cccc(Br)c1)=O)CC2 27061,c1(CCC(=O)NC(C)CNC(=O)CCc2ncccn2)nc2cc(Cl)ccc2s1 27062,n1(CCC)cc(C(=O)NC2CC(N(C(=O)Cc3cccn3C)C)C2)c(C)n1 27063,C1(C#N)(COC)CCN(C(=O)Nc2cc(C3CCCN3C)[nH]n2)CC1 27064,c1(OC)cccc2c1CN(N1CCC(CCSC)CC1)C2 27065,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27066,c1(C(N(CCNC(c2n(CC)c(O)nc2)=O)CC2CC2)=O)sc(C)c(Br)c1C 27067,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27068,c1(C(=O)NCC(C2CCOC2=O)NC(C(C)(C)OCC)=O)c(C)ccc(C)c1C 27069,c1(C(=O)NC2CCN(C(c3c(C(C)C)ccs3)=O)C2)cc2c(cn1)OCCC2 27070,C1(NC(c2cn(C(C)C)nn2)=O)(CO)CCCN(C(=O)CCn2cnnn2)C1 27071,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(C1CCC(C)O1)=O 27072,N12CCC(F)(F)C(C1)C(=O)N(C13CC(C1)C3)C2=O.CCCCCC=CC(=O)O 27073,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27074,N1(C(C(COC)C)=O)CCCCCC(NC(c2cc(C)cnc2C)=O)C1 27075,c1(C(=O)NC2CCCN(C(c3c(C)occ3)=O)C2)ccc2c(c1)N(C)C(=O)CO2 27076,C(C(N=[N+]=[N-])C(=O)NC1CCN(S(=O)(=O)C(F)F)CC1)OCC 27077,N(C(=NCCc1ccccc1F)NCC1=CCCOC1)CC1(C)CCC1 27078,C1(C)(CNC(c2c(C)nco2)=O)CCN(C(=O)CSCc2cccnc2)CC1 27079,C(C(C(C)C(C)C)NC(=O)COCCF)NC(c1c(CCC)nsc1N)=O 27080,C1(NC(C(C)NS(CC)(=O)=O)=O)(CO)CCN(C(c2c[nH]nc2CC2CC2)=O)C1 27081,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)CC)NCC 27082,c1(C(c2ccccn2)N(C)C(=O)NCC2CCC3CC23)ccccc1 27083,C(C(CC(C)C)C(=O)N(C12CC(C1)C2)C)NC(c1n(C=C)ncc1)=O 27084,CCC(CC(=O)NCC1COCCN(C(=O)C(F)C2CCCC2)C1)CC(C)C 27085,CCC(C)(C)CCCC(=O)NC1CCN(C(=O)C(N(C)C)OC)CC1O 27086,O=C1NC2COCC(CNCC3(C(F)(F)F)CC3)N2C(=O)N1 27087,Cc1cc(C)c(C(=O)NCC(C)C(=O)NC2CSCSC2)s1 27088,C1(OC)(CNC(=O)C(Cc2ccccc2)C2CC2)CN(C(=O)CC2(C)CCC2)C1 27089,C1(CNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27090,C(=O)(C#CC(C)(C)C)N1CCC(C(C)NC(c2ccccc2-n2cccn2)=O)C1 27091,c1(C(=O)NC(C)(C)C)cn(CC(C2(O)CN(C(=O)CC3CCCO3)C2)F)nn1 27092,C1(NC(Cc2ccc(C)cc2Cl)=O)CN(C(C2CCSC2)=O)CC12CCCC2 27093,Cc1ncc(-c2ccco2)n1CC(=O)NC1CCCNC1=O 27094,c1(N2CCC(OCC)C(C)C2)nc(=NCc2cc[nH]c(=N)c2)[nH]c2c(C)nn(C)c12 27095,CCCCC(F)(F)C(=O)NCCC1CCCN1C(=O)CCC1CNC(=O)N1 27096,C(CC(C)C(=O)NCc1ocnc1C(=O)NCCCC1CCC1)OC(C)=O 27097,c1(N(C)CC2CCC2)nc(=NCC2NC(=O)CC2(C)C)[nH]c2c(F)cc(F)cc12 27098,C1(c2onc(Cc3n(C)ccn3)n2)CC12CC(O)C2 27099,c1(CC)cc(CC)nc(N2CCC(C)(NC(=O)C(N3CCOCC3)C)CC2)n1 27100,N1(C(CN(C)CC)=O)CC2CCC(CNC(C3CC3(C(C)C)CC)=O)(C2)C1 27101,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)N(C)C)C1)=O 27102,C1(C(C)CNC(C2CCC[SH]2C)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1 27103,C12(C(N3CC(C)(NC(Cc4ccc(C)o4)=O)C3)=O)CC3CC1C2C3 27104,C1(NC(c2nc3c(s2)CCC3)=O)CCN(c2nnc(O)s2)CC1O 27105,c1(C(=O)NCCOCCC(=O)NCc2n[nH]cc2C2CC2)cnccn1 27106,C(=O)(CC(C(C)(C)C)NC(c1cc(F)ccc1F)=O)NCc1c(C)scn1 27107,N1(CC=C)CCN(CCN(C2CCNC2)C(c2nnsc2C)=O)CC1 27108,N1(C(C(C)Cn2cccn2)=O)CCCC(C(N2CCC(C(F)F)CC2)=O)CC1 27109,Cc1nn(C(C)C)cc1C(=O)NCCCC1(NC(=O)C(C)c2ccsc2)CC1 27110,C(=O)(CCC(=O)N(CCCOCCN(C(=O)CCCC1CCCO1)C)C)N(C)C 27111,CCCCCC(C)CC(=O)NCc1cc(C(=O)N(c2cccc(C)c2C)C)cs1 27112,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)OC(C)C)C(C)C 27113,N1(Cc2ccc(OCC(C)C)cc2)C2CCC1(CNC(=O)CC1(O)CCC1)CC2 27114,c1(C(=O)NC2CCCN(C(CC3(C)OCCO3)=O)C2)cc2ccncc2s1 27115,c1(OC)ccc(C(N2CCN(C(c3c[nH]c(Br)c3)=O)C(C)C2)=O)cc1F 27116,CCC(CCC(=O)NCC1CC(O)C1)NC(c1nc(CC)oc1C)=O 27117,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27118,N1(C(CCC(C)(C)C)=O)CCOCC(C)(CNC(C2COCC2(C)C)=O)C1 27119,Cc1cnc(O)c(CNC(C2CCC(C)N2C(=O)Cc2cccc(C)n2)=O)c1 27120,C12(NC(CCC(CC)OC)=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2 27121,N1(C(C(C)n2ccnc2)=O)CC2CC2(NC(=O)CCC2CC2)C1 27122,CC(c1ccccc1)=CC(=O)NCC1(NC(C2CC3CC2C2CC32)=O)CCOC1 27123,c1(C(=O)NCC(CC(=O)NCCC2CCC(C)(C)C2)OC)cccc(F)c1C 27124,C1(NC(C(N2CC(c3scc(C)n3)C2)=O)=O)CCCN(C)C1 27125,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27126,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27127,C=CCCCCCC(=O)N1CCCC(C(C(=O)OC)NC(C(C)CC)=O)C1 27128,c1(C2C(CC(C)(C)C)C2)cc2c(s1)CCOC2.C12CC3C1CCN3NC2=O 27129,C1(C(=O)NC2C(CNc3nc(C)c(F)cn3)CCCC2)CCc2ccccc2N1 27130,C(=O)(C1=NOC(C)C1C)NCC1CCN(C(c2sc(C)c(C)c2C)=O)C12CC2 27131,N1(C(c2c(C)ncnc2)=O)CCc2[nH]nc(CN(C)Cc3cccnc3)c2C1 27132,C1(C(=O)NCC(CC(F)(F)F)NC(COCC=C)=O)CS(=O)(=O)CC12CC2 27133,c1(CNC(=O)C(N2CCC3(C2)OCCO3)=O)cccc2ccnn12 27134,N1(C(C2(C)CN(C(C34CC(F)(C3)C4)=O)C2)=O)CCN2C(=O)CCC2C1 27135,C#Cc1cncc(CN2CCN(C(=O)CCN3CCCCC3C)C(CC)C2)c1 27136,N1(C(CCOCC#C)=O)CCC(C)C(NC(c2ccc(NC(C)=O)cc2C)=O)C1 27137,c1(SC)ccc(C(=O)NC(C(c2ccc(N(C)C)cc2)=O)C(C)C)cc1[N+](=O)[O-] 27138,C(=O)(CC1=CCOCC1)N(C)CCOCCCNC(C1CC1[N+](=O)[O-])=O 27139,CC(C)CCCC(C)CNC(=O)C(C)CNC(C1CN(C(N)=O)C1)=O 27140,c1(C(N)=O)ccc(N2CCN(C(=O)C(=O)NCC(F)(F)Cl)CC2)c(F)c1 27141,c1(CC(=O)NCC2(CN(C(=O)CCc3ccsc3)C)CC2)cn2ccccc2n1 27142,C(=O)(C(F)(F)c1cscn1)NC(C)CN(C(=O)CC1(n2ccnc2)CC1)C1CC1 27143,N1(C(CC2N(C(=O)CSc3cccs3)CCOC2)=O)CCCC(O)(C(C)C)C1 27144,C(=O)(C(C)C(C)(C)O)Nc1cc(OC)c(-c2nccn2-c2cscc2Br)s1 27145,c1(C(N2CC(CNC(C3(C(F)(F)F)CCO3)=O)C3CC23)=O)cccc2nncn12 27146,c1(C(=O)NCc2cccc(CN(C(=O)CCF)C)c2)n[nH]cc1[N+](=O)[O-] 27147,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27148,c1(NC(CN(C(C2CCN(OC)CC2)=O)C)=O)ccc2c(c1)OCCO2 27149,c1(SCN2C(C)C2)ccccc1.c1(C(NOC(C2CC2)=O)=O)cnccn1 27150,C1(CNC(CCC=C(C)C)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CC2(CCC2)O1 27151,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cn2cnc(C(N)=O)n2)C(O)C1 27152,C(CC(F)F)(C(=O)N(C)Cc1ccccc1F)NC(C1C(C)SCCC1)=O 27153,N1(C(C)CN(C2CCCC2)C(c2ccoc2C2CC2)=O)C(C)CCC1C 27154,CC(C(CO)NC(c1cn(C2CCOC2)nn1)=O)NC(=O)Cc1cnco1 27155,c1(C(=O)NCC2N(C(CCCCC#C)=O)CC3(CC3)C2)ccc2nc(Cl)cn2c1 27156,C1(NC(=O)CCN2CCCC2)CCSC12CN(C(c1ccc(O)c(F)c1)=O)C2 27157,CCCCCC(CC)C(=O)NCC(C)N(C(=O)CCCc1cncs1)CC 27158,c1(CNC(=O)CNC(=O)COCCF)cc(Cl)cnn1 27159,C1(NC(=O)OCCCNC(CC(CC)OC)=O)CCC2(CCC2)CC1 27160,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C)cc(F)c2)=O)cc1C1CC1 27161,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27162,Cc1noc(CC(C)C)c1C(=O)NCC(C1(O)CCN(C(=O)COC(C)C)C1)C 27163,c1(C(=O)NC(C(C)NC(c2cc(N)cnc2Cl)=O)C)ccc(Cl)c2ccccc12 27164,C12(C(NOCCCC=C)=O)CCCC1CCN2C(=O)CC(C)(C)C=C 27165,N1(C(C2(S(C)(=O)=O)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccc(Cl)cn2)C1 27166,CC1CN(C(=O)C2=COCCC2)CC(C(=O)NC2(C)CC(O)C2)O1 27167,c1(CN(C(c2noc3c2CCC3)C(=O)NC2CCCCC2)C)ccc2cccnc2c1 27168,C(CCCCCO)N(CCC(N1CCCC1C(C)(C)CO)=O)CCCOC 27169,c1(C(N(CC(C)NC(c2snnc2C2CC2)=O)C)=O)nnn2c1COCC2 27170,C(=O)(CCCCC(=O)N1CC(CNC(=O)C(C)(O)C2CC2)C(F)(CO)C1)NC 27171,CC1CCN(C(c2nc(=N)cc[nH]2)=O)CC1CNC(=O)CC12COC(C)(C1)C2 27172,CC(C)C(CNC(=O)Cn1cnc(=N)[nH]1)C(=O)NC1(C)CCC(C)(C)C1 27173,CC#CCCCC(=O)N1CC(C(N2CCC=CC2C(=O)OC)=O)C(F)(F)C1 27174,c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1coc(SC)c1)=O)C2 27175,C1(C)(CNC(C2(C)C(C)CCC2)=O)CCCN(C(c2ccc(F)s2)=O)C1 27176,C1(C(=O)NC2CCN(C(C(C)Cn3cccn3)=O)CC2)CCc2nncn2CC1 27177,CCCCC(C)CCC(=O)N1CCC1CNC(C1(CCCC)CCCC1)=O 27178,c1(OC)cccnc1C(=O)NC1(C)CC(NC(=O)CCC2CCOC2)C1 27179,c1(C(N(CC(=O)OC)C2CC2)=O)c(CC)cnn1CC.C1(O)(C(C=O)F)CCCC1 27180,Cc1ccc(-c2ccc3occc3c2)c2nc(C(=O)NCCC(C)CO)cn12 27181,C(C)(C)(CC(=O)N1CCCC(C(=O)NC2(C(N)=O)CCC2)C1)OC 27182,C(=O)(C1=COCCO1)N(CCCC(C)O)CCNC(=O)CCC(=O)N(C)C 27183,C(=O)(CC(C(F)F)NC(c1ccc(F)nc1)=O)N1C(C)(COC)C=CC1 27184,c1(C(=O)NCC(CCOC)(C)C)cc(O)nc(C(C)C)n1 27185,C1(CC)CN(C(c2cc(C)oc2C)=O)CCC1NC(c1cnn(CC(C)C)c1)=O 27186,Cc1ncnc(C)c1OCC(=O)NCC12CC1CN(C(=O)CN(C)C1CC1)C2 27187,c1(N2CCCC(CNC(c3c(F)cccc3Cl)=O)C2)ncnc2cccnc12 27188,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27189,N1(C(c2n(C)nnc2)=O)CCC(CO)(NC(=O)CCCC2CCC2)CC1 27190,CCCC(C)(C)C(=O)N1CCC(C)(NC(=O)CN2CC3CCC2C3)C1 27191,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc[nH]n1)=O)C2 27192,C#Cc1cccc(C(=O)N(CCNC(=O)C(C)(C)C(N)=O)CC)c1 27193,C#Cc1cn(C)nc1C(N1CC(NC(=O)CC2CC3CC(=O)C2C3)CC(O)C1)=O 27194,C(=O)(CCC(=O)c1ccncc1)N1CC(OCCN(C)C(C2CCNC2=O)=O)C1 27195,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27196,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27197,C(CC#C)(CC(=O)N1CCSC(C)CC1)OCCCC#C.C1C(=O)NCCN1CC 27198,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(C#C)C1CCC1)C1CCCO1 27199,Cc1ccccc1OCCC(=O)NC(c1nccs1)C1CCC1 27200,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)Cc3cccc(C(F)F)c3)C2)o1 27201,c1(OC(C)C)ncccc1-c1nc(N(S(C)(=O)=O)Cc2cccs2)cs1 27202,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27203,C1(C(=O)NC2(CC#C)CN(C(C3(CC4CC4)CCC3)=O)C2)CCCC(O)C1 27204,c1(C(N(C2C(N(C(C=C(COC)C)=O)C)CCCC2)C)=O)cnc2sccn12 27205,N1(CC(N)=O)CCN(C(=O)C(=O)NCCCN2CCSCC2)CC1 27206,CC(C)C(C(=O)Nc1cncc(C#N)c1)C(C)NC(C1CC(O)C1)=O 27207,C1(C(=O)NC2CC3CC(NC(C4=CC(C)(C)C4)=O)C3C2)COc2ccccc2C1 27208,C(=O)(C(C)CCCOCC)NC(CNC(C(CCC)OCC)=O)C1CCC1 27209,N1(CC)CCOC(c2ccc(OC)cc2)C1.C12(COCCN1)C(=O)NC2 27210,C1(CC(N2CCC(C(CC)CC)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27211,Cc1c(C(=O)NCC(C(C)C)NC(=O)COC(F)F)cnn1CCC(C)C 27212,CC(C)CCC(CO)NC(=O)CCCCc1nc(CC(=O)C2=CCCCO2)no1 27213,c1(C(N(CC(C)(C)CNC(C2(n3ccnc3)CCCC2)=O)C)=O)cc(C)cc(O)c1 27214,c1(C(=O)NC(CNC(C=C(CC)CC)=O)(C)C2CC2)nc(CC)cn1C(=O)O 27215,N1(C(c2cn(CC=C)nc2)=O)CC(NC(c2onc(CC)c2C)=O)CC1CC=C 27216,COn1cnc(C)c1C(=O)NC(CCN(C)C)C(=O)NC1CCC1(C)C 27217,C1(C)(C(=O)NCCC(C)N(C(=O)COc2ccccc2F)C)COCCO1 27218,CC1(C(=O)NCCn2cnnn2)CC(O)CN1C(=O)Cc1nc[nH]n1 27219,Cc1cccc2c(CC(=O)NC3CC4CC3N(C(=O)C3=CCC3)C4)c[nH]c12 27220,c1(CNC(=O)CCCn2cccn2)n[nH]c2ccccc12.C12CCCCN1C2 27221,c1(NC(C2CC23CN(Cc2ccc(O)c(Cl)c2)C3)=O)ccc2cc[nH]c2c1 27222,C1(C)(CNC(c2ccc(C#C)nc2)=O)CC(F)(F)CN1C(C1CCCNC1=O)=O 27223,c1(OC)ncccc1C1(O)CCN(C(=O)C(=O)NCc2nc(C(=O)O)co2)C1 27224,C1(N(C)C(c2ccc(C(F)F)nc2)=O)CCN(C(C2(CO)CCCO2)=O)CC1 27225,C1(N(C(=O)CC2CCCC2)CC)CCCN(C(c2oncc2CC)=O)C1 27226,N1(C(CCN(C(C(C)(C)NC(C)=O)=O)C)=O)CCC(CO)C(C)(C)C1 27227,C(C)(C)(CCC(=O)Nc1ccccc1F)ONC(C1CCN(C)C1)=O 27228,N#Cc1ccc(S(N)(=O)=O)cc1CN1CCC(c2cc(-c3ccco3)n[nH]2)CC1 27229,C1(O)(CCSC)CCCN(C(C2(N(C)C)CCC2)=O)C1.C12(CC1)CC(=O)NC2 27230,n1(CC)cnc(C(=O)NCC(C)(C)NC(=O)CNC(=O)C2CC2)n1 27231,C(C1CCCCCC1)=CC(=O)NCC1N(C(c2c(C)noc2C(F)F)=O)CC1 27232,C1(O)(CNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27233,Cn1nc(C(=O)NCC2(O)CCN(C(=O)COC3CCCOC3)C2)cc1Cl 27234,N1(C(C2CC(CCNC(c3n(CC)ccc3)=O)C2)=O)CCSCC1CC(N)=O 27235,CC1CN(C(=O)CN2CCN(C(=O)CN(C3CCCC3)C)CC2)C2COCC2O1 27236,c1(CC(=O)NC2CC2)cccc(OCC(C)C)c1.C(CC(=O)N)N(C)CC 27237,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27238,C12CCN(CC1C)CCCN2.CC(CC1CCCCC1)C(=O)N(C)C 27239,c1(C(=O)NCCCCN(C)C(c2[nH]cnc2C#N)=O)ccc2c(c1O)CCC2 27240,C=CCC(CC=C)C(=O)N1Cc2[nH]nc(C(=O)NC3CCC3(C)C)c2C1 27241,CC(C)C(CCN(C)C(C1(C)CCSCC1)=O)NC(c1occc1CN(C)C)=O 27242,N1(C(C2CC(SC)C2)=O)CCN(C(c2ccnn2C2CCOCC2)=O)CC1 27243,N1(C(CC2CCC(=O)N2)=O)CC2(CCCN(C(C3CC(N4CCCC4)C3)=O)C2)C1 27244,N1(C(COC2(C)CCC2)=O)CCOC(CC(=O)NCc2ccc(C(N)=O)[nH]2)C1 27245,C1(C)(C(=O)NCc2cn(C(CC)C)nn2)CCC2CC2C1 27246,C1(NC(c2cc(COC)[nH]n2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27247,c1(CC2C(=O)CC(NC(=O)NC(c3nn[nH]n3)C)C2)cccc2ccccc12 27248,Cn1nc(C(=O)NC(Cc2ccccc2)CCO)c2c1CNCC2 27249,C(=O)(C1CCCn2cnnc21)N(C(C1CC2CN(c3nnc(C4CC4)s3)CC12)C)CC 27250,C1(CCOC)CN(C(C2(COC)CC2)=O)CCN1C(C1C2CC3C(C2)C13)=O 27251,C(CCCC(=O)N1CC(CNC(c2cn(C3CC3)nc2C)=O)C1)COC(C)(C)C 27252,CC(C)C(C)C(CNC(c1occ2c1CCC2)=O)NC(=O)C(C)(C)C#N 27253,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27254,CC1(C(=O)NCC2CCCC(NC(=O)CNS(=O)(=O)C3CC3)C2)CNC(=O)C1 27255,C1(C(N2CC(O)(CN(C)C(C3CCCN3C=O)=O)C2)=O)(COC)CCCCC1 27256,c1(C(N2C(CNC(CC(CC)C3CC3)=O)C=CC2)=O)ccc(OC)c2ccsc12 27257,c1(C(C(C)NC(=O)NCCNC(=O)OC)C)ccc(C)s1 27258,C1(CNC(Cc2c(C)non2)=O)CCCN(C(C2SCCS2)=O)CC1 27259,N1(C(CC2CC(CC)C2)=O)CC2CC1CCC2NCc1ccccc1 27260,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)F 27261,c1(N2CCN(C)C(CNC(=O)COCCC(F)(F)F)C2)ncc2c(ncn2C)n1 27262,c1(N2CCN(C)CC2)ncc(C#N)cc1F.C12C(O)CCN1CC(=O)N2 27263,c1(CNC(C2CCSC2)=O)ccsc1C(=O)NC1CCC1CO 27264,c1(SC(C)C(=O)N(CCCCNC(c2ccn(C)n2)=O)C)ccc(Cl)cc1 27265,c1(C(N2CC(CC(=O)Nc3cncc(Cl)c3)OCC2)=O)cnn2ccccc12 27266,C(N=c1[nH]c(C(=O)OC)nc(=N)[nH]1)C1CC(NC(CC(CC)O)=O)C1 27267,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(F)(CF)C2)=O)C1 27268,C1(COC)CCCN(C(=NCCCC2CC2)NCCc2ccc(F)c(F)c2)C1 27269,N1(C(c2cc(C)oc2C)=O)CC2CCCC2(CNC(=O)CCCC(C)=O)C1 27270,Cc1[nH]nc(Br)c1C(=O)NCCCC1CCCN1C(=O)CCc1cc[nH]n1 27271,c1(OC(C)C)ccc(C(=O)NCCCCN(C)C(C2CCCC2(C)C)=O)cc1F 27272,C1(NC(C=C(C)C)=O)CC1C1CCCN(C(=O)C(C)N(C)C)C1 27273,C(=O)(C(CO)C(F)(F)F)N1C(CCC(=O)NC(C)C=CCN2CCCC2)CCC1 27274,N12CCC3C(C3C1)C2=O.n1(CC)ccc(C(=O)NC(C2(C(C)C)CCCC2)C)n1 27275,Cc1cc(C(N2CCC(C)(NC(c3cc(F)c(F)cc3Cl)=O)C2)=O)cc(F)c1C 27276,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27277,CC1(NC(C2CCC(=O)N2)=O)CN(C(=O)CNC(=O)NC2CCCCC2)C1 27278,C(CCC(C(=O)NCCC1CC1C)NC(c1cn(C)cn1)=O)OC 27279,N1(C(c2cc(Br)no2)=O)CC2CCN(C(c3cnn4c3OCC4)=O)CCC2C1 27280,c1(C(C(=O)NCCN(C(C(CC#C)C2CC2)=O)C)(C)C)ccc(F)c(Cl)c1 27281,CCCCCCC(C)NC(c1conc1CNC(=O)C(CCC)N(C)C)=O 27282,S(=O)(=O)(c1ccc(N2CCCC3(CC3)C2)nc1)NC(C)CC(N)=O 27283,Cc1ccc(C(N2CCSCC2C(N2CCC(OCC(C)C)C2)=O)=O)nc1O 27284,C(=O)(CCCS(C)(=O)=O)N(CC(C)NC(=O)CC1CCCC(=O)N1)CC 27285,C1(C(=O)NC2C(C)C2(C)C)CCN(C(c2ncccc2Cl)=O)C1(C)C 27286,c1(C(N2CCOCC(C(=O)NCCC(=O)N(C)C3CC3)C2)=O)cccc2ccoc12 27287,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27288,c1(NC(C(=O)NC(c2c(C)cccc2C)C)=O)ccc2c(c1)CCC2 27289,c1(C(N2CCC(N(C(=O)CC3C=CCC3)CC#C)C2)=O)ncc(OC)nc1OC 27290,C1(NC(CNC(N)=O)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27291,CCCCC(CC)C(=O)NCC1CC(C(=O)NC2CCOC2CC)C1 27292,c1(NCCN(c2nccc(NC3C(C)CSC3)n2)C)ccc(Br)cc1[N+](=O)[O-] 27293,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27294,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27295,C(=O)(CC(C)(C)C(=O)NCCN(C(=O)C(C)CSC)C(C)C)OC 27296,c1(OC)cc(C2(O[SH](c3ccccc3)CC(C(=O)OC)C)CCC2)ccc1Cl 27297,C(CCCC)(C(=O)N1CC(C2CCCO2)C1)NC(C(C)=CCC)=O 27298,c1(CCC(c2n(CC(=O)NCC)nnn2)NC2CC(C)(C)C2)cccc(Br)c1 27299,C1(NC(C(C)OCC2CCCC2)=O)CC(C(=O)NOCCO)C12CCC2 27300,c1(C(N2CC(CCNC(C3(C)C=CCC3)=O)C2)=O)ccc2c(=O)ccoc2c1 27301,C(=O)(C(C)CC(=O)OC)N1CCC(C)(NC(CC2CC(OCC)C2)=O)C1 27302,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27303,c1(CC(=O)N(CCCNC(=O)CCCC2CCC2)CC)ccc(F)c(F)c1 27304,C(=O)(CN=c1cc[nH]cc1)NC(CNC(=O)CCC(=O)c1ccccn1)CO 27305,C1(CC=C)(C(=O)NC)CCCN1C(c1ncn(C(C)C)n1)=O.C1(=O)CO1 27306,N1(C(c2cc(=O)n(-c3ccccc3)[nH]2)=O)CCn2cncc2C1 27307,c1(NCC2CC3CC(OC)C2C3)nc2c(F)cccc2c(=NCC(C)(C)C(N)=O)[nH]1 27308,C1(NC(C(CCC#C)O)=O)CN(C(c2nnn(C)c2CCC)=O)C2(CCCC2)C1 27309,c1(CCNC(=O)NC2CCc3c[nH]nc3C2)cc(Cl)c2c(c1)OCCO2 27310,C(C(C)(CCO)NC(=O)C(CCC1CC1)NC(c1snc(C)c1N)=O)OC 27311,c1(OCCC(=O)N(CCN=[N+]=[N-])CCOC)ccc(C)cc1Br 27312,C1(CNC(C(c2cn(C)nc2)=O)=O)CCCCCN1C(c1ccsc1Cl)=O 27313,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27314,CC1(C)CN(C(=O)CN2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC2)CCC1O 27315,c1(C(=O)NC(C(C)NC(C2(C)CCCOC2)=O)(C)C)cc(S(C)(=O)=O)co1 27316,N1(CC(CCC)(C)C)CCC(O)C(C(=O)NCc2cccc(OC)n2)C1 27317,CCC(C)N=c1[nH]c(=NCc2cc(F)nc(F)c2F)[nH]c2c(F)cc(F)cc12 27318,c1(C(=O)NC(CCOC)CNC(=O)COC2CCC2)cc(=O)n(C)o1 27319,CC(C)C(CN(C(=O)COCc1ccccc1)C)NC(=O)CCc1cc(Cl)no1 27320,c1(OC)cc(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(F)n1 27321,C(=O)(C1=C(Cl)CCCC1)NC(C(=O)N(CC)CC1CCOC1)CO 27322,CCCC(CC)CCC(=O)NC1C=CC(C(N2CCC(O)C2C)=O)C1 27323,C1(COC)(CNC(=O)CC(O)C2CCCC2)CN(C(=O)CCC2CC2(Cl)Cl)C1 27324,CCC(CC(=O)NC1CC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1)C(F)F 27325,N(C1COc2ccccc21)C(CC1CCN(C(c2cnc(C)n2C)=O)C1)=O 27326,CCCC(C(=O)N(C(C(=O)NOCCCSC)C1CC1)C)C(C)C 27327,Nc1c(C(=O)NC2CCCCC2NC(C2CC3(C2)CC3F)=O)cc(Cl)cc1F 27328,c1(CNC(c2cn(CCCC(=O)N(C3COCC3O)C)nn2)C)cccc(Br)c1 27329,C#Cc1cc(NC(=O)Cc2ncnc3sccc23)cc(-c2csc(OC)n2)c1 27330,C12(C(C)=O)CCC(NC(=O)CC(=O)NC(CC)CO)(CC1)C2 27331,N1(C(c2cc(C(C)C)nn2C)=O)CCN(C(=O)CCOCC2CC2)CC1C(C)C 27332,c1(C(=O)OC)[nH]c(=NC(=O)C2CC(O)C2)cc2cccnc12 27333,C1(N(CCCC)C(=O)CO)CCCC2CN(C(=O)CC3CCN(C)C3=O)CC12 27334,C1(C(=O)NCc2cc(C3CC3)on2)(CC)CN(C(c2cc(C)[nH]n2)=O)C1 27335,c1(C(N(CC(=O)N(C(C(CC)C)C)C)C)=O)ccc2cc[nH]c2n1 27336,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27337,C1(C(N(CCCNC(C2C(C)C2(F)F)=O)CC2CCCC2)=O)C(F)(F)C12CCC2 27338,c1(NC(CC(C)NC(=O)CCC2CC(F)(F)C2)C)c([N+](=O)[O-])cnn1C 27339,CC1CCC(C)(C(=O)NCC(=O)NCC(=O)NCc2nnc(O)n2C)C1 27340,C1(C(=O)NC2CN(C(C3OCCC3C)=O)C(C)(C)C2)(OC)Cc2ccccc2C1 27341,CC1(C)CN(C(C2CCCOCC2)=O)CC(C)(C)C1NC(=O)Cc1nnc(O)s1 27342,c1(C(=O)NC2CN(C(c3cn(C)nn3)=O)C2)cnc2ncnn2c1O 27343,C1(CNC(C2CCC(CC)O2)=O)CC2(CC2)CN1C(=O)CCCc1cncs1 27344,C1(NC(C2CC23CCOC3)=O)CCCCC12CCCN(C(=O)C1=CCCOC1)C2 27345,CCC(CO)C(=O)N1CCC(N2CC(C)(NC(=O)CCCC3(C)CC3)C2=O)CC1 27346,C(C)(C)(C(=O)OCC(C1CCC1)NC(OC(F)F)=O)NC(=O)OC 27347,c1(C(C2COCCO2)CNC(=O)NCC(=O)NC)cccc2[nH]ccc12 27348,c1(OCC)cc(C(=O)NCC2(C)CCCN(Cc3cnc(Cl)s3)C2)cc(F)c1 27349,c1(C(=O)NCCC(C)NC(=O)C=Cc2nccs2)cc(-c2ccoc2)[nH]n1 27350,c1(C(=O)NC(CNC(C(C)CC(C)(C)C)=O)(C)C2CC2)cnc2c(c1)NC(=O)CO2 27351,c1(C(=O)NCC(CCCC)NC(C2CC2OC2CC2)=O)c[nH]c2cc(F)ccc12 27352,Cc1cc(C(=O)NC2CCOC(C(=O)N(C34CC(C3)C4)C)C2)c(C)o1 27353,Cc1nc2c(o1)CCCC2CC(=O)N1CC2CCC1CN2C(=O)Cn1cncn1 27354,C1(C(N2CCCC(C)(CC)C2)=O)CCCCCCN1C(c1cncc(OC)n1)=O 27355,C(=O)(CCCC(F)(F)F)NCC(CC)(C)NC(C1(C)CCC(=O)N(C)C1)=O 27356,CC(CC(=O)NCCC1CN(C(=O)CNC(C2CCC2)=O)C1)C(F)(F)F 27357,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCC2(CN(C(c3nnsc3C)=O)C2)O1 27358,C1(CC)CN(C(c2cncc(C(F)(F)F)c2)=O)CCC1NC(c1cccnc1)=O 27359,c1(NC(Cc2cccc(C)n2)=O)cnc(Cl)cc1NC(=O)CNC(=O)C(F)(F)F 27360,CC1CC(C(=O)N2CCCC(CC(=O)NC3CCC4CC3CO4)C2)=NO1 27361,C1(CCC(=O)NC23CC(NC(=O)CCc4cc[nH]n4)(C2)C3)CCCCC1 27362,c1(C(N2CCC(NC(c3cccc(OC)c3)=O)(CO)C2)=O)scc2c1OCCO2 27363,C1(NC(CCn2c(C)ccc2C)=O)CC(NC(=O)Cc2nc[nH]n2)C12CCC2 27364,N1(C(C(CSC)OC)=O)CCN(C(=O)C(C(C)(C)C)c2cccc(C)c2)CC1C 27365,N1(C(CC(CC)C)=O)CCc2onc(C(N3CCN(CCF)CC3)=O)c2C1 27366,C(=O)(CC(O)C(Cl)(Cl)Cl)NC1(CO)CN(C(C(CCC)CC)=O)C1 27367,C123CCC(CC1)N(C2)C3=O.c1(NC(CN2C(C)CC2)=O)ncc([N+](=O)[O-])n1C 27368,N1(C(c2c(CC)nnc(C)c2)=O)CCCC2CN(C(C3CCN(C)C3=O)=O)CC12 27369,C(=O)(CCCCN=[N+]=[N-])N1CCCC(N(C(c2c(CC)nn[nH]2)=O)CC2CC2)C1 27370,C(=O)(C(O)CC(=O)OC(C)(C)C)NC1(C)CN(C(C(CCC)C)=O)C1 27371,N1(C(C2C(C)CCCC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27372,Cc1ccccc1C1(C)CC1NC(N1CC(CCC(=O)OC(C)(C)C)C1)=O 27373,Cc1nc(C(=O)NCc2ccc(CNC(=O)C=CS(C)=O)cc2)c(C)n1C1CC1 27374,CC(CC(C)(C)C)C(=O)NCC1CN(C)CCN1C(C1CC12CCC2)=O 27375,N1(C(COC(C)C)=O)CC(NC(C2(C)CC3CC3C2)=O)CC(O)C1 27376,N1(C(C(C=C)C)=O)CCC2(CCC(NC(C3(CC=C)CC3)=O)CC2)CC1 27377,C(C(C(=O)NCCCNC(=O)CC(C)NC(=O)CCN1CCOC1=O)OC)OC 27378,C(C1COC(C)(C)O1)=CC(=O)NCC(C)CNC(=O)C(C)(C)CC1CCC1 27379,CC(C)CC(C(=O)NC1(CO)CC(F)C1)NC(c1nnc(O)nc1O)=O 27380,Cc1nn2cccnc2c1C(N1CC(CCNC(=O)CN2CCC(C)C2)C1)=O 27381,c12c(cccc1Br)S2.C1(C(=O)OC)CC2(C1)CC2NC(=O)C(=O)NCC(F)(F)F 27382,C(=O)(C(O)C1=CCCCC1)N(C(C)C)CCN(C(=O)CN1CC(=O)NC1=O)C 27383,C12CCC(C1)C(=O)OCCCC(=O)N2C.C(=O)(C(C)(C)C)NCCOC(C)(C)C 27384,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC2CN(C(C3(C)CCCS3)=O)CC12 27385,c1(C(=O)NCCC(C)NC(=O)C(F)(F)C(O)C2CC2)cc(S(N)(=O)=O)c[nH]1 27386,C1(CN(C(=O)C=CC=O)C)COCCN1C1CCC1.C1(CCC)CC1C(=O)OCC 27387,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27388,c1(OCC(N2C(C(C)NC(C)=O)CCCC2)=O)ccc(F)c(F)c1 27389,N1(C(C(C)c2ncco2)=O)CCN(C(C2CC(N(C)C)C2)=O)CC(C)(C)C1 27390,c1(OC(C)C(=O)NC2CCCN(C(=O)C3=NNC(=O)C3)C2)ccccc1C#N 27391,c1(C(N2CCCCC(NC(c3c(C)c[nH]n3)=O)C2)=O)cccc2nc[nH]c12 27392,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27393,N1(C(Cc2cc(CC)no2)=O)CCCCC(CSc2cc(C)nc(N(C)C)n2)C1 27394,c1(N(C)CC)nc(NN)nc2ccsc12.C1(C)(CO)CC(F)(F)C1 27395,c1(-n2c(C3CCCCN3C(C3CCC3)=O)nc(CCC)n2)cccc2ncccc12 27396,C(=O)(CN=c1cc[nH]cc1)N(C(C(=O)N(C)CCC1CCCCO1)(C)C1CC1)C 27397,c1(OC)ccc(C(=O)NCC(CO)NC(c2ccoc2C)=O)nc1 27398,C1(C(=O)NCC(C)S(N)(=O)=O)C(C)OCCN1C(=O)C(C1CCOCC1)F 27399,Cc1nc(NCC2CN(C(C3C=CCCC3)=O)CCC2C)ncc1Br 27400,N1(C(CCOC)=O)CCCC(NC(c2cc(CCOC(C)C)on2)=O)C1C 27401,C(=O)(C(F)C(C)CNC)NC(C1C=CCCC1)C(=O)NC(CC)CC 27402,CC1CN(C(c2ccc(-c3ccco3)s2)=O)CC(C)C1NC(=O)CCC1(C)CC1 27403,C1(c2nc3ccc(OC)nn3c2)NC(=O)N(CCF)C2=C1C(=O)NC2(C)C 27404,Cn1c(C(=O)NC2(CNC(=O)C(O)C(F)F)CC(F)(F)C2)cc2sccc12 27405,c1(CCCCCC)c(-c2cnc(C3(C(F)(F)F)CCC3)nc2)cncc1F 27406,Cn1ncc([N+](=O)[O-])c1C(=O)NCC(C)(C1CC1)NC(=O)Cc1ccccc1Cl 27407,C1(NC(C2(C)COC2)=O)CC(CNC(c2conc2C(C)(C)C)=O)CC1O 27408,N1(C(C(CCC2CC2)NC(COCC(=C)C)=O)=O)CCC2CCN(C)CC12 27409,c1(C(C)NS(=O)(=O)c2cc(Cl)sc2Cl)nc2ccc(C(N)=O)cc2s1 27410,C1(C(=O)Nc2c(C)n(C)nc2)CC(F)CN(C(C2CCO2)=O)C1 27411,c1(C(=O)NCC2CCN(C(C(CSC)(C)C)=O)C2)[nH]c(C)c([N+](=O)[O-])c1C 27412,C1(N(C(C(C)CO)=O)C)CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 27413,C12(NC(=O)C3=CCCOC3)CCN(C(c3cccc4c[nH]nc34)=O)CCC1C2 27414,Cc1c(Br)ccc(F)c1CNCC(c1ccccc1)(C)O.C1(C(C)(C)C)CN1 27415,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27416,C1(C(N(CC(=O)NCC2(F)CCCCC2)C)=O)CC2C=CC1C2 27417,N1(C(C(C)C2CCCC2)=O)CC23CCCC2(C1)CN(C(=O)Cc1c[nH]nc1O)C3 27418,c1(N2CCC(OCC=C)CC2)nc(N2CC(OC(C)C)C2)nc2c1SCC2 27419,C(=O)(C(C(C)C)NC(C)=O)N1CC(c2cn(CC(=C)CC)nn2)(C)C1 27420,n1(CC)ccc(C(=O)NCC2CN(C(c3ncc(F)cc3N)=O)CC2C)cc1=O 27421,c1(C(=O)NC2CC2CNc2cc(O)ncn2)ccc(=O)n2c1CCC2 27422,CC(C)C(CCNC(C1CCCC(=O)N1)=O)NC(=O)C(C1CCCCCC1)C 27423,c1(C(CNC(CN(CCOC(=O)NC)CC)=O)NC(=O)COC)cccc(N)c1 27424,CC(F)(C(=O)NC1CCC(NC(c2cnncc2O)=O)CC1)C(F)(F)F 27425,C1(NC(C(=O)N(C)CCN2CCCCC2)=O)CCC2CC=CC12 27426,N1(C(C2COCC(C)O2)=O)CCCC(O)(CCNC(=O)C(C)(C)CC2CC2)C1 27427,S(=O)(=O)(c1ccc(N2CCC3(CCC3)CC2)cc1Br)NC(C)Cn1cccn1 27428,N1(C(C(C)N(CC(O)C2CCC2)C(=O)NS(C)(=O)=O)=O)CCc2ccsc2C1 27429,N1(C(c2cc(OC)n[nH]2)=O)CCC2(COC(CNC(c3coc(O)n3)=O)C2)C1 27430,N1(C(CC2(C)CC2(F)F)=O)CCCC(OCCCNC(=O)Cc2cocn2)C1 27431,N1(C(CCCCNC(=O)COC)=O)C(CNC(N)=O)CC2COCC12 27432,c1(N(C)C(c2ccc(C(C)=O)cc2)=O)ccc(NCC=CC)cc1 27433,C12(NC(c3ccccc3)=O)CC(NCC3(C(C)(C)OC)CC3)C1C2 27434,N1(C(C(F)=C(C)C)=O)CCN(C(=O)Cc2ccccc2OCC2CC2)CC12CC2 27435,c1(CC(=O)NCc2cccnc2Br)n[nH]c2cc(C3=CCCCC3)ccc12 27436,C(C(=O)N(C)CC1CCCN1C(c1occ(C)c1C)=O)(C(C)C)N(CC)CC 27437,Cc1cccc(CNC2CCC(C(=O)NC(C3CSC3)CO)C2)c1F 27438,Cc1nocc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1ccco1 27439,N1(C(C(=O)NC(c2ncc(Br)cn2)CCC)=O)CN(C)C(=O)C1C 27440,N1(C(c2cc(NC)nn2C)=O)C2CCC1C(NC(=O)C(C)OC1COC1)C2 27441,S(=O)(=O)(c1ccc(-c2ccc(F)c(Br)c2)cc1)N1CCC(C)C(C(=O)O)C1C 27442,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27443,N1(C(C(=O)NCCC2CCCCC2(F)F)=O)CCc2ccc(Cl)c(F)c2C1 27444,N1(C(C(C)=CC=C)=O)CC2CCCC2C1C(=O)NCCC(O)CC 27445,C1(NC(CC2CCN(C)C2)=O)CCC(C)(NC(c2cc(N)nc(Cl)c2)=O)CC1 27446,C=CCCC(F)(F)C(=O)NC(CC)CCCC(=O)N(C)Cc1ncc[nH]1 27447,c1(C(N2C(C)(CNC(c3cc(OCC)n[nH]3)=O)CCC2)=O)c(C)nn(C)c1F 27448,CC1CCC(CC(=O)Nc2nn(C)cc2Br)CC1C 27449,N1(C(C2CCN(C(C)=O)CC2)=O)CC(CNC(=O)CC(C)C(F)F)C(F)(CO)C1 27450,C(=O)(C(O)CC(C)C)N(C)Cc1ccc(CNC(C(C)=C(C)C)=O)cc1 27451,C1(C(=O)NC2(COCC)CC2)CC12CCN(C(c1ccc(N(C)C)cn1)=O)CC2 27452,CCC(C)C(O)C(C)C(=O)N(CC(=O)NC1CCC(C2CC2)C1)C(C)C 27453,C(C)(C(C(=O)N(C)CC1CCCC1)C(C)C)NC(c1snc(C)c1N)=O 27454,Cn1ncc(C#N)c1C(N1CC(CNC(c2ncc(F)cn2)=O)C(O)C1)=O 27455,C=CC1(C(=O)NCC2CCCN(C(=O)CCc3cnn(C)c3C)C2)CCCCC1 27456,NS(=O)(=O)c1csc(C(N2CCC3C(NC(=O)CCCn4cncn4)CC23)=O)c1 27457,c1(CC)cc(C)c(C(=O)NCC(C)(C(C)C)NC(=O)Cc2cscn2)o1 27458,c12cc(oc1C)COCCCNC2=O.C(=O)(C(=O)NCCC1CCCC1)NCC 27459,N1(C(C(C)n2ccnc2)=O)CCN(C(=O)CN2CC(C)(C)C2)CC(C)(F)C1 27460,c1(C(=O)NC(CN(C(C2CCN(CC)C2)=O)CC)C)cc(COC)c[nH]1 27461,c1(C(C(N2CCC(C(C)NC(=O)CSC(F)(F)F)C2)=O)O)ccc(F)cc1 27462,c1(OC)ccc(NC(C2(C)CCCN(Cc3cc(Br)ccc3F)C2)=O)c(F)c1 27463,C1(CC)CCN(C(C)=O)C1C(=O)N(C(C)CNC(c1scnc1C)=O)CC 27464,N1(C(C2CCCC23CCC3)=O)CCN(C(C2(Cl)CC2)=O)CC12CCC2 27465,c1(C(N2CC(CCC)C(C(=O)NC3CCSC3)C2)=O)ccc(=O)n(C)n1 27466,c1(C(C(=O)N(C)CC2CSC2)NC(C(C)OCC=C)=O)cccc(C(F)(F)F)c1 27467,c1(C(=O)NCC2N(C(C3CC=C(C)CC3)=O)CC2)cc(C)c(C)cc1C 27468,CCCC(C(=O)NC(C)(CNC(=O)C(N1CCOC1=O)C)C1CCC1)OCC 27469,CC1CC(C(=O)NCC2(F)CCN(C(=O)C3CC3)C2)=NO1 27470,N1(C(C(CC)OCC)=O)CC(C)CN(C(c2cccc(C)c2C)=O)C(C)C1 27471,c1(NC(C23C(CN(C(CCOCC#C)=O)C2)C3)=O)[nH]c(C)c(C)c1C#N 27472,C(=O)(C1=CCCCO1)NCCCCCNC(=O)Cn1ccc(C(F)F)n1 27473,Cc1cccc(CC(=O)NC2CC3(C2)CC3NC(C2CC(C(C)C)=NO2)=O)c1F 27474,CC1CCN(C(c2cncc(O)c2)=O)CC1CNC(C1CCCC1)=O 27475,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27476,C(=O)(C1=COCCC1)NCC1(NC(c2ccccc2F)=O)CC(O)C1 27477,CC1CN(C(=O)Cc2nn(C)cc2Br)CCN1C(=O)CSc1nnnn1C 27478,C(=O)(C1CCc2c(Cl)cccc21)OC.C1(=O)C2c3c[nH]nc3CN12 27479,C#Cc1cc(C(=O)NC(C)CCNC(C2(CS(N)(=O)=O)COC2)=O)ccc1C 27480,N1(C(c2cc(C)sn2)=O)CCC(CNC(C2C(F)(F)C23CCC3)=O)C(F)(F)CC1 27481,N1(Cc2c(C)cccc2)CC2(CCN2C(=O)CCn2ccnn2)C1 27482,Cn1c(C(=O)NCCC2CCCCN2C(=O)CN2CCCCC2)nnc1S 27483,C(=O)(C(F)CCC(C)C)N1CCC(NC(C=CCC=C)=O)CC1C1CC1 27484,c1(C(C(=O)NCCC2CC3(CCC3)O2)N(C)CC)nc(C)c(C)s1 27485,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(C(C)C)C1 27486,C1(C(N(C2CCN(C(=O)C(F)(F)F)C2)CC#C)=O)CC(=O)N(C2CCCCCC2)C1 27487,N#CCCCC(=O)N1CC(OC2CCN(C(=O)CNC(C3CCCC3)=O)CC2)C1 27488,Cc1cc(C)n(CCN(C(C2CN(C(=O)OC(C)(C)C)CCO2)=O)C2CC2)n1 27489,c1(C(N(CCCCOCCNC(C2C(C)OCC2)=O)C)=O)ccc2oncc2c1 27490,C12(CNC(c3cc(C)oc3)=O)CCC(CNC(c3cscc3Cl)=O)(CC1)CO2 27491,N1(C(CC2CC(C)(C)C2)=O)CC2C3CCC(C2C1)N(C(C1CC1C1CCC1)=O)C3 27492,c1(CNC(c2ccc(C#C)o2)=O)nc(CNC(=O)C(C)CC2CC2)cc(O)n1 27493,c1(C(C(N(CCN2CCOCC2)C(=O)NC)C)C)cncc(OCCNC)c1 27494,N1(C(c2cc(C)c(C#N)cc2)=O)CCC2CN(C(=O)CCP(C)(C)=O)CCC2C1 27495,c1(C(=O)OCC)c(OC=O)noc1C.C123CC(C1)(C2)C(=O)NC3.C(CC)OC 27496,C1(CNC(C(C)N(C(=O)CC2CCCSC2)C)=O)CC2C=CC1CC2 27497,c1(C(=O)NCC2CN(C(CC(=O)NCCOC)=O)CC2C)cc(N)c(C)cc1C 27498,c1(C(N2CC(F)(CNC(COCCOC)=O)C2)=O)ccc(C(=O)OC)c(O)n1 27499,C12(NC(c3cocn3)=O)CC1CN(C(C1CC1c1cncs1)=O)C2 27500,N(C1CCCn2ccnc21)C(c1scc(C(=O)OCC)n1)=O.c12cc(ccn1)N2 27501,C1(NC(C23CCCC2C3(F)F)=O)CC2CCC1(NC(C1(n3nccn3)CC1)=O)C2 27502,CC(C)CC(CNCCCc1ccncc1)OCc1nnnn1C1COC1 27503,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27504,C1(C)(COC)CC(NC(=O)CC(C)(C)O)CN1C(=O)CCc1cnn(C)c1 27505,c1(C(N2CCC(NC(c3c(C)cns3)=O)C2C2CC2)=O)cc(S(N)(=O)=O)c[nH]1 27506,c1(N2CC(C)C(N(C)C)C2)[nH]c(=NCc2cc(C(F)(F)F)on2)nc2scnc12 27507,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(C(C)C)C(=O)O 27508,C1CCN=C(NCc2c(C)cccc2)NCc2ccc(nc2)O1.C1(OC)CCC1 27509,C1(CC(=O)N(CCCS(N)(=O)=O)C)CCC1C1CC1 27510,Cc1ccc(Cl)cc1C(=O)NC1COCCC1NC(=O)CC1(O)CCCOC1 27511,C12(NC(c3cc(Cl)c[nH]3)=O)CCCC1N(C(C1CC3CCC1C3)=O)CC2 27512,Cc1nn(C)c(C)c1CC(=O)NC1CCC(NC(=O)COCC2(F)CC2)CC1 27513,N1(OC(=O)CC(C)CSCC)CC(=O)NC(C2CC2)C1 27514,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(=O)Cc2c(C)noc2Cl)C1 27515,Cc1c(C)c(C)c(C(=O)NCCC2CCN(C(c3cnn(C)c3)=O)C2)c(C)c1C 27516,C1(SC)CC(C(=O)OCC2(CN(C)C)CC2)C1.C(C)(C)C 27517,C1(NC(C(C=C)O)=O)CS(=O)(=O)N(C)C12CCN(C(C1CC13CC(O)C3)=O)CC2 27518,CC1CN(C(c2nccc(C(F)F)n2)=O)CCN1C(C1CCCC(F)(F)C1)=O 27519,C1(N(C(=O)CSSC(F)F)CC)CCN(C(C2CC2c2ccccc2)=O)C1 27520,C1(C(=O)NCC2(C(C)(C)C)CCN(C(CC=C(C)C)=O)C2)C2CCC1(C)C2(C)C 27521,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27522,c1(CCNC(=O)NC(C)=O)ccc(C(C)NCc2ncc(Br)cn2)cc1 27523,c1(C(=O)NC2C(NC(c3cc(C4CCOC4)[nH]n3)=O)COC2)cc(O)nc(O)n1 27524,c1(CC)ccc(C(=O)NC(Cn2ccnn2)C(=O)NC(C)(C)CSC)cc1 27525,c1(N2CCC(NC(C(C)(O)C3CC3)=O)C2(C)C)nc(O)c2c[nH]nc2n1 27526,C1(NC(=O)CCCCO)CC2CCC1N(C(c1cccn1C1CC1)=O)C2 27527,C1(CC(=O)NCC2(NC(c3c(OC)cccn3)=O)CCCC2)CC2C=CC1CC2 27528,N1(C(C(=O)NCc2cc(Br)c(Br)c(F)c2)=O)CCC12CCCS(=O)(=O)C2 27529,Cc1nnccc1N(C(C(=O)NCSc1ccc(Cl)cc1)C1CCOC1)C 27530,N1(C(C(COC)OC)=O)CC2CC(C(=O)Nc3cc(Cl)ccc3C)CC(C2)C1 27531,C(C(C(=O)N1CC(N2CCOC2=O)C1)C(C)(C)C)NC(CCCCCN(C)C)=O 27532,N1(C(=O)CN2CC3CCCC2C3CO)CCC2C(CCN2C(=O)CO)C1 27533,C1(CNC(c2ccn(CCCC)n2)=O)CC(NC(C2CC2F)=O)CC1O 27534,C12(NC(c3cc(C)c(O)cc3)=O)CCCC1N(C(c1coc(O)n1)=O)CCC2 27535,N1(C(C(C)c2ccsc2)=O)CC(CC(=O)NC2CN(C(=O)C3CC3)C2)CC1(C)C 27536,CC(C)CC(C(=O)N(CC(C)(C)C(N)=O)C)N(C(=O)CN1CCNC1=O)C 27537,N1(c2nnc(COC)s2)CCCCC(CNC(C2CC(=O)N(C(C)CC)C2)=O)C1 27538,N1(C(C(C)CF)=O)CC(C2CCN(C(=O)C(C)(C3(C)CC3)OC(C)(C)C)CC2)C1 27539,C(=O)(CC(C)CCC(=O)NC(C)(C)CCNC(c1nn(C)cc1Cl)=O)OC 27540,c1(C(N(CCCNC(C(C)=CC)=O)C2CC2)=O)ccc2nc(C)nn2c1 27541,c1(CC)cc(C(N2CCC(C(C)(C)NC(c3c[nH]ccc3=O)=O)C2)=O)nn1C 27542,c1(C(N2CCC3(NC(=O)CCCCC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27543,C(=O)(C#CC1CCOCC1)N1CCC(=C)CC1C(=O)Nc1cn(C)nc1C(=O)OC 27544,c1(CN(C)C(c2cccc(CN3CCOCC3)c2)=O)cc(O)ccc1I 27545,C1(C(=O)NC2C(NC(=O)COCC3CCC3)CCC2)CC(=O)OC1(C)C 27546,c1(NC(C(CC)(C)C)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1.C12C=CCN1C2=O 27547,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27548,N1(C(c2cn(C(C)C)nn2)=O)CCCC(CNC(c2cocn2)=O)C1 27549,N1(CCCOC)CCC(C)C(NC(C2CCCCC2c2nc(S)n[nH]2)=O)C1 27550,Cc1ccc(C(C)NCC2CCCCC2c2cccc(F)c2)nn1 27551,c1(C(N2C(C(C)(C)NC(=O)CNS(N)(=O)=O)CCC2)=O)cnc2[nH]c(O)nc2c1 27552,N1(C(CC)=O)CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1 27553,c1(C(NNC(=O)NCC)=O)ccc(F)c(Br)c1.Cc1ccnnc1CCN(C)CC 27554,C(CCNC(=O)OC(C)(C)C)(C(F)(F)F)NCC(c1cccc(F)c1)C 27555,C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C=CC)=O)C2)C1 27556,N1(CC(=O)N(C(CNC(C(c2cccnc2)C)=O)C)C)CCC(CO)CC1 27557,C1(NC(=O)NC2C3CCCOC23)COCCN(C(=O)Cc2cccs2)C1 27558,Cc1cnc2n1CCCC2C(=O)NC1CCCC1NC(c1cncn(C)c1=O)=O 27559,C(=O)(C(F)(F)C1=CCOCC1)N(C(C)CNC(C1SCCCS1)=O)C 27560,C1(NC(CCOC(CC(C)C)C)=O)CCN(C(C2CCCC(C#N)C2)=O)C1(C)C 27561,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3CCCN3C3CC3)=O)C2)cc1Cl 27562,N1(C(CCSC)=O)CCN(C(=O)C2=CCCC2)C(C)C1 27563,N1(C(=O)CC2(O)CCC2)CCC2(CCC2)C(NC(C2CC3C=CC2C3)=O)C1 27564,N1(C(C2(F)CCN(C(=O)CCOC3CC3)C2)=O)CCC2C(O)CC12 27565,c1(C(=O)NCC2(O)CC(C(N3CC4(CCOC4)C3)=O)C2)nccc2cc[nH]c12 27566,c1(C(=O)NCC2CCCN(C(=O)C(O)C3CC3)CC2)c[nH]c2cccc(Cl)c12 27567,C12(NC(c3ccc(CC)nc3)=O)CCCC(CN(C(C)=O)C1)C2 27568,CC(C)(C)CC(=O)N1CC(O)CC1C(=O)NC(CO)C(C)O 27569,C(=O)(C(C)S(C)(=O)=O)N1CCN(c2cc(C=CCOC)sn2)CC1 27570,c1(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)cnc2c(c1)CCOC2 27571,C(=O)(C(C)CC(C)(C)C)NCc1ccc(CN(C(c2onc(C)c2C)=O)C)cc1 27572,c1(C(C)C(=O)NC(C)(C)CNC(C2(C(C)(C)O)CC2)=O)cncc(F)c1 27573,C1(O)(CN(C)C(C2CCC(=O)CC2)=O)CCN(C(C2(O)CC2)=O)C1 27574,N1(C(c2nc(OC)c(C)s2)C(=O)NCCCOC)CCC2CCCCC2CC1 27575,Cc1cncc(CC(=O)NC2(C(=O)NC3CCSCC3)CCCCC2)c1 27576,c1(C(=O)NCC2OCCN(Cc3c(C)ccs3)C2)cccc2c1COC2(C)C 27577,C1(C(N(C2CCCC2)CCNC(C2C(C)(C)COC2)=O)=O)CCC2(CCC2)C1 27578,C(CCC(C)(C)C)(C(=O)NCC)N1CCOCC(=C)C1 27579,C(CC)(C(=O)NCC(=O)NCCC(O)CNC(c1cc(-c2ccco2)c[nH]1)=O)OC 27580,c1(COC)cc(C(=O)NCC2(NC(=O)CCc3ccccc3)CCCC2)c(C)o1 27581,N1(C(c2scc(C)n2)=O)CCC(F)(CNC(C2CC2(Cl)Cl)=O)CC1 27582,CC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C(C1(CCN(C)C)CC1)=O 27583,C=CCCC(C(=O)NC(CCO)C(C)(C)C)NC(=O)C=CCN(C)CC 27584,c1(C(=O)NCC2N(C(Cc3nnc(C)o3)=O)CC(O)C2)cnn2cnnc2c1 27585,c1(C(=O)NC(C(C)NC(C2CNC(=O)C2)=O)CO)cnc2nccn2c1 27586,c1(C(N2CC(CC=C)(NC(c3cccnc3S)=O)C2)=O)cc(F)c(O)c(Cl)c1 27587,c1(C(=O)NCCNC(C2OCC3CCCC2C3)=O)cc2cc[nH]c(=O)c2s1 27588,c1(C(N2C3C(C(N4CCN(C)CC4)=O)C(C3)C2)=O)ccc2[nH][nH]c(=N)c2c1 27589,C1(NC(c2cc(C)[nH]n2)=O)CCCC(N(C(=O)C(F)=CC2CC2)C)C1 27590,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27591,C(=O)(C1CSc2ccccc21)N1CC(CC=C)(NC(c2ccnnc2C)=O)C1 27592,Cc1cc(CNS(C)(=O)=O)cc(-n2nccc2C)c1.C12CCC(=O)N1CC2 27593,c1(NC(COCCNC(Cn2ccc(C)n2)=O)=O)cccc(=O)n1C 27594,N1(C(c2csnn2)=O)Cc2[nH]nc(-c3cncc(Oc4ccccc4)c3)c2C1 27595,N1(Cc2nc(C)sc2C)CC(C2CCCCC2)CC1C(=O)O 27596,C1(CNC(CCCn2cc(C(C)C(=O)O)nn2)=O)CC2COCC2O1 27597,c1(C(=O)NCC2C(NC(CC(C)(C)C)=O)C2)ccc(OC2CCCC2)c(F)c1 27598,c1(CC)c(C(=O)NC(C)CCNC(C2CCOC2)=O)nnn1CC 27599,C1(C(=O)NCC(C(C)C)NC(c2cc(COC)on2)=O)(C(F)F)CCCCC1 27600,C1(C(=O)OC(C)=O)CCCC1.C(C1CC(=O)N1)SC 27601,C1(N(C(COC)=O)C)CCCN(C(C2CCCS2(=O)=O)=O)CC1 27602,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(OCCF)c1 27603,C1(C(OC)Cc2ccc(C)o2)CCN(C(C2CNC(=O)C2)=O)CC1 27604,C(CCC(C)N=c1cc(Cl)nc(C2CCC2)[nH]1)NC(c1cncc(COC)c1)=O 27605,C1(C(=O)NCC2(F)CCCN(C(CN(C(=O)OC)C)=O)C2)CCn2nncc2C1 27606,C[Si](C)(C)CCCNC(=O)C(c1cccs1)NC(C1(O)CCOC1)=O 27607,C1(NC(=O)OCc2ccc(Br)cc2)(CCCOCCO)CCOCC1 27608,N1(CC(=O)NC2CN(C(C(C)OCCC(C)C)=O)C(C)C2)CCc2ccccc21 27609,c1(C(c2ncccn2)NC(c2ccc(Cl)s2)CC)nnnn1CC(=O)OC 27610,C1(C(N(C(C)COC)CC)=O)(NC(=O)Cc2ncn(C)n2)CC1(C)C 27611,N1(C(c2n(C(C)C)ccn2)=O)CCN(C(C2CC3CCCCC23)=O)C(CO)C1 27612,C1(C(=O)NCCOCC#C)CSCCN1C(=O)CN1CC=CC1 27613,c1(C(=O)NC(CNC(C2(Cn3cncn3)CC2)=O)C2CC2)cn(CCO)nn1 27614,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CC(=O)N1)=O)CCO2 27615,C(=O)(C(CC=C)CC(C)C)NCC1CC(C(=O)NC(CC#C)(C)C(=O)NC)C1 27616,CC1(C)CC(CNC(=O)CC2CNC(=O)C2)N(C(=O)C=Cc2cccc(Cl)c2)C1 27617,C1(NC(C(C)Oc2ccccc2)=O)CC1C1CCCN(c2cc(=O)n(C)cn2)C1 27618,N1(C(CNC(CC)=O)=O)CC(C)CN(C(c2cccc(=O)o2)=O)C(C)C1 27619,N1(C(=O)CCC2CCOC2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27620,C1(C(=O)NCC2(C)CCN(c3cc(C(=O)OC)ncn3)C2)CCS(=O)(=O)CC1 27621,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27622,C1(CSC)CCCN1C(C1CCOC1CNC(=O)CCCc1ccccc1)=O 27623,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCCN(C)C)CC12 27624,c1(OC)ccc(C(=O)Nc2ncoc2-c2cccs2)c([N+](=O)[O-])c1 27625,C12(C3CCN(CC3)C(=O)CS(=O)(=O)N(C)C(C)C(=O)N1)CC2.CCCCNSCCl 27626,C(=O)(C1=C(Cl)CCC1)NC(C(=O)NC(c1ccc(Cl)cc1)C)CCF 27627,Nc1ccc(F)c(C(N2CCC(N(C3CC3)C(C3CCCCC3)=O)CC2)=O)c1 27628,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CNC(C1CCCN(C(C)C)C1)=O 27629,C#CC1CN(C(C2(C(N)=O)CC2)=O)CCN1C(=O)Cc1cccc(C)c1 27630,C1(NC(C(C)OCC)=O)CCN(C(c2cc3cccnc3s2)=O)C12CCC2 27631,C(=O)(C(C)(C)C(C)O)NCCCCCN(C(C(c1cccc(C#N)c1)C)=O)C 27632,C(=O)(C(C(C)NC)C(C)C)NC(c1c(C)noc1C)c1ccc(Br)cc1 27633,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27634,CN1C(=O)NCC12CCN(c1nccc(=NCC3(Sc4ccccc4)CC3)[nH]1)CC2 27635,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(CCC(=C)C)=O)C1 27636,c1(OC)ccc(C)nc1C(=O)NCC(C)NC(=O)C(C)C(C)O 27637,c1(NC(=O)NCCc2ccc(OC)cc2)nc(CC(C)C)sc1C#N 27638,CC1CC(CNC(c2cnn(C)c2Cl)=O)CN1C(=O)CC1(O)CCOC1 27639,c1(NCc2c(C)cccn2)ncc(S(=O)(=O)NCC2CC2C)cc1Cl 27640,CC1(C)CC(=O)OC1CNC(C1(C2CCCN2C(C2C3CC4C(C3)C24)=O)CC1)=O 27641,Cc1ncnc(N2CC3CC3(C(=O)NCc3cccc(C#N)c3)C2)c1Br 27642,C1(C(=O)NCC2(O)CC2)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27643,Cc1[nH]c2ccccc2c1CC(=O)NCCC1(O)CCN(C(=O)CN(C)C)CC1 27644,c1(OC)c(F)cc(C(=O)OCc2cn3cccnc3n2)cc1F 27645,c1(CCOCCC)nc(-c2cc(OC)ccn2)nn1C1CCOC1(C)C 27646,C1(COCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27647,c1(CC)cc(OCC)cc(C)n1.c12ccccc1C1(CC1)C(=O)N1CC(C1)CN2 27648,C1(C(=O)NC2C(NC(C(=O)NCCNC(C)=O)=O)C2)CCC12CCC2 27649,Cc1[nH]nc(CO)c1C=O.N1(C(N)=O)CCC(C(C)C(=O)NC2CC(C#N)C2)C1 27650,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27651,Cc1cc(NC(=O)C#CCNC(C2CCSC(C)C2)=O)cc(CO)c1 27652,n1(CCC(C)(C)C)nc(C2CCCO2)nc1Cn1nnc(C(C)(C)C)n1 27653,Cc1c(C(N2CC3(CCC3NC(=O)C(N)=O)C2)=O)oc2c(C)cc(Br)cc12 27654,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27655,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27656,C1(O)(C(=O)NCC(C)(C2CC2)NC(c2cnc(C)nc2)=O)CCCC(C)CC1 27657,c1(CCC)ccc(C(=O)NC(CO)C(C)NC(c2coc(CN(C)C)c2)=O)cc1 27658,C1(C(=O)NCC2(C)N(C(C(C)NC(CC)=O)=O)CCC2)CCc2nc(C)cn2C1 27659,C(=O)(C(F)(CNC(C1CCCOC1)=O)C(C)C)N1CCCC(OC)CC1 27660,C1(O)(CN(C)C)CN(C(=O)CCNC(c2cnns2)=O)C1 27661,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27662,N1(C(C(COCC)C)=O)CC(CC(=O)NCCn2cc(C)cn2)CC1(C)C 27663,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CCO)=O)cncc(F)c1Cl 27664,c1(C(N2CC(CC)N(C(=O)CCn3cc(Cl)cn3)CC2)=O)ccnc2ccsc12 27665,c1(OCC(N2CCC(C(C(=O)OC)Cc3cn(C)nn3)C2)=O)cncc(F)c1C 27666,c1(CCCC(=O)NC23C(CN(C(CC(=C)C)=O)C2)C3)csc2ccccc12 27667,c1(C(=O)NC2CC(C(C)NC(c3cc(C)ns3)=O)C2)ccc(Cl)nc1O 27668,Cc1nc(C(=O)Nc2ccc(C(N3CCC(F)(F)C3)=O)nc2)cc(O)n1 27669,Cc1cc(C(=O)NC2CCN(C(=O)CCC3CC3NC(=O)OC(C)(C)C)C2)cs1 27670,C(=O)(C#CC1CC1)N(C1CCCN(C(=O)CNC(=O)C=Cc2ccco2)C1)CC 27671,c12nc(Br)ccc1C(=O)N2.N1(C(C2CC(=C)C2)=O)CCCCC1C(N)=O 27672,c1(-c2cn(CC(CNC(c3ccc(CCC)[nH]3)=O)OC)nn2)c(F)cccc1F 27673,C#CCCC(C(=O)NC)NC(=O)C(C1CCC1)NC(C12CC(CO)(C1)C2)=O 27674,C(C1c2ccccc2CC1C)N(C(C(=O)N(CC(C)O)C)=O)C 27675,c1(C(=O)NCC(CN(C(C(C)C(F)(F)F)=O)C)O)cccc2c1N(C)C(=O)CO2 27676,O=C1NC(C(=O)NC23CC(C2)N(C(=O)CC2CCC(=O)N2)C3)CCO1 27677,CC(C)C#CC(=O)N(CC(C)NC(c1cnn(C)c1C1CC1)=O)C 27678,N1(C(C(CCC)NC(C2CC2(Cl)C(=O)OCC)=O)=O)CCN(C)C(CO)C1 27679,C(CN=c1cc[nH]cc1C#N)(C(C)(C)C)NC(C1N(S(C)(=O)=O)CCC1)=O.CCO 27680,OC1CCCCC(Cc2nc(-c3ccncc3)nn2CCCC(F)F)C1 27681,N1(C(c2cn(C(C)C)nc2)=O)CCCCC1C(C)(C)CNC(C1CS(=O)(=O)C1)=O 27682,C1(NC(C2(CC#C)CCOCC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1C 27683,N1(C(COCC#C)=O)CCCC1CN(C(C1(C#C)CC1)=O)C1CC1 27684,CC1CCC(C)(C(N2CC3CC2C(NC(=O)CCOCC2CC2)C3)=O)CC1 27685,c1(C(C(=O)NCC2CCOC2)N(CCC)CC)cncc(OCC2CC2)c1 27686,CC1(C)C(C(=O)NCC(CO)NC(=O)CNC(N)=O)CC1(F)F 27687,CC1=NC(C)(CNC(C2(CCNC(=O)Cn3cnc(=N)[nH]3)CCC2)=O)CS1 27688,C(=O)(CC(C(F)(F)F)N(C(c1[nH]ccc1C1CC1)=O)CCO)N(c1cccnc1)C 27689,C(=O)(CS(=O)(=O)CC1CCCO1)N1CCC(C(C)NC(C2COC(=O)O2)=O)CC1 27690,c1(C(n2cc(-c3ccc(Br)s3)nn2)C)nnsc1-c1ccccc1 27691,C1(NC(c2csc(CO)n2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC12CCC2 27692,C1(C(=O)NC2CCCN(C(Cc3c(C)ccnc3)=O)C2)CCC([N+](=O)[O-])CC1 27693,n1(CC(C)NC(=O)Cc2nc[nH]n2)cc(CN(C(=O)C(F)CC2CCOC2)CC)nn1 27694,CCC(C)C(C(=O)NC(c1nncs1)C)NC(C1C2CCC(F)C12)=O 27695,c1(SC)ncc(C#N)c(N2CCN(c3ncc(C)cn3)C3CC23)n1 27696,c1(C(N2CCCN(C(CC(=C)C)=O)CC2C)=O)cccc2c1OCC2C 27697,N1(C(c2c(OC)csc2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1C(C)C 27698,c1(C(=O)NCC2CCCC(NC(CC(=O)OC)=O)C2)cc(N)ccc1Br 27699,C(F)(C(=O)NN1CCCC1C(=O)NCC1CCCOC1)=C(C)C 27700,CCC(C)CCCCC(=O)N1CCC(C)(C(=O)NCC2CC=CC2)C1 27701,S(=O)(=O)(c1ccc(CNC(=O)C(=O)NC2C(O)CC2O)cc1)NC 27702,N1(CC)CCC1C(=O)NC1(CC(=O)NC2(c3cc[nH]n3)CC2)CC1 27703,c1(C(N(C)CC2N(C(C(C)n3ccnc3)=O)CCC2)=O)cn2c(n1)C(C)CCC2 27704,C1(NC(=O)CC2CC3CC3C2)CN(C(=O)Cn2nccn2)C2(CCC2)C1 27705,C=CCC(CNC(=O)C(C)OC(C)=O)C(=O)NC(C)(CC)CC 27706,C1(CC(=O)NC(CN(C(COC(C)C)=O)CCO)C)CCOC1=O 27707,c1(N2C3CC(O)CC2C3)ccc2c(c1)CCN2c1ncccn1 27708,C(CO)(CCCCNC(c1cc(C)[nH]n1)=O)NC(C=C(CC)C)=O 27709,Cc1nc2c(o1)CCCC2CC(=O)NC1CCN(CCC2CCOCC2)C(C)C1 27710,Nc1cc(C(=O)NC2(CNC(C3CC34CCCOC4)=O)CC2)cc(F)c1 27711,CCS(=O)(=O)CC(=O)N1CC(C(N2C3CCCC2CC3)=O)CC1(C)C 27712,C=CCC(C(=O)NCC(CC)OC)NC(=O)Cc1cc(C)cs1 27713,C1(C(N2CCC(O)(CNC(c3cnc(C)o3)=O)C2)=O)CC(C)(C)CN1C 27714,Cc1ccc(NC(c2ccc(C(=O)NOCc3cc(Br)ccn3)cc2)=O)cc1 27715,C1(CNC(CC2(CC)CC2)=O)C2CN(CC(=O)Nc3cncc(Cl)n3)CC12 27716,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27717,C(=O)(C(C(C)O)N(C)C)N1CC(O)(CNC(C(C)c2cccs2)=O)C1 27718,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2C(=O)Nc1cnc(C2CCCC2)nc1 27719,CC(CS(C)=O)C(=O)NCCCCCN1CCCN(C(=O)C(C)(C)C)CC1 27720,c1(C(N2CCC(NC(CCCNC(C)=O)=O)C2)=O)cccc(C)c1N 27721,C1(C)(CNC(C2OCC(C)C2)=O)CCCN1C(C1CCN(C)C1C)=O 27722,N1(C(c2ccc(CNC(C(CCC=C)(C)C)=O)cn2)=O)CCc2c(O)noc2C1 27723,Cc1ccc(O)cc1C(=O)NC(CNC(=O)CSc1ccccc1O)CO 27724,C(CC(C(=O)NC1CCC(C)CC1)NC(=O)CC1(CSC)CC1)SC 27725,C(C(=O)NCCCc1c[nH]nc1C)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27726,C1(C(N(c2c(C)n[nH]c2)C)=O)CC12CC2(F)F 27727,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27728,c1(C(N2CCCC(NC(CC(=C)C)=O)CC2)=O)c(F)ccc(O)c1F 27729,C1(NC(CCc2onc(CC)n2)=O)CC12CCN(C(=O)CCc1cnn[nH]1)CC2 27730,N1(C(C(CC)(C)OC)=O)Cc2cccc(CNC(c3ncc(C4CC4)[nH]3)=O)c2C1 27731,C(CC(C)C(=O)N(CC(C)NC(=O)C(c1cnn(C)c1)=O)CC)=CCC 27732,Cc1nc(C2CC2)oc1C(=O)NCC1CN(C(C2CC2c2ccc(F)cc2)=O)C1 27733,S(=O)(=O)(c1ccc(OC)c(-c2ccc(OC)cc2CC)c1)N(CC#C)CC=C 27734,N1(C(c2ccn(CC)c2C)=O)CCC(C)C(NC(=O)C(C)(O)C2CCC2)C1 27735,C1(N(C(CCOCCC)=O)C)CN(C(=O)Cn2c(C)c(C)sc2=O)CC1(C)C 27736,C1(C(=O)NC(C2(CNC(=O)C(O)CC3CCCC3)CC2)C)CCNC(=O)C1 27737,C1(C(=O)NCC2CC3CC2CC3O)CCCN(C(C23C(=O)C4CC2C3C4)=O)CC1 27738,c1(CC(=O)NCCNC(c2nc(COCC)sc2)=O)ccc(S(C)(=O)=O)cc1 27739,c1(OCC(=O)NCCOc2ccon2)cc(F)cc(F)c1.C12CCCN1C(=O)C2C 27740,C1(C(=O)NCCOCCOCCOC)(C(C(C2CCC(CC)CC2)=O)=O)CC(C)(C)C1 27741,c1(CNS(Cc2c(C(C)(C)C)cccc2)(=O)=O)ccc2c(c1F)OCCO2 27742,c1(C(N2C(CNC(C3CCNC3=O)=O)CCCC2)=O)ncn2ccccc12 27743,N1(Cc2ccc(CC(=O)Nc3cc(Br)cc(C)c3Cl)[nH]2)CCC2(CCCCC2)CC1 27744,C(=O)(CCCCNC(c1cc(C2CC2)n[nH]1)=O)NCC1C(OCC)CC1 27745,c1(C(C(=O)NC)N(C2C3COCC23)C)ccc2cc(F)ccc2n1 27746,N1(C(C2C(CC)OCC2)=O)CC2(CC(CC(=O)NC(COC(C)=O)CO)C2)C1 27747,C1(OC)(NC(c2cc(F)ccc2N2CCN(C)CC2)=O)CCC(C(=O)O)CC1 27748,c1(NC(=O)COC)ncccc1Cl.C(C=O)(C1CCOC1)SC1CC1 27749,C1(C(=O)NCC(CC)NC(CSCCC)=O)CC2(C1)CC1(CCC1)C2 27750,Cc1nnc2n1CC(c1nc(C3CC=CCC3)nn1-c1cnnn1C)CC2 27751,c1(C(=O)NC2C3(CC(NC(c4c(C)scn4)=O)C3)C2)c(C)nn(CCO)c1C 27752,C1(NC(C2CCOCC2)=O)CCN(C(=O)C(F)(F)C(O)C2CCC2)CC(O)C1 27753,c1(C(N(CC(C)(C)NC(=O)CC2CCCCN2C)C)=O)ccc(N)c(Cl)c1O 27754,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(c2conc2C)=O)C1 27755,C1(O)(CNC(C(C)OCCOCC)=O)CCN(C(c2scc(C)c2C)=O)C1 27756,c1(C(=O)NCC(C)N(C(c2ccoc2)=O)CC)cocc1C 27757,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(C1CC(C)(C)C1)=O)=O 27758,O=C1CCc2ccc(C(=O)NC3CCCC(NC(c4n[nH]cc4Cl)=O)C3)cc2N1 27759,c1(N)ccnc(C2CC2)c1C.C1(COC)CCCCC1n1ccnn1 27760,C(C(=O)N1CC(O)(C(F)(F)F)C1)(C(C)(C)C)NC(c1cc(C)sc1)=O 27761,C1(C(N2CC(F)(CNC(=O)Cc3ccc(F)cn3)C2)=O)C2CC3CC(C2)CC1C3 27762,N1(Cc2c(C#N)scc2)CCC2(CC1)CCN2C(c1ccc(F)cc1)=O 27763,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27764,N1(C(C2=CC(C)(C)C2)=O)CC2CCC(C(=O)NCCCc3ccsc3)(C2)C1 27765,C(C(CNC(=O)CN1CCCCC1=O)C(F)(F)F)NC(CC1C(C)C1)=O 27766,N#Cc1cc(C(=O)NC2CC2NC(c2ccn(C3CCCC3)n2)=O)c[nH]1 27767,N12CCOC(CC1)C2=O.C#CC1(C(=O)NC(COC)COC)CCCC1 27768,O=C(CC(F)(F)F)NCC1CC1NC(c1csc(C2CCCCC2)c1)=O 27769,N1(c2cccc(CNC3(c4n(CC(=C)C)nnn4)CCCC3C)c2)CCC(F)(F)CC1 27770,C1(NC(CCC)=O)CCCC(NC(=O)C(c2ccc(Cl)cc2)(C)N(C)C)C1 27771,C1(NC(c2ccc(CNC(C(C)S(C)(=O)=O)=O)cc2)=O)CN(C)CCN(C)C1 27772,c1(C(=O)NCCCN(C(=O)Cc2ccc(C)cc2)CC)cc(F)ccc1O 27773,C1(C(CC)=O)CC(CC(N2CC(Cn3cc(Cn4ccnc4)nn3)C2)=O)CCO1 27774,C1(CNC(C2(CCOC)CCCC2)=O)CCN(C(c2nnc(C)s2)=O)C12CC2 27775,c1(OC)ccc(F)c(C(N2CCCC(NC(=O)CN3CSCC3=O)C2C)=O)c1N 27776,C1(C(=O)NCCCN(C(c2cnn(CC)c2C)=O)C)CC12CCCCCC2 27777,N1(CC(=O)N(CC(C)C)CC(C)C)CC(C(=O)NCC2CCCO2)C1 27778,N#Cc1ccc(C2CCN(c3nnc(-c4ccc(Br)cn4)o3)CC2)cc1 27779,c1(N(C(=O)C#CC2(C)COC2)CCNS(C)(=O)=O)nc2ccccc2[nH]c1=O 27780,CC1(C)CCN(C(C2CC23CCOC3)=O)C1CNC(c1cc2n(n1)CCO2)=O 27781,Cc1ccc(NC(CC(=O)NCCc2cnn(C)c2)c2ccccc2)cc1C 27782,C1(CCC(=O)NC2(CCNC(c3cc(C(C)=O)sc3)=O)CC2)CCCCN1C 27783,C1(OC(CC)C)C2CC(NC(C3(C)CC(C#N)C3)=O)CC12 27784,Oc1nc(CCO)oc1-c1nc(C2CCC2)nn1-n1cccc1 27785,Nc1cnnc(I)c1C(=O)NCCNC(=O)C(O)C1CCCC1 27786,C#CCCCCC(=O)NC12CC1CN(C(=O)C(C)Cc1ccc(C)cc1)C2 27787,c1(CN2CCCC(N(C)C)C2)ccc(C(=O)Sc2ccccc2)c(F)c1 27788,CC(C)(C)CCCCC(=O)NC1(NC(=O)Cc2cccc(Br)c2F)CC1 27789,C1(C)(COCC)CC(NC(c2nn[nH]c2Cl)=O)CN1C(c1n[nH]c2c1COC2)=O 27790,C(=O)(C(C(C)(C)O)NC(c1nocc1C(C)C)=O)NCCCc1nnc(C)s1 27791,C1(CCNC(c2n(C=C)ncc2)=O)CC2CCC(C1)N2C(C1CCN(C)C1C)=O 27792,c1(C(N2CCC(C(C)(C)NC(C3OCCCO3)=O)C2)=O)cn2c(n1)CCC2 27793,C(=O)(C(CC1CCC1)NC(=O)C(C)N(C)C)NCC(=O)N(C)C1CC1 27794,c1(C(=O)NCC2C(NC(c3cc(C)nc(C)n3)=O)CCC2)cnc2ncccn12 27795,C(=O)(C1CCc2snnc21)N1C2CN(C(CN(S(C)(=O)=O)C)=O)CC1CC2 27796,O=C1CCCC(C(=O)NCc2cc[nH]c2C(=O)N(C2CCC2)C2CC2)O1 27797,Cc1ccc(C(=O)NC(C)CCCNC(C2C=CCC2)=O)c(C)c1 27798,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(C1CC1c1cn[nH]c1)=O 27799,c1(C(N2CCC(C3CCCN3C(c3occc3F)=O)C2)=O)ccc2ncnn2n1 27800,N1(C(c2c(CC)nc(CC)s2)=O)C2CCC1CN(C(=O)Cc1c(C)noc1Cl)C2 27801,Cc1cnc(Cl)c(CN2CCC2(C)C(=O)NCc2ccc(F)cc2C)c1 27802,c1(C(C)(C)C)ccc(N2CCC3CN(c4nc(Cl)ncc4F)CC23)c([N+](=O)[O-])c1 27803,C(N=c1[nH]c(C)c(C(=O)NCc2ccsc2)s1)c1c(OC)cncc1 27804,Cc1cc(C(=O)NCC2C(C)CCN2C(c2ccnc(Cl)c2O)=O)cnc1C 27805,c1(CC(=O)NCCC(C)CO)csc(=NCc2ccc(O)c(Cl)c2)[nH]1 27806,C1(OCC(C)(C)C)(C)CCCN(C(=O)CC(C)CC)C1.c1(CCC(=O)N)nccn1C 27807,Cc1ccc(C(=O)NC23CC(NC(=O)C(Cl)(Cl)Cl)(C2)C3)c2ccccc12 27808,c1(CC)ccc(OCC(N2CCC(CNC(=O)CC(C)F)CC2)=O)cc1 27809,N1(C(Cn2ncn(C)c2=O)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C2C1 27810,C1(NC(c2c(NCC)scn2)=O)CC2CC(NC(C3CCC3)=O)CC2C1 27811,N1(C(C(C2CCCC2)SC)=O)CC(F)(NC(=O)COc2ccncc2)C1 27812,c1(C(N2CC(COC)(CNC(=O)C(F)F)C2)=O)ccnc(S(N)(=O)=O)c1 27813,C12(CNC(C(CC)N(C)C)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 27814,CC1CN(C(C2C3CC4C(C3=O)C24)=O)CCC1C(=O)N(CC(O)CO)C 27815,N1(C(C2(OC)CCOC2)=O)CCC2(C=C(C(=O)Nc3ccc(C(C)C)nc3)C2)C1 27816,CCCCCC(CCCCC)C(=O)NC1CC2CCC(C1F)N2C(C1CC1F)=O 27817,c1(NC(Cc2nc(CC)sc2)=O)cccc(NC(=O)C(C)OC)c1 27818,Cc1ccc(-n2cc(Cl)cn2)c(NC(C2CCN(C(C3(O)CCC3)=O)CC2)=O)c1 27819,C12CCN(CC1F)C(=O)CN2.Cn1cc(Br)c(NC(=O)C2CC2)n1 27820,N1(C(C(CC2CCC(C)C2)(C)C)=O)CCOC2(C1)CN(C(=O)CS(N)(=O)=O)C2 27821,C1(NC(CN(C(C)C)C)=O)CC(O)CN(C(=O)CN2CCC(O)CC2)C1 27822,Cc1nnc2n1CC(C(N1CC3CCC(C1)N3C(C13CC(O)C1C3)=O)=O)CC2 27823,N1(C(C(C2CC2)NC(C(C2CCC(=O)N2)C)=O)=O)CC2CCC(C1)C(=O)O2 27824,C1(C(=O)Nc2ccc(SCC)cc2)CC2CCC1N(C(=O)C(C)(C)N1CCCC1)C2 27825,N1(C(=O)CC)CC2CCC(C1)C(=O)N2.c1(OC)cc(-c2ccc3cc2-3)cc(N)c1 27826,c1(CC(=O)N(C2CCS(=O)(=O)C2)CCOC)c(-c2ccccc2)coc1C 27827,c1(CNC(CCCN(C)C(C2CCCO2)=O)=O)ccc(C#N)o1 27828,C1(NC(c2c(CC)con2)=O)CCOC(CNC(=O)CCn2cnnn2)C1 27829,c1(CC(=O)NCCCCCCN(C(CC(CCC)C)=O)C)ccc(S(C)=O)cc1 27830,C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1cc3n(n1)CCCN3)=O)C2 27831,N1(C(C(C)SCC(F)(F)F)=O)CC2C(CC(=O)CSCC)C2C1.N1(CCN)CCOCC1 27832,N1(C(C2(C(=O)OCC)CC2)=O)CCC(NC(=O)CC2CCCC2C)C1C 27833,C1(CC#C)(C(=O)NCCC(C)NC(c2coc(Br)n2)=O)CCOC1 27834,N1(C(c2ccc(CC)cc2C)=O)CC(C)N(C(c2cnc(S)nc2)=O)CC1C 27835,C1(NC(CC(C)n2ccnc2)=O)C2CC3CN(C(=O)Cc4cnsc4)C1C3C2 27836,Cc1oc([N+](=O)[O-])cc1C(N1CC2CCC1CC2NC(=O)CC1=CCCC1)=O 27837,c1(C(=O)NCC2C(C(=O)NCC(CO)N(C)C)C2)ccc2ccccc2n1 27838,Cc1oc(CO)cc1C(=O)NCC1(C)CCCN1C(=O)COCc1nc[nH]n1 27839,N1(C(Cc2c(CC)con2)=O)CC(NC(=O)Cc2ccsc2C)C(C)(C)C1 27840,CC(C)(CCC(=O)NC1CCCC(O)CC1)NC(=O)CCCC1CCC1 27841,CC1CCN(C(=O)CCC2CCN(C(C3(O)CC4CCC3C4)=O)C2)C(C(=O)CCl)C1 27842,C1(C(=O)NC2CCC(CNC(c3[nH]ccc3CC3CCC3)=O)C2)CCS(=O)(=O)CC1 27843,c1(C(=O)NC(C)CCN(C)C(C2CCCC2(C)C)=O)cnc(N)c(Br)c1 27844,O=C(C(O)C(F)(F)F)N1CCN(CC2CN(C(C3(C(F)F)CCCO3)=O)C2)CC1 27845,N1(C(C(CN(C)C)NC(=O)C=CCF)=O)CCCC(F)CC1 27846,C(=O)(C(CCCc1ccc(OC)cc1)N(C(C)CCC(N)=O)C)NCCCOC 27847,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 27848,c1(C(N)=O)cccc(C(=O)NCC(F)CNC(C2(c3ccc(F)cc3)CC2)=O)c1 27849,c1(SC)nc2ncnc(NCC3(F)CCN(C(=O)C(C)C4CCCO4)CC3)c2s1 27850,C1(CNC(C=CC)=O)CC(C(F)(F)F)CCN1C(=O)CCSCCNC(C)=O 27851,c1(OC)ccc(OC)c(CC(=O)NCC2(NC(C3CCC(C)O3)=O)CC2)c1 27852,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccsc2)cc1N 27853,C1(C(=O)NCC(C)NC(=O)Cc2cn[nH]c2)CCCN1Cc1c[nH]c(=N)s1 27854,c1(COCC(=O)O)ccc2c(c1)CN(C1CCN(c3ccccc3)CC1)C2=O 27855,N1(C(C2C(C)OCCC2)=O)CCN(C(c2sccc2Cl)=O)CC(C)(F)C1 27856,C1(C(=O)NCc2ncoc2C2CN(C(C3CCCSC3)=O)C2)CC2COCC2C1 27857,CCCS(=O)(=O)C(C)C(=O)N(C(C)CCNC(c1cc2sccc2n1C)=O)C 27858,N(C1CCc2c(Br)cccc21)C(C)CNC(C1(O)CN(C(=O)OC(C)(C)C)C1)=O 27859,c1(SC)ccc(NC(N(CC(F)(F)C(C)C)C(CC)C)=O)c(C)c1 27860,c1(C(=O)NCC(C)(CO)NC(c2cncc(OC)n2)=O)nccc2cccnc12 27861,c1(C(C(=O)NCCCN(C(C(C)CO)=O)C)O)ccc(Cl)c(F)c1 27862,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CNC(=O)C2=COCC2)C1 27863,CN1C(CNC(=NCC2CCC(O)CC2)NCc2ccccc2)CCS1(=O)=O 27864,c1(CCCC(=O)NCC(c2ccccc2)C2OCCO2)ccc(F)cc1 27865,N12CC(C(O)C1)CN(C)CC2=O.c1(CNC(c2cc[nH]n2)=O)ccccc1 27866,CN1c2ccccc2CC1CNCC1(CN)CC1.c1(C)c(F)ccc2[nH]ccc12 27867,C1(NC(C2C(C(C)C)OCC2)=O)CCN(C(=O)CC2COCC(C)O2)C1C1CC1 27868,N1(C(C=C(C)C(F)F)=O)CC2(CCC2NC(=O)C(C(C)(C)C)NC(N)=O)C1 27869,c1(OCOC(C(=O)OC)Cc2ncc(C)cn2)ccc(OC)cc1Cl 27870,c1(NC(c2c(C(=O)NCCN3CC(OCC)C3)cco2)=O)cc(C)cc(C#N)c1 27871,CN=c1[nH]cc(C(=O)N(C2CCN(C(=O)CCc3ccncn3)C2)C)s1 27872,c1(CC)[nH]c(=N)sc1C(=O)NCCN(C)C(c1ccncc1C)=O 27873,N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)C(C)NC(=O)NC)CCO2 27874,c1(COC)ccc(-c2csc(NC(C)=O)n2)cc1.C1(=O)CCCCOCCN1 27875,c1(CN2CC(C#N)C(CC)C2)ccc2nc(O)[nH]c2c1 27876,C(=O)(CC1=CCN(C)CC1)NCC(C#C)NC(=O)COC(F)(F)F 27877,c1(C(=O)NC2C(NC(c3c(C)cc(C(F)(F)F)s3)=O)CCC2)cccc2cncn12 27878,CC1CCCCC1C(=O)N(C1CCCCC1)CCCNC(=O)COc1ccccc1 27879,CCCCCC(O)C(=O)N1CCCC1C(=O)NCC(n1cc(C)cn1)C 27880,C1(C(=O)NC2C=CC(CNC(c3csc(C4CC4)n3)=O)C2)CC2(CCCO2)C1 27881,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(C2CC(=O)N2)=O)CC1 27882,c1(CC)cc(NC(=O)C(O)C2CN(C(=O)C(C)C(F)(F)F)C2)ccc1C 27883,c1(C(=O)NC2CN(C(c3c(CC)nc[nH]3)=O)CC2CC)ccc(C)nc1N 27884,C(=O)(C(C(C)(C)C)NC(C1CNC(=O)N1)=O)N(CCCN(C)C)CC 27885,Cc1[nH]nc2c1CCC(C(=O)NC1CN(S(=O)(=O)c3ccc(Br)cc3)CCC1C)C2 27886,C1(O)(CNC2C(N(C)C)CC2)CCN(Cc2ccccc2N2CCCC2=O)C1 27887,c1(OC)ccccc1NC(=O)C(N1CCN(CC2CC2)CC1)c1scnc1Cl 27888,C1(NC(=O)CC2CC3(CC3)C2)CC(CNC(c2csc(Br)n2)=O)C12CCC2 27889,c1(-c2nc(CC3CC(OCC)C34CCCC4)on2)cc(N=S(C)(C)=O)ccn1 27890,N1(C(C(C(C)C)NC(C)=O)=O)CCCC2(NC(c3ocnc3C)=O)CC2C1 27891,C1(C(C)C)CN(C(=O)C(CC(F)F)C2CCC2)CC(=O)N1 27892,CCCCS(=O)(=O)N(CC(N1CC(O)(CNC(=O)C=Cc2cccnc2)C1)=O)C 27893,C(=O)(N1CC=CCO1)C1(C(F)F)CCC1.C12CCN(CC1)NC2=O 27894,c1(C(=O)NCC(C2(O)CCN(C(=O)CCCF)C2)C)ccc(C2CC2)cc1F 27895,S(=O)(=O)(c1[nH]c(=NCCCCC(C)(C)N(CCCC=C)C)ccc1Br)NC 27896,N1(CN2CCC(n3cc(CNC(c4ccc(CSC)o4)=O)nn3)C2)CCCCC1=O 27897,N1(C(CC(C)(C)SC)=O)CCN(C(c2cc(C)nc(O)n2)=O)C2CCCCC12 27898,N1(C(CN2CC(C)(C)SCC2)=O)Cc2[nH]nc(NC(=O)CN3CC(=O)NC3=O)c2C1 27899,C=CC1CN(C(=O)CC(CC)NC(=O)CCCCCC)CCO1 27900,CCC(C)(C)CCCC(=O)N1CC(C(N2CC(N(C)CCO)C2)=O)CC1(C)C 27901,Cc1cc(Br)oc1C(=O)NCCn1cc(C2CCCN2C(C2C3COCC23)=O)nn1 27902,C1(COc2cc(OC(F)F)ccc2C)CCCCCN1C(=O)NC(CCCOC)=O.O 27903,c1(C(=O)NCC(CNC(c2c(N)nc(Cl)cc2)=O)CO)ccc2nonc2c1 27904,CCC(C)C(O)C(C)C(=O)NC1CCCCC1CC(=O)NC12CCCN(CC1)C2 27905,C1(C(N(C)CC2CN(C(c3cn(C4CC4)nn3)=O)CCO2)=O)CCC=CCCC1 27906,C1(C(=O)NCC2CN(C(c3cnc(CC)s3)=O)C2)NC(=O)OC1C 27907,C(CN=c1nn[nH]n1-c1ccccc1)N(C1CCC(C(=O)C2CC2)O1)CC 27908,C1(CCNC(=O)NC2(NS(CC)(=O)=O)CC2)COC(C)(C)CO1 27909,N1(C(CCC(CC)CC)=O)CC(C2CCCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 27910,c1(C(N2CCC(NC(C(CC3CC3)OC)=O)C(O)C2)=O)cc2ncccc2[nH]1 27911,C12(NC(C(CC)NC(C)=O)=O)CC(CNC(=O)N)(C1)OC2(C)C.c1ccc(=O)oc1 27912,C12(NC(C3CC(OCC)C3)=O)CCOC(C)(C1)C2.c12ccc(cc1)CC(=O)NC2 27913,C1(CC(=O)NC(C(=O)OC)CC2CCCC2)CCNC2(CC2)C1 27914,N1(C(C(C)(C)OC)=O)CCC(C2CCCN2C(=O)C(c2ccc(F)cc2)F)CC1 27915,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 27916,C1(n2cc(C3(F)CCN(C(C(C)NC(COC)=O)=O)C3)nn2)CCCS(=O)(=O)C1 27917,C1(C(=O)N(C(C)(C)CC2CC2)CCO)CCCN(C(=O)CSC(C)(C)C)C1 27918,C(C(C)(C)C(=O)N1CCCC(C(C)(C)C)C1)N(C(C(C1CC1)OC)=O)C 27919,C(C[Si](C)(C)C)NC(CN(CC#C)C(c1cc(Cl)cs1)=O)=O 27920,C(CC(N)=O)(C(=O)NC1(CC(=O)OC)CCC1)NCc1nccc(CC)c1 27921,c1(C(=O)NCC2CN(C(CCSCC)=O)CC2O)cc(CC)cnc1O 27922,N1(C(c2cnc(COC)s2)=O)CCC2(NC(=O)CSS(C)(=O)=O)CCCC12 27923,N1(C(CC2(OC)CC2)=O)CCC(C2CCN(C(c3sccc3C)=O)CC2)C1 27924,c12cccc(c1)C2.Cc1sccc1CC(=O)NC1COCC1n1cc(C(=O)O)nn1 27925,c1(C(N(C(CCNC(c2nn(CC)c(O)c2)=O)C)C)=O)cc(F)ncc1N 27926,N1(C(=O)NCC)CCC(C(N2CC(N(C(=O)CC(F)F)C)C2)=O)C1 27927,c1(-n2cc(C(C)NC(C3C=CCS3)=O)nn2)ccc2ncc(Br)cc2c1 27928,N1(C(C(n2ccc(C)n2)C)=O)CCC(C(=O)NC(C)CC#N)CC1C 27929,N1(C(Cc2n(C)cnn2)=O)CCC(CNC(C2CC(n3cnnc3)C2)=O)C12CC2 27930,C1(NC(c2c(C)cc(SC)o2)=O)CN(C(C2CC3C=CC2CC3)=O)CC1(F)F 27931,CCCCCCC(C)(c1nnnn1CCSC)NC1CCC(C)CC1 27932,C=CC(C)(O)CC(=O)NCC1CCCCN(C(c2nc(OC)ccc2OC)=O)C1 27933,c1(NCC(C2CC2)NC(c2cc(C)sn2)=O)nnc(C)c(C)c1C#N 27934,C=C(C)C(C)(C)C(=O)N1CCC(CN(C)C(c2cn(C)nc2SC)=O)C1 27935,N1(C(=O)Nc2cccc(C)c2F)CCC2(C1)CN(c1ncc(Br)cn1)CCO2 27936,c1(CN=C(NC(=O)NC2CCCO2)NC2CCS(=O)(=O)C2)ccc2c(c1)OCCCO2 27937,N1(c2c(C(C)C)cnc(Cl)n2)CCC(C)C(NC(=O)CC23COC(C)(C2)C3)C1C 27938,N1(C(Cc2[nH]c(=N)sc2)=O)CC2CCCC(CNC(=O)NCC3CCCO3)(C2)C1 27939,C(=O)(C1=CCS(=O)(=O)C1)NC1C(C)(C)CCCC1.N12CCOCC1C1(C2=O)CC1 27940,C#CCCCC(C(=O)Nc1ccc(C(=O)OC)cc1)N(C1COC1)C 27941,c1(-c2onc(C(O)CC3CCS(=O)(=O)CC3)n2)ccnc2c(I)cnn12 27942,Cc1c(C(=O)NCC2CCN(C(=O)C(F)=C3CCCC3)C2)cnn1CCO 27943,c1(OC)c(C(=O)N(C2CC2)CC2CCCN2C(C2C=CCC2)=O)cccc1Cl 27944,CC1CN(C(c2cnn3c2SCC3)=O)CC(C)N(C(c2ncnc(O)c2Cl)=O)C1 27945,C(=O)(C(F)C(F)(F)F)N1CCC(CCCCNC(C(c2cncnc2)C)=O)CC1 27946,N1(C(C2CC2F)=O)CCC2(CC1)CN(C(=O)Cc1c(F)cccc1Cl)CCC2O 27947,c1(C(=O)NC(C(C(C)C)NC(Cc2c(C)ocn2)=O)C)ccsc1S(C)(=O)=O 27948,N1(C(C2CCOC2(C)C)C(=O)NC(C(=O)OC)C)Cc2cnc(N(C)C)nc2C1 27949,Cc1ccc(N)c(C)c1C(=O)NC1CCC1NC(=O)CC(C)c1ccsc1 27950,CCC(CC(=O)N(CC(C)C(=O)NCC1CC1(C)C)C)CC(C)C 27951,C1(CNC(C2N(CCC(=O)OC)CCC=C2)=O)CC(=O)N(C)C1=O 27952,C1(CNC(C(CCCC)C)(C)c2nnnn2CCCF)Cc2ccccc2CO1 27953,c1(C(N2C(C(=O)NC3(c4cc(F)cc(Cl)c4)CC3)CC(O)C2)=O)n[nH]cc1[N+](=O)[O-] 27954,N1(C(CCCn2c(C)ncc2)=O)CC(NC(=O)CC2COCCO2)CC(C)(C)C1 27955,CON1CC(C(=O)NCC(C(=O)NC(C2(CO)CC2)C)N(C)C)CC1=O 27956,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)NC(c2nncs2)C)CC1 27957,C12(CNC(CC=CC=C)=O)CCCCC1CN(C(c1ccc(CO)c(Cl)c1)=O)C2 27958,C(CCSC)(C(=O)NC(C)CN(C)C)NC(Cn1ncc(C(=O)OC)c1)=O 27959,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 27960,N1(C(c2cnco2)=O)CC2CCN(C(c3ccc(-n4cnnn4)cc3)=O)C(C2)C1 27961,CC1(C)CC1(C#N)C(N1CCOC(CCNC(c2nc[nH]c2C(F)(F)F)=O)C1)=O 27962,c1(C(=O)NCC2C(C)CN(C(c3nsc(C(C)(C)C)n3)=O)C2)cc(C#N)cn1C 27963,c1(C(=O)NC2C(C)(C)CCN(C(C3(C)COC3)=O)C2)cc2nn[nH]c2cc1F 27964,C(=O)(C1=CCCC(C)(C)C1)NCCCNC(c1c(C)nc(N)cn1)=O 27965,CC(C)(C)C(CNC(C1CCC(C(N)=O)C1)=O)NC(c1cc(C2CCC2)on1)=O 27966,N1(C(c2cnn(C)n2)=O)CCCC(C2CCCCN2C(=O)COCC2CC2)C1 27967,c12ccc(cn1)NC(=O)C1CN(C1)C2=O.c1(C)ccc(O)cn1.C1(N)CCCCC1 27968,CN(S(=O)(=O)N1CC(O)COCC1C)Cc1ccsc1 27969,Cc1csc(CC(=O)NC(C(=O)NCC2(S(C)=O)CC2)C2CCCC2)c1 27970,C12(CCN(C)CCF)CCC(F)(CN(C(=O)OC(C)(C)C)C1)C2 27971,C(=O)(C(O)CCC(C)(C)C)N(CC(=O)NC(C)CN(C(=O)CN(C)C)C)C1CC1 27972,C1(OC)(CNC(C2C3CCC(=O)C23)=O)CCN(C(c2cncc(N)c2)=O)C1 27973,C(=O)(C#CC1CCOCC1)NC1C(C)CN(C(C2CCS(=O)(=O)CC2)=O)C1 27974,C(=O)(CS(=O)(=O)CC(=O)NC(C)C)OC.C12CC3CCC1N(C3)C(=O)C(=O)NC2 27975,c1(N(C)C)ccc(N)c(C(=O)NCC2CC(F)CN2C(C2SCCCS2)=O)c1 27976,C1(C(=O)NC(C(C)C)(C)CNC(=O)CSC(F)F)CCCC(=O)N1C 27977,n1(CC#N)ccc(C(=O)NC2(C(=O)NCCC3C=CCC3)CC(F)C2)n1 27978,c1(CC)ccc(C(=O)NCC(C)CNC(c2cccn2CC)=O)cc1Cl 27979,c1(C(=O)NCC2CCN(C(Cc3nc(C)sc3)=O)C2)ccc2c(n1)CCC(C)C2 27980,Cn1ncc2ccnc(C(N3CCC(NCCN4CCNC4=O)CC3)=O)c12 27981,c1(C(=O)NC(c2c(C)nccn2)C)cnn2c1NCCC2 27982,Cc1nc(O)sc1C(=O)NC(C)(CNC(=O)C(=O)NCC(F)F)C(C)C 27983,N1(C(c2sccc2Br)C(=O)NCCCSCC)CCCC2(CO)CCCC12 27984,CC(C)C(CN(C)C)C(=O)NC(C)C=CC(=O)NCc1cccs1 27985,C(=O)(C(CCC1CC1)NC(C1CN(C(C)=O)C1)=O)NCCCCC=C 27986,C1(NC(c2cscc2Br)=O)CN(Cc2cncnc2)CC1(F)F 27987,c1(CNC)ccccc1CC(C)(COCC)C1CCC1.c12cc([nH]n1)C(=O)N2 27988,c1(N(CCN(C(C)=O)C)C)ncc(Cl)c(C)c1C#N.c12ccoc1C(=O)N2 27989,c1(C(C2CC2)NC(=O)C(N2CCN(c3nccs3)CC2)=O)cc(F)cc(F)c1 27990,N1(C(C2=CC(C)CC2)=O)CCC2(CC1)CCN(C(c1c[nH]nc1C(C)(C)C)=O)CC2 27991,c1(C(=O)NCCC2CCN(C(C3CCCC3F)=O)C2)ccn2ccnc2c1 27992,C(c1csc2ccccc12)=CC(=O)NC1CCN(C(=O)CN2CCCCC2=O)C1 27993,c1(C(N2CC(CNC(=O)CC(=O)NC3CC3)CC(C)C2)=O)cccc2ncnn12 27994,CC(C)CCCCCC(=O)NCC1CC1CNC(=O)Cn1cc(C2CC2)cn1 27995,c1(CC(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2)=O)cc(F)cc(F)c1 27996,c1(CN2C(C(=O)NCc3cc(F)ccc3F)CC(F)C2)ccc(I)cc1O 27997,C1(OC)CC(CC(N2CC=CC2Cn2cc(-c3cccnc3O)nn2)=O)C1(C)C 27998,C1(CC(=O)NC)CN(C(=O)C(O)CC(F)F)CCN1C(c1nc(C)sc1C)=O 27999,N1(C(C2OCCC(N(C)C)C2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC(C)(CO)C1 28000,C1(C(=O)NC2CC(NC(C3CCC(=C)CC3)=O)C2)CC(c2ccc(C)cc2)=NO1 28001,N1(C(c2cccc(C)c2F)=O)CCC2CN(C(=O)Cc3cnn(C(F)F)c3)C2C1 28002,Cc1c(C(N2CCC(NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)ncn1C 28003,N1(C(CC(N)c2ccccc2)=O)CCOCC(NC(c2ccsc2)C2CCC2)C1 28004,Cc1nc(Cl)ccc1CC(=O)NCC(O)CN(C)C(c1ccn(C)c1)=O 28005,Cc1ccc(C(CNC(=O)NCc2cc(C(=O)O)nn2C)NC(=O)C(C)C)cc1 28006,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28007,C1(C(=O)NCCn2cc(CNC(C(C)(C)CF)=O)nn2)CCOC(=O)CC1 28008,c1(CNCC(c2onc(C)n2)OC)ccc(OC(C)(C)C)nc1 28009,C12(CC(N3CCC(CO)C(O)C3)=O)CCC1CN(C(=O)CCCCN1CCCC1)C2 28010,C1(N(C)C(C2(C)CCC(=O)N2)=O)CCCN(C(C2(C)CC2)=O)CC1 28011,C1(CC(=O)NC(C(N2CC(C(=O)NCC)C2)=O)C2CCOC2)CCCCO1 28012,c1(C(N2CCC(NC(C3C(C)CCC3)=O)C2C(C)(C)C)=O)ccc2oncc2c1 28013,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28014,c1(Nc2cnc(SCC)nc2)ccc(Cl)c(O)c1 28015,C1(C(=O)NCC23C(CC(=O)N2)CCC3)CCc2cnccc2N1 28016,CC1CCCCC1(CNC(=O)Cc1sc(O)nc1O)NC(=O)CC1CCCCC1C 28017,c1(C(=O)NCC(C#C)OC)coc(CNC(C2(F)CCC2)=O)c1 28018,CCCCCS(=O)(=O)CC(=O)OCCC1(c2cc(OC)c(O)c(C=O)c2)CC1 28019,C1(NC(C(C)Sc2nncn2C)=O)CC(C)N(C(C2CCN2C)=O)C1 28020,N1(C(C2(N(C(=O)C(C)S(N)(=O)=O)C)CCN(C)C2)=O)CCC(C2(C)CC2)C1 28021,c1(C(=O)NCCCN(C(c2cncc(C=C)c2)=O)CC)cnc2scc(C)n12 28022,S(=O)(=O)(c1c[nH]ccc1=NCc1cc(O)ncn1)N(C1C(C)(C)C(O)C1)CCO 28023,N1(C(c2cncc(OCC)c2)=O)CCC(CNC(=O)C(C)c2ccsc2)C1(C)C 28024,c1(C(N2CCN(C(Cc3nc(C)on3)=O)C3C2C3)=O)cnc2cc(Cl)ccn12 28025,c1(CC(=O)NCC(CN(C)C(C2CC(C#N)C2)=O)O)ccc2ccncc2c1 28026,N1(C(C2CC(C)C2)=O)CCC2(CC1)CCN(C(=O)C=Cc1ccco1)CC2C 28027,CC1=C(C(=O)N2CC3CC2C3C(=O)NC23CCC(F)(CC2)C3)CCC1 28028,N1(C(c2c(CC)csc2)=O)CCC(CNC(=O)Cn2nc(C)oc2=O)C(C)C1 28029,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC(C)C)(F)F)=O)CC1(C)C 28030,c1(C(N(C(CNC(CN2CC(C)C2)=O)C2CC2)C)=O)cc2cc[nH]c2cn1 28031,C(C)(C)(CC(=O)NCC=C1CCN(C(=O)C(C2CCOCC2)O)CC1)OC 28032,c1(C(N2CCCC(NC(C(C)n3cnnn3)=O)C2)=O)ccc2c(c1)COC2 28033,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)C(C)n1cnnn1)C(C)C 28034,C(C(C)(C(C)C)NC(c1csc(-c2nc[nH]n2)n1)=O)NC(C1CN(C(C)=O)C1)=O 28035,C1(NC(c2n(C(C)(C)C)ncc2)=O)CCC(C)(CNC(=O)Cc2cnoc2)C1 28036,c1(C(=O)NCC2(NC(c3cnn[nH]3)=O)CCOC2)cccnc1SC(F)F 28037,CC1CCC(C)(NC(=O)CC=CCNC(C2C3COCC23)=O)C1 28038,c1(CC(N2CCC2CNC(C2CCC(F)CC2)=O)=O)ccc2c(c1)CCO2 28039,C1(C(N2CCCC2CNC(=O)CC2CCCC23CC3)=O)(OC)CCS(=O)(=O)C1 28040,C1(NC(C(C)N(C)C)=O)CCN(C(c2ccnn2CC#N)=O)CC1(C)C 28041,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28042,c1(OC(C)C)ccc(C(N2CCC2CNC(=O)CCN2CCC2)=O)cc1 28043,C1(CNC(C(C(CC)C)O)=O)CCCC2(CN(C(=O)Cc3cccc(Cl)c3)C2)O1 28044,Cc1c(-c2cn(CC(F)CCNC(C3CCCN3N=O)=O)nn2)cccc1F 28045,Cc1cccc2c(C(N3CCCC(N(CCF)C(C4CC4(F)F)=O)C3)=O)coc12 28046,N1(C(C2(c3ncco3)CCC2)=O)CCCC1(C)CC(=O)NCC1C(CC)CCO1 28047,N1(C(C(C(C)C)OC)=O)CCN(C(=O)Cn2nnnc2C(C)(C)C)CC12CC2 28048,Cc1cccc(C(=O)NCC2(F)CCC(CNC(C3(C)CC3(F)F)=O)CC2)c1C 28049,c1(C(=O)NC2(CO)CN(C(c3cc(Cl)ccc3Cl)=O)C2)cc2c(s1)CCSC2 28050,C(=O)(C(F)(F)CO)NCC1(F)CC(NC(Cc2c(C)ocn2)=O)C1 28051,c1(C(=O)OC)ccc(N(C)C)cc1C.n12cc(nn1)CNC(=O)C(=O)NC(C)C2 28052,CC1(C)CC(CNC(=O)CCCNC(N)=O)CN(C(c2ccccn2)=O)C1 28053,N1(C(C2(COC)CN(C(C3CC(=O)N(C)C3=O)=O)C2)=O)CCCC(C)CC1 28054,C#Cc1ccc(C(=O)NC2CCCC2CNC(=O)CCc2ccc(O)cc2)cn1 28055,CP(C)(=O)C(O)C(=O)NCCCO.c1(NC(=O)COC)ccc(Cl)nc1.C1CCCO1 28056,C#CC1CN(C(C2CCC2C#N)=O)CCN1C(c1cnc2[nH]nnc2c1)=O 28057,C(=O)(CCCCCCNC(=O)C(C)(CO)NC(C1(C)CN(C(C)=O)C1)=O)OCC 28058,N1(C(CN(C)C(N)=O)=O)CCN(C(=O)CC2(N3CCCC3)CC2)C(C2CCC2)C1 28059,c1(OC)ccc(C(N2CCSCC2C(=O)Nc2cc(I)ncn2)=O)c(C)c1OC 28060,C#CCC(C)(C(=O)Nc1c(NC)cccn1)NC(=O)C(C)CN(C)C 28061,Cc1c(F)ccc(CN2CCC(F)(C(=O)NCc3cccnc3)C2)c1Cl 28062,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C)OCCN(C)C)C1 28063,c1(C(=O)NC(CNC(c2cc(SC)oc2)=O)(C)CO)ccc([N+](=O)[O-])s1 28064,n1(CCC(N2CCC(CNC(c3ccc(CCC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28065,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C1CC(=O)N(C)Cc1cnc[nH]1 28066,C1(Cl)(C(c2nnnn2CC2CCOCC2)NC2(C(F)F)CC2)CC12CCC2 28067,C(=O)(CCN=c1[nH]ccs1)NCCC1CC(OC)CN1C(c1c[nH]ccc1=O)=O 28068,c1(N2CC(C)(CNC(C(CC)OC)=O)OCC2)ncnc2sc(C(F)(F)F)nc12 28069,C(=O)(C1=NOC(C)(C)C1)NCC(CN(C)C(C1C(c2ccccc2)C1(F)F)=O)CO 28070,N1(C(C(C)Cc2cnco2)=O)CCN(C(c2cnn(C)c2C2CC2)=O)CC1 28071,c1(C(=O)NC(C2(CNC(=O)C(F)C3CCCC3)CC2)C)cc(C)on1.C1CCC1 28072,C(=O)(C(C)(C)C(F)F)NC1CN(C(C2C(C)(C)C2(F)F)=O)CC1F 28073,N1(C(c2ccc(C)c(C)c2)=O)CCC(C2CC2)C1CNC(c1nsnc1O)=O 28074,N1(C(c2c(CC)ncs2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28075,C(CCCCCNC(c1nscc1Br)=O)NC(CC1N(C)CCC1)=O 28076,c1(C(=O)NCC#CCNC(=O)C=CC2CCCO2)cc2ccccn2n1 28077,c1(C(=O)NC(C)CCCNC(=O)CCS(N)(=O)=O)ccc2c(c1)CCC2(F)F 28078,S(=O)(=O)(c1ccc2c(c1)COCC2)CCC(N1CC2C(C)(C)C2C1)=O 28079,C1(C(=O)NCC2CCN(C(C3CCCC(C(N)=O)C3)=O)C2)(CC)CCC(O)CC1 28080,c1(C(=O)NCC2C(NC(c3ccon3)=O)CC2)cnn2c(-c3ccco3)ccnc12 28081,C[Si](C)(CCCCN1CCOCC1)C1CCN(C(=O)CC2CCCN2)CC1 28082,Cc1ccccc1CC(C)C(=O)NCCN(C(=O)CCN(S(C)(=O)=O)C)C1CC1 28083,CS(=O)(=NC(=O)CC1CNCCN1)c1ccccc1.c1(CS)ccccc1 28084,c1(NCc2cn(C3CCCN(C(C4C(C)(Br)C4)=O)C3)nn2)c[nH]cc(F)c1=O 28085,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28086,N1(C(c2c(C)[nH]nc2C(C)C)=O)CCN(C(=O)CC(C)(C)c2cccs2)C(C)C1 28087,c1(NCC(=O)NC(N(CCCOC)C)=O)cccc(C(N)=O)c1 28088,Cc1nnc2n1CCN(C(=O)NCc1ccc(C3CCC3)nc1)C2 28089,N1(C(C2CC(C(C)C)OCC2)=O)C2CCCC1CN(C(c1cccc(O)n1)=O)C2 28090,C1(NC(C(C)(C)C)=O)CC2CC(NC(C3CCCN(c4nccs4)C3)=O)C1C2 28091,C(=O)(C(CCCOC)NC(=O)C=C(C)C(F)F)NCCC.C12CCN1C2 28092,CCC(CCCC(=O)NC1(C(=O)NC)CCC1)OC.C12(CC1)C(=O)N2 28093,CCC(CC(=O)N1CCC(C(C)O)CC1)NC(=O)C(=CC1CCCC1)C 28094,NS(=O)(=O)CCC(=O)NCCn1ccc(C(=O)NCC2CCC(CO)C2)c1.C1(C)CC1 28095,Cc1nc(NC(=O)COC2CC2(C)C)ccc1COC(=O)C=CCF 28096,N1(C(C2(CCOC)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28097,C#CC1CN(C(=O)CC(CC)N(C(=O)C(C)CC(C)C)C)CCN1C 28098,N1(c2ncnc(-c3ccccn3)c2)CCCC(F)(CN=c2ccnc[nH]2)C1 28099,Cc1ccc(CN2C(C(=O)NCC3CCC(O)CC3)CC3CC23)c(Cl)c1Cl 28100,C1(C(N2CCC(OCCNC(C(COC)(C)C)=O)C2)=O)CCc2nccn2C1 28101,N(C1CC(C)n2ccnc21)C(N1C(Cc2cncc(C)n2)CCCC1)=O 28102,C1(N(C)C(C2CN3CCC2(C)CC3)=O)CCN(C(=O)COCC(F)(F)F)CC1(C)C 28103,C(=O)(C1Cc2ccc(Cl)cc21)N1C2CCN(C(=O)C3=CCCO3)CC2CC1 28104,C1(CC(=O)NC(C2CCCC2)CNC(C(N2CCOCC2)C)=O)CC2(CCC2)C1 28105,C1(CC)CCCN(C(=O)C(F)OC(F)(F)F)C1.C12(CCCC1)C(=O)N2 28106,N1(CC=C)CCCN(C(C2CC(C)N(C(=O)CNC(=O)CN(C)C)C2)=O)CC1 28107,C(=O)(C(C)(C)C(F)(F)F)NCCC1CCC(NC(CCC(=O)NCC)=O)C1 28108,CCCCCCCC(=O)N1CC(CNC(=O)C(c2ccc(Cl)cc2Cl)O)C(C)C1 28109,C1(N(C)C)CCCCC1C(=O)NC1CC(C)(NC(=O)C=Cc2cccs2)C1 28110,C1(C(N(C(CC)CC)C)=O)CC2CCC(C1)N2C(=O)C(C)N1CC(C)C1 28111,N1(C(COC(CC)C)=O)CCC2(CCCN(Cc3ccco3)C2)C1 28112,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CC)CC1 28113,N1(C(c2cccc(OC)c2N)=O)CC23CCCCC2(C1)CN(C(=O)CSC)C3 28114,Cc1ccccc1C(C)C(N1CCCC(CNC(c2cncn2C2CC2)=O)C1)=O 28115,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28116,C(CC(C(=O)NCC1(O)CCOCC1)NC(=O)CC1C=CCC1)OC 28117,c1(C(N2CCC(C(=O)NC(C)C(C)(C)OC)(OC)C2)=O)cnc(C)c(C)c1 28118,CC1C2CCC(C2)C1C(N1CCC(F)(C(N2CCC(C(C)C)(CO)C2)=O)C1)=O 28119,C(C1CCc2nccn21)NC(C1CC(C)(NC(=O)C2=CCCC2)C1)=O 28120,c1(-n2c(C3CCCN(Cc4cccs4)C3)nc(C(CC)C)n2)cc(C)ccc1C 28121,c1(C(=O)NC(CC=C)CNC(=O)CCC2CC2(C)C)ccc(C(F)F)cn1 28122,c1(COC)cncc(C(=O)N(C2CCCN(C(C34CC(C)(C3)C4)=O)C2)CCF)c1 28123,C(C(CNC(c1nnn(C)c1C)=O)S(C)(=O)=O)NC(c1occ(C)c1)=O 28124,C(C(CC1CC1)C(=O)NC1CCC=CCCC1)NC(CNC(CC)=O)=O 28125,CC(C)(C)CO.C1(C(=O)NCC(O)CF)C2(CCC2)CCC(=O)N1.C(C)(C)(C)O 28126,N1(C(C(c2ccccc2)C)=O)CCN(C(=O)C=CCn2cncn2)CC(O)C1 28127,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28128,c1(C(N(C)CC2CN(C(c3c(Cl)cn(CC)n3)=O)C2)=O)cnnc(C)c1C 28129,c1(-c2nc(C)c(NCc3cccc(O)c3C)s2)cc(F)c(C(=O)N(C)C)c(F)c1 28130,N1(CC(=O)NC(c2cn(CC3COC(=O)C3)nn2)(C)C)CCOC1=O 28131,C1(NC(C2(C(C)C)CCCO2)=O)CN(CCOc2ccccc2F)CC1C 28132,C1(NC(C(C)(C)C2CCNC2)=O)CC=C(C(=O)N2CCC2)C1 28133,C(C(C)C(=O)N(CCOCCOCCO)C(C)C)NC(C)C.C1(=O)C(C)N1 28134,N1(C(C(C)N(C)C(=O)OC(C)(C)C)=O)CCN(C(C2CCOCC2)=O)C2CCC12 28135,C(=O)(CS(=O)(=O)N(C)C)NC(C1CN(C(c2cn(C(C)(C)C)cn2)=O)CCO1)C 28136,N1(C(C2COCCN(C(c3n(C)nc(CC)c3Cl)=O)C2)=O)CCC(C)C(F)(F)C1 28137,N1(C(CC2CCN(C(CCCOC)=O)C2)=O)CC2(CSC2)C1 28138,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28139,N1(C(C(=O)NCCSCCOCC)C2CC2(Br)Br)CC(C)(C)C1c1ccccc1 28140,C1(CNC(C(CC)NC(C)=O)=O)(NC(C2CCCC(=O)CC2)=O)CCCCC1C 28141,C=CCC(CC(F)F)NC(=O)C(CNC(=O)Cc1ccsc1C)CC=C 28142,C1(C(=O)NCC(C)NC(C2CC23CCCC3)=O)CC2(CCO1)CC2 28143,C1(NC(C(c2ccc(Cl)nc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28144,CCS(=O)CC(=O)N(CCO)CCNC(=O)C(C)NC(=O)Nc1ccccn1 28145,n1(C(C(=O)NCCC(CCNC(CSCC=C)=O)C)C)ccc2ccccc2c1=O 28146,CC1=C(C(=O)N2CCCC2)C(c2cc(F)ccc2F)NC(=S)N1c1ccccc1F 28147,O(NC(=O)CN=c1[nH]c(=NCC2(C3=CCOCC3)CC2)[nH]c2c1SCC2)CC 28148,c1(C(=O)NC2C(NC(Cn3c(C)nnn3)=O)COC2)ccc(F)c(O)c1 28149,c1(NC(C(CCC)NC(=O)C(C)NC(C)=O)=O)cc2ccoc2cn1 28150,c1(C(=O)NC2CCCC23CN(C(c2cccnn2)=O)C3)ccc2nccnc2n1 28151,C1(C)(C(N2CC(NC(C(CCC)=CCC)=O)C(O)C2)=O)CCS(=O)(=O)CC1 28152,C(=O)(C(C)(C)CCC(=O)OC(C1CCCN(C(C2CC(=C)C2)=O)C1)C)N(CC)CC 28153,C1(C(N(C2CC(C(=O)NC3CCCC3F)C2)C)=O)CCOC1C1CC1 28154,C1(CN(C(c2cnc(C(C)=O)s2)=O)CC)CCCN(C(=O)Cn2cncn2)C1 28155,C(=O)(Nn1nnc2c1CCCC2)C1(NC(C(c2cccnc2)N(C)C)=O)CCC1 28156,C(=O)(C1=CC2(CCN(C(=O)Cc3cc[nH]n3)C2)C1)Nc1cn(C(C)C)c(=O)cc1 28157,c1(SC)cccc(Br)c1NCC1CC(C)(O)C1 28158,c1(C(N(C(C)C)CCNC(=O)CC2COCC2(C)C)=O)cc2nccnc2[nH]1 28159,C(CCC(CO)NC(=O)C=C=C(C)C)NC(C1(SC)CC1)=O 28160,C1CCC(C)(C)C(=O)N(OC)CCC(=O)N1.C=C=CCCOC 28161,CCC(C)C(O)C(C)C(=O)N1C2CCC1C(NC(=O)CCNC(C)=O)C2 28162,N1(C(C2C(OCC)C2)=O)CCCC(C)(C)C1CNC(c1cnn(CC)n1)=O 28163,C1(NC(=O)Cn2cncn2)C2CC(O)C1N(C(c1ccnnc1O)=O)C2 28164,N1(C(C2C(NC(c3c(CC)ccs3)=O)C2(C)C)=O)CCC(O)(CC)C1 28165,c1(C(N(CC(=C)Cl)CC)=O)csc(C2CCCCC2)c1 28166,C1(C(=O)Nc2c(C)nsc2C)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28167,c1(-c2cn(CC(C)NC(=O)CCCc3ccccn3)nn2)ccc(C(N)=O)cc1 28168,CC1(CO)COCCN(C(c2cnc(O)cc2O)=O)C1.C12OCCC1C(=O)NC2 28169,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28170,Cn1nnc(Cn2nnnc2C(c2ncc[nH]2)NC(C2CC2)C2CC2)n1 28171,Cc1nc(N2CCCC(NC(c3cc(C)c(F)cc3C)=O)C2)c2c(n1)CCC2 28172,CCC(C(=O)NC1(C)CCN(C(=O)CN(C2CCSC2)C)C1)C(C)O 28173,c1(C(=O)NCC(C)NC(c2ccc(OCC)nn2)=O)ccc(F)c(CO)c1 28174,N1(CC(=O)N(C2CCN(C(=O)Cn3ncn(C)c3=O)CC2)CC)CCCCCC1 28175,N1(C(C(CC)(C)O)=O)CCOC2(CCCN(C(C3CCC(C)CC3)=O)C2)C1 28176,C=CCC(C)(C)C(=O)NCC1(O)CC(NC(c2nnn(C)n2)=O)C1 28177,C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 28178,C1(C(=O)NC2(C(N3CCC(NC(C)=O)C3)=O)CCCC2)CCCCC(=O)C1 28179,N1(C(C(CCC)(C)O)=O)CC(C)(C)OC2(C1)CN(C(c1cc(Cl)ncc1O)=O)C2 28180,N1(C(CCOC)=O)CCC2(CCN(C(c3ncccc3N)=O)C2)C1 28181,C1(C(N2CCN(C(c3ccc(C(N)=O)nn3)=O)CC2)=O)CCc2ncncc2C1 28182,c1(C(=O)NC2CCC(SCCOCOC)C2)ccc(CF)cc1 28183,c1(NC(c2cc(OC(C)C)cc(C(F)(F)F)c2)=O)c(Br)nc2ccccc2c1F 28184,C(=O)(C1=NOC(C2CCC2)C1)NCCCOCC 28185,c1(C(=O)NC2CC3CN(C(c4ccc(C)c(O)c4)=O)CC32)nccn2cnnc12 28186,C1(C(N2CCN(C(c3cnc(CO)s3)=O)C3C2C3)=O)CCc2ccccc2CC1 28187,c12ccc(cc1OC(C)C)n2CCCC.c1(COC)cn(C)nc1C(F)(F)F 28188,N1(C(C2(C(=O)NC(c3ccccc3)C)CCCC2)=O)CCN(C(=O)C(C)(C)C)CC1 28189,N1(C(C=CCCC)=O)C2CCC1C1CC1(NC(C1CCCC(F)(F)CC1)=O)C2 28190,c1(OC)cc(C(C(=O)NC)N(C)CC2CC3(CC(OC)C3)C2)c(F)cc1F 28191,C(CCC(=O)NCC1CN(C(c2occc2Br)=O)C1)NC(=O)C1CC1 28192,Cc1nc(C)c(C(N2CCC(NC(=O)C(=O)NC3CC3)CC2)C)[nH]1 28193,c1(C(N2C(CCNC(CCCCC#C)=O)CSCC2)=O)ccc2c[nH]nc2n1 28194,C1(C(=O)NCC2CC(Nc3nccc(SC)n3)C2)CN2CCN1CC2C 28195,Cc1ncn(CCNCc2cn(C(C)C)nc2-c2ccccc2)c1C 28196,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28197,N1(C(c2c(CC)n(CC)nc2)=O)CCN(C(=O)CN(C(=O)COC)C)C(C)C1 28198,C1(OC)CC2(C1)CC(C(=O)NC1CCN(C(c3cnn(CC4CC4)c3)=O)C1)C2 28199,C1(CC#C)(OC)CCCCC1.c1(C(C(=O)NC23CN(C2)C3)C)ccccc1C 28200,N1(C(C=Cc2scc(C)n2)=O)CCC(N(C(=O)CCC(C)(C)F)C)C(C)C1 28201,N1(C(=O)NC(C)C(=O)NCC2CCCC2)CCN(C2CCCCC2)CC1 28202,C1(C(=O)NC(CCC(=O)NC(CCSC)C)C)CCCCNC1=O 28203,c1(C(=O)NCC(CC)NC(C2(O)CC2(C)C)=O)ccnnc1N.C(C)(C)(C)OC=O 28204,c1(C(N2C3CCC(NC(c4c(C)cnnc4)=O)(C3)C2)=O)cc(N)c(C)cc1Cl 28205,c1(C(N2CC(NC(CN(C)CC)=O)C(F)C2)=O)cc(C)c(C)cc1C 28206,c1(N(C(CC)CNC)C)ccc(S(=O)(=O)N(CCN2CCOCC2)C)cc1Br 28207,c1(NC2C(C)(CC)C2)ncnc(NCc2cc(C(C)C)on2)c1C 28208,C(=O)(CS(=O)(=O)Cc1ccc(-c2ccccc2)s1)NC1C(C(=O)OCC)CC=CC1 28209,c1(C(N2C(C)CC(CNC(C=COC(C)=O)=O)C2)=O)ccc(F)c(CC)c1.CCO 28210,N1(C(C2CCC(C)CC2)=O)CC2CC(C1)N2C(=O)CS(=O)(=O)N(C)C 28211,c1(C(=O)NCC(C)N(C(=O)CC2CCC(F)(F)C2)CC)cc2ccsc2n1C 28212,C1(NC(=O)COC(F)F)CCC2(CCN(C(=O)CCOc3ccc(Cl)cc3)C2)C1 28213,n1(C(C)C(=O)NCc2nc(-c3ccccc3)cs2)cc(CCC2OCCO2)nn1 28214,CC1CC2(CC(C(=O)NCC(O)C(=O)NC3(C(O)CO)CC3)C2)C1 28215,C1(CNC(CCC2(NC(CSC)=O)CCCC2)=O)CCCCC1(C)C 28216,C1(CC(N2CC(NC(CC3(C(=O)OC)CCCC3)=O)C2)=O)CC(O)C12CCC2 28217,C=CCC(F)(F)C(=O)NCC1CCC(C(=O)N(C)Cc2cc(C)cs2)O1 28218,c1(SC)ccc(OS(=O)(=O)CC2CCCC(=O)C2)c(F)c1.C12C=CC(C1)C(=O)N2 28219,N1(CCC(=O)N(C2CC(C(=O)Nc3nccs3)C2)C)CC(O)(C(N)=O)C1 28220,C1(NC(c2ccn(CCCC)n2)=O)CCCCCC1NC(=O)C(O)c1cnc[nH]1 28221,C(=O)(CC(F)(F)C(F)F)NC1CCCC(CNC(Cc2c(C)nc(C)s2)=O)C1 28222,N1(C(CC2CC(=O)NC2=O)=O)CCC(NC(=O)C=CCO)C(CO)CC1 28223,C(=O)(C(CC(C)C)N(C)C(c1ccncc1Cl)=O)NC(CC#C)C(N)=O 28224,c1(OC)cc(C(N2CCC(CNC(=O)C(F)=C3CCC3)C2(C)C)=O)oc(=O)c1 28225,N1(C(C(C)=CC)=O)CCC2(CCC(CNC(=O)CN3CC(C)(C)C3)O2)CC1 28226,C1(NC(C(C(C)(F)F)(C)C)=O)CCC2CN(C(C3(C(F)F)CC3)=O)CC2C1 28227,N1(Cc2cnc(C)s2)CCC(NC(=O)CN2CCCCCC2)C(C)(C)C1 28228,CC1COCCC1NC(C1OCCC1CNC(C1CC12CCCC2)=O)=O 28229,N1(CCC(=O)NC(C)(C)C(F)F)CCN(C(=O)CC2CC2)CC1 28230,c1(C(=O)NCCCN(C(C=CC(C)C)=O)CCO)cscc1OC(F)F 28231,c1(OCC(=O)NCCN(C(=O)C2=CCCCC2)CC)cccc(C)c1C 28232,C1(NC(COC(CC)C)=O)COCCC1C(=O)NC1CC(C)(CC)C1 28233,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CC2CC2)C1 28234,N1(C(C2CCCCC2)=O)CCC2CN(NC(c3ccn(C)n3)=O)CC12 28235,Cc1cc(C(=O)NCC2COCCN2C(c2cc(C3CC3)nn2C)=O)cc(F)c1 28236,N1(C(C2C(C)C2)=O)CC2(C(F)(F)F)CC2(C(F)(F)F)C1 28237,c1(C(CC)OCCNc2nnnn2CCCc2ccccc2)cn(CC)nn1 28238,c1(NC(C2C3(CC(NC(c4ccn(CC)c4C)=O)C3)C2)=O)cccc2occc12 28239,C1(CC(N2CCC(OCC#C)C2)=O)C2CC(C2)N1C(c1cc(C)oc1C)=O 28240,Cc1cc(C(N2CCCC(C(N3CC(C(C)(C)C)C3)=O)CC2)=O)cc(O)c1 28241,c1(NC(C2(C)CN(Cc3cccc(C=O)c3Br)C2)=O)csc2nccnc12 28242,N1(C(C(C=C)(C)C)=O)CCN(C(=O)CN2CCC(C)C2)C(c2ccccc2)C1 28243,c1(CCNC(N(CCC2CCC(=O)C2)CC2CCCC2)=O)nnc2ccccn12 28244,C1(NC(c2cc(C)cc(OC)n2)c2n(CCCOC)nnn2)C(=O)NCCC1C 28245,C#CCC(C(=O)NOCc1ccccc1)NC(c1ccc(CC)nc1)=O 28246,c1(OCC(=O)N(CC(C)(C)NC(=O)C(c2cccnc2)O)C)ccccc1C#N 28247,c1(C2C(C)C2)csc(C(=O)NCCN(C(=O)Cc2ccc(C(=O)OC)s2)C2CC2)n1 28248,C1(NC(C(C)(C)OC(C)=O)=O)CN(C(=O)C(N2CCC(O)CC2)C)CC2(CC2)C1 28249,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28250,C(C1=NOC2CN(C(=O)C#CC3CCCC3)CC12)NC(=O)CC1(CO)CC1 28251,c1(C(N2CC(N(C(C(CN(C)C)N(C)C)=O)C)C2)=O)ccc2ncnn2c1 28252,C1(C)(NC(CNC(CNC(c2cnc(CC)o2)=O)=O)=O)CCCC1(C)C 28253,CCCCC(C)CCC(=O)N1CC(NC(C2(C)COCC2(F)F)=O)C1 28254,N1(C(c2cc(C)cc(F)c2N)=O)CC(C)OC2(CCN(C(C3CC3F)=O)CC2)C1 28255,c1(N(CC(C)CO)C)nc(=NCCc2cccn2C)[nH]c2c1cnn2C 28256,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(c1cc(C)on1)=O 28257,N1(C(c2ccc(SCCC)o2)=O)CCC(NC(C2CCN2C(C)(C)C)=O)C1C 28258,c1(C(=O)NCC2(NC(=O)OCc3ccccc3)CCCC2)cc2n(n1)CCCO2 28259,c1(OC)cc(C(=O)NC2CCC(NC(C3(Cl)CC3)=O)C2)c(C)c(Br)c1 28260,C1(CNC(c2ccc(C)o2)=O)CC2(C1)CN(C(=O)CCc1cc(C)nn1C)C2 28261,C1(NC(C2CNC(=O)N2)=O)CC2(C(=O)NCC3(C4CC4)CCC3)COC1C2 28262,C1(C(N(C(C)C)CCNC(c2ncc(Cl)n2C)=O)=O)CCC2CC2CC1 28263,N1(CC(=O)N(C(C)C)C(C)C)CCC(C)(CNC(c2ccc(F)cn2)=O)CC1 28264,N1(C(C2CC(NC(C3(O)CCSCC3)=O)CCO2)=O)CCC(F)(F)C(O)C1 28265,CCCCC(C)(F)C(=O)N(C)CC1(O)CCN(C(=O)C=Cc2cccc(F)c2)C1 28266,c1(NC(c2n(C)ccc2)=O)ccc(CN2CCSCC2)cc1 28267,C1(CNC(c2ccc(Cn3cc(-c4cccs4)nn3)o2)=O)CCCOCC1 28268,N1(C(CCOCCOC)=O)CCC2(CCN(C(=O)C(C)(C)N(S(C)(=O)=O)CC)C2)C1 28269,C1(Cc2ccccc2)(NC(=O)NCc2ncc(I)s2)CCS(=O)(=O)CC1 28270,n1(C(C)C)cnc2c(NC(c3nc(=N)[nH][nH]3)C)[nH]c(=NCc3cncs3)nc12 28271,c1(N(C)C)cc(CNC(=O)C(c2ccc(-c3cc[nH]n3)cc2)O)cc(F)c1 28272,c1(C(N(CC(C)(C)CNC(c2ccc(C(F)F)o2)=O)CC)=O)cnnc(C)c1 28273,C#CCCCCC(C(=O)NC)N(c1ccc(C(=O)OC)cc1Cl)C 28274,C1(NC(C(C)=CC)=O)CN(C(c2ccc(C(=O)OC)cn2)=O)C2CC12 28275,C(COCC(=O)OCC1CC1)(CCCC)NC(C1N(CC)CC1)=O 28276,C12CCCC3CN(CC13)C2=O.c1(N(C(=O)COc2cccnc2)CC)nccnc1Br 28277,C(=O)(C1=C(Cl)CCC(C)C1)N(CC(CNC(CC(C)C(F)(F)F)=O)(C)C)C 28278,C(=O)(CS(=O)(=O)CC(C)C)NC1C(C=C)CN(C(=O)COC2CCCC(C)C2)C1 28279,Cc1ccccc1-n1cc(C(N2CC(NC(C3CC3C(F)F)=O)C2)=O)nn1 28280,CCN=C(NCN1CC2CCC2(CO)C1)N1CCC(O)CC(C)(C)C1 28281,N1(C(C23C(CN(Cc4cccc(N(C)C)c4)C2)C3)=O)CC2CCCC2C1 28282,c1(-c2cn(CCCC(=O)NCC(C)(C)OCC)nn2)ccc2c(c1)CCO2 28283,C1(C(=O)OCC2(C)CC(F)(F)C2)CCCC1C1CCCC1 28284,c1(C(=O)NCC2CCC(NC(CCCOC(C)C)=O)C2)ccc(C(F)(F)F)cc1 28285,N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28286,C1(NC(c2n(CC)ncc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28287,C1(CC(=O)N(CCCCN(C)C)CC(=O)N(C2CCCC2)CC)CCCCC1C 28288,C1(OC2(CC)CC2)CCC1NC(=O)CN(C(=O)C(C)n1cccc1)C 28289,c1(OC)ncccc1CN1CCC(CC(=O)NCc2cn(C)cn2)CC1 28290,N1(C(C(C)Cn2cncn2)=O)CC2CCC1C(NC(=O)CN1CCS(=O)(=O)CC1)C2 28291,C1(NC(CSS(C)(=O)=O)=O)CS(=O)(=O)C2CN(C(C3CC4(CSC4)C3)=O)CC12 28292,C(=O)(C(CO)C(C)(C)C)NCCCN(C(c1cnn(CCO)c1C)=O)CC 28293,c1(COC)nc(N(C(C)CNC(=O)C=Cc2cccnc2)C)cc(O)n1 28294,C1(OC)CCCCC1C(N1CCOC(C(C)NC(c2ccncc2)=O)C1)=O 28295,CCCC(O)C(CO)NC(=O)C(CCC1CCC1)NC(C1CCCN1C=O)=O 28296,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28297,N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(=O)NC2(C(C)O)CCC2)C(O)C1 28298,c1(CC(N2CCC(O)(CNC(C(c3cccs3)SC)=O)C2)=O)cc(F)cc(F)c1 28299,N1(C(=O)OC)CCCC(CC2n3cnc(n3)C(=O)N2)C1.C(OC)OC.CCOCC 28300,c1(C(N2CCC(NC(c3cnn(C)c(=O)c3)=O)(CF)C2)=O)c(F)cc(Cl)cc1F 28301,N1(C(CCC=C)=O)CCN(C(=O)CNC(=O)C=Cc2ccco2)CC1CC 28302,O=C1NC(CN2CC(CCCCNC(c3ccc(-c4ccccc4)s3)=O)C2)CO1 28303,C1(CCN(C(=O)C(N)=O)CC)CCN(C(=O)CC(C)SC)CC1 28304,CCCC(CC)C(=O)NCC1(F)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 28305,N1(C(CCOC)=O)CCC(C(C)(C)C)(CNC(=O)COc2ccccc2F)C1 28306,N1(CC(=O)NCC2(CN(C)C(C3CCCC34CCC4)=O)CC2)C(=O)NC(C)(C)C1=O 28307,N1(CCC(=O)N(CC(C)CNC(=O)CC2CCOC2(C)C)C)CCC(CO)CC1 28308,Cc1nn(C)c(C)c1C1OCCC1n1cc(NC(=O)C(F)(F)F)nn1 28309,c1(C(C(=O)NCC2CCOC2)N2CCC2CC2CC2)ccc(Br)cc1 28310,C(C(C)(C)CN=C(NCc1ccco1)NC1CC1CN(C)C)NC(CC)=O 28311,C(C)(C(C)C(=O)NCc1noc(C)n1)NC(CSCCOC)=O 28312,C1(CNC(C(C)NC(CC)=O)=O)CC(C)(NC(c2ccc(Br)o2)=O)C1 28313,Cc1ccc(C(=O)NC2CC2NC(C2(N3CCOCC3)CCC2)=O)o1 28314,c1(C(=O)NCC(C)CNC(C2(COC(C)(C)C)CC2)=O)coc(Br)c1 28315,CC(C)CC(C(=O)NC(CC1CCC1)C(=O)NC(CCO)C1CCCC1)C(N)=O 28316,C12(CNC(C(C)c3ccsc3)=O)CC3CC(CC(C3)C1NC(=O)CO)C2 28317,CCCC(C)(CC)C(=O)NC(C)CCNC(=O)C1=CSCS1 28318,c1(SCc2n(CCOC)nc(-c3cnn(C)c3)n2)cc2c(s1)CCCC2 28319,C12(CNC(=O)COc3ccn(C)n3)CCC(CC1)OC2.C12(CC)CCCN1C2=O 28320,C(CC(=O)N1CCN(C(=O)CCc2ccc(O)nn2)C(C)C1)(C(F)(F)F)OC 28321,C1(CNC(C(C)OC(C)(C)C)=O)(CO)CC(NC(=O)CC2CCCOC2)C1 28322,C1(NC(c2n(CC)ccn2)=O)CN(C(C2(C)CCN(CC)CC2)=O)CCC12CCC2 28323,CCCC(C)(CC)C(=O)N1CC(CC(N2C(CO)CC2C)=O)(OC)C1 28324,C(C)(C)(C(C(=O)NC)C(C)C)NC(c1ccc(CC)cc1)C(=O)OC 28325,c1(CN(CCNC(CSCC)=O)C(C2CCCN2C(C)=O)=O)ccc(C#N)cc1 28326,c1(C(N(C(C)CN(C)C(C2CC(COC)C2)=O)C)=O)cccc(CN(C)C)c1 28327,Cc1cncnc1C(N1CCCCC1CNC(=O)CC1CC(=O)NC1=O)=O 28328,N1(C(C2C(C(=O)OC)C2)=O)CCC2(C=C(C(=O)NC3COC(C(F)F)C3)C2)C1 28329,CCCC(CNC(C1CCCC1O)=O)C(=O)NCCC1CC1C 28330,N1(c2csnn2)CCC(C(C2CC2)NC=O)CC1.[nH]1cc(C2C3COCC23)nn1 28331,CC1CC(CCNC(=O)CCOC2CCCC2)CCN1C(=O)CC(Cl)Cl 28332,Cc1cc(C(=O)NCC2(C(N3CC(N4CC(F)C4)C3)=O)CC=CC2)ncc1F 28333,CC(C)CC(F)(F)C(=O)NCCCCNC(=O)CC1CCCCC1(F)F 28334,C1(c2nnnn2CC2CCOCC2)(NC(c2cc(C)sc2C)C)CCCCC1F 28335,C1(C(C)C)OCCC1C(N1CCC(CCNC(c2conc2C(C)(C)C)=O)C1)=O 28336,CC1CCC(CC(=O)NC(=O)C(=O)N(C)C)C1.C1(=O)CCN1CCCO 28337,c1(N(C)C)ccnc2c(N(C3CC4CC3CN4)C(C3CCC(=O)N3C)=O)cccc12 28338,C(=O)(C(C)(O)C(F)(F)F)N(C1CCCN(C(=O)C(=O)N(C)C)CC1)CC 28339,N1(C(c2c(COC)scc2)=O)CCN(C(C2CCCO2)=O)CC1C1CC1 28340,CC(C)C(C(C)NC(=O)C(=O)N1CCCC1)NCc1cc(Cl)ccn1 28341,Cc1ccc(N)c(C(=O)NCC2CCCN2C(=O)C(C2CC2)N(C)C)c1 28342,C(CNC(=O)Cn1cc(C)cn1)(CC(=O)NCCn1nncc1C)OC 28343,c1(C(=O)NCC(CCNC(C2(C)CC3CC3C2)=O)O)ccc2oncc2c1 28344,c1(OC)cc(C(=O)OCCCN2CCC(C(C)(F)F)CC2)ccn1 28345,N1(C(CNC(=O)CNC(C2CC3CCCC3C2)=O)=O)CCC12CC(O)C2 28346,N1(C(=O)NC)CCCC(C(N2CCC(OC(C(O)CO)C3CC3)C2)=O)CC1 28347,c1(C(=O)NC(CCOC)CNC(=O)Cn2cccc2)ccn(C(C)C)c1C 28348,Cc1cccc(C(O)C(=O)NCCC2(NC(=O)CCc3ccsc3)CC2)c1 28349,C1(NC(C(C2CCC2)OC)=O)CN(C(C2CN3CCN2CC3)=O)CC1(C)C 28350,C(=O)(C(C)(C)C(C)O)N(CC(C)NC(C1(c2ccnn2CC(F)(F)F)CC1)=O)C 28351,CCC(N=c1[nH]c(N2CCC(F)(F)C2)nc2ccc(N(C)C)cc12)c1ncnn1C 28352,CCC(C)CC(=O)C(=O)N1CCC2(CC(C(N3CCOC(C)C3C)=O)C2)C1 28353,c1(C(=O)NC(CN(C2CCCN(C(C(C)C)=O)C2)C)=O)ccc([N+](=O)[O-])cc1 28354,C1(CCC)(C(=O)OC)CCCN(C(=O)C(c2ccccc2OCC)OC)C1 28355,Cc1n[nH]c(C)c1C(C)CC(=O)N(CCCCCNC(=O)C(C)OCCN(C)C)C 28356,n1(CC)nnc2cc(C(N3CC(CNC(C4CCCCCCC4)=O)C3)=O)ccc12 28357,C1(CCC)CN(C(c2c[nH]c(=NC)o2)=O)CCN1C(c1cccnc1S)=O 28358,C(=O)(C1=CCCOC1)N1C(CN(C(C(C)NC(C2CCCC2)=O)=O)CC)CCCC1 28359,C=CCCC(F)(F)C(=O)NC(C1CN(C(c2cnn(CC(C)C)c2)=O)CCO1)C 28360,c1(C(=O)NC2CC(NC(c3ccc(N)c(F)n3)=O)C2)cc2cc(O)ccc2[nH]1 28361,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28362,N1(CC#C)CC(NC(c2ncoc2COC)=O)C2(CCOCC2)C1 28363,C1(C(N2CCC(c3cccc(F)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28364,c1(SC)ccc(CC(=O)NC2CCCC(NC(=O)Cc3ccc(Cl)cn3)C2)cc1 28365,C1(O)(CN(C)C(C2CCC3(CCC3)C2)=O)CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 28366,c1(C(N(C(CN(C(C(CC=C)CC)=O)C)C)C)=O)cccn2nccc12 28367,C1(C(=O)NC2(CC(=O)NCC(CO)N(C)C)CCC2)CC(F)(F)C1 28368,C(CC(=O)NC1CC2CCCC(C1)C2)(C(F)(F)F)NC(C(C)NC(=O)C1CC1)=O 28369,c1(N2CC(N(C)C)C3(C2)CC3)nc(=NCCC2(C)CC2(Cl)Cl)[nH]c2ccsc12 28370,c1(CN2CC(NC(c3c(COC)cccc3)=O)C(O)CC2)cc(O)c(Br)cc1O 28371,c1(NC(C2(CNCc3c(C)cccc3)CC2)=O)cccc2nscc12 28372,C(=O)(CC(F)(F)F)NC1(CNC(CN(CC)CC)=O)CCOC1 28373,c1(C(N2CCCC(CNc3nccc(C)n3)C2)=O)cncc(N)c1C 28374,c1(OC)cc(C(=O)NC2CCC2NC(C2CCCCC23CC3)=O)c2occc2c1 28375,C(=O)(CC(O)c1ccccc1)NCCC(C)N(C)C(C1(C)CCCC1)=O 28376,CCC(C)(C)CCCC(=O)NC1(CCNC(c2ccc(CF)cc2)=O)CCCC1 28377,c1(C(N2C3C(NC(CSCC#C)=O)CC(C3)C2)=O)cccc2nccnc12 28378,c1(C(=O)NCc2ccsc2C(N2CCC2)=O)n[nH]cc1[N+](=O)[O-] 28379,C(=O)(C(F)(F)F)NC(C)C(=O)NC1CN(C(C2CSC2)=O)C1 28380,CCC(C(=O)NCC1CN(C(c2ccc(C(C)C)cc2)=O)CC1(F)F)C(C)C 28381,c1(NC(C)=O)c(C(N2CCC(NC(=O)Cn3cccc3)C2C)=O)cccc1C 28382,C#CC1CN(C(=O)C(CC)OC)CCN1C(=O)CCc1ccccc1C 28383,CN1CCC(COC(C2CCCC(=O)C2)=O)c2ccccc21 28384,c1(C(=O)NC2C3CN(C(C4(SC)CC4)=O)CC32)ccc(F)c(C(C)C)c1 28385,C1(c2ccccc2)(NC(C2(NCC3C(OCC)C3)COC2)=O)CCN(C)CC1 28386,N1(C(c2cnc(C)[nH]2)=O)CCOCC(NC(=O)COc2ccccc2C(N)=O)C1 28387,C1(CNC(CC2CC(C(=O)OC)C2)=O)CCCCN1C(=O)COCP(C)(C)=O 28388,N1(C(CCC=C(C)C)=O)CCOC2(C1)CN(C(=O)C(C)SCc1ccccc1)C2 28389,CC1CCC(C)(C(N2CC3(CC(NC(C4CN(C5CCOC5)C4)=O)C3)C2)=O)CC1 28390,Cc1ccnc(O)c1NC(C1CC(F)CN1C(c1cccc(Cl)c1)=O)=O 28391,S(=O)(=O)(c1ccc(C)c(C)c1)NCC12CCC(NC(C(CCCC)O)=O)(CC1)C2 28392,C1(NC(=O)Cn2cccn2)C2CC3C1C3C2NC(C1(c2ccc(Cl)o2)CC1)=O 28393,CC1CN(C(c2sccc2CNC(=O)CCc2cccn2C)=O)CC1O 28394,Cc1ccc(O)c(CC(N2CCN(C(c3nc(O)sc3C)=O)C(C)C2)=O)c1 28395,CC1CCCCCN1C(=O)CCOCCN(C)C(c1cncn(C)c1=O)=O 28396,N1(C(c2ccc(C(C)C)cn2)=O)CCCC(C)(NC(=O)CC2(O)CCCOC2)C1 28397,c1(CCC2(C(=O)NCC(C)NC(=O)Cc3cncnc3)CC2)ncc(Cl)cc1F 28398,C1(NC(C(N2CC(c3onc(C)n3)N(C)CC2)=O)=O)CCc2nnc(O)n2C1 28399,C1(NC(c2c(OC)cc(OC)cc2O)=O)CC2CN(C(=O)CCF)CCN2C1=O 28400,N1(C(Cn2nc(C)c(Cl)c2)=O)CC2COCCC2(NC(c2cccnc2)=O)C1 28401,c1(C(N2CC=CC(C(=O)NC34CCCC3C4)C2)=O)cccnc1SCCO 28402,c1(CC(=O)NC(CC2CN(C(c3cc(C)oc3)=O)C2)C)cnc(Cl)cc1C 28403,C1(O)(CN(c2ccc(C(C(n3ccc(C(F)(F)F)n3)C)=O)cc2)C)CCCCCC1 28404,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CCC(C(C)C)C2)=O)CCC1 28405,c1(C(N2CC(NC(C3(N=[N+]=[N-])CC3)=O)CC(C)(C)C2)=O)cc(F)cc2nn[nH]c12 28406,C1(NC(C2CC2C2CC2)=O)C2CC1CN(C(c1cnc(C3CCOC3)s1)=O)C2 28407,C(=O)(C(C)(C)CS(N)(=O)=O)N(CCNC(CNC(=O)OC)=O)Cc1ccccc1 28408,C1(O)(C(C)NC(c2cscn2)=O)CN(C(c2ncoc2Br)=O)C1 28409,c1(C(=O)NCCN(CCOC)C(C2CCOC2C)=O)cc(C)ncc1C 28410,CC1(C(=O)NC2CC(CO)N(C(c3cc[nH]n3)=O)C2)CCc2ccccc21 28411,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(C(N2CC(C(C)C)C2)=O)C(CO)CC1 28412,c1(C(=O)NCCN(C)C(c2cnc(-c3ccccn3)nc2)=O)cc2n(n1)CCC2 28413,CC(Cc1cccn1C)N=c1ccnc(NC2CCC(=O)NC2)[nH]1 28414,N1(C(=O)NCCN2CC(C)N(C(=O)OC(C)(C)C)CC2)CCC(O)C2(CC2)C1 28415,CC(=NO)C1CC(C(N2CC(NC(=O)COC3CCCC3)C(C)(C)C2)=O)C1(C)C 28416,Cc1cccnc1C(=O)NC1(CCO)CN(C(c2cncc(C(C)(F)F)c2)=O)C1 28417,C1(C(=O)NC(c2cn(CC(=O)NC(C3CCCC3)C)nn2)C)(SC)CCOCC1 28418,Cn1nc(C(=O)NC2CC2NC(C2CC3(CC3)CO2)=O)cc1C(N)=O 28419,c1(-c2ccc(C(C)NN3CCN(CCCO)CC3)cc2)ccc(Cl)c(C(=O)O)c1 28420,c1(CC(CC(C)(C)NC(=O)CC2CC2C)C)ccccn1.n1(CC(=O)N)cncn1 28421,C1(NC(=O)C(O)P(C)(C)=O)CCn2nccc2C1.C12CCN(CC1)C(=O)N2CC 28422,c1(C(=O)NCC(C)(CNC(=O)CC2CCCOC2)OC)ccncc1NC(C)C 28423,c1(C(=O)NC(C2C3N(C(C(F)=CCC)=O)C(CC3)C2)(C)C)ccc(F)c(CO)c1 28424,C1(CC(=O)NC(C(C)C)CO)CN(CCOCc2ccccc2)CC12CC2 28425,c1(C(=O)NCC2N(C(CC(C)C)=O)CC(C)CC2)cccc2cc[nH]c12 28426,C(CC(C)C)(C(=O)N1CC(CC(C)NC(C2CCCS2(=O)=O)=O)C1)NC(=O)OC 28427,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28428,C1(NC(C2(OCC)CCCCC2)=O)CCN(C(=O)C2=CC(C)C2)CC1O 28429,N1(C(CCOC(C)=O)=O)CC(F)(F)CC1C(=O)NC(C)Cn1cncn1 28430,c1(C(=O)NCCN(C)C(C2CCC(C)(C)CC2)=O)occ2c1CCC2 28431,N1(C(C2C(CCC)C2)=O)CC(NC(=O)C=C2CCCCC2(C)C)C2CCCC12 28432,c1(C(=O)NC2(CC(=O)NCC3C(C)(C)COCC3)CCC2)ccc2cc[nH]c2n1 28433,O=C1CC(NC(c2c(CN3CCCCC3CCCO)ccs2)=O)C(=O)N1 28434,C(CNC(=O)C(C)Oc1ccccc1F)(CC(F)(F)F)NC(c1c(C)nsc1)=O 28435,CC1(NC(c2csc(Cl)n2)=O)CCN(C(C2CCCC2)=O)C1.C12CSCN1C2=O 28436,c1(NC)snc(C)c1C(=O)NCN1CCC(CNC(C2CCNC2=O)=O)C1 28437,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28438,C1(C(C)NC(c2ccc(CNC(C)=O)cc2)=O)CN(C(=O)CC(=O)N(C)C)CCO1 28439,c1(NC(C(C(=O)OC)OC)=O)ccc(NC(=O)CCCSC(C)(C)C)c(C)c1 28440,C1(N(C)C)CCC(C(=O)NCC2CC(n3cc(CCOC(=N)O)nn3)C2)CC1 28441,n1(C(C)C)ncc2cc(-c3ccc(NC(=O)CN4CCOCC4)cn3)cnc12 28442,CCC(CCC(=O)N(C)CC1CCCN(C(C2CC(N(C)C)C2)=O)C1)OC 28443,C#CCCCCC(=O)N1CCC(OCCCNC(C2CCCS(=O)(=O)C2)=O)CC1 28444,N1(C(C2(OCC)CCCC2)=O)CCCCC1CNC(=O)C(c1cccc(F)c1)O 28445,Cc1cn2cc(C(N3CCN(C4CN(C(=O)C=CS(C)(=O)=O)C4)CC3)=O)sc2n1 28446,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1C1CC1)=O 28447,c1(C(CNCC(=O)NCC(C)(C)c2cncs2)OC)cccc(C(F)(F)F)c1 28448,C1(CC(=O)OCC)CN(C(CC2CCCC2)C(=O)NCC(C)C)CC(C)O1 28449,CC1(C)CC1(C#N)NC(N(c1cccc(SCCCl)c1)C1CC1)=O 28450,Cc1cnc2cc(C(N3C4CCC3C(CNC(=O)COCC(C)C)C4)=O)ccn12 28451,c1(C(=O)NCc2ccc(OC)cc2)c[nH]c2cc(-c3nn[nH]n3)cnc12 28452,C(=O)(CC(C(F)F)C(C)(C)C)N(CCN(C(c1cccc(CO)c1)=O)CC)CC 28453,c1(C(C)NC(CCNC(C=C(COCC)C)=O)=O)c[nH]ccc1=O 28454,C1(NC(=O)C=CC2CC2)CCCN(C(c2cc(O)cc(=O)o2)=O)CC1 28455,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28456,C(C)(C(=O)NCC1CCC1)N(C(=O)C=CCO)CCC 28457,c1(C(N(C2CCCN(C(C(C)C3CCC3)=O)C2)C)=O)ccc(N)c(Cl)c1O 28458,c1(C(C)=O)cc(C(N2CC(Cc3cn(CC(O)C(F)(F)F)nn3)C2)=O)ccc1Cl 28459,C(=O)(CC(C)(C)C1CCCCC1)N(CCNC(C1CCC(C(N)=O)N1C)=O)CC 28460,N1(C(C=COCC)=O)CCCC2(CCC(NC(c3cc(C)c(C)nc3O)=O)C2)C1 28461,n1(CC)nccc1C(C(=O)NC1CCCC1)N(C1CCOCC1)C 28462,c1(C(=O)NC2CC3(C(NC(=O)CC4CC45CC5)C3)C2)cccc2c1C(=O)NC2 28463,Cc1cc2[nH]c(C(=O)NC34CCC(CC3NC(c3cc[nH]c3)=O)C4)cc2o1 28464,C1(NC(c2c(C(C)(C)C)ccs2)=O)CC2CC(NC(c3cnc[nH]3)=O)CC2C1 28465,c1(NC(C2CCCCC2NCc2cc(Cl)ncn2)=O)nc(Cl)ccc1I 28466,CON(C)C1CN(C(C23CC(CN2C(c2ccc(F)s2)=O)C3)=O)C1 28467,N1(C(CSCC(C)C)=O)CCc2cc(CNC(C3(C)CCC34CCC4)=O)ccc21 28468,N1(C(c2c(C)ccc(C)c2)=O)CC2CCC(C1)C2NC(=O)C(C)(C)c1cccs1 28469,c1(C(N2CC(C)N(C(C3COC(=O)C3)=O)CC2)=O)nnn2c1CCCC2 28470,CC1CC(NC(=O)Cn2nnc(=O)[nH]2)CCN1C(=O)Cc1cccc(C#C)c1 28471,C1(C(N2CCCN(C(=O)C(c3sc(C)nc3C)=O)CC2)=O)(OC)CCC(C)CC1 28472,C(C1CCOc2ccccc21)NC(=O)NNC(C1CCC(F)(F)CC1)=O 28473,Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)CCSc1nccn1C)C)O2 28474,N1(C(C2C(CNC(CC(CC(C)C)C)=O)CCC2)=O)CC2C(=O)NC(=O)C2C1 28475,Cc1sc(C(F)(F)F)nc1C(N1CCC(N(C(=O)COC2CC2)C)C1)=O 28476,N1(C(CSCC)=O)CCOC(CCNC(=O)CCC(C)SC)C1 28477,C(=O)(CCCCC(N)=O)N1CC(CC)C(NC(=O)CCOCCCOC)CC1 28478,C=C(C)C(CC(=O)N1CCC(CN(C)C(c2cnc(C)cc2Cl)=O)CC1)OCC 28479,C(CC(C(=O)NC1CCCN(C(c2cccc(C(N)=O)c2)=O)C1)OC)OC 28480,N1(C(c2nccc(CC)c2)=O)CCC2(CO)CN(C(=O)CO)CC2C1 28481,CCC(CC(=O)NC(C)(C)C(C)CC(=O)N1CC(CO)(CF)C1)C(F)F 28482,c1(C(=O)NCC(CCCC)NC(C2(C)CCCO2)=O)coc2c1C(=O)NCC2 28483,N1(C(CCC=CC)=O)CCN(C(=O)C(C)(C)CCF)CC1c1ccncc1 28484,C1(NC(COCCCOC)=O)CCN(C(C2CC2C2CC2)=O)CC1F 28485,C(C)(CC1CCC1)(C(=O)N(C1CCCCC1)CCNC(C1(Cl)CCCCC1)=O)OC 28486,Cc1c(C(N2CCC(NC(N3CCC(F)(F)C3)=O)CC2)=O)cccc1Cl 28487,c1(C(=O)OC)ccc(CNCC2CCCC2N)cc1Cl 28488,c1(C(=O)NC(C)(Cc2ccccc2Br)C(N)=O)ccc([N+](=O)[O-])cn1 28489,C1(CNC(=O)CCCC2CCC2)CN(C(C23CCCC2C3(F)F)=O)CC12CCC2 28490,N1(C(=O)NC2CC(c3ccc(Br)cc3)C2)CCC12CC1CCC2C1 28491,C1(C)(C(=O)NCCCN2CCN(C(C(C)C)=O)CC2)CC2CCC(C1)S2 28492,c1(CC)ccc2occ(C(N3CCC(C)C(NC(=O)CCNC(N)=O)C3)=O)c2c1 28493,C(=O)(CCCCN=[N+]=[N-])N1CCC(CCC(N2CCCC2CC(C)(C)C#N)=O)C1 28494,c1(C(=O)NCCC(C)NCCOc2ccccc2)ccc(C2CCOCC2)nc1 28495,C1(NC(C(C)C)=O)CS(=O)(=O)C12CCN(C(c1cnn3ccnc(N)c13)=O)CC2 28496,c1(C(=O)NC2CC(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)c(C)cc(C)nc1O 28497,c1(-c2cnc(NCc3ccc(COCC)o3)c(C)c2)ccc2c(SC)cnn2c1 28498,c1(CC(=O)NC(C(=O)NCCN(C)C)C2CCC2)cccnc1 28499,C(=O)(CC(F)(F)C(F)(F)F)NC(C1N(C(CCN(CC)CC)=O)CCCC1)C 28500,C1(NC(C(CCC)O)=O)CCN(C(c2cc(NC(C)=O)ccc2C)=O)C12CC2 28501,c1(NC(C(=O)NCC(CC)NC(=O)CSC2CCS(=O)(=O)C2)=O)ccc(O)cc1 28502,CCCCC(CC)C(=O)NCC1(NC(C2CCCO2)=O)CCCCC1 28503,C1(C)(C(=O)OCc2c(C)nns2)CCCN(C(=O)OC(C)(C)C)C1 28504,N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CN(C(=O)Cn1nc(C)nc1C)C 28505,c1(C(CCC)O)cn(CC(C)OCCN(CC)Cc2cc(C)ns2)nn1 28506,Cc1c(C(N2CCOCC2CN(C)C(C2(C)CC2(F)F)=O)=O)cccc1Cl 28507,CC1CN(C(c2ccn(C)c(=O)c2)=O)C(C)CN1C(=O)CC1CCN(C2CC2)CC1 28508,C1(CN(c2ncccc2C(C)=O)CC)CCCN(C(=O)Cc2sc(S)nc2C)C1 28509,C1(CC)(NC(=O)C(F)F)CCN(C(=O)C(C)(C)C)CC1 28510,c1(C(C(=O)O)NC(=O)CSc2cccnc2)cccc(Cl)c1Cl 28511,CCC(CC)CC(F)C(=O)N1CSCC1C1CCN(C(=O)CC2CCOCC2)C1 28512,c1(C(=O)NCC(C)CNC(c2ccoc2)=O)cccc2c1CCO2 28513,c1(C(=O)NCC(C)(CC)NC(C2CC(=C)C2)=O)sc2cncc(C(C)C)c2c1C 28514,c1(C(=O)NC2CCN(C(C=C(CC)C)=O)C23CC3)cccc2[nH]ncc12 28515,c1(C(N2CCC(C(C)C(=O)Nc3cnc(Br)nc3)CC2)=O)cc(Cl)ccc1F 28516,CC1(C)C2CCC1(C(=O)NC1CCCCC1CNC(C1(CN(C)C)CCCC1)=O)C2 28517,C(=O)(CC(F)(F)C(F)F)NCc1c(C(N2C(C)CC(O)C2)=O)scc1 28518,n1(CC(=O)N(CC(C)NC(C2CCCCC2O)=O)CC)nc(C)c([N+](=O)[O-])c1C 28519,C1(Nc2cccnc2Cl)CN(C(=O)C2CC2)CC2(CC2)C1.CC1CC(=O)N1 28520,N1(C(c2c(C)nn[nH]2)=O)CCC(C)(O)C1C(=O)N(C)Cc1ccsc1 28521,c1(C(=O)NC2C(NC(C(C)Oc3ccc(Cl)cc3)=O)CC2)cccc(C(F)F)n1 28522,CCCCC(F)C(=O)NC1CCC(C(=O)NCc2ncccc2C)CC1 28523,N1(C(c2cccc(C)c2F)=O)CCCC(C2CCN(C(C3(C)COC3)=O)CC2)C1 28524,C1(NC(C(C)OCCCC)=O)CC(NC(C2(c3cccc(Cl)c3)CC2)=O)CC1O 28525,C1(C(=O)OC)CC(F)(F)CN1C(c1cc(C)c(C)s1)C(=O)NC(C)C 28526,C1(CNC(C(CC)(C)C)=O)C2CCCC1N(C(c1ccon1)=O)C2 28527,C1(NC(CC(CC=C)(C)C)=O)CC2(CCC(CNC(C3C4COCC34)=O)CC2)C1 28528,n1(CC)cc(C#N)cc1CN(C=O)CC(C1CCCCCC1)OC 28529,CCCC(C)(C)CC(=O)NCc1cn(CC(=O)NC2CC(O)C2O)nn1 28530,N1(C(C(C)OCC2CC2)=O)CC(CNC(C2(C)CCN(C)C2=O)=O)CC(C)C1 28531,C(=O)(C(O)CC(C)(C)C)NC(CC#CC)C(=O)NCc1nnc(O)n1C 28532,c1(CC(=O)NC(C)CNC(=O)CC(C)N2CCCC2=O)cc2cc(Cl)ccc2s1 28533,c1(N(CCNC(C(C=CC)O)=O)CCOC)nccc2c(CC)c(O)nnc12 28534,N1(C(CC(n2ccc(C)n2)C)=O)CCCCC(NC(c2n[nH]c(C)c2F)=O)C1 28535,C12(NC(COCCCC)=O)CC3CC(C1)CC(NC(C1OCCCO1)=O)(C3)C2 28536,c1(C(C(=O)NC(CNC(Cc2cc(C(C)C)no2)=O)C)O)ccccc1F 28537,CC1(CC(N2CC(CO)(NC(c3coc(O)n3)=O)C2)=O)CCS(=O)(=O)N1 28538,CCCC(C(=O)OCC)NC(C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C)=O 28539,CC(C)(C(=O)N1CCC(NC(=O)Cn2nnc(=O)[nH]2)C1)C1CCCCO1 28540,C12(CNC(C3CC(=C)C3)=O)CCC(CNC(=O)C(C)OCCC(C)C)(C1)OC2 28541,c1(C(N2CC(C)C(CNC(C3COC3)=O)C2)=O)ccc2c(Br)cncc2c1 28542,c1(C(=O)NCC2N(C(CSCCOC)=O)CCCC2)cccn2nncc12 28543,N1(C(Cc2c(CC)con2)=O)CCCC(C(=O)NC2C=CCC2)CC1 28544,c1(C(=O)NC2CN(C(c3cc(Cl)cnc3Cl)=O)C2)ccc2nonc2c1 28545,C1(NC(=O)Cc2nc(C3CC3)cs2)CN(C(c2cc(Cl)ns2)=O)CC12CCC2 28546,C(=O)(CCCC=C)N(CC(=O)NCC(C1CCC1)NC(C)=O)CC#C 28547,c1(C(N2CC(OCCC)C(n3ccnn3)C2)=O)cc(C)cc(Br)c1 28548,Cc1ccc(C(=O)NC(C(C)NC(=O)C(C)C)C(C)C)c(=O)n1C 28549,c1(C(CNC(c2scc(C(C)=O)c2)=O)NC(C2CC2C)=O)ccccc1F 28550,c1(C(=O)NC2CC(NC(C(c3scc(C)n3)C)=O)C2)cc2nccnc2cc1C 28551,c1(OC)ccccc1CCC(=O)NC(C)CC(C)NC(c1nocc1C)=O 28552,C(=O)(CCCCCS(N)(=O)=O)N(C)CC1(O)CN(C(=O)C(C)(C)NC(=O)CO)C1 28553,c1(NC(=O)NC(c2ccc(Cl)cc2)CCSC)nnc2n1CCC2 28554,c1(SC)cc(F)c(F)c(Cl)c1F.c12ccc(cc1)OC(=O)CNC2C(=O)OC 28555,c1(OC)ccc(CNC(=O)COc2ccccc2)c(OC2CC(O)C2)c1 28556,C1(COC(C)=O)CC2CCCCCC12.n1(CCCCN2CCC2=O)ccc(C)n1 28557,C1(COC)COCCN1C(C1C2CN(C(C3CC=CCC3C)=O)CC12)=O 28558,N1(C(C(F)=CC)=O)CC(NC(C2(c3ccccc3)CCCC2)=O)C(SC)C1 28559,c1(OC)ccc(C(C)CNC(C2CCC2(C)C)=O)cc1 28560,c1(CNC(=O)Nc2cnn(CCCC)c2C)cc2cccnc2cc1F 28561,c1(C(=O)CN(CC(C)NC(=O)COc2ccco2)CC)c(F)cc(OC)cc1F 28562,c1(C(=O)NC(c2nccs2)CC)cccnc1C(=O)NCC1CC(O)C1 28563,CC1CCC(C(=O)NCCN(C)C(c2cncc(-c3cnn(C)c3)c2)=O)CC1 28564,C1(C(F)F)(NC(C(C)O)=O)CC(NC(C2COCCN2)=O)C1 28565,Cc1csc(=O)n1CC(N1CCCC1CNC(c1ccc(C2CCC2)nc1)=O)=O 28566,C1(COC)CN(C(=O)NCCCCc2cnoc2C)CCN1c1ccccc1 28567,N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)Cc2ccc(F)cc2)C(C2CC2)C1 28568,CC(C(C)C(=O)NCCC1CCC(=O)N1)NC(C1(C2CC2)CCCO1)=O 28569,N1(C(=O)CSc2cccc(F)c2)CCC2C3CCC(C3)C12 28570,Cc1cc(O)c(C(=O)NC(C2(O)CCN(C(=O)CN3CCC(C)C3)CC2)C)nn1 28571,CCC(CC(=O)NCC1CCN(C(c2cc(F)c(C)cc2F)=O)C1(C)C)C(C)C 28572,C1(CC(=O)N(C2CCCN(C(=O)CCc3conc3C)C2)CC)CCCOCC1 28573,C(c1cnc(O)nc1O)=CC(N1CC(CNC(CN2CCC(C)CC2)=O)(CO)C1)=O 28574,N1(C(C2OCC(C)C2)=O)CCC(C)C(NC(c2ccn(C(C)(C)C)n2)=O)C1C 28575,c1(CN2CCC(C(=O)NC(Cc3c(C)ncs3)C)C2)csc2ccccc12 28576,N1(C(C(CC)CC)=O)CCN(C(=O)CC2CC3(CCOCC3)CO2)CC2(CC2)C1 28577,C(CCO)(C(=O)N1CCCCC1CCCNC(c1conc1C1CC1)=O)N(C)C 28578,c1(NC(C)(C)CNC(=O)COCc2ccccc2Cl)nccc2nn[nH]c12 28579,CCCC(F)C(=O)N(C(CC)CC(=O)NCC1COCC1OC)C 28580,Cc1nnc(O)c(C(=O)NCC(C)(CC(C)C)NC(=O)CC(O)C(C)C)c1C 28581,N1(C(C=CC=CCC)=O)CCC(CO)(CNC(C2CC(C)(C)CO2)=O)CC1 28582,C=CCCCC(=O)NCCOCCNC(c1cnc(SC)n1C)=O 28583,c1(C(N2CC3C(=O)NC(=O)C3C2)C(=O)NCCCCCC)cnc2n1CCCCC2 28584,C(=O)(C1=NN(C)C(=O)CC1)N(C)CCN(C(=O)C(F)CC1CCCOC1)C 28585,c1(C(=O)NCC2(NC(=O)COCC3CC3)CCOC2)ccn2nccc2n1 28586,C(=O)(C(O)C(C)(C)C)NCc1cc(C(N2CCC(C(C)O)CC2)=O)on1 28587,C#CCS(=O)(=O)CCNC(=NCC1CC1)NCC(=O)NC1(C#N)CCCCC1 28588,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28589,C1(CNC(C2(C)CC2(F)F)=O)CN(C(c2cn(CCO)nn2)=O)CC1O 28590,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28591,c1(C(N(C2CCSC2)CC#C)=O)nn(C)cc1I 28592,C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1CN(C(CC(=C=C)C)=O)C(C)(C)C1 28593,CCC(CNC(=O)C(CNC(=O)C(F)C1CCCC1)N(C)C)CC(C)C 28594,N1(C(CCN(C)C(C)=O)=O)CCS(=O)(=O)C(CC(=O)NCc2cn(CC)nn2)C1 28595,c1(C(N2CCC(C(N3C(C)(CC)C=CC3)=O)(CO)C2)=O)ccc2[nH]nc(Cl)c2c1 28596,N1(C(C2CCCCN(CC)C2)=O)CC2CC(O)C1C2NC(=O)COCCOC 28597,N1(C(C2N(C)CCC2)=O)CCCC2(CCN(C(c3cnn(C)n3)=O)C2)C1 28598,C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)Nc2ccc(CO)nc2)C1 28599,c1(CCC)occc1C(=O)NCC1(CNC(c2ccn(C)c2)=O)CCCC1 28600,N1(C(C(c2ccccc2F)OC)=O)CCCC(CO)(NC(C2C3COCC23)=O)C1 28601,C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(C(=O)NC2CCC(C(C)O)CC2)CC2CC21 28602,C1(COC)(CNC(=O)C(C)CSC)CCN(C(c2nc(C(C)C)ncc2Cl)=O)CC1 28603,c1(OCC)ccc(OCC(=O)N(CC(C)NC(=O)C(F)=C(C)C)CC)cc1 28604,C(=O)(C(CCF)NC(c1cc(C(N)=O)[nH]n1)=O)NCc1[nH]nc(C(C)C)n1 28605,N1(C(C2C(CNC(CC(C)(C)O)=O)CCC2)=O)CCc2ccc(F)cc21 28606,C(C(C(=O)NCC1CN(C(=O)OC(C)(C)C)C1)OC)(c1ccccc1)OC 28607,C(=O)(CC(C)C(C)(C)C)NC1CC=C(C(=O)NCCN2CCN(CC)CC2)C1 28608,Cc1nc2ncc(C(N3CC4C(CNC(C5CCC(CF)C5)=O)C4C3)=O)cc2o1 28609,C12CC(O)C1NC(=O)CONC2=O.C(=O)(CC1(COC)CC1)OCC 28610,c1(C(N2CCCCC(NC(=O)C=CC3CCOC3)C2)=O)csc2ccccc12 28611,N1(C(c2c(C(=O)OC)coc2)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C2CC12 28612,CC(C)CS(=O)(=O)CC(=O)N1CC=CC1CNC(=O)CCNS(C)(=O)=O 28613,C(=O)(CCC(C1CC1)NC(C1(C(C)(F)F)CCOCC1)=O)OCC 28614,CC1(C)CC(C(=O)NC2CC(NC(c3ccc(O)nc3Cl)=O)C(O)C2)CCO1 28615,N1(C(c2cnn(-c3ccccc3)c2)C(=O)NC(CC)C)Cc2nccc(Cl)c2C1 28616,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28617,N1(C(C(CC#C)O)=O)CCN(CC(c2cccc(C)c2)N(C)CCOC)CC1=O 28618,n1(CCCOC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28619,c1(OC)ccc(C)c(NC(=O)CC2COCCN2C(=O)Cn2ccnc2C)c1 28620,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)C=CSc3nc[nH]n3)CC(F)(C1)C2 28621,CC(=O)CCN=C(NCc1cc(C)ccc1O)NCC(O)COc1ccccc1Cl 28622,C1(C(N2CCC(N(C(C(C3CCC3)OC)=O)CCO)CC2)=O)CC12CC(C)(C)C2 28623,CN1CCCC1CCNC(=O)NC(CC1CCCO1)C(=O)O 28624,N1(C(C2C(NC(C=CC(=O)N(C)C)=O)CCC2)=O)CC(C)C1(C)C 28625,c1(NC(C(CC2CCCC2)NC(c2c(C)n[nH]c2)=O)=O)ccc(CO)cc1 28626,N1(c2ncnc(NC3C(OC)CC3)c2C)CCCC(C)(O)CC1 28627,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28628,C1(C(N2CC(N(C(c3nnc(C(C)C)s3)=O)C)C2)=O)C(C)OC(C)C1C 28629,c1(CC)nc(C)c(C(=O)NC(C)(C)CNC(c2cn(CCCF)nn2)=O)s1 28630,CCCC(C(=O)N1CC(O)(C(F)C(N2CCC23CC(C(N)=O)C3)=O)C1)C(C)C 28631,c1(C(=O)NC(CN(C(c2cc(C)[nH]c2)=O)C)C)cc(C#N)ccc1C 28632,c1(CNCC(C)OC)cc(C)c(-c2ccccc2)s1 28633,c1(C(=O)OC)ccc(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)F)cn1 28634,C1(NC(CSCC#C)=O)C(CNC(c2cc3ccncc3s2)=O)CCC12CCC2 28635,c1(C(N2CCC(C)(CCNC(CN(CCC)C)=O)C2)=O)ccc(Cl)c(F)c1O 28636,N1(C(C=CC(C)(C)C)=O)CC(NC(c2cc(C3CC3)no2)=O)CC(O)C1 28637,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28638,c1(NC(C(CCC)CNC(C2(C#N)CCOC2)=O)=O)ccc2nncn2c1 28639,C1(CCNC(c2n(C(C)C)cnc2)=O)CCN(C(=O)C(F)n2cccn2)C(C)C1 28640,C1(c2nnnn2C(C)C)(NCCSc2nnc(C)s2)CC(C)(C)SC(C)(C)C1 28641,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)n1)=O)N(CC#C)CC#C 28642,CCC(CO)NC(=O)NCC1C2CCC12 28643,c1(C(=O)NC(C(=O)N(C(CC(C)C)CO)C)CN(C)C)cc(F)cc(F)c1 28644,C=CCCCCCN(C(=O)CC1CCCN1C(=O)C(O)C1CCC1)C 28645,C(CCCCC(=O)NC1CCCN(CCCOC2CCCC2)C1)OCC 28646,C1(NC(CCS(C)=O)=O)CCC2(CCN(C(=O)CNC(=O)CC3CCCC3)C2)C1 28647,C1(C(N2CC(NC(c3cc(CCC)n(C)n3)=O)C2)=O)CC1C1CCOCC1 28648,C1(O)(CC(=O)NC2(CO)CCN(C(c3c(CC)ocn3)=O)C2)COC(C)(C)C1 28649,O=C(C1=CCCO1)NCCCN(C(=O)C(O)C1CC1)C1CC1 28650,N1(c2n(CC=C)c(C(C)C)nn2)CC(C)(C)CC(C)(C)C1 28651,N1(C(CCc2n(C)ccn2)=O)C(C(=O)NC2CCOC2)CC2CCCC12 28652,c1(C(C(=O)NC2CN(C(C3(C(F)(F)F)CC3C(F)(F)F)=O)C2)C)cccc(Cl)c1 28653,C1(N(C(=O)C(=O)NCCc2cccc(C3CCCCC3)c2)C)CCC(CO)CC1 28654,c1(OC)cc(C(=O)NC2CCCC2NC(C2(F)CC2)=O)cnc1O 28655,C(=O)(CCCCCNC(N)=O)NCC(CNC(CC1(COC)CC1)=O)O 28656,c1(C(N2CCCCC(N(C(CCCNC(C)=O)=O)C)C2)=O)cncc2sccc12 28657,c1(CC)c(C(=O)NCC2CN(C(C3(C(N)=O)CC3)=O)C2)cccc1Br 28658,C1(C(N2CCC(n3ccnc3)C2)=O)CCC(O)CN1C(=O)Cc1sccc1Cl 28659,C(=O)(N=c1[nH]oc2c1CC(C(=O)OC(C)(C)C)CC2)NCC(C#C)CC 28660,C(CCCCC(=O)NC1CC(Nc2cc(=O)n(C)cn2)C1)OC 28661,C12(NC(C(C)Sc3ncccn3)=O)CCCCCC1N(C(=O)CC(C)(F)F)CC2 28662,N1(c2nccc(C#N)n2)CCC2(NC(=O)C3=NNC(C(F)(F)F)C3)CCCC12 28663,Cc1cc(C(N2CC3CC(NC(c4ccc(C)n4C)=O)C2C3)=O)n2nccc2n1 28664,c1(C(=O)OC)nc(-c2c[nH]nc2CN(C(C)CC(C)C)C)c(C)o1 28665,N1(C(C(C)N(C(C2CCCCCN2C)=O)CC)=O)CC2CCCCC12C 28666,C1(c2n(-c3ccc(CC)cc3)nnn2)(NCCN(C)C)CCCC2(CCCCC2)C1 28667,C(C(=O)NCC1CCC(F)(F)C1)(C(C)(C)C)NC(C(N1CCOC1=O)C)=O 28668,C1(C(=O)NC(c2cn(Cc3ccc(Cl)s3)nn2)C)CC12CCOc1ccccc12 28669,N1(C(=O)CCc2ccc(O)cc2)CCC2CCCC12CNC(C1(F)CCCOC1)=O 28670,C1(C(N2CCC(C(=O)NC(C)CC3(C(F)(F)F)CCC3)C2)=O)CC(C)(C)CN1C 28671,C1(NC(C(Cc2cc(O)ncn2)NC(CC2CCC(=O)N2)=O)=O)CCC2CCC12 28672,N1(C(CC2CC(CC)C2)=O)CCC2CN(C(c3cnc4ccccn34)=O)C2C1 28673,c1(C(C)C)cnoc1C(N1CCCC1c1nc(COCc2ccccc2)no1)=O 28674,c1(C(=O)NCC(C)CN(C)C(C2CC(C)(F)C2)=O)ccnc2c1ccn2C 28675,c1(CNC(CC(=O)NCC(C)C)Cc2cccs2)cccc(F)c1I 28676,C1(N(C)C)(C(=O)NC(=O)CC2=CCCC2)CC2CCC1C2 28677,C1(OCC)CC(N(C)C(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28678,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)(C)CNC(C1CC1c1ccccc1)=O 28679,N1(C(c2cc(C)ns2)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)C2CCCCC12 28680,N1(C(CC(=O)NCC)=O)CC(C(=O)NCC(F)CO)CC12CCC2 28681,C1(O)(CCNC(c2c(CC)c[nH]n2)=O)CCCN(C(C2CC(O)(C(F)F)C2)=O)C1 28682,CCCCC(C(=O)N1CC2CCC2(CNC(=O)Cc2cccnc2)C1)N(C)C 28683,c1(C(=O)NC2C3(CC(NC(CCC(=O)NC)=O)C3)C2)oc2ccccc2c1Cl 28684,c1(C(c2ccnn2CC)NCC(=C)C)nnnn1C 28685,C#CCC(C(=O)N1CCCC(c2n[nH]cc2N(C)C(=O)OC(C)(C)C)C1)C1CC1 28686,C12(C(=O)NC3C(C)(NC(CC(C)SC)=O)CCC3)CC=CCN1CCC2 28687,N#Cc1cccc(F)c1NC(C1CCC(NC(c2cnccc2Cl)=O)C1)=O 28688,C1(c2c(C(N(C3CN(C(C4(C)CCCO4)=O)C3)C)=O)nco2)CCC(F)(F)CC1 28689,C(=O)(CC(C)CC(F)(F)F)NCCCNC(C(c1ccc(OC)cc1)C)=O 28690,C(=O)(CCCCCOC)NC(CN(C(c1n[nH]c(CC)c1Br)=O)CC)C 28691,C1(F)(C(=O)NC(C)(C)CNC(=O)CN2CCOCC2)C2CCCCC12 28692,Cc1cc(C(=O)NC2CN(C(=O)CCC3CCOC3)C2)cc(OCCN(C)C)n1 28693,c1(C(=O)NCC(C(C)C)NC(c2nc(C(C)OCC)sc2)=O)cn(C)[nH]c1=N 28694,N1(C(C(=O)N(C2CCOC2)CC)=O)CCC(C(N2CC3CCCCC23)=O)C12CCC2 28695,Cc1ccnnc1C(=O)NCC(O)CN(C(=O)C#CC(=O)N(C)C)C 28696,N1(C(C(C)(F)F)=O)CC2(CC(CNC(=O)C3=COCCC3)C2)C1 28697,C(CNC(=O)CNC(C)=O)(C(C)(C)C)NC(C1(COC)COC1)=O 28698,C1(C(=O)Nc2cc(C(CC)(C)C)n[nH]2)COCC1(C)C 28699,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1NC(=O)C(C)Sc1ccccc1 28700,C=CC1(CNC(=O)CCNC(=O)C(C)OCCC(C)C)CCC1 28701,C1(C2CCCN(C(c3ccc(F)c(OC)c3)=O)C2)(NC(COCCC#C)=O)CC1 28702,N1(C(C(=O)OC)C)CCN(C(=O)C(N2CCC(=O)CC2)=O)C(=O)C1 28703,C=CCC(CC)C(=O)NCC1CN(C)CCN1C(=O)CCCC(N)=O 28704,N1(C(C2CCCC(OCC)C2)=O)CC2OCCN(C(=O)C=CCO)C2C1 28705,C(CCN(C)C(C1CCC(F)(F)CC1)=O)(C(C)(C)C)NC(C1(C)ON=C(C)C1)=O 28706,N1(C(C(Cc2ncn(C)c2)O)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)C1C2 28707,Cc1nccc(C(=O)NC2C3CN(C(=O)Cc4ccccc4O)CC23)c1O 28708,C#Cc1ccc(C(N2CCN(C(c3c[nH]cc3Br)=O)C3CC23)=O)cc1F 28709,CC1(C)CCN(C(C2C3CC2N(C(=O)C(F)C2CCCC2)C3)=O)C1 28710,N1(C(=O)C2CC2)CC2CC1CN2C(C)COC(c1cc(CC)n(C)n1)=O 28711,C(=O)(C#CC1CCOCC1)NCCN(C1CCCCC1)C(C1CC(C)C1)=O 28712,c1(C2(CC)CN(Cc3cccc(-n4cncn4)n3)C2)ccc(Br)cc1 28713,N1(C(C(N2CCCCCC2)C)=O)C2CCCC1CN(C(=O)CC1(C)OCCO1)C2 28714,C1(NCc2c(C(=C)C)cccc2)C(C(O)=C)Cc2ccccc2C1=O 28715,c1(C(N2C(CNC(C3C(C=C)CC3)=O)CC(F)C2)=O)ccc(-c2cnco2)cc1 28716,N1(C(=O)OC(C)(C)C)CCC2(C(=O)Nc3ncc(Br)cc3C)CCCC12 28717,c1(NC(c2n(CCC)nnn2)c2ccc(Cl)s2)ccc(-c2nnco2)cc1OC 28718,Cc1cccc(C(=O)NCCOC2CCN(C(=O)C(C)S(C)(=O)=O)C2)c1N 28719,c1(C(=O)NC(C#C)(C)C)cccc(CNC(C2CC3(CC3)CO2)=O)n1 28720,N1(C(c2cc(COC)on2)=O)CCC(N(C(=O)Cc2cc(C)no2)C)C(C)C1 28721,C1(C(C)NC(C2CCN(C(=O)Cc3cccnc3)C2)=O)CCC(O)C1 28722,C=C(C)CC(C(=O)N1CC(COC)C1)NC(c1nocc1OC)=O 28723,C(=O)(CC(CC)C1CCC1)NCC1N(C(C(=O)NCCOC)=O)CC1 28724,C1(C(N2C(CC=C)COCC2)=O)CC2CCCCC2N1 28725,CN1CCC(O)(CNC(c2cc(CNC(c3cc(Cl)no3)=O)[nH]n2)=O)C1 28726,N1(C(C2(C)CCCC(=O)C2)=O)CCC(C)(C)C(NC(c2ccc(F)s2)=O)C1 28727,C1(CCNC(CCc2c(C)cccn2)=O)CN(C(C2CCOC2=O)=O)CCCO1 28728,C(N=c1[nH]c(=NCC2=CCOCC2)[nH]c2c1CCCCCC2)c1cn(CC)nc1 28729,c1(C(c2n(CC(=C)C)nnn2)NCc2cncn2CC)sc(Br)c(C)c1C 28730,Cc1cnc(NCC2(C)CCN(C(=O)CCC(C)(C)C)C2)c([N+](=O)[O-])c1 28731,c1(CNC(C2COCCN2C(c2cc(Cl)ncn2)=O)=O)ccc(Cl)cc1Cl 28732,C1(C(C(=O)NC(CSC)C)C)CCCN(C=O)C1.c1cnn(C)c1Cl 28733,N1(C(=O)OC(C)(C)C)CC(C(=O)OC2CCC2)C(C(F)F)C1 28734,c1(N)cnc2ccc(Br)cc2n1.c1(C(=O)NCc2n(CC)nnn2)ccc(S)nc1 28735,C1(CNC(CSCCOC)=O)CC(C)N(C(C2CCC(F)(F)C2)=O)C1 28736,C1(C(N2CCC(NC(CCC(N)=O)=O)CC2)=O)C2C3CC4C1C1C2CC3C41 28737,c1(SCC)ccccc1CC(=O)NCCC1CCN(C(C2CC3(CC3)C2)=O)CC1 28738,CC1(C)CCC(CC(N2CC(CCNC(C3(c4ccno4)CC3)=O)C2)=O)O1 28739,C(=O)(CCCC(C)(C)C)N(CCC(=O)NCCC(F)(F)C(C)C)C(C)C 28740,N1(C(c2nc(CC(C)C)sc2)=O)CC2CC(NC(=O)CCN3CCCC3=O)C2C1 28741,N1(C(c2cnc(C)nc2)C(=O)NC(C)(C)C)CCc2cc(C3CC3)ccc2C1 28742,C(=O)(CCC(C)(F)F)NCC.c12cccc(c1)OCCN(CCSC)C(=O)C2C 28743,CCC(C(=O)N1CCCC1CN(C)CCOC1CCCCC1)NCc1ccccn1 28744,Cc1sc(NC(=O)C2CC2)c(C(=O)NCC2CCCCC2NC(=O)CC#N)c1C 28745,c1(-c2cn(CC(C(=O)N(CC)Cc3cncnc3)C)nn2)cc(C)ccn1 28746,C=Cc1ccc(C(=O)NC2CCC(CNC(c3cc(CC)[nH]n3)=O)C2)cc1 28747,CS(=O)(=O)c1cnc(NC(=O)C(=O)NCC2COC(C3CC3)C2)nc1 28748,c1(C(N2C(C)CC(NC(C3(CCOC)CC3)=O)C2)=O)cnc(C)cc1C 28749,Cc1cc(C(N2CC(OCCNC(C3CC=CCO3)=O)C2)=O)sc1C 28750,C1(N(C(CS(=O)(=O)NC)=O)C)CN(C(C2CC(F)(F)C2)=O)CCC1O 28751,C1(C(N2CCC(CC=C)(NC(C3(C)C=CCC3)=O)CC2)=O)CC(C2CCCC2)C1 28752,c1(CCC)nccn1CC(=O)NCCN(C(=O)C(F)CC1CCOCC1)C1CC1 28753,c1(C(N(CC(=O)NC)CCC)=O)ccc(F)s1.C(=O)NC 28754,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28755,N1(C(Cc2cncc(OC)c2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(O)C1 28756,C1(NC(CCOC2CN(C(CC(C)SC)=O)C2)=O)CCC(C)CC1 28757,c1(C(=O)NC)ccc(C=CC(=O)NCC(CO)NC(C2CCCSS2)=O)cc1 28758,C(=O)(C1=CC2CCCCCC12)N1CC(NC(C(C)Cc2cnc[nH]2)=O)C(C)CC1 28759,CCC(CC(C)CO)NCc1ccccc1.c12cn(nn1)CCCN(C)S(=O)(=O)C2 28760,C=C(Cl)C(C)(C)C(=O)NC1CCN(C(c2ccc(CN3CCCC3)o2)=O)C1 28761,O=C(C1=CC(O)CCC1)NCC1CCN(C(c2ccsc2Cl)=O)C12CC2 28762,C1(NC(C)Cn2ccnc2)CCCN(CCCOc2ccccn2)CC1 28763,Cc1ccc(F)c(C(N2CC(C)(NC(c3cc(Cl)ncc3N)=O)C2)=O)c1 28764,C(CCS(C)=O)(C(=O)N1CCC(NC(=O)COc2ccc(Cl)c(F)c2)C1)N(C)C 28765,C(=O)(C1=CCC(C)CC1)N1CCC(O)(CN(C(C2(CCOCC)CCC2)=O)C)C1 28766,C1(=O)CCCCC(=O)NC2CCCCC12.c1(-n2cc(C)nn2)ccc(Br)c(C)c1 28767,C1(OC)(CNC(=O)CC(C)OC)CCN(C(=O)Nc2cccc(Cl)c2Cl)CC1 28768,c1(C2CC(C(=O)NC3C(CNC(=O)COC4CC4)C3)C2)ccccc1 28769,C1(NC(C(C2CC2)OCC)=O)CCC2(CCN(C(c3cn4cnnc4cn3)=O)CC2)C1 28770,C1(C(=O)NC(c2c(C)noc2C)C)CC(O)CCN1C(c1cnc(O)o1)=O 28771,N1(C(c2c(C)nn(C3CCOC3)c2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1C 28772,CC(CCCO)(C(F)(F)F)NC(c1csc(C(N)=O)c1)=O 28773,C1(CC(=O)NC(c2c(C)nccc2)C)C2CCCC2N1C(=O)C(C#N)C(C)C 28774,c1(C(=O)OCC)ncc(C(C)OC(=O)C(C)CO)s1 28775,C(c1cccc(F)c1Cl)=CC(=O)NCCCCN(C(CCNC(COC)=O)=O)C 28776,c1(C(N(C2CCOC2)CCNC(C(C2CCCC2)OC)=O)=O)ccccc1 28777,c1(CC)cccc(CNC(c2nc(C(C)OC)n(-c3ccccc3)n2)=O)n1 28778,C1(C(N(CC(=O)Nc2c[nH]nc2C)CCC)=O)CC2(CCC2)CO1 28779,c1(C(=O)N=c2ccn(-c3ccnc(OC(F)(F)F)c3)[nH]2)cc2c(cc1Br)OCCO2 28780,c1(CC(=O)NCC(C)N(C(=O)C(C)n2cccc2)C)cn(C)nn1 28781,c1(CNC(C2(F)CC2c2ccc(Cl)cc2)=O)ccc(Cl)cc1F 28782,CC(C)CC(CCO)NC(C1OCCC1CNC(C1(n2cccn2)CC1)=O)=O 28783,c1(C(=O)OC)cc(C)cnc1NC(C1CC(O)CCN1C(C1CCCN1C)=O)=O 28784,Nc1cc(C(N2CC3CC3(CNC(c3cnc(SC)s3)=O)C2)=O)c(F)c(O)c1F 28785,c1(CNC(CN(C(=O)CCN(C)CCO)C(C)C)=O)cccc(N(C)C)n1 28786,N1(CCCC)C(=O)Nc2cc(-c3csc(C#N)c3)ccc2S1=O 28787,S(=O)(=O)(c1ccc(N2CCC(CCCO)CC2)c(Cl)c1)NC(c1cn[nH]c1)C 28788,C#Cc1ccc(Cl)c(C(=O)NC2CCCC(NC(c3cnsc3C)=O)C2)c1 28789,c12ccccc1SCC(=O)N2.O=C1CCC(Cn2cc(C3CCC=CO3)nn2)C1 28790,C1(CNC(C2CCC(C)C2)=O)CCCN(Cc2sncc2Br)C1 28791,c1(OCCn2c(-c3c(F)cccc3)nnc2S)cccc2c(Br)cccc12 28792,C1(C(N(OCC(=O)OC)C)=O)(c2cccs2)CCOCC1 28793,C(N=c1[nH]c(=NCC2CCCC(CO)O2)[nH]c2ccsc12)c1c(C)cccc1Cl 28794,c1(COCCNC(C(C)(C)C2CC2)=O)cccc(-n2cc(C3CC3C3CC3)nn2)c1 28795,N1(C(c2cncc(-c3ccc(F)c(F)c3)n2)=O)CC2CCCCCCC2C1 28796,C(=O)(C1CCCc2nncn21)N1CC2CN(C(CN(C)C3CC3)=O)CC2C1 28797,N1(C(C2N(C)CCCC2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 28798,c1(CCC(N2CCC(NC(C)=O)C2)=O)ccc(-n2nc(C)cc2C)cc1 28799,c1(C(=O)NCCc2ccc(C#C)cc2)cc(OC)c(N)c([N+](=O)[O-])c1 28800,C(N=c1nc2scnc2c(N2CCOCC(F)(F)C2)[nH]1)c1n(C)nnn1 28801,C1(CC(=O)NC(C2CCOC2)CO)(NC(C(CO)N(C)C)=O)CCCCC1 28802,c1(C(=O)NCC2N(C(C(CSC)O)=O)CC=C2)c(C)cccc1C 28803,c1(C(N2C(C)CC(CNC(=O)C(c3ccccc3Cl)C)C2)=O)cncc(C#N)c1 28804,c1(C(N2CCC(NC(C(CCC)OCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 28805,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 28806,c1(C(N2CCC(N(C(=O)CCC)CC#C)CC2)=O)cccc(C#CC)c1 28807,C(c1nc2cc(Br)cnc2o1)=C(C)C 28808,CC1(CNC(C2(CCNC(c3cccc(F)c3F)=O)CCC2)=O)CCCCC1O 28809,c1(CN2CC(CC(=O)NCc3ncc(F)cc3Cl)C2)ccccc1[N+](=O)[O-] 28810,C(=O)(C1=C(Cl)CCC1)NCC1(CC(N2CC(CCC)C(CO)C2)=O)CCCC1 28811,C(CN=c1nc(N2CCC(C(C)(C)CO)CC2)c2c([nH]1)CCS2)SCC 28812,N1(C(C(CCC)NC(C2(COC)CC(=C)C2)=O)=O)CCCC2OCCC12 28813,c1(CC)cn2c(n1)CC(C(=O)NCC(C)N(C)C(c1cc(C)cc(O)c1)=O)CC2 28814,N1(C(=O)NC(c2nc[nH]n2)C)CC2CC2(C(=O)N(c2ccccc2)C)C1 28815,c1(NC(=O)N(C2CCN(c3ncc(F)cn3)C2)CC2CCOC2)ccc(F)cc1 28816,n1(CCC(N2C(C(C)NC(C(C)OC)=O)CCC2)=O)ccc2ccccc12 28817,C1(C(N2CC(NC(=O)C(F)=C3CCC3)C3(CCC3)C2)=O)CC12CCC(F)(F)CC2 28818,CCCCC(C)CCC(=O)NC(CNc1snc(Cl)c1C#N)CO 28819,C(=O)(C1=C(C)OCCS1)N1CC(OCC)C(CNC(C2CCC(C)(C)OC2)=O)C1 28820,N1(C(C2C(C=C)C2)=O)CC2CN(C(c3ccc(SC)cc3)=O)CCC12 28821,N1(C(C2(C)COC2)=O)CC2CC(C1)C(CO)C2NC(c1noc2ncccc12)=O 28822,c1(OC)ccc(C(=O)NC(=O)N(CCN(C)C)C2CC2)c(Cl)c1 28823,N#CC1CCN(C(C2CN(C(c3csc(Cl)n3)=O)CCO2)=O)CC1 28824,c1(-n2c(CCC3CC3)nc(-c3ccc(N(C)C)cc3)n2)ccc2ccn(C)c2c1 28825,c1(C(=O)NCC2(NC(c3c(CCC)n(CC)nn3)=O)CC2)ccnc2ccsc12 28826,C(=O)(C1=CCOCC1)N(CCCCN(C(=O)CC1CCN(C)C1=O)C)CCO 28827,CN1N=C(C(=O)N2CCC2CNC(c2cccnc2C2CCCC2)=O)CCC1=O 28828,c1(C(=O)NCCC2CSCCN2C(=O)C=CCF)csc2c(F)cccc12 28829,c1(SC)ccc(CN2CCN(C(C)C(=O)NCc3cncs3)CC2)cc1 28830,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2F)=O)CCO1 28831,c1(C(N2CC(CNC(C)=O)OC(C)(C)C2)=O)cc2c(C)nn(C)c2s1 28832,c1(C(C)(F)F)nc(C(=O)NCCCNC(C2CCCN2c2ncccn2)=O)cs1 28833,CC1CC2CN(C(=O)C(CO)N(C)C)CC2N1C(c1ccc(COC)o1)=O 28834,c1(CCC)cc(C(N2CC(COC)CC2CNC(=O)CC2CCNC2=O)=O)no1 28835,Cc1noc(C)c1C(C)C(=O)NCC1(CNC(C2(C)CNC(=O)C2)=O)CC1 28836,C=CC(CN(C)C)N=c1nc(N2CCCC(CCOC)C2)c2cnn(C)c2[nH]1 28837,c1(C(N(CCn2cc(-c3csc(C)n3)nn2)CC)=O)cc2c(cn1)OCO2 28838,Cc1cc(C)n(CCNC(=O)CC(C2CC2)NC(=O)CC2CC(C)(C)CO2)n1 28839,c1(OCC)cc(C(N2CCC(N(C(=O)C(C)(C)CO)CCO)C2)=O)cnc1OC 28840,c1(C(=O)NCC2(CCNC(CCN(C)C3CC3)=O)CC2)scnc1C1CC1 28841,CCCC(C)(C)CC(=O)NC1C(C)(C)C(NC(C2CSCCS2)=O)C1(C)C 28842,Cn1cccc(C(=O)NCC2CN(C(C3(F)C4CCCC34)=O)CC2O)c1=O 28843,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1CO 28844,c1(CC)nc(Cl)nc(N2CCCC2CN(C(=O)C(C)(C)n2cnnn2)C)c1C#N 28845,C1(NC(=O)Cc2cccc(Cl)c2)CN(C(=O)C(F)C2CC2)CC2(CCOCC2)C1 28846,C1(C2CCN(C(=O)CC3OC(C)(C)OC3=O)CC2)(NC(C2CC(SC)C2)=O)CC1 28847,C12(NC(c3c(CSC)scc3)=O)CCN(C(=O)CNc3ccccc3)CCC1C2 28848,c1(C(=O)NC2CCC(CNC(=O)CCn3cccn3)C2)cc2c(=O)[nH]ccn2n1 28849,N1(C(C(C)OCC2CCCO2)=O)CCCOCC1 28850,C1(CC(N2CC(O)(C(C)NC(c3n(C(C)C)ccn3)=O)C2)=O)COCC(C)(C)O1 28851,c1(CNC(C(COC)C)=O)ccccc1CNC(C)=O 28852,C(C(C(=O)N1OC2CCC1C2)NC(=O)C(c1cccnc1)OC)SCC 28853,C1(CC)CCN(C(c2ccc(O)cc2)=O)C1C(=O)NCC1CCCCC1 28854,N1(C(C)=O)CC(O)CC1C(=O)NCC1C=CCN1C(=O)CCOCC(F)(F)F 28855,C1(CC(=O)N(CC(O)CO)CC)CCN(C(=O)CC2OCCC2(C)C)C1(C)C 28856,c1(C(=O)NCC(=C2CN(C(c3nc(OCC)oc3)=O)C2)F)cccc(C(C)C)c1 28857,C(=O)(CCCC1CC1)NC(C1(C(N(C(CC)C2CC2)C)=O)CC1)C 28858,Cc1[nH]nc(C(=O)NCC2CCCN2C(=O)CCN2CCOCC2=O)c1[N+](=O)[O-] 28859,c1(OC)cccc(-c2cc(-c3nccn3CCC3(C)CCCCC3)n[nH]2)c1 28860,c1(C(=O)NCC2(O)CCN(C(C3(CO)CC3(F)F)=O)C2)csc2ccc(F)cc12 28861,C1(NC(C(C)SCC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 28862,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 28863,CC1CCN(C(=O)C=Cc2ccccc2)CC1NC(=O)CC1CC(=O)NC1=O 28864,C1(NC(c2c(CCCC)ocn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 28865,C1(CNC(c2cc(C)[nH]c2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1O 28866,N1(C(=O)Nc2c(CC(=O)OC)ccs2)CCN(Cc2cnccc2C)CC1C#N 28867,c1(NCCN(C2CCN(C(=O)CC(F)(F)F)CC2)CC)cccc(OC)c1C 28868,C1(C(N(CC(C)NC(c2cnc(O)s2)=O)CC)=O)CCC(NC(C)=O)CC1 28869,c1(C(C)OC)ncc(C(=O)NC(C)C(C)(C)NC(c2ccnn2C)=O)s1 28870,CCCCC(O)C(=O)NCC(CNC(C1Cc2nccn2C1)=O)S(C)(=O)=O 28871,C1(NC(CC(C)C)=O)CCCCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 28872,c1(CN2CC(c3cn(NC(C(c4ccccc4)C)=O)nn3)C2)cccnc1F 28873,c1(C(C(C)NC(C=C(COCC)C)=O)NC)ccccc1Oc1ccccc1F 28874,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 28875,N1(C(C(C2CCC2)OC)=O)CCC(CF)(NC(=O)Cc2ccnc(O)c2)C1 28876,Cc1scnc1C(N1CCC1(C)CC(=O)NC(C)Cc1ccccn1)=O 28877,C1(C(=O)NCC(CN(C(c2c(C)occ2)=O)C)C)C2CCC1(c1ncco1)C2 28878,C1(CC)CN(C)C(=O)CN1C(C1CN(C)CCN1C(=O)CC1COC(=O)C1)=O 28879,N1(C(=O)NC(c2cncc(OC)c2)C)C2COCC1CC(F)C2 28880,C(=O)(C1COc2ccccc21)NCC1(C)CCN(C(c2cc(F)ccc2N)=O)C1 28881,C1(C(N(C2(CC(=O)NC3(COC)CCOC3)CC2)C)=O)CCCC(=O)C1 28882,C1(NC2CCC(OCC)CC2)CCCCNC12CC2 28883,CCCCC(=O)C(=O)NC(CNC(c1ccco1)=O)CC(C)C 28884,C=CC(F)(F)C(=O)NCCCN(C)C(C1COC(C)(C)C1)=O 28885,c1(NC(C2C(OC)CCC2)=O)nc2c(C)cccc2o1.N12CCCC(C)C1C2=O 28886,C12(NC(C3C(C)C3)=O)CC(CO)(C1)OC21CN(C(=O)C2CCCc3ncnn32)C1 28887,C1(CC(=O)N(CCCCNC(C2CCC2)=O)C2CC2)OCCCO1 28888,c1(NC(N2CCCC2COCC(F)F)=O)nc2cc(Cl)cc(Cl)c2o1 28889,c1(C(N2CCC(C(C(=O)NC(c3nnc(CO)o3)C)F)C2)=O)nc(=N)cc[nH]1 28890,c1(CC)nc(Cl)nc(N2CCCCC(CNC(C3(CCN)CC3)=O)C2)c1C#N 28891,C12(C(=O)NCC3CCN(C(C(=O)NCC)=O)C3)C=CC(CC1)C2 28892,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 28893,CC(C)(F)CC(=O)NC1(CF)CCN(C(=O)CCNC(=O)OC(C)(C)C)C1 28894,CC1(C)CCCC1(O)CNC(=O)CC1(NC(C2OC3CCC2C3)=O)CC1 28895,CCCCC(O)CCC(=O)NC1CCSC12CN(C(=O)C(c1ccc(F)cc1)C)C2 28896,Cc1noc(Cl)c1CCC(=O)NCC(n1cc(-c2cn(C)nc2CO)nn1)C 28897,c1(C(N2C(C)CC(NC(=O)CNC=O)C2)=O)ccccc1S(=O)(=O)CCN(C)C 28898,C1(NC(C2COCCO2)=O)CCCCN(C(=O)CN2C(=O)CNC2=O)C1 28899,Cc1cccc(CNC(=O)C(=O)NC2CC3(CCC3)C2)c1C#N 28900,CCCC(CCCNC(=O)C(O)CSC)NC(c1ccc(Br)cc1)=O 28901,CC1(C(N2CCC(C)(CCNC(=O)CSc3n[nH]c(=N)s3)C2)=O)COCCO1 28902,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 28903,n1(CC)nccc1C=CC(=O)NC1CCCC(CNC(c2ccsc2CC)=O)C1 28904,CC(CC(=O)N1CCC(C)(N(C)C)C1)C(C)(C)NC(C1C2CCCC12)=O 28905,C1(CNC(CN2CC(CC)C2)=O)CN(C(c2cnn(C)c2N)=O)CCC1(F)F 28906,CC1CC=C(C(=O)NCc2cncc(C(=O)NC(c3nnc(O)n3C)C)c2)CC1 28907,C(=O)(CC(C)(C)C(=O)NCC(C)CC(=O)NCCn1ccnn1)OC 28908,C(CCCCC(=O)NC1CC(NC(=O)CC2CC(F)C2)C12CCC2)OCC 28909,c1(C(=O)NC2CC(C)(NC(C=CCC)=O)C2)ccc(C(=O)NC2C=CCC2)cc1 28910,N1(c2c(OC)cccc2)CCC2(C1)CN(N1CC(O)CC1C(C)C)C2 28911,c1(NC(=O)CSc2ccc(Cl)c(F)c2)nc2ccccn2c1[N+](=O)[O-] 28912,c1(OC)cccc(Cl)c1CN1CCCCC1CNC(c1nnco1)=O 28913,C1(CCC(=O)NCC2CC(NC(C(C#N)C3CC3)=O)C2)NC(=O)NC1=O 28914,C1(C(=O)NCC2C(CC(=O)N(C(CC)CO)C)C2)(SC)CC(=O)C1 28915,N1(C(C2(SC)CN(C(C3CC4CCC4C3)=O)C2)=O)CCCC(N=[N+]=[N-])C1 28916,c1(N(C(C)C)CCO)cc(N)c(Cl)c(O)n1.c1(CCCCNC=O)cn(CC)nn1 28917,C(C(F)C(C)CC(C)(C)C)OC(C(=O)Nc1c(OC)cccc1)C 28918,c1(C(=O)NC(C2CCN(C(CSCCC)=O)C2)C)cc2c(C)ccc(F)c2o1 28919,C(c1ccco1)=C(C)C(N1CCC(C(C)NC(=O)C(F)=C(C)C)C1)=O 28920,CCC(C)(O)C(=O)N1CC(N(C)C(c2ncccc2OCC(F)(F)F)=O)C(O)C1 28921,N1(C(c2cc(C)n(C)c2)=O)CC(C)(C)OCC1C(=O)NCC12CCCC1OCC2 28922,C1(C)(C(=O)NCc2c(C)cco2)CCCN1C(C1CCC2CC12)=O 28923,C(=O)(C#CC1CCCOC1)N1CC(N(C(=O)C2=NN(C3CC3)C(=O)CC2)C)C1 28924,C1(CNC(c2c(CC)c[nH]n2)=O)CC2CCC(C1)N2C(=O)C(COC)OC 28925,CC1CN(C(C2CCCCO2)=O)CC1(C)CNC(=O)CSc1ccc(F)cc1 28926,N1(C(C2C(C(N)=O)C2)=O)CCCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 28927,Cc1cc(C(=O)NCCOCCN(C)C(c2cccc(C(=O)N(C)C)n2)=O)sc1C 28928,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 28929,CCCCC(C)(C)C(=O)N1CC2C(C(=O)NCC(=O)NC(C)C)C2C1 28930,N1(C(c2ccc(CNC(C)=O)o2)=O)CCCCC(CNC(=O)C(Br)=C(C)C)C1 28931,c1(C(=O)NCC(CC(C)C)NC(C2NC(=O)C3CC23)=O)cn2c(n1)CCC2 28932,C(=O)(C(C)C(F)(F)F)N1c2nnc(n2C2CC2)C12CCC2.C(C)(C)(C)OC(C)C 28933,C1(C(N2CCC(CNC(C3CC4CCC3CC4)=O)C2)=O)CCC2CCC1O2 28934,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1C(C)CN(C(=O)CSC2CC2)C1 28935,c1(OC)ccc(NC(C2COCCN2C(c2ccc(C)cn2)=O)=O)cn1 28936,Cc1c(CCNC2CCCCC2F)nc(Br)n1C 28937,C#CC1CC2CCC1N(c1cc(F)c(Cl)cc1Cl)C2 28938,C1(CN(C(C(C)c2ccco2)=O)C)CCCN(C(=O)CCNS(C)(=O)=O)C1 28939,Cn1nc(C(=O)NCC2C3CN(C(C4(C)CCC4)=O)CC23)cc1Br 28940,C1(CNC(C2(Cc3ccccc3)CCOC2)=O)NCC12CCC2 28941,N1(C(c2c(C)occ2)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1C1CC1 28942,c1(SC)ccc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc1Br 28943,c1(C(=O)NC(CCCC)CNC(=O)CN(C)CCC)ccc(Cl)c(S(N)(=O)=O)c1 28944,n1(CC(=O)NC2C(CNC(c3c(CC)cco3)=O)C2)c(C)nc2ccccc12 28945,c1(CC)ccccc1CC(=O)NCCC1(NC(=O)C=C(C)c2ccco2)CC1 28946,Cc1nccc(C(=O)NC2(C(=O)Nc3cn(C)nc3O)CCN(C)C2)c1N 28947,C1(O)(C(C)C)CCN(C(c2ncccc2NS(=O)(=O)C(F)(F)F)=O)C1 28948,c1(C(N2CC3CCN(C(CC(C)C(F)(F)F)=O)C3C2)=O)cnn(C)c1S(N)(=O)=O 28949,C1(CC(=O)N(CCC)Cc2ccn(C)n2)(CC)CNC(=O)O1 28950,C1(C)(CC)CC(C(=O)NCC(CO)NC(=O)CC2CSCCO2)C1 28951,N1(Cc2cn(CCCN(C)C)nn2)CCOCC12CCS(=O)(=O)C2 28952,N1(CC(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C(=O)NC2(CCCC2)C1=O 28953,C1(NC(c2n(C=C)nnc2)=O)CC2CC1CN(C(=O)C(C)(C)c1cnsc1)C2 28954,N1(C(C(COCC)C)=O)CCN(C)C(CNC(c2ncc(C)cn2)=O)C1 28955,O=S(=O)(c1cc2sc(=NCCCS(=O)(=O)C(F)(F)F)[nH]c2cc1Cl)NC1C=CCC1 28956,N1(C(C)(C)C)CCC(CNc2cn(C3CCCC3)nn2)CC1 28957,Cc1cc(=NC(Cc2ccccc2)C(C)C)[nH]c(=NCC(C)(C)C(F)(F)F)[nH]1 28958,c1(SC(C(=O)OC(c2ccccc2)C)C)cccc(OC(=N)O)c1 28959,C1(CNC(C(C)Cc2cccc(F)c2)=O)CCN(C(=O)C2=CC(C)(C)C2)CC1C 28960,C(=O)(C#CC1CCCCC1)N1CCCC(F)(CNC(C2C(OC)CCCC2)=O)C1 28961,CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)CC2CO)CCCC1 28962,c1(N2CCC(N(c3c(C(=O)OCC)nccn3)C)C2)ncc2c(Br)cccc2n1 28963,c1(C(N(CCC)CCNC(=O)CN(C)C(N)=O)=O)cc(F)ccc1OC 28964,O=C(CCCCF)NCCCCC1CN(C(=O)COC2CC=CC2)C1 28965,Cc1noc(Cl)c1CC(=O)NC1CCCCC1NC(C1(F)CC=CCC1)=O 28966,c1(CCC(=O)NC(C(C)C)CNC(C2(C(C)(F)F)CC2)=O)ccc(F)cc1F 28967,Cc1ccn(C)c1C(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1C(F)(F)F 28968,C1(C)(CNC(C(CCC)C)=O)COCCN(C(c2ccc(CO)cc2F)=O)C1 28969,c1(C(N2CCCC(n3ncc(C)c3)C2)=O)sc2ncn(C)c(=O)c2c1C 28970,c1(OC)ncnc(C(=O)NCc2ccc(C#N)cc2)c1F.C12(O)CCN(C1)C2=O 28971,N1(C(C(CC#C)O)=O)CCN(C(=O)CC(C)C)CC1C(C)COC 28972,c1(C(=O)NC2CC(CNC(Cc3nc(C)sc3)=O)C2(C)C)ccc(CO)c(Cl)c1 28973,Clc1ccc2c(c1)CCC2NCC1(c2cn(C3CCC3)nn2)CC1 28974,O=C1NCCC2C(C(N3CCCC3c3ccsc3)=O)C12 28975,CN1CCC(OC2(C(N3CCCC(CCC(=O)NC4CNC(=O)C4)C3)=O)CC2)CC1 28976,c1(C(=O)NCCCN(C)CC2COC(C)(C)O2)ccc(C23CCC(C2)OC3)cc1 28977,c1(OCC)cnc(Cl)[nH]c1=NC(=O)C1(Cc2ccccc2-c2ccccc2)CC1 28978,C1(NC(c2ccc(C(=O)OC)nc2)=O)CN(C(=O)C=CC2CCC2)CC12CCC2 28979,C1(NC(c2cc(C(C)C)on2)=O)CCCCC1CNC(=O)C(C)CN(C)C 28980,Cn1ccc2cc(-c3nc(C4CCOC4)nn3Cc3nc[nH]n3)ccc12 28981,c1(CNC(c2cccc(Cl)c2Cl)C(=O)OCC)scc2c1OCCO2 28982,c1(C(=O)NCC(C)N(C(CC(CCC)C)=O)C)c(F)cc(F)cc1F 28983,c1(C2(C(N3C(CNC(c4c(C)cns4)=O)CC3)=O)CC2)ccccc1C 28984,C1(NC(C)C)CCCCN1C(=O)CCC1CCCCO1.c12cccc(c1)OC2 28985,N1(C(C(C2CCOC2)OCC)=O)CCOC(CN(C(=O)CN(C)C(C)C)C)C1 28986,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 28987,N1(C(CCC(C)NC(=O)CC2CC3C=CC2C3)=O)CCC2C(C1)C2(F)F 28988,C12CCCCN1C(=O)S(=O)(=O)C2.C1(NC)CCN(C(=O)OCCN)C1.C(C)(C)C 28989,N1(C2CCN(C(=O)CCF)CC2)C2CCC1CN(C(C1C=CCC1)=O)C2 28990,C(C(F)(F)C(=O)N1CCC(C(C)NC(=O)COCc2ccccc2F)C1)OC 28991,c1(C(=O)NC(C2CCOC2)CNC(C2(C)CC2(F)F)=O)cc2nc(F)ccc2o1 28992,OC1(CN2CCCCC2c2n[nH]c(-c3ccccc3)n2)CN2CCC1CC2 28993,C=C(Cl)CCC(=O)N1CC=CC1C(=O)NCCC1CCCCO1 28994,C(=O)(C1=C(Cl)CCC1)N1C(C(=O)NCCCN(C(C)C)C)CCC1 28995,N1(C(c2ccc(CC)cc2)=O)CC2CCC1CN2C(=O)C(c1csc(C)n1)=O 28996,c1(CC(=O)NC2(CO)C(C)C2)csc(-c2cccnc2)n1 28997,C1(C(=O)NC(C2CCN(C(=O)C(F)CC3CCCC3)CC2)(C)C)SC(=N)NC1=O 28998,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(c1csc(C)n1)=O)C2 28999,c1(C(=O)NC23CCN(C(C=C(C)C4CC4)=O)C2CCC3)ccc2c(c1O)CCC2 29000,C1(C(C)NC(c2cnsn2)=O)CCCCN1C(=O)CCC1CC1CC1CC1 29001,CC(C)C(C(=O)NC1CC(CNC(c2nocc2Cl)=O)C1)N(C)C 29002,n1(CCC)nc(C)cc1C(=O)NCC1CCCC1NC(C1(C)CC1C)=O 29003,c1(C(N(C2CC3CC2CN3)CCCOC)=O)ccc(Br)cc1 29004,c1(CCOC(C(CSC)OC)=O)cc2cnccc2[nH]1 29005,c1(C(=O)NC2CCN(C(COCC(C)(C)C)=O)CC2O)cc(Cl)c(Cl)c(Cl)c1 29006,C1(NC(C(CCOC)NC(C2C=CCC2)=O)=O)CCN(C)CC1C 29007,c1(C(=O)NCC(F)CNC(C2CCC2)=O)cc2sc(Br)cc2[nH]1 29008,Cn1c(CNC(=O)C(=O)Nc2cc3cc(Br)ccc3s2)cc2ccccc12 29009,Cc1nc(O)[nH]c1C(=O)NCCC1(O)CCN(C(=O)C(C)Cc2cnco2)C1 29010,N1(C(COCCCCC)=O)CC2CC(C(=O)NC(CO)C3(C)CC3)(C2)C1 29011,C1(C(N2CCN(C(c3ccc(-c4ccccc4)[nH]3)=O)CC2)=O)CC12CCCOC2 29012,c1(C(N2CCC(C(=O)OC)CC2(C)C)=O)cccc2c1CCCC2 29013,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29014,C(C)(CCC(=O)NCC1CCN1C(=O)COCCc1ccccc1)OC 29015,c1(C(N(CC(CC)NC(C2CC23CCOC3)=O)C)=O)ccc(C)c(C(=O)OC)c1 29016,c1(C(=O)OC)ccc(CCc2cn(-c3ccc(C(=O)NO)cc3)nn2)cc1 29017,c1(C(=O)NCC2(OC)CN(C(c3coc(C)c3)=O)C2)cncc2c1CCNC2=O 29018,c1(NCc2c(C)nc(C)s2)cc(=NCCS(=O)(=O)N2CCCC2)[nH]c(C)n1 29019,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29020,N1(CCC(=O)NC(C2CCCN(C(=O)CCF)C2)C)CCCCC1=O 29021,c1(OC)ccc(C(=O)NCCCCCCNC(C2CCCCN2C)=O)nc1N 29022,Cc1cccc2oc(C(N3CCC34CCC(c3cc(C(=O)O)n[nH]3)CC4)=O)cc12 29023,C1(CN(C(=O)CC2CC3CC3C2)C)COCCN1C(c1ccncc1Cl)=O 29024,Cc1nccn1CC(=O)NC1(C(=O)NCCN2CCC(C)C2)CCC1 29025,N1(C(C2C(CC)CCCN2C(=O)Cc2ccnn2C)=O)CC(S(C)(=O)=O)C1 29026,C1(NC(C2(NC(CSC(C)C)=O)CCC(C)(C)C2)=O)CC(C2CCCC2)C1 29027,CC1(NC(=O)Cc2cc(C3CC3)n[nH]2)CCCN(C(=O)C(F)F)C1 29028,N(C1CN(C(=O)C(O)c2ccsc2)Cc2ccccc21)C(C1(C(=O)OC)CC1)=O 29029,CC1(C)CCC2CC(N)c3cccc1c32.C1(C2(C(=O)N)CCC2)CCCCO1 29030,c1(OC)cnc(C(=O)N(C)Cc2cccc(CNC(C3(O)CC=CC3)=O)c2)nc1 29031,N1(C(C=C(C)C(C)(C)C)=O)CCCC2CN(Cc3cncc(C#N)c3)CCC12 29032,c1(CN(C(c2ncc(Cl)n2C)C(=O)NCCCC)C)noc2ccccc12 29033,C(C(=O)N1CC(n2cc(CC(=O)OC(C)(C)C)nn2)C1)(C(C)(C)O)NC1CCCS1 29034,c1(CC(=O)N(C(CN(CC)CC)C)C)cccnc1.C(C(C)(C)CO)N 29035,c1(CN2C(C(=O)NCc3nc(C(F)(F)F)cs3)CC2)csc2ccccc12 29036,Cc1cnn(C)c1C(=O)NC1CCN(CCN(c2ccc(N)cc2)S(C)(=O)=O)C1 29037,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29038,Cc1ccc2c(c1)CC(C(=O)N(CCCC(N1CCCCC1C)=O)C)S2 29039,C12(C(=O)NC(c3cnc[nH]3)C)CCCC1CCN2C(C1OCCO1)=O 29040,CN1CCC(COC(c2cn(Cc3cccnc3)nn2)=O)C1=O 29041,C1(NC(CC2CCCC(C(N)=O)C2)=O)CC12CCN(C(c1ccc[nH]1)=O)CC2 29042,C=Cc1cnn(C)c1C(=O)NCCN(C(=O)Cc1ccc(Cl)c(OC)c1)C 29043,CCCCN=C(NCc1ccn(CCOCC)n1)NC1CCCC1 29044,c1(N2CCCC(C(N(CC(C)O)C)=O)C2)cc(Cl)c2c(c1)OCCCO2 29045,CC(C)CCC(C(=O)N(C)CC1(O)CN(C)C1)NC(=O)C(O)C(C)(C)C 29046,c1(CCCC(=O)NCC(CCNC(C(C)O)=O)(C)C)cncc2ccccc12 29047,C#CCC(C(=O)OC)NC(C1CCOCC1NC(c1cncc(F)n1)=O)=O 29048,c1(NCC(=O)NC2CC3CNCC23)ccc(N2CCOCC2=O)cc1 29049,N1(C(c2nn(C)c(Cl)c2)=O)C2CCC(C2)C1C(=O)NCC(F)(F)F 29050,c1(C(C)NCC(COC)(C)C)ccc2nsnc2c1 29051,N1(C(c2c(C)nsc2)=O)CC2=C(C1)CN(C(C13CC(C1)C(c1ccccc1)O3)=O)C2 29052,N12CCC(CO)(CC1)N(C)C(=O)C2.c1(CN2CCC(C)(C)C2)ccccc1Cl 29053,CC(C)(CCC(=O)NCCNc1nccc(-c2ccnn2C)n1)[N+](=O)[O-] 29054,C=C=CC(C)C(=O)N1CC(NC(c2cnc(OCC)nc2)=O)C(C)C1 29055,c1(C(N(C)CCN(c2cc(=O)n(C3CC3)c(O)n2)C)=O)ccc2c(c1)COCC2 29056,N1(C(CCNC(NC)=S)=O)CCC(C(N2CCCC(C(=O)OC)C2)=O)C12CCC2 29057,CCS(=O)(=O)c1ccc(F)c(C(=O)NCCC(=C)CNC(=O)Cc2ccnn2C)c1 29058,c1(C(=O)NC2(CO)CCN(C(c3c(OC)scc3)=O)CC2)ccc([N+](=O)[O-])cn1 29059,C=CCC(C)(C(=O)NC1CC(C)(NC(c2cnn(CCO)c2)=O)C1)N(C)C 29060,C1(NC(C(CN(C)C)NC(C2CC3(C2)CC32CC2)=O)=O)CCCCCC1(C)C 29061,C(C(C)(O)CCC)NC(CNC(C(C)OCCC)=O)=O 29062,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)NC(C3CCC3)C)C2C1 29063,c1(C(N2CCC(C)(C(N(CCOC)CCO)=O)C2)=O)cc(C(N)=O)cc(C)c1 29064,N1(C(CCCC)=O)CCCCC1CCCNC(C1(c2ccnn2C)CC1)=O 29065,c1(C(N2C(C)(CNC(=O)C3=C(Cl)CC3)CCC2)=O)cc(=O)n2ccccc2n1 29066,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)ncn2C)=O)CC1 29067,N1(C(c2ccc(C(C)C)cc2)=O)CC2CC(NC(C3CCCC(C)C3)=O)CC2C1 29068,N1(C(C2CC(CC)(CC)C2)=O)CCC2(CCCN2C(=O)C(F)OC)C1 29069,c1(CN2C3(C(=O)NC4CC(OCC)C4OC)CC(C2)C3)cn2cc[nH]c(=O)c2n1 29070,S(=O)(=O)(c1c[nH]ccc1=NC(C)c1ccc(N(C)C)cc1)N(CC(CCC)C)CC 29071,C=C(C)CC(C(=O)NC(C)C(=O)NC1CC1)NC(=O)Cc1ccsc1 29072,C1(C)(C(N(C2CCN(C(C3(n4nccn4)CC3)=O)C2)CC)=O)CC(C2CC2)=NO1 29073,Cc1cccc(-c2cn(C3CC(NC(C4(CO)CC5CCC4C5)=O)C3)nn2)c1I 29074,Cn1cc(-c2nc(C(N3CC(F)(CNC(C4CCOC4)=O)C3)=O)co2)cn1 29075,C1(C#CC(=O)N2CCC(OCC(=O)N(C)C(C3CC3)C3CC3)C2)(CC)COC1 29076,C1(C)(NC(C=CC)=O)CCN(C(c2oc(-c3ccccc3)nc2C)=O)C1 29077,C1(CNC(C2C(C=C)C2)=O)CCCCCN1C(=O)CCOc1ccccc1C 29078,Cc1[nH]nc2c(C(=O)NC(C)(CNC(c3nccnc3Cl)=O)CO)cccc12 29079,N1(C(CCC#CC)=O)CC2(CC(NC(=O)C(=O)NCC(F)F)CO2)C1 29080,S(=O)(=O)(c1ccc(=NCC2CC(O)C2)[nH]c1)NC(C1CCCC(F)(F)CC1)C 29081,N#CCCCN=c1[nH]c(N2CCC3(CCCC3)C2)nc2cccnc12 29082,Cc1oc(C(N2CC(NC(=O)C(=O)NC(C)(C)C)C(O)C2)=O)cc1S(=O)(=O)N(C)C 29083,C(=O)(C(C(=O)NCC(C)(CO)NC(=O)C(C)Cc1cnc[nH]1)C1CC1)OC(C)(C)C 29084,C(=O)(CCC(C)(C)NC(c1ncccc1F)=O)NC(c1nc(C)on1)C 29085,c1(CN(C)C(=O)NC2CCC(C)(C)CO2)c[nH]c2ccc(Br)cc12 29086,c1(C(=O)NCC2CCCC(NC(CCCSC)=O)C2)coc2c(F)cc(Cl)cc12 29087,c1(C(=O)NCC2CC(CNC(COC)=O)OC2)cc(N)c(Cl)c(O)n1 29088,N1(C(C=CC=CC)=O)CC(NC(c2cccc(OCCC)c2)=O)C(C)C1 29089,c1(OCC)ncccc1CC(=O)NC1(CCNC(=O)C=C=C(C)C)CC1 29090,N1(C(Cn2ncc(C)c2)=O)CCCCC1C1CCN(C(=O)C(C)CF)C1 29091,Cn1nc(C(=O)Nc2ccc(NCC3CCCOC3(C)C)cc2)c2ccccc12 29092,C1(C(N(CCCCC(=O)NCC2CC(F)(F)CO2)C)=O)CC2COCC2C1 29093,N1(C(C2CCCN(C(=O)OC)C2)=O)CC2(CCC2NC(=O)C(F)=C(C)C2CC2)C1 29094,C1(NC(CS(=O)(=O)NC(C)(C)C)=O)CN(C(C2(C)CCOC2)=O)CCC1C 29095,C(=O)(C(=O)NNC(=O)C1CCCC1)NC1(OC)CC(CN2CCCC2)C1 29096,c1(C(N2CCN(C(C(CC#C)C)=O)CC2)=O)sc2ccccc2c1CS(C)=O 29097,C1(C(=O)NC2CC(F)(F)C2)CC(F)(F)CN1C(c1cncs1)=O 29098,CCN=c1ccc(C(=O)NC2CC(CCNC(c3csc([N+](=O)[O-])c3)=O)C2)c[nH]1 29099,c1(N(CC(C)C)C(N2CCC3CC(C)(C(=O)O)C3C2)=O)cccc2ccccc12 29100,C1(NCc2ccc(COCCOCC)cc2)CCC(P(C)(C)=O)C1 29101,C1(O)(CN(C(C(C2CCCCC2)C)=O)C)CN(C(c2nocc2C)=O)C1 29102,c1(C(=O)O)cc(S(=O)(=O)N2CC3CC4CCCN4C3C2)c(F)cc1I 29103,CC1CC(C)N(C(c2cccc(NC(N)=O)c2)=O)CCN1C(=O)C=C1CCN(C)C1 29104,C1(O)(CCC)CCN(C(c2cc(CNCC)c[nH]2)=O)CC1.C(=O)(C(C)P(C)(C)=O)N 29105,N1(C(C2N(C)CCCC2)=O)CC2CCC2(CCNC(c2ccc(CO)cc2)=O)C1 29106,N1(C(C#CC(=O)N(C)C)=O)CC2CC(NC(c3cc(CCN(C)C)on3)=O)C2C1 29107,N1(C(C2C(C)C2)=O)CCC(CNC(=O)CCc2c(N)cnn2C)C1(C)C 29108,C1(C(=O)NCC(CC)NC(=O)CCCn2ccnc2)CCCC(=O)O1 29109,c1(N(C)C(C2CCC(c3nc[nH]n3)O2)=O)ncc(Br)cc1C#N 29110,CC1CC(=O)NC(C(N2CC(C)(NC(c3ccc(C(F)F)c(F)c3)=O)C2)=O)C1 29111,C1(NC(CCC#CC)=O)CC(O)CN(C(=O)CC(C)Cc2ccc(Cl)cc2)C1 29112,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CC(O)C2)=O)ccc(=O)n(C)c1 29113,C(=O)(C1=CCCOC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 29114,c1(C(c2nnnn2CCCF)CCOC)cccc(OC)c1Cl.C1C(C)S1 29115,c1(C(=O)OCC(N2CC(c3ccc(C)cc3)(O)C2)=O)cc(C)c(F)cc1N=[N+]=[N-] 29116,c1(C(=O)NCC2(NC(C3(Cl)C(C)(C)C3)=O)CCOC2)ccc(CF)cc1 29117,N1(C(C=CCC)=O)CCN(C(C2CC2c2c(OC)cccc2Cl)=O)CC12CCC2 29118,N1(C(CC=C)=O)CCCCC1CCC(N1CCC(C(C)C)(CO)C1)=O 29119,C#Cc1ccc(C(N2CCN(C(C3CC(N4CCN(C)CC4)C3)=O)CC2)=O)nc1 29120,C(=O)(C(C)CCCOC)NCC12OCC(NC(Cc3cn(CC)nn3)=O)(C1)C2 29121,C1(C(N(CC(C(=O)N(CC#C)CC2CCCO2)(C)C)C)=O)CCC(C)(O)CC1 29122,C12(C(N(CCN(C)C(C34CC(F)C3C4)=O)C)=O)CC(CO)(C1)C2 29123,c1(C(N2CC(OC)C(NC(=O)C(C)(C)CC#N)C2)=O)ccnc2nc(C)nn12 29124,c12cc([nH]n1)CNC2=O.c1(C(N2CCC(CC3CC3)C2)C)sccc1F 29125,CCCC(C(=O)NCc1ccc(F)cc1)NC(C1CN(C(=O)C(C)C)C1)=O 29126,N1(C(c2ccn(COC)n2)=O)CC(N=[N+]=[N-])CN1C(C1CC12CCCC2)=O 29127,c1(CNC(=O)NCCC(OC)OC)ccccc1SC 29128,c1(CN2CC(CC(=O)NC(CCC)c3cccs3)OCC2)cc(Cl)ccc1OC 29129,C1(CNC(CCC(=O)NCC)=O)CN(C(=O)COc2ccccc2Cl)CCN1C 29130,C(=O)(C(CC1CCOC1)NC(=O)Cn1cc(CCCC(C)O)nn1)OC 29131,C(=O)(CCCCC(=O)NC)NCCOC(CNC(C(CCC)NC(C)=O)=O)(C)C 29132,C12(NC(C(C)OCCC(C)C)=O)COC(C1)C(NC(c1cccc(CO)c1)=O)C2 29133,C1(NC(Cc2nc(C(CC)(C)C)on2)=O)CCC(=O)NC1 29134,C1(C(=O)NCCCCN(C)C(C2(C#N)CCCC2)=O)(COC)CC=CCC1 29135,C1(NC(=O)CN2CCCCC2)CN(C(=O)CCc2cnc[nH]2)Cc2nccn2C1 29136,N1(CC(=O)N(C)CC2CCCCN2C(=O)C=CCF)CCCCC(O)C1=O 29137,c1(OC)ncccc1CC(=O)NCC1C2CC1N(C(=O)CN1CCCC1C)C2 29138,N1(C(c2c(OC)nn(C)c2)=O)CCC(O)CC1C(N1C2CCC1CC2)=O 29139,CC1CC(CN2CCN(C(=O)NS(=O)(=O)C(F)(F)F)CC2)C(=O)O1 29140,N1(C(C2CCN(Cc3ccc(C)s3)C2)=O)CC2CCCCC2C1 29141,C(=O)(C(C)(O)C(C)C)NCC(CNC(CCc1ncc(C)[nH]1)=O)O 29142,c1(N2CC(C)C(NC(c3ccon3)=O)CC2)nc(Cl)nc2ccccc12 29143,c1(NCC2CC(=C)C2)nc(N(C)C)c2ncn(CC3(CO)CCC34CCCC4)c2n1 29144,C1(C(=O)NC(CC)C(O)c2ccccc2)CC(O)CN1S(=O)(=O)CC1CC1 29145,C1(C(=O)NCCc2ncc[nH]2)C2CC3C(C2NC(C2C4COCC24)=O)C13 29146,C(=O)(CCCC(=O)NCC(C)NC(=O)C(C)C1CCC1)OCCC(C)C 29147,Cc1cccc(NC2(CNC(=O)COC3CC3)CC2)c1.C12CCCC(C1)C(=O)N2 29148,C(=O)(C1=C(CNCC(CNC(=O)OC(C)(C)C)CO)NC(=O)NC1C)OC 29149,c1(CC=O)cnc2cccnn12.N=c1[nH]c(Cl)cs1.N12CC(C1)OCCC2=O 29150,C1(C(C(=O)NC(C)(C)C)N(C(C)C(=O)NCc2ccccc2)CC)CC2CCC1CC2 29151,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 29152,N1(C(c2c(C)ocn2)=O)C2CCC1CN(C(c1cccc(C(F)F)n1)=O)C2 29153,C1(OCC)CN(C(=O)C=CC2CC2)CC1CNC(C1(c2ccno2)CCC1)=O.COC 29154,c1(NCc2nn(C)c(=O)cc2)ncccc1S(=O)(=O)NCC1CCC(F)(F)CO1 29155,C(=O)(CC1=CCN(C(c2cc(C#N)c[nH]2)=O)CC1)NC(c1cn(C)nn1)C 29156,C(C#Cc1cc(Cl)cnc1F)NC(N1CCC(O)(C(C)C)CC1)=O 29157,C1(NC(C(C)OC2COC2)=O)CCC2CN(C(c3ccnn3C3CC3)=O)CCC2C1 29158,N1(C(c2ncn(C)c2)=O)CC2CCCC1(CNC(c1ccc3cnoc3c1)=O)C2 29159,c1(C(N(C(CCNC(c2c(OC)ccs2)=O)C)C)=O)cc2n(c1)CCSC2 29160,c1(-c2cccc(NC(C3(CC)CC3)=O)c2)cc(OC)cc(C#N)c1 29161,N1(C(Cc2ccc(C)s2)=O)CCOCC(NC(C2CC3CCCCC23)=O)C1 29162,CC1(C)C2CN(CC(c3ccc(OC(F)F)cc3)O)CC12 29163,C#Cc1ccc(NCC2(NC(c3cncc(N4CCCC4)n3)=O)CCCCC2)o1 29164,CCCC(C)CC(=O)NC1COCCN(C(=O)C(C2CCCCC2)O)C1 29165,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)CCc2conc2C)C1 29166,c1(C(N(CCOC)CCNC(C2CSCCS2)=O)=O)cn(CCCF)nn1 29167,N(C1CC(F)(F)c2cc(Br)ccc21)C(=O)C(N1CCC(O)(c2cc[nH]n2)C1)=O 29168,c1(CC(N2CCC(CNc3ncccn3)C2)=O)cccc2c1OCO2 29169,CCCC(C)(CCC)C(=O)NCC(CC(F)(F)F)NC(c1[nH]cnc1C#N)=O 29170,C1(CC)CCN(C(C2CC=CC(O)C2)=O)C1CNC(c1cc(F)c[nH]1)=O 29171,S(=O)(=O)(c1ccc(OC)cc1)N1CCC(CC2CCN(C(=O)NCCC)CC2)CC1 29172,C1(C(=O)NC2(CC(C)C)CC2)CSCN1C(c1ccn(C)n1)=O 29173,c1(CC(=O)N(C2CCN(C(=O)CCc3cnc(C)s3)C2)CCC)ccnn1C 29174,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29175,C1(C(=O)N(Cc2ncc(C(C)C)[nH]2)CC)CCCN(C(=O)CC2CCCCO2)C1 29176,n1(C(C)(C)C)ncc(C(=O)NCCN(C2CCCC2)C(=O)COCP(C)(C)=O)c1Cl 29177,C1(NC(CNC(=O)NC)=O)CCCC(CNC(=O)CCNc2ccc(C)cc2)C1 29178,C1(C(N2CCC(c3cn(-c4ccncc4)nn3)C2)=O)(SC)CC(=O)C1 29179,CC1CN(CC(=O)Nc2ccccc2Cl)CCC1NC(C1CC2OC(=O)OC2C1)=O 29180,c1(C(C)C)ccc(C(=O)NCC2(C)CCCN(C(c3csc(=N)[nH]3)=O)C2)c(O)c1 29181,C1(CC)(NC(=O)COCC(=O)OC)CCCN(C(=O)CCCn2cncn2)C1 29182,N1(C(c2c(CNC(C(C)OCC)=O)n[nH]c2)=O)CCOCC(O)C1 29183,C1(NC(C2CCCO2)=O)CC2CC1CC2C(=O)NC(CC1CCCO1)CO 29184,O=S(=O)(c1cnc(C(F)(F)F)s1)N1CCCC1C1CCC2(CC1)CC2 29185,Cc1c(NC(C2(F)CN(Cc3ccc(Br)s3)C2)=O)cccc1F 29186,c1(CN(C(c2snc(C)n2)C(=O)NC2CCC2)C)ccnc(Cl)c1 29187,N1(C(C(c2ccc(Cl)s2)C)=O)CCCC(CO)(NC(=O)Cc2ccccc2F)C1 29188,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29189,C(CC(C)(C)C)NC(=O)CCc1nc(CC(=O)NC(=O)C=CC(C)C)no1.CS 29190,c1(NC(c2cn(C)nc2C(N2CCCC(C)(O)C2)=O)=O)ccc(Cl)nc1[N+](=O)[O-] 29191,c1(N2CCN(CC(=O)NC)CC2)nccc(=NC(C)c2ccn(C)n2)[nH]1 29192,N1(C(CC2C(OC)COCC2)=O)CCOC2CN(C(c3cc(C)sc3C)=O)CC12 29193,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(-c2ccco2)nn1C 29194,CC1CCN(C(=O)Cn2[nH]cnc2=N)C(C(N2CCCC(CO)(CO)C2)=O)C1 29195,C1(CNC(c2ccc(C(C)C)o2)=O)CCN(C(=O)C(C)(C)CF)CC1C 29196,N1(C(C(C=C)(C)O)=O)CCc2nc(CNC(C3CC(C)CC(C)(C)C3)=O)sc2C1 29197,c1(CC)nn(C)cc1C(=O)NCc1noc(C(N)=O)n1.N1(C=O)CCCC(N)C1 29198,CCCCCC(CN=c1cc(C)[nH]c(=NCc2ncn3ccccc23)[nH]1)N(C)C 29199,C(CN=c1ccc(C(=O)NCC2CCN(C(=O)CC(O)CN(C)C)C2)c[nH]1)OC 29200,N1(C(Cn2c(CC)nnc2)=O)CCN(C(=O)CC2(C#N)CCC2)C(CC(F)F)C1 29201,N1(C(C2CC3(C2)CC3(F)F)=O)CC2CCCC(C1)N2c1ccncc1[N+](=O)[O-] 29202,C(C(CC1CC1)C(=O)Nc1ccc(C(C)C)nc1)NC(CCCNC(C)=O)=O 29203,c1(C(N2CC(CNC(CCCN(C)C)=O)C2)=O)cnc(N)c(N)c1 29204,c1(C(=O)NC2CC(NC(CC(=C)Br)=O)C2)ccnc2c1nnn2C 29205,CC(C)C(C(C)NC(c1ncccc1CO)=O)NC(c1ccc(CO)nc1)=O 29206,C(N=c1cc(NC2(CCOc3ccccc3Cl)CC2)nc[nH]1)C1CC(C)OCC1 29207,N1(C(c2c(C)c(Cl)cnc2)=O)CCCC(C2CN(C(=O)COC3COC3)C2)C1 29208,c1(CS(=O)(=O)N2CC(CCC3=CCCC3)C2)ccc([N+](=O)[O-])cc1 29209,c1(CN2CCC3(C(C(=O)NCc4ccc(F)c(Br)c4)C3)C2)cc(Cl)cc(Cl)c1O 29210,c1(CC(=O)NCC(C)(C)OCC(=O)N(C2(C#C)CC2)CC=C)cccnc1F 29211,C1(CN(C(c2nnnn2C2CC2)CC)C)CCN(C(c2csc(Cl)n2)=O)CC1 29212,C(=O)(CCCCCN(C)C(C1C2CCCC12)=O)N(C(C)C(=O)OC)CC=C 29213,C1(CC)CC(C(=O)NCC(c2ccsc2)O)CCN1C(c1csc(C)n1)=O 29214,N1(C(C2CC(CC(=O)NC(C3C(C)CC3)=O)C2)=O)CCSCC1CCN.N(C)C 29215,N1(C(C(C)=CCC)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29216,N1(C(C(CC=C)CC)=O)CCC2(CC1)CN(C(=O)C=Cc1ccn(C)c1)C2 29217,C1(C(N2CC(OC)CC(NC(CNC(COC)=O)=O)C2)=O)CCCCC(C)(C)C1 29218,Cc1nn(C)c(Cl)c1C(=O)NC1(CNC(c2ncncc2F)=O)CCCCC1C 29219,CC1=C(C(=O)NCc2cc(-c3cccs3)on2)C(C)n2ncnc2N1C 29220,c1(C(C)N(C)CCc2nc(C(F)(F)F)cs2)ccc(F)cc1 29221,c1(C(=O)NC(C2N(C(C(CC=C)C)=O)CCC2)C)ccc(C)c(OC)c1 29222,C1(NC(CC2ON=C(CC)C2)C(N2CC(=O)NC2=O)=O)CC2(C1)CC(C)(C)C2 29223,C(=O)(C1=CCC(C)(C)CC1)NC1C2CN(C(C(C)S(C)(=O)=O)=O)C(CC2)C1 29224,C1(NC(N(CC(O)COCc2ccccc2)C)=O)CC12CCCCCC2 29225,N1(C(CCn2c(SC)nnc2N2CCOCC2)=O)CC2CC1c1ccccc12 29226,C(C(CCC(F)(F)F)NC(c1ncc(Br)cc1Cl)=O)OC 29227,C(=O)(C1=NOC(C)(C)C1)NCC1CN(C(CCC2CCCN(C)C2)=O)CC1O 29228,C(CC(CC)C(=O)NCC1CN(C(=O)CN2CCN(C)CC2)CC1(C)C)=CC 29229,C1(C(=O)NCC(C)CNC(=O)CN2CCCC2)CCCC1CF 29230,C1(C(=O)NC2(CO)CCN(C(CCC#C)=O)C2)CCn2nccc2C1 29231,c1(NC(c2cnn(-c3ccccn3)c2)=O)ncnc2cc(I)sc12.C12CN(C1)C2 29232,C(=O)(C1=CC2(CCOC2)C1)NC(C1CN(C(c2snc(O)c2Cl)=O)C1)C 29233,CC(C)C(C(F)F)NC(=O)NCC1CCC(=O)O1 29234,c1(CNC(C(C(CC)C)C)=O)c(C)nn2c1CN(C(c1ccncc1N)=O)CC2 29235,N1(C(CC=CCC)=O)CCOC(CNC(c2sc(-c3ncccn3)nc2C)=O)C1 29236,C(=O)(C1=C(C#N)CCC1)N(C1CCCC(NC(=O)C=CC2CC2)C1)C 29237,CCC(CC)(C(=O)NC(C1CN(C(c2n[nH]cc2C)=O)CC1C)c1nnn(C)n1)OC 29238,C12(NC(CNC(=O)CC(O)CNC(=O)C3CC3)=O)CCCC1CCC2 29239,CC1CN(C(=O)CCCCN(C(=O)CC2COCC(C)O2)C)CC(C)N1 29240,C(=O)(CN=c1cc[nH]cc1)N1CCC(CC=C)(C(=O)NC2CCCCC23CC3)C1 29241,C(=O)(CCC(C)(C)C)N1CC(C(CC)C(=O)NCC)C(C)C1 29242,C1(C(N2CC(O)(CCNC(C(C=CC)O)=O)C2)=O)COc2ccccc2O1 29243,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29244,Cc1nc(C)c(C(=O)NC(C2CCN(C(=O)Cn3nnnc3C)C2)(C)C)[nH]1 29245,c1(NC(C2(C)CCCN2Cc2cccc3c2OCC3)=O)cc(F)ccc1C#N 29246,c1(CN)cn2c(F)cccc2n1.C1(COCC)CCCCN(C(=O)C(=O)N)C1 29247,C1(NC(C2CCC(F)(F)C2)=O)CC2CC1CN(C(C1CCN(C3CC3)CC1)=O)C2 29248,C1(C(=O)NC2C(SC)CCC2)Cc2nn(C)cc2C(=O)N1 29249,C12(CNC(c3cc(CC)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29250,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29251,C1(CC)CCN(C(c2ccc(OC)nc2)=O)C1CNC(=O)CCCOC1CC1 29252,c1(NC(=O)NC(c2onc(C)n2)Cc2cccc(Br)c2)cc(F)ccc1O 29253,C1(F)(CNC(C2CCN(C(C)=O)C2)=O)CCCN(C(=O)Cn2c(O)nnc2O)C1 29254,N1(C(c2nn(CC(F)(F)F)cc2I)=O)CCN2C(=O)CCC2C1 29255,C(=O)(CC(CNC(C1CSC1)=O)OC)NCCCCC 29256,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29257,C#CC1(O)CCN(C(=O)C(CC(=C)C)NC(c2ccccc2C#N)=O)C1 29258,N1(c2nnc(-c3ccc(C)s3)n2CC2(CO)CC2)CCc2nc(Cl)ccc2C1 29259,c1(CC(=O)NCC=CCNC(C(CCC)C(C)C)=O)coc2cc(OC)ccc12 29260,c12occc1C(=O)NCC(C)NC2=O.C(C=O)N(CC)CC 29261,CN1C(=O)CCC1CC(N1CCCCC1CNC(c1csc(Cl)n1)=O)=O 29262,c1(NC(CC2CCN(Cc3nccc(OCC)c3)C2)=O)cc(Br)c(Cl)cc1F 29263,O=C(C1=NN2CCCN=C2N1)NC1CN(C(=O)Cc2ccc(O)cc2)C1 29264,C1(C)(C(=O)OC(C)C)CCN(C(C(=O)NCC2CCC2)c2cn[nH]c2)C1 29265,c1(C(N2C(CN(C)C(C3(O)COC3)=O)CCC2)=O)ccc(S(C)=O)cc1 29266,C1(NC(NCc2n(C)ncc2)=NCCN2CCCC2)CCN(CCS)CC1(F)F.C 29267,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29268,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)CCc1ccn(C)c1 29269,CC(C)CCC(=O)NC(CO)C(=O)NCCCC1CCOC1=O 29270,c1(C(=O)NC(c2cccc(F)c2)C(CC)SC)cc(Br)c(CO)cc1OC 29271,N1(C(CCc2scc(C)c2)=O)CCC(C)C(CNC(=O)Cc2csnn2)C1 29272,C1(C(=O)OC)CCC2CC2C1NC(=O)NC(c1ccccc1C)CO 29273,c1(NC(=O)OC(C)(C)C)c(Br)c(C(=O)NC2C(C(=O)OC)CCC2)cn1C 29274,c1(C(=O)NC2C(CNC(C(C)(C)c3cccs3)=O)CCC2)cc2n(c1)CCSC2 29275,N1(CC23CCC(C)(C2)CO3)C(=O)CCN(CC2CCCc3nc[nH]c32)C1=O 29276,O=S(=O)(c1cc(Br)c(F)cc1F)NCC1CC2(C1)CN(CC1CC1)C2 29277,C(=O)(C(C)CCCC(C)C)N1CC2(C1)C(=O)N2.C(=O)(C=NOC)N.CSC 29278,CONC(=O)C(=O)NC1CN(C(=O)COCP(C)(C)=O)CC1SC 29279,C(=O)(C(C)(C)CCCNC(=O)CS(=O)CC)N1CCC(C(=O)OC)C1 29280,C1(O)(C(=O)Nc2cccc(OC)c2)CCN(CC)C1.n12nnnc1C2 29281,Cc1coc(C)c1C=CC(N1CC(C)(NC(C2CN(C)C(=O)N2)=O)C1)=O 29282,CCC(CC(=O)N1CCOCC1CNC(=O)C=Cc1nccn1C)C(F)F 29283,CC(C)(C)C(CO)C(=O)C=C1CCCCC1.C1(N2CC(=O)O2)CCCCC1 29284,C1(CCC)(NC(=O)CC2(OC)CN(C(=O)C(CC)SCC)C2)CCNC1=O 29285,C(CC(=O)NCC1CC12CCOCC2)(CC(C)C)NC(CN(C(=O)OC)C)=O 29286,N1(C(CSCCC)=O)CCCC(CC(=O)NCC2C=CCCC2)C1 29287,Cc1cc(C(=O)N(C)C)c[nH]c1=NCc1ccc2c[nH]nc2c1 29288,C1(NC(c2c(NC)scn2)=O)(COC)CCN(C(=O)CCc2cscn2)C1 29289,c1(C(C)=O)ccc(C(C(=O)Nc2ccccc2)N(CCCCC(C)C(=O)O)C)cc1 29290,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29291,C(CCC1CC1)(C(=O)NC1CC2C=CC1C2)NC(C(C1CCCC1)OCC)=O 29292,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29293,C(=O)(C1(C)CCc2ccccc21)N1CC(CC(C)NC(c2c(C)sc(Cl)n2)=O)C1 29294,C(C)(C(C)(C)C(=O)NCc1nc(C(C)C)no1)NC(C(n1ncc(C)c1)C)=O 29295,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(C2CCC(=O)N2C)=O)c(C)c1 29296,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1C 29297,C1(NC(C(C2CCN(C(c3ccc(C)nc3C)=O)C2)C)=O)CCc2cscc2C1 29298,C1(C(=O)NCCC(=O)NC(C)C(C)NC(=O)CO)CCc2nnc(O)cc2C1 29299,Cc1nc(C(C)(C)C)nc(C)c1C(=O)NCC(C)(C)NC(C1CCS(=O)(=O)C1)=O 29300,C(=O)(C(O)Cc1cnn(C)c1)NC(C)CN(C(=O)C(N1CCSCC1)C)C1CC1 29301,C12CCCCN(C1)C2=O.c1(N(C)C)ccc(CNC(C2C=CCC2)=O)cc1 29302,c1(C(=O)NC2(CNC(CCc3cc(C)no3)=O)CC2)cccc2c(C)cccc12 29303,N1(C(c2n(C(C)C)cnc2)=O)CC(Nc2ccnn2CCCO)C2(CC2)C1 29304,c1(CN(OC)C(=O)N(CC(C)Oc2ccccc2)C)ccc([N+](=O)[O-])cc1 29305,N1(C(c2cc(C(C)=O)oc2)=O)CCC2CN(C(=O)CC3CC3(C)C)CC12 29306,c1(C(COC)NC(c2nnsc2C)=O)ccc(Cl)cc1 29307,c1(OC)c(F)ccc(C(N2CC(NC(c3ccc(Cl)o3)=O)CC2C)=O)c1F 29308,CC(CCCNC(c1ncoc1C1CCC1)=O)NC(=O)C(N1CCOCC1)C 29309,c1(C(=O)OC)nc(C(=O)NCC(CC)NC(=O)C(C)CN2CCCCC2)c(C)s1 29310,O(NC(=O)C(CNC(=O)C(CN(C)C)c1ccon1)C(C)(C)C)CC(C(C)(C)C)O 29311,C1(CC(C)C)CC1N=c1[nH]c(N2CCN3CCCC3C2)nc(=NCCCC#N)[nH]1 29312,NS(=O)(=O)C1CC(C(=O)NCc2cccc(CNC(C3CC3CF)=O)c2)C1 29313,c1(CC(N2CC(N(C(CCOCCC)=O)CCC)C2)=O)csnc1C 29314,C#CCC(C(=O)NCCOC)NC(=O)NCCC.C12(CC1)C(=O)N2 29315,N1(C(C=CC)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1C(C)(C)C 29316,c1(C(=O)NC(C)CN(C(=O)CCOC2CCCC2)C)c[nH]c2cccc(F)c12 29317,c1(OCc2ncc(-c3ccc(OC)cc3)[nH]2)c(Cl)cc(Br)cc1Cl 29318,c1(NC(c2c(N=[N+]=[N-])cccc2)Cc2ccc(Cl)c(F)c2)cc2ccccc2o1 29319,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)CC1CNC(C1CNC(=O)O1)=O 29320,C(CC(C=O)NC(C1OCCC1CNC(=O)CSC1CC1)=O)OCC 29321,c1(NC(C2C(C)CC=C2)=O)cccc(NC(=O)C(=O)NC(C)(C)C)c1 29322,N1(C(c2ccc(OC)cn2)=O)CC(C)(C(=O)NCC(C)C(C)(C)C)CC1(C)C 29323,C1(CC(N2CC(O)(COC)C2)=O)CCCC12CC2.C1(=O)NCCN1 29324,C(C(N=c1cc(C)nc(NC2CC3(C2)CC(O)C3)[nH]1)C1CCCCC1)SC 29325,c1(NC(=O)CCC2CC2)ccc(C(=O)NCc2ccc(Br)cc2)cc1 29326,Cc1nc(Br)sc1C(=O)NC1CCC(N(C)C(c2ccc(O)nc2)=O)CC1 29327,N1(C(C=C(C)CNC(C2CCC(C)(C)C2)=O)=O)CCC2CCN(C)C2C1 29328,C1(C(N2CC(CCO)(NC(CC=CC=C)=O)C2)=O)CCCC2(CCC2)O1 29329,C(=O)(CC(C)(C)CC(=O)NCC1CC1CNC(C1CC2(CCC2)C1)=O)OC 29330,C(CC(C)C)(C(=O)NCC(CNC(=O)CCc1cnoc1)CO)OC 29331,CN=c1nc(C(=O)NC2(CNC(=O)CC(O)CC(C)C)CCC2)cc(C)[nH]1 29332,C1(C(=O)NC(C2CN(C(c3nccs3)=O)C2)C)CC2CCC1O2 29333,C=CCCC(C(=O)N(C)Cc1cn(C)nc1C)NC(=O)CC1CCOC1(C)C 29334,c1(C(C)C)ccc(C(N2CCC(C)(NC(=O)COc3cncnc3Cl)C2)=O)nc1 29335,C1(CC)CC(CNC(=O)C(c2ccc(F)cc2)O)N(C(C2CC(C)=NO2)=O)C1 29336,C(N=c1[nH]c(=NCC2CC3(CCC3)CO2)c2[nH]ccc2[nH]1)c1nn(C)c(=O)cc1 29337,c1(C(N2CCC(C(F)(F)F)C(CC3CC3)C2)=O)cc2ccsc2s1 29338,c1(CC)ccc(C(=O)NC2COCC2NC(=O)CCc2nnc(O)nc2O)cc1N 29339,N1(C(=O)Cc2sccc2Br)CC2CCC(C1)C2NCc1cc(Cl)ccc1Cl 29340,N1(C(C2(SC)CC2)=O)CCC2CCCC12C(=O)NCC1CCC1 29341,c1(C(C2CCCO2)N(C(C(n2cc(CC(C)(C)C)nn2)C)=O)C)cccnc1 29342,c1(C(N2CCC(N(C(CS(CC)=O)=O)CCO)C2)=O)cc(Cl)n[nH]c1=N 29343,N1(C(=O)NC(C2(C)CN(C(C)=O)CCO2)CC)CCOc2cccc(OCC)c2C1 29344,C1(O)(C(C(=O)N(CCCO)CCO)NC(c2ccc(CO)cc2)=O)CCCCC1 29345,N1(C(C2OCCN(C)C2=O)=O)CC(NC(=O)Cc2cnns2)CC2(CC2)C1 29346,C1(CNC(C2CCN(c3ccccc3Cl)C2)=O)COCCN1C(c1cnns1)=O 29347,C(C(COC)C(=O)NC(Cc1ccco1)C(=O)N(C)C(C1CCCO1)C)OC 29348,C(C)(CO)(C(=O)N1CC(C)(C)C1c1cn(CC(=O)OC)nn1)OCC 29349,N1(C(CCOC)=O)CCc2sccc2C1CNC(c1ccc2oc(O)nc2n1)=O 29350,c1(C(=O)OC)cc(C)c(F)c(S(=O)(=O)NCCNc2c(C)nc(C)nc2C)c1 29351,C1(NC(c2n(C)cnc2)=O)CCCCC1CNC(C1CCCCC1C(F)(F)F)=O 29352,c1(CC(=O)NCC(CC)NC(=O)CN(CC)CC2CC2)csc(Cl)n1 29353,N1(C(C(CC)(C)C)=O)CC2(CCN(C(C3CCCO3)=O)CC2)c2ccccc21 29354,C(=O)(CC(C)CC1CCCCC1)N1CC(OCC)C1 29355,Cc1ncc(F)c(=NCC2CN(C(=O)CC3CCC(C)C3)C2)[nH]1 29356,N(C(=NCC(C)OC)NC1CCC1)CC(CC)Oc1ccccc1F 29357,C1(NC(=O)NC(C2CC(C#N)C2)C)CCC(c2nn[nH]n2)CC1 29358,c1(CC(N2CCC(CNC(CC(C)C)=O)CC2)=O)ccc(C#N)nc1 29359,C=CCN=C(NCc1nnn(C)n1)NC1C(C)C1C 29360,Cc1ccccc1CC(C)C(=O)NC1(C)CN(C(c2cn(C(C)(C)C)nn2)=O)C1 29361,C1(CNC(C2(N(C)C)CC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29362,C(c1ccc(C)nc1)=CC(=O)NCC1(C)CCN(C(c2c(OC)ccs2)=O)C1 29363,c1(C(N(CCNC(C(c2cccs2)SC)=O)CC2CC2)=O)c(C)nc(O)nc1O 29364,C1(C(=O)NOCCCO)COCCC1NC(C1CSCCN1)=O 29365,N1(C(c2c(C)cncc2C)=O)CC2CC(NC(C3CCCCS3)=O)CC1C2 29366,c1(CNCC2CCC(C(=O)NCCSC)C2)c[nH]c2cnccc12 29367,S(=O)(=O)(c1ccc(NC2CCS(=O)(=O)C2C)c(Br)c1)NCCCOCC(C)C 29368,N1(Cc2cn(CC)nc2)CCC(NC(c2ccccc2C(F)(F)F)=O)C1C1CC1 29369,C1(C(C(=O)NC2(CC=C)CC(O)C2)O)CCN(C(=O)OC(C)(C)C)CC1 29370,Cc1cnc(N2CCSCC2C)c(S(=O)(=O)N2CCCC2c2ccccc2C)c1 29371,C1(C)(COC)CCCN(C(=O)C(O)C2CN(C(=O)Cc3ccccc3C)C2)C1 29372,C(=O)(C1=CCC(NC(c2ccc(CF)cc2)=O)C1)N(C(C)C(C)(C)O)C 29373,C12(CCN(CC)C1C(C)(C)C)CCOC2=O.C(C)(C)(C)OC(=O)O.C(=O)O 29374,C1(CC(=O)NC(C2CCCC2)CNC(CC2CN(C(=O)NC)C2)=O)CC(F)(F)C1 29375,C(=O)(CCS(N)(=O)=O)N1CC(C(C)NC(C2(CC)CC2)=O)C1 29376,N1(C(C(CC=C)(F)F)=O)CCC2(CCCN2C(c2cccc(OCCF)c2)=O)C1 29377,CCCCC(C)C(=O)NC1(CNC(c2ccc(NS(=O)(=O)CC)cc2)=O)CCC1 29378,c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NC1CCN(C(C2CCCC2)=O)C1 29379,C1(CC=C)(C(=O)NC(C)C(C)C(=O)OC)CCCN1C(C1CC1Cl)=O 29380,C1(C(N(CC(CN(C(C2CC(C)C2)=O)C)O)C)=O)CC(c2cnn(C)c2)=NO1 29381,C1(C(=O)NC2CC(NC(=O)C(N3CCCCC3)C)C2)(COCC)CC=CC1 29382,C1(CNC(=O)CO)CC(O)CN1C(C1(c2ccc(C(F)(F)F)cc2)CC1)=O 29383,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C(C)NC(=O)CC(C)(C)C)=O)C1C 29384,N1(C(C2CC(NC(Cc3c(C)noc3)=O)C(O)C2)=O)CCSC2CCCCC12 29385,C=C1CC2(C1)CC(C(=O)NCC(CC)NC(=O)C=Cc1cncc(O)c1)C2 29386,C(=O)(CCCC1CCCO1)N(C(c1ccccc1)CNC(CC1CN(C)C1)=O)C 29387,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC(O)C1 29388,N1(C(CS(=O)(=O)NC)=O)CCC2(CCC2)C(NC(c2csc3c2CCCC3)=O)C1 29389,N1(C(COC)=O)CC2CCC2(CCNC(c2nc(Cl)sc2C2CC2)=O)C1 29390,CC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)c1ccns1)C)P(C)(C)=O 29391,N1(C(c2c(C)ocn2)=O)CCC2(CCC2)C(CNC(c2ccc(N)c(N)n2)=O)C1 29392,O=S(=O)(c1ccc2c(c1)CCC2)NCC1CC(O)C12CCC2 29393,CCC(C)C(C(=O)N(CCC(C(C)C)NC(c1cnnn1C(C)C)=O)C)OC 29394,N1(c2ccnc(C(CC)C)n2)CCCCC(CNC(C2(C)CC2(F)Cl)=O)C1 29395,c1(C(N(CCNC(C2CCS(=O)(=O)N2)=O)CC)=O)cnn(C)c1C#N 29396,N1(C(C2OCCN(C)C2)=O)CCCC(O)(CNC(c2cn(CCO)nn2)=O)CC1 29397,Cc1noc(CCC(=O)NCC2CCN(C(=O)CCc3nc(C4CC4)no3)C2)n1 29398,C(=O)(C(CNC(=O)C=Cc1ccncc1)(CC)CC)NCCC(CC)(C)O 29399,C1(C(=O)NC2C(NC(=O)CSCC3CCCCO3)C2)CCS(=O)(=O)N1 29400,CC1(NC(C2CN(C(C3CCCSC3)=O)C2)=O)CC(F)(F)C1 29401,c1(C(=O)NC2CCN(C(c3cc(C(C)=O)oc3)=O)C2)cnn(C)c1C 29402,c1(C(N(CC(C)N(C(c2c(CCC)nco2)=O)C)C2CCC2)=O)ccc(OC)cc1 29403,c1(C(=O)NC2C(C)(C)C2C(=O)NCc2ccnc(CO)c2)cnn2c1CCC2 29404,c1(C(N(CCn2cc(C3CCN(C)C3)nn2)C2CC2)=O)cccc(C2CC2)c1Cl 29405,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3CC3C)=O)C2)=O)cc1 29406,C12=C(C)NNC1=NC(=O)c1ccc(o1)C(C)NC2=O.C(C)(C)(C)OCC#C 29407,Cc1ccn2c(C(N3CC4(C3)CN(C(c3n[nH]cc3F)=O)CC4CO)=O)cnc2c1 29408,C12(NC(C=Cc3ncc(C)[nH]3)=O)CCOCC1CN(C(c1nccnc1C)=O)C2 29409,c1(N(CC(=C)Br)C)nc(NC(c2ccnc(OC)c2)C)c2ccsc2n1 29410,[SH](=O)(=O)CC(C)C1CC1.CC(C)(C)NC(=O)NCC(C1CC1)NC(=O)NCCO 29411,c1(C(N2C3(C(N4CCN(CC)CC4)=O)CC3CC2)=O)cc(C)n(C)c1C 29412,C1(C)(CNC(Cc2n(C)nnc2)=O)COCCN(C(C2CCC3CCC2O3)=O)C1 29413,N1(C(CC(CNC(CC)=O)NC(=O)C(C)C)=O)CCC(O)C(C)(C)C1 29414,Cc1cccc(C)c1OCC(=O)NCC1CC(NC(C2(C)CC3CCC2C3)=O)C1 29415,C12(NC(CC3C(C)(C)N(C(C4CC5CCC4CC5)=O)CC3)=O)CCC(CC1)OC2 29416,CC1(OCC(=O)NCC2(C)CC(F)C2)CN(C(=O)C=CC2CCOC2)C1 29417,C1(NC(=O)CC2CCS(=O)(=O)CC2)CN(C(=O)C(F)=C2CCC2)CC12CCC2 29418,C12(COC)CN(C1)C(=O)c1cc2n[nH]1.C1(NC(=O)OC(C)(C)C)CCCC1SC 29419,CC1CCCCC1(C)C(=O)N1CCC(C(=O)NCCSC2CC(C)(C)OC2=O)O1 29420,N1(C(C(C)(C)C2CC2)=O)CC2CCC1CN(C(=O)CCOc1ccc(O)cc1)C2 29421,c1(C(N2CC(NC(c3c[nH]c(=N)s3)=O)C(CO)CC2)=O)cccn2nnnc12 29422,C(CCCCN=c1[nH]c(Br)cc2ccccc12)C1N(C(C=C(C)c2ccco2)=O)CC1 29423,C12(OC)CC(C1)C(=O)O2.C1(C(=O)OC)(C(=O)OC(C)(C)C)CC1C 29424,N1(C(c2occ(C(N)=O)c2)=O)CCC2(CCCCC2NC(=O)CNC=O)CC1 29425,Cc1c[nH]c(CC(N)=O)c1C(=O)NC(=O)CCC1CCC(O)CC1 29426,N1(C=O)CCC2(CC1)CCN(C(c1cccc(C)c1)=O)CC2.Cc1cc(N)cc(C)c1 29427,c1(C2(CC(C)C)CC2)ccc(N)c(O)c1.C1(CC(=O)N)CC(C)N(C(=O)C2CC2)C1 29428,C1(C(N2C(C(=O)NCCC3CCCCC3)C=CCC2)=O)CC2CCC(C1)C2 29429,c1(OC)cccc(CC(=O)NC2CC(CO)N(C(c3cnc(C4CC4)s3)=O)C2)n1 29430,C(=O)(C(C)(C(F)(F)F)N1CCOCC1)NC(c1ccc(C)cc1)CO 29431,C1(c2cn(C(CC)C)nn2)CCCN(C(c2cc(I)cn2C)=O)C1 29432,N1(C(c2c(CCC)nns2)=O)CC2CC1CC2NC(=O)C#CC1CC1 29433,C1(c2scc(C)n2)CCCN(C(C(C)(CN(C)C)C2CC2)=O)C1 29434,Cn1cnc2cccc(C(=O)NC34CC3CN(C(C3CCC(O)C3)=O)C4)c12 29435,C#CCCC(=O)NC(C)C(CO)NC(=O)C(C)=C1CN(C(=O)OC(C)(C)C)C1 29436,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29437,Cc1nn(CC(N2CC3CCC3(NC(=O)CCCOC(C)C)C2)=O)c(C)c1Br 29438,CC(N=c1ccnc(N2CCNC(=O)CC2)[nH]1)C1(C2CCCO2)CC1 29439,C(=O)(CCCCN1CCCCC1)NCC1(NC(C2C(COCC)C2)=O)CCC1 29440,CCCC(C(=O)N=c1ccn(C(C)C)[nH]1)NC(=O)CCCN(C)C 29441,C1(C(=O)NC2CC(CCNC(c3c(C#C)cnn3C)=O)C2)CC2(COCCO2)C1 29442,CC(C)C(CO)C(=O)NCCC1CCCCN1C(=O)CC1CCC(C)(C)C1 29443,C(=O)(C1=CCC(C(F)(F)F)OC1)C(C(C)OC1CCCCC1)=O.C1(N)CC(C)C1 29444,CC1CC(CCNC(c2cc[nH]c2)=O)CCN1C(c1ccc(C(N)=O)[nH]1)=O 29445,C(C(C)CC(=O)N1CC(CC(=O)NOC(C)(C)C)C(C)C1)OC 29446,C1(NC(CC=C)=O)(CC)CCN(C(c2cccc(C(C)(F)F)n2)=O)CC1 29447,c1ccc2c(c1F)CCC2.C1(CS(N)(=O)=O)CCCC1C(=O)NCC=CCNC=O 29448,c1(OC(C)C)ccc(NC(=S)Nc2ccn(C)c(=O)c2)cc1F 29449,C1(C(=O)NC2(CN(C)C(c3nccn3C)=O)CC2)C2CCC1(c1ccccc1)C2 29450,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29451,C1(C(=O)NCCCCCCCC)CCN(C(=O)C(C2CC2)OCC)CC1(C)C 29452,N1(C(C(CC=C)NC(=O)C(C)CC(C)C)=O)CC2(C1)CC(C)(C)C2 29453,N1(C(C(C)CN(C)C(C2CCCOCC2)=O)=O)CCc2sccc2C1 29454,N12CCC(C(C)C1)NC2=O.Cc1cccc(CN2CCCC(CN)C2)c1 29455,N1(C(C(C(C)(C)C)SC)=O)CCC2(CC1)CCN(C(C13CC(C1)C(C)O3)=O)C2 29456,c1(CC(CO)NC(=O)Cn2cc(-c3ncccn3)nn2)cccc(C(F)(F)F)c1 29457,C(C(CC(C)C)NC(=O)C(C)NC(c1ccoc1)=O)NC(C1(CC)CC1(F)F)=O 29458,c1(N(C23CC(CO)(C2)C3)C)ccc2c(n1)CCCC2=O 29459,Cc1sc(O)nc1C(=O)NC(C)C(C)NC(=O)C(C)(C)CN1CCOCC1 29460,N1(C(C(c2ccccc2)C)=O)CCC(CNC(=O)Cc2cccnc2Cl)C1(C)C 29461,CC(CC(C)(C)C)C(=O)NC1CC(NC(C2(CF)CCC2)=O)C12CCC2 29462,N1(C(CC2N(CC)CCC2)=O)CCC(C(C)CNC(C2(C)CCCCC2)=O)CC1 29463,C(C)(C)(CC(=O)N1CCCCC1C(C)NC(=O)Cc1cccs1)SC 29464,ONC(=O)C(CO)N(C)C.c1(CC(=O)NC(c2noc(C)n2)CC)ccn(CC)n1 29465,c1(C(N2CCN(c3ncc(Cl)cn3)CC2)C(=O)NC)cccc(P(C)(C)=O)c1 29466,Cc1ccc(O)cc1C(=O)NCCC(C)NC(c1cncn1C)=O 29467,C1(N(C(=O)COc2ccsc2)CC)CN2CCN1CC2C.N12CCN(CC1)C2=O 29468,Cc1cccc(OCCCC(=O)NCCCCCNC(c2cc(C)[nH]n2)=O)c1 29469,C(CC(N)=O)(C(=O)NC1(C2CC2)CC1)NC(CSC(C)(C)C)=O 29470,c1(CNC(CC(C)F)=O)cccc(CNC(c2cccc(O)n2)=O)c1 29471,n1(CC)nnc(C(=O)NCCCCC(C)NC(=O)Cn2c(C)ccc2C)c1C 29472,C12(C(N3C(CNC(C=CC(CC)=CC)=O)CC3)=O)CCOC1CCOC2 29473,c1(CC)cc(C(=O)NCCC2CCCN(C(=O)C(F)OC(F)(F)F)C2)oc1CC 29474,c1(C(N2CCCC(NC(CN3CCCC(C)C3)=O)CC2)=O)cnc2[nH]ncc2c1 29475,CCCC(CCO)CN=c1ncc(-c2nccn2Cc2ccccc2)c[nH]1 29476,C1(CNC(=O)CC(C2CC2)C2CC2)CC2(CCC2)CN1c1nc2ccccc2o1 29477,c1(OCC)cncc(C(=O)N(CC(C)N(C)C(c2oc(C3CC3)nc2C)=O)C)n1 29478,CC1CCc2nnc(C(=O)NCC(C)CN(C(=O)C(F)=CCCF)C)cc2C1 29479,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29480,N1(C(C2CC(C(C)=O)C2(C)C)=O)CC2CCC(C(=O)NCC3CC3)(C2)C1 29481,C1(NC(c2cc(C)no2)=O)CC12CCN(C(=O)Cc1nc(=N)[nH][nH]1)C2 29482,S(=O)(=O)(c1cc(Cl)ccc1Cl)NC1CCCCCN(C(C(=O)NCCCl)=O)C1 29483,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29484,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29485,C1(C(=O)NC2CCC(NC(C3CCC(CC)O3)=O)C2)C2CCC3C(C2)CC13 29486,C(C)(C)(CC(=O)N1CCC(CN(C(=O)C(F)C2CCOC2)C)C1)OC 29487,C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C(C(C)C)n1cc(C)nc1)=O 29488,c1(C(=O)NCC2CCCC2NC(C2CCCC2)=O)cncc(Cl)c1Cl 29489,N1(C(CS(C)(=N)=O)=O)CC2C3CCC(C2C1)N(C(c1cscc1C(F)F)=O)C3 29490,c1(OCCC)cccc(CC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29491,N1(C(=O)NC2C(C(=O)OC)CCCN2)CCCC(C(=O)O)C1C 29492,C(=O)(C1CCCn2nccc21)N1CCC(SCc2n(C(C)C)cnc2)CC1 29493,Cc1cc2c[nH]nc2c(C(=O)NCC2(CNC(=O)CC3CC(=O)NC3=O)CC2)c1 29494,N1(C(c2cnn(CC)c2C)=O)CCC(CNC(c2cccc(Cl)c2O)=O)C12CC2 29495,n1(CC(=O)NC2CC(C(N(C(C)(CO)C3CC3)C)=O)C2)cnc(C#N)n1 29496,c1(C(N2CC(CCNC(c3cc(C)c(N)cn3)=O)C2)=O)ccc2c(n1)OCCO2 29497,C(CC(Cc1ccccc1)NC(C1(Br)CC1)=O)NC(c1cnns1)=O 29498,c1(C(N(CC(CNC(CSCC=C)=O)(C)C)C)=O)cccc2nc(O)oc12 29499,C1(CNC(=O)COC2CCC2)CN(C(=O)CC2CCCOC2)CC2(CC2)C1 29500,C1(C(=O)NCC(C)(C)O)CC2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 29501,C(=O)(C(F)OC)N(CCC)CCNC(=O)C(C1CCC1)C1CCC1 29502,c1(OC)cccc2c(N)cccc12.N12CCCN(CC1)C(=O)c1noc(n1)CC2=O 29503,C(c1ccc2ccccc2n1)=CC(=O)N(C)CC1CCN(C(C(C)O)=O)C1 29504,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3C)CO2)C1 29505,c1(C(N)=O)cc(C(=O)NC2CCCC2NC(C2C3CCN2CC3)=O)ccn1 29506,Cc1nnc2cnc(C(=O)NC3CC(CNC(c4ccc(Cl)c(Cl)c4)=O)C3)cn12 29507,c1(C(c2cnn(C)c2-c2cn(CCCO)nn2)C)ccc(I)cc1 29508,C1(C(N2CC(F)(C(=O)NC(c3c(C)nns3)C)C2)=O)CCC(C)CC1 29509,c1(CC)conc1CC(=O)N(C(C)CC(=O)NC1COCC1CN(C)C)C 29510,C(=O)(C(CC1CC1)NC(c1cc(F)c[nH]1)=O)NC(C)COCC1CC1 29511,n1(CCC)cc(C(=O)NC(C2CCCCN2C(=O)CN2CCCCC2)C)c(C)n1 29512,C1(NC(=O)OC(C)(C)C)CN(C(=O)OC2CC3CCCC3C2)C2CCCC12 29513,C(=O)(CCCCC(N)=O)N1C(C)CC(CCNC(=O)COCP(C)(C)=O)CC1 29514,c1(CNC(C(C)C#N)=O)cccc(CNC(=O)CC(c2ccccc2)N(C)C)c1 29515,C1(C2CC2)(NC(N(C)CC2CN(c3ccccc3)CCO2)=O)CCCCCC1 29516,CC1(C)CN(C(=O)Cc2ccsc2)CC1NC(c1ccccc1C(=O)N(C)C)=O 29517,Clc1ccccc1C1CCC1OCCN1CCN(c2nccnn2)CC1 29518,C(=O)(CCN=[N+]=[N-])N(CCCN(C)C(C1(N(C)C)CCCC1)=O)C 29519,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(N)=O)CC1CO 29520,C1(CNC(CCC(C)O)=O)CCN(C(=O)Cc2ccc3c[nH]nc3c2)CC1(F)F 29521,c1(C(N2CC(CCNC(C3C(CCC)CCC3)=O)(OCC)C2)=O)ncccc1N 29522,N1(C(C(CNC(=O)Cn2cc(Cl)cn2)N(C)C)=O)CC2CC=CCC2C1 29523,CC(CCc1ccccc1F)C(=O)NCC(O)CNC(=O)CCC1CCCOC1 29524,C(=O)(C#CC1CCCCC1)N1CC(C(C(=O)NCC(CCC)CCO)OC)C1 29525,CCC(CCC(=O)NOCC1CCC1)NC(=O)Cn1ccc(C)n1 29526,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29527,S(=O)(=O)(c1ccc(Br)cc1CSC)NCCN(C(C(CC)O)=O)C1CC1 29528,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29529,c1(OC)ccc(CC(=O)NN(C)CC2(CNC(=O)Cc3nncn3C)CC2)o1 29530,C1(n2ncc(NC(c3cc(C)c(C(F)(F)F)cc3)=O)c2)COc2ccccc2O1 29531,c1(N(CC(=O)NC(C)C)C)nc(N2CCC(C(F)F)C2)nc2c(F)cccc12 29532,C1(NC(c2nn(CCC)c(C)c2)=O)CCN(C(=O)CCOC2CCC2)C(C)C1 29533,C=CCC(C(=O)NC1CCCN(C(c2snnc2CC)=O)C1)OC 29534,C(=O)(C(C)(C)C(F)F)N(CCN(C(C(C)OCCC=C)=O)C)CCn1cncn1 29535,CCC(C)(CNC(C1CCCCC1)=O)NC(C1(N(C)C)CC1)=O 29536,c1(C(=O)NC2CC(NC(C(=O)NCCOCCCC)=O)C2(C)C)ccc(O)c(C)c1 29537,c1(SCC(=O)NC(C)CCNC(C23CC(C)C(C2)C3)=O)cccc(F)c1 29538,c1(C(N2CC(CC=C)(NC(C3CC3COC)=O)C2)=O)ccc(S(=O)(=O)CC)cc1 29539,C1(COC)CN(C(c2ccc[nH]2)=O)CCN1C(=O)CCc1ccc(O)c(F)c1 29540,N1(C(C2(O)CCCC2)=O)CC2CC(NC(C3CC(n4cnnc4)C3)=O)CC(C2)C1 29541,c1(-n2cc(CN3CCC(Cc4c(Cl)c[nH]n4)CC3)nn2)cccc2c1OCO2 29542,c1(OC)ccc(OC)cc1-c1ccc(C(=O)NC2C=CS(=O)(=O)C2)s1 29543,c1(C(=O)NCCOCCOCCCNC(c2c(C)cns2)=O)sc(C)nc1Cl 29544,Cc1cc2ccc(C(N3CCC(NC(c4[nH]c(O)nc4C)=O)CC3C)=O)cn2c1 29545,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29546,C1(C(N2CC(C(=O)NC(C3CCCOC3)(C)C)C(C(C)C)C2)=O)C2CCC(F)(F)C12 29547,C(=O)(C(F)CC1CCOC1)N(CCOC)CCNC(=O)Cn1nnc(C)n1 29548,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2[nH]cncc1-2 29549,C1(CC(=O)NCCOCCNC(=O)Cn2cccc2)CC(=O)N(c2cn[nH]c2)C1 29550,c1(C(N2C(C(=O)NC3CC(C(N)=O)C3)(CC)CCC2)=O)ncc(C)cc1C 29551,c1(OC)cc(NC(=O)C(N2CCOC3(CCC3OC)C2)=O)cc(S(C)(=O)=O)c1 29552,C1(C)(NC(C2CC2NC(C(C)OCCC=C)=O)=O)CC(=O)N(C)C1 29553,c1(C(N(CCCNC(C(CC)C)=O)Cc2ccccc2)=O)nc(C)ccc1F 29554,c1(C(N(C)CCn2cc(CCN3CCSCC3)nn2)=O)snc(Cl)c1Cl 29555,CCCCC(O)C(C)C(=O)NCCCC(=O)N(CC(C)OC)C(C)C 29556,C(=O)(C(C(C)C)OC)NC(CC)CN(C(=O)Cc1nc(C(C)(C)C)cs1)C 29557,C1(C)NC(=O)NC1=O.c12occc1C(=O)NCC2.C12CCC(C1)C(=O)NC2.CC 29558,C(=O)(C(C(C)(C)C)NC(C1CCC2(CCC2)O1)=O)N1CCC(C)(CCO)C1 29559,CC(C)C(F)(F)CC(=O)NCC1(C)CN(C(=O)C(n2cc(Cl)cn2)C)C1 29560,C#CCCC(O)C(=O)NCC1(C)CCCN(C(=O)CSCCOC)C1 29561,Cc1cc(C)n(C(C)CC(=O)NC23CC2CN(C(c2sc(F)cc2C)=O)C3)n1 29562,C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccc(C(N)=O)cc2)=O)CCC1C 29563,N1(CC(=O)Nc2cnn(C)c2)CCOC(C)(C(F)(F)F)C1.CN 29564,c1(-n2c(C(C3CCCOC3)CC)nc(C3CC3)n2)ccnc2ccccc12 29565,C1(NC(CCC(=O)OC(C)(C)C)=O)CC2CC1CN2C(c1cnc(C(N)=O)s1)=O 29566,CC(O)C(C(=O)N(C)CC1(CO)CC1)NC(C1CC(F)(F)C1)=O 29567,c1(-c2nc(CCCOC)nn2-c2cccc(OC)c2)cnn2ccc(O)nc12 29568,N1(C(CC)=O)CCCC2(CCN(C(C3CCn4nccc4C3)=O)C2)C1 29569,C=CC1(CC(N2CCC(NC(c3cscc3C)=O)C(CC)C2)=O)CCOCC1 29570,C1(NC(C2CC(SC)C2)=O)CCCN(C(c2cocn2)=O)C1C(C)C 29571,CCCCCCC(=O)NCC(O)CN(C)C(C1CCCSC1C)=O 29572,c1(C(=O)NCCC(C(C)C)NC(C(CC)C)=O)nc2ccccc2nc1C 29573,c1(C(N2C(CN(C(CCC#CC)=O)C)COCC2)=O)c(C)nc2sc(C)cn12 29574,C(CCC(C)C(=O)NCC12CC(CO1)N(C(c1cnc(OCC)nc1)=O)C2)CC 29575,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)CC3C=CCC3)CC2)cc(C2CC2)nn1C 29576,C1(CNC(CC(C)n2cccn2)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29577,c1(OC)cccc(O)c1C(=O)NCC(C)(C)CNC(C1CCCO1)=O 29578,c1(C(=O)NC(C2CCN(C(c3cnc(C)nc3)=O)C2)C)cc2ccc(Cl)cc2o1 29579,N1(C(C(=O)NC)=O)CCCC2CN(C(=O)CCCOc3ccc(C)cc3)CC12 29580,C(C(CC1CC1)C(=O)NC(C)COC(F)(F)F)NC(C(C1CC1)OC)=O 29581,n1(CC)nc(-c2ccc(Cl)cc2)nc1Cn1nnnc1-c1ccsc1 29582,c1(C(=O)NCC23C(CN(C(C=C(C)C)=O)C2)C3)cc(F)ccc1S(C)(=O)=O 29583,c1(C(N2CC(Nc3snc(C)c3C#N)C(C)C2)=O)ccc2c(O)nc(C)nc2c1 29584,CCC(C#N)(CC)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CC1 29585,C(=O)(CCCCCCNC(C1CCOC1(C)C)=O)NC(C)C(C)n1cccn1 29586,c1(C(=O)NCC(C)NC(C2(C(F)F)CCC2)=O)cn(C)nc1C(C)(F)F 29587,N1(C(C23CC(NC(=O)C(c4ccccc4)F)(C2)C3)=O)CCOC2COCC12 29588,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C#N)C2CC2)CC1 29589,N1(C(C(C2CCOC2)NC(C(COC)C)=O)=O)CC2(CC(C)CO2)C1 29590,C1(NC(c2c(C)ncs2)=O)CC2CCC1CC2NC(=O)Cc1ccc(F)c(C)c1 29591,c1(C(=O)NC2C(NC(C3(C=C)CC3)=O)CCCC2)cc(C)nc(O)c1 29592,N1(C(c2n(C)ncc2)=O)CC2C(NC(=O)CC3(CO)CCCCC3)C2C1 29593,C(N=c1cc(NC(C)C)nc[nH]1)C1(O)CN(C(C(C(C)C)N2CCCC2=O)=O)C1 29594,c1(CN(C(=O)C(=O)NCCc2ccc(C#N)cc2)C)sccc1S(C)(=O)=O 29595,c1(OC)ccnc(C(=O)NCC2CCCCN(C(=O)C=CC3CC3)C2)c1F 29596,c1(C(=O)NCCCCC(CO)NC(c2ccc(F)cn2)=O)cncc2sccc12 29597,c1(OC)ccc2c(c1)CCC(CNC(=O)C(=O)Nc1c(C)nc3sc(C)cn13)C2 29598,C1(C(=O)NC2CC(C=C)C2)(NC(=O)C=CCCC)CCCC1C 29599,CN1CCN(C(=O)C(=O)NCCCN2C(=O)CCC2=O)c2cccnc21 29600,c1(N2CCC(CCNC(=O)C(c3ccccc3)O)CC2)ncc2cccnc2n1 29601,N(C(=NCCc1cccs1)N1CCCC2(CCCCCC2)C1)C(C#C)COC 29602,C1(NC(C(n2ncc(C)c2)C)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC1O 29603,C(=O)(CC(C(=C)C)OC)N1CCCC(N(C(c2cc(CCC)[nH]n2)=O)CCO)C1 29604,c1(C(=O)Nc2cnsc2)ccc(CNC(c2cccc(-c3nn[nH]n3)c2)=O)cn1 29605,C1(C)(C(N2C(C(C)NC(C(c3cccc(C)c3)C)=O)CCC2)=O)C(C)(C)C1(C)C 29606,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29607,C(N=c1[nH]cncc1Cl)C1(NC(c2c(C)n[nH]c2C)=O)CCOCC1 29608,CCCC(C(=O)N1CCC(C(=O)OC)O1)NC(C)CO 29609,C(=O)(CC(C(F)(F)F)NC(=O)CCCNC(=O)C(C)=NOCC#N)NC 29610,N1(C(c2cc(CNC(c3c(C)occ3)=O)oc2)=O)C(CO)CCC1C 29611,c1(N(CCCC=C)C)ncnc(N2CCCC(c3ccccc3)C2C(C)C)c1C 29612,N1(C(C(CC#C)(C)C)=O)CCC(C2CCCN(C(C3(CC)CCC3)=O)C2)CC1 29613,N1(C(C2(C)CCCCC2)=O)CC2CCC(C1)N2C(c1cc(I)c(O)c(I)c1)=O 29614,C1(C(=O)NC(CNC(c2cnn(C)c2C#N)=O)CO)Cc2ccccc2CO1 29615,c1(C(N2CCC(NC(C3CC(OC)(OC)C3)=O)C(O)C2)=O)cc2ccccc2[nH]1 29616,CCC(C)C(C(=O)NCc1nc(C)no1)NC(=O)CC(C)C1CCCO1 29617,CC(C)CCCC(C)C(=O)NC1C2CC3C(C2)C13C(=O)N(C(CO)C1CC1)C 29618,c1(C(=O)NC(C2CCN(C(C(=CC3CCCC3)C)=O)C2)(C)C)nc(Cl)c(Cl)s1 29619,C1(C(=O)NC(c2cn(CCCCO)nn2)C)COc2ccc(Cl)cc2C1 29620,CCCCC(=O)C(=O)NC(CO)C(N1CC(CO)CC1CO)=O 29621,C1(N(C)C(C23CCCC2C3)=O)CCC(NC(C2(C3CCCO3)CC2)=O)CC1 29622,c1(C(=O)NC2(CNC(c3ccc(N)c(Cl)n3)=O)CCCC2)ccc2ccnn2c1 29623,C(=O)(CS(=O)(=O)CCC)NC12CC(NC(C(CC)N(C)C)=O)(C1)C2 29624,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29625,C(=O)(CCC(F)(F)C(=O)NCC(CO)N(C)C)OCC.c12ccc([nH]1)CNC2=O 29626,N1(CCNC(C=CC2(C)COC2)=O)CCN(C(=O)CC2CCNC2=O)CC1 29627,CC(C)C1C(=O)NC(=O)CCN(C)C1C.C1(C#N)(C(=O)NCC(F)F)CC1 29628,C(=O)(CC(O)CC(C)(C)C)N1CCC(C(=O)NCc2cncc(C)c2)C1 29629,c1(C(N(C2CN(C(C=CC=CC)=O)C2)CCO)=O)cccc2ccc(Br)nc12 29630,C(CO)(CCF)NC(C(C)N(C(=O)C=CCN1CCC1)C)=O 29631,Cc1cccc2c1c(Nc1nccc(CNC(c3ccc(Cl)c(I)c3)C)n1)cn2C 29632,c1(C2(C(=O)NC(C)CN(C)C(C3(C)CC3Br)=O)CC2)ccccc1 29633,N1(C(C(CC)C#N)=O)CC2CCCC(CNC(c3nc(C)ccc3C)=O)C2C1 29634,CCC(CC(=O)N1CCCC1(C)C(=O)NCC1(C)CCOCC1)C(C)(C)C 29635,CC1(C)OCCC1C(=O)NC1CCCC1NC(c1ncccc1O)=O 29636,N1(C(c2c(C)n(C)cc2)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29637,Cc1ccc(O)nc1CNC(C1CCCN(CC2CCSC2)C1)=O 29638,N1(C(CCNC(=O)OCC)=O)CCC2(CC1)COC(CNC(=O)CC1CC13CC3)C2 29639,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2nnc(C)n2)CC(C)(C)C1 29640,N1(C(C(C)SC(C)C)=O)CC2CCC1C2NC(C1Cc2cscc2C1)=O 29641,C1(C(=O)NCC(CC(C)C)NC(=O)CC2CC3(CCC3)C2)CN2CCN1CC2C 29642,C(C1=NOC2CCCC12)NC(CNC(CNC(c1cc(C)oc1)=O)=O)=O 29643,C(=O)(CC(C)C(F)(F)F)NCCCN(C(C1CC(C)(C)C1)=O)CC 29644,c1(C(=O)NC23CN(C(c4c(CC)nccc4)=O)C(C2)C3)ccnc(Cl)c1OC 29645,CCCC(CC)C(=O)NCCN(C(C1CCC1N)=O)CC1CCCC1 29646,C12(C(=O)NC(CC)(C)CN(C)C)CC(CN1C(C1CC(OCC)C1)=O)C2 29647,C(=O)(CC(C)P(C)(C)=O)N(CCNC(CSCC(=O)OC)=O)C(C)C 29648,C(=O)(C1=CCCN(C(C2(C(C)(F)F)CC2)=O)C1)NC1C(OC)COCC1 29649,N1(C(C#C)C)CCCN(C(c2cscc2Br)C(=O)NC2(C)CC2)CC1 29650,N1(C(c2ccc(C)c(O)c2)=O)CC2=C(C1)CN(C(C1(C)CCCS1(=O)=O)=O)C2 29651,C12(CNC(C3(C(=O)NC)CCC3)=O)CCC(CN(C(=O)C3=NOCC3)C1)C2 29652,CCCC(C)(CCC)C(=O)NC1CN(C(=O)C(C)(C)CNC(C)=O)CC1C1CC1 29653,C(N=c1nc(O)c(Br)c[nH]1)C1CCC(NC(c2ccc3nnnn3c2)=O)C1 29654,c1(C(N2C(CNC(C3CCCS3)=O)CC(C)(C)C2)=O)cnc(O)c2ncccc12 29655,Cc1nc2ccnn2c(C)c1C(N1CCN(C)CC1CNC(=O)C#CC(C)C)=O 29656,Cn1cnc(CC(=O)NC(C)(C)CN(C(C2CC(F)(F)C2)=O)Cc2cccs2)c1 29657,Cc1ccc(C(N2CC(NC(=O)Cn3nnc(C4CC4)n3)C2)=O)cc1C1CC1 29658,N1(C(c2cc(SC)oc2)=O)CCN(CC(C)NC(=O)CCCCN(C)C)CC1 29659,C1(CN(C)C(c2c(C)cco2)=O)CN(C(=O)CCCCN2CCCC2)CC12CCC2 29660,c1(C(=O)NC23CC2CN(C(C2CC4(C2)CC(O)C4)=O)C3)cn2cc[nH]c(=O)c2n1 29661,C1(CS(N2CCC(NC(=NC)NCCOC(C)C)C2)(=O)=O)CCC(F)(F)CC1 29662,C1(NC(c2n(C)cnn2)=O)(CO)CCOCC1.C12CCOC1C(=O)NC2 29663,c1(C(N(CCC(C)(C)NC(C2(C3CCCO3)CC2)=O)C)=O)cccc(F)c1O 29664,CC1OCCN(C(=O)CC(C)CNC(=O)CSCC(N)=O)C1C 29665,N1(C(C#CC2(OC)CC2)=O)CCN(C(=O)CSC2Cc3ccccc3O2)CCC1C 29666,C1(C(=O)NCC2=CCN(C(C3CCCN3C3CC3)=O)CC2)C2CCC3C(C2)CC13 29667,Cc1c(Br)c(C(N2CCC(CNC(=O)C(C)N(C)C)C23CC3)=O)nn1C 29668,C1(C(=O)NCCN(C(Cn2c(C)c(Cl)cn2)=O)C2CC2)CCC2(CCC2)CC1 29669,C(=O)(C1=CC2CCC(C1)C2)NC1CCC(C(N2CCC3(CCN(C)C3)C2)=O)CC1 29670,C1(CC(=O)NC(C(C)C)CNC(=O)CN2CCCC2=O)CCCS(=O)(=O)C1 29671,c1(C(=O)NCCCCN(C(CSCC)=O)CC)cc(C)ccc1C1CC1 29672,c1(CC)cccnc1C(=O)NC(C)CN(C(=O)C(=Cc1ccccc1)C)CC 29673,Cc1ccc(NC(=O)C(=O)Nc2ccnc(F)c2F)c(I)c1 29674,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29675,C(=O)(CC(C)(C)COC)NCCN(C(C(C1CCC1)SC)=O)CCCN(C)C 29676,C1(NC(CC2(C)CN(Cc3c(C)nn(C)c3Cl)C2)=O)CCC2(CC1)OCCO2 29677,n1(CC(=O)NC2CC(C)CN(C(C3CCS(=O)(=O)CC3)=O)C2)ncc2ncccc12 29678,C12(C(=O)NC(C)CC3CC3(F)F)COCC(c3ccccc3F)(C1)C2 29679,C12(C(=O)NCc3cncc(C)n3)CC(CN(C(c3c(C)noc3C)=O)C1)C2 29680,CCCCCC(C)(C)C(=O)NCCC1(C)CCN(C(=O)CC2CCCO2)CC1 29681,C(=O)(C1OCCn2ccnc21)N1CCC(CNC(c2n(C(C)C)ccn2)=O)CC1 29682,c1(OCC)ccc(C2CCN(C(=O)NCC3COC(C4CC4)C3)CC2)cc1 29683,N1(C(c2nn(CC)nc2C)=O)CCC(NC(c2occc2C)=O)C(CO)C1 29684,N(C(=NCCCCl)N1CCCC(C)(F)C1)CCN(CC)Cc1ccccc1N.CC 29685,C1(COCc2ccccc2)CC(O)CN1C(C1CCC(O)C1)=O.C1(C2CC2)C(=O)N1 29686,c1(C(N)=O)c(-c2ccccc2)ccnc1NC(C1CCC(C2CC2)O1)=O 29687,C1(C)(C(=O)NCC(CNC(CCOc2c(C)cccc2)=O)C)CCS(=O)(=O)CC1 29688,c1(CNC(N(C(CC(C)C)CO)C)=O)cc(Cl)ccc1C(F)(F)F 29689,C(CCC)(C(=O)NC1CCN(C2CCN(C(=O)C=Cc3cccs3)C2)CC1)=CCC 29690,Cc1cc(NS(C)(=O)=O)ccc1NC(N1CC(Nc2ccccc2Br)C1)=O 29691,C1(C2CC2)(CNC(CNC(CN(C)C)=O)=O)CCN(C(C2(C)CCOC2)=O)C1 29692,C1(CC(N2CC(C)C(NC(=O)Cc3nncn3C)C2)=O)CCC(F)(F)CC1 29693,C1(NC(=O)CCn2cc(Cl)cn2)CN(C(c2cnn[nH]2)=O)C2(CCCC2)C1 29694,N1(C(c2cc(C(C)=O)on2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29695,C#CC1CCC(C(=O)NCC2CN(C(c3ccc(C(=O)OC)c(F)c3)=O)C2)CC1 29696,C1(CCC(N2CC(CC)(NC(C3CNC(=O)N3)=O)C2)=O)CC(C)(C)CO1 29697,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29698,N1(C(C2C(C)CCC2)=O)Cc2[nH]nc(C(=O)NCCOC3CC3(F)F)c2C1 29699,c1(C(=O)NC2(CCC=C)CN(C(=O)C(C)CC=CCCOC)C2)cc(C)ccc1F 29700,Cc1cc(SCC(=O)N(CC(=O)NCCC(C)C)CC(C)C)c[nH]1 29701,CC1CC(c2ccccc2)(NC(c2nnnn2C)COC(c2ccccc2)C)C1 29702,C(=O)(C(CC=C)CC(C)C)NC(C(=O)N1CC(OCC#C)C1)CCF 29703,c1(C(C)C)[nH]nc(C(=O)NC2CCN(C(C3(NC(N)=O)CC3)=O)C23CC3)c1[N+](=O)[O-] 29704,CC1CCCN(C(c2cnc(C#N)s2)=O)C1CNC(=O)CCF 29705,N1(C(c2c(C(C)C)con2)=O)CCCC(N(CCO)C(c2csnc2Cl)=O)C1 29706,C1(N(C)C(C2C3COCC23)=O)CCCN(C(=O)CSc2ncccn2)CC1 29707,c1ccc(C)o1.C1(C(=O)NC(CNC(C)=O)C2CC2)CCCOC1 29708,C1(C(=O)NC2C(NC(C3(CCC)CCC3)=O)CC2)CCSCC1 29709,N1(C(c2c(CC)c[nH]n2)=O)CCC(C(=O)N(CC(=O)NC(C)C)C)C(C)(C)C1 29710,c1(CN2C3CN(C(=O)Cn4cccc4)C(C3)C2)c[nH]c2nccc-2c1 29711,Cc1cc(=NC2CCC(=O)N(C(C)C)C2)[nH]c(N2CCC(C)OC(C)C2)n1 29712,C1(C(=O)NC(CCNC(CC(CC)OC)=O)C(C)C)CC12CCS(=O)(=O)CC2 29713,C1(C(=O)NCc2nnnn2C2CCCC2)C=CC(NC(C2CC2(F)F)=O)C1 29714,CC1CSCC1NC(=O)CC1(N(C)C(C2CCN2C2CCCC2)=O)CC1 29715,N1(C(=O)NCC2C(C)COCC2)CCOC(C#N)C1 29716,C(CCC(=O)NC(C1CCCN1C(=O)CC1CC(F)(F)C1)(C)C)OC(C)C 29717,C1(NC(c2ccc(CO)cc2)=O)CCC(NC(=O)C(F)Cc2ccccc2)CC1 29718,C1(NC(c2c(C)n[nH]c2)=O)(CO)CC2CCCC12.c1(C2C(=O)N2)ccnn1C 29719,c1(C(N2CC3C(CNC(CC)=O)C3C2)=O)oc2ccccc2c1CS(C)(=O)=O 29720,C1(CCNC(C(=O)N(C(c2nc(C(F)(F)F)no2)C)C2CC2)=O)CCCCN1C 29721,c1(C(=O)NCCCNC(Cc2ccn(CC)n2)=O)cc(C(C)=O)c(C)nc1C 29722,C12(C(=O)NC(CNC(C(COC)O)=O)COC)C3CCC(CC13)C2(F)F 29723,CC1CCC(CNC(c2cnc(C(N)=O)cn2)=O)CN1C(=O)CS(=O)(=O)N(C)C 29724,C1(NC(C=CCN(C(C(CC#C)O)=O)C)=O)CCCCN(C)C1=O 29725,C(CC(C)(C)C)(C(=O)N1CC(CN(C(=O)C=C(C)C)C)C2(CC2)C1)OC 29726,C1(CCOCC)(OCC(=O)NC(CCNC(C(C)NC(CC)=O)=O)C)CCOCC1 29727,Cc1ocnc1CC(=O)NC(=O)Cn1cnnc1CC1CCC(C(N)=O)C1 29728,c1(C(N(CC(C)NC(=O)C=C(C)C)CC)=O)ccc(OC)cn1 29729,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29730,N1(C(c2nc(Br)c(C)s2)C(=O)NCC=C)CCCC(O)(CC=C)C1 29731,N1(C(C#C)=O)CCC2(C1)C(=O)Nc1ccc(C(=O)NC3CCN(CCC)C3)cc12 29732,CCCC(CC(C)C)C(=O)NC1CC(NC(=O)CCCC(F)(F)F)CC1O 29733,C(=O)(CCCC(=O)NC)N1CCC(NC(C2(OC)CCSC2)=O)C1C(C)C 29734,N1(C(c2cc(CC)nn2C)=O)CCC2C(C1)CN2C(c1cnc(SC)s1)=O 29735,CCCCCC(C)CC(=O)NC1C2CC1N(C(=O)C1=NNC(=O)CC1)C2 29736,Cc1noc(N)c1C(=O)NC1CC(CCC(N2CCOC(CCF)C2)=O)C1 29737,C(CNC(=O)C(O)CN(C)C)(CC(=O)Nc1ccccc1Cl)OC 29738,C(=O)(C(CC(=O)NC(C)CCNC(C1(Cl)CC1)=O)C(C)=O)OC 29739,CC1CN(C(=O)CCn2ncn(C)c2=O)CC1CNC(=O)CSCC(N)=O 29740,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29741,N1(C(c2c(C)snn2)=O)CCC(C(C)CNC(C2(P(C)(C)=O)CC2)=O)CC1 29742,N1(C(CC(C)N(C)C)=O)CCC2CCN(C(c3cc4n(n3)CCNC4=O)=O)CC12 29743,c1(C(=O)NCC(C)(C)NC(c2c(COC)ncs2)=O)cccc2ncnn12 29744,c1(C(N2CCCC(CC=C)(NC(c3ccc[nH]3)=O)C2)=O)nccn2cccc12 29745,C1(NC(CCC(C)(C)C#N)=O)CC(NC(c2occc2Br)=O)C12CCOCC2 29746,C1(NC(C2CCC(NC(=O)C(F)OC(F)(F)F)CC2)=O)CCN2CCC1C2 29747,C1(C2(O)CN(C(=O)C(C)OC)C2)(C)CC1.CCCS(=O)(=O)N1CC(=O)N1.C(C)(C)O 29748,C=C(C(=O)NCC(F)(F)Oc1ccc(OCC)cc1)C(C)(C)C.COC 29749,CC1(C)CNC(=O)CN1c1ccnn1Cc1cccc(C(F)(F)F)c1 29750,CCCCC(CC)C(=O)NC(C)(C)CCCNC(c1cnc(OC)cc1)=O 29751,O(S(=O)(=O)CC1CCN(C(=O)OC(C)(C)C)C1)CC(=O)N(C1CCCCC1)C 29752,c1(C(=O)NC(C)C(C)(C)Cc2ccccc2)nccc2ccn(C)c12 29753,C(=O)(C(C(C)C)c1ccncc1)N(CCCNC(C(c1ccnn1C)OC)=O)C 29754,C(CCNC(c1ccc(SC)s1)=O)(C(C)C)NC(C1(CC)CCCO1)=O 29755,c1(OCC)cc(CCC(N2CC(O)(c3cn(C(C4CC4)CC)nn3)C2)=O)on1.C1CC1 29756,N1(C(CCCC)(C)C)CCC(=O)N(Cc2cn(CCO)nn2)C1=O 29757,c1(C2C(C(N(CCNC(CCC(=C)Br)=O)C)=O)C2)ccc(C#N)cc1 29758,C1(C(N(CC(C)NC(CS(=O)(=O)NCC)=O)CC)=O)CCCC2(CCOCC2)O1 29759,c1(C(C)C)ccc(OCC(N2CC(CO)(NC(C34CC(C)C3C4)=O)C2)=O)cc1 29760,C(=O)(CC1=CCN(C(c2cccnc2O)=O)CC1)N(CC(C1CC1)OC)C 29761,C(=O)(C1c2c[nH]nc2CN1C(c1ccc(Cl)s1)=O)N1C(C)COCC1 29762,C1(C#N)(CNC(C)=O)CCN(C(=O)CC2CCOC2=O)C1 29763,CCC(CC(C)C)C(=O)NC1CCC(NC(=O)Cc2ccc(C#N)cc2F)CC1 29764,C(=O)(CC(O)CNC(C1CC1C(F)(F)F)=O)N(CC(CC)CC)C1CC1 29765,c1(OC)ccc(F)cc1C(=O)CCC(=O)N1CC(CNC(c2ncn(C)n2)=O)C1 29766,c1(OC)ccc2nc3nc(c2c1)N(C)C3.c1(OC)ccc(-n2ccnc2O)cc1 29767,C(=O)(C(F)CC1CCC1)NC(C)CNC(=O)CCOC1CCC1 29768,Cc1cnc(CNC(C2CCCCC2n2cc(CCS(=O)(=O)N(C)C)nn2)=O)cn1 29769,C1(C)(CNC(C2CC(C)C2)=O)CN(C(=O)CSCc2ccc(F)c(F)c2)CC1C 29770,C(CC1=CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1)N(C)C(c1cnsn1)=O 29771,N1(C(C(C(C)C)n2cc(Br)cn2)=O)CCCC(NC(C2CC2(C)C)=O)CCC1 29772,N1(C(Cc2cccc(OCC)c2F)=O)CCc2c(C(=O)NC)n[nH]c2C1 29773,CC1CCCN(C(c2cnc(C(F)F)s2)=O)C1CCNC(=O)CCNC(N)=O 29774,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29775,C1(C(=O)NCC=C(C)C)C=CC(NC(c2[nH]nnc2C)=O)C1 29776,c1(-n2cc(C3CCN(C(C(C)OCC)=O)C3)nn2)ncnc2scc(C)c12 29777,C(C(CNC(C1CCC(C)S1)=O)S(C)(=O)=O)NC(C1CC(OCC)C1)=O 29778,CC1CCCCC1(CNC(=O)COC1CCCC1)NC(=O)CCc1ncccn1 29779,N1(C(c2c(C)ccnn2)=O)CCCN(C(C2C3CCCCC23)=O)C(C)C1 29780,CCCC(C)(CC)C(=O)N(CCCCC(=O)NC1(C(=O)OC)CC1C)C 29781,c1(C(N2CCN(Cc3ccc(OC)cc3Cl)C(C)C2)=O)cccc2oc(O)nc12 29782,c1(CN2CC(O)C(C3CC3)C2)c(F)c(F)c(Cl)c(F)c1F 29783,N1(C(=O)NCc2c(OC)ccc(I)c2)CC2CN(C)CCC2(CO)C1 29784,c1(C(N2CCC(NC(C3(OC)CCC(C)(C)C3)=O)C2)=O)cccc2c1CC(=O)N2 29785,C12(C(=O)NC(CC=C)CO)CC(C)(CN1C(c1c[nH]c(=N)c(C)c1)=O)C2 29786,C1(OC)(CNC(C2(F)CC2)=O)CCN(C(c2cccc(-c3csc(C)n3)c2)=O)C1 29787,N1(C(=O)COC(C2C3CCC2CC3)=O)CC2CCCC2(Nc2ccc(F)cc2)C1 29788,CC(=O)CCN=C(NCCC1(CO)CCC1)N1CCN(c2cccc(F)n2)CC1 29789,c1(C(N2CC(n3ncc(NC(c4cccnc4O)=O)c3)C2)=O)ccc(Br)c(F)c1 29790,c1(C(=O)NC(C2CCCCC2)CNC(C2(CC)CCCC2)=O)ccc(F)cc1N 29791,OCCC(N=c1[nH]c(=NCCCCCF)c2[nH]ccc2[nH]1)C1CCCCC1 29792,C#Cc1ccc(C(=O)NCC2(COC)CCCN2C(=O)CCCC=C)c(C)c1 29793,C(=O)(CN1C(=O)CCc2ccccc21)NC(CN(C(=O)CSC)CC)C 29794,Cc1nc(CNC(c2nnnn2-c2ccccc2)C2CC23CC3)sc1C 29795,c1(OC(C)C)ccc(Cl)c(C(N2CC(CCNC(=O)C(F)C(C)C)C(C)C2)=O)n1 29796,N1(C(CCCCCNC(C(C)C#N)=O)=O)CCc2c(C#N)cccc21 29797,C(=O)(CCCCC(=O)NCc1ccc(C(=O)NCC(C2CC2)OC)s1)OC 29798,N1(C(c2c(OC)nn(C)c2)=O)CCC2(NC(=O)CCc3cnn[nH]3)CC2C1 29799,n1(CC(C)SC(F)F)cc(C(C)N(C)C(c2cnc(-c3ccoc3)s2)=O)nn1 29800,c1(CNC(c2cocc2NC(=O)COCCF)=O)cn(C2CC2)cn1 29801,C1(CNC(C2(CC=C)CC2)=O)CN(C(=O)COc2cccc(F)n2)CCO1 29802,C(=O)(CCCCC(N)=O)N1CCCC(CCCCNC(C(CN(C)C)O)=O)C1 29803,c1(C(N(C23CCC(C2)N(C(=O)COC2CC2)C3)C)=O)cnc2ccc(C#N)cn12 29804,c1(N(CCOC)C)[nH]c(=NCc2cc(O)nc(O)n2)nc2scnc12.C(C)(COC)N 29805,Cn1cnc2c(N3CCC(C(C)NC(c4cn(C5COC5)nn4)=O)C3)ncnc12 29806,C(CCCC(C)(C)C(=O)NNC(=O)CCCCC(C)C)NC(CCC(CCC=C)CC)=O 29807,N1(C(C2N(C(c3ccc(OC)cc3)=O)C3(CC2)CC3)=O)CC(C)CCC12CC2 29808,N1(C(C(N2CCCC2=O)C)=O)CCCCC(CNC(=O)Cc2ccc(Cl)nc2)C1 29809,c1(CC(=O)NCC(C(C)C)NC(=O)C=CSc2nc[nH]n2)nn(C)cc1Cl 29810,c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc(F)cnc1O 29811,c1(C(C)(C)C#N)cncc(C(=O)NCCNC(c2ccns2)=O)c1 29812,N1(C(c2c[nH]ccc2=O)=O)CCc2ncccc2C1.CC1(C)CC2N(C1)C2=O 29813,C(C(C(=O)NCCCSC)N(C1CCCS1)C1(C)CC1)(C1CCCC1)OC 29814,C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C(C)NC(C1CCCS1)=O)CO 29815,Cc1cc(-c2nc(CN3CC(C4(C)CCC(=O)N4C)C3)no2)cc(N)c1Cl 29816,C1(NC(C2C(NC(C(C)C3(O)CCC3)=O)COC2)=O)CC(C)(C)C12CCC2 29817,c1(C(C)NC(c2n(CC=C)nnn2)c2ccc(CC)s2)ncccc1Br 29818,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 29819,CCC(C(C)(C)O)NC(C1CC(C)(NC(=O)CC2CC3(CC3)CO2)C1)=O 29820,N1(C(C2C(CCC)C2)=O)CCC(C(=O)NC2C=CCCC2CO)CC1(C)C 29821,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 29822,c1(N(CC(C)(C)C)C)cccc(S(=O)(=O)NCCCCCOC(F)(F)F)n1 29823,CC(C)CCC(O)C(=O)N1CC(O)(CN(C(=O)CC2(C)OCCO2)C)C1 29824,C(=O)(CCC(C)(C)c1ccccc1)OC(CC)C(C)C 29825,c1(C(=O)NC2C3CN(C(c4ccc(OC)s4)=O)CC32)cc(OC)cnc1C 29826,C(CCCCCC(=O)N1CC2(C1)CN(C(=O)CC1(C(F)F)CC1)C2)SC 29827,C(CCCC(=O)NC(CNC(C1(CC)CC1)=O)CCO)OCC 29828,c1(C(N(CCOC)CCNC(=O)Cc2cc(=O)n(CC#N)[nH]2)=O)ccn(C)c(=O)c1 29829,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)C2(CC2)C1 29830,CC1C(C(=O)NCC(C)(C)OCCNC(c2cc(CN(C)C)cn2C)=O)CCN1C 29831,C1(F)(CNC(c2nc(CC)oc2)=O)CCC(NC(C2CCSCC2)=O)C1 29832,C1(CNC(=O)NCc2ccccc2)CC(C(=CCCOC)C)CCO1 29833,N1(C(CCNc2ccc(C)cc2)=O)CC(CNC(c2cc(C)sn2)=O)CCC1C 29834,C(c1cc(F)c(F)c(F)c1)=CC(N1CCOC2(C1)CN(C(c1nccs1)=O)C2)=O 29835,c1(OCC)ncccc1C(=O)NCCOCCNC(=O)C(CC)c1ccccc1 29836,O=C1CNC(=O)c2cc(C(=O)NC3CC3CNC(C3(F)CC3)=O)ccc2N1 29837,Cn1ccc(CCC(=O)NC2(C(=O)NC3CC3(C)C(N)=O)CCC2)c1 29838,C1(C(N2CC(NC(c3nc(CCC)sc3)=O)C(OC)C2)=O)CC2(CCCCO2)C1 29839,c1(C(N(CCNC(C2CCNC2=O)=O)CC2CC2)=O)[nH]nc2ncccc12 29840,c1(C(C(=O)NCc2ccccc2)N(C2CCS(=O)(=O)C2)C)cc(F)ccc1Br 29841,N1(C(C(CCC)OC)=O)CCN(C(C2(C)CCC2)=O)CC1C 29842,C1(CC(=O)NC2(CCCO)CCC2)CC1(Br)Br 29843,CC(O)(CNC(c1cc(CCNC(=O)C(F)=CC2CC2)on1)=O)CO 29844,CCN=c1[nH]cc(C(N2CCC(C(C)CNC(=O)CC(O)C(C)C)CC2)=O)s1 29845,C(=O)(C1=CCCC1)NCC(CO)NC(c1cc(CC)on1)=O 29846,c1(C(N2CCN(C(c3coc(C(F)F)c3)=O)C(CO)C2)=O)cc2cnccc2o1 29847,C1(C(N2CCC(C(C)NC(c3ccc(C)o3)=O)C2)=O)CC=CCC1C 29848,c1(C(=O)NC2C3(CN(C(CSCC(=O)OC)=O)C3)CC2)cnc2snc(C)c2c1 29849,c1(OC)cc(C)c(F)cc1S(=O)(=O)N1CCCC1C(=O)NCCC#N 29850,C1(C)(CN(C(COCCC#C)=O)C)CCCC1NC(c1cncn1C)=O 29851,CC(C)(C)CCC(=O)NC12CCC(NC(C3CCC(C)(C)CC3)=O)(CC1)C2 29852,N1(C(C(CCNC(=O)CCc2nc[nH]n2)OC)=O)CCC2(CCOC2)CC1 29853,N1(c2nnc(C3N(C)C(=O)COC3)n2CC(=O)NC)CC(C)CC2CCCCC12 29854,c1(C(N2CCCN(C(=O)CC(C)(C)C)CC2)C(=O)NC)cc2c(cc1C)OCO2 29855,n1(CCOCC=C)c(N2CCC(C(O)C(F)(F)F)CC2)nnc1Cc1nccs1 29856,c1(C(=O)NC(C2(O)CN(C(C3CCCS3)=O)C2)C)cc2cccn2c(O)n1 29857,c1(C(N2CCC(NC(c3nc(OCC)sn3)=O)C2)=O)c(C)nsc1OCC 29858,C1(C(=O)NCCC2CCC3CC23)(OC)CC(C)C1.C1CC(=O)N1 29859,C(CNC(=O)CCn1cnccc1=O)(C(C)(C)C)NC(C(CSC)OC)=O 29860,c1(C(N2CCCCC(NC(CSC(C)(C)C)=O)C2)=O)cc2cc(O)ccc2[nH]1 29861,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 29862,C(=O)(CC(C)(C)C(C)(F)F)NCC1C(CNC(Cc2n(C)cnn2)=O)C1 29863,Cc1ccc2nc(C)c(C(=O)NCC(O)CN(C(=O)CC#N)C)cc2c1 29864,N1(C(c2cccc(C3(O)CCN(CCO)C3)c2)=O)CCc2nc(C3CC3)ccc2C1 29865,CC(=O)n1cc(CN2CC3(CC3)CC2CC(N2CCCC2)=O)c2cccnc12 29866,CN1CC(C)(C)CC1C(N1CCC(N(CCO)C(C2(C)CCC2)=O)C1)=O 29867,CCC(N=c1[nH]c2c(c(=NC(C)C3CCCO3)[nH]1)CSC2)c1ncc(C)[nH]1 29868,Cn1cc(CN2CC(C(=O)Nc3cccc4[nH]cc(C#N)c34)C2)c2ccccc12 29869,CCC(CC)C(F)C(=O)NCC(=C)CCNC(c1ccc(F)c(C)c1Cl)=O 29870,n1(CCCCCC)nc(-c2cnn(CCC)c2)nc1CCC(C)(C)CCO 29871,CCC(CC)CC(=O)N1CCC(C(=O)NCc2ccn(C3CC3)n2)C1CC 29872,CCCC(C#N)C(=O)NCC1(CC(N2CC(N(C)C)C2)=O)CC1.C1C(=O)N1 29873,c1(OC)ccc(F)c(-c2nc(CC3(C)CC3)nn2C(C)C)c1OC 29874,CCCCC(O)C(C)C(=O)NC1CCCC1C(=O)NC1(C)CC(C)(C)OC1=O 29875,C(=O)(C#CC1CCCO1)NCC1(C(N)=O)CN(C(C2(CC)CCNC2=O)=O)C1 29876,c1(CC(N2CCC(C(C)NC(=O)CCC3CCCO3)C2)=O)c(C)nc(O)nc1O 29877,C12(C(=O)NCC3CCC=CCC3)CCCC1N(C(c1sccc1F)=O)CC2 29878,Cc1ccc(C(=O)N(C)C)nc1C.C1(c2ccco2)C(=O)NOC(C)C(=O)N1 29879,N#Cc1ccc(CC(c2nnn[nH]2)C2CC2)cn1.n1(CCN)cnnc1 29880,C1(OC)CC2CC1CN(C(C1CC(C)N1C(c1sncc1C)=O)=O)C2 29881,c1(CC)ccnc(C(C(=O)NCC2CC2)N(C)CC2(C#N)CCC2)c1 29882,c1(C(N(C)CCOc2cccc(F)c2)=O)nccc(=NCCCCn2ccnc2)[nH]1 29883,C(C(C)C(C)C(=O)N1CC(CCCCNC(c2nnc(O)nc2O)=O)C1)OC 29884,c1(C(CNC(COCCC=C)=O)NC(C2CCC2F)=O)ccccc1 29885,CC(CC(=O)N1CCN(C(c2cnn(C3CC3)c2)=O)C(c2ncc[nH]2)C1)C(F)F 29886,N1(C(C(C)OCC)=O)C2CCC(C2)C1CNC(c1cncc(F)c1)=O 29887,C1(C(=O)NCC(C2CCCC2)C)(NC(C2CNC(=O)N2)=O)CCCC1 29888,Cc1cc(C(=O)N(C)CCN(C)C(c2cc(C3CC3)n(C)n2)=O)sc1Cl 29889,C1(NC(=O)Cc2cnc[nH]2)CN(C(=O)C2=CCOCC2)CC2(CCC2)C1 29890,N1(CC=CC(N2CCNC(c3ccccc3)C2)=O)CCc2ccccc21 29891,C(=O)(CC(O)CN(C)C)N(CC(C)(C)NC(C1(c2nc(C)sc2)CC1)=O)C 29892,N=c1nc[nH]c(=NCCOC2CCN(C(c3cc(F)c[nH]3)=O)CC2)[nH]1 29893,N1(CC2CN(C(Cc3ccn(C)n3)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 29894,C1(CC(=O)NCCn2cc(Cl)cn2)CCC(NC(=O)C(C2CC2)C2CC2)C1 29895,c1(C(N(C)CC2(O)CN(C(C(C)OCCC=C)=O)C2)=O)ccnc2ccncc12 29896,c1(CCNC(C23C(CN(C(=O)CCn4cncn4)C2)C3)=O)ccc(F)c(F)c1 29897,c1(C(N2C(CNC(C(C)Sc3nncn3C)=O)CCC2)=O)cc2n(n1)CCCO2 29898,O=S(=O)(c1sccc1I)N1CCN(S(=O)(=O)CC2CN(CC(F)(F)F)C2)CC1 29899,Cc1nc(=N)[nH]cc1C(=O)NCCNC(C1CCN(CCF)CC1)=O 29900,C(CC(CNC(=O)C(CO)N(C)C)NC(=O)CC=CC(C)(C)C)OC 29901,N1(C(CCN(CC)Cc2ccccc2)=O)CCC(c2nnc(S)n2C)C1 29902,c1(C(CO)NC(=O)Nc2nccc(CC)c2)cc(Br)ccc1C 29903,C(=O)(CCCCCc1ccccc1)N(CC(C)NC(=O)CC(C)CN(C)C)CC 29904,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(N2CC(C)C(C)C2)=O)C1 29905,N1(C(COCC)=O)CCC2(CCN(C(C3(S(C)(=O)=O)CCCC3)=O)C2)C1 29906,C12(COC)CC1CN(c1ccnc(COC)n1)C2 29907,c1(C(N2C(C)CC(CNC(c3ccc(F)nc3)=O)C2)=O)ccc(F)c(N)c1 29908,c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)CCOC2)cn2cccnc2n1 29909,N1(C(Cc2cn(CC)nn2)=O)CCC2(CC1)CC2C(N1CCC(CO)CC1C)=O 29910,C=CC(C)(CC)NC(C1CCC1NC(c1cc(COC)[nH]n1)=O)=O 29911,N1(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CN2CCOC2=O)CC1 29912,CC(CNC(=O)C=CC(=O)OC(C)(C)C)N(C)C(C1(O)CC1)=O 29913,CC1CN(C(c2cnc(S)n2C)=O)CC(C)C1NC(c1coc2c1CCCC2)=O 29914,Cc1nn2ccccc2c1C(=O)NCC1CCC(NC(C2CCCC2(F)F)=O)C1 29915,N(C(=NCCOC)NCc1nccs1)CC(c1cccc(C)c1)OC1CCCCC1 29916,c1(C(N2CCN(C(c3scc(C#N)c3)=O)C3C2C3)=O)ccc2ccccc2c1 29917,Cc1nc(C(F)(F)C(=O)N(CC(C)NC(=O)CCc2nc(C(C)C)no2)C)n[nH]1 29918,C(=O)(CCCS(N)(=O)=O)N(C(CN(C(C(C)NC(COC)=O)=O)C)C)C 29919,C1(CC(=O)OC(c2ccc(F)c(F)c2F)C)CCc2ncc(Br)n2C1 29920,c1(C(N2CCC(C)(CNC(C(CCCC)C)=O)CC2)=O)cc(OC)c(O)c(N)c1 29921,C(C)(CCC(=O)NCC1OCCC1C(=O)NCC1(C#N)CCC1)OCC 29922,c1(C(N(C2CCN(C(C3CC3OCC)=O)CC2)CCC)=O)ccc(F)cc1Cl 29923,C1(N(C(=O)Cn2cnnc2O)C)CCCN(C(=O)CN2C(=O)CCC2=O)CC1 29924,Cc1ccncc1CC(N1CC2C(CNC(C3(C(C)C)CCCO3)=O)C2C1)=O 29925,Cc1cnc(C(N2CC(CCNC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)cc1Cl 29926,CC1CC(=O)NC1C(=O)NC1CCCC1NC(c1cc(-c2ccco2)[nH]n1)=O 29927,CCCC(O)(CCC)CC(C)NC(c1ccc(N2CCOC(C)C2)nc1)=O 29928,C1(C(=O)NCCc2ncsc2Cl)CCN(Cc2csc(Cl)n2)CC1 29929,N1(C(c2nncs2)C)CCC2(CN(C(=O)CCc3cccc(F)c3)C2)C1 29930,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)COCC(F)F)CC12 29931,n1(CCC)ccc(=NC(=O)C2CC(F)(F)C2NC(=O)C(F)(F)C(C)O)[nH]1 29932,C(CC(C(=O)N1CCC1CN=[N+]=[N-])NC(c1csc(C)n1)=O)OC 29933,C(=O)(C(CC(C)C)NC(=O)Cc1cccs1)NCC(CC)NC(C1CN(C)C1)=O 29934,c1(CCC)onc(C)c1C(=O)NCCCN(C(=O)C=CC(CC)=CC)C 29935,c1(C(=O)NCC2C(NC(CNC(=O)OC)=O)COC2)cc(C(F)F)nn1C 29936,C(=O)(C(C)(C)CN1CCOCC1)N(C1CCOC1)CCNC(C=CC)=O 29937,C(C(O)C(=O)N(CC(C)C(=O)NC(C1CCOC1=O)C)C)SC 29938,C(C(=O)NC(CO)C(C)NC(=O)CCCn1ccnc1C)(C(C)C)SCC 29939,N1(C(CC2N(CC)CCC2)=O)CCC(CN(C)C(c2coc(C(F)F)n2)=O)CC1 29940,N1(c2ccnc(C)n2)CC23CCCCC2(CN(C(C2(CC4CC4)CC2)=O)C3)C1 29941,N(C1CCc2sc(C)cc21)C(=O)NC1(OCC)CCC12CCC2 29942,c1(C(N(CC(CNC(Cc2cc(C)nn2C)=O)(C)C)C)=O)cc2n(c1)CCSC2 29943,C=C1CCN(C(=O)CC=CC)C(C(N2CCC(CO)CC2)=O)C1 29944,c1(C(CC)NC(CN(CCC)C)=O)noc(C(C2CCOC2)OC)n1 29945,C1(CC(=O)NCCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 29946,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 29947,C1(C(=O)NC2(c3ccccc3)CC2)(COC)CCOC1.C12CCCC1CNC2=O 29948,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(C(CNC(C(COC)(F)F)=O)F)CC1 29949,CCC(C)C(C(=O)NCC1CCCOCC1)N(C)C(c1ccncc1OC)=O 29950,c1(C(=O)NCC2CCCC(CNC(C3(N(C)C)CC3)=O)C2)cc(F)cc(F)c1 29951,N1(C(C(C)CN2CCOCC2)=O)CCCC(CCNC(C23CC(CO2)C3)=O)CC1 29952,C1(C(=O)NCC2(C(N3C(CCC#C)CCCC3)=O)CC2)CCOCC1(C)C 29953,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(C2CCCCN(C(=O)CSC(F)(F)F)C2)C1 29954,C(C1=NOC2OCCC12)NC(=O)CC1CCC=CC1O 29955,C1(C(=O)NC(CC#C)CCOC)CCN(C(=O)c2sc(C)nc2C)O1 29956,N1(C(C(C)OC)C(C)C)CCC(O)(CNc2ccccn2)CC1 29957,N1(C(C(C)SC)=O)CCCCC(CNC(c2cnoc2C)=O)C1 29958,C1(OC)CCCC1NC(=O)C(c1ccnn1C)OC 29959,CCCCCCCC(=O)N1CCCC1CN(C)C(c1cc2nnn(C)c2s1)=O 29960,C(=O)(CCC(=O)N1CCOC(C2CN(C(c3coc(C)n3)=O)C2)C1)NC 29961,c1(C(N2CCC(O)(CNC(c3nc(C)oc3C)=O)C2)=O)cc([N+](=O)[O-])ccc1N 29962,N1(C(=O)C2=C(Cl)CC2)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(CO)C1 29963,C1(C(N2CCN(C(c3c(C)onc3)=O)C(C(C)C)C2)=O)CCc2ncccc2C1 29964,Cc1ccc2nc(C(=O)NC(C)CC(C)NC(=O)C(=O)NCCC(N)=O)c(N)n2c1 29965,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 29966,c1(C(=O)NCCCC(C)NC(C2(OCC)CCC2)=O)c(C)nn(CC(F)F)c1C 29967,C1(NC(=O)Cc2cn[nH]c2)CCCCC1C(=O)NCCCCCCO 29968,N1(C(C2C(NC(CCCN=[N+]=[N-])=O)COCC2)=O)CCC12CCCCC2 29969,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc2c(Br)coc2cn1 29970,N1(C(CCCOC)=O)CCC2(CCC2)C(CNC(c2cncnc2C)=O)C1 29971,c1(C(N2CCC(O)(CNC(C3CC3(F)F)=O)C2)=O)nnn2c1CCCCC2 29972,Cc1cccc(CS(N2C3CN(CS(=O)(=O)CCc4ccccn4)CC23)(=O)=O)c1 29973,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 29974,C1(N(C(COCC)=O)C)CCC(NC(c2[nH]ccc2CC)=O)CC1 29975,Cc1cc(C(N2CC3CCC2C3NC(C2CCC2)=O)=O)c(N)c(F)c1 29976,C(CCC1CCC1)(C(=O)NCc1cccnn1)NC(C(C)CC1CCC1)=O 29977,CC(C)CC(C)C(=O)N(CC(O)CN(C(=O)COc1ccc(CO)cc1)C)C 29978,c1(C(=O)NCC2CCN(C(C34CCN(CC3)C4)=O)C2)ccc([N+](=O)[O-])[nH]1 29979,c1(C(=O)NC2C(CNC(CN(CCC#C)C)=O)C2)ncccc1OC 29980,C(CC1=CCN(C(c2ccc(C)c(C#N)c2)=O)CC1)NC(C(CC=C)OC)=O 29981,N1(C=O)CCc2ccccc21.CC1CC(C(=O)O)CN(C(=O)CN(C)C2CC2)C1 29982,N1(C(C(C)=CC2CC2)=O)CC(NC(C2CCCO2)=O)C(N=[N+]=[N-])C1 29983,C=Cc1ccc(C(N2CCC(CC)C2)C(=O)NCSc2ccccc2)cc1 29984,C1(NC(c2n(C=C)nnc2)=O)CC=C(C(=O)NCC23CCN(CC2)C3)C1 29985,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 29986,N1(C(c2n(C(C)C)ncc2)=O)CCCC(O)(CNC(C2CC(O)CN2)=O)C1 29987,CCC(CC(=O)NOCC(=O)NC1CCCC1c1ccc(O)cn1)C(C)(C)C 29988,N1(C(C=C(CC)CC)=O)CCC(N2CCC2)C1.C1CC(=O)N1CCCO.CCCO 29989,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 29990,c1(CNc2c(C#N)cc(Br)cc2)cnc2c(-c3ccc(C4CC4)s3)cccc2c1 29991,c1(C(N2CC(NC(c3ccc(O)nn3)=O)C3C2C3)=O)ccc2cnccc2n1 29992,C1(C)(NC(CCCN(C)C)=O)CCN(C(=O)C2=CCCC2)CC1 29993,N1(CC)CCCCC1C(=O)NCCNC(c1cnn(-c2ccccc2)c1N)=O 29994,N1(C(c2cccs2)=O)C2CCC1CN(C(=O)C(F)C1CCCC1)C2.O=C1CN1 29995,C(=O)(C(CN(C)C)C(C)C)NC1(CNC(CCc2cc(C)n(C)n2)=O)CCC1 29996,c1(OC)nc(C(=O)NCCC(=O)NCCOCC(F)(F)F)ccc1F 29997,c1(Oc2cccc(OCC)c2CO)ccc2oc(=O)oc2c1 29998,c1(C(=O)OCC)cnc(NC2CCCN(C(=O)COCCN(C)C)C2)nc1C 29999,N1(C(C(COC)OC)=O)CCC(C2CC2)C1CNC(c1cc(OC)ns1)=O 30000,c1(C(=O)NC(C)C(=O)NC2(C(=O)NC(C)C)CCOCC2)cccc(=O)n1C 30001,Cc1c(NC(C2CC3CC3N2Cc2cc(C(C)(C)C)on2)=O)cc(Br)cc1Cl 30002,CC(F)(F)C(C)(C)CNC(C1(NC(=O)COc2ccsc2)CCCC1)=O 30003,N1(C(C)C)CCCC1CC(=O)NCC(C)(C1CC1)NC(=O)CSC(F)(F)F 30004,Cc1cccc(C(=O)C(=O)N(C(C)CN(C)C(c2n[nH]cc2F)=O)C)c1 30005,C(C(C)(C)C(=O)NC(C)CS(C)(=O)=O)N(C(CCC1C(C)C1)=O)C1CC1 30006,c1(OC)ccc2c(C(=O)NC3CC(O)(CNC(=O)C(C)CF)C3)cnn2c1 30007,C1(C(C)(C)C)CCCC(CNC(N2CCCCC2Cn2ccnn2)=O)C1 30008,N1(CC(N2CC(O)(CCNC(CCCOCC)=O)C2)=O)OC(C)(C)CC1=O 30009,C#CCCCCCC(=O)N1CCCOC(CNC(=O)CCSC2CCCC2)C1 30010,C1(CC)CCCCC1C(N1CCCC1C1(NC(c2c(NC)c[nH]c2C)=O)CC1)=O 30011,CC1CN(C(c2nccn3cnnc23)=O)CCCN1C(C1(C)COC(=O)OC1)=O 30012,c1(SC)ncc(C#N)c(N2CCN(c3nc(C)cc(C#N)n3)C3CC23)n1 30013,c1(CCC(=O)NCC(C)CNC(c2cc(CC(F)(F)F)on2)=O)cccnc1F 30014,Cc1ccnc(C(=O)NCc2cc(C(=O)NC3CSCC3C)ccn2)c1N 30015,C1(CCCNC(C2(COC)CC2)=O)CCCN1C(=O)CC1(OC)CC1 30016,c1(CN2CCC(N(C(=O)CSCC(N)=O)CC)CC2)cc(OC)c2sccc2c1 30017,N1(C(c2occ(C)c2)=O)CC=CCC1C(=O)NC1CC(F)C1 30018,N1(C(c2cc(CC(C)C)n(-c3ccccc3)n2)=O)Cc2cccc3c2C(CCC3)C1 30019,n1(CC)ncc(C(=O)NCC2CCN2C(c2ccc(C)s2)=O)c1C 30020,CCC(CNC(C(C)(C)C)=O)N(C(=O)CNC(=O)Cn1cncn1)C 30021,c1(N2CCC(NC(=O)CCC3CCC(O)CC3)C2)nc2c(F)cccc2o1 30022,C=CCC(C)(CNC(=O)C(C)N(C)C(c1cc(C)n(CC)n1)=O)CO 30023,c1(CC(=O)NCC2(C)CCN(C(Cn3nnc(C)n3)=O)C2)c(F)cncc1Cl 30024,Cc1ccc(OCCC(=O)NC2CC2CNC(c2cn(C)cn2)=O)cc1C 30025,c1(C(=O)NCC2N(C(C(CCC)C)=O)CC(O)C2)cc2cnc(Cl)cc2s1 30026,c1(CC(=O)NC(CSC)CC(=O)O)c(Cl)cccc1Cl 30027,N1(C(=O)OC(C)(C)C)CCN(C(=O)C2=CCCN(S(C)(=O)=O)C2)CC2CCCCC12 30028,S(=O)(=O)(CCC(=O)NCC1CC(O)CN1C(c1cccc(=O)n1C)=O)N(C)C 30029,c1(CC(=O)NC(CC)CN(C(=O)CN2CCN(C)CC2)C)cnc2ccccn12 30030,N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCC1CC(N(C(=O)C(C)CC1CC1)C)C2 30031,C1(C(=O)NCC(C)(C)C)CNC(=O)C12CCN(C(c1cccc(Br)c1)=O)CC2 30032,C=CC1OCCC1N=c1[nH]c(N2CCCC(SCc3nccs3)C2)c(OC)c(Br)c1C 30033,N1(CCNC(=O)CCc2ccc(O)cc2)CCn2cccc2C1 30034,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30035,C1(C(C)O)CCN(C(=O)N(c2cc(Br)n(C)n2)C2CC2)CC1 30036,N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)(CNC(C2(O)COC2)=O)C1 30037,CCC(C)CCC(O)CC(=O)N1CCC(NC(=O)CC2CC=CC2)CC1C 30038,CC1CCN(C(=O)CCc2cnn(C)n2)CC1N(C)C(C1COC(C)(C)CO1)=O 30039,O(NC(=O)Cc1noc(CS(=O)(=O)C(F)F)n1)C(=O)CC1CCCO1 30040,Cc1cccnc1C(N1CCC(C)C1CNC(C12CC(C1)C(C)O2)=O)=O 30041,C1(C(=O)NCC2(NC(=O)CCc3ccc(F)cc3)CCOC2)CCCC12CC2 30042,c1(CN2C(CC)CN(c3nc(OC)cc(C)n3)CC2)cc(F)c(Cl)cc1O 30043,c1(C(=O)NCCCC2(CNC(CC=C=C)=O)CCCC2)c(C)cc(C)nc1O 30044,c1(C(=O)OCC)nn(C)c2c1CN(Cc1ccn(-c3nocc3CC)n1)CC2 30045,c1(C(=O)NC2CC(CCNC(c3cscn3)=O)C2)ccnc(O)n1 30046,c1(C(N(C(CN(C(C(C)OCC#C)=O)C)C)C)=O)cc(O)cc(C#N)c1 30047,C1(SC)CCCC1C(=O)NCCNC(=O)C(CC)SCc1ccccc1 30048,N1(C(Cc2c(C)nc(Cl)cc2)=O)CC2CN(Cc3ccc(F)cn3)CC2C1 30049,C(C(CCC)CCO)NC(C1(C#C)CN(C(C2COCCN2C)=O)C1)=O 30050,C1(C(=O)NC(C2CCN(C(C3(n4ccnn4)CC3)=O)C2)C)CCCCC(F)(F)C1 30051,CCC(C(=O)NCC1CC2(CC(NC(=O)C=CCOCCOC)C2)C1)C(C)C 30052,N1(C(C(C)CC(C)(C)C)=O)CCC(O)(C2(NC(=O)CCC3CCCC3)CC2)CC1 30053,C1(C2CC2)(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)CCC1 30054,c1(C(=O)NC2CCC(COC)C2)ncn(CC(=O)CNC(=O)C(F)=CC2CC2)n1 30055,N1(C(C2C(=C)C2)=O)CCC(CC)(NC(=O)CC(C)COC)CC1 30056,c1(CC(N2CCN(CCNC(COCC)=O)CC2)=O)ccc2c(c1)CCCS2 30057,C1(C)(C(=O)NC(CNC(C)=O)C(C)C)CCNC1.C(CCC=O)OC 30058,c1(NC(C2CC(NC(c3ccc(O)cc3)=O)C2)=O)ccc2sncc2c1 30059,Cc1cn(C)nc1C(=O)NC1CCN(C(=O)CC(c2cccs2)NC(N)=O)C1 30060,c1(C(CC(=O)NC2CCN(C(C=C(C)C(F)F)=O)C2C)O)nc2ccccc2[nH]1 30061,CC1C(C(=O)N(C2CCOC2)CCO)CCN1C(=O)C=CC1CCC1 30062,N1(C(=O)C2CC2)CCC2(CC1)CC(C(N1CCC(c3ccccc3)C1)=O)C2 30063,C=C(C)C(C)(C)C(=O)NC1CCC(N(C)C(c2ccccc2C(C)O)=O)CC1 30064,S(=O)(=O)(c1ccccc1F)NCC(=O)NC1C2CCC(C2)C1F 30065,c1(NC(C2CN(C(=O)C(C3CCCCC3)OCF)CC2F)=O)ccn2nccc2c1 30066,CC1CN(C(=O)C(C)(C)NS(C)(=O)=O)CCCN1C(C12CCC(CC1)CO2)=O 30067,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnn[nH]1 30068,C1(CN(C)C(=O)OC(C)=O)CCN(C(=O)Cn2ccnc2CC)CC1 30069,C(C(C)(C)C(=O)N1CCCCC1c1cncnc1)NC(C=C(C)c1ccco1)=O 30070,Cc1sc(=O)n(CC(=O)NC(C2CCCN2C(c2cc(Cl)ccn2)=O)(C)C)c1C 30071,C(C)(CO)(C(=O)NCCC(C)CCNC(=O)C(C)(C)c1cnn(C)c1)OC 30072,C=C(Cl)CC(C(=O)N=c1cc(C)n(C(C)C)[nH]1)NC(=O)C1=CC2C=CC1C2 30073,C(=O)(C1=NOC2(CCOC2)C1)NCCOCCNC(C1(c2c(C)c[nH]n2)CC1)=O 30074,CC1C(=O)NC(=O)CN1C(=O)C(Cc1ccccc1)NC(=O)OC(C)(C)C 30075,C1(Cn2c(-c3ccn(CC)n3)nc(N(C)C)n2)CC(F)(F)C1(C)c1ccccc1 30076,C(C(=O)N=c1ccn(CC(F)F)[nH]1)NC(C1CN(C)CCO1)C 30077,N1(C(CCC(C)OC)=O)CCC2(CCC(NC(=O)CCc3ccc[nH]3)C2)C1 30078,C1(CC)CCC(C(=O)NC23CC(NC(C4(C5COC5)CC4)=O)(C2)C3)CC1 30079,C1(CNC(C=CCC)=O)CC(CNC(=O)CCOC2CCC2)CO1 30080,C(=O)(C1CCC(=O)c2cccn21)NCC(C)(CO)N(C(=O)CNC(=O)C1CC1)C 30081,C1(NC(c2cc(C(C)C)nn2C)=O)CN(C(=O)C(=O)C(C)(C)C)CC(F)(F)C1 30082,C(=O)(C#CC1CCCC1)N(CCCN(C(=O)CCN1CCSC(C)(C)C1)C)CCO 30083,C(CCC(C)C)(C(=O)N1CCC(F)(CO)CC1)NC(C(=CC1CCCC1)C)=O 30084,C1(CC(=O)NCC(C2CCCCC2)NC(C2CCOC2=O)=O)CCCS1(=O)=O 30085,C(=O)(C(F)C(C)CNC(=O)C(=C1CCCCC1)F)N(C(C)C(=O)OC)CC 30086,c1(C(=O)NC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)n[nH]c2ccc(F)cc12 30087,N1(C(c2ncn(C)n2)=O)CCOC2CN(C(=O)CC3CCC(C)(C)O3)CC12 30088,c1(C(=O)NCCC2(C(=O)NC(C)Cc3ccnn3C)CCC2)ncccc1N 30089,N1(CC)CC(C(COC)NCCCCC(C)NC(=O)Cc2c(C)n[nH]c2C)CC1=O 30090,S(=O)(=O)(c1ccc(C#N)c(N2CCC3CC23)c1)N1CCCC(=C)C1 30091,c1(C(=O)NCC2CC(OC)CN2C(C2CC(C)=NO2)=O)ncc(C)cc1F 30092,c1(C(=O)NC2(CNC(C3COCC(C)(C)O3)=O)CCOC2)ccn2cccc2c1 30093,c1(C(=O)NCC2(NC(c3nn[nH]c3C(F)(F)F)=O)COC2)cccc(Cl)c1F 30094,c1(C(=O)NC2CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30095,CC(C)CC(C(=O)NC1CC2CC(CNC(=O)Cc3ccsc3)C1C2)C(N)=O 30096,C(=O)(C(C(=O)C1(COC)CC1)NC(=O)CCN(CC(C)(C)C)C)OCC.CCOC 30097,C1(C(C)O)CCC(NC(N2CCC(F)(c3ccccc3Cl)C2)=O)CC1 30098,N1(C(C2N(C(CN3CCN(C)CC3)=O)CCOC2)=O)CC2(CNC(=O)N2C)C1 30099,c1(OC)ccc2nc(N3CCC(N(C(=O)Cn4cc(Br)cn4)C)C3)sc2c1 30100,N1(C(c2ccc(OC)cn2)=O)CC2(CCCN(C(c3cc(O)nn3C)=O)C2)C1 30101,C1(COC)CN(C(=O)Cc2cncc(F)c2)CCN1C(=O)CC(C)n1cccn1 30102,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30103,c1(N2CCC(COCC)C2)ncc(C)cc1S(=O)(=O)N1CCC(C(C)O)C1 30104,C(=O)(C1=CC(O)CCC1)N1C(CN(C(=O)CCCC2CCOCC2)C)COCC1 30105,Cc1ccc(C(C(=O)NC2CNC2)N(C2CCC2)C2CCC2)cc1C 30106,N1(C(CCCOCC)=O)CC2(COC)CC1(CNC(c1ocnc1C(C)C)=O)C2 30107,N1(C(C=CCCC(C)C)=O)CC2CCC2(CCNC(C2CN(C(N)=O)C2)=O)C1 30108,C1(NC(c2nc(C#C)sc2)=O)CS(=O)(=O)CC1NC(=O)CC1(N(C)C)COC1 30109,C1(OC)CC2CCC(N2)C1COC(N1CC(C)(C)C1C1CC1)=O 30110,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CCN(C)C1 30111,C1(CNC(c2ccc(Cl)cn2)=O)CC2COCC2N1C(=O)CCCN1CCC1 30112,N1(CC)C(=O)CCC1C(=O)N(C)CCN(C)C(c1c[nH]c(=S)cn1)=O 30113,CC1CCCN(C(c2cnn(C(F)F)c2)=O)C1CCNC(c1nccnc1N)=O 30114,CC1=C(C(=O)NC2CCCC2(C)CNC(=O)CC(C)(C)C)C(C)n2nnnc2N1C 30115,C(=O)(CC(CC)C(F)F)N(CCC(=O)NCc1nc(C)c(C)o1)CC=C 30116,C(=O)(C1=CCN(C)C1)NC(CCSC)C(=O)NCC(CO)C1CC1 30117,c1(C(N2C(CNC(c3c(CCC)cccc3)=O)CCC2)=O)ccc2cncn2c1 30118,c1(OC)ccc(-n2nnc(C(=O)NOCC(=O)N(C)C(C)C)c2C)cc1 30119,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)CCCn2cncn2)C(F)C1 30120,c1(C(N(C2C(OC)COC2)C)=O)ccnc(CNC(=O)C(CSC)OC)c1 30121,C#CCCCCCCOC(=O)CC(c1cccc(NC(=O)OC(C)C)c1)=O 30122,c1(C(C2CC2)NC(=O)CNC(c2cccc(OC(F)(F)C(F)F)c2)=O)cccc(I)c1 30123,N1(C(CN2CC(C)(OC)C2)=O)CC(CN(C(=O)C=C(C)C(C)C)C2CC2)C(C)C1 30124,c1(C(N2CC(N(C(=O)CC(C)(C)C3CC3)CCC)C2)=O)ccc2c(c1)CCC2 30125,N1(C(N(CCOC)Cc2cccc(F)c2)=O)CCCC(c2nc(=N)[nH][nH]2)C1 30126,c1(CC(=O)NCC(CC=C)NC(c2ncc(C)cc2C)=O)csc2ccccc12 30127,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30128,C1(C(N(CC(=O)OCC)C2CCC2)=O)(CC2CCCCO2)CCCCO1 30129,C1(NC(=O)CCCc2ncco2)CN(C(c2[nH]ccc2C2CC2)=O)CC12CC2 30130,N1(C(C2C(C)=NOC2=O)=O)CCCCC(CNC(=O)C(C)Cc2ccccc2)C1 30131,C1(C(C)NC(c2c(C)c[nH]n2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30132,C(C(CC(F)(F)F)NC(c1ccncc1NC)=O)NC(=O)CN1CCC(O)CC1 30133,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30134,N1(C(c2ncc(C)s2)=O)C2CC1CN(C(=O)C(C)Cc1ccccc1)C2 30135,N1(CC(C)C)CCC(C(=O)N(C)CCN(C(=O)CCC2CNC(=O)C2)C=O)C1 30136,C1(NC(CCCN(C)C)=O)CC=C(C(=O)N(C2(N(C)C)CC2)C)C1 30137,C1(C(N(C(C)C(N2CCC(CN=[N+]=[N-])C2)=O)CC)=O)CCOC1(C)C 30138,C1(NC(c2c(N)cncc2)=O)CC(NC(c2coc(Cl)n2)=O)C12CCC2 30139,N12CC(CC1=O)C(=O)N1CC2C1.C1(F)(C(=O)NCC(NN(C)C)=O)CCCOC1 30140,CC1C(C=CC(N2CCCC2CCNC(C2CN(C)C2)=O)=O)C1(Cl)Cl 30141,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CCC3)[nH]c12 30142,N1(C(c2ccc(OC)c(OC)n2)=O)C2CCC1CC(NC(C1(C)CCCO1)=O)C2 30143,c1(C(C)(O)CNc2cn(C3CCNC3)nn2)cccc(O)c1 30144,c1(C(=O)NC(CNC(c2c(C)nncc2)=O)(C)C(C)C)ncc(C#N)cc1Cl 30145,CC12COC(=O)N1CCN(N1CCN(Cc3ccccc3)CC(C(=O)OC)C1)C2 30146,c1(NC(C2CCS(=O)(=O)C2)=O)cccc(-c2ccccn2)c1Cl 30147,Cc1cc(C(=O)NC2COCCC2NC(C2CC(C)OC2C)=O)cc(O)c1 30148,Cc1cnc(F)cc1C(N1CC(CNC(=O)C(C)NC(c2ccccc2)=O)C1)=O 30149,N1(C(C(C)c2ccco2)=O)CCC(C)(C(N2CCC(CCCO)C2)=O)C1 30150,C1(C(=O)NC(CC#C)C(=O)NCCCn2cnnn2)CC2(CCO1)CC2 30151,c1(OC)ccccc1NC(C1C=CC(NC(c2csc(Br)c2)=O)C1)=O 30152,C(=O)(CCC(=O)NN(C)C)NC(C1C(C(=O)NCC(CCC)C)C1)C 30153,C1(COC)(NC(C2CC3CC2CC3O)=O)CCN(C(c2csc(SC)n2)=O)CC1 30154,n1(CCCSCC)nnnc1C(C1(CC#N)CC1)NCCC1C=CCC1 30155,C1(NC(c2c(CC)nc(C)n2C)=O)CCN(Cc2cncn2C)CC1(C)C 30156,N1(C(C2(CS(C)(=O)=O)CCC2)=O)CCc2ccc(F)c(F)c2C1(C)C 30157,N1(CC2=C(C)CC2)CCC(=O)N(CC2CN3CC4CC3(CO2)C4)C1=O 30158,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)C(n2ccc(C(F)F)n2)C)C1 30159,N1(C(C(=O)Nc2cccc(CC)n2)=O)CCCc2ccc(O)cc2C1 30160,C(=O)(C(C)(C)C(C)O)NCc1cccc(CN(C(CC(C)O)=O)C)c1 30161,C(Cn1cccn1)(C(=O)N1CCCCCO1)NC(C12CC(CO)(C1)C2)=O 30162,CCC(COC)C(=O)N(C(C)CN(C)C(c1cc(Cl)cnn1)=O)C 30163,CCCCCC(O)CC(=O)NCCCC1CCCCN1C(=O)C(CC)SC 30164,C1(C(N2CC(NC(=O)C(n3cc(Cl)cn3)F)C2)=O)CC2CCCCCN2C1 30165,C1(C(C)C)CCN(c2cc(N3CCOC(c4nncn4C)C3)ncn2)CC1 30166,C#CC1(C)CCCN(C(=O)C(CC(=C)C)NC(c2cc(C3CC3)[nH]n2)=O)C1 30167,C1(CNC(c2[nH]cc(C)c2)=O)COCCN(C(=O)Cc2csc(NC=O)n2)C1 30168,C(=O)(C(C)(C)CCSC)N1CCCC(CN(C(C=CCN(CC)CC)=O)CC)C1 30169,CC(C)N=C(NCC(C)Oc1ccccc1)NC(C1CC(N(C)C)CN1C)C 30170,c1(CC)ccc2c(c1)CN(c1nnc(-c3ncc[nH]3)n1CCC#N)CC2 30171,c1(C(N(C2CCN(C(=O)C(C)(C)C)C2)C)=O)nn[nH]c1Cl 30172,Cc1ncc(Br)c(C(=O)NCC=CCNC(C2CC2C(C)C)=O)n1 30173,Cc1cccnc1C(=O)NCC1CCN1C(=O)CC1CCC(C)(C)C1 30174,c1(C(C)C)ccc(-n2cc(-c3c[nH]nc3CN(C)C)nn2)cc1 30175,N1(C(c2cnc(CC)s2)=O)CCCCC(NC(=O)C(O)CC2CCOCC2)C1 30176,c1(C(N(C)CC2N(C(C3=NOC(C)C3)=O)CCC2)=O)c(O)cc(Cl)cc1O 30177,C1(CC(=O)NCCCNC(=O)C=CC2CC2)CCCCC1O 30178,c1(C(N)=O)cc(C(N2CCC(F)C(NC(C3OCCOC3(C)C)=O)C2)=O)ccc1Cl 30179,C(=O)(CCCCC(=O)NC(CNC(=O)Cn1cc(Br)cn1)C1CC1)NC 30180,c1(NC(C2CC3CC3N2C(C2CCCCCC2)=O)=O)ccc2c(O)n[nH]c2c1 30181,N1(C(c2c(CC)csc2)=O)C2CCC1CN(C(c1ccn(CC)c(=O)c1)=O)C2 30182,c1(C(=O)OC)cc(Cl)nc(Cl)c1NC(C1(C)CCN1Cc1cscn1)=O 30183,c1(C(=O)NCC2CCCN2C(C23C=CC(CC2)C3)=O)ccc2c(c1)COC2=O 30184,C(=O)(C(F)C1CCC1)NCCN(C(=O)CCC1CC1(Cl)Cl)CCC 30185,N1(C(CSCC=C)=O)CCCC(C)(CC(=O)NCc2scnc2C(=O)OCC)C1 30186,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30187,N1(C(C2(C(C)C)COC2)=O)CC2(C1)CN(C(=O)CC1(CO)CC1)CC2CO 30188,c1(CC#N)cccc(C(=O)N(C23CC(C(c4scnc4C(F)(F)F)=O)(C2)C3)C2CC2)c1 30189,C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC(=O)NC)C2)CCC(O)CN1C 30190,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC(F)C(NC(C2(F)CC2(C)C)=O)C1 30191,C1(NC(C(C)CN2CCOCC2)=O)CCN(C(=O)CC#N)C1C 30192,C1(CN(C(C(C)N(C)C)=O)C)CN(C(=O)C(O)C2CCCC2)CCO1 30193,C1(N(C(c2ccsc2C)=O)CC)CCN(C(c2ncoc2C)=O)C1 30194,N1(CCCNS(C)(=O)=O)CCN(C(=O)COCC2CCCN2C)CC1 30195,N1(C(C(CC)F)=O)CCC2CC(CNC(=O)CCCc3csc(C)n3)CCC2C1 30196,C1(CCOC)CCCCN1C(c1cncc(Cl)c1)C(=O)Nc1ccc(OC)cc1 30197,Cc1ncc([N+](=O)[O-])n1CC(N1CC(O)(CN(C(=O)CCC(F)(F)F)C)C1)=O 30198,c1(-n2c3nc(n2)-c2ccc(nc2)S3)ccc(F)cc1-n1nccn1.C(C)(C)OC 30199,C1(NC(C(CC(=C)C)OC)=O)CN(C(=O)C(C)SC)CC1S(C)(=O)=O 30200,N1(c2ncc(OC)c(C)n2)C2CCCC1CC(CN1CCC(OC)CC1)C2 30201,c1(-c2ccc(NC)s2)cn(C)nc1C.N12CCCC1C2C(=O)NC(CC)C 30202,CC1C(C=CC(=O)NCC=CCNC(=O)CCC2(C#N)CCC2)C1(Cl)Cl 30203,N1(C(c2cc(CC)no2)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1CC(F)(F)F 30204,CC1CN=C2NC(C(=O)N3C4CCC3CN(C(C3(CF)COC3)=O)C4)=NN2C1 30205,C(C1=CCN(C(C2CCC(C(N)=O)CC2)=O)CC1)NC(c1nnn(C)n1)=O 30206,Cc1cc(C(=O)NCCC2(NC(=O)Cc3cc(C)cs3)CCC2)c(C)[nH]1 30207,CC(C)(C(=O)NC1CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1)C(F)F 30208,c1(N(CCC(C)(C)C(=O)OC(C)(C)C)C(=O)NCC=CCC)ccc(Cl)cc1 30209,c1(C(=O)OC)cnc(C(=O)NCCC2(CNC(c3nsnc3O)=O)CC2)cn1 30210,C(=O)(C1=CCCSC1)N1CC(CCC=C)(C(=O)NC2CCC3(CC3)C2)C1 30211,CC1C(C(N2CCN(CC3(C(=O)NC4(CO)CC4)CCCO3)CC2)=O)CCN1C 30212,c1(C(C)C)nc(CC(=O)NCC2CCN(C(C3CC3C3CCCCO3)=O)C2)cs1 30213,C1(C(=O)NC2(CNC(CNS(C)(=O)=O)=O)CC2)CC12CCC1(CC1)CC2 30214,c1(C(=O)NCc2c(C(=O)NC(CC=C)C3CC3)nco2)cccc(Cl)c1 30215,c1(C(=O)NC(CNC(CCOCC)=O)(C)C2CC2)ccc(C2(C#N)CC2)cc1 30216,C1(NC(CSc2n(C)ccn2)=O)CCC12CN(C(c1cnc(Cl)cc1N)=O)C2 30217,c1(C(=O)OC(CCC(=O)OCC)C(=O)O)cc2ccc(OC)cc2o1 30218,C(=O)(C(C)Cc1cn(C2CN(C(c3cn(CC(C)(C)O)nn3)=O)C2)nn1)OCC 30219,CCC(C)C(C(=O)NC1CCCCC1CC(=O)Nc1cnn(C)c1C1CC1)SC 30220,c1(SC(C)C(=O)NC2C3CC2N(C(=O)C2=CCCC2)C3)ccc(Cl)cc1 30221,C=CCC(C(=O)NCC1(O)CCN(C(c2ncoc2CC)=O)C1)C(C)C 30222,CC(C)(O)C(F)(F)C(=O)NCC12CC1CN(C(c1ccc3nncn3c1)=O)C2 30223,c1(C(=O)NC2C3CN(C(CC=CCC)=O)C2CC3)cc2c(F)ccc(F)c2s1 30224,c1(C(=O)OC)ccc2nc1OC(=O)C(=O)N2C.C(C)(C)(C)OC(C1CC1)O.C1CC1 30225,c1(-c2nc(CCS(=O)CCN3CCOCC3)on2)cccc(F)c1F 30226,c1(C(=O)NCC2N(C(C(C)CO)=O)CCC2C)cnc2c(c1)CCCO2 30227,N1(C(C2CC3C=CC2C3)=O)CCCC(C2CN(Cc3c(F)cccc3F)C2)C1 30228,CN1CCCCC1CS(=O)(=O)NC1CCN(c2cccc(C(=O)O)c2)C1 30229,c1(C(N2C(C(=O)NC3CCC(O)CC3)CCCC2)=O)cn2ncccc2n1 30230,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30231,C(=O)(CC(F)(F)C(F)F)N1C2C(N(C(c3nnn(CC)c3C)=O)C)CC(C2)C1 30232,C1(C(N(C2(CC)CC2)C)=O)CCN(C(=O)Cc2csc(Cl)n2)C1C(C)C 30233,C(=O)(C1=C(C)OCCC1)N1C(CC)CN(C(C2(C)CC=CCO2)=O)CC1 30234,C1(OC)CC(CCNC(C2(C)CC2(Cl)Cl)=O)N(C(=O)CCc2nccn2C)C1 30235,C1(OC)(CNC(=O)C(C)N2CCCC2)CCN(C(=O)COc2cc(C)on2)CC1 30236,C1(CCNC(CC(COC)C)=O)C(C)CCCN1C(c1cc(=O)c(OC)co1)=O 30237,c1(C(=O)NCCN(CCC2NC(=O)NC2=O)CC)ccc2c(c1)C(C)(C)CO2 30238,C1(C(N2CCC(C)(NC(CC3C(C)(C)CO3)=O)CC2)=O)C2Cc3ccccc3C12 30239,C1(NC(Cc2nc(C)oc2)=O)CCC2CN(C(C3(n4ccnc4)CC3)=O)CC2C1 30240,NC(CSC(F)F)CC(=O)NC(CNCC(F)(F)F)CO 30241,CC(C)C(C)(O)C(=O)NCCOCCNC(=O)CN1C(=O)CCCC1=O 30242,c1(OCC(=O)NCCC(C)NC(=O)CC2CC23CC3)ccc(Cl)c(F)c1 30243,c1(CN(CCCCCC)C(c2ccc(Cl)cc2)C)cc2c(c(Br)c1)O2.OC 30244,O=C(NNc1cccnn1)Nc1cccc(Oc2ccc(Cl)cc2F)c1 30245,C1(C(C)(C)CNC(=O)NCCc2ccc(I)o2)CCN(C(=O)OC(C)(C)C)CC1 30246,C1(C)(C(=O)NCC23OCC(CNC(c4c(CC)noc4C)=O)(C2)C3)CCC(F)(F)C1 30247,C1(OC)CN(C(c2ccc(OC)c(OC)c2)=O)CCC1NC(=O)CS(C)(=O)=O 30248,C1(NC(C(C)F)=O)CCOCC1c1ccc(Br)cc1 30249,C1(C(=O)NCCC(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)N(C)C)CC1 30250,C=C(Br)CN=c1ccc2cc(CC)ccc2[nH]1 30251,C(=O)(C(F)C1CCOC1)N(CCNC(C(C1CC1)OCC)=O)C 30252,CC1CN(C)SCC1N(C(=O)N(CCn1ccnc1)C1CC1)C1CC1 30253,c1(C(N(C(C(=O)NCCOCC#C)C)CCC)=O)coc(OC)n1 30254,C(=O)(CCCCN=[N+]=[N-])N1CC(C)N(C(c2cc(-c3cccnc3)[nH]n2)=O)CC1 30255,CN1CCC(CCNC(c2ccc(CNC(C3CCC3C(N)=O)=O)s2)=O)C1 30256,c1(CC(C)C)cccc(C(=O)OC2CCCN(C3CCN(C)C3=O)C2)c1 30257,C12CCN(C1(C)C)C2=O.c1(NC(CCN(C)CC)=O)cc(OC)ccn1 30258,N1(C(C2C(CNC(CC3=NNC(=O)C3)=O)CCC2)=O)CC(O)CC12CCCC2 30259,C#CCCCC(C)NC(C1CC1c1ccccc1Nc1ccccc1)=O 30260,N1(C(CC=C)=O)CC2C(CN(C)C(C3(c4ccccc4F)CC4(CC4)C3)=O)C2C1 30261,Nc1ccc(C(N2CCN(c3ccc(Br)cc3-c3nn[nH]n3)CC2)=O)nc1F 30262,C1(CN(C(=O)Cc2ccc(Cl)nc2)C)CC(F)CN1C(=O)C(F)OC(F)(F)F 30263,c1(C(=O)NCCc2ocnc2CNC(C2CC23CC3)=O)cc(O)cc(O)n1 30264,Cc1cc(=NCc2cscc2Cl)[nH]c(N2CCCC(CS(C)(=O)=O)C2)n1 30265,C=CCC(C(=O)NC(C)CNC(=O)C(c1ccc(Cl)nc1)(C)C)C(C)(C)C 30266,N1(C(CC(C)F)=O)C(CC(=O)NC23CCC(C2)OC3C)C2CCCC12 30267,c1(C(C(=O)NCC(C)NC(=O)Cc2ccccc2F)=O)c[nH]c2ccccc12 30268,c1(NC(C)=O)ncnc(Nc2cc(-c3cccc(OC(C)C)c3)no2)c1F 30269,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1Cc1nc(Br)cn1C 30270,C1(NC(CC=C)=O)CN(C(=O)C(c2c(Cl)cccc2Cl)C)CC12COC2 30271,N1(C(CCCOC(C)(C)C)=O)CCC2CCN(C(=O)C=Cc3ccsc3)CC12 30272,c1(C(N2CCN(c3ncnc(CC)c3F)C(C(C)C)C2)=O)cc(S(C)(=O)=O)co1 30273,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(C1C(C)(C)C1(C)C)=O 30274,C1(C#N)(Cc2nn(-c3ccn(CC)n3)c(C(F)F)n2)CCOCC1 30275,N1(C(C2C(C)SCCC2)=O)CC(CC(=O)NCCc2ccon2)C2(CC2)C1 30276,Cc1cncc(C(=O)NC2CCC(NC(C3CC(=C4CC4)C3)=O)CC2)c1C 30277,CCC(CCO)CN=c1nc(N2CCC(C3CCCC3)CC2)c2c([nH]1)CCCC2 30278,CC1(C)CCC(C(=O)NOC(=O)C=Cc2cc[nH]n2)CN1Cc1cccnc1 30279,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(=O)CCN(C1CCCCC1)C 30280,c1(C(N2C(C(=O)Nc3ccc(C)nc3)C=CCC2)=O)ccc2c(c1)CCC2 30281,C12(NC(c3cnc4n3CCS4)=O)CCCCCC1N(C(C1(F)CCC1)=O)CC2 30282,c1(C(N2CCC(C)(NC(=O)CCC3CCCO3)C2)=O)[nH]c2ccccc2c1Cl 30283,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30284,N1(C(COC(C)C)=O)CC2C(CN(C(=O)CCSCC(N)=O)C)C2C1 30285,Cc1cc([N+](=O)[O-])ncc1C(=O)NCC1CCCN1C(=O)C=Cc1cn[nH]c1 30286,c1(OC)cccc(C(CCNC(=O)C(N2CCCCC2c2ccccn2)=O)OC)c1 30287,c1(-c2nc(C(CC)C)nn2C23CCCC2C3)ccc(Cl)c(S(C)(=O)=O)c1 30288,N1(C(C=CS(C)=O)=O)CCN(C(c2cc(C(N)=O)cs2)=O)CC1C1CCCC1 30289,c1(NC(c2ccc(-n3cncn3)cc2)=O)cccc(OCCC2CCOC2)c1 30290,Cc1nn(C2CC2)c(C)c1C(N1CCCC(NC(=O)CC(F)(F)F)C1)=O 30291,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30292,c1(CC(=O)NC2CCC(CNC(=O)C(F)(F)C(O)C3CC3)C2)ccc2c(c1)COC2 30293,C1(N(C(C2(C(=O)OC)C(=C)CC2)=O)CC)CCCN(C(=O)COCC(F)(F)F)CC1 30294,C(=O)(CC(C)CC(=O)NCCC(O)CNC(=O)CNc1ccc(CO)cn1)OC 30295,c1(C(=O)NC(C(=O)OC)C2CCOC2)cc(F)cc(F)c1.C12CCN(C1)C2=O 30296,c1(N2CCC(C(C)C)CC2)[nH]c(=NCC23CC2CN(C)S3(=O)=O)nc2sccc12 30297,C1(C(=O)NCCCNC(c2nc(C)oc2C)=O)CCOC2(CCC2)C1 30298,N1(C(C(CN(C(c2ccc(C)cc2)=O)C)C)=O)CCCC(C(N)=O)C1C 30299,c1(C(N(CCNC(CC(CCC)(C)C)=O)C2CC2)=O)c(F)ccc2nc[nH]c12 30300,N#CC1(CO)CC12CCN(C(=O)NCc1ccc(C(N)=O)cc1)CC2 30301,c1(C(N2CCCC(NC(C3C(C#C)C3)=O)C2)=O)ccc2c(c1)nc(O)n2C1CC1 30302,C1(CC(=O)NCC(CCC)C)CC(C)(C)CN1C(c1ccc(C#N)[nH]1)=O 30303,CCC(C)(CNC(C1(CO)CCN(C(=O)CSC)C1)=O)CO 30304,C1(NC(c2ccc([N+](=O)[O-])s2)=O)CC2CCC1N2C(=O)C#CC1CCC1 30305,CC(C)(C(=O)NC(Cn1ccnn1)C(=O)NCCc1cnco1)C1CCOC1 30306,C(=O)(CC(C)C(F)(F)F)NCC1N(C(C2=CCCC2C)=O)CC(F)C1 30307,C1(C(N2CCC(NC(c3cnc(C)[nH]3)=O)C2)=O)CCC(C)(C)CO1 30308,C(C(CC(F)(F)F)NC(=O)CC(Cc1ccccc1)CC)NC(COCCC)=O 30309,C1(CCC(=O)NCC2CCC23CCC3)CCN(C(C2COC(=O)N2)=O)CC1 30310,CC(C)(CS(N)(=O)=O)C(=O)N1CC(CNC(C2CC3(C2)CC3F)=O)C1 30311,C(=O)(C1CCCc2nccn21)N(CCN(C)C(c1nc2ncccn2n1)=O)C 30312,C1(NC(CC(=O)OC)=O)CCC(N(C(=O)C=CBr)C)CC1 30313,S(=O)(=O)(c1cc(C)cnc1NCCCSC)N1CCCC(CC)C1 30314,Cc1cc(=NCC2(CNC(=O)Cc3c(O)ncnc3O)CCC2)[nH]c(C2CC2)n1 30315,C(=O)(CCCCCCNC(=O)COCc1ccccc1)N(c1ccccc1F)C 30316,c1(C(N2CC3C(C(=O)Nc4cnn(C(F)F)c4)(C3)C2)=O)ccc(F)c(F)c1Cl 30317,Cn1ncc(C(=O)NCCNC(C2COC(C)(C)C2)=O)c1C#N 30318,CC1CC(C(N2CCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCNC(=O)CO)C1 30319,c1(C(N2CCC(O)(CNC(C(CC=C)(F)F)=O)C2)=O)[nH]c2c(Cl)cccc2c1C 30320,C1(C(N2CCN(Cc3ccc(Br)cc3)CC2)=O)CC2CC2N1Cc1cnco1 30321,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30322,CC1CCC(C)N1CC(=O)N(CCCCN(C(=O)Cn1cc(C(N)=O)nn1)C)C 30323,C1(C(N2CCC(OC(C)C)C2)=O)CC(O)CN1Cc1ccccc1C(C)C 30324,c1(C(CC(=O)NCC(C)NC(=O)CC2CCN(C)C2=O)C)ccc(Cl)cc1 30325,C(C(N=c1nc(C2CCCCC2)[nH]s1)c1ccccc1)NC(CCC(=C)C)=O 30326,N1(C(C2CC(OC)(OC)C2)=O)CCC(C2CCCN2CN2C(=O)CNC2=O)CC1 30327,c1(C(=O)NCC(C)(C)NC(c2c[nH]nc2Cl)=O)ccc(C(F)(F)F)s1 30328,C1(CNC(C(C)OCC)=O)(CNC(C2CC=CC2)=O)CC12CCC2 30329,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30330,C(=O)(C(C)(C)CO)NCC(CC)(C)NC(=O)CC1(c2ccccc2)CC1 30331,c1(C2CCCCC2)cncc(C(=O)NC(c2cc(C)[nH]n2)c2nnnn2C)c1 30332,c1(-c2c(C(N3C(CNC(COC)=O)CC3)=O)nccn2)ccc2c(c1)CCO2 30333,c1(C(=O)NCC2(C(C)NC(C3=CCCC3C)=O)CC2)ccc(F)cc1[N+](=O)[O-] 30334,C1(CN(C(CCN(C(c2nccn2CC)=O)CC)=O)C)CCOC1C 30335,c1(C(=O)NC2CCCN(C(CC=CC=C)=O)CC2)nc2ccccc2nc1C 30336,CC(C)(C(=O)NCCCC(=O)NCC1CCCC1N(C)C)c1ccno1 30337,C(C(C(=O)NCc1ncc(CO)s1)NC(=O)C=CC(F)F)N(C)C 30338,N1(CC(C)NC(C(CC)OC)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 30339,C12(C)CCC(CC1)NC2=O.CCC(CN(C(=O)CCc1cccs1)C)OC 30340,N1(C(C2(c3cccc(F)c3)CCOCC2)=O)CCC(NC(C2(O)CC2)=O)C(F)C1 30341,C(C)(CCCC(=O)NCC1CCC(O)C1)NC(C(c1ccn(C)c1)C)=O 30342,c1(C(=O)NC(C(C)NC(CCCN(C(C)=O)C)=O)C(C)C)scc2c1OCCO2 30343,C(=O)(CC(C)CC(=O)NC1CCN(C(c2cnc(CC3CC3)s2)=O)CC1)OCC 30344,C(C(N=c1[nH]nc(C#N)s1)C(C)C)NC(c1cc(OC)c(F)c(F)c1)=O 30345,C12(NC(=O)CSc3ccccc3)CCC1CN(C(c1cccnc1)=O)C2 30346,N1(C(C2CC2C(F)(F)F)=O)CCOC2(C1)CN(C(C1CCCC1)=O)C2 30347,N1(C(C=CCNC(C(C)c2cc[nH]n2)=O)=O)CCCC(C)C1CCO 30348,C(=O)(C(C)CC(F)F)NC(C(=O)NCCc1cnc(C)[nH]1)CO 30349,CC1CCN(CC2CCCC(=O)N2)CC1NC(c1ccsc1-n1cnnn1)=O 30350,C12(C(=O)NC(CNC(c3nc(OCC)oc3)=O)(C)C)CCCCC1C2 30351,CC1CCC(NC(=O)CCc2cnccn2)CN1C(=O)CSCCN(C)C 30352,c1(NC(C2(NC(COCC#C)=O)CC2(C)C)=O)ccc2ccoc2c1 30353,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cocn1)OC)OC 30354,N1(C(c2cn(CC=C)nn2)=O)CC(F)CC1CNC(=O)Cc1csc(S)n1 30355,N1(c2cc(OC)ncn2)CCC(F)(F)C(CNC(c2ccc(C)s2)=O)C1 30356,CC1CCN(C(=O)CC2N(C(=O)CN3CCSCC3)CCC2(C)C)CC12CCC2 30357,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30358,C(CCCCC(=O)N1CCN(C(C2CC3(C2)CC3F)=O)CC1CO)OC 30359,c1(CC)ccc(CCC(=O)NC(C)C(CO)NC(=O)COC(C)=O)cc1 30360,c1(C(N(CC(=O)NC2C3(CC(OCC)C3)C2)CC(C)C)=O)cn2c(n1)CCC2 30361,C1(CNC(=O)Cc2cncs2)C=CC(NC(c2coc(C(F)(F)F)c2)=O)C1 30362,Cc1cnn2cc(C(N3CC(O)CC3c3ccc(F)cc3)=O)cnc12 30363,CC1CN(C(=O)CCSC2CCCC2)CCCN1C(C1CSCCS1)=O 30364,C1(OC)CCCCC1C(=O)NCc1cccc(CNC(=O)COC2CCOC2)c1 30365,C1(CNC(c2c(OCC#C)nccc2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)O1 30366,N1(C(c2c(CC)nn[nH]2)=O)CC2(CCC2)CC1CNC(=O)CSc1cccs1 30367,c1ccc(Cl)c(C)c1.C(=O)(CCS(C)=O)NC1(CO)CC(OC)C1.C1(=O)CO1 30368,c1(C(=O)NC2CCCN(C(C(CCC)C)=O)CC2)ccc2nc(CC)cn2c1 30369,c1(N2CCN(c3cc(NCCCSC(F)F)ncn3)CC2)cc(N)ccc1N 30370,C1(C(N(C2CN(C(=O)Cc3nc[nH]n3)C2)C)=O)CC2CCC(C1)S2(=O)=O 30371,N1(C(C2(NC(C(CC)C)=O)CCCC2)=O)CC(O)CC1(C)C 30372,N1(C(CCCCOC)=O)CC2(CCN(C(=O)CN3CCNC3=O)C2)C1 30373,N1(C(CCN(CCC)C)=O)CC(NC(c2ccc(=NC)[nH]c2)=O)CC(C)(C)C1 30374,C(C(C(=O)NCCc1cn[nH]c1)C(C)C)NC(C1CC(CCC)C1)=O 30375,C(N=c1cc(C(C)C)nc[nH]1)C1CN(C(C(C=C)O)=O)C(C)C1 30376,c1(C(C)=O)cncc(OCCN(CCNC2(C(=O)OCCOC(C)=O)CC2)C)c1 30377,Cc1cnnc(O)c1C(=O)NCC1CC1CC(=O)N(CC1=CCCOC1)C 30378,c1(C(C(=O)NC)N(C)Cc2cn(C)cn2)cc(OCCO)n(C)n1 30379,C(=O)(C1=NOC2(CCC2)C1)N1CC(CCCCNC(=O)C2=COCCC2)C1 30380,N1(C(c2c(N)non2)=O)CCN(C(c2ccn3cccc3c2)=O)CC12CCC2 30381,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(=O)Cc3nc(CO)cs3)C2)OC1 30382,c1(C(=O)Nc2cn(C3CCC(C(N(CC(C)C)C4CC4)=O)C3)nn2)ncccc1Cl 30383,c1(OCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30384,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CC3C)CC2)=O)cnc1O 30385,Cn1c(O)nc2cccc(C(=O)NCC(C)(C(C)C)NC(C3CCCO3)=O)c12 30386,c1(NCCN2C(=O)CCCC2)nccc(=NCC2CSCCO2)[nH]1 30387,C12(C(N3CC(=C(CNC(C4(OC)CCC4)=O)F)C3)=O)CCOC1CS(=O)(=O)C2 30388,c1(C(N2CCC(N(C(c3cncc(OC)c3)=O)C)C2)=O)c(F)ccc(F)c1Cl 30389,c1(OC)ccc(C2CCCN(CC3CCCC3)C2)c(F)c1F 30390,C(=O)(C(F)C(C)CNC(=O)Nc1ccsc1OC)NCC 30391,c1(CN(C(N2CCCC(c3n[nH]c(C4CCCC4)n3)C2)=O)C2CC2)ccccc1F 30392,C=CCC(C(=O)NC(C)CC(C)NC(c1cnn(C)c1OC)=O)C(C)C 30393,c1(OC)ccc(C(N2CCC(CNC(c3c[nH]nc3OC)=O)C(C)C2)=O)c(F)n1 30394,C1(NC(C(C)OC(C)(C)C)=O)CC12CCN(Cc1csc(NC(=O)C3CC3)n1)CC2 30395,c1(CC(=O)NC(CCNC(CC2(C(=O)OC)CC2)=O)C)c(C)n[nH]c1C 30396,C1(C(N(CC(CC)OC)C)=O)CCC(C)(C)N(C(=O)CC2(O)CCCCC2)C1 30397,c1(C(N2CC(OC)CC2(C)CNC(c2coc(C)c2)=O)=O)cc2cnn(C)c2s1 30398,N1(C(CC2CC(NC(CSCCC#N)=O)C2)=O)CC2(CCNC(=O)O2)C1 30399,N1(C=O)CCCC(C(O)C(F)(F)F)C1.C(=O)(C(=O)N(CC(C)CCNC(C)=O)C)N 30400,CCCCCCN(C(c1sccc1Cl)C(=O)NC(C)C1CC1)C1CC1 30401,Cc1[nH]nc(CC(=O)NCCCN(CCO)C(C2CC2c2ccnn2C)=O)c1Cl 30402,N1(C(Cc2c(C)c(Br)cnc2)=O)CCCN(C(=O)CNC=O)CC1C 30403,C1(C(=O)NCC2C(NC(=O)C(F)(F)CO)CCC2)CC2(CCCCC2)S1(=O)=O 30404,n1(CC(=O)NC(C2(CNC(c3c(C)ccnn3)=O)CC2)C)cnc2ccccc12 30405,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CCCCC2CCCO)=O)CCC1 30406,c1(C(N(C2CCN(C(C3CCCOC3C)=O)C2)CCC)=O)cc(C(N)=O)nn1C 30407,c1(C2(C(=O)NCCC(=O)N(C)CC3CNC(=O)C3)CCC2)cnn(C)c1 30408,n1(C(C)C)cnnc1CC(N1CCCC1C1(NC(=O)CN2CC3CC3C2)CC1)=O 30409,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(Br)CC1)=O)C2 30410,C1(CNC(C2(SCC)CC2)=O)CCN(C(=O)Cc2cccc(C)c2)C12CCC2 30411,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1conc1C(F)(F)F)=O)CC2 30412,CCC(=O)CCC(=O)NCCc1conc1CC(NCP(C)(C)=O)=O 30413,C=CC(C)(CCOC)C(=O)N1CC(C(=O)Nc2cc(OC)ccc2C)C(C2CC2)C1 30414,C1(NC(=O)CCc2ncc(F)cn2)CCC2(CCN(C(=O)CC3CCOCC3)C2)C1 30415,c1(COC)cncc(CNC(=O)C(C)CNC(=O)C(c2cnn(C)c2)O)c1 30416,N1(C(C2N(CC)CCCC2)=O)CCc2ccccc2C1CNC(=O)CCC1CC1 30417,c1(SC)ccc(NC(=O)NC2CCN(c3cccc(Br)c3)C2)cc1 30418,C1(NC(C2N(C)CCCC2)=O)CCC12CN(C(=O)CCc1cnc(C3CC3)o1)C2 30419,N1(C(C(CCC)C)=O)CC2CCC(CNC(=O)CSC(F)(F)F)C2C1 30420,Cc1sc(N)c(C(=O)NC23CC2CN(C(c2nnc(O)nc2O)=O)C3)c1C 30421,N1(C(C(CCC)CNC(c2nccnc2C)=O)=O)Cc2nncn2C(C)C1 30422,N1(C(CCC(=O)NC)=O)CC(NC(=O)C(C)=CC2CC2)CCC1C 30423,Cc1cccc(C(=O)NCC2(F)CN(C(=O)C(CO)C(C)(C)C)C2)c1C#N 30424,N1(CN=c2nc(N3CC(C)OCC3)c3c([nH]2)ccs3)CCOC2(CCSC2)CC1 30425,N1(C(C(C2CCN(C(c3cc(C)c(O)nn3)=O)C2)F)=O)CC2CCC1C(CO)C2 30426,S(=O)(=O)(c1ccc(N(C(c2ccccc2)C(C)OC)C)nc1)N(CCC=C)C 30427,N1(C(c2scc(OC)c2)=O)CC(CNC(c2sccc2OC(F)F)=O)C(O)C1 30428,c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)C2CC2)cccc2ccncc12 30429,c1(C(N2C(CC#C)CCCC2)C(=O)NCCC)cc(C)n(CC(=O)NC2CC2)c1C 30430,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30431,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)Cc1ccccn1 30432,N1(C(C23N(C(c4c(C)c[nH]n4)=O)CCC2C3)=O)CCN2C(=O)OCC2C1 30433,CC(C)C(C)C(CNC(c1cc(N)ccc1F)=O)NC(c1coc2c1COC2)=O 30434,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)NC)CC2)=O)CC1)C 30435,S(=O)(=O)(c1cccc(C(=O)NC23CC(NCc4conc4C)(C2)C3)c1)NC 30436,Cc1cc(CCNC(=O)CN(C(=O)CC2CC(C)C2)C(C)C)nn1C 30437,c1(C(N2C(C(=O)NC3(C(=O)OC)CC3)CSCC2)=O)cc(Cl)c(O)cc1F 30438,C(CNC(=O)CCc1ncccn1)(C(C)(C)C)NC(c1nc(COC)[nH]n1)=O 30439,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCCn3ccnc3)CCC1CC2 30440,C1(C(=O)NC)C2CCN(C(C3CC4C(C3)C4(C)C)=O)CC12.C(CCC=O)O 30441,c12cccc(c1)NC(=O)C2.c1(COC(=O)C=CC2CCOC2)cccc(OC)c1 30442,C1(C(=O)NC(c2cn(C)nn2)C(=O)N(C2CCCOC2)C)CC2CC(=O)C1C2 30443,Cc1nc(C(C)C)ccc1C(=O)NCC1(O)CN(C(=O)COc2ccon2)C1 30444,c1(C(=O)NCCCNC(C2(C(CC)(F)F)CC2)=O)c(F)ccc(Br)c1Cl 30445,CCC(F)(F)CC(=O)NC1CCC(C)N(C(=O)C(=O)C(C)C)C1.c12ccc(cc1)s2 30446,N1(CC(=O)N(C)Cc2cnn[nH]2)CCN(C(c2cscn2)=O)CC1 30447,c1(CNC(C2(SC)CC2)=O)cc(C)c(C(=O)NC2(N3CCOCC3=O)CC2)o1 30448,N1(C(CCN(C)CC)=O)CCC(N(C(=O)C(F)(F)c2ccncc2)CCO)CC1 30449,S(=O)(=O)(c1cccnc1)NCCC(=O)NCC1C(CNC(=O)C2=CCC2)C1 30450,c1(Nc2nccc(N3CC(C)CC(C)C3)n2)cnc2c([N+](=O)[O-])cnn2c1 30451,C(=O)(CCCCN(C(=O)C(C)(C)C1CCCO1)C)NCC(C)CCO 30452,S(=O)(=O)(c1ccc(=NC(C)c2ccncc2)[nH]c1)N1C(C)CC(O)C1 30453,c1(C(N2CCCC(N3C(=O)C3)C2)=O)ccc(C)cc1C.C1(NC)CCCC12CC2 30454,CC(C)C(C(=O)N1CC=CC(NC(C2CNC(=O)C2)=O)C1)N1CCCS1(=O)=O 30455,c1(OC)ncccc1CC(=O)NC1CN(C(=O)CCc2cncn2C)CC1O 30456,N1(C(C23CC(C(N4C(C)CCCC4)=O)(C2)C3)=O)CCC2CCC12C 30457,c1(C(=O)NC2(CNC(c3cc(OC)ncc3)=O)CC2)c(F)ccc2nc[nH]c12 30458,C(=O)(C(F)CCC(C)C)N(C1CCN(C(CCC(C)(C)OC)=O)C1)C 30459,N1(C(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30460,c1(C(=O)NC(C2CC=CCC2)C(=O)NC2(C)CC(C)(C)C2)ccc(C#N)cc1 30461,Cc1c(C(=O)NC2C=CCCC2C(N2CC(OCCOC)C2)=O)nnn1C 30462,c1(C(=O)NCC2CCN(C(C(C)(CO)OC)=O)C2)cc(Cl)c(F)cc1N 30463,CCCCC(=O)C(=O)NC(C1CN(C(C2CC23CCOCC3)=O)CCO1)C 30464,c1(CC(=O)NCC(Cc2ccccc2)N(C)C(c2nncs2)=O)nnc(O)s1 30465,c1(-c2scc(CCC)n2)ccc2[nH]cc(C(=O)Nc3cccc(F)c3SC)c2c1 30466,C1(NC(C(=O)N(CC(N)=O)C)=O)CCN(c2ncccn2)C1 30467,C=CC1(C(=O)N(C)Cc2cncs2)CCN(C(c2ccn(C)c2)=O)C1 30468,c1(NC)sc(NC(C2CCCCC2)C(=O)OC)nc1C.C(C)(C)OC 30469,N1(C(C2(C)CSC2)=O)CC(NC(c2ccccc2CO)=O)C(F)C1 30470,C1(O)(CNC(=O)CC2C3CCCC23)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 30471,c1(C(N2CC3C(CC(N4CCN(CCO)CC4)=O)C3C2)=O)ccc2nncn2c1 30472,Cc1nc(C)c(C(C)NCC2(CC(=O)NC(C)(C)C)CCOCC2)[nH]1 30473,N1(C(c2c(CC)cns2)=O)CCCN(CCNC(C2(C(F)F)CCCC2)=O)CC1 30474,c1(NC(CNC(=O)NCC23CCC(OC)C2C3)=O)cc(F)c(F)cc1Cl 30475,c1(C(N(C(C)CNC(=O)CNS(N)(=O)=O)CC)=O)ccc(C(C)C)nc1O 30476,N12CC3CC3(C1)C(N1CC(C)C1)C2=O.c1(CNCc2ccccc2)nnsc1C 30477,C1(C(=O)NCC(C)N(C(=O)C(=O)NCC2CC2)C)CC2CSCC(C1)C2 30478,C1(NC(c2cc(O)cs2)=O)CN(C(C2CC3C=CCC(C2)C3)=O)C2(CCC2)C1 30479,C(C(C)(CO)NC(=O)CCCSC(C)=O)NC(C1C(CCOC)C1)=O 30480,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30481,Cc1cc(C(=O)NCC2CC(C(=O)NC3CCCC(O)C3)C2)n(CC(F)F)n1 30482,C#Cc1ccc(C(=O)NCc2ccc(C(=O)NC(C)C(C)(C)OC)s2)c(C)c1 30483,Cc1c(CNC(=O)NCCC2OCCO2)cnn1-c1ccc(C(F)(F)F)cc1 30484,C12(CNC(=O)CC3CC3(Cl)Cl)CC3CC(CC(NC(=O)C(O)C(F)(F)F)(C3)C1)C2 30485,N1(C(C(C(CC)O)C)=O)CCN(C(c2cc(C)c(C(=O)N(C)C)o2)=O)C2(CC2)C1 30486,CC1CN(C(C2CCC3(CCC3)OC2)=O)CCCN1C(=O)CC1CC(C2CC2)C1 30487,C12(C(=O)NCC(CC=C)NC(c3cccnc3)=O)CC1CCC2(F)F 30488,n1(C(C2CCC2)C)nc(-c2ccc(N(C)C)nc2)nc1C1CCCN1C=O 30489,C1(C(C)O)CCN(C(=O)C(c2ccnn2C)NC(=O)CCn2cccn2)CC1 30490,N1(CCC(N2CCC(C)(C)C(c3nn[nH]n3)C2)=O)C(=O)C2CC=CCC2C1=O 30491,COn1cnc(C)c1C(=O)NCC1CN(C(c2cc(C)ccc2SC)=O)CCO1 30492,C1(C(C)CNC(=O)CCCSC)CCN(C(=O)CCOc2cccc(O)c2)CC1 30493,C1(N(CC)CC)C(=O)N1C.C1CC(=O)N=CC(=O)N1C.C(C)(=O)OC 30494,c1(CNC(N2CCN(c3nnc(C)c(C)n3)C(C)C2)=O)cccc2c1COC2 30495,c1(C(N(C(C)CNC(=O)C(F)CC2CCCC2)CC)=O)ncncc1Cl 30496,CC1Cc2ccccc2N1C(C1CC2CCCC2N1)=O 30497,N1(C(C(CC)NC(C)=O)=O)CCN(C(c2n[nH]cc2C)=O)CC1C(F)F 30498,c1(C(=O)OCC)cnc(NC(C)C(C)NC(c2ccc(CO)cc2)=O)c(Cl)c1 30499,c1(C(CC)OC(=O)C2CC2)nc(-c2ccccc2)nn1-c1cnn(C)c1 30500,c1(OC)ccc2nc(C)c(C(=O)NCC3CCC3NC(=O)Cc3ccsn3)n2n1 30501,C1(NC(CCSC)=O)CN(C(=O)CCc2cc(F)ccc2F)CCC1C 30502,c1(C(N(C2CCCS(=O)(=O)C2)CC)=O)cc(C)cc(OC)c1OC 30503,Cc1cnc(C(N2CCSCC2CCNC(C2(C)CCCCO2)=O)=O)cc1C 30504,Cc1ncc(C(=O)NC2(C)CCCN(C(c3c[nH]c(=N)c(C)c3)=O)C2)c(=N)[nH]1 30505,c1(C(=O)NCCC2CCCN(C(C(C)(C)OC)=O)C2)cccc(N)c1C 30506,N1(C(c2cccc(SC)c2)=O)CC(NC(c2csc(CC(C)C)n2)=O)CCC1C 30507,C(=O)(CC(O)(C(F)(F)F)c1ccc(C)o1)N(CCN(C(COC)=O)C)C 30508,C1(C)(SCC(=O)NCCC(=O)OCC)NC(=O)NC1=O.N12CCNCC1C2 30509,C1(NC(C(C)=C(CC)C)=O)CC2CC(NC(=O)C(C)(C)CO)CC12 30510,N1(C(c2ccn(COC)n2)=O)CCC=C(C(=O)N2CC3CCC2C3)C1 30511,n1(CC(=O)OC)ncc(CNC(N2CC(CC(C)(C)C)C2)=O)c1C 30512,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30513,c1(-c2ccc(F)cc2)cc2c[nH]nc2s1.C12CCC(O1)C2 30514,C(=O)(CCC(=O)N1CC(NC(=O)CC(O)CN(C)C)CC1C)N(C(C)C)C 30515,C1(C(N(C)OCc2cccnc2F)=O)C=CCN(C(=O)Cc2cnn(C)c2)C1 30516,c1(CC(=O)NC23C(CN(C(c4cncc(C)c4)=O)C2)C3)cccc(F)c1F 30517,C1(OC)(CNC(=O)C(CC(=O)OC(=O)CCCC(C)O)c2ccccc2)CCCCC1C 30518,c1(NC(CC)=O)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(C(=O)O)C3)c1 30519,C1(C(N)=O)C2CC3CC(C2)CC1(NC(NC1CCCc2c[nH]nc21)=O)C3 30520,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1 30521,CC1(C#CC(=O)N2CCC(C)(CCNC(=O)COC3CCCCC3)C2)CC1 30522,C1(NC(C(CC)C)=O)CN(C(C2(CCC)CC(=O)C2)=O)CC1C(F)F 30523,C1(N(C)C(c2ccnc(S)c2)=O)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 30524,C1(C(=O)NCC2C=CC(NC(C3(C(=O)NC)CCC3)=O)C2)CS(=O)(=O)CC(=O)N1 30525,C(C)(C)(CC(=O)N1CC(C)(C(N)=O)C1)N(C)C(C1(c2cc[nH]n2)CC1)=O 30526,c1(-c2cc(C(=O)NC3COCC3c3ccccc3)on2)cccc(Cl)c1 30527,c1(-c2cnc(N3CCN(Cc4cccc(C#C)c4)CC3)nc2)ccc(F)c(C#N)c1 30528,c1(C(N2C(CCC)CN(C(=O)CC3=CCCC3)CC2)=O)ccc2c(c1)nnn2C 30529,C#Cc1cn(C)nc1C(=O)NCC(O)CC(=O)N1CC(OCCC)C1 30530,C1(C(N)=O)(OC)CCCN(C(=NCc2ccc(C#N)cn2)NC(C2CC2)C2CC2)C1 30531,C(=O)(CCCS(C)(=O)=O)N1CCCN(C(c2c(C)ncn2C)=O)CC1 30532,CCC(O)(C(=O)NCC1CC2CC2N1C(C1OCCO1)=O)c1ccccc1 30533,C1(NC(c2occc2Br)=O)CCC2CN(C(C3=C4C(CN=C3)C=CC=N4)=O)CC2C1 30534,CC1CCCCN1CC(N1CCC(C(=O)NC2(CC(C)(C)C)CC2)CC1)=O 30535,c1(C(N2CCC(C(C)NC(CCCSC)=O)C2)=O)sc(C)cc1Cl 30536,C1(CCCC)CCC(NC(=O)Nc2c[nH]nc2-c2ccccc2Cl)CC1 30537,c1(C(c2ccc(OC)cc2)NCC(C)C(C)(F)F)nc(O)c2c(C)c(C)sc2n1 30538,N1(C(C(C)C(C2CCC2C)CNCCC=C)=O)CCC(C(=O)OCC)C1 30539,c1(C(N2CC3(CNC(CC=C=C)=O)C(C(F)F)(C2)C3)=O)cc(C)c2[nH]cnc2c1 30540,c1(C(=O)NC(C(C)C)(C)CNC(=O)CSC(F)F)cnc(C2CC2)[nH]c1=N 30541,c1(C(=O)NCCC)ccc(NC(c2ccc(Nc3ccccn3)nc2)=O)cc1 30542,N1(C(c2c(C)ccc(C)c2)=O)CC2CC(NC(=O)CCN(C)C3CC3)CC1C2 30543,N1(CCNC(=O)CC2CSC2)CCN(C(=O)CC2(C(F)(F)F)CCC2)CC1 30544,C12(NC(c3c(CC)noc3)=O)CC(CNc3ncncc3C(C)=O)(C1)OC2C 30545,C1(C(=O)NC2(C)CC(NC(CC(C=C)C)=O)C2)Cc2cscc2C1 30546,C1(OC)(OC)CC(C)(C(=O)N(CC(O)CNC(=O)CC2C(C)(C)C2(C)C)C)C1 30547,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30548,c1(SC)cc(C(=O)NCC2(C)CN(C(=O)CC(c3ccccc3F)C)C2)c(C)o1 30549,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30550,CCC(CC(C)C)C(=O)N1CCC(NC(C2CCCO2)=O)C(OC)C1 30551,c1(OCC(=O)NC(CNC(CCCCOCC)=O)CO)c(Cl)cncc1Cl 30552,Cc1cc(NC(c2cc(CNC(c3cc(CO)ccn3)=O)on2)=O)c(=O)n(C)c1 30553,N1(C(c2cc(COCC)on2)=O)CC(CC(=O)N(CCCC(C)C)C)C(C)C1 30554,N1(C(c2cn(CC)nn2)=O)CCC(O)(C(=O)NCCN2CCNC(=O)C2)C1 30555,c1(NC2CCN(CC=C)CC2)ncc(S(=O)(=O)N2CCC(C)C2)cc1Cl 30556,CCC(CCOC)C(=O)NCC1CCC1NC(c1nccc(OC)c1O)=O 30557,C1(C(=O)NCCc2cnc(C)o2)C2CC2CN1C(=O)C(C)CO 30558,C(CC#CC(C)(C)C)NC(CC(CC)NC(C1(CC)CC1)=O)=O 30559,Cc1cc(C(=O)NCC2(NC(C3CSC3)=O)CCC2)cc2nc[nH]c12 30560,c1(CNC(=O)NOCC2COCC2NC2CCCCS2)cccnc1Cl 30561,Cc1cc(Cl)cc(C)c1C=CC(N1CCCC1CCNC(=O)C(O)C(C)C)=O 30562,c1(NCC(C)S(N)(=O)=O)ncccc1S(=O)(=O)NC(CC(N)=O)C1CC1 30563,c12nnc(n1CC1CCCO1)C2OC(=N)O.c1(N(C)C2CC2)cccs1 30564,Cc1ccc(C(N2CC3(CCC(CNC(=O)Cc4ccno4)O3)C2)=O)cc1C#N 30565,CN1CCCC(F)(C(=O)NCCOC2CCN(C(C3(C)CCC3)=O)CC2)C1 30566,c1(C(N2CCN(c3ncnc(CC)c3F)C3C2C3)=O)cc2ccc(C)cc2o1 30567,C1(C)(CNC(C(C2CCOC2)OC)=O)CCN(C(C23CCN(CC2)CC3)=O)CC1 30568,C1(CC(=O)N(C2CCN(C(c3nc(O)sc3C)=O)CC2)C)CCCCC1(F)F 30569,C(=O)(C(C)CC(F)F)NC1CC(C(C)NC(c2ccn(CCC)n2)=O)C1 30570,CCC(C)C(=O)NC(CNC(C1CC2CC2C1)=O)C1CCC1 30571,c1(C(C)C)ccc(S(=O)(=O)N2CCCC(C(N3CCOCC3CO)=O)C2)cc1 30572,C1(N(C(c2n(CC)ccn2)=O)C)CCCN(Cc2nnc(C3CC3)o2)C1 30573,C(=O)(N=c1nc[nH]n2cccc12)C1CC(NC(c2cccc(F)c2O)=O)C1 30574,C(=O)(C(O)C(C)C)NC(CCC)CNC(c1coc(C(N)=O)c1)=O 30575,CCC1=C(C(=O)NCCC(O)C(=O)NC2CCc3n[nH]c(C)c3C2)CCCO1 30576,C1(NC(C(N)=O)=O)C2COCC1CC(NC(=O)C1=CCCOCC1)C2 30577,N1(C(C(C(C)(C)C)OC)=O)CC(C2CN(C(c3csc(Br)c3)=O)C2)C1 30578,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30579,CCC(CCC(=O)NCCSCC(=O)NCCc1n[nH]c(C2CC2)n1)OC 30580,Cc1c(O)ccc(C(=O)N(CCNC(=O)CNC(=O)CCC(C)C)C(C)C)c1C 30581,C1(C)(c2onc(CCCNC(C)=O)n2)CCC(NC(=O)OC(C)(C)C)CC1 30582,c1(C(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30583,c1(OC)cc(C(=O)NC2(CNC(c3cc(=O)n(C)o3)=O)CCCCC2)cc(F)c1 30584,C(CCCCCC(=O)NCC(O)C1(Cl)CC1)NC(CC(COC)C)=O 30585,C(CC(=O)NCC1C(C)CCN1C(=O)CSCCN(C)C)(C(F)(F)F)OC 30586,CCCC(CNC(c1nc(C(C)(C)C)no1)(C)C)C(=O)O 30587,O=C(CC1=CCOCC1)N1CCCN(C(=O)C(C2CC2)C2CC2)CC1 30588,N1(C(COC2C(C)CCCC2)=O)CC2(CC2)CC1CNC(=O)C(C)(F)F 30589,CC1(C(=O)NCCOC2CCN(C(C3CCCCNC3=O)=O)C2)CCCNC1=O 30590,C1(CNC(CC(C)c2ccco2)=O)C2CN(C(=O)CC3(C(F)F)CC3)CC12 30591,C(=O)(CCCCCCCC=C)NC(CC#C)(C)C(=O)N(C)Cc1cc(C)cs1 30592,c1(CC)cc(C(N2CC(F)(c3cccnc3)C2)=O)no1 30593,C(CNC(=O)C=Cc1cc[nH]n1)(CC(=O)NCC1CC(O)C(O)C1)OC 30594,c1(CN(c2ccccc2F)CC)ccc2c(C(=O)NCCOCCO)ncn2c1 30595,C(=O)(C1c2ccccc2CN1C(c1cc2ccoc2s1)=O)NC(=O)CCC(C)C 30596,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30597,C1(NC(=O)NCCC)CCN(C(=O)C#N)CCC1CO 30598,c1(C(N(CCC(C)NC(CCc2onc(CSC)n2)=O)C)=O)cnnc(C)c1C 30599,c1(C(=O)NCC(CNC(CC(CC)CC)=O)(C)OC)ccc(F)c2ccoc12 30600,CCCC(C#N)N(C(C)CC)Cc1ccc(Cc2ccccc2)s1 30601,C1(C(N2CC(C)CC(CC)C2)=O)(CC)CCCN(C(=O)CC#N)C1 30602,C1(NC(c2c(OC)ccc(OC)c2)=O)CCC(C2CCN(C(=O)C(C)(C)C)CC2)C1 30603,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(C(F)(F)F)C(NC(=O)OC(C)(C)C)C1 30604,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30605,c1(C(=O)NCC(C(C)C)(C)NC(c2cccc(Cl)c2)=O)cc(F)c(O)c(F)c1 30606,c1(C(=O)NC(C)C(C)NC(c2ccnc3[nH]cnc23)=O)cc2c(s1)CCCCC2 30607,c1(C(=O)NCC2OCC(CNC(Cc3cn(C)nc3)=O)C2)ccnc2ncnn12 30608,C(C)(C)(C(=O)NCc1ccoc1C(=O)NC1C=CC(C(N)=O)C1)SC 30609,c1(CC(C)C)[nH]nc2cncc(C(N3CCC(C)(NC(=O)C=CCO)C3)=O)c12 30610,c1(OC)cccc(C(=O)N(CC(c2ccccc2)O)Cc2cccc(C)c2)c1C 30611,c1(NCCC2(O)CN(C(C(CC)SC)=O)C2)ncc(Br)cc1[N+](=O)[O-] 30612,C1(C)(C(=O)NCCCN(C(=O)CC2(C#N)CC2)C)CCC(=O)N1 30613,CC1(C2CC2C(=O)N(CCNC(c2ccc(C(F)(F)F)nc2)=O)C2CC2)COC1 30614,NS(=O)(=O)N1CCCC(C(=O)NC2(C3CN(C(=O)CCC(N)=O)C3)CC2)C1 30615,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3ccc(O)nn3)=O)C2)c1 30616,C1(CC(=O)NCCCC(=O)NC)CN(C(C)C(=O)OCC)CCC1C 30617,C1(CC(=O)NCCOC2CN(C(C=CSC)=O)C2)CC2(CC2)CO1 30618,C1(C(N(CCCSC)C)=O)CCN(C(=O)C(C)c2cccs2)C1C(C)C 30619,C(c1ccccc1)=CCN(C)C(=O)NCCc1cc(C(F)(F)F)n[nH]1 30620,S(=O)(=O)(c1cnccc1N1CC(CO)CC(C)C1)NCCSCCOC 30621,CC1(C)CC=C(C(=O)N2CC3CC2(CNC(C2CCCN2S(C)(=O)=O)=O)C3)CC1 30622,C(CC(C)(C)C(=O)N1CCN(C(C)CO)CC1)NC(c1c(C)n(C)nn1)=O 30623,CCC(C(=O)N(C1CCCN(C(C2(N3CCOCC3=O)CC2)=O)C1)C)C(F)(F)F 30624,N1(Cc2c(CNCC(=O)OC)cccc2)CCN(C(=O)Cc2ccc(Cl)s2)CC1 30625,Cc1[nH]nc(C(N2CCCCC2CNC(=O)CCc2ccnn2C)=O)c1C 30626,C1(C)(NC(CC2CCC(C)C2)=O)CCCN(C(=O)CCc2ccc(CO)cc2)C1 30627,N(C(=NCCC1CC(F)C1)NCCc1cnccn1)CCN(C)CC 30628,C(=O)(CS(=O)(=O)C1CCCC1)NCC(c1cc2ccccc2o1)C 30629,c1(C(N2CCOC(CNC(C3CC(F)(CO)C3)=O)C2)=O)ccc2nnnn2c1 30630,C1(N(C(C=C(CC)CC)=O)C)CN(C(=O)C(c2cccc(C)c2)(F)F)CC1O 30631,C1(CNC(C(CC)OCC)=O)CC(NC(=O)Cc2cscn2)C(O)C1 30632,C=CC1(NC(C2C(C)CCC2C)=O)CCN(C(=O)COc2cccnc2)C1 30633,Cn1cc(CC(O)C(=O)NCCNC(=O)C=Cc2cnc[nH]2)cn1.C1CCCO1 30634,C1(NC(c2ccn(CCN(C)C)n2)=O)CC12CC(NC(C1CC(F)(CO)C1)=O)C2 30635,c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)C)ccc(N)cc1[N+](=O)[O-] 30636,C1(C(=O)NCC2(NC(C(C)OC)=O)CCCC2)CCCCN1C 30637,C(=O)(N=c1nc2ncc(C(F)(F)F)cn2[nH]1)c1cccc(C#N)n1 30638,n1(CC)nc(C)c(CC(N2CCOC(CNC(=O)CCCN=[N+]=[N-])C2)=O)c1C 30639,N1(CC=C)CCC2C(CCCN2C(c2cnn(C)c2)=O)C1 30640,Cn1c(=O)oc2cc(-c3cn(C4CCN(C(=O)C(F)=C5CCC5)C4)nn3)ccc12 30641,OCC1CN2CCN1C(C(N1CC(NC(c3c4ccccc4nn3C)=O)C1)=O)C2 30642,N1(C(C=C(CC)CC)=O)CC(NC(c2ncccc2OC(C)C)=O)CC(O)C1 30643,N1(C(CS(CCOC)(=O)=O)=O)CC2(CCN(C(C3CC3C#N)=O)CC2)CC1C 30644,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)CO)ccn2cncc2c1 30645,N1(C(C2N(Cc3nnc(C)s3)CC2)=O)CCC(CCNC(=O)C(C)C(C)C)CC1 30646,N1(C(CCOC)=O)CCC(O)(CN2CCC(C(=O)N(CC(C)C)C3CC3)CC2)C1 30647,C1(NC(=O)CN2CC3CC3C2)COC2CN(C(=O)CCSC3CCCC3)CC12 30648,N1(C(c2ccn(CC)c2C)=O)CCCN(CCCCNC(C2CNC(=O)C2)=O)CC1 30649,S(=O)(=O)(c1ccsc1C(N1CCN(C(=O)C#CC2CCCC2)CC1CF)=O)NC 30650,N1(C(C)=O)CCC2(CCN(C(=O)C(C)C(C)(C)C)C2)C1.N(CCN)(CC)CC 30651,c1(C(=O)NC2C(CNC(C3(C)C(CC)CCC3)=O)CC2)ccc2oc(=N)[nH]c2c1 30652,C12(NC(c3c(C)cn(C)c3)=O)CCCC(CN(C(c3c[nH]c(=N)o3)=O)C1)C2 30653,CC#CCCC(=O)N1CCC(C(=O)NCCN2CCCC(O)C2)O1 30654,N1(C(=O)CC(C2CC2)NC(C23CCCC2C3)=O)CC2(CCC2O)C1 30655,n1(CC)nnnc1C(C)(CC1CCCO1)NCCc1csnc1OC 30656,CCCCCCCCC(C)C(=O)NC(CNC(C1(OC)CC1)=O)C(C)C 30657,c1(NC(C)=O)cc(C(=O)NC(C(F)F)C2CCCO2)ccn1 30658,C(=O)(CCS(N)(=O)=O)NC(CNC(CCC(C)SC)=O)(C)C(C)C 30659,c1(CN(C(c2cc(C)no2)C(=O)NC(CC)(C)C)C(C)C)ccccc1Cl 30660,C(C(=O)NC(C)CCSC)(C(C)C)N(C(CCN(CCC)C)=O)CC 30661,C1(CCNC(=O)NC2(c3cn(C)nc3)COCCO2)COCC(C)(C)O1 30662,C1(OCC(=O)NC(C(C)NCCCOCC(=O)SC)C)CC(F)(F)C1 30663,S(=O)(=O)(c1cc(F)c(OC)cc1Cl)N(C(=O)C(N)CC1CCCC1)C(C)=O 30664,C1(CNC(c2ccoc2Br)=O)CCCCC1NC(C1(C2CCCO2)CCC1)=O 30665,c1(C(N(CCCNC(C(CC)OC)=O)CC)=O)cc2ccccc2oc1=O 30666,Cc1ccn(C)c1C(=O)NCCC1CCCN(C(C2(O)CCCCC2)=O)C1 30667,N1(C(C(C)(C)NCCc2cccc(Cl)c2)=O)CCCS(=O)(=O)C1 30668,C(=O)(C(O)C(C(C)C)OCC(C)(CO)CC=C)NCC(=O)NCCCC#C 30669,c1(C(N2CCC(C)C(NC(C3CC(CC4CC4)C3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 30670,c1(CC(=O)Nc2ccnc(-c3cc(F)c(F)cc3Br)c2)ccc2n[nH]cc2c1 30671,C1(C(=O)NCC2(C)CCN(C(C3(C)C(C)C3)=O)C2)CCC12CCOCC2 30672,N1(C(c2cn(CCOC)nc2)=O)CC(NC(c2ccc(SC)o2)=O)C(O)C1 30673,c1(C(=O)NC2C(C)CN(C(c3nn(C)cc3Cl)=O)CC2)cc2c(cc1O)OCO2 30674,N1(C(C(C#C)(C)C)=O)CC2CC(NC(=O)Cc3cnccc3C(F)(F)F)C(C2)C1 30675,c1(-c2cnc(C)nc2)ccn2nc(C(=O)Nc3ccc(Cl)c(F)c3)cc2c1 30676,c1(C(=O)NCC(N2CCN(C(C(CCOC)C)=O)CC2)C)c(C)ccc(C)c1F 30677,C1(C(=O)NCC2N(CC(=O)OC)CC2)CC=CC(O)C1 30678,C12(CNC(c3cc(CO)ccc3Cl)=O)CCC(CC1)CN2C(=O)C1=COCC1 30679,CC1CCN(C(C2(C(F)F)CC2)=O)CCN1c1ncc(I)cn1 30680,Cc1nn(-c2cccc(F)c2)cc1CNCCCCCN1CCCCC1 30681,c1(C(=O)NC(C2(O)CCN(C(=O)C3=CSCCO3)C2)C)c[nH]c(=N)nc1O 30682,Cc1cnncc1C(=O)O.N12CCC(CC1)NC2=O.C(C)(C)(C)CCSC 30683,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30684,N1(C(C=C(CCC)C)=O)CC(O)(C2(CNC(c3c(C)cc(F)cc3C)=O)CC2)C1 30685,C1(CNC(C(CN(C)C)(F)F)=O)CC2CCC1N2C(=O)CC1SC(=N)NC1=O 30686,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(NC)cn2)=O)CC12CCC2 30687,n1(CC)ccc(C(N2CC(CCNC(=O)COCC(=O)OCC)C2)=O)n1 30688,C1(CNC(C(CC)=CC)=O)CN(C(=O)CN(C)S(N)(=O)=O)CCN1C 30689,N1(C(C(C)CC(C)(F)F)=O)CCOC2(C1)CN(C(=O)CCCC1CC1)C2 30690,C=CCCC(CO)NC(c1cn(C2CCN(C(=O)C=CC(=O)N(C)C)C2)nn1)=O 30691,c1(NC(C2(C)CN(Cc3ccc4nc[nH]c4c3)C2)=O)ccc(Cl)c(C#N)c1Cl 30692,n1(CC)cc(CC(N2CCCCC2CNC(=O)CCS(C)=O)=O)c(C)n1 30693,C(c1ccncc1)=C(C)C(N1CCC(O)C1C(=O)NC1CC2(CC2)CO1)=O 30694,c1(C(=O)NCc2ccc(-c3ccc(SC(C)C)cc3)cn2)c(O)ccc(F)c1F 30695,C(=O)(C(CO)NC(c1[nH]ccc1NC(N)=O)=O)NC1CC(SC)C1 30696,C1(CCC)CCN(C(=NCC2CCCCC2)NCCOCC2(O)CCC2)C1 30697,c1(C(C(C(=O)Nc2nnc(N(C)C)s2)N)=O)ccc(F)cc1F 30698,C1(C(=O)NC2(CC)COC2)(NC(COCC)=O)CC(CO)C1 30699,c1(OC)cc(C)cnc1C(=O)NC1CC(NC(=O)C2=CCC2)C1 30700,N1(C(Cc2cc(CC)no2)=O)CCN(C)CC1CNC(=O)CC(CC)C1CCCO1 30701,CON(CCC(=O)N(CCN1CCC1)CC)C(=O)C1CCCN1C=O 30702,C(CCC1CC1)(C(=O)NC1CC(O)C1O)NC(C(COC)NC(C)=O)=O 30703,N1(C(C2C(CC)CCC2)=O)CCC(CO)(CNC(C2CCC(=O)N2)=O)CC1 30704,c1(-c2ccc(NC(N)=O)cc2)ccn2nc(C(=O)NCC3(O)CC3)cc2c1 30705,C=C1CCN(C(=O)C(C2CCC2)OCC)C(C(=O)NCC2CC(C)(C)C2)C1 30706,Cc1nn(C)c(Cl)c1C(=O)NC1(C2CN(C(C3COC(=O)N3)=O)C2)CC1 30707,c1(CC)oc(C)cc1C(=O)NC(Cc1cnc[nH]1)C(=O)N1CCCC1 30708,c1(C(N(C)CC2N(C(C=CC(=O)N(C)C)=O)CCC2)=O)c[nH]c(=O)c2ccnn12 30709,N1(c2cc(NCC3(O)CN(C)C3)ncn2)CCCC2(CCCCCC2)C1 30710,C(CCSC)(C(=O)N(CC(O)CNC(=O)Cc1cnn(C)c1O)C)OC 30711,c1(C(=O)NC2C(NC(=O)CC3CCCCC3(F)F)CCC2)ccc2nnnn2c1 30712,c1(C(=O)NC2CC(N(C(CCC(=O)OC)=O)C)C2)cc(N)nc(Cl)c1 30713,C(C(=O)N(CC)OC)NC(C(CNC(C1(CC#C)CC1)=O)C)=O 30714,c1(C(=O)NC(CNC(c2n(COC)ncc2)=O)(C)CC)cc(N)c(O)c(F)c1 30715,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cocc3C(N)=O)=O)C2)C1 30716,C(=O)(C1CCc2cccc(F)c21)NC(C)CN(C(=O)Cn1ccc(=O)cc1C)C 30717,C=CC1(C(=O)NC2CCCCC23CC3)CCN(C(=O)Cc2cscn2)C1 30718,CCC(C)CCCCC(=O)NCC(CC)NC(=O)Cn1cc(C)cn1 30719,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(C(C)O)s1)=O 30720,c1(C(=O)NC2CCC(CCNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30721,C(=O)(C#CC1CCCC1)N1CCC(NC(c2c(C)c[nH]c2CC(N)=O)=O)C(C)C1 30722,C(=O)(C(CC(C)C)N(C)C)N1C(CNC(c2nc(CC(C)C)oc2)=O)CC1 30723,C1(C(C(=O)NCC(CC)NC(C2(C)COCCO2)=O)(C)C)CCCCCC1 30724,c1(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)F)=O)csc([N+](=O)[O-])c1 30725,C1(NC(C(CC)=CCCC)=O)CCN(C(=O)COc2cc(C)on2)CC1F 30726,C(C(=O)NCCCF)(C(C)(C)O)NC(C(CCSC)O)=O 30727,N#CC1CCCCN1C(C1CN(Cc2cccnc2F)CCC1O)=O 30728,C1(CNC(c2nc(Br)c[nH]2)=O)CN(C(C23CC(F)C2C3)=O)CC12CCOCC2 30729,N1(C2CCC(c3cccc(OC)c3)C2)CCOc2cccc([N+](=O)[O-])c2C1 30730,C(=O)(C(C)(CC)CC)NC(CNC(Cc1c(SCC)cccc1)=O)CCOC 30731,N1(C(C2CCCCC2O)=O)CCC(C)(CC(=O)NC2(C(C)(C)O)CC2)C1 30732,c1(C(=O)O)ccccc1CC(N1CCCCC1C(c1cn(CCO)nn1)C1CC1)=O 30733,c1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC3CCC2C3)cccc2c1SCCC2 30734,N1(CC(=O)N(C)CCNC(=O)NC2CC2)CCCC1CNC(CC)=O 30735,c12ccc(Br)cc1S2.C(=O)(CCc1nc[nH]n1)N(C)C 30736,N1(C(C(CCN(C)C)NC(C(NOC)=O)=O)=O)CCN(C)CC(O)C1 30737,N1(Cc2cnn(C)c2Cl)CCc2cc(NS(=O)(=O)c3cccc(Cl)n3)ccc2C1 30738,CC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CN1C(c1c[nH]ccc1=N)=O 30739,C1(NC(CC(C=C)CCC)=O)CCC2(CCCN(C(=O)CCCC(=O)OC)C2)C1 30740,CC1CN(C(C23CN(C(=O)CCc4nc[nH]n4)CC2CCO3)=O)C(C)CC(C)O1 30741,c1(C(N2CCC(NC(c3c(C)coc3)=O)(CO)C2)=O)c(C)cccc1[N+](=O)[O-] 30742,C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC2CN(C(c3c(C)coc3C)=O)CC21 30743,N1(C(CCCC(C)=O)=O)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2C1 30744,N1(C(c2c(OC)nccc2)=O)CC(CC(=O)NOCC2CCCO2)C2(CC2)C1 30745,c1(CC)cc(C(=O)NC2CN(C(=O)Cn3nnc(=N)[nH]3)CC2C(F)F)c(C)nn1 30746,C1(NC(C=C(CC)C)=O)CCN(C)C12CCCN(C(C)=O)C2.C12CCC1CC2 30747,c1(C(=O)NC2CCCN(C(c3cc(OC)cc(F)c3)=O)C2)cc(Cl)c(F)cc1F 30748,n12cc(c3ccccc13)C(=O)NCCC2.C1(SC)CCC(NC(C2CCC2)=O)C1 30749,N1(C(c2c(C)cco2)=O)CCc2ccccc2C(NC(=O)C(N)CCC(N)=O)C1 30750,N1(C(c2c(CC)nnc(C)c2)=O)CC2(CCN(C(C3(SC)CCC3)=O)CC2)C1 30751,c1(OCC)ncc(C#N)cc1NC(C1CC2(CC2)CN1Cc1ccc(Cl)s1)=O 30752,C(=O)(CCN(OC)C(=O)CC1CC1C(F)(F)F)NC(C)C(F)(F)F 30753,c1(OC)cc(C(=O)NC(c2ccnn2C)C(=O)NCC2COCCOC2)ccn1 30754,C1(C)(C(=O)NCC(CNC(C2C(C(=O)OC)C2)=O)O)CC2(CC2)C1 30755,C(CC(=O)NCC)NC(=O)CONC=O.C(C(C)(C(C)(C)C)C1CC1)OCC.O.C.OC 30756,Cc1ccc(F)c(NC(c2cccc(NC(c3cc(C)cc(Cl)c3)=O)c2)=O)c1 30757,N1(C(c2c(C)nc[nH]2)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30758,N1(C(C(C)OCC#C)=O)C2CCC1CN(c1ccnc(C)n1)CC2 30759,c1(C(=O)NCCC(C)NC(=O)CCc2nc(O)n[nH]2)c(F)ccc(F)c1N 30760,C1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)COc2cc(Cl)ccc2C1 30761,C1(C(=O)NCC2(CN(C)C(C3CCN(C4CCCCC4)C3)=O)CC2)CCCC1O 30762,N1(C(C(C)(C)C2CCOCC2)=O)CCC(N(C(=O)CC=C(Cl)Cl)C2CCCO2)CC1 30763,CCC(CC(=O)NC(CCN(C)C)C(=O)N1CCC1c1ccccc1)C1CCC1 30764,c1(C(N2CC3C(C(=O)NC(C(CO)N(C)CC)C)C3C2)=O)ccc(O)cc1C 30765,c1(C(=O)OC)cccc(N2CC(C(C)NC(=O)C(C)(C)CC(F)F)C2)c1[N+](=O)[O-] 30766,N1(C(=O)CCC2CCC2)CCC2(CC1)CC2CNC(C1(CCF)CC1)=O 30767,CC1OCCN(C(=O)CC2CCOC2)C1C(=O)N(CC(F)(F)Cl)CCO 30768,c1(C(=O)NC(C2CCCCN2C(=O)Cc2conc2C)C)nn(C)c2c1COCC2 30769,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30770,N1(C(c2cn(CCC=C)nn2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)C2CCC12 30771,C(C1=CCN(C(=O)CC2CCC3CC3C2)CC1)NC(c1ccnn1C1CC1)=O 30772,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)Cc2cocn2)CC12CCOCC2 30773,N1(C(=O)CC23CCCC2C3)CCN(C(=O)CCNc2ccccn2)C2(CC2)C1 30774,C1(CC)CC(N(C=O)Cc2cccc(OCCCOC)c2)C12CCC2 30775,c1(C(=O)NC(CNC(C(CCCCC)O)=O)CO)cc2cc(C)ccc2[nH]1 30776,C(CS(=O)(=O)CC(=O)NC1CC1NC(c1nc(C)c(C)nc1C)=O)OC 30777,N1(C(C(C)(C)SC)=O)CCC(NC(c2cscc2Br)=O)C2(CCC2)C1 30778,c1(C(=O)NC2CC(CNC(C(CC(C)C)OC)=O)C2)cc2ncccc2s1 30779,Cc1ccc(F)c(C(N2CC(O)(C(C)NC(=O)CCC3CCN(C)CC3)C2)=O)n1 30780,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2Cc3cscc3C2)=O)CC1C 30781,CC1CCCCCC1NC(=O)C=CC1CCCN1C(=O)C=Cc1ccsc1 30782,N1(C(C(CC=CC)NC(C2CC2CC(C)(C)C)=O)=O)CCC2(C=CCO2)CC1 30783,C=C(CNC(c1cc(C)c(I)cc1F)=O)c1ccc(C)c([N+](=O)[O-])c1 30784,N1(C(CCC=C(C)C)=O)CCC2(CC1)CN(C(C1C3CCC1CC3)=O)C2C 30785,C(CC(C)C)(C(=O)N1CCCN(C(=O)Cn2cc(C(C)O)nn2)CC1)OC 30786,CC1CC(NC(=O)NCC2(C)CC(F)(F)C2)C(=O)N1c1ccccc1 30787,C#Cc1cc(C(=O)NCC(C)CNC(c2cc(Cl)cc(F)c2F)=O)cc(N)c1 30788,C(=O)(C(C)(CC)CC#C[Si](C)(C)C)NC1(Nc2ccc(OCC(=O)NC)cc2)CC1 30789,c1(CNC(C2(C=C)CCC2)=O)ncc(C(=O)NCCN2CC3CC3C2)cn1 30790,c1(C(=O)NCC=CC(=O)N(C2(COC)CC2)C)ccc([N+](=O)[O-])o1 30791,C(C)(C)(C(=O)N(CCC(C)(C)NC(=O)CC1CC1C)C)OC(C)=O 30792,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 30793,C=C=C(C)CC(=O)NCC1(CNC(=O)C(C)(CC)OC)CCOCC1 30794,c1(C(C)NC(=O)CC2CCN(C(C3CC3C#N)=O)CC2)c[nH]ccc1=O 30795,N1(C(CCCCC=C)=O)CCC(C2CC2)C1CNC(=O)CN1CC(=O)NC1=O 30796,c1(NC)c(C(=O)NC2COCC2NC(=O)C(C)C(C)(F)F)cccc1F 30797,c1(C(N2CC3(CCN(C(C=CCOC)=O)C3)C2)=O)cc2n(n1)CC(C)NC2=O 30798,CC1CN(C(C2C3CNC(=O)C23)=O)CC2(CCN(C(=O)C=CC(F)(F)F)C2)O1 30799,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 30800,C123CCC(C1)(OC2)C(=O)N1CCCC(C1)C(=O)N3.C(=O)(C1=CCCO1)N 30801,C12(CNC(=O)CC3CCN(C(C4CC(O)C(F)C4)=O)C3)CCC(CC1)C2 30802,N1(C(CC2CC(=O)NC2)=O)CCC2(C=C(C(=O)NOC(=O)C(F)(F)F)C2)C1 30803,CCCC(C)=CC(=O)NC(C(=O)NCCOC1CCCC1)C1(C)CC1 30804,c1(N2CCC=C(C)C2)nc(=NC)[nH]c(=NCc2cc(F)c(F)cc2F)[nH]1 30805,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)CC1 30806,c1(C(=O)NCCCC(CO)NC(CCc2cnc(C)s2)=O)cccc2nccn12 30807,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 30808,C(CCCCCCC)C(N1C(CNC(C(CC=C)OC)=O)C(CC)CC1)=O 30809,c1(SC)ocnc1-c1cn(C(C)CNC(=O)Cc2conc2C)nn1 30810,C(=O)(C(=O)CCC(C)C)NC1CCN(CC(=O)Nc2c(SC)cc(C)cc2)C1 30811,N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2coc(Cl)n2)=O)Cc2ccccc21 30812,N1(C(c2cc(OCC)n[nH]2)=O)CC(C)CN(C(c2onc(Br)c2C)=O)C(C)C1 30813,c1(CNC(=O)CCNC(C2(F)CC3(CNC3)C2)=O)ccc(Br)cc1Cl 30814,N1(C(C(CC2CC2)OC)=O)CCCCC1CC(=O)NC(C)CCCCO 30815,CC1(C)CC(NC(=O)NCc2nc(C(c3ccccc3)(C)C)no2)CO1 30816,C(c1cc(C(F)(F)F)ccc1Cl)=CC(=O)NCC1CN(C(=O)CO)CCCO1 30817,C#Cc1cn(C)nc1C(=O)NC1COCCC1NC(=O)CCCCCOC 30818,CC12CCC(C(=O)NCC3CN(c4nc5cc(Cl)ccc5s4)CCO3)(CC1)CO2 30819,C1(OCCNC(c2nc(C(N3CCCCCC3)=O)cs2)=O)CCCCC1N(C)C 30820,n1(CC)nc(C(=O)NCC2(F)CC(NC(=O)C(F)=CCCF)C2)ccc1=O 30821,C1(C(=O)NC2CC(C)(CNC(Cc3c(C)ocn3)=O)C2)CC(=O)NC(C)C1 30822,Cc1cc2[nH]c(C(N3CCCC(O)(CNC(=O)Cc4csnc4C)C3)=O)cc2o1 30823,N1(C(c2cncc(CC)c2)=O)CCCC(F)(C(=O)NCc2ccccc2C#N)C1 30824,O(NC(=O)C(F)(CNC(=O)CCC(CF)CF)C(C)C)C(C)C 30825,C(C(=O)N=c1cc(C)o[nH]1)NC(=O)C(C)NC(C)=O.C(C1CCC(=O)N1)OC 30826,N1(C(CC(C)OC)=O)CC(CNC(=O)CCc2cncc(Br)c2)C(C)C1 30827,CCCC(C(O)c1nnnn1Cc1ccc(NCc2nnn(C)n2)nc1)N(C)C 30828,C(C(C(=O)N1CC(C)(CN(C)C)C1)C(C)(C)C)NC(C=C(CC)CC)=O 30829,C1(C)(C(=O)NC(C(=O)N(CC(=O)NC(C)C)C)Cc2ccoc2)CCCCC1C 30830,N1(C(c2ccc(N)c(O)c2)=O)CCC(C2CC2)(NC(=O)CCc2cnccn2)C1 30831,Cc1cccnc1CC(=O)NC(C1CCCN1C(c1c(Cl)n[nH]c1C1CC1)=O)(C)C 30832,c1(C2C(NC(=O)NCCc3cc(OC)ncc3)C2)cc(C)cc(Br)c1 30833,CCCC(C)C(=O)NC1CC1CNC(=O)Cc1cccc(NC(=O)CC)c1 30834,S(=O)(=O)(CCC(=O)N(C1CCC(NC(=O)COC2CCCOC2)C1)C)NCCO 30835,C1(C)(COC)CC(CC(=O)OC(C)(C)C)=NO1.C12C3CN(CC13)C(=O)NC2 30836,N1(C(C#C)=O)CCCC(C(=O)Nc2c(C(C)=O)cccc2C)CC1 30837,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 30838,c1(C(N2C(C(=O)NC(CSCC)C)CC2)=O)ncn(C)n1 30839,c1(C(=O)NC2CCC(N(C(CS(CC)=O)=O)C)CC2)ncc(OC)cc1F 30840,O=C(N=c1c(Cl)c[nH]cc1I)C12CC1CN(Cc1cscc1Br)C2 30841,N1(c2nc(C)cc(C)n2)CCCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)CC2)C1 30842,CC(CC(=O)N1CCN(C(=O)CCc2ccc[nH]2)C(CCO)C1)C(F)(F)F 30843,c1(C(N2CCOC(CCF)C2)C(=O)N(CCC(=O)OCC)CC)cc(C)nc(C)n1 30844,CC1C(NC(c2cc(F)ccc2F)=O)CCCN1C(=O)CCCc1cnn[nH]1 30845,N1(C(C2ON=C(CC)C2)=O)CCCN(C(c2cccc(=O)n2C)=O)C(C)C1 30846,c1(C(N2C(C(=O)NCC(C)N(CC(N)=O)C)CCC2)=O)ccccc1C(C)O 30847,C(=O)(CCCC(=O)N1CCC(C(C)NC(c2ncoc2C)=O)C1)NCCC 30848,N1(C(C(CC)CC)=O)CCCC(NC(C23CCN(CC2)CC3)=O)CC1 30849,c1(C(=O)NCC(CC=C)NC(c2cc(OC)ccc2O)=O)cnn2cnnc2c1 30850,N1(C(C=CCN(CCOC)C)=O)CC(OC)CC(NC(=O)CC2CC(OC)C2)C1 30851,C12(C(=O)NCCC3N(C(Cn4nnc(C)n4)=O)CCC3)CCC(C(F)F)(CC1)C2 30852,c1(OC)c(C(N2CC(CC(C)NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 30853,Nc1cnc(Cl)cc1C(=O)NCC1CN(C(=O)C(F)(F)C(O)C2CC2)CC12CC2 30854,n1(CCC)ccc2ccc(NC(=O)C(N3CC(CCO)(C(=O)OC)C3)=O)cc12 30855,n1(CC(=O)NC(C)CN(C)C(C2CSC2)=O)cc(C2CC2)nn1 30856,CN1CCN2CCN(C(c3nc(Br)cs3)C(=O)NC3CCC3)CC2C1=O 30857,N1(C(C(C)N(CC)CC)=O)CCCC1CCNC(=O)CCCOc1cccnc1 30858,C(CN=c1ccc(S(=O)(=O)NC(c2nnc(C)s2)C)c[nH]1)SC 30859,CC1(C)CCN(C(=O)CC2CC2(C)C)C(C(=O)Nc2ccc(F)c(O)c2)C1 30860,c1(CC(=O)N(CCN(C(C2CCC2(C)C)=O)CC)CC)ccc(OC)c([N+](=O)[O-])c1 30861,C1(NC(CCN(C(C2CCN2C(C)(C)C)=O)CC)=O)CCSCC1 30862,c1(C(=O)NCC(CC=C)NC(c2cscn2)=O)ncccc1C 30863,CC(CCCNC(C1(C2CCCO2)CCCC1)=O)NC(C1CCO1)=O 30864,CC1CN(C(c2cnn(C)c(=O)c2)=O)CC(C)CN1C(C1CC=CCO1)=O 30865,C1(CNC(C(C)NC(CC)=O)=O)CC(OC)C(OC)C1.C1C(=O)S1 30866,N1(C(c2nc(C#C)sc2)=O)CCCC(COC)(NC(=O)CN(C)C(C)C)C1 30867,C(=O)(C(O)CC(N)=O)NC(C(N1CCCC(CCC#C)C1)=O)(C)CO 30868,C1(C(N(CCCN(C(Cc2nnc(C)n2C)=O)C)C)=O)CCC(C)NC1=O 30869,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CCCC(NC(C2C3CCCC23)=O)C1 30870,C1(CNC(C(COC)O)=O)CCN(C(C2(c3cccc(F)c3)CC2)=O)C1(C)C 30871,N1(C(N2C(c3[nH]c(C)c(OC)c3C)CCCC2)=O)CCc2c(O)noc2C1 30872,c1(C(N(C(C)C)C)=O)ccccc1Cl.C1CC(=O)N(C)C(C)CN(C)C(=O)CN1 30873,C(=O)(C1CCc2c(Cl)cccc21)CC1CCC(C)(C)O1 30874,CC1=NOC(=O)C1CC(N1CCOC(CNC(C2CN(C)CCO2)=O)C1)=O 30875,c1(C(=O)OC)ccc(CNCC(N2CCN(c3ncc(C)cn3)CC2)(C)C)cn1 30876,Cc1ccc2c(C(=O)NC(C)C(C(C)C)NC(=O)CSC(F)(F)F)onc2c1 30877,N1(C(c2c(C)cc(F)s2)=O)CCC2CN(C(=O)C(C)Cc3ccnn3C)CC2C1 30878,C(C)(C(=O)NCC(CO)NC(C)(C)C)(C(C)C)OC(C)C 30879,N1(C(C(C2CCCC2)NC(C)=O)=O)CCC(C)(CC(N2CC(N(C)C)C(F)C2)=O)C1 30880,c1(N2CCCC(C(N(C)Cc3ccco3)=O)C2)cnc2cccnn12 30881,C#CCC(CC(F)F)NC(=O)C=CC1CCCN1C(=O)CC1COCC(C)O1 30882,C1(C)(C(=O)NC2CCN(Cc3nc(CCC)on3)C2)COC(=O)C1 30883,Cc1ccc(N2CCC(c3nc(C4CCC(C)C4)no3)C2)c(Cl)c1 30884,C1(CCC(=O)NCCN(CCC)CCC)CN(C(=O)CCOC)CCC1C 30885,n1(NC(C2(C)CCSC2)=O)ncc(C(=O)NC2(CNC(C)=O)CC2)c1C 30886,c1(COC(N2CCC(CN3CCCC3)C2)=O)cc(O)nc(C2CC2)n1 30887,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(=O)Cc2ncn3c2CCC3)C1 30888,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 30889,c1(CC(=O)NCC(C)CN(C)C(C2CC2c2ccccc2)=O)c[nH]c(=N)nc1O 30890,c1(OC)ccccc1C1CC1OC.C1(CCNC(=O)CCCC(=O)N)(C)CCOC1.N(C)C 30891,c1(CCC(=O)NC(CN(C)C(c2ccc(F)s2)=O)(C)C)ncc(F)cn1 30892,c1(OC)ccc(C(N2CCCC(C)C2CNC(=O)C(F)(F)C(F)F)=O)c(N)c1F 30893,N1(C(Cc2ccc(OC)cc2F)=O)CCN(C(C2(C)CCOC2)=O)CC2(CC2)C1 30894,c1(CCC)cc(C)[nH]c(=NCC23CC2CN(C(c2cccc(C(N)=O)n2)=O)C3)n1 30895,c1(CC(=O)NCC(C)NC(C2(CS(C)(=O)=O)CC2)=O)ccc(C2CC2)c(F)c1 30896,C(=O)(C1CCc2nccn21)N1C(C)(C)CC(NC(C2(c3cccs3)CC2)=O)C1 30897,c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)C)=O)C2)ccc2c(c1)CCN2 30898,CC1=C(C(=O)NCC2CC(F)CN2C(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 30899,CC(CN1CCOCC1)C(=O)NC(CO)C(C)NC(C1(CC#N)COC1)=O 30900,C#Cc1ccc(C(=O)NC2(C(N3CCC(CC)C3(C)C)=O)CC(O)C2)nc1 30901,N1(C(C2C(CNC(c3ccsc3Cl)=O)CCC2)=O)CC(CO)C2(CCC2)C1 30902,C(=O)(C(F)CC(C)(C)NC(C1(CO)COC1)=O)NCC#CC 30903,C1(C)(C(=O)NCC(c2ncc[nH]2)C)CC(O)CN1C(=O)CN1CCCCCC1 30904,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 30905,CC1(C)CC(C(N2CCOC(C#N)C2)=O)CN1C(=O)CC1CCC(O)C1 30906,c1(CNC(c2cc(F)ncc2NC(=O)C(Cl)(Cl)Cl)=O)ccc(F)c(C2CC2)c1 30907,[N-]=[N+]=NC1CN(C(c2ccc3cc[nH]c3c2)=O)CC1NC(=O)C=CCN(C)C 30908,C1(C)(C(=O)NC2CN(C(C(c3cn(C)nc3C(F)(F)F)C)=O)C2)CCCS1(=O)=O 30909,N1(C(C2CN(C)C(=O)C2)=O)CCC(C2CC2)(NC(c2cc(F)c(F)cc2F)=O)C1 30910,N1(N(C(CC23CC(C(=O)OC)(C2)C3)=O)C)CCN(C(=O)C(F)C2CCC2)CC1 30911,C(=O)(CCC(C)(C)F)N1CCCC(CN(C(c2nncn2C2CC2)=O)CC)C1 30912,C(CN=c1[nH]c(=NCCC2CCCO2)[nH]c2cc(C)ccc12)N1CC(C)OCC1 30913,C=CC(CC)CC(=O)NC(C1CN(C(C2(n3nccn3)CC2)=O)C1)C 30914,c1(C(N2CCC(C(C)NC(C3(F)CC3C)=O)C2)=O)ccnc(NCC(F)(F)F)c1 30915,C(C1(C)OCCc2ccccc21)N(C)C(c1cc(Br)c(F)cc1S(N)(=O)=O)=O 30916,C1(C)(CNC(C2C(CC)C2)=O)CN(C(c2ccc(OC)nc2)=O)C(C)(C)C1 30917,C1(NC(C2C(CC)CCO2)=O)CCN(C(c2ccc(Cl)o2)=O)CC12CCC2 30918,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 30919,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3ccn(CC#N)n3)=O)CC1C2 30920,N1(C(C2(NC(c3cccc(NC)c3)=O)CC2)=O)CCC(F)(F)C(O)C1 30921,n1(CC(=O)NC(C(=O)N(CC)CC2CCCN2C(C)=O)(C)C)nc(C)cc1C 30922,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 30923,c1(CC(C)CN(c2noc(C3CCC4CC34)n2)C)ccccc1 30924,C1(NC(COCC(=O)NC)=O)CCCC1NC(C1CC(Cl)(Cl)C1)=O 30925,C(=O)(CS(=O)(=O)CCOC)NCC1(O)CCN(C(Cc2cc(OCC)no2)=O)C1 30926,c1(C(N(C2CCN(C(C3(C)CCOCC3)=O)C2)CC)=O)nc2ccccc2cc1C 30927,Cc1cc(C)c(C(=O)NCCN(CC(C)O)C(C2CNC(=O)N2C)=O)c(C)c1 30928,C1(C(=O)O)COC2(CCN(C(c3cccc(CNC4CC=CC4)c3)=O)CC2)C1 30929,c1(C(N2CCC(NC(Cn3cc(C(C)=O)nn3)=O)CC2)=O)c(Cl)nn(C)c1Cl 30930,C1(CNC(C(C)C2CCCC2)=O)CC2CCC(C1)N2C(=O)CCC(F)(F)F 30931,N1(C(C(CC)C(C)O)=O)CC2(C1)CN(C(=O)Cc1ccc(C)cc1)CCO2 30932,C1(NC(C(C)(C)C2CC2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 30933,CCCCCC(O)CC(=O)NC1CN(C(=O)Cn2ccc(=O)c([N+](=O)[O-])c2)C1 30934,c1(SC(C)C(=O)NC2(CCNC(=O)C(O)Cn3cncn3)CCC2)ccccc1 30935,C1(n2nnc(C)n2)(C(F)(F)F)CCN(C(C)Cc2c[nH]c(C#N)c2)C1 30936,C(C(F)(F)CCC(=O)NC)n1cc(-c2nc(CC(CCC)(C)O)sc2)nn1 30937,c1(CC(=O)NC(CNC(CN(CCOC)C)=O)C)nc(C(F)(F)F)n[nH]1 30938,C12(C(=O)Nc3cnc(I)cn3)CCCCC1CN(C(c1ccc(O)c(O)c1O)=O)C2 30939,N1(C(c2ccc(OC)o2)=O)CCC(C)(C)C(COC(=O)C(C(C)C)N(C)C)C1 30940,C1(CNC(=O)C=C2CCC2)CN(C(C2(n3cccc3)CC2)=O)CC1(F)CO 30941,C1(C(=O)NCCOCCCNC(c2ccc(C(C)C)s2)=O)CN2CCCC1C2 30942,c1(N(C)C)ccc(CNC(=O)NCC2CNC(=O)CO2)cn1 30943,C1(C(=O)NC2(CO)CCOCC2)CC(C(=O)OC(C)(C)C)=NO1.CC1C=CC(=O)N1 30944,N1(C(C2C(CC)OCC2)=O)CCC2(COC(CNC(c3ccn(C)n3)=O)C2)C1 30945,c1(C(N2CC(N(C(C(C=C)O)=O)CC)C3(C2)CC3)=O)cc2ccccc2o1 30946,N1(C(CC2N(C)CCOC2)=O)CC2(CC(NC(c3ccnnc3)=O)C2)C1 30947,N1(C(C(C)(C)CF)=O)CCC2(CC1)CCN(C(C1(n3cccn3)CCC1)=O)C2 30948,n1(CCC)cc(C(=O)NC2CCCC2CN(C)C(c2csc(O)n2)=O)c(C)n1 30949,O=C(CN1CCc2[nH]ccc2C1)N1CCCC(S(C)(=O)=O)C1 30950,C(=O)(C(C)(C)CC(F)(F)CC)NC(CC)CNC(c1nnnn1C)=O 30951,C1(C(=O)NCc2n(C(C)C)ncn2)CCCCN(C(C2CC23CCC3)=O)C1 30952,N1(C(C2CCC2(F)F)=O)CCC(F)(CNC(C2(c3cccnc3)CCC2)=O)C1 30953,C(=O)(CC(C)CC(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)OC 30954,N1(C(CC(=C)C)=O)CC(NC(c2cncc(OC)n2)=O)CCC1C 30955,C1(C(C(=O)N(CCN=[N+]=[N-])C)F)CCN(C(C2(c3ccno3)CC2)=O)C1 30956,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 30957,C(C(C(C)C)NC(=O)CCC1(C)CN(C(=O)CC2CCC(O)C2)C1)OC 30958,c1(C(N(C(C)C)CCN(C)C(C2CCCN2C=O)=O)=O)cc([N+](=O)[O-])c[nH]1 30959,C1(CCC)(NC(=O)C(COC)N(C)C)CCCN(C(c2ccc(Cl)s2)=O)C1 30960,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 30961,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 30962,N1(C(C(C)Cc2cnn(C)c2)=O)CCC2(CCCN2C(C2CC2(C)C)=O)C1 30963,c1(C(N(C(C)C)CCN(C)C(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 30964,C1(NC(CS(=O)(=O)NC(C)(C)C)=O)CC2CC1CN(C(C1CC(CF)C1)=O)C2 30965,C(=O)(C(F)(F)C(F)(F)C(F)F)NC(C(C)C)(C)CNC(=O)C(C)(C)C 30966,c1(-c2ncc(C(=O)NCC(CC)NC(=O)C(F)CC3CC3)s2)ccc(F)cc1F 30967,N1(C(CCCC)=O)CC2(CC(NC(=O)C(C)C(C)CC)C2)C1 30968,C1(NC(C(C=C)(C)C)=O)CCN(C(C2(n3cnnn3)CC2)=O)CC1C 30969,N1(C(c2cc3cccnc3s2)C(=O)NCCC)CC2CCC(C1)CC(F)(F)C2 30970,c1(C(C)C)ccc(C(N2CCC3C(NC(c4ccccc4)=O)C23)=O)c(O)n1 30971,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 30972,C1(NC(c2cc(-c3ccns3)on2)=O)COCCN(Cc2ccccc2)C1 30973,N1(C(c2ccc(F)cn2)C)CC(CC(N2CCCC23CC3)=O)CC1(C)C 30974,c1(C(=O)NCC2C3CCC(C3)N2C(C2CCCC(F)C2)=O)ccc2n[nH]cc2n1 30975,c1(C(=O)NC2CCN(C(C3(COC)CC=CCC3)=O)C2)ccc2ccccc2c1 30976,C1(NC(CSCCCC)=O)CC2CCC1N(C(c1cc(C(F)(F)F)cs1)=O)C2 30977,O=C(C#CC1CCCCO1)NC1(CNC(=O)CC2CCS(=O)(=O)C2)CCC1 30978,C1(CNC(C=CCOC)=O)CCC(NC(c2cc(C(C)=O)on2)=O)C1 30979,Cc1nc(Cl)nc(N2CC3CN(C(C4CCCS(=O)(=O)C4)=O)CC3C2)c1C#N 30980,C(C(C(=O)NCC(CO)NC(C1(N(C)C)CCCSC1)=O)C(C)(C)C)OCC=C 30981,C1(CNC(CCSCC(C)C)=O)CN(C(=O)Cc2ccsc2)CC1C 30982,CC(C)CC(C)(C)C(=O)NCC1CC(C)CN(C(=O)C(Cl)=CCl)C1 30983,C1(C(=O)NC(C#C)C(C)C)CC(=O)CN1C(=O)CSC1CC1 30984,C1(Nc2ncnc(NC(c3nc(C4CC4)n[nH]3)C)c2C)CCc2ncncc2C1 30985,C1(C2CC2)(C(=O)NC(CC)(CNC(c2cnn(CCO)c2C)=O)CC)CC=CC1 30986,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 30987,CCCCCC(O)CC(=O)N(C1CCCCN(C(=O)C(C)C2(O)CCC2)C1)C 30988,c1(C(C)C)nccc(C(=O)NC(C2CN(C(c3ccccc3F)=O)C2)C)n1 30989,N1(Cc2c(C)c(=O)n(C)c(=O)s2)CCC2(CCOC2=O)CC1 30990,C1(C(=O)N)CCCCN1C(c1ccc(CO)s1)=O.C1(=O)C(CN(C)C)N1.CC 30991,C1(C(N2CCCC2C(=O)O)=O)(CC2CC2)CCCNC1 30992,C1(CNC(C2(CC#C)CC2)=O)CC(N=c2[nH]nc(CO)s2)C1 30993,C(N=c1[nH]c(=NCc2nccn2C(F)F)[nH]c2c1COC2)c1c(Cl)c(Br)ccc1 30994,C(CCCCC(=O)NCCC(O)C1CCCC1)N(C(C=CC(=O)OCC)=O)C 30995,CCCC(COC)CCO.c1(CO)cccc(Cc2nnc(CN)n2CCOC)c1 30996,c1(CC)c(C(=O)NC(C)C(C)NC(c2cccc(OC(F)F)n2)=O)nnn1C 30997,C(=O)(C(O)CC(F)(F)F)NCCn1ncc(CC(=O)N(CC(C)O)C)c1 30998,c1(-c2scc(CC(=O)NCC=CCNC(C(CC)SC)=O)n2)cccc(C#N)c1 30999,c1(SCC)cnc(O)c(C(=O)NC(C)CCCNC(c2cc(N)ccc2C)=O)c1 31000,C(CO)(CCC(C)C)NC(CSCCNC(Cc1scc(C)c1)=O)=O 31001,c1(C(=O)NC(CC(=O)NCCc2ccnc(C)n2)C)ccc2cc[nH]c2c1 31002,c1(CNC(c2ccc(N(C)C)s2)=O)ccc(CN(C)CC2CC2)cc1 31003,C1(O)(C(C)NC(CC)=O)CCN(C(c2cccc(-n3cncn3)n2)=O)C1 31004,C1(C(=O)OC)CCCC12CCN(C(c1cc(N)nc(I)c1)=O)C2 31005,c1(C(=O)NCCCN(C(=O)C(C#N)C(C)(C)C)CC)cc(S(C)(=O)=O)co1 31006,N1(C(COCCCOC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1C(C)C 31007,CC1(C)C(CC(N2CC(CNC(=O)Cc3ccc(O)nc3)C2)=O)C1(C)C 31008,CC1CC(NC(c2nncs2)=O)CCN1C(=O)CCN1CCOCC1 31009,N1(c2nnc(C(=O)OCC)s2)CCC2(CCC2)C(NC(=O)C2=COCCC2)C1 31010,CC(C)C(C)C(CNC(C1(Br)CC1)=O)NC(=O)C1CC1 31011,C(=O)(C(=O)C(F)(F)F)NCC(C)CN(C(=O)CNC(=O)C1CC1)C 31012,N1(C(CCC(=O)NC)=O)CCCCC(C2CN(C(c3ccc(F)s3)=O)C2)C1 31013,N1(C(Cc2c(C)non2)=O)CCC(C2CCCCN2C(=O)COCCF)CC1 31014,Cc1cc(Br)cc(C)c1OCC(=O)NC1CC1CNC(=O)C1=CCOCC1 31015,Cc1c(C(N2CCC(CCNC(=O)C=C3CCCC3)CC2)=O)c(C(F)F)nn1C 31016,N1(C(c2nnn(C)c2C(F)(F)F)=O)CCCC(NC(=O)Cc2cnco2)C(F)C1 31017,CCCCCCN(C(=O)C(C)N(C(=O)CCC=C(C)C)C)CCCC 31018,N1(C(CC=C)=O)CCOCC12CCN(C(c1cc(C)no1)=O)C2 31019,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31020,C(=O)(CCCCCN(C(=O)CC=CC(C)(C)C)C)N(C)CC1CC1(C)C 31021,c1(CNC(C(C)c2ccsc2)=O)ncc(C(=O)NCC23CC(CO)(CO2)C3)cn1 31022,c1(C(=O)NCCOCCN(C)C(C2CCS(=O)(=O)CC2)=O)cc(Cl)n[nH]c1=N 31023,c1(C(N2C(COC)CCCC2)=O)cccc(C)c1C.C=CCCC(=O)N1CC=CC1C 31024,C(=O)(C1=C(C)CCOC1)N1CCC(F)(C(N(CCCCCC)C2CC2)=O)C1 31025,N1(C(C2CCCC2C(=O)Nc2ccc(NC=O)cc2)=O)CCC2(CCCO2)C1 31026,CS(=O)(=O)c1cc(NC(=O)NCc2ccc(Cl)cc2N2CCCC2)cc(F)c1 31027,C(CC(O)CNC(=O)C(c1ccccc1)n1cc(Cl)cn1)NC(C1CCC1)=O 31028,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31029,C(CCCCCC(=O)O)NC.C(=O)(CCCF)C(=O)CC1CC(=O)C1 31030,N1(C(c2ccn(CC)n2)=O)CCC2CN(C(C3(c4cc(C)on4)CC3)=O)CCC12 31031,c1(CN(C(=O)C(C)(C)C2CCOC2)C)cccc(C2CC2)c1.C12(O)CN(C1)C2=O 31032,c1(CC)cc(C(N2CCC2C(=O)N(C)C)=O)ns1 31033,c1(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)cc2c(Cl)cccc2[nH]1 31034,c1(OC)cc(N)c(F)cc1C(=O)NC1(CN(C)C(c2ccnnc2S)=O)CC1 31035,C#Cc1ccc(C(N2CCC(O)(CCNC(c3ccc(Cl)s3)=O)C2)=O)cc1F 31036,C1(NC(c2scc(COC)c2)=O)CCN(C(c2cnc3sccn23)=O)C(C)C1 31037,C1(NC(C2(CCNC(=O)C(F)n3ccnc3)CC2)=O)COCCC1(F)F 31038,c1(CC(=O)NC2(C)CCN(C(c3n(CC)cnn3)=O)C2)nnc2n1CCCC2 31039,C12(NC(C3CCC4(CCC4)CO3)=O)CCCC1N(C(c1cncs1)=O)CCC2 31040,N1(C(N2CCOCC2)C(=O)NC(c2ccccc2)COC)C2CCC1CN(C)C2 31041,CC1CC(C(=O)NCCC2(C(=O)N(CC(C)O)C)CC2)=NO1 31042,C1(NC(C2CCC(C)C2)=O)CC2(NC(=O)CCCc3nc(C(C)C)no3)COC1C2 31043,C(C)(CCCCO)NC(C(CNC(C(CC1CC1)OC)=O)OC)=O 31044,c1(OC)ccccc1C(CNC(=O)CCC1CCCO1)NC(c1cc(=O)cc[nH]1)=O 31045,c1(C(=O)Nc2cc(I)ccn2)cccc(OC(F)(F)F)c1.C12CC1CNC2=O 31046,C1(NC(C(COC(C)=O)C)=O)CC=CCC1C(=O)NC1C=CC(CO)C1 31047,C1(NC(c2cc(Br)cs2)=O)CCCN(C(c2ccc(I)c(O)c2)=O)CC1 31048,c1(CN(C2CCC(C(C)O)CC2)CC2CCCC2)ccc(F)c(Cl)c1 31049,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=CCCC(C)C 31050,c1(C(=O)NC(CC(C)NC(Cc2cccc(CC)c2)=O)C)cc(C)c(C)nn1 31051,C1(NC(=O)NCC2CCC3CCCC3C2)CCc2ccccc2OC1 31052,c1(OCCN(CC(C)N)C2CC2)cccc(S(C)(=O)=O)c1 31053,CCCCC(C(=O)N1CCN(C(C2CCC3CC23)=O)C(CCO)C1)C(C)C 31054,C(C)(C(=O)NC(C)CCn1cc(CSCC)nn1)(C1CCCO1)OC 31055,N1(C(C=CCCC(C)NC(C(OCC)OC)=O)=O)CCCCCC1 31056,C1(NC(c2ccc(F)c(C)c2O)=O)CCC2C(CCN2C)C1 31057,C(=O)(C(CO)N(C)C)NCC(C1CC1)NC(CC1(CC(=O)OCC)CC1)=O 31058,C(CCCC(CO)NC(C1CC2CC1CC2O)=O)NC(C1CCC(=O)C1)=O 31059,C1(C(N2CCC(C)(CCO)C2)=O)(NC(CC2C(C)C(=O)CC2)=O)CCOCC1 31060,C1(c2n(CCCCCC)nnn2)(NC2CCCCCC2CO)CC2COC1C2 31061,c1(CC(N2CCC(CCOC)(NC(=O)CC3CC3)C2)=O)ccc(Cl)c(C)c1F 31062,C1(C(N(CC(C)NC(c2c(C(F)(F)F)cccc2O)=O)C)=O)CC(F)(F)C1(C)C 31063,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31064,c1(C(N2CC(CNC(C3CCN(C)C3=O)=O)OCC2)=O)ccnc2ncnn12 31065,c1(C(=O)NC(CCCC)CNC(c2conc2C2CC2)=O)cnc2c(c1)NCC2 31066,c1(CC)nc(C)c(C(=O)NC(C)CNC(c2nnsc2SC)=O)o1 31067,c1(C(N2CC(O)(C(C)NC(CC(C)c3ccco3)=O)C2)=O)c(F)ccc(F)c1F 31068,C1(CNC(C=CCC)=O)CCC(C)(C)CN1C(=O)C=Cc1nc[nH]n1 31069,N1(C(CSCC)=O)C2CCC(C2)C1C(=O)NCCc1cnc(C)o1 31070,c1(C(N2CC3(C(=O)NC4CCCC4(F)F)CC2CO3)=O)ccc2[nH]ccc2n1 31071,C12(C(N3CC(CC=C)(NC(=O)C4=C(C)CCC4)C3)=O)CC3CC(C(=O)N1)C2C3 31072,c1(C(=O)NC2C(CNC(=O)CC3C=CS(=O)(=O)C3)CC2)cnc2ncccn12 31073,c1(C(N2CCCC(C(=O)Nc3ccc(Cl)cc3CO)C2)=O)cc2ccoc2cn1 31074,c1(OCC)cnc(C(=O)NC2COCC2NC(=O)CCc2ccsc2)c(Cl)c1 31075,CCC(COC)C(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)C)C1CC1 31076,c1(CC)cc(C)c(C(=O)NCCC(C)NC(C23CC(C)(CO2)C3)=O)o1 31077,C1(C(N2CC(C(=O)NCC(F)(F)C(N)=O)(CC)C2)=O)CC(O)C(F)C1 31078,C=CC1(N(C)C(C)=O)CCCN(C(=O)C(CC(C)C)OC)C1.C(=O)CSCCCC 31079,N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)CCCSc2ccccc2)C(C)C1 31080,C1(C)(CNC(C(C)N(C)C)=O)CCN(C(c2cnn(C3CCOCC3)c2)=O)C1 31081,c1(C(N2CCC(NC(C3(C)CC(C)C3)=O)CC2C)=O)ccc2ncccc2c1F 31082,C1(CC(=O)NC(C#CC)(C)C)COCCN1C(c1ccc(CC#N)cc1)=O 31083,CCCC(=O)N(CCN(C(=O)Cn1cccc1)CC)CC 31084,C1(CC=C)(C(=O)N(CC(C)O)C2CC2)CCNC1 31085,Cc1cc(NC(C2CCN2C(=O)C(c2ccc(Cl)s2)=O)=O)cc(Br)c1 31086,C1(C2C(=O)NC(C=C)C(=O)N2)CC(=O)NC(C)C1.C(C)(C)(C)OC(=O)NCCO 31087,c1(OC)nc(C)cc(=NC2CCC(NC(=O)CCCn3ccnc3)C2)[nH]1 31088,N1(C(CC2C(CC)C2)=O)CCN(C(C2CCC(F)(F)CC2)=O)CC(CO)C1 31089,N1(C(CCCNC(C)=O)=O)CCN(C(=O)CC(C)C(C)C)CC(CO)C1 31090,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31091,CCCCCCCC(F)C(=O)N1CC12CN(C(=O)Cc1ccccc1F)C2 31092,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NC1CC=CC1)N(C)C 31093,CC1(C)CN(C(C2(CNC(c3cc(CO)ccn3)=O)CCC2)=O)CCC1CO 31094,Cc1scc(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)nn3C)=O)C2)C)c1N 31095,C(=O)(C(CC(C)C)c1ncco1)OC.c12ccccc1OC(C)C(=O)N(CC)C2 31096,C(=O)(C(C)(O)C(C)C)NCCCNC(C1C(Cc2c(OC)cccc2)OCC1)=O 31097,Cc1oc2cc(C(=O)NCC3CC3NC(c3nccc4n[nH]cc34)=O)[nH]c2c1C 31098,c1(C(=O)NC(CNC(c2occ(C(N)=O)n2)=O)C2CCC2)ccc(CO)cc1 31099,C1(C(=O)NCC(CC)(CC)NC(=O)CC2C(C(C)C)C2(F)F)CCCS(=O)(=O)C1 31100,C1(NC(C=CC(CC)=CC)=O)CC2CN(C(=O)Cn3c(C)csc3=O)CC2C1 31101,CCC(C)(C(=O)N(C1CCN(C(C2CCCC(C)(C)C2)=O)CC1)CCO)C(N)=O 31102,C1(C(=O)NCC(CO)NC(COCCCC)=O)CC2CCC1O2 31103,c1(C(N(C(C(=O)N(CC(C)O)CCOC)C2CC2)C)=O)ccc2c[nH]nc2c1 31104,Cc1nc(N)cnc1C(=O)NC1(C)CC(NC(C2CNC(=O)C2)=O)C1 31105,N1(C(C2C(F)(F)CN(C(COCC)=O)C2)=O)C2CCCC1C(CC)C2CC 31106,CCC(C(=O)N1CCC(NC(=O)CN2CCN(C)C(=O)C2)C1C(C)C)C(F)(F)F 31107,c1(C(C(=O)OCC)N(C(CC(CC)C)C(=O)NC)C)noc2ccc(Br)cc12 31108,C1(c2scc(CC(=O)NC(C(C)NC(CCCC)=O)C)n2)CCCCCC1 31109,C(C)(C(C(C)C)NC(=O)C(C)OC1CCCC1)NC(c1c(CC)nn[nH]1)=O 31110,C(=O)(C(O)CC(N)=O)N1CCC(NC(Cc2ccc(C(C)=O)s2)=O)(CO)C1 31111,N#Cc1c[nH]c(C(=O)NCCC2(C(N3CCCC4CC34)=O)CCC2)c1 31112,C1(NC(c2cccc3[nH]ncc23)=O)CCCN(C(=O)Cc2csnn2)CC1F 31113,N1(C(C(CC(=O)O)NC(CC=CC)=O)=O)CCc2ncc(C(N)=O)cc2C1 31114,c1(C(=O)NC2CC3(C2)CC3NC(C2CCCSC2)=O)noc2c1CC(F)(F)CC2 31115,CCCC(O)C(=O)NCC(C)CNC(=O)C(c1ccc(OC)cc1)C 31116,C1(C(=O)OC)(C(=O)OC)CC2C=CC1CC2.c12cccc(c1)NC(=O)C2N 31117,c1(C(=O)N(c2ccn(-c3ccccc3)n2)c2nn[nH]n2)cc(Br)c(O)cc1Br 31118,CCC(CCC(=O)N1CCC(C)C1NC(C=CC(=O)NC1CC1)=O)OC 31119,C1(NC(c2c(C)nsc2)=O)CCCCC1NC(=O)C(C)c1ncco1 31120,N1(C(C2CCN(OC)CC2)=O)CCC(C2(NC(=O)C(C)S(C)(=O)=O)CCC2)CC1 31121,C1(CNC(CC(C)C2CC2)=O)C2CCC1CN(C(c1cc3ccnn3cn1)=O)C2 31122,c1(NC(=O)NC2CC2c2cncc(C)c2)cccc(Br)c1C#N 31123,C(C(C)(O)C(=O)N1CC(NC(=O)CCc2c(C)noc2C)C(C)C1)OC 31124,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31125,c1(NC(C(C)SCC=C)=O)nc(Cl)ncc1NC 31126,CC1(CNC(=O)CC2COCCO2)CCCN1C(c1ccc(NC=O)cc1)=O 31127,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccnc5)=O)C34)n[nH]c2c1 31128,N1(C(C)=O)CCCCC1CC.C(=O)(CCCc1nnc(C(C)C)o1)NC 31129,C(=O)(C(CC)CC(F)F)NCCNC(C(CSC)NC(C)=O)=O 31130,N1(C(CC2(C)OCCO2)=O)CC(F)(F)CC1CC(=O)NCCC1CCCC12CC2 31131,C1(C(CNC(CN(c2ccccc2)C)=O)=O)CCCN1C(=O)COC1CCC1 31132,C1(C)(C(=O)NC(C2CCCCC2)C(C)NC(=O)CC2CC2)CCCCO1 31133,N1(C(CCCC#C)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CC1C 31134,C1(CC)(NC(c2ccnn2CC(C)C)=O)CCCN(C(=O)CSCC(C)C)C1 31135,CC1(C)CN(C(=O)C(c2ccccc2)F)CC1NC(=O)C(c1ccccn1)O 31136,c1(NC(CCCC=C)C)ncc(S(=O)(=O)NCCSC2CCOCC2C)cc1Cl 31137,c1(CNC)cc(F)c(F)cc1Br.c12nc(C)c(s1)C(=O)NC2C 31138,C(N=c1ccnc(CN2C(=O)CCC2=O)[nH]1)c1c(C)cccc1F 31139,C1(C(OCC(=O)OCC)C2CC2)CN(N2CCCCC2C)C1 31140,Cc1cc2ccccc2nc1SCc1nnc(-c2ccc(F)c(C(F)(F)F)c2)o1 31141,c1(NCC(=O)OC)sccc1C(=O)OC.c12cc(on1)C(c1ccccc1)S2 31142,C(=O)(C1=CCC(C)CC1)N(CCC)CCNC(C1(CC(C)(C)C)CC1)=O 31143,C1(C(=O)NC(CCCNC(CCN(CCCCC)C)=O)(C)C)CCC(N=[N+]=[N-])C1 31144,C(=O)(C1=CCCCC1C)N(CC1=C(C)CCC1)CCN(C(=O)CCOC)C1CCC1 31145,C(C)(CC1CCC1)(C(=O)NCCCC(F)(F)F)NC(C(c1cccc(F)c1)C)=O 31146,N1(CC(=O)OCCCCCF)CCN(C(c2cnc(C3CC3)o2)=O)CC1 31147,C1(C#N)(C(=O)NC(CC)(C)CCNC(=O)CC2(O)CCC2)CC12CCC2 31148,N1(C(CC(C)(C)C2CC2)=O)CCN(C(C2C3CN(CC(F)F)CC23)=O)C(C2CC2)C1 31149,C1(CC)CN(C(=O)CCNC(N)=O)CCC1NC(=O)CCCCNC(N)=O 31150,N1(C(C=O)CCC(C)C)CC2CC3CCCN3C2C1.CCC(C)(C)OC 31151,c1(C(N(C)CCN(C(=O)C(O)C2CCC2)C)=O)c[nH]c(Cc2cscn2)c1 31152,CC1(C)COC(CC(=O)NC(C(=O)N2CC(CO)C2)c2ccco2)C1 31153,C1(CNC(C2(SC)CCC2)=O)CCCN1C(C1CCC(=O)C1)=O 31154,C1(C(=O)NCCSCC)C2CC3C(C2NC(C2(C)C(C)(C)C2(C)C)=O)C13 31155,N1(C(c2scc(C)c2)=O)CC(CNC(C2SC3C=CC2CC3)=O)C(C)(C)C1 31156,n1(CC)nc(C(=O)NC2CC23CC(NC(=O)COCc2nc[nH]n2)C3)c(C)n1 31157,C1(NC(CCc2c(C)n[nH]c2C)=O)COC2CN(C(c3ocnc3C)=O)CC12 31158,c1(C(C)C)ncc(NC(=O)C(O)CCNC(C2(F)CCC2)=O)cn1 31159,c1(CNC(CC2(NC(C3C(C(C)(F)F)C3)=O)CC2)=O)nc(C(N)=O)cs1 31160,CCCC(C(=O)N1CCCC(NC(=O)CCCn2ccnc2)CC1)S(N)(=O)=O 31161,n1(C2CN(C(C)=O)C2)cnc(=N)[nH]1.C12(CC1)C(=O)NCC(=O)N2 31162,N1(C(C(C)NC(CC)=O)=O)CC(F)(F)CC1CNC(c1cccc(C)n1)=O 31163,c1(NCc2c(C(=O)OC)n[nH]c2)c[nH]ccc1=NCC1CC1.C1(=O)COCCN1 31164,c1(-c2cc(C)[nH]n2)cccc(C(=O)N(CCCNC(=O)C(O)CC2CC2)CCO)c1 31165,S(=O)(=O)(c1ccc(Br)cc1NC1CN(C2CC2)CCO1)NCCC=C=C 31166,c1(CC)cncc(C(=O)NC2CC2C(=O)NCc2cnn(C(C)C)c2)c1 31167,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31168,C1(C(=O)NC(CCCNC(c2c(C)n(C)cn2)=O)(C)C)CCCS(=O)(=O)C1 31169,c1(CC(C)NC(c2ccnnc2)c2nnnn2CC(F)F)cccnc1 31170,c1(C(N)C(=O)N(C2CCCC2)CCF)ccc2nn[nH]c2c1.c12ccc(cc1)[nH]2 31171,Cc1cnc2n1CCC(C(=O)N(C)CC1(O)CN(C(=O)C(O)C(C)(C)C)C1)C2 31172,c1(C(=O)NC2CC(C)(COC)N(C(=O)C=C(Cl)Cl)C2)ccc2ncc(=O)[nH]c2c1 31173,C1(CNC(CN2CC(C)(C(F)(F)F)C2)=O)COCC1(C)C.c12cncc(c1)N2 31174,C(=O)(CCC(C)OC(c1ccc(C2CCC2(C)C)cc1)=O)OCC 31175,CCCCC(C(=O)N1CC(N=[N+]=[N-])C1)NC(=O)CCN1CCCCC1 31176,c1(N(CC(=O)NCCNC(c2c(C)nns2)=O)C)ccc(C#N)cc1F 31177,C1(CNC(c2cnsn2)=O)CC2CN(C(C3(n4cnnn4)CCCCC3)=O)CC12 31178,c1(C(N2C(C(=O)NCC3CCCO3)COCC2)=O)ccc(O)c(F)c1 31179,CC1SCCC1NC(=O)CCOCCCNC(=O)C(C1CCOCC1)O 31180,c1(OC)ccccc1CC(=O)N(CC(C)NC(c1cc(O)cs1)=O)C 31181,c1(C(=O)NC2(COC)CN(C(CC3C(CC)C3(F)F)=O)C2)nnn(C)c1N 31182,C1(F)(CNC(C(F)=C(C)C)=O)CCCN(C(=O)CCCC2CCC2)CC1 31183,CCC1=NOC(CC(=O)N(C)CCNC(=O)CCc2ccncc2Br)C1 31184,C(C)(CCC(=O)NC(Cc1cc[nH]n1)C(=O)NCC(c1nccs1)C)OC 31185,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 31186,C1(CNC(CCSCCC)=O)CCCCN(C(C2(C)CSC2)=O)C1 31187,C(CC(=O)NC(C1(C(=O)NC(C)Cc2cnc[nH]2)CC1)C)N(C)CC 31188,N1(C(c2cncc(CC)c2)=O)CC(NC(=O)C(CO)NC(=O)C2CC2)CC(O)C1 31189,N1(C(C2C(C)(C)CC(=O)NC2)=O)CC23CCCC2(C1)CN(C(c1ccsc1)=O)C3 31190,N1(C(C2C(OCC)C2)=O)CC2CCC1CC2NC(C1(CN(C)C)CCCCC1)=O 31191,C(=O)(C1=CS(=O)CCC1)N1CCC(C(C)NC(C2(OC)CCCCC2)=O)C1 31192,Cc1cc(C)c(C#N)c(NCC(C)(C2CC2)NC(=O)CC2CCC(C)(C)CC2)n1 31193,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)Cl)=O)CC2O)cc1Cl 31194,c1(C(N2CCOCC(NC(C3ON=C(C)C3C)=O)C2)=O)sc([N+](=O)[O-])cc1Cl 31195,c1(NC)cccc(C(=O)NCC2CCC(CNC(C3(C(F)(F)F)CC3)=O)C2)n1 31196,c1(OC)cnc(F)cc1C(=O)NC(C)(C)CN(C)C(C1CCCSC1)=O 31197,C(=O)(C(C)C(=O)OC)NC1(C(=O)NC2(C(=O)NC)CCC2)CC(C(N)=O)C1 31198,N1(C(C(F)=CCC)=O)CCC2CCN(C(=O)C#CC3CC3)CC12 31199,c1(NC(N2CCN(C(C)C(=O)OC(C)(C)C)CC2)=O)nccn2nccc12 31200,c1(CN=C(NCC2(O)CC(C)(C)C2)NC2CC2)cc2n(n1)CCC2 31201,C1(Cn2cc(C(N(CC)CC)C)nn2)CCN(C(=O)CC2COCCO2)CC1 31202,c1(C(N2C(CNC(=O)COCC3CCOC3)C=CC2)=O)nccc2cc[nH]c12 31203,c1(C(=O)NC(C#C)(C)C2CN(C(=O)C(C)OCC=C)C2)sccc1Br 31204,c1(C(=O)Nc2cccc(-c3cccnc3)c2)cc2cncn2c(O)n1 31205,N1(C(c2ncccc2C2CC2)=O)CC2(CCCCN2C(=O)CC2OCCO2)C1 31206,C12(C(=O)NCC3(NC(C4(Cl)CC4(F)F)=O)CC3)CC(CO)(C1)OC21CCC1 31207,C1(NC(c2cc(SC)oc2)=O)CCCCC1CNC(=O)CSc1nncs1 31208,c1(OCC)c(C(N2CC(CCNC(C3(COC)CCC3)=O)C2)=O)nc(O)nc1C 31209,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31210,N1(C(C2(n3cc(CSC4CCC5(CC5)C4)nn3)CC2)=O)CCCc2ccccc21 31211,c1(CC(=O)NC2C(NC(Cn3c(C)ccn3)=O)CCC2)ccc2cccnc2c1 31212,c1(NC(N2C(COC)(CNC(=O)CCSC)CCC2)=O)nn(C)c2c1COCC2 31213,CCCCN=C(NC1CCN(CCNC(C)=O)C1)NC1CCS(=O)(=O)C1 31214,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2C(C1)CN2C(C1CCCNS1(=O)=O)=O 31215,C1(NC(C(C)S(C)(=O)=O)=O)CCOC2(CCN(C(=O)CCC3OCCO3)CC2)C1 31216,Fc1cc2nc(CN3CCC3c3ccccc3)[nH]c2c(F)c1F 31217,C1(N(C(=O)CC2CC23CC3)CCO)CCN(c2ncccn2)CC1.C12CN(C1)C2=O 31218,N1(C(C2(C)CCSCC2)=O)CCC(F)C(NC(C2CC3CCC3C2)=O)C1 31219,C(=O)(C(C)CC(C)C)NC1C(CNC(c2nc(OCC)sn2)=O)CC1 31220,N1(C(C=C(C)Cl)=O)CCC2CCN(C(c3ccc(-c4ncc[nH]4)cc3)=O)CC12 31221,c1(C(N2C(C(N3CCC(COCC)C3)=O)C=CC2)=O)ncccc1Cl 31222,N1(C(c2sccc2CO)=O)CCC(C(C)NC(C2CCN2S(C)(=O)=O)=O)C1.C=O 31223,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(C12CCC1CC2)=O 31224,c1(NCC)cccnc1C(N1CCOC(CCNC(=O)CCN2CCCC2)C1)=O 31225,C(=O)(CC1=CCN(C)CC1)NC(CCC)C(=O)N(C(C)CCO)C 31226,C12CCCN(C1)C2=O.c1(C=O)cnco1.C(C(Cl)=CCl)N(N(CC(=O)OC)C)CC 31227,CON1CCC(CC(=O)NC2CCC(CNC(C34CC(CO3)C4)=O)CC2)CC1 31228,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31229,C1(C(=O)NCCN(C(C2(COCC)CC2)=O)C2CC2)CCCC(F)(F)C1.COC 31230,C1(CC)CC(CNC(c2c[nH]nc2CNC(c2ccn(CCF)n2)=O)=O)CCO1 31231,C1(CC)CCN(C(c2cc(C)oc2C)=O)C1CNC(=O)C=CC1CCOC1 31232,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(c2ccc(CC(C)C)s2)=O)C1 31233,C1(CN(C(C)C=O)C(c2cc(C)oc2C)=O)CC2(CCOCC2)C1.CCCN 31234,c1(C(N(CCNC(CC)=O)CCOC)=O)ccc2c(c1)CCCCN2 31235,O=C(CCC(F)(F)F)NCC12CC1CN(C(c1cnccc1C(F)(F)F)=O)C2 31236,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(=O)CCc1c(C)noc1C 31237,C1(C(N2CCC(C(=O)NCCc3ccc(F)nc3)(CO)C2)=O)(CC)CNC(=O)C1 31238,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31239,C1(COC)(CNC(C2C(C)C2C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 31240,C1(NC(=O)COCC2CCOCC2)CC2CCC(C1)N2C(=O)C1=NNC(=O)C1 31241,C1(O)(CCNC(C2CCCO2)=O)CCCN(C(c2occc2C(F)(F)F)=O)C1 31242,C1(C(=O)NC(CC)(C)CNC(C2C3(CC3)C23CC3)=O)CCc2c(ncn2C)C1 31243,C1(NC(c2cn(CCC)nn2)=O)CC2CC1N(C(c1nnc(O)nc1O)=O)C2 31244,N1(CC(=O)NCCOC)Cc2[nH][nH]c(=NC(=O)c3cc(I)c(F)cc3Cl)c2C1 31245,c1(CNC2C(NC(=O)OC(C)(C)C)CC=CC2)cc2c(o1)CCCC2 31246,Cc1c(C(=O)NC2CC2C(=O)Nc2cnccc2CC2CCC2)cccc1O 31247,C1(C(N)=O)CC(CNC(=O)NCc2n[nH]c(C(F)(F)F)n2)CO1 31248,C12(CN(C(=O)CC3CCOCC3)C1)C(=O)C2=O.N1(CCN)CCC1CSC 31249,Cc1sc(Cl)nc1C(=O)NC1CN(C(c2ccccc2Br)=O)CC1O 31250,C#Cc1cncc(C(=O)NCC(CCNC(c2ccc(C(F)(F)F)[nH]2)=O)OC)c1 31251,N1(C(C(CCC)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31252,c1(CCC)cccc(C(C(=O)NCC2CCCCC2)N(CC(N)=O)C)c1 31253,C(C1CN(C(c2cccn2C)=O)CC1C(=O)Nc1cnc(C(C)C)nc1)=CC 31254,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCNC(=O)C(C2CCOCC2)O)cc1 31255,C(=O)(N=c1cc(-c2cnc3n2CCCC3)o[nH]1)N(c1c(C(C)C)nsc1)C1CC1 31256,c1(C(C)C)ccc(N)c(C(N2CCN(C(=O)C3=CCC3)C(CO)C2)=O)c1 31257,N1(C(C(c2c(C)cncc2)C)=O)CC(CNC(=O)C=Cc2cc[nH]c2)CCC1C 31258,CC1CCN(C(c2ccncn2)=O)CC1NC(c1c[nH]nc1F)=O 31259,Cc1cc(C(=O)NC2CC(NC(C3CCC(C(N)=O)O3)=O)C2)cc(N)c1O 31260,C(CC(CC)C(=O)N1CC(=O)NCC1C(=O)NCC1(F)CC(O)C1)=CC 31261,C12(CNC(Cc3n[nH]c(=N)s3)=O)CCC(CN(C(=O)C3=COCC3)C1)C2 31262,c1(C(=O)OC)ccccc1C(=O)NC(CNC(=O)C(C)CC1CCCC1)C1CCC1 31263,N1(C(C2(C(C)(C)OC)CC2)=O)CC(CNC(=O)CC2(CC3CC3)CC2)OC(C)(C)C1 31264,CC(C)(CCC(=O)NC1COCC1NC(=O)C(Cl)=CCl)c1ccc(Cl)cc1 31265,C(=O)(CCCC(C)C)NCCN(CCOC)C(c1cc(C2CC2)on1)=O 31266,C(=O)(C(F)CC(C)C)NCCCCCCNC(C1N(CCC)C(=O)CC1)=O 31267,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2(CF)CC2)=O)C1 31268,c1(C(N2CCCC(NC(CC)=O)(COC)C2)=O)cccc2c1ccn2C(C)C 31269,C1(C)(CC)C=C(C(=O)NC(C)CCNC(c2ncc(Br)cc2N)=O)C1 31270,C(=O)(C=CS(C)=O)NC1(C(C(=O)NCC2C(N(C)C)COC2)(F)F)CCC1 31271,C1(C)(C(=O)NC(CNC(c2ccc(C(C)=O)nc2)=O)(C)C2CC2)CCCS1(=O)=O 31272,N1(C(c2ccc(C(=O)NC)cc2)C(=O)NCC(C)C)CCC2(CC1)N=N2 31273,C(=O)(C1Cc2ccc(F)cc21)NC1CN(C(C2ON=C(C)C2)=O)CC2(C1)CC2 31274,c1(C(=O)Nc2scc(CC(=O)NCC(C(C)O)O)n2)ccc(Cl)nc1O 31275,C(=O)(CS(=O)(=O)CCOC)NCCN(CCC)C(c1cc(CCCO)on1)=O 31276,CC(C)CCCC(=O)NCC1(F)CCC(NC(C2CCC(C)(C)OC2)=O)C1 31277,N1(CC)CCC(C(=O)NCCCCN(C)C(c2c[nH]nc2-c2cnn(C)c2)=O)C1 31278,CC(C)C(C)(CNC(=O)CN1CC2CCC1C2)NC(=O)CN1C(=O)CNC1=O 31279,c1(CCC(N2C(CNC(c3c(C)cc[nH]3)=O)CCC2)=O)ccc(C(F)(F)F)cc1Br 31280,c1(C(=O)NC2CCCN(C(C(C)(O)C3CC3)=O)C2)noc2cc(Cl)ccc12 31281,c1(C(N(CC(C)NC(=O)C(O)CN(C)C(C)=O)CC)=O)cccc(NC)c1 31282,C(C(C(=O)NC1(CC)CCN(C(=O)C(CN(C)C)CC)CC1)C(C)(C)C)OCC=C 31283,C(=O)(CCCC(N)=O)NCC(C1CCN(C(c2cccc(N)c2)=O)CC1)(C)O 31284,CC(CF)CC(=O)NC1CCCC1NC(=O)CCn1cccc1 31285,c1(NC(C2CC(F)CN2C(c2ccnc(Cl)c2)=O)=O)cc(F)c(F)cc1Br 31286,c1(NC(CCNC(CC(CC)NC2CC=CCC2)=O)=O)ccc(Cl)c2ccccc12 31287,CC(CCCNC(c1cc(Cl)c[nH]1)=O)NC(=O)C(c1ccccc1)OC(C)(C)C 31288,Cn1nc(C(C)(C)C)cc1S(=O)(=O)NC(c1cccc(Cl)c1)C(N)=O 31289,C(C(=O)N(CC(O)C1CCC1)C)(C1CCOC1)N(C(C1(N(C)C)CC1)=O)CCO 31290,C1(C(CNC(CN(C2CCSC2)C)=O)NC=O)(CN2CCOCC2)CCCC1 31291,C(=O)(CCC(F)(F)F)N1CC(CCNC(=O)Cc2cscn2)OCC1 31292,C(=O)(C(C)(C)C(C)(C)O)NC1C=CC(CC(=O)NCC(C)C2CCC2)C1 31293,Cc1nc(NCC(C2CCC2)C2CCC2)cc(NC2CC2c2ccccc2)n1 31294,c1(SC)nc(N2CC3CCC2CN3C(c2cncn2C(C)C)=O)c(C)c(Cl)n1 31295,O(C1CCCc2nc(Cl)ccc21)C(=O)CCc1cnc(C2CCC2)o1 31296,C(=O)(CC1OCCc2ccccc21)NC1CN(C(C2C(C)(C)C2(F)F)=O)C1 31297,C1(NC(=O)NCC2(C)COC2)CCOC2(CCOC2)C1 31298,C1(N(C(=O)CNC(C2CCC2)=O)C)CCN(C(C2CCC2n2ccnc2)=O)C1 31299,c1(CC(=O)NCCN(C(=O)CC2COCCO2)CC)ccc(OC(F)F)cc1 31300,Cc1[nH]nc(C(C)C)c1C(=O)N(CC(C)CNC(c1ccc(C(C)C)cc1)=O)C 31301,C1(COC)(CNC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)C=C(C)Cl)C1 31302,c1(CC)ncc(CNC(C2(CNC(=O)C=CC3CC3)CC2)=O)[nH]1 31303,c1(OCC)ccc(C(N2CC(F)CC2C#N)C(=O)NC2CC2)c(C)c1Br 31304,C#Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cnc(C4CC4)[nH]3)=O)C2)cc1 31305,c1(C(=O)NCC2CC2NC(C2(F)CCOCC2)=O)cc(=O)c2ccncc2o1 31306,c1(OC)ncc(C(N2CCCC2C(CC(F)(F)F)=O)=O)c(C)c1Br 31307,CC1(C)CN(c2nc(=N)[nH]c(=NCC3(CC4CC4)CC3)[nH]2)c2ccccc21 31308,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1)=O)C1CC1 31309,c1(C(C)C)nnsc1C(=O)NCC1(C(N2CCCCC2)=O)CCCO1 31310,N1(CCC2CN(C(C(C)F)=O)C2)CCN(C(C2CC2c2ccco2)=O)CC1 31311,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(C3(F)CC3)=O)nc12 31312,c1(C(=O)NC2C(NC(c3ccnc(OC)n3)=O)CCCC2)ccc(C#N)n1C 31313,N1(C(C(c2ccccc2)N(C)C)=O)CCCC(CO)(NC(C2CC(CF)C2)=O)C1 31314,Cc1nc(C#N)c(NC2CCN(CC(=O)NC(=O)C(F)(F)F)C23CC3)o1 31315,C1(NCC2CCN(C(N(C)C)=O)C2)CCc2[nH]nc(C(F)(F)F)c2C1 31316,N#CC1CCCC1NC(=O)CCCCNC(=O)C(F)C1CCC1 31317,c1(C(=O)NCC2(NC(C(CC=C)C)=O)CC2)ccc(Cl)cc1-c1ccccc1 31318,Cc1ccc(CN(C(=O)C(=O)NC(C)CNC(C2CCC2)=O)C)c(Cl)c1 31319,C1(OC)CCC(C(=O)NCCC2(NC(=O)Cc3csc(SC(C)C)n3)CCC2)C1 31320,O=C1OC2CC(C(=O)NCC3CCCN3C(c3cnc4[nH]ncc4c3)=O)CC2O1 31321,Cc1cc(N(C)C)ccc1C(=O)NC1CCCN(C(=O)CCC2CCC(=O)C2)C1 31322,c12nc([nH]c(=N)n1)C(=O)N1CCC2C1.c1(CC)sc(=N)[nH]c1-c1ccccc1 31323,N1(C(C2N(C(C3CCCN3C=O)=O)CCC(=C)C2)=O)CCCC2(CCC2)C1 31324,c1(OC)cccc(C(=O)NC2CCCCC2NC(=O)CNC(c2cscn2)=O)c1 31325,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(SC)n1)NC(C)=O 31326,n1(CC)nc(C(=O)NC(C)CC(C)NC(=O)CC2CC(C)(C)CO2)ccc1=O 31327,N1(C(c2n(CC)ccn2)=O)CC2(C=C(C(=O)NCCN3CCCC3)CO2)C1 31328,C(=O)(C#CC(=O)N1CC(CNC(c2c[nH]nc2Cl)=O)C(O)C1)N(C)C 31329,c1(C(N(CC(=O)NC(C)CN=[N+]=[N-])C)=O)ccncc1F 31330,Cc1ccc(F)c(C(=O)NCCC(C)N(C(=O)C(c2cncnc2)C)C)c1Cl 31331,c1(C(=O)NCC(CNC(C(CC=C)CC)=O)O)cnc2c(Br)cnn2c1 31332,c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCC(C)C2)nccc2occc12 31333,n1(C2(C3(CNC(C)C=O)CC3)CC2)cc(C2CC2)nn1.c1(C2CC2)cccs1 31334,c1(OC)ccc(C)c(CN2CCOC2=O)c1.c12nnc(n1CC1CC1(F)F)s2 31335,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCCC2 31336,c1(C(C)=O)cc(C(=O)NC(CC2CN(C(C3CCCN3CC)=O)C2)C)ccc1C 31337,C=CC(C)(C)CCNC(=O)C(CN(C)C)NC(c1ccnc(CO)c1)=O 31338,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31339,n1(C2(NC(C34C(CN(C(=O)OC(C)(C)C)C3)C4)=O)CC2)nc(O)c2c1CCCC2 31340,c1(C(=O)NCC(CC)(C)NC(=O)C=CC2CCOCC2)cn(C)nc1C 31341,CCC(C)CC(=O)C(=O)N1CC(C(=O)NCCCCCC#N)C(F)(F)C1 31342,c1(NCC(C)(C)C2(O)CNC2)ncc(N2CCCCC2)cn1 31343,c1(OC)ccc(-n2nc(C3CC=CCC3)nc2C2CC(C)C2(C)C)cc1C 31344,c1(CC)c(C(N2CC(N(C)C(c3ccc(Cl)cn3)=O)C2)=O)cnn1C(CC)CC 31345,N1(C(C(CCC)CCC)=O)CCC2(NC(C34CC5CC3C4C5)=O)CCCCCC12 31346,c1(C(N(C(CCNC(C2(CC#C)CCCO2)=O)C)CC)=O)cccc2c[nH]nc12 31347,Cc1cccc(NC(C2COCCN2Cc2cc(Cl)ncc2C(=O)O)=O)c1Br 31348,CN1CCN(C(=O)CC(=O)NCC2(O)CC(NC(=O)CCF)C2)C(C(C)(C)C)C1 31349,C(N=c1[nH]c(=NCC2CCCC2)[nH]c2cc[nH]c12)c1cnn(CC)c1C 31350,CC1CN(C(C2C3(CC3)C23CC3)=O)CCC1NC(c1ccc(O)nc1)=O 31351,C(=O)(C(F)C(C)CNC(c1cc(O)nc(C)n1)=O)N1CCC(OC(C)=O)C1 31352,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31353,C(CCCCCNC(c1ccncn1)=O)NC(=O)CCc1csc(Br)c1 31354,c1(NC(C2CCC(n3cc(CN(CCOC)C)nn3)C2)=O)cc(Cl)c(F)cc1F 31355,C1(CC)(CNC(C2CCCC2CNC(C2CCCOCC2)=O)=O)CCC(=O)N1 31356,C(N=c1[nH]c2cc(F)ccc2o1)C1(CNC(c2cc(Br)n3ccccc23)=O)CC1 31357,Cc1cc2ccnc(C(N3CCC(O)(C(F)(F)F)C(F)C3)=O)c2s1 31358,C1(C(=O)OCC)(NCCc2cn(C)nc2C)CCS(=O)(=O)C1 31359,N1(C(CCc2cncc(C)c2)=O)CCC2CN(C(=O)C(C)NS(C)(=O)=O)CC2C1 31360,C(=O)(C(F)(CNC(C1CN(CC)CCO1)=O)C(C)C)NC(C#C)(CC)CC 31361,c1(C(N(CCCNC(C(CC=C)(C)C)=O)C)=O)ccc2c(c1)OC(F)(F)O2 31362,CC(CC(C)(C)O)NC(=O)NC1CC=CCC1C(F)(F)F 31363,Cc1nn(C)c(C(F)(F)F)c1C(=O)NNC(=O)CN1CCCC(C(C)O)C1 31364,N1(CCC)CC(NC(=O)C(c2cccnc2)NC(C2(C)CNC(=O)N2)=O)CC1=O 31365,C1(C(=O)NC(CCC)CO)Cc2nccnc2CN1C(c1ccc(F)cc1)=O 31366,CCC(C)C(O)C(C)C(=O)N1CCC(C)C(CNC(=O)Cc2c(C)noc2Cl)C1 31367,c1(C(=O)NC2CCN(C(COCCOC)=O)C23CC3)ccnc2[nH]c(C)nc12 31368,C123CCC(CC1)N2CC(=O)C(F)Cc1nccn13.CCC 31369,C(=O)(CC(F)(F)C(F)F)N(C)CC1(NC(c2csc(C)c2N)=O)CC1 31370,C(=O)(C(C(C)(C)C)N(C)C)NC1C(NC(c2cc(CC)[nH]n2)=O)CC1 31371,C(=O)(C(C)(F)C(=O)NCCCN(CCO)C(C1(C)CCC1)=O)OCC 31372,c1(C(=O)NC(CN(C(C#C)C)C)C)noc(C)c1-c1ccccc1 31373,C(=O)(CCCCN(C)C(c1cc(COC)on1)=O)NCC(C#C)CC 31374,C=CC1CN(C(=O)C(C)(CC)OC)CC1NC(c1ccccc1COC(=N)O)=O 31375,Cc1cccc(C(C)C)c1C(=O)NC(C)CCN(C(=O)CC1COCCO1)C 31376,N1(C(c2c(COC)cccc2)=O)CC(C)CCC1CNC(=O)CSC(F)F 31377,c1(C(=O)NCC2CN(C(C(C3CC3)OCC)=O)C2)ccn(C)c(=O)c1O 31378,c1(C(=O)NCCC(C)NC(C2(C(=O)OCC)CC2C)=O)noc2ncccc12 31379,c1(C(C(=O)NCCOC)N(C(C)COC)CC=C)ncn(C)n1 31380,c1(C(C(=O)NCCC)N2CCCC2)ccc(CS(C)(=O)=O)o1.C(COC)S 31381,C1(C(NCSC2CCN(C(C3CC(=C4CC4)C3)=O)C2C2CC2)=O)C=CCCN1 31382,c1(OC)cc(C(=O)NCC2CCCN2C(=O)C=C(C)C(F)F)c2ccccc2n1 31383,c1(CC)cc(C(=O)NCC2(F)CC(CNC(=O)CC3(O)CCOC3)C2)n(C)n1 31384,c1(COC)ccccc1-c1ccc(CN2CCC(CC(=O)N(C)C)CC2)cc1 31385,C1(NC(CC(CC)OC)=O)COC2CN(C(=O)Cc3ccc(F)c(F)c3)CC12 31386,C(=O)(CC1=CCN(C(c2cnc(OC3CC3)cn2)=O)CC1)NC1CC(OCC)C1 31387,C1(CC)CCC(NC(C2(F)CCN(C(=O)C(C)C(=O)OC)C2)=O)CC1 31388,CCCCC(C(=O)NC1(CCOC)CC=CC1)NC(=O)C(O)CC(C)C 31389,N1(C(c2c(C)cns2)=O)CC=CC(C(=O)NCC(C)OC(F)F)C1 31390,C1(CC=C)(NC(C2CSCCS2)=O)CC2CCC(C1)N2C(=O)C(C1CC1)OC 31391,C1(C(N(CC#C)CC)=O)CCN(C(c2occc2C)=O)C(CC)C1 31392,c1(OC(N(C)Cc2snnc2C2CC2)=O)ccc2c(c1)OCCCO2 31393,c1(OC)cccc(SCC(=O)NCCC(C)N(C(=O)C(C2CCCCC2)O)C)c1 31394,N1(C(C2CC(=O)NC(=O)C2)=O)CCOC2(CCC(NC(C3CC(=O)N3)=O)CC2)C1 31395,c1(C(=O)NCC2C(CNC(=O)CN3CCC3)C2)cc2ccc(Br)cn2n1 31396,c1(C(CC(=O)NCC(N2CC(CC(=O)N(C3CC3)C3CC3)C2)=O)C)ccccn1 31397,c1(C(N(C)CC2COCCN2C(C2CC(C#N)C2)=O)=O)cnc(S(C)(=O)=O)s1 31398,N1(C(C2C(C(C)C)C2)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 31399,Cc1cc(CC(=O)NC(C)CNC(C2(c3cccc(Cl)c3F)CC2)=O)ccc1O 31400,C1(CNC(COC(CC)C)=O)C(C(=O)NCC(C)(O)CO)C1(C)C 31401,C=CCCN=C(NCC1CCCC1)NC1CCCC(OCCO)C1.C(C)C 31402,c1(COC)ccc(C(=O)NC(C)(CNC(C2CCCOC2)=O)C2CC2)[nH]1 31403,N1(C(c2c(F)cn(C)n2)=O)Cc2ccccc2CC1C(=O)Nc1cccc(CO)c1 31404,c1(C(=O)NC2C(NC(c3cscc3F)=O)C2)ccc(-c2ccco2)[nH]1 31405,c1(CC)cc(N)c(C(N2CC(CNC(c3cc[n+]([O-])cc3)=O)C(C)C2)=O)cc1F 31406,N1(C(C#C)C)CCN(C(c2nc(CNC(=O)Cc3cc[nH]n3)oc2C)=O)CC1 31407,c1(N(C(=O)NC(C=C(C)C)C)CC2CC2)ccccc1Br 31408,CC(CC(C)(C)C)C(=O)N1CCCOC(CNC(C2CC(F)(F)C2)=O)C1 31409,CC1(C)CC(CNC(c2ccccc2C2CCC2)=O)CN1C(c1ccc(Cl)o1)=O 31410,C1(C(N(CC(C)C)CC(=O)NC2CC(F)(COC)C2)=O)CCN(C)C1C 31411,c1(OC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)CC(C)NC(=O)C1CC1 31412,C(=O)(C(F)C(C)C(F)(F)F)NCCN(C(c1c(C)nc(CC(C)C)s1)=O)C 31413,N1(C(CC2CCCN(C)C2)=O)CCN(C(=O)C(F)=CC2CC2)C(CC(F)(F)F)C1 31414,C1(NC(c2cnc(C)o2)=O)CCC(CNC(=O)CC2COCCO2)CC1 31415,c1(C(=O)NC(C2CN(C(=O)COCP(C)(C)=O)C2)C)ccc(C(F)(F)F)o1 31416,N1(C(c2ccc(F)cc2)C(=O)NC2CC2)Cc2cc(Cl)c(Cl)cc2C1 31417,c1(C(N2CC(CN(C(CCC(=C)C)=O)C)C3(C2)CC3)=O)nc2ccccn2c1F 31418,CC(C)CC(C(=O)NCC1(O)CC(O)C1)N(C)C(C1(CO)CCOC1)=O 31419,N1(C(=O)C=Cc2cnccn2)CCn2nc(CNC(=O)Cn3ccnn3)cc2C1 31420,C1(CCO)(NC(c2ccc(-c3ccc(Cl)cc3)o2)=O)CCCCC1 31421,N1(C(CC)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2(C)C)=O)C1 31422,c1(CN)cccnc1.Cc1occc1COC(F)F 31423,C(CCC(C(=O)NCCC1CC1C)NC(=O)CC(F)(F)F)OC 31424,C1(C(=O)O)(C)CC=CCC1.c1(COC(C)(C)C)ncc(CN2CCCC2)s1 31425,C1(C(C)C)C2CCC(C2)C1C(=O)NCCCNS(C)(=O)=O 31426,Cc1c(C(=O)NC(CNC(=O)Cc2cnco2)C2CCC2)cc(O)cc1N 31427,CC(C)CC(F)C(=O)NCCC12CCC1CN(C(=O)CN1CCS(=O)(=O)CC1)C2 31428,N1(C(C(CCOC)C)=O)CCC2(CC1)CN(C(=O)CC13CCC(CC1)OC3)C2 31429,c1(CNC(c2c(C)ccc(F)c2)C)cc(=O)oc2cc(N)ccc12 31430,c1(CNC(=O)NCC2(CO)CC3CC3C2)ccc(-c2cccc(O)n2)cc1 31431,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31432,C1(NC(=O)CC2CCOC2)CC12CC(NC(C1(c3cccnc3)CCCC1)=O)C2 31433,CC1(F)CCCN(C(C2CCOCCN2C(=O)Cc2ccc3c(c2)CC3)=O)C1 31434,C(=O)(C(C#N)C(C)(C)C)NCCN1CCN(C(C2(COCC)CCCC2)=O)CC1 31435,C1(C(=O)NCC2C(C)CC2)CCOCC1NC(=O)C(C)(F)c1ccon1 31436,Cn1cnc2ccsc2c1=NCC1CCCN1C(c1cc(Cl)c[nH]1)=O 31437,Cc1[nH]nc(C(=O)NC2CCCC2CNC(=O)C(=Cc2cscn2)F)c1C 31438,Cc1nc(C(N2CC(O)(C(C(=O)NC3(C)CCCC3O)F)C2)=O)c(C)o1 31439,N1(C(c2c(OC)csc2)=O)CCN(C(=O)CC2CCC3CC23)CC1 31440,c1(CC(=O)OCC2CC(O)C2)cccc(NC(c2cnco2)=O)c1 31441,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)N(CCNC(=O)CC(C)C(=O)OC)CC 31442,c1(CC)[nH]c(C(N2CCC3(NC(=O)CS(C)(=O)=O)CC3C2)=O)c(C)c1C(=O)OC 31443,N1(C(CCCc2cc(C)no2)=O)CCC2(CCCN(C(C3CCC(=O)N3)=O)C2)C1 31444,c1(C(=O)NCC(CNC(c2ccc(NCC)cc2)=O)C)c2ccccc2nn1C 31445,C=C(CNC(=O)C(F)C(C)CNC(=O)CCn1cnnn1)C1CCOCC1 31446,c1(C(N2CC(NC(CC3N(C)CCC3)=O)C2)=O)ccc2c(O)nc(S)nc2c1 31447,C1(NC(C(C)SC(C)C)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31448,c1(C(N2CC(C(C)NC(c3cn[nH]c3)=O)OCC2)=O)ccnc(F)c1N(C)C 31449,N1(C(C2CCCN(S(CC)(=O)=O)C2)=O)CCC(NC(=O)CC(C)(F)F)CC1C 31450,c1(OC)cc(C(N2CCCC2C(C)NC(C2CC(OC)C2)=O)=O)ccn1 31451,N1(CC#C)CCN(C(C2CCN(C(C3CC(=O)N(CC)C3)=O)C2C)=O)CC1=O 31452,CN1CC2CC1CN2C(=O)CCC(=O)Nc1ccc(COc2cccs2)cc1 31453,C(=O)(CC1=NNC(=O)C1)NC1C(C)CN(C(=O)CNS(N)(=O)=O)C1 31454,N1(C(CSCC#C)=O)CCC(NC(c2nn(C)c(Cl)c2C(F)(F)F)=O)C(F)C1 31455,C1(CNC(C2(C)CCC2)=O)CCC2CN(C(C3CC3c3cccs3)=O)CC12 31456,c1(C(=O)NCCc2c(CNC(C(C(C=C)C)C)=O)nco2)cn2cc(C)sc2n1 31457,Cc1cnc(F)cc1C(N1CCN(CCS(C)=O)CC1)=O 31458,C1(C(=O)NCCNS(CCCC)(=O)=O)CCC2(CC2)N1C(=O)C(C)CSC 31459,c1(CNC(CONC(c2cnn(C)n2)=O)=O)ccccc1O 31460,C(=O)(C(C(C)C)N(C1CCCCO1)C(=O)COC)N(CCC#C)CCO 31461,C(CN(C1COC(=O)C1)C)(C(=O)Nc1ccccc1)NC(C(C)=CCC)=O 31462,C1(C(N(CC(CN(C(C(CC)C)=O)C)O)C)=O)CCC2CCCCC2C1 31463,Cc1ccc(F)c(C(=O)N(CCCCN(C)C(C2(C)C=CCCC2)=O)C)c1Cl 31464,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NCC(C)(C)COC)C(F)(F)C1 31465,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31466,C(=O)(C1CCCc2nncn21)N(C1CCN(C(C2(C)CC(=O)C2)=O)C1)CC 31467,c1(C2C(NC(=O)NCC3(CN4CCCCC4=O)CC3)C2)ccc(Br)cc1 31468,C12CCCCCN1C2=O.N1(CC=C)CCN(C(c2ccc(OC)o2)=O)CC1 31469,C(=O)(CC1=CCCCC1)NC1C(C)CN(C(c2ccc(N(C)C)c(Cl)n2)=O)C1 31470,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(Cc3ccns3)C2)CC1 31471,C=CC1(C(=O)NCC(Cl)Cl)CCN(C(c2ccc(C)cc2C)=O)C1 31472,C12(C(N3CCC(C(C)NC(=O)CN4C(=O)CCC4=O)C3)=O)CCC(C)(C1)OC2 31473,C1(O)(CC(N2CCC(CN(C(=O)CN3CCC(CO)CC3)C)C2)=O)CCCCCC1 31474,C1(NC(C2NC(=O)OC2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 31475,O=C(CC(O)CNC(c1csnn1)=O)NCC1CCN(C2CC2)C1 31476,C(=O)(C(C)(O)C(F)(F)F)NCCCn1ccnc1.CC12CCN(CC1)C2=O 31477,C(C)(CCC(=O)NCC(=O)N(C)Cc1ncc[nH]1)NC(C(C)C)=O 31478,N1(C(c2cc(C)sc2C)=O)CCCC(O)(CNC(=O)Cc2ccsc2Cl)C1 31479,Cc1ccc(F)c(C(C(=O)NC2COC2)N(C)Cc2cccs2)c1 31480,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CCCC2(CCN(C(=O)CN3CCCCC3)C2)C1 31481,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCC(NC(=O)COCC2CC2)CC1 31482,C1(C(=O)NCC2(c3ccc(OC)cc3)CC2)CCCC2(CC1)OCCO2 31483,c1(N2CCCC(CC=C)(NC(c3ccc(=O)oc3)=O)C2)c2ccccc2nn1C 31484,CC1(CNCc2nccc3sccc23)CCCCC1(F)F 31485,C1(CC#C)(C(=O)NC2CC2CNC(=O)C#CC2CC2)CCCCC1 31486,c1(C(N2CCN(C(CCSCCCC)=O)CC(C)C2)=O)cnc([N+](=O)[O-])cc1C 31487,N1(C(c2c(Cl)nn(C)c2Cl)=O)CC(C2CN(C(=O)CCC#N)C2)C1 31488,C1(NC(c2cc(C)nn2C)=O)CCSC12CN(C(c1ccc(N)cc1O)=O)C2 31489,C1(n2cc(CC)nn2)CN(C(c2nn(C)nc2Br)C(=O)NC)CC1(C)C 31490,C1(N(CC)Cc2csc(SC)n2)CCN(C(C23COCC2C3)=O)CC1 31491,N(C(=NCCC1CCOC1)NCc1ccc(Br)o1)Cc1n(CCC)ccc1 31492,c1(C(N(CC(CNC(CC(CC)C2CCC2)=O)(C)C)C)=O)cnc2ncccn12 31493,C1(C(=O)NCC(C)NC(C2(c3cccnc3)CC2)=O)CCc2nnc(O)cc2C1 31494,c1(C(=O)NCC(CNC(c2c(CC)nc(C)[nH]2)=O)O)cccc(O)c1Cl 31495,C1(C(N2CC3C(NC(c4ccncc4Cl)=O)C(C3)C2)=O)COc2ccccc2O1 31496,N1(C(C(CC)SC)=O)CCN(C(c2ccc(C3CC3)nc2O)=O)CC1COC 31497,N1(C(CC#C)C)CCN(C(=O)NCCn2ncc(C(=O)OC)c2C)CC1 31498,CCC(CN(C)C)CC(=O)NCC1C(C(=O)NCCCC2(O)CC2)C1(C)C 31499,C1(C(=O)NC2CCC(CNC(C3(C)CCCO3)=O)CC2)(NC(C)=O)CCCCC1 31500,N1(C(C(CC)C#N)=O)CC(C(=O)NC(C2(O)CCC2)C)CC(C)C1 31501,c1(C(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc2c(F)c(Cl)ccc2[nH]1 31502,C1(C(=O)NCC(CC)C)CC(F)CN(C(c2ccc(C(F)(F)F)cc2)=O)C1 31503,C1(SCC)CCN(C(=O)C(C)[SH](c2ccc(N)cc2)OC(C)=O)C1(C)C 31504,c1(C(=O)NCC2CCC(F)(F)CC2)ccc2c(c1)NS(=O)(=O)C2 31505,c1(C(=O)NC2CCCC(NC(CCC(=C)C)=O)C2)cnc(O)c(OC)c1 31506,c1(CC(N2C(CNC(Cn3ccc(C)n3)=O)COCC2)=O)ccc2nc[nH]c2c1 31507,N1(CC)CC(CNC(C2SCCC2C)=O)CCC1.c12cc(no1)C(=O)N1CC2C1 31508,CCCC(O)C(=O)N(C)CC1CCN(C(=O)CN(c2ccnc(Cl)n2)C)CC1 31509,c1(NC(c2cnn(CC(C)C)c2C2CC2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 31510,c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CC=C2)nn(C)c(Cl)c1Cl 31511,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31512,C1(CCC(=O)N(CC(C)NC(C2CSC2)=O)C)CC(C)(C)CO1 31513,C(C)(C(=O)N1CCCC(N(CCF)C(c2ccoc2)=O)C1)(C(C)C)OC 31514,C1(C(=O)NC2(CN(C(=O)CC3C=NN(C)C3=O)C)CC2)CC1C1CCCCC1 31515,Cc1onc(C2CC2)c1C(=O)NC1CCC(NC(=O)CC2CC(C)OC2C)C1 31516,Cn1nc(CNC(=O)C(C)(C)NC(C2CCCCN2C)=O)n(C)c1=O 31517,N1(C(C(C)C2(O)CCC2)=O)CC=CC1CNC(=O)NC1(c2ccccc2)CC1 31518,Cn1cc(C(O)C(=O)NC2COCC2NC(c2cscc2Br)=O)cn1 31519,CC1CN(C(c2cc[nH]c2)=O)CC2(CCN(C(C3CCCCC3)=O)C2)O1 31520,C(=O)(C(F)C(F)(F)F)NCC1(F)CC(NC(=O)CCc2nnc(S)nc2O)C1 31521,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31522,C(CC1=CCCCCC1)NC(C(C)NC(C(C)NC(=O)C1CC1)=O)=O 31523,C1CCCC(=O)N1.C(C)(CCC(C)C)N(C(C(COC(C)=O)C)=O)C 31524,c1(OC)c(C(=O)NC2CCN(C(c3cc(C4CCC4)[nH]c3C)=O)C2)ncnc1C 31525,c1(C(=O)NCCC2CCC(NC(C3(CC=C)CC3)=O)C2)[nH]nc2ncnc(O)c12 31526,C12(CNC(C(C)S(N)(=O)=O)=O)CCCC1N(C(c1ccnnc1O)=O)CCC2 31527,N1(C(c2cc(Cl)ncc2F)=O)CCCC(C2CN(Cc3cc(Br)ccc3F)C2)C1 31528,Cc1ccc(C2CC2C(=O)NC2(C)CC(NC(=O)C3=NOCC3)C2)cc1 31529,c1(C(=O)NC2CCN(C(C(n3c(C)cc(C)n3)C)=O)C2)c(C)c(Cl)cc(C)c1N 31530,C1(NC(N)=O)CCC(C(N2CCOC(C(=O)CCc3nc[nH]n3)C2)=O)CC1 31531,C(C(=O)N(C)CC1CCCN1C(c1nnn(C)n1)=O)(C(C)C)SC 31532,c1(C(=O)NC(CC=C)CNC(c2c(C)ncn2C)=O)cc(Cl)ccc1OC 31533,C(=O)(CC(C)N(C)C(C1CC(O)C1)=O)NC(CN(CCCC)C)C 31534,C1(C(=O)NC2(CO)CN(C(CN(CCCCCC)C)=O)C2)CC=CCC1C 31535,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3c[nH]cc3Br)=O)CC1C2 31536,CC1CCC(OCC(=O)NC(C)(CNC(C2CCCO2)=O)CO)CC1 31537,Cc1cccn2cc(C(=O)NC(C)CC3CN(C(=O)CC(C)CN(C)C)C3)cc12 31538,C12(C(N3CC(CNC(c4ccc(C)cc4F)=O)C(C)C3)=O)CCOC1CCOC2 31539,C1(CNC(c2cnc(OC)nc2)=O)CC2(CC2)CN1C(=O)CC1CC(F)C1 31540,N1(C(C(C=CC)O)=O)CCN(CC(=O)NCCC2(C)N=N2)CC1 31541,C1CN=C(NCC2(O)CCCOC2)NCC1.Cc1nc(C)c(CC(C)C)s1 31542,N1(C(c2csc(C)n2)C(=O)NC(C(=O)OC)C)CCN(c2ccccc2O)CC1 31543,c1(C(=O)NCC=CCNC(c2c(Cl)cc(C)nc2)=O)c(C)nc(C2CC2)nc1O 31544,c1(CC)[nH]c(=N)sc1C(=O)N(C1CCCN(C(=O)CC2CCC23CCC3)C1)C 31545,CC1CN(C(=O)CC23CCC(CC2)C3)CC(C)N(C(=O)CS(=O)(=O)CCO)C1 31546,C1(CC)CN(C(C2CN(C(=O)Cc3cnoc3)CC2CC)=O)CC12CCC2 31547,C1(CC=C)(C(N2CCC(CC)CC2)=O)CCCN1C(=O)Cn1nc(C)oc1=O 31548,c1(CC)cc(Br)cc(C(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2F)c1N 31549,Cc1c(C(N2CCC(C)(C(=O)NCC3CCCO3)C2)C(=O)N(C)C)cccc1Cl 31550,CC12CCOC(C(N)=O)(C1)C2.C12CC(CO1)C(=O)NCCN(C)CC(=O)NC2 31551,C1(COCC)CN(C(=O)Nc2ccnn2C(CC)CC)CC1O 31552,c12cn(C)nc1C(=O)NC2.C1(COC)CCC1CC(=O)NCCC(N)=O 31553,c1(C(C(C(N)=O)C2CCCC2)C)ccc2nc(O)[nH]c2c1 31554,c1(C(=O)NCCN(C(Cc2c(C#C)cccc2)=O)C)cc2cccnc2o1 31555,c1(SC)cccc(NC(c2ncc(C)o2)C(=O)NC2CC2C(=O)OC(C)(C)C)c1 31556,C(=O)(CC(O)CC(C)(C)C)N(CCN(C(Cc1ccc(C)c(Cl)c1)=O)C)C 31557,c1(C(c2ccccc2)N(CCCNC(C2CCC2F)=O)C)c(Cl)cncc1Cl 31558,c1(C(=O)NCCOCCNC(CCCC(CC)C)=O)c(F)ccc2n[nH]cc12 31559,C1(C(=O)NCCCCCNC(=O)CC2COC3CC2C3)CCCCC(F)(F)C1 31560,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C1 31561,C1(NC(C(C2CCCC2)NC(C)=O)=O)CCN(C(c2ccc(C(F)F)s2)=O)C1 31562,c1(CC(N2CC(CC=C)(NC(=O)CC3CCC(O)C3)C2)=O)sc(C)cc1C 31563,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(c2nc(Cl)cs2)=O)C1 31564,C12(C(=O)NCC3N(C(C4(S(N)(=O)=O)CCCC4)=O)CC3)CCOC1CC(=O)NC2 31565,N1(C(COC2CCN(C(CC3CCCN(C)C3)=O)C2)=O)CC2CC2C2CC12 31566,C1(C(=O)OC)CN(C)CC1NC(=O)NCc1cccc(-c2nc[nH]n2)c1 31567,C1(C(N2C(C)COCC2)=O)CN(C(c2ccc3c[nH]nc3c2)=O)CC12CCCC2 31568,C(CCC(C)(F)F)NC(c1n(CCCSCC)nnn1)c1cn(C2CCC2)nn1 31569,C#CCCCC(C)C(=O)N(CCNC(=O)CCCCC1CC1)CC1CC1 31570,c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)c(NC(C)=O)c[nH]c1C 31571,c1(C(=O)NC(C)C(C)(C)NC(=O)Cc2cn3ccsc3n2)cc(O)cc(=O)o1 31572,CC1CN(N2CCSC(CC(F)(F)F)C(C)C2)CCO1 31573,N1(C(C(C(C)OC)N(C)C)=O)CCC(C)C(CC(N2CC(F)(F)CC2CO)=O)C1 31574,CCC(CNC(c1cnc2cc(Cl)ccn12)=O)N=c1[nH]nc(CO)s1 31575,CCCC(CC)CC(=O)N1CC(CNC(c2cc(Cl)ccc2C)=O)C2(CC2)C1 31576,C1(CC)CN(C(C2(NC(=O)CCC3CCOC3)CCCCC2)=O)CCCO1 31577,C(CN(C)C(C1(O)CCC1)=O)(CO)(CO)NC(C1C(C(C)C)CCO1)=O 31578,CCC(CC)C(C)C(=O)N1CC(NC(c2cc(F)ccc2OC)=O)CC(F)(F)C1 31579,C1(NC(C(C(=O)OC)OC)=O)CCN(C(C2CCOC2)=O)CC1F 31580,C(CNC(C1CC1)=O)(C(=O)NCC(C)N(C(=O)CCCC1CCC1)C)NC(C)=O 31581,C#Cc1ccc(C(=O)NCC2C3CC2N(C(c2sccc2C2CC2)=O)C3)c(C)c1 31582,CCC(CN(C(=O)Cc1cncs1)C)NC(=O)CSC 31583,Cc1ccc(C(=O)NC2C(Cl)(Cl)C23CC3)cc1Br 31584,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31585,C(C(C)(F)C(F)(F)F)SCCOC(c1c(C(=O)OC(C)(C)C)cccc1)=O 31586,C12(C(N3CCC(F)(OC)C3)=O)CCC(CN(C(=O)Nc3cc(C)ccc3F)C1)C2 31587,C1(CC(=O)NCC(=O)NCC)N(C(c2cc(C)[nH]c2C)=O)CCC1(C)C 31588,Cc1cnc(F)cc1C(=O)NC1CC(NC(=O)CC(C)O)C(O)C1 31589,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31590,C(=O)(CC1CCOc2ccccc21)N1CC(O)(CCNC(CC(COC)C)=O)C1 31591,c1(C(N(C(CNC(Cc2c(C)ccc(F)c2)=O)C)C)=O)cccc(S(C)=O)c1 31592,CCC(C(=O)OC)C(=O)NCC1(NC(c2c(COC)cnn2C)=O)CCOC1 31593,Cc1ncc(N)cc1C(N1CC(C2(NC(=O)Cc3cc(Cl)n(C)n3)CC2)C1)=O 31594,C1(C(N2CCC(C(C)(C)O)C2)=O)N(C(=O)CCCc2cnn[nH]2)CCC1(C)C 31595,CCC(CC)CC(=O)Nc1nc(CC(=O)Nc2c[nH]nc2C#N)cs1 31596,Cc1n[nH]c2nc(O)c(C(=O)NC(C)Cn3ccnn3)cc12 31597,C1(C(C)(C)C)CCCN(c2nnc(-c3nn[nH]n3)n2C2CC2)C1 31598,c1(OC)cccc(C(N2CC=CC(NC(C3CC=CCC3C)=O)C2)=O)c1C 31599,N1(NC(C2(SC)CN(C(c3c(CC)nco3)=O)C2)=O)CCC(O)CC12CC2 31600,CCC(O)CC(=O)N1CCCCC1Cn1cc(C2C3CCCCC23)nn1 31601,N1(C(C(C)NC(=O)OC)=O)CCN(C(=O)Cc2cccnc2C)CC(C)(C)C1 31602,c1(CC(=O)NC23CCC(C2)N(C(=O)C(F)n2ccnc2)C3)cc(F)cc(F)c1 31603,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(F)(F)CC1CNC(C1CC(C)C1)=O 31604,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31605,CCC(CC)C(=O)N1CC(CNC(=O)CC2CCNC(=O)C2)(OCC)C1 31606,N1(C(c2ccc(CC)o2)=O)CCC(C)(C)C(CNC(C2CCCSC2)=O)C1 31607,c1(CC)nc(C)c(CNC(=O)C(CCF)NC(c2c(C)cnn2C)=O)o1 31608,c1(CC)ccc(CNC(C2CN(C(=O)C3=C(Cl)CCC3)CCN2C)=O)cc1C 31609,N1(C(CCOC)=O)CCC(C)N(C(C2CCC(=O)N2C(C)C)=O)CC1 31610,C(=O)(C(F)C(C)(F)F)NCCCCCCN(C(CCC(=O)N(C)SCCCN)=O)C 31611,N1(C(c2[nH]cc(C)c2)=O)CC(CNC(C2CC3C=CC2C3)=O)C(C)C1 31612,C1(CNC(Cn2cc(C)nc2)=O)CC2CN(C(=O)CN3CC(=O)NC3=O)CC12 31613,C1(N(C(C)C)CCNC(=O)CCCNC(N)=O)CCCC(C)C1 31614,C1(C(=O)NCC2CCC=CCC2)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 31615,c1(OCC)cc(C(=O)N(CC(O)CN(C(=O)CCc2cc[nH]n2)C)C)on1 31616,N1(C(CCSCCCC)=O)CC(C)CN(C(c2cc(O)ccc2N)=O)C(C)C1 31617,C1(NC(CCN(C)CC)=O)CCN(C(c2cnc(C(F)F)nc2)=O)C1C(C)C 31618,c1(C(=O)NCC2CCN(C(C3CC(OC)C3)=O)CC2C)csc(=NC2CC2)[nH]1 31619,C1(c2onc(N(c3cc(C=O)[nH]n3)C)n2)CCN(C(=O)NC)CC1.CC 31620,N1(C(C=CCC)=O)CCC(C2CC2)(CNC(c2ccc(Cl)s2)=O)C1 31621,Cc1ccn(C)c1C(=O)NC1CC(NC(C2(C(C)(F)F)CCOCC2)=O)C1 31622,Cc1cccnc1C(=O)NCCCN(CCCNC(C1COCCN1C)=O)C 31623,N1(C(C(=O)Nc2ccc(C(=O)OC)cc2)C2COC2)CCC2(CCC(O)C2)C1 31624,C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(c2n(C(C)C)ncc2F)=O)CC1 31625,c1(C(=O)NCC2(NC(C3CCCC(=O)C3)=O)CCCC2)cc(C(F)F)cc(F)c1 31626,C1(NC(C2CC(CC)CCC2)=O)CC2(C1)CC2N=c1[nH]c2cccc(C)c2s1 31627,C1(CC)CN(CC)CCN1C(C1(NC(=O)C(O)C(F)(F)F)CC1(C)C)=O 31628,CCCCC(C(=O)N(C1CCSCC1)C)NC(=O)C=CCCC(C)C 31629,C1(C(N2CC(Cn3cc(CCn4ccnc4)nn3)C2)=O)CC2CC1C1C2C1(F)F 31630,CC1CC(NC(=O)CC2CCCO2)CN1C(c1cc(N)ccn1)=O 31631,c1(C(N(C2CCN(C(Cc3nc(C)sc3C)=O)C2)C)=O)cc(Cl)ccc1N 31632,C1(C(N2CC(C(N)=O)(CNC(COC(C)C)=O)C2)=O)CCCC1S(C)(=O)=O 31633,C1(C(=O)NCC(C(=O)NC)CC2CC2)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31634,N1(C(C2(N(CC)CC)CC2)=O)CC2CC(SCC)C(C2)C1.C(CSC)(CC(C)C)NC=O 31635,CCC(C#N)CN1C(=O)COCC1.C1(NC(=O)COCC)CCOC1 31636,N1(C(CCC=C(C)C)=O)CC(F)(F)CC1C(=O)NCC(c1ccc(C)o1)O 31637,c1(C(N2CCC(C)(CNC(C(CCSC)O)=O)C2)=O)sc2nnc(S)n2c1C 31638,c1(C(C2(C(F)F)CC2)NC(=O)Nc2ccc(CCO)cn2)ccc(Br)cn1 31639,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31640,C(CCCC(C)C)(C(=O)O)Sc1n(-c2c(CCCC)cccc2)nnn1 31641,n1(CC)cc(C(N2CCN(C(=O)C(F)CC)C(C)C2)=O)c(=O)c2cc(Cl)ccc12 31642,c1(C(=O)NCCN(C(c2n[nH]cc2C2CC2)=O)CC)nccc2ccn(C)c12 31643,c1ccc(C)c(C)c1.C1(N2CC2)CCC(O)CN1C.C(=O)(COCC)NCCC 31644,CC(C)CC(F)(F)C(=O)NC1C2CC(NC(=O)C(N3C(=O)CCC3=O)C)CC12 31645,C(CCCCC(=O)NCCCCCNC(c1cn2ccsc2n1)=O)N(C)C 31646,C1(N(C(c2c(SC)cccc2)=O)C)CCN(C(c2c[nH]c(C#N)c2)=O)CC1C 31647,c1(CCCC(=O)NC2CC(NC(C3CCCCC3O)=O)C2)ccc(O)cc1 31648,CC1CCN(C(c2ccnc(-n3cncn3)c2)=O)C1CNC(=O)C=C(Cl)Cl 31649,C(CC(C(=O)NCCC1CC(C(=O)NCc2nccnc2C)C1)OC)OC 31650,C(CC(=O)NCCCCNC(=O)CC1CCCC1)(C1CC1)NC(=O)OCC 31651,Cc1ccncc1C1(NC(C2CN(C(=O)CCC3CCCC3C)C2)=O)CC1 31652,c1(C(=O)NC2CCC(CNC(C3CC4(CC4)C3)=O)CC2)ccc2c(c1O)CCC2 31653,C1(NC(C2CCC(NC(C)=O)CC2)=O)CN(C(C2CC3CCC2C3)=O)CC2CC12 31654,N1(C(C(C)C2CCC2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C 31655,c1(CC(=O)NCCC2(NC(CCOCCCOC)=O)CCC2)cnc(C)s1 31656,c1(OC)ncc(-c2cn(CCNC(C3CCC3C(F)F)=O)nn2)c(C2CC2)n1 31657,c1(CCC(=O)NC(C2CCCN2C(=O)CN2CCCC2)C)cccnc1Cl 31658,O=S(=O)(c1nc(N2CC3CCCC2C3)ccc1Br)N1CCC(OCCO)C(OC)C1 31659,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31660,c1(C(=O)NC(CC)CNC(c2ncsc2C)=O)cccc2c1oc(=O)n2C 31661,C1(NC(C=CC(=O)OCC)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31662,C(=O)(C1OC(=O)c2ccccc21)N(CCOCCN(C(C#CC(=O)OC)=O)C)C 31663,C1(CCC(N2CC(CC(C)NC(C(C3CCOCC3)C)=O)C2)=O)CCCCCC1 31664,CC(C)CC(C(=O)NOC(c1ncccn1)C)NC1CC1 31665,CC(C)C(O)C(=O)N.C1(c2ccc(F)cc2)(N2CCOCC2)CCN(C(=O)C(F)F)C1 31666,C1(CCCCCNC(C(C)=CC)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 31667,CS(=O)(=O)c1ccc(C(=O)NC2CC23CCN(C(=O)CC2CCCS2(=O)=O)CC3)o1 31668,c1(C(=O)NC2CCCN(C(C3C(C)C3(F)F)=O)C2)n[nH]c2cccnc12 31669,c1(C(=O)NC(CC)CNC(=O)CSc2nnnn2C)cccc(N2CCCC2)n1 31670,CCC(CCCC(=O)NCc1ccnc(NC(C2CCN2CC)=O)c1)OC 31671,CC1CNC(=O)CN1C(C1CC12CCN(C(c1ccn(C3CC3)n1)=O)C2)=O 31672,N1(C(CC(COC)(C)O)=O)CC2CC(O)C1C2NC(=O)CCc1cnc[nH]1 31673,N1(C(C2CC(=C)C2)=O)CCC(C2(NC(=O)Cc3cnccn3)CC2)CC1 31674,Cc1nsc(C(N2CCOC(Cc3cn(CCC4CCN(C)C4)nn3)C2)=O)c1N 31675,c1(C(N2CCN(C(COCC(C)C)=O)CC2)=O)cccc2c1OCCC2CCO 31676,N1(C(Cc2cn(CC)nc2)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])cn1 31677,C=C(Cl)C(C)(C)C(=O)NCC1(NC(=O)C(C)OCC(C)C)CCCCCC1 31678,C1(NC(CSC)=O)CCN(C(c2c(Cl)nn(C)c2C)=O)CC(C)(C)C1 31679,N1(C(c2nn(C)c(Cl)c2)=O)CC2(CC2)CC1CC(N1CCC(c2cnn[nH]2)C1)=O 31680,c1(C(N(CCC#N)CC2CCCC2)=O)cccc(Cl)c1F 31681,c1(COC(CC(COC)C)=O)cc2cccnn2c1 31682,N1(C(C(C(CC)C)N)=O)CCCC12CCCN(C(C1CC=C(C)CC1)=O)CC2 31683,C1(CC(N)=O)(NC(=O)CCN2CCC(F)(F)C2)CCCN(C(=O)CC2CCC2)C1 31684,C12(CNC(=O)COCC(F)(F)F)CCCC1CN(C(C13CCCC(CO1)C3)=O)C2 31685,C1(CO)CC(NC(c2ccc(C(OC)OC)o2)=O)CN(C(C23CCC2C3)=O)C1 31686,CCC(C)(CC)C(=O)N1CCCC1(CO)CNC(=O)C(COC)COC 31687,N12CC(OC(C(F)(F)F)C1)C(=O)N1CCC(CC1)C(C)C2=O.C(=O)(OCC)OC 31688,C(C(F)(C(=O)NCCCCN=[N+]=[N-])C(C)C)NC(C(=Cc1ccccc1)C)=O 31689,C(=O)(C(O)CCCNC(=O)C(C)N=[N+]=[N-])N1CCC(C(CC)C)CC1 31690,C(=O)(CCCC(F)(F)F)N1C(C)(CNC(N2CC(CN(C)C)C2)=O)CCC1 31691,N1(C(C2C(C)(C)C(NC(=O)CCCC3CCC3)C2)=O)CCC2(CC1)CC2C#N 31692,N1(C(C(CC)c2ccccc2)=O)CCC(C)(C)C(CNC(=O)Cc2cn[nH]c2)C1 31693,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31694,C1(NC(C(=Cc2cccnc2)C)=O)CC(O)CN(C(c2coc(Br)c2)=O)C1 31695,CCC(C)C(C)C(=O)NCC1(C(C)(C)C)CCN(C(=O)COC(F)F)C1 31696,c1(CC)cc(NC(C2(F)CCN(C(c3cccc(C#N)c3)=O)CC2)=O)ccc1F 31697,C(C1CN(C(=O)C(C)CC2CCC2)CC1C(=O)NCc1cncn1C)=CC 31698,c1(N)nc(N2CC3CCC3(CO)C2)c2c(n1)CSC2.CC1CCS(=O)(=O)C1 31699,C(=O)(C(C)(C)CCC#N)NCc1cccc(CN(C(C2(OCC)CC2)=O)CC2CC2)c1 31700,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31701,Cc1ccc(O)c(CC(N2CC(O)CC2CNC(=O)COCC2CCC2)=O)c1 31702,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31703,CC(C)(C)C(O)CNC(=O)CCCOC1CN(C(=O)CC2(O)CCC2)C1 31704,S(=O)(=O)(c1ccc(Br)cc1NCC(CC1CC1)OC)NC(C=C)COC 31705,C(=O)(C=C1SCC(=O)N1C)N1CC(CC(C)NC(CCc2c(C)ncs2)=O)C1 31706,Cc1nc2cc(C(=O)NCC3CN(C(C4CCOC4)=O)CC3C)cc(Br)c2o1 31707,Cc1noc(C(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)C2)c1I 31708,Cc1cc(C(N2CCN(C3COCC3NC(=O)CC3(C)CC3)CC2)=O)oc1C 31709,N1(C(C(CCCC)O)=O)CC2(CCN(C(C3CN4CCN3C(C)C4)=O)CC2)C1 31710,CCC(C)(C(=O)NCC1CN(C(=O)CCc2cc(Cl)no2)CCC1(F)F)C(F)F 31711,C(=O)(C(C)(CNC(=O)CC(CC)C1CCC1)CC)NC(CCCC)C 31712,C(CC(C(=O)NC(CO)CCCN(C)C)NC(c1sccc1F)=O)N(C)C 31713,C1(C(=O)NC2(CC)CCN(C(=O)C(F)Cc3ccccc3)C2)CCC(C)(O)CC1 31714,C1(NC(=O)CSCC2CCCO2)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1O 31715,N1(C(CCCCC#C)=O)CCN(C(=O)C=Cc2ccc(OC)cc2)C(C)C1C 31716,CCC(C)(C#N)C(=O)N1CC(C(=O)NOC(C)(C)CO)C(C)(C)C1 31717,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31718,N1(C(C2Cc3ccncc3N2)=O)CC2CCN(C(=O)CSC(F)F)C2C1 31719,CC1(C)COCCC1C(=O)NC1(CO)CCN(C(C2CCC(=O)N2)=O)CC1 31720,c1(C(=O)NCC2(CNC(=O)CC3CC4(CC4)C3)CC2)nsc2ccccc12 31721,c1(CC)ccc(N)c(C(=O)NC(CNC(c2cc(O)n(CC)n2)=O)CCC)c1 31722,n1(CC)nncc1C(=O)NC12CC(CNC(=O)C(C3(O)CCCC3)F)(C1)C2 31723,C1(CCC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)CC2CCOCC2)CC1 31724,c1(C(=O)NC(C(C)NC(Cn2nc(C)n(C)c2=O)=O)CO)ccc(C#N)nc1O 31725,c1(-c2n(C3CCC(OC(C)(C)C)C3)nc(CCCO)n2)cc(F)cnc1O 31726,c1(C(=O)NOC(C2C(C)(C)OC(=O)C2)C2CCCCC2)cc[nH]c2nccc1-2 31727,Cc1cccnc1C(=O)NCC1(C(=O)NCC(c2nccs2)C)CC2(CC2)C1 31728,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)Cc1c[nH]nc1O 31729,C1(C(=O)NC2CC(NC(CCCN(C(C)=O)C)=O)CC2O)CC2CC1CC2O 31730,N1(C(C2(COC)CCC2)=O)CCC(C(C)NC(=O)Cc2cccc(C(F)F)c2)CC1 31731,C(=O)(CCC(=O)N1CSCC1C(N1CCC(CC(N)=O)C1)=O)N(C)C 31732,N1(C(CC2CC(=O)NC2)=O)CC=C(CNC(C23CCCC2C3(F)F)=O)CC1 31733,N1(C(c2ccnc3c2CCC3)=O)CCN(C(C2CCC(O)C2)=O)C2(CCC2)C1 31734,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(C12CC(CO1)C2)=O 31735,c1(OC)ncc(Cl)cc1C(=O)NCC1CCC(NC(c2cnc(O)cc2C)=O)C1 31736,N1(C(c2cnn(C(C)C)c2N)=O)CCC(NC(C2(C)CC2(C)C)=O)CC1C 31737,CC(CC(C)(C)C)C(F)C(=O)N1CCOC2(C1)CN(C(=O)C(C)(F)C(C)(C)F)C2 31738,c1(CC(=O)NC2CCCC(NC(=O)Cc3nc(Cl)cs3)C2)cnn2ccccc12 31739,C1(OCCCNC(C(C)c2ccsn2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31740,CCCC(C)(O)C(=O)NCC(C)(C)CNC(c1ccnc(Cn2cnnc2)c1)=O 31741,N1(C(CC2CCC(=O)CC2)=O)CCC2CCCC12C(=O)NOCC1CCOC1 31742,C(=O)(C(C)(C)C(N)=O)N1CCC(CC(C)NC(c2nc(=O)n(C)[nH]2)=O)CC1 31743,C1(N(C(C2CC3(CCC3)C2)C(=O)NC2COC2)CC)CCCCC1O 31744,N1(C(c2cc(N)c(Cl)cn2)=O)CCC(C2CC2)(CNC(c2ccc(CO)o2)=O)C1 31745,CC(C)CCCC(C)C(=O)NCCOC1CCN(C(=O)CC2CCCO2)CC1 31746,c1(C(=O)NC23CC2CN(c2ncc4sccc4n2)C3)cc(Br)cc2[nH]ccc12 31747,Cc1ncccc1CC(=O)N(C1CC(NC(=O)CC2COC(C)(C)C2)C1)C 31748,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31749,C(C1CCCCCC1)=CC(=O)NC(C(C)C)CCNC(=O)CCc1nncs1 31750,C(C(CC(C)C)NC(c1c(CC)cno1)=O)NC1CCC(CCC(=O)OC)O1 31751,c1(C(=O)NC2(C)CC(NC(c3ccc[n+]([O-])c3)C)C2)cnc2n1CCCC2 31752,c1(CC)[nH]nc(C(N2CCC(N(C(=O)C(C)COC)CCOC)C2)=O)c1Cl 31753,CC(C)(C)C(CNC(C1CC1CF)=O)NC(C12CC3CC1C2C3)=O 31754,N1(C(c2cccc(CSC)c2F)=O)CC2(C1)CN(C(=O)C(O)CC(N)=O)CCO2.CO 31755,c1(NC2CCN(C(C(C)NC(CC)=O)=O)CC2C)ccc(C#N)c(C)n1 31756,c1(CC(=O)NCCC(CNC(c2c(C)cccn2)=O)O)ccn2cncc2c1 31757,C1(NC(C(C)OCCC#C)=O)C2CCN(C(c3sc(Br)cc3F)=O)C12 31758,c1(C(=O)NC2C=CCN(C(C3(C=C)CCCCC3)=O)C2)cn2c(C)nnc2cn1 31759,N1(C(CNS(C)(=O)=O)=O)CCCC1CC(=O)NCCOCCN(C)C 31760,Cc1ccnc(C(C)(C)C(=O)NCC(C)(C)CCNC(c2cc(C)ns2)=O)c1 31761,N12CCC(CC1)SCC2=O.c1(COC(C(=O)N(CC=C)C)C)ccccc1 31762,c1(C(N2C(CNC(CC(c3ccc(C)cc3)(C)C)=O)CC2)=O)cc(N)ccc1C 31763,c1(C(N)=O)ccc(NC(=O)CC2CN(Cc3ccc(Br)s3)CCO2)cn1 31764,c1(N)nc(O)ccc1[N+](=O)[O-].N1(C(C(=O)C2CCCC2)=O)CC(C=O)CC(F)(F)C1 31765,C1(CCC(=O)N(C(C)CNC(=O)C(C)c2ncco2)CC)CCC(=O)N1 31766,C1(CNC(C(F)=CCC)=O)(CNC(=O)C(Cc2ccccc2)SCC)CCCC1 31767,C(CC(C(=O)NC1CCCSCC1)NC(C1(F)CCOC1)=O)N(C)C 31768,c1(SC)ccc(C(=O)NC(c2ccccc2)CNC(=O)CC2CCOC2=O)o1 31769,N1(C(C2(C)N(C)CC(O)C2)=O)CC2CN(C(=O)Cc3c(F)cccc3Cl)CCC12 31770,CC1CC(CNC(C2(C(=O)O)CC2(F)F)=O)=NO1 31771,c1(C(N2CCC3(CCOC3)C2)=O)ncnn2ccc(Br)c12.C12(CCCC1)CC(=O)N2 31772,CC(Cc1ccnn1C)N=c1[nH]c2c(c(=NCC3C4CCCCC34)[nH]1)CSC2 31773,c1(C(=O)NC2CN(C(c3cc(C)n(C)n3)=O)CC2F)ccc2ccccc2c1O 31774,Cc1cn2c(n1)CC(C(=O)NC1CCC1NC(c1cc(N)cc(O)c1)=O)CC2 31775,C(=O)(C(O)CSC)NC(C1(CNC(=O)Cn2cnnn2)CC1)C.N(C)(C)C 31776,c1(C(C)NC(C2CC(C)(C)C2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 31777,C1(NC(C(C)OCCN(C)C)=O)COCCC1NC(=O)Cn1cnnc1O 31778,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(C(=O)Nc2c(C)cc(C(C)C)cc2)C1 31779,Cc1cc(C(=O)NC2CN(c3ccc(F)c(F)c3)C2)c2ccc(Br)cc2n1 31780,C(=O)(CCCCN1CCCC1)N(CCCNC(CCC=C)=O)CC1CCCC1 31781,c1(C(=O)OC)cc(OC)cc2c1OCC2.N12CC(SCC)(C1)CC(C)C2=O 31782,C(=O)(CC(F)(F)C(F)F)NC(C1(C(=O)NCC(CC=C)CO)CC1)C 31783,C1(C(N2CC(CCNC(C3CC(C)(F)C3)=O)C2)=O)CCN(CC(F)(F)F)CC1 31784,C(=O)(C(C)CC(C)(F)F)N1CCN(C(CN(C(C)C)C)=O)C(CCO)C1 31785,N1(Cc2cnc(COC)s2)C(C(=O)NC2CC(F)(F)C2)CC2CC12 31786,C#Cc1cncc(C(=O)NCCC2CCC(NC(c3ccc(C)c(C)n3)=O)C2)c1 31787,C12CCC(N(C)C)(CC1)c1nnnn1C2.n1(CCC)ccnc1NC1CC1 31788,C1(CNC(C(c2ccc(Cl)cc2)N(C)C)=O)COCCN(C(=O)CC(F)(F)F)C1 31789,C1(NC(=O)CCCn2nnnc2C(CCCCCOCC)(C)C)CC2CCC1C2 31790,C1(NC(C2CC(=C)C2)=O)CCCCC12CCN(C(c1cnc3cccnn13)=O)CC2 31791,N1(C(C=CC=CC)=O)CCC=C(C(=O)NCC2(OCC)CCCCC2C)C1 31792,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 31793,c1(C2C(=O)NCCCC(C)N2C2CC2)ccc(C(F)F)cc1F.C1(SC)CC1 31794,C1(C(=O)NC2CC(C)(NC(C(C)(C)C)=O)C2)CCCC(O)C1 31795,CCC1=C(C(=O)NC2C(C)CCN(C(c3csc(Cl)n3)=O)C2C)SCCO1 31796,c1(CCNC(=O)CCN2CCNC2=O)cccc(OCC(F)F)c1 31797,N1(C(C(CC)C#N)=O)CC(C2CN(C(=O)Cc3ccn(C(C)C)n3)C2)C1 31798,CCC(CC(C)C)C(=O)NC(C)CN(C)C(c1cn(-c2ccccc2)nn1)=O 31799,C1(NC(C2(C(C)NC(C3(C#N)CC3)=O)CC2)=O)COCC(C)O1 31800,c1(C(=O)NC2C3CN(C(C4C(C)=CCS4)=O)CC2C3)cc2cccc(C)c2o1 31801,c1(Nc2cc(NCc3cc4ccnn4cn3)nc(C)n2)cnc(C)c(C)c1C 31802,C(CCCCCCCO)N(C(=O)CCc1cn[nH]c1)CC1(C2C(C)C2)N=N1 31803,CC1CCN(C(c2cnn[nH]2)=O)CC1CNC(c1cc(C(F)F)nn1C)=O 31804,C=CCN=C(NCC1CCC(C(=O)N(C)C)CC1)N1CCC(C)(OC)C1 31805,C(=O)(C1=CCS(=O)(=O)C1)NCCC(C(C)C)NC(C1C(CN=[N+]=[N-])C1(C)C)=O 31806,n1(CC)cc(Br)c(C(=O)NCC2COCCN2C(c2ccc(O)cn2)=O)n1 31807,n1(CC)nc(C(N2CC(F)(C(=O)NC(C)CCC(C)C)C2)=O)cc1C 31808,Cc1oc(C(C)C)nc1C(=O)N(CC(O)CN(C(=O)C=Cc1ccncn1)C)C 31809,c1(C(N2CCSCC2Cc2ccccc2)=O)cnc2c[nH]nc2c1 31810,C1(NC(c2cc[nH]n2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 31811,C(C)(CN=c1cc(C)c(S(=O)(=O)NCCC2(C)CC2)c[nH]1)N1CC(C)OC(C)C1 31812,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 31813,CCCCCC(C)CC(=O)NC1(F)CN(C(=O)C2=CCC(C)CC2)C1 31814,C(=O)(CC1=CCCC1)NCc1c(CNC(CN2C(=O)OCC2)=O)cccc1 31815,C(=O)(CC(C)C(=O)NC(C1CCN(C(C2C(O)C(=O)N(C)C2C)=O)CC1)C)OC 31816,C1(C(=O)OC(C)(C)C)CC2(CCN2CCCNC(C2(Br)CCC2)=O)C1 31817,C1(CNC(C2(C=C)CC2)=O)CC(C(C)C)CCN1C(=O)C=CC1CCCC1 31818,c1(CC)ccc(C(=O)NCC2(NC(C3CCC(C)S3)=O)CCCCC2)c(C)c1 31819,c1(SCC(=O)NCc2cccc(CNC(C3C(C)C3)=O)c2)cccc(Cl)c1 31820,C1(C(N(C(CNC(CC=CC)=O)C)C)=O)CCc2nncn2CC1 31821,CC1CN(C(=O)C(O)C(F)(F)c2ccccc2)CC1P(C)(C)=O 31822,c1(C(C(=O)NCCC(=O)OCCC(C)C)C)ccc(F)cc1F 31823,C(=O)(CCC(=O)N(C)C)NCCNC(=O)NC1CCN(C(COC)=O)C1 31824,N1(C(=O)CCF)CCN(C(C2CC(c3c(C)n[nH]c3C)C2)=O)C(CC(F)F)C1 31825,N1(C(c2ncc(C)cn2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 31826,N1(C(C2CC(F)(F)C2(F)F)=O)CC2(C1)CN(C(C1(CC3CC3)CC1)=O)CCO2 31827,C(=O)(C(C)CC(C)C)NC(CCCNC(c1cccc(NC(C)=O)n1)=O)C 31828,CN1C(=O)CC(C(=O)NC(C(=O)NCCS(C)(=N)=O)c2ccco2)C1=O 31829,c1(C(N2C(C(=O)Nc3ccnc(F)c3)CC(=C)C2)=O)ccc2[nH]cc(Br)c2c1 31830,C=CCCCCCC(=O)N1CCCC1C1CCN(C(C2(CF)CC2)=O)C1 31831,c1(SC)ccc(NC(=O)CC2CCCN2C(=O)C=Cc2ccnn2C)c(F)c1 31832,c1(C(=O)Nc2cc(C(=O)OC)oc2C)c(OC(C)C)cccc1F 31833,C1(=O)CCCCCNC2C(C)CN1C2.c1(NC(=O)CC2CC(F)C2)ccccc1 31834,N1(C(C(CCCC)O)=O)Cc2ccccc2CC1CNC(C1(CSC)CC1)=O 31835,c1(C(C)=O)ccc(Cl)cc1NC(C1CCCN(Cc2ccc(Br)[nH]2)C1)=O 31836,c1(C(c2ccccc2)OC)ncccc1S(=O)(=O)NCCN(C1CNC1)C 31837,Cc1ccn(CC(C)(O)C(=O)NCC2CN(C(=O)C(C3CC3)N(C)C)C2)c(=O)c1 31838,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCCO)C4)c2C1 31839,N1(C(c2c(CC)c[nH]n2)=O)CC=CC(NC(=O)CSC)C1 31840,c1(CNC(C(CC)(F)F)=O)ccc2c(c1)CCC2NC(=O)CCCCCO 31841,C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(C(N1CCN(C(C)C)CC1)=O)C2 31842,c1(OC)ccc(F)c(F)c1CN1CC(NC(c2cc(Br)c(C)s2)=O)C(F)C1 31843,C1(C(N2CCCCC2CCNc2ncc([N+](=O)[O-])cn2)=O)CCC2CCCCN12 31844,c1(CC(=O)NCC2(C(=O)Nc3ccc(C)cc3)CC(=C)C2)ccc(C#N)cc1 31845,Cc1cc(C(N2CC(CNC(=O)C(=Cc3c[nH]cn3)F)C(C)C2)=O)nn1C(F)F 31846,C(c1ccncc1)=C(C)C(=O)N(C1CCCCC1)CC.C12CC(C1)NC(=O)C2C 31847,c1(C(=O)NC(CNC(c2c(OC)cccn2)=O)CO)ncnc2c1ccn2C 31848,C1(CNC(c2c(CC=C)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 31849,N1(C(C2N(C(CNC(c3c(C)ocn3)=O)=O)CCC2)=O)CC2C(C(N)=O)C2C1 31850,CC1CN(C(C2(n3cnnn3)CC2)=O)CC(C)C1NC(=O)C=Cc1cnn(C)c1 31851,C1(NC(C2CC2N)=O)CCCN(CC(F)(F)F)C1.c1(N)ccc(Cl)cn1 31852,C1(CCN(C)C(C2CCCO2)=O)COCCN1C(C1CSCCS1)=O 31853,c1(C(N2CCC2c2c(F)cccc2F)=O)ccc2ncccc2c1 31854,N1(C(=O)NCC(C)(C2CCC2)NC(C2CCC(F)CC2)=O)CC(OC)CC(F)C1 31855,c1(CC(=O)NC(CC)CNC(=O)C(COC(F)F)CC)ccc(OC)cc1 31856,C1(C(=O)Nc2n(CC)nnn2)C2CCC(C2)C1NCc1ccc(F)cc1 31857,c1(C(=O)OCC)[nH]c2ccccc2c1NC(N1CCCC(C(C)(F)F)C1)=O 31858,C(=O)(C1=CC2C=CC1C2)NC1C(CC(=O)NCCC(C(C)C)OC)CCC1 31859,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CC(NC(=O)CCc3csnn3)C2)C1 31860,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 31861,c1(C(c2nnnn2CCCF)NCc2c(CC)noc2C)ccc2ncsc2c1 31862,c1(CNC(COCC=C)=O)ccc(C(=O)NCCCC2CCCO2)o1 31863,C1(C)(CC)C=C(C(=O)N2CC3CC3(NC(=O)C(C)Sc3ccccc3)C2)C1 31864,C(CCC(C)C)(C(=O)NOCC(O)CO)NC(CC(CC=C)(C)C)=O 31865,C1(CC)CC(NC(C2C3CCCCC23)=O)CCN1C(c1cc(C(C)=O)c(C)o1)=O 31866,CCCCCS(=O)(=O)CC(=O)NCC(C(C)C)NC(=O)C#CC1CCCCC1 31867,c1(C(=O)OC)ncc[nH]c1=NC1CCCC(NCCC2CCCO2)C1 31868,C1(NC(CCCC)=O)COC2(C1)CN(C(=O)Cc1c[nH]c(=N)nc1O)C2 31869,C(=O)(C(CNC(C1(CCCC)CCC1)=O)CC(C)C)NCC(CC#C)(C)CO 31870,CC1(CCNC(=O)CC2CCC(=O)O2)CCN(C(c2cnoc2C2CCC2)=O)C1 31871,N1(c2nc(N(C)Cc3c(C)nc[nH]3)c3c(n2)CCS3)CCCC2CCC(C)CC12 31872,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 31873,N1(C(=O)Cc2ccon2)CCCC(CC(=O)NCCOCCCO)C1 31874,c1(CC)c(C(=O)NCC2(F)CC(NC(c3cc(N)ccc3C)=O)C2)cccc1C 31875,N1(CC(=O)NC2CCCN(CC(C)(C)N3CCCC3)C2)CCCCC1=O 31876,c1(C(N(C)CC2(NC(c3c(CC)nccc3)=O)CC2)=O)cc(O)ccc1C 31877,N1(C(C2=C(C)CCC2)=O)CC(NC(=O)COCCCF)C(C2CC2)C1 31878,c1(C(=O)OC)cc(F)ncc1NC(C1CN(C(c2sccc2C)=O)CCN1)=O 31879,c1(C(=O)NCC(=O)NCC(=O)NC2(C(C)C#N)CC2)cnc(C(C)C)nc1 31880,c1(NC(COCCC#C)=O)ccc(Br)cc1COC 31881,CC1(C)OCCOC1CC(=O)NC1CC(NC(c2cncn2C2CC2)=O)C1 31882,CCC(C)(COC)C(=O)NCCOCC.C(=O)(C(CC)SC(=O)OC(C)(C)C)CO 31883,CC(C)C(CC(=O)NC(C)CCNC(c1oc(Br)nc1C(F)F)=O)C(C)C 31884,C(CN=S(C)(C)=O)NC(C(CC)NC(=O)Cc1c(C)cnn1C)=O 31885,CN1CCC(C(N2CCC(C(=O)N(C)OCCSc3ccccc3)C2)=O)CC1=O 31886,C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(=O)CC(C)n2cccn2)C1C 31887,C#Cc1cccc(C(N2CC(NC(=O)C3CC3)CC2C)=O)c1 31888,C(=O)(CCCS(=O)(=O)c1ccc(F)cc1)NC1(C)CCN(C(C(C)SC)=O)C1 31889,CC1CC(C(=O)NC2(Cc3ccccc3)CC2)CCN1C(C1(O)CCC1)=O 31890,N1(c2ccnc(N3C(CC)CC(OC)C3)n2)CCN2CCOCC2(CO)C1 31891,c1(CC(=O)NC2CN(C(c3ccno3)=O)C2)cncnc1O 31892,C(=O)(CC(O)C(C)CC)N(CCC(C(C)C)NC(C1(CC#C)CC1)=O)C 31893,c1(C(C)C)ccc(C(=O)NC2CN(C(=O)CSC(F)(F)F)CC2C(F)F)cn1 31894,c1(N2CCC(C)(CO)C2)ccc(S(=O)(=O)CNC(=O)CCC(N)=O)cc1Br 31895,C1(C(=O)NCC23CC2CN(C(=O)C(F)Cc2ccccc2)C3)C2CCCCCC12 31896,c1(C(=O)NC(CNC(C(C)=CC)=O)(C)C2CC2)cc(C)c(-c2ccc(Cl)cc2)s1 31897,C1(C(N2CCC(CNC(=O)CCC=CBr)C2)=O)(CO)CCCCO1 31898,n1(C(C)C)ccc(=NC(=O)C2COC(C)(C)OC2)[nH]1 31899,c1(C(=O)NCC(C)CC#N)[nH]ccc1C(N1CCCCC1)=O.C1(C)C(=O)N1C 31900,c1(C(C(=O)NCCCCNC(C(SC)SC)=O)F)ccccc1 31901,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(N1CCC(N(C)CCO)CC1)=O 31902,C(=O)(C(C(C)C)n1cncn1)NC(CNC(C(CC)n1cnnc1)=O)C(C)C 31903,C(=O)(C(O)CC(F)F)NCCCC(C)NC(c1cnc(C)o1)=O 31904,c1(C(=O)Nc2cncc(CO)c2)ccc(F)c(-c2cc(F)ccc2O)n1 31905,C1(C(=O)NCCCCNC(c2ccc(C(C)C)cc2)=O)CCCCC(F)(F)C1 31906,N1(C(c2cnc(SC)s2)=O)CCC(C)C(CC(N2CCC2CC(C)(C)C)=O)C1 31907,C1(CN(C(CCN(C(COCC)=O)C)=O)CCO)CCCC(O)C1 31908,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 31909,CC(C)C(C(=O)NC1CCOC1C(=O)N(C)Cc1ccnn1C)n1cccc1 31910,C(C(C)(C)CNC(C1(Cl)CC1(F)F)=O)N(C(=O)CCCc1cccs1)C 31911,c1(C(=O)NCC2(NC(C(C=C=C)C)=O)CC2)ccc(NC)nc1C 31912,c1(C(N(CCC)CCNC(=O)C(F)C(C)C)=O)ccc(C(C)=O)c(F)c1 31913,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 31914,C12(NC(c3c(C)cnn3C)=O)CCC(CN(C(=O)CN3CC4CC4C3)C1)C2 31915,Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CCOCC2)=O)cnn1C 31916,Nc1ccc(-c2cn(C3CC(NC(c4nc(Cl)cs4)=O)C3)nn2)nc1 31917,C1(CC(=O)NCC=C(C)C)CC(O)CN1C(=O)CCC1OCCO1 31918,C(=O)(CCC(=O)NC(C)CNC(C1CCCC(CC)C1)=O)N(CCC)CCC 31919,CCC(CC)(CC)C(=O)N1CCC(CCNC(=O)CCSC(F)(F)F)CC1 31920,c1(OC)c(Cl)cc(NC(=O)C(=O)Nc2cnc(OC)c(F)c2)cc1Cl 31921,Cc1c(OC(F)F)cccc1C(=O)NC1CCN(c2ccnc(=N)[nH]2)CC1 31922,CC(C)(O)C(C)(C)C(=O)NCC1(CNC(C2CCCO2)=O)CCC1 31923,c1(C(=O)NC(C)CCCNC(=O)COCC2CC2)cncc(C(F)F)c1 31924,C1(C(N(CCCCC=C)C)=O)CC2CCC1N(C(c1cc(C(C)(C)C)on1)=O)C2 31925,C1(CNC(C2CC(C)OC2C)=O)(CO)CCN(C(C2(CC(F)F)CCC2)=O)CC1 31926,C1(CNC(CN(CC(C)C)C(c2cn(C3CC3)cn2)=O)=O)CCOC1=O 31927,c1(CN2CCC(O)(C(=O)NCc3cc(Cl)ccc3Cl)C2)cncc2ccccc12 31928,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 31929,CC1[PH](C)(C)CCN(C(=NCCC2CNC(=O)C2)NC2CCCCC2)C1 31930,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 31931,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 31932,C1(CCC)CCC(C(=O)NCCC(C)N(C(=O)CC2CCCN(C)C2)C)CC1 31933,C(=O)(C(F)(F)C(C)O)N(C(CNC(c1c(C(=O)OC)nn(C)n1)=O)C)C 31934,Cc1cn2cc(C(=O)N(C3CCN(C(c4cnccn4)=O)CC3C)C)ccc2n1 31935,c1(C(=O)NCCCCCNC(C(C=C)(C)CC)=O)ccc([N+](=O)[O-])c(N)n1 31936,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(CO)c2ccccc2)C(CO)C1 31937,C1(C(N(C)CC23CC(NC(=O)C=CC(=O)N(C)C)(C2)C3)=O)CCC1(F)F 31938,C1(C(N(CC(C=C)O)C)=O)CC(=O)CN1C(=O)C(c1cccn1C)=O 31939,C1(NC(C(CCC)(C)O)=O)CC(C2CCN(C(=O)C=Cc3ccncc3)CC2)C1 31940,C1(CC(=O)NCC(c2ccco2)NC(=O)CC2(O)CCCC2)CCC2CC12 31941,C(CC(=O)N(CC(O)CN(C)C(C1CC(CCO)C1)=O)C)OCC(C)C 31942,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CCC2)csc2c(O)ccnc12 31943,c1(N2C(C(=O)NCc3cc(I)c(O)c(I)c3)CC2)ncnc2ncc(Br)cc12 31944,c1(C(N2CCC(CNC(C(C(C)O)C)=O)C2)=O)ccc(N)c(Cl)c1O 31945,CCC(C)(CNC(=O)C(CN(C)C)NC(=O)C=Cc1cncn1C)CC 31946,Cc1c(C(=O)NC(C)C(CO)NC(=O)C2=NOC(C)(C)C2)nc2sccn12 31947,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CC(NC(=O)C#CC2(C)CC2)C(O)C1 31948,CC1(C)CCN(C(=O)C=CC2CCCCC2)C1C(=O)NC1CC2CCCCC12 31949,C1(NC(CCOCC#C)=O)(CO)CCN(C(c2cn(-c3ccccc3)nn2)=O)C1 31950,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 31951,Cc1nc2ncc(C(N3CCCC(CO)(NC(C4CCC(=O)N4)=O)C3)=O)cc2o1 31952,Cc1ncc(C(=O)NCCC2CCN(C(=O)CC(O)C(C)C)C2)c(=N)[nH]1 31953,Cc1ncc(NC(=O)CC2CC(NC(C3C4(CC4)C34CC4)=O)C2)cc1Br 31954,Cc1cc(N2CCC(NC(C3CCCC3(C)C)=O)C(F)C2)nc(S(C)(=O)=O)n1 31955,c1(C(=O)NC2C3CN(Cc4cc(C#N)sc4)CC32)cc(Cl)nc(Cl)c1 31956,C=C(C)CC(C(=O)C(=O)CCN)NC(C1CC(C)(C)C1)=O 31957,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 31958,C(=O)(C1CCCc2cncn21)NCCCCNC(C(C)N(C)C)=O 31959,Cc1nc(C(=O)NCCC(N2CCC(C(N3CCCC3)=O)C2C)=O)c(C)s1 31960,C#CCC(CC(=O)N1CC(OC)C1)NC(=O)CCNC(=O)COC1CCOC1 31961,c1(C(N(CCCc2cn[nH]c2)C)=O)c[nH]nc1CCNC(=O)C(C1CC1)OC 31962,C1(NC(C)=O)CCCC(NC(c2cc(-c3ccccc3)[nH]n2)=O)CC1 31963,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 31964,Cc1coc(C(=O)NC(C)(C)CN(C(=O)C(C)C2CCCC2)C)c1C 31965,C1(C(=O)NC2CN(C(c3cccc(Cl)c3Cl)=O)C2)CCC2CC2CC1 31966,CCCCCCCCCCC(=O)NCC(CO)NC(c1c(CO)n[nH]c1C)=O 31967,c1(C(N2C3CCN(C(=O)CCN4CCC4)CC2CC3)=O)cc2cccc(F)c2o1 31968,c1(C(=O)NC2COCC2CNC(c2ccc(Cl)s2)=O)cc2nccn2c(O)n1 31969,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)C(C)SCc1cccnc1 31970,c1(CC(=O)NC(CC2(C=C)CC2)=O)ccccc1Br 31971,c1(C(N2CC(CC(N3C(C#C)CCC3)=O)C2)=O)cccc2[nH]ncc12 31972,c1(C(N2C(CCNC(C(C)OC3COC3)=O)COCC2)=O)cnn2ccn(C)c12 31973,CC1(CNC(=O)CC2CCC(NC(C3OC4CCC3C4)=O)C2)CCCCO1 31974,CCCCC(C)C(=O)NCCC1(NC(C2CCC(=O)CC2C)=O)CCOCC1 31975,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(C2CC2F)=O)CCC12CCC2 31976,c1(C(N(CCCNC(=O)C(C(C)C)SC)CC)=O)cncc(N)c1.C(C)(=O)O 31977,c1(CC(=O)NCC(CNC(C(C)n2ccnc2)=O)F)cccc2cn[nH]c12 31978,CC1(C)C(C(=O)NCC(P(C)(C)=O)c2ccccc2)(CO)C1(C)C 31979,C(=O)(C(F)(F)c1ncccn1)N(C1CCN(C(=O)Cc2cc[nH]c2)C1)C 31980,C1(CNC(CC(C)n2ccnc2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 31981,c1(C(N2CC(SC)C(NC(=O)CCSC(F)(F)F)C2)=O)ncnc2c1ccn2C 31982,c1(-c2cc(C)cc(OC)c2C)cccc2[nH]nc(C(=O)Nc3conc3C)c12 31983,Cn1ccc(S(=O)(=O)NCC(=O)NCCNC(c2cnc(Cl)s2)=O)c1 31984,C#CCCCC(C)C(=O)NCC1CCCC1NC(=O)CC1CCC(=O)NC1 31985,N1(C(C2C3CN(C)CC32)=O)CCC2C(CCN2C(c2ccc(F)cc2Cl)=O)C1 31986,C1(NC(CCSC)=O)CCN(C(c2cnc(-c3ccccc3)nc2)=O)CC1O 31987,N1(C(C(c2n(C)cnc2)O)=O)CCN(C(c2cocn2)=O)C(CO)C1 31988,c1(OC)cc(C)cc(C(=O)NCC2CC(O)CN2C(=O)CC(=O)N(C)C)c1C 31989,c1(C(=O)NCC2CC(F)(CNC(C(CC#C)C)=O)C2)cc(C)c(C)nc1C 31990,c1(C(=O)NC2C(NC(C(F)=CC)=O)COC2)sc(O)nc1C 31991,c1(OC)nccc(C(=O)NC2CC2CNC(=O)C(CCC2CC2)NC(C)=O)n1 31992,C1(CNC(=O)NCC2(C(=O)OC(C)(C)C)CC2)CC2(C1)C(F)(F)C21CCC1 31993,Cc1c(CN(C)C(=O)NCCC2COCCO2)cccc1F 31994,N1(C(C(CC2CCC2)NC(=O)CC2CCOCC2)=O)CCC2(CC1)CSC2 31995,N1(C(CC(C)SC)=O)CCC2(CC1)CN(C(=O)CC1COCCO1)C2 31996,c1(CNC(C2C(OCC)C2)=O)nc(CNC(C2(Cl)CC2)=O)cc(O)n1 31997,C1(NC(C(CC)CC)=O)CC2CC(NC(C3CN(C(=O)NC)C3)=O)CC2C1 31998,C1(NC(c2ccc(C(N)=O)o2)=O)(C)CCN(c2ccc(Cl)c(O)n2)CC1.C(=O)(C1CC1)N 31999,Cc1nc2cc(n1)N1CCOC(C1)Cn1cc(nn1)CN2.C(CCO)NC=O 32000,C(=O)(C1=C(C=O)C(c2ccccc2)NC(=O)N1)OC.N1(CC)CCC2(CC=CCO2)C1 32001,N1(C(CC2C(=O)OCC2)=O)CCOCCC1CNC(=O)Cn1cccn1 32002,c1(C(=O)OCc2cc(CC(=O)OC)no2)sc(C)c(Br)c1C 32003,c1(OC)cnc(C(=O)NCC2(O)CCCN(C(=O)CC(C)C(F)F)C2)c(F)c1 32004,N1(C(CC2CC(=C)C2)=O)CCN(C(c2cccc(F)c2C)=O)CC2(CC2)C1 32005,C(=O)(C1=NOC2COCC12)NC(C)CN(C)C(C1C2(CC2)C12CC2)=O 32006,C(C(=O)ON1CCC(n2cncn2)C1)(C(C)C)SC.C12(CCCC1)C(=O)N2 32007,N1(C(C2C(C=C)C2)=O)CCC(O)C(NC(=O)Cc2csc(-c3ncccn3)n2)C1 32008,Cc1cc(F)sc1C(=O)NC1(c2ccccc2)CCN(C(C2CNC(=O)C2)=O)C1 32009,N1(C(C(c2scc(C)n2)C)=O)CCC(CNC(=O)C#CC(C)(C)C)C12CC2 32010,Cc1ccc(CN(CC(C)NC(=O)C2=CC3CCCC23)C)c([N+](=O)[O-])c1 32011,CN1CCC(CC(=O)NCC2COCC2NC(c2ccc(C(F)F)nc2)=O)C1=O 32012,C=C(C)CC(C(=O)NC1CC12CC(NC(=O)CSc1ncccc1O)C2)OC 32013,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C(NC(=O)C(F)(F)c2cncs2)C1 32014,CC1CN(c2nc(C3CCOCC3)ns2)CCC1NC(c1ccnc(F)c1)=O 32015,c1(-c2cn(C(C)C(=O)N(CCC(N3CCC(C)CC3)=O)C)nn2)ccc(Cl)nc1 32016,N#CC1CCCCN1C(c1nc(Br)c(-c2ccccc2)s1)=O 32017,C1(CNC(C(C)OCCCC)=O)CCCCN(C(=O)CC2(CSC)CC2)C1 32018,N1(C(C2CCN(C)C(=O)C2)=O)CC2(CCN(C(=O)CN3CCC(C)(O)C3)CC2)C1 32019,CCC(C(=O)NCC(C)N(C(c1nnc(Cl)cc1N)=O)CC)C(C)(F)F 32020,C1(C(=O)NCC(C)NC(=O)C=CCN(C)C(=O)[O-])CC2C(C1)C2(C)C.C(C)(C)(C)O 32021,C1(CN(C(COCCC#C)=O)C)CN(C(=O)C(c2ccc(Cl)cc2)C)CC12CC2 32022,N1(C(C2(C(C)C)COC2)=O)CCCC(O)(CCNC(c2nccn2C2CC2)=O)C1 32023,C(CC(C)C)(C(=O)N1CC(N2CC(CNC(=O)CC3(CO)CC3)CC2=O)C1)OC 32024,c1(C(N2C(C)CC(NC(=O)CCCN3CCCCC3)C2)=O)cncc(N=[N+]=[N-])c1 32025,N1(C(C2C(C#C)C2)=O)C2CCC1CN(C(c1ccc(N)c(O)c1)=O)CC2 32026,C(=O)(N=c1[nH]nc(Cl)cc1O)NC1N(C(C(COC)C)=O)CC=C1 32027,C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1ocnc1C(F)F)=O 32028,c1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CC2)=O)ccc(Cl)c(Cl)c1O 32029,c1(C(=O)NCCC(C)NC(c2c(C)cn(CC)n2)=O)cnn2c1OCC(C)C2 32030,c1(C(=O)NCC2(NC(COC(CC)(C)C)=O)CCCCC2)cn2cnnc2cn1 32031,n1(CC)cc(Cl)c(C(=O)N(C2CCCC2)C(=O)CC2CC2C)n1.CCCS 32032,C#CC1CC1C(=O)NCC(C)N(C(=O)COCCCOC)CC 32033,N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC(C)(O)C3(C)CC3)CO2)C1 32034,Cn1nc(CO)cc1C(=O)NCC12CC(CNC(=O)OC(C)(C)C)(C1)C2 32035,CC(C)(C)CC(F)C(=O)NCCCNC(=O)CCN1CCCC(C(N)=O)C1 32036,CC12CN(C1)C2=O.C1(CCC(N2CC(c3ccon3)C2)=O)CCC(=O)C1 32037,Cc1cc(NC(=O)NCC2(CO)CC2(C)C)ccc1N1CCN(C)CC1 32038,N1(c2nnc(CC)s2)CCC2CC12CNC(=O)CNS(C)(=O)=O 32039,c1(C(=O)NC2CN(C(c3cccc4sccc34)=O)C2)cc(F)cc(F)c1Br 32040,N1(C(CC(C=C)C)=O)C(C)CC2CN(C(=O)C(C3(O)CCCC3)F)CC12 32041,C(C(F)(F)CC(O)CO)NC(C1=CCCSC1)c1n(CCC(=O)OCC)nnn1 32042,Cc1c(Br)ccc(F)c1C(=O)NC(CNC(c1cnc(O)s1)=O)C1CC1 32043,c1(C(=O)NCC(C2CC2)NC(CSCC(C)C)=O)c(F)cc(F)cc1Cl 32044,C1(C(=O)NC(C#C)C2CCC2)C2CC3C(C2NC(=O)CCCCOC)C13 32045,c1(CC(C(=O)OC)N(C2CC(n3ccnn3)C2)C)ccc(OC)cc1 32046,c1(CN2C(C(=O)NCc3c(C)ccc(Br)c3)C3CCC2C3)ccc2nc[nH]c2c1 32047,C(C(=O)NCc1cncnc1C)(C(C)(C)C)NC(c1c(C)n[nH]c1)=O 32048,N1(C(C2CCN(C(C)C)CC2)=O)CC2CC(CNC(=O)C3=COCCO3)C(C2)C1 32049,c1(C(N(C(C)C)CCNC(c2cc[nH]c2)=O)=O)nccc2ccn(C)c12 32050,C1(NC(C(C)O)=O)CN(C(c2snnc2-c2ccccc2)=O)CC1C 32051,C1(CC)CN(C(C2C3CCCCC23)=O)CC1C(=O)NC1CCC1N(C)C 32052,N1(C(C(CCCC)O)=O)CCN(C(=O)CCc2cocn2)C2(CCC2)C1 32053,C1(C)(C(=O)NCC2(O)CN(C(CCCOCCC)=O)C2)CCCS1(=O)=O 32054,C1(CNC(c2ccc(C3CC3)o2)=O)COCCN1c1nccc(C2CCCCO2)n1 32055,c1(C(N2CCC(CN(C(=O)C(c3cnccc3C)O)CC)C2)=O)cnc(C)nc1 32056,CC1CC2CCCCC2N1C(C1CC(NCc2sccc2OC(F)F)C1)=O 32057,N1(Cc2cc(C)[nH]c2C)CC2(CCN2C(c2c[nH]c(C(C)(C)C)c2)=O)C1 32058,C1(C(=O)NC(C)CCCNC(C2CCS(=O)CC2)=O)CC2(CC(=O)N2)C1 32059,C1(CCNC(=O)CCCn2ccnc2)CC(F)(F)CN1C(c1cocn1)=O 32060,c1(C(C(=O)NCCN(C(C(C)n2cccn2)=O)C2CCCC2)C)ccnn1C 32061,C(c1cnc2ccccc2n1)=CC(N1CCC(NC(C2C(C)C2)=O)C12CC2)=O 32062,S(=O)(=O)(c1ccc(NC2CCOC(CC)C2)cc1Br)NCC(C)(C)OCC 32063,c1(C(=O)NCC(CNC(C(C(=C)Cl)(C)C)=O)CC)cn2cc(C)ccc2n1 32064,C1(CN(C(c2n(CC)ccc2)=O)C)CCCCN1C(c1ccc(C(C)C)cn1)=O 32065,c1(C(=O)Nc2n[nH]cc2C2CC2)ccc(-c2ccccc2)c(F)c1 32066,C1(CNC(C(F)=CCC)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32067,CCC(C(C)(F)F)NC(c1cnn(CCNC(C2CCC(CC)C2)=O)c1)=O 32068,C(=O)(CCCCC(N)=O)NC(CC(=O)NCC1(C)CCN(C)C1)C(F)F 32069,C(N=c1[nH]c(=NCCN(C)C2CC2)[nH]c2ncn(C)c12)C1N(CC)CCCC1 32070,C#Cc1ccnc(NC(C(c2nnnn2C2CC2)C2CCC2)C(F)F)c1 32071,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1 32072,CC1(C)CC(CNC(=O)C(F)=C2CCC2)N(C(=O)CC2CC3CC3C2)C1 32073,C(=O)(CCC(C)S(C)(=O)=O)NCC(CCC(O)C=O)C.Cc1nn(C2CC2)c(Cl)c1C(=O)N 32074,CCC(C)C(C(=O)N1CCOCC1)N(C)C.N12CC(c3ccccc3)(C1)C2=O 32075,c1(C(N2C(CCNC(c3c(C)cncc3F)=O)CCC2)=O)cnc2scc(C)n12 32076,CC(c1ccccc1Cl)=CC(=O)NC1CC(CNC(c2cc(C)nc(C)n2)=O)C1 32077,Cc1ccc(O)c(C(=O)NCCCNC(c2ccn(C)n2)=O)n1 32078,c1(C(=O)NC(C2(O)CCN(C(c3cc[nH]c(=N)c3)=O)C2)C)cc2n(c1)CCCC2 32079,N1(CCC(=O)NCC(C2CCC2)NC(C=CCC)=O)CCCC(N(C)C)C1 32080,c12nn(cc1Cl)C(=O)N(CC)CCn1cc-2nn1.C1(C)(NC2CC2)CC1Br 32081,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32082,C1(NC(C2(CC=C)CCOC2)=O)C2CC1N(C(c1cnc(C(C)(F)F)s1)=O)C2 32083,c1(N2CCN(C)C(C)(C)C2)nc(N2CCOCC(C)(C)C2)nc2cccnc12 32084,N1(CC)CC(C(=O)NCC2CCC2NC(c2ccnc(OC(C)C)c2)=O)NC1=O 32085,C(CCCCCC(=O)NC(c1nncn1C)C)NC(C(COC(C)=O)C)=O 32086,N1(C(C(CSC)(C)C)=O)CCCC2(NC(c3ncc(C(N)=O)cc3Cl)=O)CC2C1 32087,C(CC(=O)NOCCC(C)O)(C(C)(C)C)NC(C1(COCC)CC1)=O 32088,c1(C(N2CCC(C)(NC(C3CCC(C)(C)C3)=O)CC2)=O)cnc(O)c2ccsc12 32089,C(CC(C(=O)NCc1nc(CC)n[nH]1)NC(=O)CC1CC(=O)C1)=CC 32090,c1(C(N2CCC(C#C)(O)C2)C(=O)NC2CCOCC2)ccc2cc[nH]c2c1 32091,C(CNC(c1c[nH]nc1OC)=O)(CCC)NC(C(C)=CC)=O 32092,C12(C(=O)NC(C3CCN(C(c4n(CC)ccc4)=O)C3)C)CC(C1)C(C)(C)O2 32093,C1(F)(C(=O)NCC2CC(NC(=O)Cn3cnnc3O)C2)CCCCC1 32094,N1(C(C2C3CN(C(CC4CCC(C)(C)C4)=O)CC32)=O)CC2(CCOCC2)C1 32095,O=C1CN(Cc2ccnc(Cl)c2)C(=O)N1CCOC1CC1 32096,N1(C(CNC(CCC)=O)=O)CCC(C2CCCN(C(c3coc(Cl)c3)=O)C2)C1 32097,Cc1cnc(NCC23CCC(CC2)CC3)nc1C.C1CNCC1C 32098,C(=O)(CCCCCF)N(C)CC1CCCC(NC(CN2C(C)CCC2)=O)C1 32099,C1(C2CCCCCC2S(N)(=O)=O)CCCN1NC(=S)NCC(F)(F)F 32100,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N2CCN(C(C3CCOC3)=O)CC2)C1 32101,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32102,N1(C(c2c(C#N)scc2)=O)CC(NC(c2cc3ncccn3n2)=O)CC12CCOC2 32103,C#CCC(CC(=O)NCCC12CC(CCO1)C2)NC(=O)Cc1ccoc1 32104,c1(OCC(=O)NC(C)CCNC(=O)C(Cl)=CCl)cccc(O)c1 32105,N1(C(C(OCC)OCC)=O)CCC(C(=O)N(C)CC2CC2(F)F)C(O)C1 32106,C(=O)(CCC(C)(C)N(C)C)NC(C)CNC(c1cn(-c2ccc(Cl)c(F)c2)nn1)=O 32107,C1(CN(C)C)CCCN1C(=O)NCN1CCCC1=O 32108,c1(C(N2C(C)CC(NC(=O)COCC3CCC3)C2)=O)cc(F)cc2nc[nH]c12 32109,CN1CCCC1C=CC(=O)NCC1(O)CCN(C(c2cscn2)=O)C1 32110,c1(CNCc2ccc(SC(C)(C)C)cc2)ccc2cc(F)ccc2n1 32111,C1(C(=O)OC)CC12CCN(C(c1cscc1Cl)C(=O)NC1CC1)CC2 32112,C(=O)(CCCCCC#N)NCc1ccc(C(N2CCC(C#CC)C2)=O)cc1 32113,N1(C(C(Cc2cc[nH]n2)NC(CCCN(C)C)=O)=O)CC2C(C1)C2(C)C 32114,c1(C(N2C(CNC(CCN(C)CC)=O)CC(OC)C2)=O)cc(C)nc2ncnn12 32115,N1(C(C(C)=CC)=O)CC(C2CN(C(c3cc4ncccc4s3)=O)C2)C1 32116,C12(NC(C(C)OCCCC)=O)CC1CN(C(=O)C(C)=NOCC#N)C2 32117,c1(C(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)CC2)=O)cc(C)nc(Cl)c1N 32118,C1(CC#C)CCCCN1C(=O)C(C)NC(c1ncccc1F)=O 32119,C1(C)(CC(N2C(C(=O)NCCNS(C)(=O)=O)CC2)=O)CCOC1 32120,C(C(O)C(=O)NC1CCC1NC(=O)CN(CC)CC)=CC 32121,Clc1ccc(C(=O)N(c2ccccc2)c2ncn[nH]2)cc1Cl 32122,C(CC(=O)NOCC1CC1)C1CN(C(C(C)(C)C)=O)C1.C1(O)CC(C)N(C)C1 32123,C1(O)(CNC(CCc2onc(CC)n2)=O)CCN(C(c2snnc2C2CC2)=O)C1 32124,N1(C(CC2C(OCC(=O)OCC3CC(Cl)C3)CCC2)=O)CCCCCC1 32125,CCCCC(C)C(=O)N1CCN(C(c2cc(SC)no2)=O)C(C(C)C)C1 32126,N1(C(C(C)(C)NC(C)=O)=O)CC2(C(=O)NC(CO)CO)CC1CO2 32127,c1(SC)nc(N2CCC(NC(c3cncn3C)=O)C(F)C2)cc(C(F)F)n1 32128,C(=O)(C1=COCCC1)N(C)CC1CCN(C(c2c(C)n[nH]c2)=O)C1 32129,N1(C(C2CCN(C3COC3)CC2)=O)CC(NC(=O)CSC(F)(F)F)C(O)C1 32130,C1(NC(C(C)OCC(C)C)=O)CCC(NC(=O)CN(C)C)CC1 32131,Cc1cnc(C)c(NC(C2CCCN2C(=O)CNC(=O)CCCNC(N)=O)=O)c1 32132,c1(-c2nc(CC(C)OC)nn2CCC(C)(C)C)cc(Cl)ncc1Cl 32133,C1(CNC(CC(CCC)CC)=O)CCCC2(CN(C(c3ccnnc3)=O)C2)O1 32134,c1(OCC)ccoc1S(=O)(=O)NC(c1cnn(C(C)C)n1)=O 32135,Cc1c(C(N2CC(NC(=O)C(C)C(F)(F)F)CCC2C)=O)cc(Br)cc1N 32136,S(=O)(=O)(C1COC(C)(C)C1)NC(C(=O)NC)C(C)C.C1(=O)N(C)CCO1 32137,CCN=C(NCc1ccccc1Cl)NC1CCC(C(=O)OC)C1 32138,C12(CNC(C(C)n3cncn3)=O)CN(C(c3ccc(O)c(F)c3F)=O)CC1CCO2 32139,O=C(N=c1cc(C2CCOC2)[nH][nH]1)C1CN(S(=O)(=O)CCC(F)(F)F)CC1O 32140,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32141,c1(NC)cncc(C(=O)NCCN(C)C(C23CC4CC2C3C4)=O)n1 32142,C1(CNC(c2ccc(Cl)cc2)=O)CN(C(c2coc(Br)n2)=O)CC1O 32143,C(=O)(C(C)(C)C(=O)NC1CCCC(NC(=O)CCc2nccn2C)C1)OC 32144,c1(C(CNC(=O)CN(C)C(=O)C2CC2)NC(C2C(OC)CC2)=O)ccccc1Cl 32145,N1(C(c2cn(CC(C)C)nc2)=O)CCN(C(=O)C(Cl)=CCl)C2CCCCC12 32146,N1(C(C2N(C(c3c(C)oc(CO)c3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32147,C#Cc1ccc(C(=O)NC(C)C(C(C)C)Nc2cc(C(N)=O)ncn2)c(F)c1Cl 32148,C1(CNC(COC(C)=O)=O)CCC(C)(C)CN1C(c1ccc(N(C)C)nc1)=O 32149,C(C1=NOC2CN(C(C34CCC(F)(CC3)C4)=O)CC12)NC(c1nn(C)c(O)c1)=O 32150,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2(Cl)CC2(F)F)=O)CC1)C 32151,Nc1[nH]c(=O)c(Cl)nc1C(=O)NC1CC(CCNC(C2CC(O)C(F)C2)=O)C1 32152,Cc1nc(C(=O)NC2(CNC(C3(CN(C)C)CC3)=O)CCCC2)c2n1CCCC2 32153,N1(C(C(C2CN(C(C3CC=C(C)CC3)=O)C2)O)=O)CCC(C)(O)C(O)C1 32154,N#Cc1cnccc1-c1cncc(C(N2CCOC3CC23)=O)n1 32155,CC(CF)CC(=O)N1CC(N(C(=O)CSc2ccc(-c3cccc(F)c3)o2)C)C1 32156,n1(CC)ccnc1C(=O)NC(C)(C)CCC1CCCN1C(=O)CCN(C)CCO 32157,C(CCN(C)C(c1cc(O)n(C)n1)=O)(C(C)(C)C)NC(CNC1CC(SC)C1)=O 32158,N1(C(C23CC(CCC)(C2)OC3(C)C)=O)Cc2c(F)cccc2CC1C(=O)OC 32159,C12(NC(Cn3c(C)ccn3)=O)CCCC1CN(C(c1cc([N+](=O)[O-])cn1C)=O)C2 32160,CC1CCCCN1CC(N1CCN(C2(c3nccn3C)CC2)CC1)=O 32161,C=CCC(CC)C(=O)ONC(=O)Cn1cc(CC(O)CC2CCC3C(O2)C3)nn1 32162,c1(C(=O)OCC)oc(C(N2CC(CNC(=O)CCCc3ccsc3)C2)=O)cc1C 32163,C12(C(N3CCC(O)(C(C)NC(C(C)=CC4CC4)=O)C3)=O)CC3CC1C2C3O 32164,c1(C(N2CCC(N(CCOC)C(C3CC3C3CC3C)=O)C2)=O)nc(C)cc(C)n1 32165,c1(C(C(=O)NC(C(C)C)CNC(c2nnsc2C(F)F)=O)C)cc(F)cc(F)c1 32166,N1(C(C2C(C)(CC)C2)=O)CCC(CCNC(=O)Cn2cnnn2)CC1 32167,c1(C(=O)NCC#CCNC(=O)COCC2CCC2)cn2ccnc2cn1 32168,N1(C(C(C)OCCC=C)=O)CCCC(N(c2ccc(-n3ccnc3)cc2)C)C1 32169,c1(CN2CC(NC(=O)Nc3cccc(C)c3Cl)NCC2)ccc2ncnn2c1 32170,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)O)c(F)ccc(F)c1F 32171,c1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)cc(F)cc2nccnc12 32172,C1(NC(c2c(C)cc(C)o2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)C)CC1O 32173,C1(C)(CCC)CCN(C(C2CCC(NC(=O)C(O)CCSC)CC2)=O)C1 32174,C1(NC(C(F)=C(C)C)=O)CCCCCN(C(c2ccc(C(C)(C)C)cc2)=O)C1 32175,c1(C(N(CC(CNC(C2(COC)CCOCC2)=O)C)C)=O)nc(C)ccc1OC 32176,C1(NC(CC2CC(C)C2)=O)C2CC3C1C3C2C(=O)N(C1Cc2ccccc2C1)C 32177,C(=O)(C(CC1CCCO1)C(F)(F)F)NCC(CNC(C(C)(C)N1CCOCC1)=O)F 32178,C(=O)(C1=CCCOC1)NCC1CC(NC(C2CC(OCC)C2)=O)C1 32179,Cc1nc(C(=O)NCC2CCCN2C(=O)Cc2cn3ccsc3n2)cc(O)n1 32180,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32181,CC(=O)CCCC(=O)NC12CC(C1)N(C(=O)C(C)Cc1cnco1)C2 32182,C1(C(=O)NC(CCOC)CNC(=O)CN2C(=O)CCCC2=O)CCCC(F)(F)CC1 32183,CCC(F)(F)C(C)(C)C(=O)N(C1CCN(C(C23CCC2C3)=O)CC1)CCO 32184,c1(C(N2C3CCC(NC(c4cnc(Cl)s4)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 32185,C(=O)(CCOC(=O)Cc1cnsc1)OC(C)(C)C 32186,c1(C(N2C3CCC(NC(=O)CCF)C(C3)C2)=O)ccc2c(c1)CCC2(F)F 32187,CC(C(C)CO)N(C(c1sccc1Cl)C(=O)NCc1ccc(Br)s1)C 32188,Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)ccc3O)=O)C2)nc(Cl)c1 32189,N1(C(C(C(C)C)(C)C)=O)CC(NC(c2ccc3ncoc3c2)=O)C(S(C)(=O)=O)C1 32190,c1(OCC#C)ccc(C(=O)NCCCCN(C(c2cc(Cl)no2)=O)CC)cc1 32191,c1(C(N(C2CN(C(C3(OC)CCCOC3)=O)C2)C)=O)cc2c(C)c(F)ccc2[nH]1 32192,Cc1cn2ccc(C(=O)NC3CC(C(=O)NCc4nccs4)C3)cc2n1 32193,N1(C2CCN(C(c3c(C)occ3)=O)C2)CCN(C(=O)CCC2CCC(=O)N2)CC1 32194,N1(C(C(C)(C)N2CCCCC2)=O)CCCCC1COC(=O)C1CC1 32195,c1(OC)cc(NC(C2CC2NCc2ccnc(C3CC3)c2)=O)c(C)cn1 32196,N1(C(C)C(=O)NC2CN3CCC23)C(=O)c2ccccc2S1(=O)=O 32197,c1(OC)ccc2c(c1)C(=O)CCN2C(=O)Cn1ccnc1C(=O)O 32198,N1(C(c2c(CC)non2)=O)C2CCCC1CC(NC(c1cnnc(O)c1)=O)C2 32199,C1(C(C)C)CN(C(=O)C(N2CCNC2=O)C)CCN1C(=O)CS(C)(=O)=O 32200,C(CCC(C)C(=O)NC1CCN(C(=O)CC(O)CN(C)C)CC1C(N)=O)OC 32201,c1(C(C(=O)NCC2(O)CN(C(CC=C)=O)C2)(C)C)cc(F)ccc1Br 32202,C1(CNC(c2c(CC)cno2)=O)C(C)CCCN1C(=O)Cn1ccnn1 32203,N1(C(c2c(C)cc(CNC(C3CC34CCC4)=O)o2)=O)CCCC2C(=O)NCC12 32204,N1(C(CNC(CSCC#C)=O)=O)CCCN(C(=O)COCCOC)CCC1 32205,C1(C(N2CCCC(CNC(C3CCC3)=O)C2)=O)CCC2CC1CO2 32206,C1(CC(=O)N(CCC)CCNC(=O)C2=C(Cl)CC2)CSc2ccccc2O1 32207,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32208,N1(C(CC2(OC)CC2)=O)CC(NC(=O)CCc2ccc(OC)nc2)C(C)(C)C1 32209,c1(COC)nc(Cl)nc(N2CCC(NC(C3CCC(N(C)C)CC3)=O)CC2)c1Cl 32210,N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)C1CNC(=O)CC(C)C1CC1 32211,c1(C(=O)NCC2(CC(=O)Nc3cncc(CO)c3)CC2)c[nH]ccc1=O 32212,CC(C)CC(C)(CNC(=O)C=Cc1ccn(C)c1)NC(c1cn2ccnc2s1)=O 32213,C(=O)(C(C)(C)S(C)(=O)=O)N1C(CNC(C(c2ccccc2)SC)=O)C=CC1 32214,O=S(=O)(c1ccc(F)c(F)c1F)N1CCC2(CCSCC2)C(O)C1 32215,C#CCC(CO)NC(C1(CNC(=O)CCOC2CC2)CCC1)=O 32216,C1(C(=O)NC2CCN(CC(C)C)CC2)CC2(C1)CN(C(=O)CC1COCC1O)C2 32217,C(CC(O)C(=O)NCC1(O)CN(C(C2CCC2c2cccc(F)c2)=O)C1)SC 32218,C1(NC(C2CCN(C)C(=O)C2)=O)CN(C(c2cc(O)nc(O)n2)=O)C2(CCC2)C1 32219,c1(OC)cc(C(=O)NCC(=O)NCC2CNC(=O)CO2)cc(Cl)c1 32220,c1(NC(C2(C)N(C(c3n(CC)ncc3)=O)CC2)=O)cc(F)cc2[nH]ccc12 32221,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)COC(F)F 32222,c1(C(N(C)CC2CCCN(C(CCCSCC)=O)C2)=O)cc(C)ccc1Br 32223,c1(NC(C(=O)NC2(C3CC3(Cl)Cl)CC2)=O)cccc(OCC(F)(F)F)c1 32224,CC(C)C(C)CNC(=O)C=CCN(C(CC(=O)NC1CC1)=O)C 32225,N1(CCC(=O)NC2CN(C(C3(SC)CC3)=O)CC2(C)C)CCCc2ccccc21 32226,c1(N(C(=O)CC2CCCN(C(=O)CC3CCC3)C2)C)cccc(C(F)(F)F)c1F 32227,CC1=C(C)CC(C(N2CCC(C(=O)NC3CNC(=O)C34CC4)C2C(C)C)=O)CC1 32228,NS(=O)(=O)c1ccsc1C(N1CC(O)(CCNC(=O)CC2COCCO2)C1)=O 32229,c1(C(=O)NC2CCC(CCC(=O)NC(C(C(=O)OC)C)C)C2)c[nH]c(=N)c(C)c1 32230,CCC(C)(C)C(C)N(C(c1n[nH]cc1I)C(=O)NCCOCC1CC1)C1CC1 32231,CCC(CC(=O)NCc1ccc(CNC(=O)C(N2CCCCC2=O)C)cc1)SC 32232,C1(CN(C)C(C2(C)CC2)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C1 32233,C(=O)(C(C)(C)CCC)N(CCC)CCC1CC1.C(=O)(COCCCN(C(C)=O)CC)N 32234,N1(C(C2(CSC)CC2)=O)CCC2CCN(C(c3coc(C(C)C)n3)=O)CC2C1 32235,c1(C(N2C(C)CC(CNC(c3ccnn3C)=O)C2)=O)cccc2c1CCO2 32236,Cc1cc(S(N)(=O)=O)cc(C(=O)N(C(C)CNC(=O)CCCCC#N)C)c1C 32237,N1(C(C2CC(O)CN2Cc2cccc3c2OCC3)=O)Cc2cccc(Br)c2C1 32238,Cc1ccc(C(CNC(=O)CN2CCCC(N(C)C)C2)NC(=O)C2CC2)cc1 32239,C(=O)(N=c1[nH]sc2c(Br)cccc12)NC(C(OC)OC)C(C)C 32240,CCC(F)(F)CC(=O)N1CCCC(CCNC(c2c(F)cncc2Cl)=O)CC1 32241,c1(-c2[nH]c(=N)sc2)ccc(C(=O)NC2CC(CNC(C3CCOC3=O)=O)C2)cc1 32242,c1(C(N(c2c(F)cnc(C)n2)C2CC3(CNC3)C2)=O)cc(F)ccc1[N+](=O)[O-] 32243,CCN=c1ccc(C(=O)NC2CCCC2NC(c2ccc(C(N)=O)cn2)=O)c[nH]1 32244,N1(C(C2(OC)CCN(C(c3cc(OC)c(C)nc3)=O)C2)=O)CCCC(F)(F)CC1 32245,C(C(CC(F)(F)F)NC(c1cnncc1)=O)NC(C(CC)n1cncn1)=O 32246,C1(C(N2CC(CCNC(Cc3ccn(C(C)C)n3)=O)C2)=O)CC2CC1C1CC21 32247,C(=O)(C#CC1(C)COC1)N1CCCC(CCC)(NC(c2ccn(CCC)n2)=O)C1 32248,C=CCC(CC)C(=O)N(CC(O)CN(C(=O)CC1CN(C)C1)C)C 32249,N1(C(CC2C(C)(C)C(O)C2)=O)CCC2(CCN(C(c3cnc(CO)cn3)=O)CC2)C1 32250,c1(C(=O)NCC(CNC(c2csnn2)=O)CO)ccc(-n2cncn2)cn1 32251,N1(C(c2ncn(C)n2)C(=O)NC(C)(C)C)CCC(C(=O)NCC2CCOC2)CC1 32252,N1(C(C2C(C)C2)=O)CCC(CC(C)(C)NC(=O)Cc2nccn2C)CC1 32253,CC1CN(C(=O)CSCC=O)CC1CNC(=O)C(F)(F)c1cncs1.C(C)(C)(C)N 32254,c1(C(=O)OC)cc(C(=O)NC(CNC(=O)COCC(C)C)C2CC2)[nH]n1 32255,c1(C(=O)NCC(C)NC(C2CCN(C)C2)=O)nncc2ccccc12 32256,Cc1nn(CC(=O)NC2CC3CN(C(c4csc(O)n4)=O)CC23)c(C)c1[N+](=O)[O-] 32257,c1(OC)ncnc(C(=O)NCCCOCCNC(C2CCNC2=O)=O)c1F 32258,Cc1ccc2ncc(NC(C3CC(NC(C4CCC(C)CC4)=O)C3)=O)n2c1 32259,C1(NC(c2c(C)c(O)ccc2)=O)COC2(CCN(C(=O)CSC(F)(F)F)C2)C1 32260,CCCC(CC)C(=O)NCC(C)N(C)C(c1c(F)cnn1C(C)C)=O 32261,CCCC(CCC)CC(=O)NC(c1cn(C)nn1)C(N1CCC(O)CC1)=O 32262,C(CCCCCC(=O)NC1(CC2CC2)CC1)NC(c1n(CC)ccc1)=O 32263,c1(SC(C(=O)NC(c2cc(C)c(O)c(C)c2)=O)C)ccnc(S(C)(=O)=O)n1 32264,C1(CCC)(NC(c2cccc(N(C)C)n2)=O)CCCN(C(=O)C(C)C(F)F)C1 32265,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32266,C(C(=O)NC(c1nnn(C(C)(C)C)n1)C)(C(C)C)OC(C)C 32267,c1(C(=O)NCC2CN(C(C(C)c3ccsc3)=O)C2)ccc(Cl)c(F)c1O 32268,C1(C)(C(=O)NCCC(N2CCCCC(C(=O)NC)C2)=O)CN2CCC1CC2 32269,Cc1cnccc1C(C)C(=O)NC1CN(C(=O)CCN2CCC(N(C)C)CC2)C1 32270,c1(CC#C)cccc(C(=O)NC(C)C(C)CCNOC(C2(C(F)(F)F)CC2)=O)c1 32271,N1(C(c2cc(C)no2)=O)CCCC(C(=O)Nc2ccccc2SC(C)(C)C)CC1 32272,c1(CNC(CCOCCOCC)=O)csc(Cl)c1.C12(CC1)C(=O)N2 32273,C1(CC(=O)NCC2CCN(C(C(N3CCOCC3=O)C)=O)C2)CCOCC1(C)C 32274,C1(O)(CCNC(=O)CN2CC3CC3C2)CCN(C(C2(NC(C)=O)CCC2)=O)C1 32275,C(=O)(C(C)(C)C(=O)NCC1CN(C(=O)CCCCc2ccccc2)C2CC12)NC 32276,c1(C(C)N)nncn1C(C)C.C1(OC)CC(C(=O)NCC(C)(C)C2CC2)C1 32277,Cc1c(CNC2CC3(c4ccccc4)CC23)cccc1Cl.C12(CC1)C(=O)N2 32278,Cc1cccc2c1CC(C(=O)NCC(CC(C)C)NC(=O)C(O)C1CCC1)N2 32279,c1(CN2CC(C)C2NC(c2cc(C(N)=O)cn2C)=O)ccc([N+](=O)[O-])cn1 32280,c1(C(N2CCN(C(CCC#CCC)=O)CC2CO)=O)cnc2ncccc2c1 32281,c1(C(=O)NCC2(NC(c3c(CC)nc[nH]3)=O)CCC2)ccnc2c1ncn2C 32282,c1(CN2C(C(N3CCOC(CO)C3)=O)CC2)ccc(O)c(Cl)c1 32283,N1(C(C(C)=O)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32284,C1(CNC(=O)Cc2cc(Br)cs2)CN(C(=O)CC2CCC2)CCO1 32285,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)sc2Cl)OC(C)(C)C1 32286,C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1ccsc1Br)=O)CC2 32287,CC1CC(=O)NC1C(N1CCC(CN(c2ccncn2)C)C1)=O 32288,N1(C(C(=O)NCCC)=O)CCCC(CC(=O)Nc2cccc(C(F)F)n2)C1 32289,C(=O)(CCC(=O)N(C(CNC(c1sc(N(C)C)nc1Cl)=O)C1CC1)C)NC 32290,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(F)c[nH]2)=O)CCCCCC1 32291,C1(CNC(c2ccsc2)=O)CCCC2(CN(C(C3CCS3(=O)=O)=O)C2)O1 32292,C1(C(N2CC(N(C(C(CC)=CC)=O)C)C(O)C2)=O)OC2CCCCC2C1C 32293,CC1CC(N(C)c2nnc(-c3cc(CO)on3)n2CC2CC2)c2ccccc2O1 32294,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32295,C1CC(C)(O)CO1.N1(C(C)=O)CCN(CCCCO)CC1 32296,c1(C(=O)NCC23CC2CN(C(=O)C(C2CCCCC2)O)C3)ccn2ccsc12 32297,N1(C(c2cc(C)on2)=O)CCC(NCc2ccccc2Cl)C(C)C1 32298,N1(C(C2C(CCC)CCC2)=O)CCN(C(=O)CCCCCOCC)C(CO)C1 32299,Cc1cnc(N(C)C(c2csc3ccccc23)C)c(S(=O)(=O)NCCCCO)c1 32300,N1(C(CC(C)(C)c2ccc(-c3n(C)c(C(=O)O)cc3)s2)=O)CCC2(CNC(=O)O2)C1 32301,c1(CCC(=O)NCC2N(C(c3cc(C)nn3C)=O)CC=C2)ccccc1[N+](=O)[O-] 32302,C1(NC(C=CC(=O)NC2CC2)=O)CCN(C(=O)CN2CC(=O)NC2=O)C1C1CC1 32303,C1(CC(=O)NC2(CC(=O)NCC3CSCCO3)CC2)CCC(=O)N1 32304,CC(C)=C=CC(=O)NC(C)CC(C)NC(=O)C(=O)Nc1ncc[nH]1 32305,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32306,S(=O)(=O)(c1cncc(Br)c1C)N(C(c1ccc(F)cc1)C(=O)OC)C 32307,C(CCCCCNC(=O)CCOCC(F)(F)F)N(C)C(C1(SC)CC(=O)C1)=O 32308,c1(C(N2CC(CCNC(CS(CC)=O)=O)C(C)C2)=O)ccc(C)cc1C 32309,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32310,CC1CCC(C(=O)N(CCNC(=O)CNC=O)CC2CC2)S1 32311,c1(OC)ccc(S(=O)(=O)N2CC3CCN(Cc4ccc(C)c(F)c4)CC3C2)cn1 32312,C12CCCN(C1)C(=O)OC(C)(C)COC(=O)C2.CC(C)(C)OC=O.C(C)(C)(C)O 32313,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NCCc1ccc(C)cc1 32314,c1(C(=O)NCCCNC(C(C)OCCC=C)=O)ccc(F)c2[nH]ccc12 32315,c1(C(=O)NCC2(O)CN(C(c3ncnc(C)c3C)=O)C2)cc(F)cc(Cl)c1N 32316,CC1CN2CC(C)N(C1)C(=O)C(=O)N(C1CC1)CC2=O.S(C)(=O)(=O)CN.C1CC1 32317,C1(CNC(C(CCC2CCC2)N(C2CCS(=O)(=O)C2)C)=O)CCCN(C)C1=O 32318,c1(C(C)C)ncccc1NC(=O)NC(C)C(F)F 32319,Cc1ccc(C(C)CC(=O)NCCC2CN(C(C3CCCN3C)=O)CCO2)cc1 32320,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C(F)(F)F)=O 32321,C=C=CC(C)C(=O)NC1CC1SCC(F)(F)F.C12(CC(F)(F)C1)C(=O)N2 32322,Nc1cc(C(=O)N(CCCNC(c2nc(C3CC3)cs2)=O)C2CC2)cc(F)c1 32323,c1(OC)cc(C(=O)NC2CCC(NC(=O)CCC3CCC3)CC2)cc(C2CC2)c1 32324,Cc1c(C(=O)NCC23CC(CO2)N(C(C24CC5CC2C4C5)=O)C3)cccc1Cl 32325,c1(COC)nn[nH]c1C(=O)NCCCN(C(c1ccc(SC)s1)=O)C(C)C 32326,N12CCc3cc(ccc31)CC(=O)NC(C1CCCO1)C2=O.c1(CC)csnc1C 32327,c1(C(=O)NCC2(O)CN(C(c3ccc(O)cc3O)=O)C2)ccc([N+](=O)[O-])cc1I 32328,C1(C(C(=O)NCC2(NC(=O)COc3ccsc3)CCC2)F)CCCCCC1 32329,C12(CNC(c3n(CC)ncc3)=O)CC(CO1)N(C(=O)C(C)OCC(C)C)C2 32330,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC(N)=O)C(C)(C)C1 32331,C(CN=C(NCC(c1ccnn1C)(C)C)NCc1ccncc1OC)OC 32332,C(=O)(C(=O)C(C)(C)CC)N(CC(=O)NOCCCC1CC1)CC=C 32333,Cc1cc(C(N2CC(F)CC2C(=O)NCC2CC(=C3CC3)C2)=O)nc(O)n1 32334,C(=O)(C(C(C)(C)C)C1CCC1)N1C(C)(CN(C(CNC(CC)=O)=O)CC)CCC1 32335,C1(C2CCCO2)(C(N2C(CNC(C=C(C)C3CC3)=O)CC2)=O)CCCO1 32336,N1(C(C(CCCC)NC(=O)Cc2cn(C)nc2C)=O)CC2(CCOCC2)C1 32337,C1(C(=O)OC)CC(F)(F)CN1C(C(=O)NC(c1cccs1)C)C1CC1(C)Br 32338,C(=O)(CC1=NNC(=O)C1)N1C(C2(O)CN(C(CCC(C)N(C)C)=O)C2)CCC1 32339,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32340,c1(NC(C(C)O)C2CC2)cccc(S(=O)(=O)N(C)CC2CCN(C)C2)n1 32341,CCC(CC(=O)NC1CCC1NC(c1ccc(C(C)C)o1)=O)C(F)F 32342,c1(C(=O)NC2CC(c3cn(-c4ccn(C)n4)nn3)C2)c(F)cc(F)cc1Cl 32343,c1(C(N2CC3CC(C2)CN(C(=O)C(F)F)C3)=O)cnn2c1OCC1(CC1)C2 32344,N1(C(CS(=O)(=O)NC)=O)CCOCC12COCCN(C(=O)C(C)OC1COC1)C2 32345,C(C(=O)N1CC(N(C)C)C(O)C1)(C(C)(C)C)NC(C(C(C)C)F)=O 32346,c1(OC)ccc(CC(=O)NC2CC(c3ccccc3OC)(F)C2)cc1OC 32347,N1(C(c2cc(C)c(F)cc2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 32348,Cc1ccc2c(c1)C(C(=O)NCCCNC(C1CCC(C(N)=O)C1)=O)C2 32349,c1(OC)ccc2cc(C(N3CC=CC3NC(=O)C=C3CCCCC3)=O)ncc2c1 32350,C1(CNC(C(C)CN(C)C(c2ccc[nH]2)=O)=O)CC12CCOCC2 32351,c1(C(N(C(C2CC(C)(C)C2)C(=O)NC)C)C)c(F)cccc1F 32352,c1(C(=O)NC(CC=C)CNC(=O)Cc2c[nH]nc2C)ccc(Cl)c(OCC)c1F 32353,CCC(C(=O)NCCN(C(=O)C(C)C1CCCC1)CCCN(C)C)C(C)C 32354,Cc1ccc(C(=O)NCCCCCC(=O)NC(c2csnn2)C)c(O)n1 32355,N1(c2cc(CC)ncn2)CCCC(C2CC2NC(c2n[nH]cc2C(F)(F)F)=O)C1 32356,c1(NC(C2(CNCc3ccc(O)cc3O)CC2)=O)cc(Br)cc2[nH]ncc12 32357,c1(C(C)(C)OC)ccc(F)cc1.C12CCC(C1)C(=O)NC2.C1(=O)C(CN(C)C)N1 32358,C(=O)(CCC(=O)NC(C(=O)NCC(CC)SC)C1CCOC1)NC 32359,C1(C(=O)NCC(C)(C)NC(c2ccc(CC(C)C)s2)=O)Cc2cccnc2C1 32360,Cc1cc(C(=O)NCC2CN(C(=O)C(CO)NC(N)=O)C2)nc(C)c1 32361,C1(NC(c2c(Br)cc(C)s2)=O)CC2CCC1N2C(=O)CCC1(C)CC1 32362,C1(NCc2ccc(C(=O)OC)nc2)CCCN(S(=O)(=O)NC)C1 32363,c1(N(C(c2cc(C(=O)OC)sc2)=O)CCNC(C)=O)cccc(Br)c1[N+](=O)[O-] 32364,N1(CC#CC)CCC(C)=C(F)C1.c1(C2C(=O)N2)ccnn1C 32365,C1(CNC(C(C)c2cccs2)=O)CC(C)(C)CN1C(c1ccoc1)=O 32366,Cn1ncc2nc(Cl)nc(NCC34CCC3CN(C(=O)CC3CC5CC5C3)C4)c12 32367,C1(C(N(CCC(=O)NC2(C)CCC(C)C2)CC=C)=O)CC12CCCCC2 32368,C1(C)(NC(C2(C)CC2C(F)(F)F)=O)CCN(c2nc(-c3ccccn3)ns2)C1 32369,c1(N2CCN(C(C(=O)N(CC#C)CC=C)C)CC2)ncnc2scc(C)c12 32370,c1(C2CC(C(=O)NC(C(C)C)CNC(C3CCCSC3)=O)C2)ccccc1F 32371,c1(NCc2c(F)cc(C)cc2F)cccc2c1CNC(=O)C2 32372,C(=O)(CC(Cl)Cl)N(C(CN(C(C1(C(=O)NC)CC1)=O)C)C)C 32373,O=S(=O)(C=Cc1ccc(Cl)cc1Cl)N1CCC(CO)CC1 32374,c1(C(N2CC(C(N)=O)(CNC(C(CC#C)O)=O)C2)=O)ccc(F)c(O)c1F 32375,CCCCCCC(CC)C(=O)N1CC(CNC(c2cccc3c2ncn3C)=O)C1 32376,c1(OC)ncc(CNC2CCC(C(=O)NCCc3nccs3)C2)cc1Cl 32377,N1(C(C2C(=C)C2C(=O)OCC)=O)C(C(=O)NCCSC)CCC12CC2 32378,Cc1nc2ccc(C(=O)N(C3CC(NC(c4ccc(N)c(Cl)c4)=O)C3)C)cc2o1 32379,c1(N(C2CCSC2)C)nc2cc(Cl)c(C(=O)O)cc2s1 32380,n1(CC)ccc(C(=O)N(C)CC2(CNC(=O)C=CBr)CC2)n1 32381,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32382,C1(O)(CCNC(c2ccc(OCC3CC3)nc2)=O)CCN(C(=O)C=CC2CC2)CC1 32383,C1(CNCC(Br)=C(C)C)CNCCC1c1nccn1C 32384,N1(Cc2c(OCC)cccc2)CC2CN(C(C3CC4CCC3O4)=O)CC12 32385,C1(C(=O)OCC)C2CN(C(C(=O)CCc3ccc(F)cc3)=O)CC12.C1(C(=O)O)CN1 32386,n1(C)cc(NC(=O)CS)nn1.c1(NCC(CNC(C2(C)COC2)=O)F)ccccc1 32387,CCC(F)(F)CC(=O)N1CCC(CNC(C23CC(c4ccccc4)C2C3)=O)CC1 32388,N1(C(C(=Cc2ccncc2)C)=O)CCN(C(c2ncccc2F)=O)CC(C)C1 32389,c1(-c2onc(COC)n2)cccc(CNC(=O)CC2(C(=O)O)CCCC2)c1 32390,N#Cc1cccc(Cl)c1NC(C1CC(NC(c2ccc(OCCO)cc2)=O)C1)=O 32391,Cc1cnn(C)c1C(N1CC(O)(CCNC(=O)CCn2cccnc2=O)C1)=O 32392,Cc1cnc(C=CC(=O)NCCC2CCCCN2C(C2C3COCC23)=O)[nH]1 32393,C=C(Cl)CCC(=O)NCCC1CCCN(C(C2CC3CCC2C3)=O)C1 32394,C1(C)(C(N(C)CC2N(C(CCC(C)C#N)=O)CCCC2)=O)CCCCNC1=O 32395,c1(SC)ccc(C(=O)NCC2CC(C(N3CC(O)(CO)C3)=O)C2)cc1.C(C)=O 32396,c1(C(N2CCN(C(C3(c4cnccn4)CC3)=O)C3CC23)=O)ccc(F)c(Br)c1 32397,C(=O)(C1=CC(C)(C)C1)NC(CCN(C(c1c(OC)nsc1)=O)C)C 32398,C1(NC(C(SC)SC)=O)CCN(C(=O)C2=CCC2)CC1C 32399,c1(C(=O)NC(C)CCCCNC(=O)Cc2cn[nH]c2)cnc2ncnn2c1O 32400,C=CC(CC)CC(=O)NCc1cccc(-n2cc(CN3CCCCC(C)C3)nn2)c1 32401,c1(CC)nn(C)c(CC)c1NC(=O)C(F)(F)C1CCC(C(=O)OCC)C1 32402,c1(NCCC(N2CCCC(CO)C2)=O)ccc[n+]([O-])c1 32403,N1(C(c2c(OC)cc(C)cn2)=O)CCN(C(=O)Cc2cnns2)C(C)C1C 32404,C1(C2=CCCCCC2)(C(=O)NCCCN(C(c2c(C)onc2C2CC2)=O)C)CC1 32405,C1(NC(CCN(CC=C)C(C2CSC2)=O)=O)CCCC(O)C1 32406,c1(C(=O)NC(C2CCCN(C(c3csc(O)n3)=O)C2)C)cc(C#N)c(O)nc1N 32407,N1(C(c2cc(C)sc2C)=O)CCC12CN(C(c1cncs1)=O)C2 32408,N1(C(C(C)=C2CCC2)=O)CCN(C(C2C(F)(F)C23CCC3)=O)CC1CF 32409,N1(C(C(C(=O)OCC)SC)=O)CCC(O)(CN(C)C(C2CCN(C)C2)=O)CC1 32410,c1(CNC(C(c2ncn(C(C)C)n2)OCC)=O)cccc(C)n1 32411,C1(C(N2C(CC(N)=O)CCC2)=O)CCCCCN1C(c1c(F)cccc1F)=O 32412,c1(OC)cc(C(N2CCCCC2CCO)C(=O)NCCC2CC2)ccc1OC 32413,c1(CC(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)=O)cnc2ccccc2c1 32414,C1(C)(Nc2cccn(C3CN(C(COC)=O)C3)c2=O)CCC(C)(C)CC1 32415,C=CCCCCCCC(=O)NCC1CC1CC(=O)NC1CC(C)(CC)C1 32416,N1(C(c2ccc(O)c(F)c2)=O)CC2C1CN(C(c1cc[nH]c1)=O)C2 32417,C1(NC(CSCC#N)=O)(CNC(=O)C(C2CCOCC2)F)CC2CCC1CC2 32418,C1(OCC)CC2(C1)CC2NCCCC(c1ccccc1)NC(=O)CC#N 32419,C12(CN(C(C3(CCC)CCC3)=O)CC)CCC1CN(C(=O)C1=CCCC1C)C2 32420,c1(OC)ccc(C(O)C(N2CCC(F)(NC(=O)CCN3CCOCC3)C2)=O)cc1 32421,c1(C(N2CCC(N(C(=O)Cc3ccoc3C)CC)C2)=O)occ(C)c1CC 32422,C(=O)(CC(C)C1CC1)NCC(CC)NC(=O)C(c1ccncc1)C 32423,N1(C(CCC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3)=O)CCCC2(F)C1 32424,c1(OC)cc(OC)c(C(N2CCCC2CNC(=O)CC2(CO)CC2)=O)c(N)c1 32425,Cc1cc(Br)c2ncnc(N3CCCC(c4n[nH]c(C)n4)C3)c2c1 32426,Cn1cc(Cl)c(C(N2CC=CCC2C(=O)NCCC(O)C(F)F)=O)n1 32427,c1(C(=O)OCC)cc(CN(C)Cc2cccc(SC)c2)c(C)s1 32428,N1(C(c2cc(C(C)C)no2)=O)CCN(C(c2cn(CCCC#N)nn2)=O)CC1C 32429,n1(CC)nnc2c1CCC(C(N1CCC(CNC(c3c[nH][nH]c3=N)=O)C1)=O)C2 32430,C1(CC(=O)NCC(Cc2cnc[nH]2)CO)CC=CCC1.C1(N2C(=O)C2C2CC2)CCCC1 32431,CC1CC(NC(c2ccc(Cl)nc2O)=O)CN(C(c2cc(Cl)nc(Cl)c2)=O)C1 32432,N1(C(COCCC)=O)CCC(NC(c2ccc(F)cc2SC)=O)C(CO)C1 32433,C(=O)(C(F)(F)CCn1ccnn1)NC(CC(C)NC(=O)CC1CC(O)C1(C)C)C 32434,C1(N(C(=O)C(C)(C)NC(=O)C=Cc2nccs2)C)CCC(C)(C)CC1 32435,C1(CNC(c2ccc(C#C)cc2)=O)CN(C(=O)C(C)C)C2(CCC2)C1.CC 32436,Cc1cccc(-c2cc(C(=O)N(C(C)CNC(C3(C(C)(F)F)CC3)=O)C)on2)c1 32437,C12(CNC(c3ccsc3Cl)=O)CC(CN1C(=O)COCC1CCCC1)C2 32438,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(CC3CC3)C2)=O)c1Cl 32439,C1(N2CCOCC2)(C(N(CCN(CC)CC)CCO)=O)CCCC1 32440,C(C)(CO)(C(=O)N1CCOCC1)N(CC(=O)NCCCS(=O)(=O)O)C 32441,C1(CNC(=O)C=Cc2ccoc2)CC2CCC1N2C(=O)CCc1cccc(F)c1 32442,c1(C(N2CC3C(NC(=O)CCn4cccn4)C3C2)=O)cnc2ncccn12 32443,N1(C(CCCN(C(C)C)C)=O)CCN(C(=O)CCN(C)C)CC(CO)C1 32444,Cc1ncnc(O)c1C(=O)NCC1(O)CC(CNC(c2cccnc2Br)=O)C1 32445,C1(C(=O)NCCC(C)NC(C2(CCF)CC2)=O)OCC2COCCC12 32446,C1(CCC(N)=O)C(=O)N2CC(C#N)(C2)c2cn1nn2.CC1CCC(CC2CC2)O1 32447,Cc1c(C(=O)NCCn2ncc(NC(C3(C(C)C)CC3)=O)c2C)cncc1Br 32448,N1(C(C2CCN(N(C)C)CC2)=O)CCC2(COCCN2C(=O)C(F)Br)C1 32449,C1(CNC(=O)COC2CCOC2)CC(C(=O)NCC2CCCC2N)CO1 32450,c1(SC)cscc1C(=O)NCCCC(C)NC(=O)C(C)NC(C1CCCC1)=O 32451,Cn1cc(CCC(=O)NCC=CCNC(c2ncsc2Br)=O)nn1 32452,CCC(C)N(OC)C(=O)C1CCC1CNC(=O)C=Cc1cocn1 32453,N1(C(C(CCF)NC(=O)CC2CCCSC2)=O)CCOC2(CCC2)C1 32454,N1(C(C2N(C(=O)CCC3CCC3)CCCC2)=O)CC(C2CC2(F)F)C1 32455,c1(C(=O)NCCC2CN(C(=O)Cc3cncs3)C2)cnccc1SC1CCCC1 32456,c1(C(=O)NC2CCC(CNC(c3c(CC)occ3C)=O)C2)cc2cccn2cn1 32457,N1(C(C(C)NC(C)=O)=O)CC(CCNC(=O)Cc2cncn2C2CC2)C(C)C1 32458,c1(C(=O)NC23CCC(NC(C4C(C)C4)=O)(CC2)C3)noc2c1CCc1sccc1-2 32459,C(CC(C)C)(C(=O)NC(c1ccccc1)NC(=O)C(c1ccncc1)OC)OC 32460,C(=O)(CCC(C)N(C)C)N(CCCNC(CC(=O)NCC#C)=O)C(C)C 32461,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3n(CC#C)ccc3)=O)CC21 32462,c1(C(=O)OC)cn(C)nc1C(N1CC(O)CC1CNC(=O)C(C)(C)N(C)C)=O 32463,c1(CC(=O)NCC2(C(C)(C)O)CN(C(C(F)OC)=O)C2)ccc(F)c(F)c1 32464,C1(CCNC(C2N(CCC)CCC2)=O)CSCCN1C(=O)Cn1cc(C)cn1 32465,C(C(CNC(c1nc(C)oc1C)=O)S(C)(=O)=O)NC(C1CC(CCC)C1)=O 32466,c1(NCCC(C)(C)NC(c2c(CC)scn2)=O)cc(C(F)F)ncn1 32467,C1(CCNC(CN(C(C(C)n2cncn2)=O)C2CC2)=O)CC(C)(C)C1 32468,N1(CC2C(C)(C)C2)CCOC2(CCCN(C(S(=O)(=O)CC#N)=O)C2)C1 32469,CC(O)C(C)(C)C(=O)N1CCC(N(CCO)C(c2cnn(C)c2C(F)(F)F)=O)C1 32470,C1(CC(=O)N(CC2(CCNC(CC)=O)CC2)C2CC2)CC2(CCC2)CO1 32471,N1(C(CCC2CCC(OC)CC2)=O)CC(C2CN(C(=O)C(C)(CO)OC)C2)C1 32472,N1(C(C)=O)CCCC12CCN(C(=O)CC(C)C(C)(C)NC(=O)C(C)(C)CCl)C2 32473,N1(C(C(C(C)C)N(C)C)=O)CC2(CC(CNC(=O)C(c3cnn(C)c3)OC)C2)C1 32474,c1(C(=O)NCCCC(C)NC(C2CC(CF)C2)=O)cccc(N)c1F 32475,N1(C(C(C)n2cncn2)=O)CCN(C(C2CC(O)C2)=O)CC1c1cnn(C)c1 32476,C=CCC(C(=O)NCC1CCCO1)NC(=O)CC1OCCO1 32477,c1(CC)c(C(=O)NC2(CO)CN(C(=O)C3=CCCCC3)C2)sc2ccccc12 32478,CC(C(C)C(=O)N(C1CCC1)CCO)NC(c1cc[nH]c1C1CC1)=O 32479,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CC4COCC4C3)=O)C2)=O)n1 32480,Cc1cc(C(=O)NCC(C)NC(C2(C#N)CC=CC2)=O)cnc1C(F)(F)F 32481,c1(C(N2CCC3(CN(C(COCCC)=O)C3)C2)=O)cc2n(n1)CCCC2O 32482,c1(C(=O)NCC2CCN(Cc3c[nH]c4cccnc34)C2)ccc2c[nH]nc2c1 32483,c1(C(N2CC(C=C)C(NC(C3(OC)CC4CCC3C4)=O)C2)=O)cccc2[nH]ccc12 32484,c1(OC)nccc(CC(N2CC(N3CCOCC3)C(C)C2)=O)n1 32485,CC1CCC(C)(C)N1C(C1(C)CCN(C(C2CCC(CO)CC2)=O)CC1)=O 32486,c12ccc(cc1)s2.C(=O)(CCC(C)C)NC(CNC(c1c(CC)c[nH]n1)=O)(C)C 32487,CC1CCN(C(=O)Cc2csnn2)C(C)C1NC(C1(CN(C)C)CC1)=O 32488,c1(C(=O)NCC23CN(C(c4cc(C)on4)=O)C(CC2)C3)nc2cc(F)ccc2s1 32489,C1(C(C(C)NC(=O)N(C)C(c2ccccn2)C)(C)C)Cc2ccccc2O1 32490,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32491,c1(C(=O)OCC)ccnc2c1OCO2.c12cc(C)nc(n1)NC2CC#C 32492,c1(C(C)C(=O)NCC=CCNC(C2CC(F)C2)=O)ccccc1-c1ccccc1 32493,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)C2CCC2)c(C)nn(C(C)C)c1C 32494,c1(CN(C(CCC)=O)C)cnn2c1CN(C(=O)C=CCF)CC2 32495,CC1CCC2CN1C(=O)CC1(CC1)NC2=O.c1(C(=O)N(C)C)cccnc1O 32496,CC(CN=c1[nH]c(=NCC2CC23CCC(O)CC3)[nH]c2c1CCCCC2)C1CC1 32497,C1(OC)CCC(C(N2CC3CC3(NC(=O)C=C(C)C(F)F)C2)=O)CC1 32498,C1(CNC(=O)CCN2CCC2)CCC2(CO1)CC(NC(C13CCCN1CCC3)=O)C2 32499,C1(CNC(C(n2cc(CC(O)CO)nn2)C)=O)CCC(CO)CC1 32500,N1(C(c2nc(C(C)C)sc2)=O)CCCC1(C)CNC(=O)CSCc1ccnn1C 32501,CC1(C)CC(C(N2CCN(C(c3ccc(F)c(F)c3)=O)C(CF)C2)=O)C(C)(C)O1 32502,C12CCCC(C1)C(=O)NC2.C1(C(CC)C)CN(C(=O)C(C)(C)F)C1 32503,C1(CCCNC(CC2N(C(COCC)=O)CCC2)=O)CCN(C(=O)CC2CC2)CC1 32504,c1(C(=O)NCC2=CCN(C(c3c(N)c(Cl)ncc3)=O)CC2)cccc2sccc12 32505,c1(C(=O)NC2(CNC(C(SC)SC)=O)CC3CCC2C3)ccc2cnc(C)n2c1 32506,CCCCC(O)CC(=O)NC(C)(C)C=CC(N1CCCC(C)C1)=O 32507,N1(C(c2cc(CC(=O)OC)on2)=O)CCCN(C(c2ccc(C(N)=O)s2)=O)CC1 32508,C1(NC(CC(COC)C)=O)CC2CC1CN(C(=O)Cc1c(C)noc1C)C2 32509,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(C(c1cn(C)nc1)O)=O)O 32510,N1(C(C2CC(N(C)C)C2)=O)CCc2nc(C(=O)NC(C)(C)C3CC3)cn2CC1 32511,C=C(C)C1OCCC1CNC(=O)C(C1CCCCC1)NC(C1C=CC1C(=O)OC)=O 32512,N1(C(c2cnc(C(F)F)nc2)C(=O)NCCC#N)CCCC(n2ccnn2)CC1 32513,CC(CCCc1ccccc1)C(=O)N1CCC(N(C(=O)C2=C(Cl)CC2)C)CC1 32514,c1(OC)cc(C(N2C3CCC2C(NC(=O)C(C)C(C)C)C3)=O)c(Cl)cc1Cl 32515,Cc1ccc(F)cc1C(N1CCC1CNC(C1(F)CCCN(C)C1)=O)=O 32516,C(=O)(C1=NOC(CNC(=O)CCOC2CCC2)C1)N(CC(O)C1CCC1)C 32517,Cc1cc(NC(N)=O)ccc1NC(=O)CCC(C)N(C)C(C12CC(C)(C1)OC2C)=O 32518,C1(C2=CCNCC2)(C(=O)NCC2C(C)(C)C2N)CC1 32519,C(=O)(C(CCF)NC(=O)C(c1cnn(C)c1)=O)NCc1ncc(C)[nH]1 32520,c1(OC)c[nH]nc1C(C(=O)Nc1nc(C(=O)OC)cs1)N(C)CC1CCCCC1 32521,Cc1cc(-c2ccc(C(=O)Nc3ncc(Br)c(O)n3)nn2)c(C)cc1O 32522,c1(CC)nc(C)c(C(=O)NC2(CNC(=O)C=CS(C)=O)CCOC2)o1 32523,C12(CCC(=O)N1)CNC(=O)CC2.CC(C(=O)NCCN(C)C)OCC1CCC1 32524,c1(NC(C2CN(C(CN(C(C)=O)C)=O)CC2(C)C)=O)nc(C)c2c(n1)CCCC2 32525,c1(OC)ccc(CCCc2ccccc2)c(O)c1.C12CCCCC1C(=O)N2 32526,N1(C(C2N(CC)CCCC2)=O)CC(NC(c2cc(C)ncn2)=O)C(C)(C)C1 32527,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32528,N1(C(c2cnn(C(C)C)c2F)=O)CCC2(CCCC2CNC(=O)CC(C)C)CC1 32529,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32530,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32531,c1(CN2CCC(c3cccc(OC(F)F)c3)CC2)cn2ccsc2n1 32532,C(CCCS(=O)(=O)CCOC)N1CCN(CC)CC1.N1(CCC)CCC(C(=O)OC)CC1 32533,C(CC(O)CO)N(C(=O)CC1(NC(C2(C)CCCO2)=O)CCC1)C 32534,c1(CC)conc1CC(=O)NCC(C)NC(c1sncc1C)=O 32535,C1(NC(c2cc(C3CC3)no2)=O)CCCCCN(C(c2cc(F)c(Cl)cc2F)=O)C1 32536,C=CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C(C)(C)C)N(C)C)CCC1C 32537,c1(C(N2CC(CNC(c3ccc(C)s3)=O)C3C2C3)=O)cc(F)c(C#N)c(F)c1 32538,CC1CN(C(=O)CN(S(C)(=O)=O)C)C(C)CN1C(=O)CC1COCC1(C)C 32539,c1(CN(C)C(C2CC(CNC(=O)Nc3ccco3)C2)=O)cnc[nH]1 32540,C(CCCCCC(=O)N(CC(O)CO)CCO)NC(c1c(Cl)cn(CC)n1)=O 32541,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)CO)C2)C)ncnc(O)c1F 32542,CC(CO)(C1CCC1)NC(C1CCC1NC(=O)COC(F)F)=O 32543,C1(C(C)C(=O)NCC(C2CCC2)C2CC2)CCN(C(=O)COC2CCCOC2)C1 32544,N1(C(c2nc(CC)sc2N)=O)CC(CNC(=O)CSc2nncn2C)C2(CC2)C1 32545,C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C)CCN(C)C(c1csnn1)=O 32546,C1(C(N(CC(C)C(=O)NCC(O)(C2CC2)C2CC2)C)=O)CCCC(O)C1 32547,N1(C(c2n(C)cnc2)=O)CCN(C(c2nccnc2N)=O)C2CCCCC12 32548,C=C(Br)CC(C)(C)C(=O)NC(c1cccc(C)n1)c1cn(CCSC)nn1 32549,c1(N2CCN(Cc3cnn(C)c3Cl)CC2)cc(Cl)cc(C(F)(F)F)n1.C1(=O)NN1 32550,N1(C(c2c(C)nns2)=O)CC2OCCN(C(c3cc4c(ccn4C)s3)=O)C2C1 32551,C1(N(C(C(C)NC(N)=O)=O)Cc2ccn(C)n2)CC2CCC(C1)N2 32552,C1(NC(C2CCC(OC)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32553,n1(C(C)C)ccnc1C(=O)NC(C)(C)CC=CC(=O)NC1(c2cccnc2)CC1 32554,S(=O)(=O)(c1cc(C)c(-c2ccccn2)cc1C)NCCOC 32555,CC1=C(CNC(=O)CC2C=CC(NC(=O)C(c3ccccc3)O)C2)COCC1 32556,c1(C(N2CC3CC(NC(C=CC)=O)C3C2)=O)ccc2cc(Cl)ccc2n1 32557,c1(C(=O)NC2CCCC(N(C(=O)C3=CCCOC3)C)C2)cccc2nccn12 32558,Cc1nnc(CCC(=O)NC2(CCNC(c3ccc(Cl)cc3)=O)CCC2)n1C 32559,C(=O)(CCC(C)(C)NC(c1cccc(F)c1N)=O)N(CC(CO)C1CC1)C 32560,N1(C(c2scc(CC)n2)=O)CCC(C#N)(NC(c2cc(F)ccn2)=O)C1 32561,C(CCO)(C(F)(F)F)NC(c1c(CCNC(Cc2nc(C)[nH]n2)=O)n[nH]c1)=O 32562,CCC(O)C(F)(F)C(=O)N(C)CC1CN(C(=O)C(C)CCCc2ccccc2)C1 32563,c1(NC2CN(C(C(C3CCOC3)OC)=O)CC2(C)C)ncc2c(n1)CCOC2 32564,N1(C(C(CC)C)=O)CCC2C(NC(c3c(C)nn(C)c3-n3cncn3)=O)CC12 32565,Cc1cc(Cl)ccc1CC(N1CC(n2cc(CN(C)C(C)C)nn2)C2(CC2)C1)=O 32566,c1(OCC)ccc(C)cc1C(N1CCC(O)(CNC(c2oncc2C)=O)C1)=O 32567,c1(C(=O)NCCCNC(c2c(C)ccc(OC)n2)=O)nccc2c1NCCC2 32568,c1(C(=O)NC(C2CCN(C(C3CCN(OC)CC3)=O)C2)C)ncc([N+](=O)[O-])cn1 32569,CC(C)C(C)(O)C(=O)N(CC(C)NC(=O)COc1cccnc1Br)C 32570,c1(C(=O)Nc2ccnc(F)c2)ccnc2ccnn12 32571,c1(C(C)C)nc(NC(=O)NC(C)C(N)=O)cc(N2CCN(CCCO)CC2)n1 32572,N1(CC(=O)NC(CCCNC(C2CCCC(OC)C2)=O)C)C(=O)CCCC1=O 32573,c1(CCC(=O)NCC(C)N(C)C(N)=O)ccccc1NC(=O)CCC(F)F 32574,C1(C(=O)NC(CNC(c2c(C)cc(CC)o2)=O)(C)C(C)C)CCCCCN1C 32575,CC1OCCCC1C(=O)NCCN1CCN(C(=O)CC2OCCO2)CC1 32576,Cc1cc(=NC2CN(S(C)(=O)=O)C2)[nH]c(N2CCc3cnn(C(C)C)c3C2)n1 32577,CCC(CC)CCCNC(=O)C(O)CNC(=O)C=Cc1cc[nH]n1 32578,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)O1)OC 32579,N1(C(c2c(CC)noc2)=O)CCC2(CCCCN(C(C3CCOC(C)C3)=O)C2)C1 32580,Cc1cc(N)cnc1C(=O)NCC(C)NC(c1cnsc1C)=O 32581,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(C2CC(C)(C)C2)=O)C1 32582,C(C)(C)(CCC(=O)NCC(C(C)C)NC(=O)CCCN1CCCC1)SC 32583,C1(CNC(C(C)OCC=C)=O)CCN(C(C2CCC2c2cccc(Cl)c2)=O)CC1 32584,C1(NC(c2cnn(C(C)C)n2)=O)CCC(C)(CNC(C2CC(=O)N2)=O)C1 32585,C12(CCNC(=O)C=Cc3cnc[nH]3)CCC1CN(C(c1cc3sccc3[nH]1)=O)C2 32586,N1(C(c2cnc(CC)s2)=O)CCC2CN(CCNC(C)=O)CC2CC1 32587,C(CCC(C(=O)N1CCN(CCF)CC1)NC(=O)CC(C)C1CC1)OC 32588,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32589,C1(C(=O)NCC(C(C)C)NC(C2CCN(C)C2=O)=O)CC(=O)OC1(C)C 32590,C1(C(=O)NCC2N(C(c3c(CC)c[nH]n3)=O)CC=C2)CSc2ccccc2O1 32591,n1(CCCN(C)C)cc(C(C)=O)nn1.CCCC1C2(CC2)CN1 32592,N1(C(c2c(C#C)cnn2C)=O)CCC2(CCC2)C(NC(c2ccccc2F)=O)C1 32593,C1(N(C)C)C(C(=O)NCC23CC4CC(CC(C4)O2)C3)C2CCC1(C)C2(C)C 32594,CCCC(CNC(=O)CC1CC(C)=NO1)NC(=O)C=C(C)C(C)C 32595,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)Cc2n[nH]c(C)n2)C2(CCCC2)C1 32596,C1(NC(CNS(NC)(=O)=O)=O)CC2CCC1C(NC(c1ccnc(CO)c1)=O)C2 32597,c1(C(=O)NCC(C)O)ccc2c(c1)CCN(Cc1ccc(F)nc1F)C2 32598,c1(C(N(C(C)C)CCN(C(=O)CN2CCOCC2)C)=O)ccc(O)cn1 32599,CCCCC(C(=O)NC1CCC12CCCC2)Nc1sc(C)nc1C.c12cn(nn1)C2 32600,C1(C)(C(N(CCNC(C(c2c[nH]nc2CC2CC2)C)=O)C)=O)CCCS1 32601,c1(CC)oc(C)cc1C(=O)N(CCCC(=O)NCCC(F)F)C 32602,c1(C(=O)NC2CCCN(C(=O)C(O)CC(F)F)CC2)cc2nc(F)ccc2o1 32603,Cc1sc(=O)n(CC(N2CC(O)(CNC(C3CCC(C)CC3)=O)C2)=O)c1C 32604,N1(C(=O)CCCC2CC2)CCC2CCN(C(c3cnc(C4CCC4)o3)=O)C2C1 32605,c1(C(=O)NCc2cccc(CNC(c3c(C)ccn3C)=O)c2)ccc(F)c(O)c1 32606,C(C1c2ccccc2CCN1C(=O)CC1(O)CCC1)NC(=O)CC(F)(F)Br 32607,N1(C(c2cc(C)nn2C)=O)CC2CCN(C(C3CCCCCCC3)=O)CC2C1 32608,CC1(C)CCOC1CCCNC1COCCC1CNC(=O)OC(C)(C)C 32609,c1(C(=O)NC(C)CN(C(=O)CCCC2CC2)C)cc2c(O)ncnc2cn1 32610,Cc1cc(NC(=O)CC2C(NC(C3C(C)(C)C3(F)F)=O)CC2O)cc(CO)c1 32611,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(c2cc(SC)oc2C)=O)CC(O)C1 32612,N1(C(c2cc3occc3s2)=O)CC2(CCN(C(C3CCOC3)=O)CC2)C1 32613,N1(C(C(C2CCC2)OC)=O)C2CCC1CC(CNC(c1cnn(C(C)C)c1)=O)C2 32614,C(=O)(C(C(C)(C)C)N(C)C)N(c1cccc(C(F)(F)F)c1)C.N12CCCC(C1)C2=O 32615,C(=O)(CC(C(C)C)NC(C1(CC(C)C)CC1)=O)NCCc1c(C)ocn1 32616,C=CC(CC)CC(=O)N1CCC(C)C(NC(=O)C=Cc2cnc(OC)cn2)C1 32617,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(=O)C(C4CC4)N(C)C)C1C3C2 32618,C1(C(=O)NC2CC(CNC(=O)C=C3CCCC3)C2)CC12CCCc1ccccc12 32619,C1(NC(C2CC(NC(N)=O)C2)=O)CC(NC(C2(CCC)CCCC2)=O)C12CCC2 32620,C(=O)(CC(O)CCSC)NC1CCN(C(c2ccc(CC)nc2)=O)C1 32621,C12(NC(C(CO)NC(c3nc(CC)oc3)=O)=O)CCCN(CC1)C2 32622,c1(CNC(C2CCCCO2)=O)cccc(Cn2cc(CNC3CCOC3)nn2)c1 32623,c1(C(=O)NC(CC)CNC(=O)Cc2nn(C)cc2Cl)c(SC)cccc1F 32624,c1(-c2n(C)ncc2)cccc(C(C)(C)C(=O)NC2CC(NC(=O)C3CC3)CC2O)c1 32625,CC1(NC(c2csc(-c3ccsc3)n2)=O)CN(C(C2CCC2)=O)C1 32626,N12CCC(CC1)N(C)S(=O)(=O)C1(CC1)C2.C1(N)(CC)CCCCC1 32627,c1(C(N2C(C(=O)NCC3COCCO3)CCC2)=O)cc([N+](=O)[O-])cs1 32628,c1(OC(C(c2ccc(Br)cc2)NCC2(OC)CCCSC2)=O)c(C)cccc1Cl 32629,C1(C)(C(=O)NCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32630,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32631,O=S(=O)(c1cccnc1NCC1CC2(C1)OCCO2)N1CCCC1CF 32632,c1(C(N2CC(C)N(C(c3ccc(N(C)C)nc3)=O)CC2)=O)ccn2ccnc2n1 32633,Cc1onc(-c2cccc(Cl)c2)c1C(=O)N(C)CCNC(c1coc(Cl)n1)=O 32634,c1(C(N(c2c(C)n(C)nc2)C)=O)cnc2[nH]c(Cl)c(Br)cc1-2 32635,c1(CN(CC(=O)NCCCN(C)C)CCOC)cc(Cl)ccn1 32636,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32637,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)N1C(C)CN(CC)C(C)C1 32638,c1(C(C(=O)NC)N(CC)Cc2cccc3ccsc23)ccc2c(c1)CCOC2 32639,c1(C(N(CC(CNC(CCCc2cc(C)no2)=O)O)C)=O)cc(F)c(O)c(Cl)c1 32640,N1(C(CCC(=O)NC)=O)CCCC(C2CC2NC(=O)Cn2nccn2)C1 32641,c1(C(=O)NCCC2CN(C(C(C)(C)OC(C)=O)=O)CC2C)cccc2c1CCC2 32642,N1(C(C23C(C)(C)C(CC2)CC3)=O)CCCC(C2(NC(=O)C=CSC3CC3)CC2)C1 32643,c1(C(N2CC(OCCNC(C3C(C)(C)OCC3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 32644,c1(C(=O)NCCCCCN(C(C(COC)N(C)C)=O)C)ccc2c(c1)C(C)CO2 32645,C1(C=O)CC2(C1)CC2F.C1(C(=O)NC)CCC(n2cc(CN)nn2)C1 32646,C1(CNC(=O)Cc2cocn2)C(C2CC2)CCN1C(=O)C(c1ccc(O)cc1)=O 32647,c1(NC(C2N(C(CCC(C)O)=O)CC(C)(C)OC2)=O)ccc2c(c1)ncn2C 32648,CCC(C(F)F)NC(=O)CC(C1CC1)NC(=O)CC1CC(OCC)C1.C(C)(C)C 32649,CC(C)C(C)C(CNC(C1CCSCC1)=O)NC(c1cc(=O)n(C)o1)=O 32650,N1(C(c2ccc(CC)cc2)=O)C(CC(N2CC(C)(N(C)C)C2)=O)C2CCCC12 32651,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(C2CC3CC3C2)=O)CCCCCC1 32652,Fc1cc(N2CCOCC2)ccc1CNCc1cn2ccsc2n1 32653,C(C(=O)NOCCC(=O)NCC1C2C3CCC(C3)C12)c1cncn(C)c1=O 32654,c1(C(=O)NCCC(C)NC(=O)Cc2cncs2)cccc(N)c1 32655,C1(C(=O)NCC(N(C(c2scc(C)c2Cl)=O)C)C2CC2)CCn2nnnc2C1 32656,C1(NC(Cn2ncc(C)c2)=O)C2CC1N(C(=O)CC1CC3(CCC3)C1)C2 32657,CC(=O)C(C)(C)CC(=O)NCC1(C(=O)NC2CS(=O)(=O)C2)CC1 32658,C1(C(N2CC(NC(C(C)(CO)OC)=O)C2)=O)Cc2cccc(F)c2O1 32659,C1(CC=C)(NC(=O)CCF)CCN(C(C2(F)CC2)=O)CC1 32660,c1(C(c2cnoc2)NCCC=CCCC)nnnn1C1CCCCC1 32661,C1(NC(c2c(C)sc(Br)n2)=O)CC2CC(C1)N(C(C1COC(=O)N1)=O)C2 32662,N1(C(c2csc(C)c2C)=O)CC2(C1)C(NC(=O)Cc1cn[nH]c1)CCS2(=O)=O 32663,C(=O)(C(C(C)C1CCOC1)N1CCCC(COC(F)F)C1)NCCNC(C)=O.C(C)=O 32664,C(C(=O)CC(c1ccccc1)c1ccccc1)NC(C)C(=O)O 32665,N1(C(C2C(NCCNC)C2)=O)CCCC(C(=O)NCCN(C)C(=O)OC)C1 32666,c1(CCCCC(=O)NC2CC(CNC(=O)CCC3CC3)C2)ccc(Cl)cc1Cl 32667,CC1(CCc2cccs2)CCCC1.N1(C(c2cccs2)=O)CCC(C2C(=O)N2)C1 32668,C#Cc1ccc(NC(=O)C(C(C)NC(C2CC(C)CCO2)=O)C(C)C)c(C)c1 32669,CC(F)(F)C(C)(C)CC(=O)NC1CCN(C(c2cc(C#N)ccc2Cl)=O)CC1F 32670,Cc1nc(CC(C)C)c(C(=O)NC2CCN(C(c3ccc[nH]3)=O)C2C(C)(C)C)s1 32671,C1(NC(C(=O)NCC2CC2)=O)C2CC(CN(C(C3SC4C=CC3C4)=O)C2)C1CO 32672,C1(CNC(=O)NC)CC(C(=O)N(C(C(N)=O)SC)C)=NO1.C1(C)C(=O)N1 32673,C=CCC(CNC(c1cnn(CC)c1C)=O)C(=O)N=c1cc(C)n(C(C)C)[nH]1 32674,c1(CC)nc(CCNC(=O)CC(O)CN(C)C)sc1Cc1ccc(Cl)cc1 32675,C1(NC(C2C(OC)(OC)CC2)=O)CN(C(C2CNC(=O)O2)=O)CCCO1 32676,C(CCCCCC(=O)NC(C)C(=O)N1CCCC1)NC(CC(C=C)C)=O 32677,c1(C(=O)NCCC2(NC(C(CC)O)=O)CCCC2)ccc(C2CCOC2)cc1 32678,N1(C(Cc2c(C)ccnc2)=O)CCC2(CCC(NC(=O)C(F)CC3CCC3)C2)C1 32679,N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)Cn2nnnc2C2CC2)CC1C 32680,c1(C(=O)NCC2OCCCN(C(C3N(C)CCOC3)=O)C2)sccc1S(N)(=O)=O 32681,C1(C)(CC)CC(C(=O)OC)CN1C(c1cccc(Oc2ncns2)c1)=O 32682,N1(C(CCSC)=O)C(C)CC2CN(C(=O)CC3CCNC3=O)CC12.CC(C)O 32683,C12CC3(C1)CN(C3)C2=O.c1(SC)cscc1C(=O)NC1(CO)CC1 32684,c1(C(=O)NC(CN(C(c2ccn(CC)n2)=O)C)C)ccc(C2CCC2(C)C)cc1 32685,CCC(C)C(C(=O)N1CCN(C(=O)C=CCO)CC1C(C)(C)C)OC 32686,C(CC1=CCN(C(c2cc(N)nc(Cl)c2)=O)CC1)NC(C(N1CCSCC1)C)=O 32687,C(CC(C(=O)NCC1CCOC1=O)NC(=O)C(Br)=C(C)C)SC 32688,N1(C(c2ccccc2)=O)CCCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 32689,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32690,C=C(C)CCC(=O)NC(C1CCCCC1)CNC(=O)CNC(c1cccnc1)=O 32691,c1(CNC(NC2C(OCC#C)CCCC2)=NCC2CCOC2)ncc(Br)cc1Br 32692,c1(-c2cn(CCC(=O)N(C)CC3CC4(CC4)C3)nn2)ccc(Cl)c(F)c1 32693,C1(C(N2CC(N(C)CC)C2)=O)CC1C1CN(C(C2CCSCC2)=O)C1 32694,N1(C(COC(CC)(C)C)=O)CC2CC(NC(=O)C=C3CCC(C)CC3)(C2)C1 32695,Cc1ccc(C(F)C(=O)N(CCCNC(C2CC(F)C2)=O)C2CC2)cc1 32696,c1(C(N2CCC(NC(CCS(=O)(=O)NC)=O)C(F)C2)=O)cnc2c(c1)CCCO2 32697,C1(NC(c2c(CC)con2)=O)CCN(C(c2cc(CS(C)(=O)=O)on2)=O)CC1C 32698,c1(CC(N2CCC(O)(CNC(C3(C(N)=O)CC3)=O)C2)=O)csc2ccccc12 32699,C(=O)(C(O)C(F)(F)F)NCC1CC(C)N1C(=O)CC(C)(C)C 32700,CCC(COC)C(=O)NC1CN(C(CCC(=O)NC2(C(=O)NC)CC2)=O)C(CO)C1 32701,N1(C(C2CCC(NC(c3cc(Br)cc(Br)c3)=O)CC2)=O)CCCC2CCCCC12 32702,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(CCO)c1)=O 32703,Nc1cc(O)nc(C2CN(C(C(=O)Nc3ccccn3)C3CC3)C2)n1 32704,c1(OC)ccc(NC(=O)C(=O)NCC(C2CN(C)CC2O)c2ccccc2)nn1 32705,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32706,C(C(=O)N1CCOC2(C1)CN(C(=O)CCCOC(C)C)C2)(c1ccccc1)=C(C)C 32707,CC(C)CC(CC(=O)NCC1(O)CCN(C(=O)C(F)OC(F)(F)F)CC1)CC(N)=O 32708,CN1CC(c2cn(CC(c3ccc(F)cc3F)CO)nn2)CCC1CC(=O)O 32709,c1(C(=O)NCCCCN(C(C2CN(C(C)C)C(=O)C2)=O)C)nc2cccnc2s1 32710,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32711,Fc1conc1CNCC1CCCS1 32712,CC(F)(F)C(C)(C)CC(=O)NC1(C)CCCN(C(=O)CCCNC(N)=O)C1 32713,C(=O)(C1Cc2ccccc21)NCC(CCCC)NC(=O)CC1(OC)CCOCC1 32714,c1(C(N(CCC(=O)NCCSC)CCC)=O)cn(C2CC2)nc1C 32715,N1(C(CC2CCC(=O)C2)=O)CC2(CCC(CNC(c3ccoc3)=O)O2)C1 32716,C1(C(N2CCC(NC(=O)NC)C2)=O)CCN(C(c2cn(C)c(C)n2)=O)CCO1 32717,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32718,c1(NC(c2ccn(CCC)n2)c2nnnn2Cc2cccs2)cccc2[nH]ccc12 32719,C1(C)(COC)CC(NC(C2CN(C)C2)=O)CN1C(=O)CCc1nncs1 32720,CCCC(CCC)CC(=O)NCC1CC(CCC(=O)NCCCCCO)C1 32721,c1(C(=O)NC2(CN(C(C3C(CCC)C3)=O)C)CC2)cncc(Cl)c1C 32722,N1(C(c2c(CC)nco2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32723,c1(OC)cc(F)cc(C=CC(=O)NCC(C)N(C(=O)C(O)C2CC2)C)c1 32724,c1(C(N2CC(NC(=O)Cc3cccs3)CC3(C2)CC3)=O)ccc2nc(O)oc2c1 32725,C#Cc1cc(F)c(CN2CC(O)(C#C)C2)c(F)c1 32726,N1(C(C2(SCC)CC2)=O)CC2CCCC2(NC(=O)Cc2csc(S)n2)C1 32727,C1(OCC)CC2(CCN(C(=O)CC=CC(C)(C)C)C2)C1.C12C(C1(C)C)NC2=O 32728,c1(N2CCC(NC(c3cccc(C(C)(C)C)n3)=O)C2)ccnc2ncnn12 32729,CC(C)(Cc1ccccc1)C(=O)OCC(c1ccccc1OC(F)(F)F)=O 32730,C1(C)(CNC(CN(C)CC)=O)CCCN1C(=O)Cc1cc(C)no1 32731,C(=O)(N=c1c(Cl)c[nH]cc1I)C1CC1c1c(C)noc1C.N12CCC(CC1)C2=O 32732,C(=O)(CCCCN=[N+]=[N-])NCC=C(C(N1CCC(C(=O)OC)CC1)=O)C 32733,Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)OCc2ccncc2)C3)cc(C)n1 32734,N1(c2n(-c3c(C)c(Cl)ccc3)cc(C3CC4CC3C3CC43)n2)CCC2CCC(O)C1C2 32735,Cn1nnnc1SCC(=O)NCC1CC1NC(=O)COCC(F)(F)F 32736,c1(-c2cnccn2)ccc(CNC(C2C(OCC)C2)=O)cn1.C12CCN(C1)C2=O 32737,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32738,N1(C(CNC(=O)Nc2n(C)cnc2)(C)C)CCN(c2ccc(F)cc2)CC1 32739,C(=O)(C(O)C(F)(F)F)N(C1COCCN1C1C2C(CN(CCF)C1)C(=O)C2)C 32740,c1(C2CC2)ccc(OC)c(OC)c1.C1(N(C2CC2)CC)CCCO1 32741,c1(NC(C2CC2(F)F)C)ccnc(N(C)CCn2cccn2)n1 32742,C1(N(C(C2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32743,C1(NC(=O)CCN2CCC(F)C2)CC(Nc2nccc(CO)n2)C12CCOCC2 32744,C=CCCCCCCCCC(C(=O)NC1CCC1)N1CCC(C)(CC)C1 32745,N1(C(C2C3(CCN(C(c4c(CC)c[nH]n4)=O)C3)C2)=O)CCc2c(C)cccc2C1 32746,N1(CC)CCC(NCCCNC(=O)C=CC(=O)Nc2ccccc2)C1 32747,c12cn(nn1)CC(=O)CCN2CC.N1(CC)CCCC1.C1(CC(=O)OC)(N)CC1 32748,c1(C(=O)NCC(C)C(=O)NCCCc2ncc[nH]2)cccc(O)n1 32749,S(=O)(=O)(c1ccc(Br)cc1)NCCNC(=O)Nc1cccc(-c2nnco2)c1 32750,N1(C(c2cccc(C)n2)=O)CC(O)C(O)C1CNC(c1ccc(C)c(CO)c1)=O 32751,N1(C(C2(CC(=O)OC)CC2)=O)CCCC(C(N2CCC(C(C)(C)O)CC2)=O)C1 32752,N1(C(CCC(C)SC)=O)CC(NC(c2nc(C3CC3)ncc2Cl)=O)C(C2CC2)C1 32753,c1(CC(=O)NC(C(=O)N(CC(CC)OC)C)C2CCCC2)cc(F)ccc1C 32754,N1(C(CC(C=C)(C)C)=O)CCC2(CCCCC2NC(C2CCC(=O)N(CC)C2)=O)C1 32755,N1(C(c2n(CCC)ccc2)=O)CCOC(CCCNC(C23CC(O)C2C3)=O)C1 32756,C(C(C(C)(C)C)NC(C1CC(C)(C(C)(C)C)C1)=O)NC(C1CC(C)OC1)=O 32757,CCC(C)(C)CCNC(=O)C=CCNC(=O)CS(=O)(=O)NCC(C)O 32758,c1(COC)ccc(CC(NC(=NCC2CCCCO2)NC2CCCCC2)C)cc1 32759,Cc1cncc(CC(N2CC(C(C)NC(=O)C(C)C3CCC3)C2)=O)c1 32760,N1(CCO)CCCC(C2(C)CC2)C1.Cc1cc(C(=O)NC2CCNC2=O)sc1C 32761,C(CCF)(C(=O)NCCC1CCCCO1)NC(c1cc(C)[nH]c1)=O 32762,C(=O)(C1=C2CCN=C2NC=C1)NC(CCCOC)c1cnc[nH]1 32763,C1(CNC(N(c2nc(C(F)(F)F)ccc2CN)C)=O)CCCS(=O)(=O)C1 32764,C1(CC)CN(C(c2cc(C#N)c[nH]2)=O)CCN1C(=O)C=CSCc1ccco1 32765,C1(OC)CCn2cc(C(=O)NCCNC(C3OCCC3C)=O)nc2C1 32766,C(c1cncnc1O)=CC(=O)NCCN(C(=O)CC(F)(F)F)C 32767,N1(C(c2c(C)nc(C)o2)=O)CCOCC(C)(CNC(C2CCCCC2C)=O)C1 32768,N1(C(C(c2n(C)cnc2)=O)=O)CCOC(C2CN(C(C3CC=CCC3)=O)C2)C1 32769,C1(CCCC)CCC(C(=O)NCCCN(C(c2ccc(Cl)s2)=O)C2CC2)C1 32770,N1(C(C2N(C(=O)OC(C)(C)C)CC2(C)C)=O)CC2CCC1C(O)C2 32771,c1(C(N(CCCCNC(C(CCC)O)=O)C)=O)cc(F)cc2c1NCCC2 32772,C1(C(=O)NCC(CN(C(=O)CCC2CC2)C)O)CCCC1P(C)(C)=O 32773,c1(C(=O)NCCC2(CNC(C3C(C)CCS3)=O)CC2)cc2ncn(C)c2cn1 32774,c1(C(C(=O)OCC)NC(=O)CCCN(C2CCCCC2)C)ccc2nonc2c1 32775,Cc1cc(C(C(=O)NC2CCCC2)N(C)CC2CCN2C(C)(C)C)c(C)cn1 32776,Cc1nn(CCC#N)c(C)c1NC(c1cn(CCCS(N)(=O)=O)nn1)CN(C)C 32777,CC(C(C)(C)C)=CC(=O)NC(CCCC(C)NC(=O)COC(F)F)C1CC1 32778,c1(C(=O)NCCC(C)CCNC(=O)COCC(F)F)cc2nc[nH]c2cc1N 32779,S(=O)(=O)(c1cccc(C#N)c1)N(C1CC2CCC(C1)N2)CCOC 32780,[N-]=[N+]=NC1CCCN(Cc2csc3ccc(Br)cc23)C1 32781,C(c1cnc2ccccc2n1)=CC(=O)NC1C2N(C(C(C)(C)CO)=O)C(CC2)C1 32782,c1(C(=O)NC(C(CO)NC(CC2(C=C)CCC2)=O)C)cc(C)nc2c1CCCC2 32783,Cc1cc(C(=O)NC2CN(C(=O)CC(=O)N(C)C)CC2C)c2nc(C)n(C)c2n1 32784,C1(C(=O)NCC2COCCN2C(=O)C(O)CCN(C)C)(CC)CCC(O)CC1 32785,S(=O)(=O)(c1ccc(Br)cc1NCCN(C)C)NCC(C1CCOCC1)C 32786,C(c1cccc(F)c1)=CC(=O)NC1C(NC(c2c(CC)c[nH]c2)=O)COCC1 32787,c1(C(=O)NCC2N(C(c3c(C)nc[nH]3)=O)CC(C)CC2)nnc2n1CCCCC2 32788,Cc1cc(C#N)cnc1C(N1CC(C)(C(N2CCCC(C)C2)=O)C1)=O 32789,N1(C(CC2(C(=O)O)CC2)=O)CCC(O)C(C)C1.C1(CC(=O)OC)CCCN1C 32790,C1(CC#C)(C(=O)NC(CN2CCCC2)CO)CCN(C(C2CC=CCC2)=O)C1 32791,c1(C(N2CC(C=C)C(NC(c3[nH]c(C)nc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 32792,N1(C(CNC(=O)OC)=O)CCCC2CN(C(=O)C(C)SCC(C)C)CC12 32793,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 32794,c1(CNC(=NC)N(C)Cc2c(CO)noc2C)cccc2c1OCCO2 32795,c1(CC(C(=O)OC)F)ccc(OCCSCCOC(=O)C2CC2)cc1 32796,CC(CC(C)(C)C)C(=O)NCC1CCC(C)(C)CN1C(=O)CCCN1CCCC1 32797,C1(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2ccc[nH]2)CC2CCC1CC2 32798,n1(CCCC)ncc(C(=O)NCC(C)N(c2nnc(COC)s2)C)c1C 32799,N1(C(C(C)N(C(=O)CC2CCCCN2C)C)=O)CCC(CNC(=O)C2CC2)CC1 32800,C(=O)C(C)(O)C(F)(F)F.N1(C(Cn2cc(CCCC)nn2)C)CCC(C)(C)C1 32801,C(=O)(C(C)CC(F)(F)F)NC1CN(C(COCCCCC)=O)CC1OC 32802,N1(C(C2N(C)CCC2)=O)CCC(C2CCC2)(NC(=O)C2CC2)CC1 32803,CCC(CC)CCCC(=O)NC(CNC(C1CC(=O)N(OC)C1)=O)CO 32804,N1(C(C(CC(C)C)=O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 32805,C(=O)(CCCS(N)(=O)=O)NC(c1ccccc1F)CNC(C=Cc1ncc(C)[nH]1)=O 32806,N1(C(Cc2c(OC)ccnc2)=O)CCOCC(NC(C2CCCC(OC)C2)=O)C1 32807,c1(C(=O)NCCN(C(C2CCC2OC)=O)CC)cc(Br)n(C)n1 32808,C(=O)(C(CC(C)(C)C)OC)NC1C(OC)CN(C(=O)CSC2CC2)C1 32809,c1(C(N2CC(C)C(NC(C3CN4CCN3C(C)C4)=O)C2)=O)cc(F)c(F)cc1F 32810,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 32811,C1(CNC(CC(C)(C)C)=O)CN(C(=O)CSc2ccccn2)CCCO1 32812,c1(C(N2CC=CC(NC(C34CC(C#N)(C3)C4)=O)C2)=O)ccc2nc(O)[nH]c2n1 32813,C1(NC(=O)CCc2ccccn2)C2CC3C1C3C2C(=O)NC(C1CC1)C1CC1 32814,C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCNC(=O)COCCCF)CC 32815,C1(CN(CC(c2c(OC)cccc2)OC)C=O)CC1C1CCCC1 32816,N1(C(CC=C)=O)CC(OC)CC1CNC(c1ccccc1NCC1CCCO1)=O 32817,C1(C(N(CCF)CC)=O)CCC(NC(=O)C=C(C)C)CC1 32818,C1(O)(C(C)NC(=O)CCN(S(C)(=O)=O)C)CCN(C(=O)CSC(F)(F)F)CC1 32819,C1(c2n(CCCC)nnn2)(NC(C2CCOCC2)CSCCF)CCCOC1 32820,C(C(O)C(C)(C)C)N(C(C1(CCC=C)CN(C(c2cn(CC)cn2)=O)C1)=O)C 32821,N1(C(c2nc(C)sc2)=O)CCC(C)C(NC(=O)CCNC(=O)C(C)(C)C)C1C 32822,c1(C(=O)NC(CN(C(c2c(OC)cncn2)=O)C)C)cnc2c(c1)ncn2C 32823,c1(C(N2CC(CNC(c3c[nH]c(=NC)o3)=O)C(C)C2)=O)cc(C)c2sccc2c1 32824,C#CC1(C)CCCN(C(=O)CN(C(c2cccc(CO)c2)=O)CC)C1 32825,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 32826,N1(C(c2n(CC)ncc2)=O)CC2CC(C1)CN(C(=O)COC1CC1)C2 32827,C1(Cn2cc(CCN(C(C(CCC)OC)=O)C)nn2)CCCC(F)(F)C1 32828,C1(NC(C(CCC2CCC2)NC(c2c(C)noc2C)=O)=O)CCCCN(C)C1=O 32829,C1(CC)(NC(=O)COC(F)F)CCN(C(c2cnn(CC(F)(F)F)n2)=O)CC1 32830,N1(C(C)Cn2cccn2)CC2CCC(C1)N2C(c1ncccn1)=O 32831,CC(C)CCC(C(=O)Nc1cnsc1)NC(=O)CCc1cccnc1 32832,Cc1cc(Cl)c(C(=O)NC2CC2NC(=O)Cn2cnc([N+](=O)[O-])c2)cc1[N+](=O)[O-] 32833,CCCC(C)CN(C(=O)C(C)N(C(=O)CC(C)n1cccc1)CC)C 32834,C1(C(N(CCCC(=O)NC(c2cnn(C)c2)C)C)=O)CCCCCN1C 32835,c1(C(=O)OCCCC(=O)OCC)cc2c(Br)nn(C)c2s1 32836,c1(C(N2CC(CNC(C=C(C)C(C)(C)C)=O)C3C2C3)=O)cccc2c1CCC2=O 32837,C1(C(N(CCC)CCNC(c2c[nH]c(=N)s2)=O)=O)COCCN1CC(F)F 32838,C1(c2cn(CCCCOC)nn2)CN(C(=O)CC2CC3CC(=O)C2O3)CC1(F)F 32839,c1(CC(=O)NC2CC(NC(c3c(OC)cc(F)cc3)=O)C2)cn2nc(C)sc2n1 32840,c1(CC)cc(C(N2CC(CO)(NC(=O)Cc3cnnn3C)C2)=O)sc1C 32841,Cc1cc(C(N2CCOCC(NC(c3cnc(F)c(Cl)c3)=O)C2)=O)nc(C)n1 32842,CN1N=C(C(=O)N(CC(O)CN(C)C(c2ccc(F)c(F)c2N)=O)C)CCC1=O 32843,C(=O)(CCC(F)(F)F)NCC1C(NC(c2ccnc(CC(C)C)n2)=O)CCC1 32844,N1(C(c2cccc(OCCC)c2C)=O)CCCN(C(C2(C)CC(C)C2)=O)CC1C 32845,N1(C(=O)Cn2ccc(C(F)F)n2)CC2CN(C(C3CC3(F)F)=O)CC2C1 32846,Cn1cnc2c1CCCC2C(=O)NC1CCN(C(=O)CN2CC(=O)NC2=O)CC1F 32847,C1(N(C(N2C(COC)CC2)=O)C)CN(C)N(C)C1 32848,c1(CNCC2C(SS(C)(=O)=O)C2)cccc(S(=O)(=O)C(F)F)c1 32849,C1(CCNC(Cn2ncc(C)c2)=O)CN(C(C2C(C)OC(C)C2C)=O)CC(C)O1 32850,C(CC(C(C)C)NC(=O)CCc1ccc(Cl)nc1)N(C(c1c(CC)ccs1)=O)C 32851,c1(C(N2C(C)CC(NC(c3c(C)nc(C4CC4)s3)=O)C2)=O)cccc2cc[nH]c12 32852,N1(C(C(CCNC)O)=O)CC2(CNC(C3CCCC3C3CC3)=O)CC1CO2 32853,C1(=O)C(C(C)C)N1.C1(C(C)C)CCN(C(=O)Nc2ccc(CN)cc2)CC1 32854,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2c(C#N)cccc12 32855,N1(CCC(=O)NC(C)CCNC(=O)C=Cc2ccco2)Cc2ccccc2C1=O 32856,c1(C(=O)OC)cc(C(=O)NC(CNC(c2ccoc2C)=O)C(C)(C)C)cc(F)c1 32857,Nc1cc(Cl)ccc1C(N1CC2CCC2(CCNC(c2cnnc(O)c2)=O)C1)=O 32858,CCCCC(O)C(=O)NCCCC(C)(C)NC(c1cc(CCC)n(C)n1)=O 32859,c1(CN(C(c2[nH]cc(CN(C)C)c2)=O)CCN(C)C)ccc(C#N)cn1 32860,c1(COC(c2nc(C3CC3)cs2)=O)cccc(I)c1 32861,C1(OC)CN(C(c2ncncc2Cl)=O)CC1NC(c1ccc(OC)nn1)=O 32862,Nc1c(F)ccc(F)c1C(N1CCN(CCNC(=O)CC2CCCCO2)CC1)=O 32863,c1(CC2(CNC(C3CN(C(Cc4nnc(C)o4)=O)C3)=O)CC2)ccc(F)cc1 32864,Cc1nc(N2CCN(CCNC(c3nn(C)cc3C)=O)CC2)[nH]c(=N)n1 32865,C1(NC(C)=O)CCC(C(=O)N(C)CCN2CCCC2=O)OC1 32866,Cn1nc(C(C2CC2)NC(=O)NC2CC2CCF)cc1N 32867,c1(N2CC3OCCN(C(CC(CC)C)=O)C3C2)ncnc2cccnc12 32868,CC1(C(=O)Nc2cc(-n3cccc3)no2)CCN(C(=O)CSCC(F)(F)F)CC1 32869,c1(CNC(=O)NC(c2ccoc2)C)csc(C(C)(C)C)n1 32870,c1(C(=O)NCC(CC)NC(c2nc(SC)ncc2Cl)=O)cnn2c1CC(C)CC2 32871,c1(C(N2CC(N(C(=O)CCc3cnco3)C)C2)=O)ccc(OC2CCOC2)cc1 32872,c1(C(=O)NC2CC2)ccc(CNC(=O)CC(Cl)Cl)nc1 32873,C1(NC(C(N2CCNC2=O)C)=O)C2CC1N(C(C1CCSC1)=O)C2 32874,C1(CNC(C=CSC)=O)CN(C)CCN1C(=O)Cc1ncccc1C 32875,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 32876,Cc1cccc(CC(=O)NC(c2ccccc2F)CNC(=O)CCNC(N)=O)c1 32877,N1(C(C2(C)C=CCC2)=O)CCC(N=c2nn[nH]n2C)CC1 32878,C1(C(=O)NC2CC(F)(CNC(C(C)NC(COC)=O)=O)C2)CCC(C(N)=O)CC1 32879,C1(C(=O)NCCCC2OCCN(C(C(C)(C)N(C)C)=O)C2)CCCCC12CCC2 32880,C(CC(O)CC(=O)NCCN(C(=O)C(C(C)(C)C)C1CCC1)C(C)C)SC 32881,c1(CC)cc(C(=O)NC(C)CCCNC(=O)C(c2ccc(C)cc2)(C)C)nn1C 32882,c1(C(=O)OCC)ccc(CC)nc1.c12csc(c1)C(=O)NC(CO)CNC2 32883,CCCCC(C(=O)N1CCCOC(CNC(=O)Cc2nc[nH]n2)C1)ON=C(C)C 32884,Cc1ccc(OCCC(N2CCC(NC(c3snnc3C)=O)C2)=O)cc1 32885,c1(C(N2C3C(NC(c4c(N)cccc4Cl)=O)CC(C3)C2)=O)cc2cccnc2[nH]1 32886,c1(N2CCC(CCC)(CO)C2)nc(=NCC(C)(C)N2CCCC2)[nH]c2c1CSC2 32887,C1(CCC(=O)N(CC(C)(C)C)CCO)CCCN(C(=O)CCOC2CCC2)C1 32888,c1(OC)cccc2c1OCCC2NS(=O)(=O)c1c(Br)cc(Br)cc1Br 32889,c1(OC)ncccc1C(=O)N(CCCC(=O)NC(c1cnc(C)s1)C)C 32890,N(C1=NCC2C(C(F)(F)F)CCN1C2)Cc1cnn(C2CC2)n1.CC 32891,N1(C(=O)COc2cc(F)ccc2C(F)(F)F)CCS(=O)(=O)N2CCCCCC12 32892,CC1CN(C(=O)CSc2nccn2C)CC1(C)CNC(c1ccc(C(F)F)s1)=O 32893,C(=O)(C#CC1CCCOC1)N1CCC(CNC(c2cc(NC(C)=O)c(F)cc2)=O)C1 32894,c1(C(N2CCC(C(C)NC(=O)CCc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 32895,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 32896,c1(CO)ccc2c(c1)CC2.N12CCC1C(=O)N(C)CCCNC(=O)C2 32897,C#CCCC(C(=O)NCC1(C)CC2(CC2)C1)NC(=O)CCCC#CC 32898,N1(C(=O)OC(C)(C)C)Cc2ccc(CC(=O)NCc3ccc4nn[nH]c4n3)cc2C1 32899,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 32900,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(CC(C)C)c2)=O)CCC1 32901,N1(C(CCC=C)=O)CCOC(CNC(=O)Cc2cccs2)C1 32902,C(CC(=O)N(CCC(=O)Nc1cccc(Cl)c1)OC)OCCCOC 32903,N1(C(c2n(CC)cnn2)=O)CC2CCCC2(NC(=O)Cc2cn(C)nn2)C1 32904,C1(N(C(C(C)N(C(CC)=O)CCC)=O)C)CCN(C(c2ncoc2C)=O)CC1 32905,C1(NC(CCNS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1CO 32906,C(CC(C(=O)NC1CCC(OC)C1)NC(C1CCCSC1C)=O)=CC 32907,CC1(NC(C2(C)CC2(C)C)=O)CN(C(=O)Cc2cc(Cl)cs2)C1 32908,C1(F)(CNC(c2nc(C)nn2C)=O)CCCN(C(=O)C=CC=C(Cl)Cl)C1 32909,CCC(C)C(CO)NC(=O)CCC1CCC(NC(=O)C=C(C)C)C1 32910,CCC(C)CCCCC(=O)NOCCN(C(C)CC1CC1)C 32911,C(=O)(C(CO)NC(=O)C=C(C)COC(C)=O)N(CC(C)O)CCO 32912,C1(=O)CCCCOC2CCN1C2.C1(OC)CCN(C(=O)COC(C)=O)C1 32913,C1(C(=O)OC)(OC)CCN(C(=O)CC23CC(C)(CO2)C3)CC1 32914,Cc1cc(C(=O)NC(CC2CC2)C(=O)Nc2ccccc2CCO)ccn1 32915,C1(NC(=O)Nc2c(OC)cccc2)CCN(Cc2cccc(N)n2)CC1O 32916,CC1CC(NC(c2ccn(CC(F)(F)F)n2)=O)CN1C(c1cc(CCO)on1)=O 32917,c1(C(=O)NCC(CSC)NC(C=CCCC)=O)cc(C(F)F)ccn1 32918,N1(C(Cn2c(C)ccn2)=O)CCOC2(C1)CN(C(C1CC(=O)N(O)C1)=O)C2 32919,n1(CC#C)c(C)cc(C(=O)NC2(CF)CCN(C(C3CC(F)C3)=O)C2)c1C 32920,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 32921,CCC(C(=O)OC)C(=O)NCC(CC)N(C)C(C1(c2cc[nH]n2)CCC1)=O 32922,c1(CSC)ccncc1.C12CCN(C1)C(=O)C1(CC1)OC(C)C(=O)N2CC 32923,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 32924,c1(OC)ccc(C(=O)NCC(C)NC(C2CN3CCN2CC3C)=O)c(OC)c1C 32925,C(=O)(CC1OCCc2ccsc21)NC1C(C)CCN(C(=O)CCC[N+](=O)[O-])C1 32926,C1(OC)CC2CCC(C1)N2C(=O)CC1CCCN(C(C2(C)CCCN2C)=O)CC1 32927,c1(C(=O)NC2C(CNC(C(C)C)=O)CC2)cc2c(cnn2C)nc1C(F)F 32928,N1(C(COCCOC)=O)CC2(C1)SCCC2NC(C1(O)CCOCC1)=O 32929,O=C(C1=CC2(CCOC2)C1)N1CCCCC(N(c2cnc(F)cn2)CCO)C1 32930,c1(OCC)cncc(C(=O)NCCOCCCNC(=O)C(C)(C)Br)c1 32931,c1(OC)nccnc1C(F)(F)F.C12CN(CC1C)C(=O)C1CCCC(C1)C(=O)N2 32932,CCC(C#N)(CC)C(=O)N1CC2CC1(CNC(=O)Cn1nc(C)ccc1=O)C2 32933,c1(C(=O)NCCC(=C)CNC(C23CCCCC2C3)=O)cc(C)cc(C)c1C 32934,N12CC(C(C)(C)C1)NCc1ccc(cn1)-c1n(ccc1)C2.N(C)(C)CC 32935,C1(NC(C(Cc2ccoc2)NC(C(C)C2(C)CC2)=O)=O)CC2C(O)C(O)CC12 32936,c1(C(=O)NCCCC(C)(C)NC(C2C(CC(C)C)C2)=O)nccc(C#N)c1F 32937,C(C)(CCC(=O)NC1CC(C(=O)NCc2nnc(O)n2C)C1)OCC 32938,c1(C(N(C(C)CNC(C2CC2F)=O)C)=O)cc(Br)nn1C 32939,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 32940,CN1N=CC(CC(N2CCC(CNC(c3cc(C4(C)CC4)on3)=O)C2)=O)C1=O 32941,C1(CC)(COC)CCN(C(=O)C2CC2)C1.c1(O)cccnc1 32942,c1(C(N2CC(CC)N(C(c3c[nH]ccc3=O)=O)CC2)=O)csc2c1CCC(C)C2 32943,Cc1cc(N2CCCC2)nc(N(C)CCNc2cc(Cl)sc2Cl)n1 32944,c1(CNC(N2CCCC2)=O)cc(-c2ccccc2)cnc1O 32945,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 32946,c1(CC(=O)NCC2N(C(CCOc3ccc(C)cc3)=O)CC2)ccc(F)c(F)c1 32947,C(CC)(CCC(=O)NCc1cc(F)ncc1O)c1c(C(=O)OCC)nco1 32948,C(CC(=O)N1CCC(N(C)C(c2cc(C(C)(C)C)[nH]c2C)=O)C1)(C(F)(F)F)OC 32949,N1(C(C2C3CCC(F)C23)=O)CC2CCCC2(C(NCP(C)(C)=O)=O)C1 32950,c1(C(=O)OC)nc(C(c2ccc(F)cc2)NC(C)C2CC2)n(C)n1 32951,N1(C(CC(C=C)(C)C)=O)CC(NC(c2cnn(C(F)F)c2)=O)C(N=[N+]=[N-])C1 32952,C1(C)(C(N2CC(N(C(CC(C)OCC)=O)C)C2)=O)CC(C)=NO1 32953,N1(C(C(C2CC2)OCC)=O)CCCC12CCCN(C(C1(CC)CCCC1)=O)C2 32954,C1(OC)CCN(CC(=O)NCC(=O)NCC(=O)N(C2CNC(=O)C2)C)C1 32955,Cn1cc(C(=O)NCC(O)CN(C(=O)COCCCF)CCO)ccc1=O 32956,C(=O)(CC(C(F)(F)F)SC)NC1(C(=O)NC(C(CC)C)CO)CCOCC1 32957,c1(OCC(=O)NCCNC(C2CCOC(C3CC3)O2)=O)c(Cl)cccc1Cl 32958,CCCC(C(=O)NC(C)CC)NC(=O)CC1CC2CC2C1 32959,C1(NC(c2cnc3[nH]ncc3c2)=O)CC2CN(C(c3occc3Cl)=O)CC2C1 32960,n1(CCC(=O)N(C)CC2CCCN2C(=O)C(F)CC2CC2)cccnc1=O 32961,c1(NC(C2CCC(NC(c3ccc(COC)cc3)=O)C2)=O)c(C=O)c(C)nn1C 32962,C1(C(N2CCC(CC#C)C2)=O)N(C(c2sccc2F)=O)CCC1(C)C 32963,c1(CCNC(c2c(-c3c(OC)csc3)ncs2)=O)ccc(Br)cc1F 32964,c1(C(=O)NC(CC(C)C)CNC(=O)CCCCC(C)C)coc2cc(F)ccc12 32965,c1(OC)cc(C#N)ccc1CN1CCC(Oc2ccc3c(c2)OCO3)C1 32966,C1(C(=O)NC2CC(CNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 32967,CC1CCC(N(C)C(c2cc(C(F)(F)F)co2)=O)C1 32968,C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2ccncn2)CC1(C)C)OC 32969,C1(NC(=O)CCc2ccco2)CC2CC1CN(C(c1noc3c1CCCC3)=O)C2 32970,C(=O)(C1c2c[nH]nc2CN1C(=O)C(=O)NCC1CC1)NC(C(C)(C)C)CO 32971,C(CCN(C)C(c1cc(F)cc(Cl)c1)=O)(C(C)(C)C)NC(C1C(C)OCCO1)=O 32972,C1(NC(c2c(C)nco2)=O)CCCC(NC(=O)C(c2cc(Br)co2)=O)C1 32973,N1(C(C2N(C(C)C)CCC2)=O)CCC2(CC1)CC2=CC(N1CC2CCC2C1)=O 32974,N1(C(=O)OC)CCN(C(C(=O)NC(C)C)C2COC2)CC1(C)C 32975,C12(NC(C(Cn3cncn3)NC(C3C(C#N)C3)=O)=O)CCCCC1OCC2 32976,N1(C(Cc2c(C)nsc2)=O)CCC(NC(C2CCS(=O)(=O)CC2)=O)C12CCC2 32977,CCCCCC(O)C(=O)NCCC1CCCN1C(c1c(C)nn(C)c1N)=O 32978,C1(OC)CC2(C(=O)NCC(N3CCC(F)(F)C3CCCO)=O)COC1C2 32979,c1(N(CC(N2CCCC(C3(C)COC(=O)N3)C2)=O)C(C)=O)cccc(O)c1 32980,Cc1nc(N2CCC(CNC(C3(C)CC3C(F)(F)F)=O)C2)c2ccsc2n1 32981,C1(C)(C(N(CC#C)CC=C)=O)CC(O)CN1C(c1cnnn1CC)=O 32982,C1(CN2CCC(c3cn(C(C)C4CC4)nc3)CC2)COC2(CCC2)CO1 32983,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 32984,c1(OC)cc(CNc2ccc(NC(c3cc(O)ccn3)=O)nc2)c(Cl)cn1 32985,N1(C(c2ccc(CC)s2)=O)CC(C)CN(C(=O)CC(C)n2ccc(C)n2)CC1C 32986,c1(NC(C2(C)N(C(CCC#C)=O)CCC2)=O)cc(C(C)(C)C)cc(C(C)C)c1O 32987,c1(C(N2CCN(C(=O)C=CBr)C(C3CCC3)C2)=O)cccc2nonc12 32988,C1(CNC(CSCC#C)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 32989,C1(CNC(C2C3CN(C(CC4(N(C)C)CCC4)=O)CC32)=O)CC(=O)NC(C)C1 32990,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 32991,C1(CNC(CSCC=C)=O)CC(C)N(C(c2cn(C)c(O)n2)=O)C1 32992,C1(C(CC=C)C)CCCN1N1CCN(CC(C)C)CC1 32993,C1(C(=O)NC2CCC(OCC)CC2)C2CCC(C2)C1NC(=O)C1=CCCC1C 32994,N1(C(CC2C(C)OCC2)=O)CCC(N=[N+]=[N-])(C(=O)NCCCc2cn[nH]c2)C1 32995,c1(C(=O)NCC(C)NC(c2cc(C)no2)=O)c(C)cc(F)cc1Br 32996,N1(CC(=O)NCc2ccsc2)CCC(C2CNC2)CC1 32997,N1(C(c2n(CC)ncc2)=O)CC2CCCC1C2CNC(C1(C)CCCO1)=O 32998,C1(C(=O)NC(c2cccnc2)CC)CCC2(CC2)N1C(c1ccc(C)c(O)n1)=O 32999,Cc1ccc(NC(C2CN(C(C3CCCCO3)=O)CCS2)=O)c(C#N)c1 33000,Cc1cc(-c2cccs2)c(C)n1CC.C12CCCN1C(=O)COCCNC2.C(N)=O 33001,C1(NC(c2n(C)c(S)nc2)=O)CC(O)CN(C(=O)CCCc2ccc(Cl)cc2)C1 33002,C(=O)(C(O)C(C)(C)C)N1CC(C(C(=O)NCC2CC(CC(=O)OC)C2)OC)C1 33003,C1(C(=O)OC)C2C=CC(CC2)C1CNC(N1CC=C(C)C1)=O 33004,Cc1ccc(C(CNC(C2CCOCC2)=O)NC(=O)C(C)c2ccco2)cc1 33005,n1(CCC)cc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C(F)OC)C2)cn1 33006,C(C)(C(C(=O)N(CC(=O)NC(C#C)CC(C)C)CC#C)C(C)C)OC(C)=O 33007,Cc1cnc(CNC(=O)CCC2CC(NC(C3CCC3C(F)F)=O)C2)o1 33008,C1(CNC(CN(CC)CC)=O)(CO)CCCN(C(=O)Cc2nc(C3CC3)cs2)C1 33009,Cn1ccnc1C1CC1C(=O)NCC1(O)CN(C(c2ccccn2)=O)C1 33010,c1(C(N2CCCC(NC(Cc3c(CC)con3)=O)CC2)=O)ccc2sncc2c1 33011,N1(C(CC=C=C)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33012,CCC(F)(C(=O)OC)C(=O)NC(C)CNC(=O)COc1ccc(Cl)cc1 33013,N1(C(C2N(C(=O)CCN3CCCCC3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33014,N1(C(CCNC(=O)NC)=O)C2CCC1CC(NC(=O)CC1(CSC)CC1)C2 33015,C1(C(=O)NC(C)Cc2cccnc2)CC(NC(C2CCCN2C(C)C)=O)C(O)C1 33016,Cn1cnc2cc(CC(=O)NCC3CC(NC(C4CCCC4)=O)C(O)C3)ccc12 33017,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33018,C1(C(=O)NC2CCC(NC(COCC#C)=O)C2)(OC)COc2ccccc2C1 33019,CN1N=C(C(=O)NCCNC(C2CC(OC)CN2C(=O)C2CC2)=O)CCC1=O 33020,C1(CCNC(c2c(CC)cc[nH]2)=O)CCCCN1C(=O)CCNC(C1CCCC1)=O 33021,C1(C)(C(=O)NC(C2CCN(C(c3coc(CC4CC4)n3)=O)CC2)C)CC2(CCC2)C1 33022,c1(C(N(C2CCN(C(=O)C(C)(C)CO)C2)CC)=O)cc2c(C)cc(Cl)cc2[nH]1 33023,C1(C(=O)NC(C(=O)N(C)C)C2CCCO2)CN2CCN1CC2 33024,N(C1CCc2c(F)ccc(F)c21)c1c(OC)c(O)ccn1 33025,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CCNC(=O)CN1CC(=O)NC1=O 33026,n1(CC)cnnc1C(N1CC(CO)C1)=O.S(=O)(=O)(C(F)F)N1CCC1 33027,c1(NC2(CNC(C3C(C)(CC)C3)=O)CCCC2)nc(C)nc(O)c1C 33028,c1(C(N(CCNC(C2C(=C)C2)=O)C(C)C)=O)cc(N2CCOCC2)nc(Cl)c1 33029,CC(C)C(C)(O)C(=O)N1CCN(C(=O)C(C)(c2ccccc2)N(C)C)CC1 33030,N1(C(CCSC)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33031,c1(C(=O)NCC(=C2CN(C(C3CC3(F)F)=O)C2)F)n[nH]c(C2CC2)n1 33032,C1(C(N2CCC(NC(c3cnn(CCF)c3)=O)CC2)=O)CCCNNC1=O 33033,N1(C(C=CC=CC)=O)Cc2ccccc2C(NC(=O)Cc2ccsc2C)C1 33034,C(=O)(C1CSc2ccccc21)N(C(c1ccc(N)cc1F)=O)CCO.CO 33035,Cc1ccc2[nH]cc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CC(O)C3)=O)c2c1 33036,c1(C(N(C2CC(NC(=O)C(F)CC3CC3)C2)C)=O)cncc(N)c1 33037,C1(C(N2CCCC(N(C)C(c3c[nH]c(=N)s3)=O)C2)=O)CC2CSCC(C1)C2 33038,C1(C(=O)O)(S)CCCCC1.n1(CCNC(C(C)OCC2CC2)=O)cc(C)nn1 33039,C1(NC(CCCC#C)=O)CCCN(C(c2cscc2C#N)=O)C1C 33040,c1(C(=O)NC2CCC(NC(C3(C(C(=O)OC)OC)CC3)=O)C2)cnc(O)cc1C 33041,N1(C(C2CC3CC3C2)=O)CCC2(C1)c1[nH]cnc1CCN2C(C1(O)COC1)=O 33042,CC(C)(C)C#CC(=O)NC1CCN(C(=O)Cc2ccno2)CC1c1ccccc1 33043,c1(C(=O)OC)cccc(-n2cc(C3C(C)CCN3C(C3CC3(F)F)=O)nn2)c1 33044,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CC1CC2(CCC2)C1 33045,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33046,c1(OC)cc(C(N2CCCOC(CNC(c3cn(C)cn3)=O)C2)=O)c(C)nc1C 33047,c1(C(=O)NCC2(CCNC(CN3C(C)CCC3C)=O)CC2)cccc2nncn12 33048,C1(F)(Cn2cc(C(C)(C)OC)nn2)CCN(C(=O)C(c2cccnc2)OCC)C1 33049,N1(C(c2n(C)nc(C)c2Cl)=O)C2CCC1CN(CC13CC(C(N)=O)(CO1)C3)CC2 33050,c1(C(=O)OC)cccc(Br)c1NC(=O)C(=O)NCc1ccn(C2CNC2)n1 33051,CC1(C)Cn2[nH]c(=NC(=O)NCC3CC(F)(F)C(=O)N3)cc2CO1 33052,CN1CCC(NC(=O)CCC2CCN(C(C3CC4CC4C3)=O)C2)C(C)(C)C1 33053,c1(C(=O)NCC#CCNC(Cc2cn(C)nn2)=O)cc(Br)c(Br)o1 33054,C(=O)(CC(C)(C)C)NC(C)C(N1CCC(C(=O)N(c2cc(Cl)c[nH]2)C)CC1)=O 33055,N1(CC)CCOCC1C(=O)N(CCCN(C(=O)CN1CCN(C)CC1)C)C 33056,C(CCN=C(NCC1(CN2C(=O)CNC2=O)CC1)N1CCCC(SC)C1)OC 33057,c1(NC)cccc(C(=O)NCC(C)(C)CN(C)C(c2cn(CCO)nn2)=O)c1C 33058,c1(CC(N2C(CO)CC(NC(CCC(CC)C)=O)C2)=O)cccc2nsnc12 33059,C(CCC(=O)NCC(CC)N(C(=O)C(C)CN(C)C(=O)OC(C)(C)C)C)=CC 33060,C1(C(=O)NCC(C)N(C(c2cn(C)nc2SC)=O)CC)CCc2nnc(O)n2C1 33061,c1(C(N(CCCN(C)C(C2CCC(C3CC3)CC2)=O)C)=O)cc2sccc2[nH]1 33062,N1(C(C2C(NC(C3CC4(CCC4)CO3)=O)CC2)=O)CCC2(CC1)CC2CO 33063,C1(C(N(C(C)C)Cc2ccco2)=O)CN(C(C2CCC3(CCC3)C2)=O)CCN1C 33064,N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(=O)Cn2cnnc2O)CC1C 33065,C(=O)(C(F)C(=O)NCC1CC(NC(C2CCCN(C)C2)=O)C1)OCC 33066,C1(NC(c2cn(CCC)nn2)=O)CN(C(c2ccc(CC)cc2F)=O)C(C)(C)C1 33067,C(CCC1CC1)(C(=O)NOCC(=O)OC)N(C(C(CC)(C)COC)=O)C 33068,c1(CC)onc(C(N2CCC(C(=O)N(CC(O)CO)C)C2C(C)C)=O)c1C 33069,C1(C(=O)N)C2CCC(C2)C1C.c1(C(C)C)cc(CNC(C2(C)CC(F)C2)=O)no1 33070,C(=O)(C1CCCc2ncnn21)N1C(C)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)C1 33071,CC1=C(C)C(Br)(C(F)(F)F)C(c2nn(C)cc2I)=N1 33072,c1(C(=O)NC2CCC(CCNC(CC(C=C)C)=O)C2)c(C)nc2sccn12 33073,c1(C(=O)NC2C(C)CN2C(=O)C=Cc2cccs2)ccnc(OCC(F)(F)F)c1 33074,C(CC1=CCOCC1)NC(C(C1CCCCN(C(=O)C=CCO)C1)C)=O 33075,N1(C(CCOCC)=O)CCC(NC(c2cc(-c3ccccc3)[nH]c2C)=O)CC1C 33076,C1(CNC(CCc2cnc(C)s2)=O)CN(C)CCN1C(=O)CCC1(C)CC1 33077,N1(C(C(CC=C)NC(=O)C(C)OCC=C)=O)CC=C(CO)CC1 33078,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33079,N1(C(c2cc(C)sn2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33080,c1(OC)cncnc1C(=O)NC(CN(C)C)C(=O)NC1CCCCC1F 33081,C1(c2n(CCNc3ccccn3)ncc2)CCN(Cc2ccccc2OC)CC1.CC 33082,c1(C(=O)NCC23N(C(COCCOC)=O)CCC2CC3)cc2c(O)ccc(F)c2[nH]1 33083,c1(C(N2CCC2CC2CC2)=O)cc2cccc(Cl)c2[nH]1.c12cc(no1)C(=O)N2 33084,C1(=O)C(C)O1.C(C(F)(F)F)OC(=O)CC1(c2cc[nH]n2)CCC1.C1CCN1CC 33085,CCN=c1[nH]cc(C(=O)NCC2COCC2NC(c2nc(C)oc2C)=O)s1 33086,c1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)c[nH]c2ncc(Br)cc12 33087,N1(C(C)=O)C(C(N2CC(O)(C(N3CCP(C)(=O)CC3)=O)C2)=O)CCC12CC2 33088,C1(NC(=O)CCC2CCCO2)CCSC12CN(C(c1cnn(C3CCC3)n1)=O)C2 33089,CC1(C(=O)NCC2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC2CCC1C2 33090,CCC(CC(F)(F)F)C(=O)NC(CCN(C(=O)CCNC(=O)C=CCl)C)C(C)C 33091,N1(c2n(CC=C)c(C(O)CCC)nn2)CCC(C)CC(C)C1 33092,C1(NC(c2c(C)con2)=O)CN(C(=O)Cc2ccns2)CCC12CCC2 33093,Cc1cc(CN2CCN(CSc3ccccc3)CC2)nc(-c2cccnc2)n1 33094,Cc1nc2sccn2c1C(=O)NC(C)C(C)NC(=O)CCCS(C)(=O)=O 33095,C1(NC(c2cnc(C)o2)=O)CCOC12CCN(C(c1cc(Br)c[nH]1)=O)CC2 33096,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33097,CC(C)CC(CNC1(F)CCN(C)C1)NC(=O)OC(C)(C)C 33098,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CN(C)CC)C2 33099,N1(C(=O)CCc2nccs2)CCCCC1C(N1CCOC2CC12)=O 33100,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33101,c1(C(C(=O)N(CC(N2CCCC2SCC(C)C)=O)CC)O)cccc(C)c1 33102,N12CCOC(C1)C(=O)N1CC(C1)CC(=O)N1CCC1(C)CC2=O.CCO 33103,N1(C(CC(=O)NCCO)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33104,N1(C(CCCC)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33105,c1(C(N2CCC(N(C(CC(C=C)C)=O)CC3CC3)C2)=O)ccc(F)c(Cl)c1 33106,c1(NC(COCC(=O)N(CC(CC)NC(=O)Cn2cncn2)C)=O)ccc(F)cc1 33107,Cc1cc(C(=O)Nc2nc(Cl)nc(Cl)n2)cnc1Cl.N12CC(F)(F)CC1C2=O 33108,C=CC(CCC)CC(=O)NC12CCC1CN(C(=O)C(O)CC(F)(F)F)C2 33109,N1(C(CCC(=O)NCC)=O)CCC2CN(C(=O)CC3CC(F)C3)CCC12 33110,N1(Cc2nc(CC)sc2Br)CC(CC2CC2)OCC12CC2 33111,C(CCCN=c1cc(C)[nH]cc1S(=O)(=O)N1CCn2nncc2C1)OCC 33112,CCCCCC(O)CC(=O)N(CCCCNC(c1ccccc1N)=O)C 33113,C1(N(C)C)CCCCC1C(N)=O.c1(C2N3C(CCC3)CNC2=O)cccc(F)c1 33114,N1(C(c2scc(C)c2)=O)CCC2(CC1)OCCC2NC(=O)CNS(N)(=O)=O 33115,C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)Nc1ncc(C)s1.C1CN1 33116,S(=O)(=O)(c1cc(F)cc(Br)c1)NCC(=O)N(c1ccc(F)cc1)CC 33117,N1(C(C(CSC)O)=O)CCC=CC1C(=O)N(CCO)CC1CC1 33118,c1(N2CCCC3(NC(c4nccnc4Cl)=O)C(C2)C3)ncc2cccnc2n1 33119,C(C)(C)(CCCCNC(=O)Cn1nccn1)NC(C(CSC(C)(C)C)NC(C)=O)=O 33120,c1(C(N2CC(NC(c3c(C)ccc(C)c3)=O)C(F)C2)=O)nn(C)c2c1CCCC2 33121,c1(CC(=O)N(CCNC(C)=O)C(C)C)cncnc1 33122,c1(CN2CC(F)(C(=O)NC3CCCN(C)C3)C2)ccc(F)cc1O 33123,C1(NC(N2CCC(C)(C)C2)=O)CCCN(C(C)(C)C)C1=O 33124,N1(C(CCC=C)=O)CCc2ccccc2C1CCNC(c1cnc(Cl)s1)=O 33125,N1(C(C(COC)C)=O)CC(NC(c2cc(=O)n(C)o2)=O)CC12CCCCC2 33126,C1(C2CC2)(CNC(CCCNC(C)=O)=O)CCN(C(=O)C2=C(C)OCC2)C1 33127,C=CCN=C(NCC1COC(C)(C)O1)N1CCCC(C(C)(C)C)C1 33128,c1(NC(C(CNC(c2cnc(C)nc2)=O)O)=O)cccnc1NC(C)=O 33129,CCC(O)C(C)C(=O)NC1CCC(CNC(c2c(C)noc2C)=O)C1 33130,N1(C(c2c(CC)csc2)=O)CCCC(N(C(=O)CC2CCOC2=O)C)C1 33131,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C(=O)Cc1ccn(C(F)F)n1)C 33132,Cc1cncc(NC(=O)CCNC(c2cc(C3CC3)on2)=O)c1 33133,CCC(C)(C(=O)N1CC(O)(CCNC(=O)Cc2ncc(F)cc2F)C1)C(N)=O 33134,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(N)=O)CCC1=O 33135,N1(C(C(C(C)C)NC=O)=O)CCC2(CCN(C(c3ccc(O)c(N)n3)=O)C2)C1 33136,c1(C(C)Nc2cc(Nc3nccn3C)nc(C(F)(F)F)n2)nc2ncc(Br)cn2n1 33137,C1(C(N2CC(C(C)NC(CCC#C)=O)C2)=O)CC(F)C(=O)N1 33138,C1(CNC(c2ccc(Cl)c(F)c2)=O)CCC2(CCC2)CN1C(=O)C(F)n1ccnc1 33139,c1(CC)nnsc1C(=O)NCC(F)CNC(c1cn(CCF)nn1)=O 33140,c1(C2C(C(CO)N(C(=O)CCCOC(F)(F)F)C)C2)cccc(C#N)c1 33141,C1(CCNC(c2cscc2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33142,c1(C(N2C3CC(OC)(C3)C2)=O)cccc2ccn(C)c12 33143,Cc1cc(Cl)nc(Cl)c1NCC1CC(C)CCN1C(=O)OC(C)(C)C 33144,C(=O)(CCCCCSCC)NCC1C(CC)CCN1C(=O)CCN1CCCC1=O 33145,C12CCCCCC1C(=O)N2.C(=O)(C(F)(F)CN(C)C)NC(c1c(C)ncs1)C 33146,CCCC(C#N)NC(C12CC(NC(=O)CCC3CCC3)(C1)C2)=O 33147,C1(C(=O)NCC(C)N(C(c2ccnn2C(C)C)=O)CC)CCCC(C(C)C)C1 33148,C(c1ccoc1)=CC(N1CCC(NC(=O)C(Cl)=CCl)C1)=O 33149,C1(NC(COC(CC)(C)C)=O)CC(CNC(=O)Cc2nccn2C)(CO)C1 33150,N1(C(Cc2cnc(C)s2)=O)CCCN(C(=O)CCC(CF)CF)C(C)C1 33151,c1(N2CC(C)C(N(C)C)CC2)nccc(=NCCC2CCN(CC(F)(F)F)CC2)[nH]1 33152,N1(C(CCCCC)=O)CC(CNC(C2CCC2C#N)=O)C2(CCC2)C1 33153,c1(C(C)OCC=C)nccc(OC(C2(NCc3ccccc3F)CCC2)=O)n1 33154,c1(C(=O)NCC2N(C(C)=O)CC(OC)C2)cnc2sccc2c1 33155,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)NC(CCN(CC)CC)=O 33156,N1(C(C(CC)N2CCCC2=O)=O)CCC(CF)(NC(=O)C(SC)SC)C1 33157,C#CCCC(O)C(=O)NCCCN(CCCCNC(C1(C(=O)NO)CC12CC2)=O)C 33158,C1(C(=O)NCc2c(C(=O)OCC)scc2)CCCC2(CCC1)OCCO2 33159,N1(C(c2ncccc2C)C(CCCC=C)=O)CC2CC3CC2C1C3O 33160,C1(CNC(c2cnn[nH]2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33161,CC1CC(C(=O)N2CCSC2c2ccccc2)=NO1.C(=O)(C#CC1(C)CC1)C1(N)CC1 33162,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33163,C1(C(N(C)C)=O)C=CCN1C(=O)CCCNC(=O)CC1CCCN1C 33164,c1(COC(=O)C=CC(=O)N(C(C2(C)CC2)C)CCN(C)C)ccccc1 33165,c1(C(=O)OCC)ccc(NC2CCN(C(=O)Cc3cccc(F)c3)C2)nc1C 33166,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)CCC3(C)CC3(F)F)C2C1 33167,Cc1cccc(OCC(=O)NC2CC(C)CN(C(c3cncs3)=O)C2)c1C 33168,Cc1ccc(CNC(C2C(O)CCN2C(C2CCC(C)(C)OC2)=O)=O)c(O)n1 33169,N1(C(C(C#N)C2CC2)=O)CCOC2CN(C(c3c(F)cccc3F)=O)CC12 33170,N#CCS(=O)c1ccc(C(=O)NC2(CNC(=O)CC3CC3(Cl)Cl)CCCC2)cc1 33171,c1(NC(N2C3(c4cn(C5C(C)CCCC5)nn4)CC(C2)C3)=O)cc(F)ccc1N 33172,C(=O)(CC(C(F)F)NC(c1conc1C)=O)N1CCC(O)(CC)C1 33173,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33174,N1(C(C(C)=C2CC2)=O)CC(N(C(=O)Cc2c[nH]nc2C)C)C(C)(C)C1 33175,N1(C(c2cc(C)[nH]c2C)=O)C2CCC1CN(C(c1cc(C3CCCC3)no1)=O)C2 33176,CC1=C(C)CC(C(=O)NCC2COCCN2C(c2csc(C)c2C2CC2)=O)CC1 33177,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33178,c1(C(=O)NC2CC(NC(c3coc(Br)n3)=O)C2)ccc(-n2ccnc2)cc1 33179,c1(COCC)nc(C(=O)NC(CNC(c2ccc(Cl)o2)=O)CO)cs1 33180,c1(NC(C2CN(C(=O)C=Cc3ccco3)CCS2)=O)c[nH]c2cccc(Br)c12 33181,Cc1ncnc(C(N2CCC(C)(NC(c3cccc(Br)c3)=O)C2)=O)c1C 33182,C(C(C)C(C)C(=O)NCC(C(C)(C)C)NC(=O)CC(C)OC)OC 33183,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCOC)C1 33184,C1(O)(CNC(C(C2CC2)SC)=O)CCN(C(=O)CC2C=CCCC2)C1 33185,c1(C(N2CC3C(NC(c4c(Cl)ccc(C)c4)=O)(CC3)C2)=O)c(N)ccc(F)c1C 33186,C1(C(=O)NC(CC)(CNC(c2n[nH]c(C)c2N)=O)CC)CCC2CC2CC1 33187,C12(C(=O)C(N(CC(C)C(C)C)C)=O)CN(C(c3ccccc3)=O)CC1S(=O)(=O)C2.CO 33188,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33189,C1(NC(COCCC=C)=O)CC2CC(C1)N(C(C1CC(C(C)=O)C1(C)C)=O)C2 33190,C(=O)(C1=CCOCC1)N(C)CCNC(C1CC(=C2CC2)C1)=O 33191,C1(CN(C(C2CCN(C(C)=O)C2)=O)CC)CCCN(C(c2cscc2C#N)=O)C1 33192,C1(NC(c2cnc(C(C)C)[nH]2)=O)(CO)CCCN(C(=O)CSc2nncs2)C1 33193,C1(C(=O)NCC(C)CNC(c2ccc(N3CC=CC3)cc2)=O)CC(=O)N(O)C1 33194,Cc1ccc(C=CC(N2CC(C3(NC(c4ccc(C(N)=O)s4)=O)CC3)C2)=O)cn1 33195,N1(C(C(C)CC2CCC2)=O)CCCC(CN(C)C(C2CCSCC2)=O)C1 33196,Cc1cn2cc(C(=O)NCC3CC(F)(F)CN3C(=O)C(C)N(C)C)cc(F)c2n1 33197,c1(C(=O)NCC(C)NC(c2c(OC)ncc(Br)c2)=O)cnc2ccnn2c1 33198,C(=O)(CC(O)CC(C)C)N1C2C(NC(c3nc(OC)c(C)s3)=O)C(C2)C1 33199,C1(CC#C)(C(=O)NCCC(C)NC(=O)CC(C)CN(C)C)CCCOC1 33200,C1(CC(=O)NC2CC(CC)C2)(OC)CN(C(c2cc(C3CC3)on2)=O)C1 33201,C1(CC#C)(C(=O)NC2CC2)CCCC1.C(C(C)O)CCN 33202,Cc1cc(C(=O)NCCCCCCN(C(=O)Cc2ccsc2)C)ncc1F 33203,C1(C(N2CC3C(NC(c4cccc(CC)c4)=O)C3C2)=O)NC(=O)OC1(C)C 33204,CCC(C)C(C(=O)N1CCCC1CS(C)(=O)=NC(=O)c1ccc(Br)cc1)OC(C)=O 33205,N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CC3CC2C3)=O)C(C2CC2)C1 33206,C(N=c1cc(NC)nc(C(F)(F)F)[nH]1)Cc1ccc(N(CC(F)CO)CC)cc1 33207,c1(CC2CC(C(=O)N)C2)ncc(C(=O)NCCOCCOC(C)C)[nH]1.C1CCCC1 33208,N1(C(C(OC)OC)=O)CCCC(O)(CCNC(C23CC2COC3(C)C)=O)C1 33209,c1(C(C(=O)NCCOC)N(C(C#C)C)C)cc(Br)c(OC)cc1O 33210,N1(C(CC(N)=O)=O)CCC(NC(=O)COc2cccc(F)n2)C(c2ccccc2)C1 33211,CC1=C(C(=O)NC(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)C(C)(C)CCC1 33212,c1(Cc2cn(CC(c3ccccn3)N(C)C)nn2)ccc(Cl)cc1 33213,C(=O)(CC(C)C(F)F)NCCC(C)NC(c1cccc(CCN(C)C)c1)=O 33214,Cc1ccc2c(C(=O)NC3(CCCNC(=O)C(C)CO)CC3)n[nH]c2c1 33215,c1(CNC(CC2(NC(CCc3cc(C)no3)=O)CCC2)=O)ccc(I)c(O)c1 33216,CN1CCN(C(=O)C(F)C2CCOC2)CC1C(=O)NCC1CC12CC2(F)F 33217,C(C1OCCc2sc(F)cc21)NC(c1ccc2c[nH]nc2c1)C 33218,c1(Oc2cc(CNCCn3c(C)ncc3)on2)cc(F)ccc1F 33219,c1(C(C(=O)N(CC)CCC2(C(=O)NCC(F)F)CC2)OCC)cc(F)cc(Cl)c1 33220,N1(C(C2N(C(C(CC#C)O)=O)CC=C2)=O)CCn2ccnc2C1 33221,c1(CC)nc(C(=O)NC2(C(=O)NC3CCC3CN3CC(C(N)=O)C3)CCC2)co1 33222,c1(NCC(N2CCC(C)(NC(C3C(C)CCC3)=O)C2)=O)nc2cc(O)ccc2[nH]1 33223,C1(C(=O)NC(C)CC(C)NC(c2cnc(C(C)O)s2)=O)(CC2CC2)CCOCC1 33224,C123CC(Cc4ccco4)(CN1NC2=O)C3.c1(C(C)=O)ccccc1N(C)C(C)C 33225,c1(-n2cc(-c3cccc(SC(C)=O)c3)nn2)cccc(F)c1Br 33226,C1(CC=C)(NC(=O)C(CCC)NC(N)=O)CCCN(C(=O)C=Cc2cc[nH]n2)C1 33227,CC(C)C#CC(=O)NC12CC1CN(C(c1ncn(C(C)(C)C)n1)=O)C2 33228,c1(C(=O)OCC(C)C)ccccc1CC(=O)OCC(n1cnnn1)=O 33229,N1(C(COCC(=O)NC)=O)CC(C(=O)NCC(C)(C)C)C(F)C1 33230,N#Cc1cnc(C2CC2)cc1NC(=O)C(=Cc1cccc(F)c1)F 33231,C#CCCCC(C)C(=O)NC1(C(=O)NCc2ccc3c(c2)CC3)CCCC1 33232,C1(C(=O)NC(C2CC2C(=O)N(C)CC2CCCC3CC23)C)CCOCC1(C)C 33233,CCC(CNC(=O)C(C)OCOC)N(C(=O)C=CCOC(C)=O)C 33234,c1(NC23CC(CNC(=O)OC(C)(C)C)(C2)OC3(C)C)cc(CO)ccc1[N+](=O)[O-] 33235,c1(C(CNC(C2(NC(c3cc(Cl)no3)=O)CCCC2)=O)O)cccnc1 33236,c1(C(=O)NCC(CC)NC(=O)C(C)OCCC(C)C)ccnn1CCOC 33237,c1(NC(C2(CC)CCN(C(=O)CC3CCC(=O)N3C)C2)=O)cc(F)ccc1O 33238,N1(C(C=C(COC)C)=O)CC2CN(C(=O)CC3CCCC34CC4)CCC12 33239,CC1CCCCN1CC(=O)OCCOc1ccc(Cl)cc1 33240,c1(N(C)C)ccnc(CNC2CC(C(=O)NC(C3COCC3n3cccn3)=O)C2)c1 33241,c1(CC)nn(C)c(C(=O)NCC2CCCCN2C(c2cnc(C(C)=O)s2)=O)c1Cl 33242,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1CCC1C)=O 33243,C1(C(=O)NCC(=O)NCCC)CCC2(CC2)N1C(=O)C(C)(C)OC(C)C 33244,C1(C)(N(C)C)CCN(C(C2CC(=O)CN2C(C2CN(C(N)=O)C2)=O)=O)C1 33245,C1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33246,c1(CC(=O)NCc2c(C(=O)NC(CC)CN3CCCC3)cco2)c[nH]nc1C 33247,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(C1CC1CCC)=O 33248,C1(CNC(c2n(CC)ncc2)=O)CCC(C(=O)N(CCC(F)(F)F)C)CC1 33249,c1(CC)c[nH]cc1C(=O)NC(CO)C(=O)NCCCn1cncn1 33250,CC1SCCCC1C(=O)NCCCNC(=O)COCC(F)F 33251,C(=O)(C(C)(C)NC(C)=O)N1CC(C(C(=O)NCC=CC2CC2)OC)C1 33252,CC1=NS(=O)(=O)N(C)C=C1c1ccccc1NC(=O)Cn1ccc2cc(C)ccc12 33253,c1(C(=O)NC(C)CC2CCCCN2C(=O)C=CCOC(C)(C)C)cc([N+](=O)[O-])c[nH]1 33254,C12(C(=O)NC3C(NC(C=C(CCC)CCC)=O)CCCC3)CC1CCC2(F)F 33255,Nc1ccc(F)cc1C(N1CC2CC2(CNC(=O)CCC2CCCCCC2)C1)=O 33256,C1(NC(c2coc(O)n2)=O)CC1C1CCCN(C(c2cc(F)c(F)c(F)c2)=O)C1 33257,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33258,N1(C(C(C(C)C)c2cccnc2)=O)CCN(C(=O)C(N)=O)CC(O)C1 33259,CC1CN(C(=O)CCc2cocn2)CCC1NC(=O)C(c1cnn(C)c1)C 33260,c1(-c2cccc(CNC(c3cc(Cl)ncc3C3CC3)=O)n2)ccc2c(c1)CCO2 33261,c1(C(=O)NC(C)CCNC(c2nc(Br)c[nH]2)=O)c(F)ccc(F)c1Cl 33262,c1(C(N2CC(N(C(=O)C=CC3C(C)C3(Cl)Cl)C)C2)=O)n[nH]c2c1CCCC2 33263,c1(CC)nnc(C)cc1C(=O)NCCNC(c1cn(CC(=O)NC)nn1)=O 33264,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(c2c(CC)occ2)=O)CCC1 33265,N1(C(C=CCNC(C2CCC(CC)O2)=O)=O)CCC(O)C(F)C1 33266,C1(C(=O)NCCC2CCCN2C)(NC(C(C=C)O)=O)CCCCC1 33267,N1(C(=O)Cn2cnnn2)CCc2ccccc2C(NC(c2cc(CF)on2)=O)C1 33268,c1(C(N2CCC(C)C2CNC(=O)Cc2cnsc2)=O)cnc(O)c([N+](=O)[O-])c1 33269,C(=O)(C1c2c[nH]nc2CN1C(=O)C(C)CO)NCc1c(C)cc(C)nc1 33270,C1(CC(N2CC=CC(NC(Cc3cncc(C)c3)=O)C2)=O)CC2CCC1CC2 33271,c1(N(C)Cc2c(C)ccc(Cl)c2)nc2c(c(=NCCC3CC3)[nH]1)SCC2 33272,CCC(C)C(Cc1ccccc1)N=c1cc[nH]c(C(F)(F)F)n1 33273,N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1C(=O)NC1CC1c1ccsc1 33274,CC(C)(C)CCC(=O)NC1CCC(CCNC(c2ccsc2-n2cnnn2)=O)C1 33275,c1(C(=O)NCC(C(C)C)Nc2ncc(C#N)cc2F)c(Cl)cccc1[N+](=O)[O-] 33276,Cn1ccnc1CN1CCC(CCC(=O)NCC(=O)NCc2ccnn2C)C1 33277,C1(C(=O)OC)CC(NC(C2CC(C(=O)Nc3nccnc3C)C2)=O)C1(C)C 33278,n1(CC(N2CC(CNC(=O)CC3CCOCC3)C2)=O)nnc2ccccc12 33279,C1(C(N(CCCC(=O)OC)C2CCCCC2)=O)CCCCN1C(=O)C(C)C1CC1 33280,C1(NC(C(C(C)C)SCC)=O)CC2(CCN(C(C3CCCN3N=O)=O)C2)C1 33281,Cc1nc(CC(=O)NCC(C)(C)NC(C2CC(C(F)F)C2)=O)n[nH]1 33282,C1(NC(C(C(C)NC(CC2(OC)CCC2)=O)C)=O)C2CCCC1COC2 33283,C(=O)(C(O)CC(C)(C)C)N(CCN(C(c1c(OC)c(Cl)sc1)=O)C)C(C)C 33284,C1(C(C)C)C(NC(=O)Cc2cncs2)CCN1C(C1OCCO1)=O 33285,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33286,c1(C(=O)NCC(C2CC2)NC(c2c(=O)ccn(C)c2)=O)cc2cc(Cl)cnc2[nH]1 33287,c1(C(N2CCC2)=O)c(F)ncn2cccc12.CC(C(=O)N1CC(F)C1)c1cccs1 33288,C1(C(=O)NC(C)CC2CN(C(C3CC4COCC4C3)=O)C2)CC2(C1)CC(F)(F)C2 33289,c1(CC)ccc(C=CC(=O)NCC2CCCN(C(C3(C(=O)OC)CC3)=O)C2)cc1 33290,C1(C(=O)N(C)C)(NCc2cc(C(C)=O)c(C)nc2)CCCCCCC1 33291,N1(Cc2cn(CC)nc2)CC(=O)N(Cc2c[nH]nc2C2CC2)C1=O 33292,C(=O)(C1CNC(=O)CCO1)N(C1CCCC1)C.CC(C)CCC1CCC1 33293,c1(-c2ccn(CCC)n2)nc(C(=O)NC(CC)C(=O)OC(C)(C)C)ccc1F 33294,C1(C#CC(=O)N2CCC(CF)(NC(C3CCOC3=O)=O)C2)(CC)COC1 33295,c1(CC(C)C)cccc(C(C)NC(CO)CC(c2ccc(F)cc2)O)c1F 33296,C1(CC(=O)N(C2CC(C#N)C2)CC(=O)OCNC(C#C)(C)C)CCOC1(C)C 33297,c1(C(CC)C)ccc(C(C)Nc2cc(C(F)F)no2)cc1 33298,C1(C(=O)Nc2c(C)ccc(OC)c2)C2CC(O)C(C2)N1C(c1ccnnc1O)=O 33299,C(=O)(CCCN=[N+]=[N-])N1C2(C(=O)NC3CN(CCC)C3)CC2CC1 33300,C1(C(N2C3(CN(C(C4CCCCO4)=O)C3)CC2)=O)CC2CC(O)C(C1)C2 33301,C(CCCCCN(C)C(C1CCC(CO)CC1)=O)NC(CCNC(=O)NC)=O 33302,CCCCC(CC)C(=O)N1CCC(=CCNC(C2(C3CC3)CCCO2)=O)CC1 33303,N1(C(C(CC#C)c2cn(-c3cncc(OC)n3)nn2)=O)CC(=O)NC2(CC2)C1 33304,N1(C(c2cccc(C)c2)=O)CCN(C(c2ccn(CCO)c2C)=O)C2CCC12 33305,c1(C(N(C2CN(C(C(CO)NC(C(C)C)=O)=O)C2)C)=O)ccc2c(c1)CCN2C 33306,C1(O)(C(=O)Nc2ccc(C(=O)OC)cn2)CCN(C(=O)Cn2cc(C)cn2)CC1 33307,C(=O)(CC(C)(C(F)(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33308,Cc1cc(C(=O)C(N2CCCC2C(N(C(CN(C)C)C2CC2)C)=O)=O)ccc1Cl 33309,C1(C(N(CCCN(C(c2ncc(OC)cn2)=O)C)C)=O)CS(=O)(=O)CC12CC2 33310,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33311,CC1(CCNC(c2cnn(-c3ccc(F)cc3)c2)=O)CCN(C(=O)C(Cl)=CCl)C1 33312,c1(-n2ccc(C(N(CCNC(c3cn(C)nn3)=O)CC)=O)n2)ccc(F)cc1 33313,C1(C(=O)NC2CC(C)(CC)C2)SC2(CCNCC2)c2ccccc21 33314,C(=O)(CC(C)(C(F)F)NCC)NC1C(CCCCC)C1.c12ocnc1c1cn2nn1 33315,N1(C(CC2C(CC)C2)=O)CCCC1(C)C(=O)N(CCN1CCC(C)(C)C1)CC 33316,N1(C2CCN(C(C3CC34CCOC4)=O)CC2)CCN(C2CC3CCC2C3)CC1=O 33317,C12(CNC(C=CCC)=O)CCCC1N(C(c1sc3nccn3c1C)=O)CC2 33318,C1(CC#C)CN(C(=O)COC2CN(C(=O)CSC(C)C)C2)CCO1 33319,c1(NCCN(C)CC)noc(-c2cnn(-c3cncnc3)c2)n1 33320,C(C(CC(F)(F)F)NC(=O)C1=NNC(=O)C1)NC(CC1N(C)CCCC1)=O 33321,c1(C(N2CCC(N(CCOC)C(c3cnc[nH]3)=O)C2)=O)ccc2nnn(O)c2c1 33322,N12CCC(CC1)N(C(=O)C=CC(C)C)CC=CC2=O.C(C1CCCO1)=CC=CC 33323,c1(C(CO)NC(=O)Nc2cn(CCC)nc2)cccc(C(F)(F)F)c1 33324,N1(C(C2N(CCC)CCOC2)=O)CCCCC(NC(c2cccc(CO)c2)=O)C1 33325,C(=O)(CCC(C)(C)NC(=O)CN1CC=CC1)N(CC#C)CC1CC1 33326,c1(OC)cncc(C(=O)NC(CN(C)C)C(=O)NC(C2CN(C)CCO2)C)n1 33327,C1(C(=O)NCC(O)CC2CCC2)(OC)CCN(C(C2CC(O)CN2C)=O)C1 33328,C(=O)(C#CC1CCCO1)N(CCNC(c1c(CC)cccc1)=O)C(C)C 33329,N1(C(C(C)(C)OC)=O)CC23CCCCC2(C1)CN(C(=O)CN(C1CCC1)C)C3 33330,Cc1cc(O)nnc1C(=O)NCC1(C)CCN(C(=O)CC2CCC(C)C2)CC1 33331,C(CC(C(=O)NCCNC(c1ccn(C)n1)=O)NC=O)SC.C(C)(=O)OC 33332,C1(OC)CC(CNC(c2cnn(CCO)c2)=O)N(C(=O)C=Cc2ccncn2)C1 33333,C1(CNC(c2csc(Cl)n2)=O)CN(C(C2CC2[N+](=O)[O-])=O)CC1C(F)F 33334,CCCCS(=O)(=O)CC(=O)N(C)CCN(C(C1CCCN1C1CCCC1)=O)C(C)C 33335,N1(C(C2C(C)(C)NC(=O)C2)=O)CCC2(CCCN2C(C2CC(O)C2)=O)CC1 33336,N1(c2ncc(C)c(C)n2)CC(NC(=O)C2=CCC2)CC(C)(C)C1 33337,N1(C(c2nc(C(N)=O)sc2)=O)CCC12CN(C(C1CC1(F)F)=O)C2 33338,C(=O)(CCCCC(F)F)NC(C1CCN(C(c2nccc(CC)c2)=O)C1)(C)C 33339,Cc1ccc(C)c(OCC(N2CC(O)(CNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)c1 33340,C1(CC(=O)OC)CN(C(=O)CC(=O)N(C)C)CC1C.c1(CN)cn(C)nn1 33341,Cc1ncc(C(F)(F)F)cc1C(N1CC(O)(C(C)NC(c2csc(O)n2)=O)C1)=O 33342,c1(CC)oc(C)nc1C.c12ocnc1C(=O)NC1(CC(C)C1)CNC2=O 33343,c1(C(=O)NCC2(NC(c3c(CC)nns3)=O)CCCC2)cc(C2CC2)nn1C 33344,c1(CNC(C(C)(C)NC(c2n(CC)nnc2)=O)=O)cn(CC)nc1C 33345,CCC(C(=O)NC(C)(C(=O)NCC1(C#N)CCCCC1)C1CCC1)C(F)(F)F 33346,N1(C(C(C)SC(F)(F)F)=O)CCN(C2CN(C(C34CC(Br)C3C4)=O)C2)CC1 33347,Cc1nc(C(=O)NC2CC(CCC(=O)N(CCF)CC3CC3)C2)c(C)o1 33348,C1(CNC(=O)Cn2cncn2)CCC(CNC(=O)C=CCn2cncn2)CC1 33349,Cc1nn(C2CCOCC2)cc1C(=O)NC1CCC(CNC(=O)C=CS(C)=O)C1 33350,c1(C(N2CC3CCC(NC(C=CSC)=O)(C2)C3)=O)cc(F)cc(F)c1Br 33351,CCCCCC(=O)NC12COC(CNC(C3(C)CCC(=O)N3)=O)(C1)C2 33352,N1(C(C2(C)CCN(C)C2)=O)CCN(C(c2cc(Cl)c(C)s2)=O)CC(CO)C1 33353,C(=O)(C#CC1CCCO1)N1CCCC(N(C(=O)CCOC2CCCC2)CC#C)C1 33354,c1(OCC)cc([N+](=O)[O-])c(NC(c2ccc(Cl)cc2)C)cc1S(=O)(=O)NC(C)=O 33355,C(=O)(CS(=O)(=O)CC1CCCO1)NC1C(CNC(c2cn(C(C)(C)C)nc2)=O)C1 33356,C1(NC(c2cc3cnccc3[nH]2)=O)CCCC12CN(C(c1cccc(Cl)c1)=O)C2 33357,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)cc2cnccc2o1 33358,c1(OC)c(C(=O)OC(C)C(C(C)C)SC)oc2ccccc12 33359,C(CCCOC)(C(=O)N1CC(C(C)C)C1)NC(c1nn(CC)nc1C)=O 33360,c1(C(N(CC)CC2CCN(C(=O)Cn3cccc3)C2)=O)cc2cnccc2o1 33361,N(C(=NCCCCl)NCc1ncoc1-c1ccccc1Cl)CC1CC(=O)NC1 33362,C1(CC(=O)NCC(CO)NC(=O)C(C2CCCC2)C2CCCC2)CCOC1 33363,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(N(C(=O)C(c2ccccc2)F)C)CC1 33364,C1(NC(C(=O)NCC)=O)(CO)CCCN(C(c2ccccc2Cl)=O)C1 33365,c1(CC(N2C(C)CC(CNC(=O)COC3CC3)C2)=O)nc([N+](=O)[O-])n[nH]1 33366,Cc1c(Cl)cc(C(=O)OCCCC(=O)OC(C)(C)C)cc1Br 33367,CCC(C(=O)N1CC(NC(c2csc(C)c2OC)=O)C1)C(C)C 33368,C1(CC)CN(C(=O)CC(C)C(C)C)CCN1C(C1(C)CCCC1)=O 33369,C1(C(=O)NCC2CCC(NC(=O)CCCC3OCCO3)C2)C2CCC1CC2 33370,CCC(CNC(C1(C)CCCN(C(C2OCCCC2(C)C)=O)C1)=O)CC(C)C 33371,C#CC1(NC(=O)CCCC(C)NC(c2coc(C(N)=O)c2)=O)CCCCC1 33372,C1(NC(c2c(C)cn(C)n2)=O)CN(C(c2c[nH]nc2C(C)(C)C)=O)CCC1C 33373,C(=O)(C1=C(Cl)CCCC1)NC1CC(CNC(c2n(C(C)C)ncn2)=O)C12CCC2 33374,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33375,C(CC(O)CCn1cc(-c2csnc2C(F)(F)F)nn1)NC(=O)CCF 33376,CCC(C)C1C(=O)C2(CO)OCC(C(COC)C2)C(=O)N(C)CCCC(=O)N1C 33377,N1(C(C2C(C)C2)=O)CC2CC(NC(=O)C(F)(F)Cc3ccc(Br)cc3)C1C2 33378,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3SCC=CC3)=O)C2)O1 33379,C(=O)(CCc1ccc[nH]1)NCC(C)NC(=O)CCOCC1CCCC1 33380,CN=c1cc(C(=O)NC2CN(C(=O)CN3CCCCC3)CC2C)cc[nH]1 33381,c1(N(C)C)ccc(C(F)(F)C(=O)NC2CN(C(c3ncccn3)=O)CC2F)cc1 33382,N1(C2(c3cnc(C)n3C)CC2)CCN(C(=O)CC2CCC3CC3C2)CC1=O 33383,C#Cc1ccc(CCC(=O)N(C2CC2)CC2CCN2C(=O)CN2CC=CC2)cc1 33384,Cc1cc(C(=O)NCC(F)CNC(=O)C2=CCOCC2)cc(=O)n1C 33385,CC(C)(CS(N)(=O)=O)C(=O)OCC.N12CCN(C(=O)OC(C)(C)C)CCN=C1NC(=O)C2 33386,C(C(CC(C)C)C(=O)NC(C)(C(=O)NC(c1csnn1)C)C1CC1)OC 33387,C=CC(C(=O)N(C1CN(C(C2(C)C=CCC2)=O)C1)C)NC(=O)OC(C)(C)C 33388,C(N=c1nnc(C)c(C)[nH]1)c1ccc(C(OC)OC)c(F)c1 33389,N12CC(C3(CC3)C1)C(=O)NC(=O)C2.C1(C(=O)NC=O)CCNC(=O)C1.C1CC1 33390,N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(c2ccsc2Cl)=O)CC1CCO 33391,c1(N2CCN(CCOC)CC2)nc(=NCCc2cnc(C)s2)[nH]c2cc[nH]c12 33392,c1(CC(C(=O)N(C(C)CNC(=O)C(C)c2ccon2)C)C)cccc(Br)c1 33393,C(CC(C)C(=O)N(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1)CCO)=CC 33394,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33395,CC1CC(NC(=O)Cc2ccc(F)cc2)CN1C(=O)CC1CCS(=O)(=O)C1 33396,CCCC(CCCNS(C)(=O)=O)NC1CN(c2ncc(F)cn2)C1 33397,Cc1cccc(C)c1OCCCN1CCOC(CCOCCCCF)C1 33398,C(=O)(CC(CC)CC(C)C)N1C(C(=O)NC(C#C)(C)C)CC1 33399,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33400,c1(SC)nc2ncnc(N(C3CN(C(c4ccc(C(F)F)cn4)=O)C3)C)c2s1 33401,Nc1nc(C(N2CC(NC(c3cnns3)=O)C(F)C2)=O)ccc1O 33402,C(=O)(C(C)(F)CC)NCCC(=C)CNC(c1ccc(OC(C)C)nc1)=O 33403,c1(CN(CC(C)C)NCc2cnns2)nnc2n1CCOCC2 33404,c1(-c2cn(C3C(=O)NCC3)nn2)cccc(Cl)c1Cl.N12CC3(CC3C1)C2 33405,c1(C(N(CC(CC)NC(C2(C(C)C)CCC2)=O)C)=O)c(C)nc2sc(C)nn12 33406,C1(CNC(c2cc(COC)no2)=O)CCCCN(C(=O)Cc2cn(C)cn2)C1 33407,CCCC(CC)C(=O)N1CC2C(CNC(C3CCN(OC)CC3)=O)C2C1 33408,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33409,Cc1cccc(-n2nc(CC(C)C)nc2C(N)Cc2ccccn2)c1C 33410,N1(C(CSCC)=O)CCN(C(c2cnc3ccsc3c2)=O)C2CCCCC12 33411,CC1(C)CC(C(N2CCCC2)=O)CCN1C(=O)C(C1CCCCC1)F 33412,C1(NC(C(C)CC(F)(F)F)=O)C2CC3CN(C(c4cc(F)ccc4F)=O)C1C3C2 33413,CC1CCN(C(=O)CNC(=O)Cc2cnn(C)c2)CCS1 33414,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33415,CC1CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1CNC(C1(C)CCOCC1)=O 33416,c1(C(C)(C)NC(CSCC2CCN(C)C2)=O)cccc(CC(=O)OC(C)(C)C)c1 33417,c1(NCCC2(COC)CC2)ncnc(NC(CO)CC(C)C)c1C 33418,C1(C(N2CC(NC(=O)CSC3(N4CCOC4=O)CC3)C2)=O)CC2COCC2C1 33419,c1(C(=O)NC2CCCC(NC(C=C(C)c3cccs3)=O)C2)cnc(C)c(N)c1 33420,c1(OC)cnc(CN2CC(C)(CC(N3CCC(Cl)CC3)=O)C2)cn1 33421,Cc1cc(F)cc(C)c1C(=O)NC1CCC(CNC(c2ccc(CO)cc2)=O)C1 33422,c1(CCC(=O)NC2CCCC(C(=O)O)CC2)nc2ccc(Br)nc2[nH]1 33423,N1(C(c2nc(CC)oc2C)=O)CC(NC(c2cnc(C)cc2N)=O)CC12CCC2 33424,Cc1cc(C(F)F)oc1C(=O)NCC1CN(C(=O)CC(C)(C)C2CC2)C2CC12 33425,c1(C(c2nnc(C3CC3)n2N)Nc2cc(OC)ncn2)n[nH]c2c1CCCC2 33426,C1(C(=O)NCC23C(CN(C(C(C)(C)C4CCC4)=O)C2)C3)COc2ccccc2O1 33427,C#Cc1ccc(C(N2CCC2C(=O)NC2CCCC(N)C2)=O)nc1.C(C)(=O)OC 33428,C=CCCCC(=O)NCC(CC=C)NC(=O)CC1CCCC1O 33429,c1(C(=O)NC2(CO)CN(C(C3C(C)(CC)C3)=O)C2)oc2ccccc2c1C 33430,N1(C(c2cc(CC)n(C)n2)=O)CCC2CN(C(c3ccc(C(N)=O)cn3)=O)CC12 33431,C=C(C)CCC(=O)NCC(CO)NC(=O)CC(C)C 33432,C(=O)(C(C)(C)C(C)O)NCC(CNC(C(C)OC1CCCCCC1)=O)O 33433,C1(N2CCN(C3CC(O)C34CCC4)CC2)CCCC12CCCO2 33434,C(=O)(C1=CCCCO1)N1CCN(CC2CCCN(C(c3c(C)nsc3)=O)C2)CC1 33435,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33436,CC(C)(CCC(=O)N(CC(F)F)CCO)NC(=O)CC1CC=CCN1C 33437,CCCCC(N)C(=O)NCc1ccc(F)nc1F 33438,Cc1nncc(C(N2CC=C(CNC(C3CCO3)=O)CC2)=O)c1C 33439,C(CC(C)C(=O)NC1CCCCC1C(N1CCN(C)CC1)=O)OC 33440,C1(OC)CCCCCC1C(=O)NCC(c1ccc(C)nc1)(C)C 33441,c1(C(N2CC(NC(C3N(CC)CCC3)=O)C2)=O)nc2ccc(C)cn2c1N 33442,C(CC(C)(C)NC(c1ccncn1)=O)NC(C1(N(C)C)CC1)=O 33443,c1(CN2CC(NC(Cc3c(OC)cccc3)=O)C(C)C2)ccc(C)c(C)c1 33444,C=CC(CC)CC(=O)N1CC(O)(C(C)(C)CNC(C2CCCN(C)C2)=O)C1 33445,c1(C2(NCc3csnn3)CCC2)ccc(NCc2nnc(C)o2)cc1 33446,CC1(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)CC(C#N)C1 33447,c1(OC)ccc(N(C(c2cc(C)c(-c3cccnc3)s2)=O)Cc2nn[nH]n2)cc1C 33448,C1(C(N2C(C(C)NC(=O)CC3CC(F)C3)CCC2)=O)CCC(C)(C)O1 33449,C1(NC(C2C(OC(C)=O)C2)=O)CCCN(C(=O)CC2(C)CCOCC2)CC1 33450,c1(C(N(C)CCn2cc(COC3CCCC3)nn2)=O)cc(C(=O)O)ccn1 33451,C1(C2CCCC2)(Nc2nccc(N3C(C)CC(CO)C3)n2)CC1 33452,C(C(=O)N1CC(C(=O)NCc2cnc(CN3CCCC3)o2)(CO)C1)(C(C)(C)C)OC 33453,C(=O)(C1=NOC2(C1)CN(C(=O)OC)C2)NCC=C(C)Cl 33454,c1(NC(C)Cc2ccoc2)ccc(S(=O)(=O)NC2CC3CCC(C2)N3C)cc1F 33455,c1(C(N(CCCN(C(C(CSC)O)=O)C)C)=O)ccc2c(c1)CC(=O)NC2 33456,CN1CCN(c2cc(O)ncn2)CC1CNC(=O)CCCn1c(O)nnc1O 33457,C1(NC(c2n(C=C)ncc2)=O)CN(C(c2cncnc2C)=O)C2(CCC2)C1 33458,C1(CSCC)CCCC(NC(=O)Cn2cc(-c3cncc(Cl)c3)nn2)C1 33459,N1(C(=O)NC)CC(NC(=O)NC2CN(C(=O)C=C(CC)CC)CC2C)NC1=O 33460,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33461,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33462,c1(OCC(=O)NCC2CN(C(=O)CCc3cc[nH]n3)CCO2)ccc(Cl)c(F)c1 33463,c1(N2CCC(NC(C3(C)ON=C(C)C3)=O)C2)nc(C)c(C#N)cc1Cl 33464,c12ccc3[nH]c(cc3c1)CNC2.c1(N(C)C(C2(C(=O)O)CC2)=O)ncc(F)cn1 33465,N1(C(C)C)CC(C(=O)NC2CC(CCNC(C3CCC(=O)N3)=O)C2)CC1=O 33466,c1(C(N2C(C)CC(NC(=O)CNc3ncccn3)CC2)=O)c[nH]c2cccnc12 33467,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33468,CCCC(CC)C(=O)NCc1cccc(C(=O)NCC2(C(=O)NC)CC2)n1 33469,N1(C(CC2CCN(C)C2)=O)CCCC2(CCCN2C(=O)C=Cc2cccnc2)C1 33470,N1(CC(=O)NC(c2nc(C)on2)C)CCCC1(C)C 33471,CC(C)(C)C(C(=O)NC1CC(NC(=O)Cc2nc(C(F)F)cs2)C1)c1ccccc1 33472,CC1CN(C(=O)C(F)OC(F)(F)F)CC1NC(c1ccc(F)o1)=O 33473,CNS(=O)(=O)NCC(=O)NCC1CC1NC(C1CCOC1C)=O 33474,c1(NC(C)=O)ccnc(C(N2CC(CO)(NC(C3CCC4CC34)=O)C2)=O)c1 33475,C1(CC(N2C(CNC(c3c(C)scn3)=O)CC(O)C2)=O)CCC(=O)NC1=O 33476,C1(C(=O)NCC2(COC)CN(C(C(C=C)C)=O)C2)CCC2(CCC2)C1 33477,C(=O)(CS(=O)(=O)CC1CCCO1)NCc1ccc(CNC(COCC)=O)cc1 33478,N1(C(C2(CNC(c3cc(C)sn3)=O)CCC2)=O)CC(C)(C)OC(C)(C)C1 33479,Cc1cnc2c(C(=O)NCC(CO)NC(C3CC34CCCCC4)=O)cnn2c1 33480,CS(=O)C=CC(=O)NCCC1(C(=O)Nc2cccc(-c3cccs3)n2)CCCC1 33481,c1(C(N2CC(O)(CNC(C(c3ccc(Cl)s3)C)=O)C2)=O)ccc(N)o1 33482,CC1Cc2cccc(C(=O)NC3CCCCC3)c2O1.c12nccnc1NC2=O 33483,c1(-c2nc3nn2CC3)cncc2nc[nH]c12.c1(OC)ccc(Br)cc1SC 33484,c1(NCC)ccc(C(=O)NCc2nccn2C)cc1.c12cncc(c1)NC2=O 33485,c1(C(N2C(C)C(=O)NCC(OC)C(CCC)C2CC)=O)ncncc1C 33486,C1(C(=O)NCC2C(CCC)CCC2)(NC(=O)CC2CC(C(=O)OC)C2)CC(F)(F)C1 33487,S(=O)(=O)(c1ccn(C)n1)N(C)CC1CN(C(c2cc(C)nc(C)c2)=O)C1 33488,C(c1cccc(F)c1Cl)=CC(=O)NCCCCCNC(Cc1cn(C)nn1)=O 33489,c1(CC(C2CC2)NC(CCC(CCOCC)C)=O)cc(C)ccc1C 33490,c1(C(=O)NC23CC(NC(c4cc(F)n[nH]4)=O)(C2)C3)cnc2ncccn12 33491,C1(O)(C(C)CNC(=O)CC(C)c2ccco2)CCN(C(C2CC(O)C2)=O)C1 33492,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33493,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33494,c1(OC)c(C(=O)NC2COCC2NC(=O)Cn2nc(C)nc2C)ncnc1C 33495,Cc1cccc(Br)c1CN1CC(F)CC1C(=O)NC(CO)C1CC1 33496,c1(NC)ccc2nc(C3CCCN3C(=O)C(N)C(C)(C)c3ccccc3)[nH]c2c1 33497,Cc1cccc2c1OCCN(C(=O)C(C)(N)CC(C)C)C2 33498,CCCS(=O)(=O)C(C)C(=O)NCC1CCN(C(c2cc[nH]n2)=O)CC1C1CC1 33499,C1(CNC(CC2(CC=C)CCCC2)=O)CC2(C1)CN(C(=O)Cc1cc(C)on1)C2 33500,c1(C(=O)NCCN(C(=O)Cc2cncs2)C(C)C)cc(C2CC2)nn1C 33501,c1(CC(N2CCC(Cc3cn(-c4ccccc4)nn3)C2)=O)ncc(Cl)s1 33502,N1(C(C2C(CC)OCC2)=O)CCC(F)(CNC(C23CCC(C2)C3)=O)CC1 33503,CC(CC(F)(F)F)C(C(=O)NCC1CCCO1)N1CCCC1CCCO 33504,C=CC1(C(=O)NCC(=O)NC(C)(C)C)CCN(C(=O)CC2CC=CCC2)C1 33505,C1(NC(CC2(OC)CCC2)=O)CCCCCC1NC(c1ccc(N)c(SC)c1)=O 33506,C1(COC)(CNC(=O)COC(C)C)CCN(C(=O)CNc2ccncc2)CC1 33507,c1(C(=O)NC(c2cccnc2)C(=O)NCC2(OC)CC2)cnc(C2CC2)o1 33508,Cc1ncc(CC(=O)NCC(C2CC2)NC(=O)C(C)N2CCC2)[nH]1 33509,c1(NC)ccc(C(F)(F)F)cc1C(N1CC(NC(C2COC(C)CO2)=O)C1)=O 33510,C(=O)(N=c1cc2ccccn2[nH]1)c1c(NC(C(CC(C)C)N(C)C)=O)c[nH]n1 33511,c12ccc(cn1)CC(=O)N2.C1(C(=O)OC)CCN(C(C2CC2(C)C)=O)C1 33512,c1(N(C2CN(C(=O)COC(F)F)C2)C)cnoc1C1CC1 33513,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(C)O)CC1c1cn[nH]c1 33514,Cc1cc(C(=O)NCC(C)(CO)NC(=O)CCc2cc(Cl)no2)ccc1Cl 33515,C1(OC)(CNC(=O)CCCSC)CN(C(=O)Cc2ccc(C)o2)C1 33516,c1(Cc2c(C)nc(F)cc2)c(C(=O)NCc2ncc(Br)nn2)[nH]c2ccccc12 33517,c1(C(=O)OC)nn2c(c1NC(=O)NC1(Cc3ccc(Cl)cc3)CC1)CCC2 33518,c1(CCC(=O)NCC(C)(C)NC(C(C)n2ccnc2)=O)ccncn1 33519,CN1C(=O)CCC(NC(=O)C(CO)NC(c2csc(C#N)c2)=O)C1=O 33520,Cc1nn(C)c(C)c1C(N1CC2CC1(CNC(C1(CO)CCCCC1)=O)C2)=O 33521,C1(CCNC(c2cc(C)on2)=O)CCN(C(C2CCCN2C=O)=O)CC1(F)F 33522,C1(C(C)=O)C(C(=O)NCCN(C(=O)CCSC(F)(F)F)CC(C)O)C1(C)C 33523,N1(C(C(CCC)OC)=O)CC(CC(N2CC3(C2)CC3(F)F)=O)C2(CC2)C1 33524,Cc1ccnc(C)c1CNC(=O)C(C)(CC1CCC1)NC(C1COCOC1)=O 33525,C1(CC)CN(C(C2CCCC2CNC(=O)C(F)n2ccnc2)=O)CC(=O)N1 33526,c1(CSC)cccnc1C(N1CCCC(CNC(C2CC(OC(F)F)C2)=O)C1)=O 33527,S(=O)(=O)(c1cccnc1N1CCC(NC2CCCOC2C2CC2)C1)OC(C)(C)C 33528,CCCCC(F)C(=O)NC1CCC(NC(c2c[nH]ccc2=O)=O)C1 33529,CCC(C)(C)C(=O)C(=O)N1CC(=O)NCC1C(=O)Nc1cc2n(n1)CCO2 33530,c1(C(=O)NC2C(CC(=O)NCc3c(C)nn[nH]3)CCCC2)cn(C)c(=O)cn1 33531,c1(C(=O)NC(C)(CNC(C2CCC(=O)N2)=O)C2CC2)cc2ccccn2n1 33532,C1(NC(c2nc(C)sc2)=O)CCN(C(c2ccc(O)c(OC(F)(F)F)c2)=O)CC1O 33533,c1(C(C)C)cccc(NC(c2cc(CNC(=O)CC3CC=CCC3)no2)=O)c1 33534,C(=O)(CCCC1CCCO1)NC(C)CCNCC(C)N(C)CC 33535,C1(OC)CCCC(CNC(=O)C=CCN(C(=O)Cn2cncn2)C)C1 33536,C1(C(=O)NCC2(NC(c3cncc(-c4ccccc4)c3)=O)CC2)CCCS1(=O)=O 33537,C(=O)(C(O)C(F)(F)F)N1CC(C(=O)Nc2nscc2C#N)(CC)C1 33538,CC1COCCCN1C(=O)CSCCNC(c1cccc(F)c1F)=O 33539,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33540,c1(C(=O)NC2(CNC(C3CC3F)=O)CC2)cccc(-n2cc(CN(C)C)nn2)c1 33541,c1(C(N(C)CCC2CCN(C(C3CCCN3C)=O)CC2)=O)cc(O)c(O)c(O)c1 33542,c1(C(N(C)CC2N(C(c3c(C)ncnc3)=O)CCCC2)=O)cc2n(c1)CCSC2 33543,C1(c2cccn2C2CCCCC2)(NC(CC)C=CCSC)CCN2CCCCC12 33544,C1(CC(=O)NC2(COC)CCN(C(C3(O)CCCOC3)=O)C2)CCC(C)(C)CC1 33545,c1(CC(=O)NC(CC)(C)CNC(C2CC(F)(F)C2)=O)ccc(Cl)c(C)c1 33546,N1(C(CCC(=C)C)=O)CCN(C(=O)C(F)c2cnc[nH]2)C(CCC(F)(F)F)C1 33547,c1(C(=O)NC2C=CC=C2)cnc(CO)[nH]c1=N 33548,c1(C(=O)NCC2CN(C(=O)CCc3cncs3)C2)cccc2cnccc12 33549,C#Cc1cc(C(=O)NCC(C)CNC(C2CC[Si](C)(C)CC2)=O)cc(F)c1 33550,N(C(=NCCNC1CCOC1)NCCOc1ncccc1Cl)N1C(C)CCC1 33551,C1(n2c(-c3n(CC)ncc3C)ncc2)CCC(F)(F)CC1 33552,c12sc(nc1Cl)NC(=O)C2N1CCCC1CCN(C)C.CCC.OC 33553,c1(NNC(C(Cc2c(OC)ccc(OC)c2)O)=O)nc(C)nc2scc(SC)c12 33554,C1(N(C)C(=O)NC(C)(C)C)COCCC1NC(=O)C=C.c1cccnc1-n1nccn1 33555,c1(NC(C(N(CCCCOCC(N)=O)C(=O)OC(C)(C)C)C2CC2)=O)ccc(Cl)o1 33556,C=C1CCN2C(C1)C2=O.c1(C)ccc(C)c(C)n1.C1(=O)C(COC)N1.OC 33557,Cc1ccc(C(=O)NC(C)C(C)NC(c2cc(C(=O)OC)sc2C)=O)c(O)n1 33558,c1(CC)cccc(CC)c1C(N1CC(CO)(NC(=O)C(C)C2CCCC2)C1)=O 33559,c1(C(N(CCNC(CC=C)=O)C(C)C)=O)cnc(Br)c(N)n1 33560,N1(C(=O)NC(C2CCC2)C)CC2(CNC(=O)C2)C1 33561,c1(CC(=O)NCC(Cn2cc(CC(C)O)nn2)OC)cc(Cl)cc2c1OCC2 33562,CC1(C)OCCOC1C(=O)NCCC1(O)CN(C(=O)Cn2cncn2)C1 33563,N1(C(c2cc(C)[nH]c2C)=O)CCN(C(c2csc(C)n2)=O)C2COCC12 33564,N1(C(C(C)Sc2ccncc2)=O)CC(NC(=O)CC(C)(C)C)CCC1C 33565,C1(CN(CCOC)C(C)C)CN(C2CCOCC2)C(=O)O1 33566,C1(C)(C(=O)NCC(=C)Cl)CCCN(C(=O)C(C)P(C)(C)=O)C1 33567,CN1CCOCC1C(=O)NCCOCCCN(C)C(c1cc(C2CC2)no1)=O 33568,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCCN(C)C 33569,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)CN1CCN(C)CC1 33570,c1(CN(C)CCc2cn(CCOC3CCCCO3)nn2)cc(F)cnc1O 33571,C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1)=O)NC(C(CC)CC)C 33572,C1(NC(C(C)CNC(=O)C2=COCC2)=O)CCC(C2CCC2)CC1 33573,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)O)CCCCC12CC2 33574,N1(C(C(C)C#N)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33575,c1(C(C(=O)NC2C=CC(CNC(C(COC)OC)=O)C2)(C)C)cccc(O)c1.CC 33576,c1(SC)cc(C)c(C(N2CCC(CF)(NC(c3cnsc3)=O)C2)=O)s1 33577,c1(CNC(C2(CC(C)C)CC2)=O)ccc(C(C)NC(C2C(F)(F)C23CC3)=O)cc1 33578,c1(C(=O)NCCNC(CC2CCN(C)C2)=O)cc(C#N)c(Br)s1 33579,CC1CCN(C(=O)CC2CCC(CC(F)(F)F)CC2)C1CNC(c1cc[nH]n1)=O 33580,N1(CC(=O)N(CCN(C(CC2C(CC)C2)=O)C)C(C)C)CCNC(=O)C1 33581,C1(COC)(CNC(=O)Cc2c[nH]nc2O)CCCN1C(C1CNC(=O)N1)=O 33582,c1(N(C(=O)Cn2nccc2C)CC)c[nH]c2nccc-2c1.C1(S)CCCCN1C(C)=O 33583,c1(OC)ccc(O)c(C(c2nnnn2-c2ccccc2F)NCCC(C)F)c1 33584,Cc1c(C(=O)NCC2CCN(C(c3cnc(Cl)s3)=O)C(C)C2)nc2sccn12 33585,C(CCC(C)N(C(=O)C(N1CCOC1=O)C)C(C)C)NC(C(C)S)=O.Cc1nccs1 33586,Cc1nnc2n1C(C(=O)N1CCN(C(=O)CC3CC4(CCC4)C3)C(C)C1)CC2 33587,N#Cc1cnn(C2CCN(C(=O)CCSc3ccc(Cl)cc3)C2)c1 33588,FCCN=C(NCC1CCCO1)N1CCCCC(=NC(=O)C2CCN2C2CC2)N1 33589,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33590,c1(OC(C)C(N2CCC(C)(CNC(C3CCOC3)=O)C2)=O)cc(Cl)cc(Cl)c1 33591,O=C1NCCCCC1C(=O)NCc1ccc(C(N2CCC23CC(O)C3)=O)s1 33592,C1(CC(N2CCC(NC(=O)CC3CC=CC3)(CF)C2)=O)CN2CCN1CC2 33593,C=CCCC(C(=O)NC1(CC=C)CC1)NC(c1cc(C)n(CC)n1)=O 33594,N1(C(c2ncc(OCC)nc2)=O)CCCC(N(C(=O)Cc2csc(C)n2)C)CC1 33595,C(C(=O)N1CC(CC(=O)NC2CC(N(C)C)C2)C1)(C1CCOC1)OCC 33596,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33597,C(CCCC(=O)NC1(C)CCN(C(=O)C2=COCC2)C1)OCC 33598,c1(C(N2CCCC(C)(CNC(C(CC)F)=O)C2)=O)ncccc1S(=O)(=O)CC 33599,N1(C(c2ccc(C(C)C)o2)=O)CCC2(CC1)CC2NC(=O)C(O)CN1CCCC1 33600,c1(NCC2C(C)(C)CN(C(C3(O)CCSC3)=O)C2)nc2c(F)cc(Cl)cc2s1 33601,N1(C(C(c2ccccc2O)OC)=O)CCC(CO)(NC(=O)CCSC(F)(F)F)CC1 33602,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33603,Cc1cc(Cl)c(Cl)cc1CN1CCC2(CC2C(N2CCC(C3CC3)C2)=O)C1 33604,N1(C(c2cc(CC(C)C)[nH]n2)=O)CCCOC(CNC(=O)C=CC(N)=O)C1 33605,c1(OCC=C)cc(Cl)ccc1C(=O)NCC1(CO)CCN(C(=O)C(C)OC)C1 33606,C1(COC)CNC(=O)CN1C(c1cc(CNC(C2CCC(C3CC3)C2)=O)cs1)=O 33607,C(CC(CC)C(=O)N(C)CCN(C(=O)C=CSCc1ccco1)C)=CC 33608,C1(CNC(C2CCC(CCC)O2)=O)CC2CCC(C1)N2C(C1COC(=O)N1)=O 33609,N1(C(C2CC23CCOCC3)=O)CC2(CCN(C(C3CC34CCC4)=O)CC2)C1 33610,C12(CNC(c3cncc(NC)c3)=O)CCCC1N(C(c1ccsc1Cl)=O)CCC2 33611,c1(OC)ccc(CC(N2CC3CC3(CNC(=O)CN3CCOC3=O)C2)=O)cc1 33612,O([Si](C)(C)C(C)(C)C)CCO.C(CCCO)N(c1nccs1)C 33613,C#CC1CCCCN1C(C1OCCC1NC(=O)CN(CC(C)(C)C)C)=O 33614,CCC(CC(=O)N1CCCC(C(=O)NCC(Cl)Cl)C1)CC(C)C 33615,C1(C(N(CC(CC)(C)OC)C)=O)(C(C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 33616,C1(CC(N2CCC(NC(COCCN(C)C)=O)(CO)C2)=O)CC2CCC1CC2 33617,c1(C(N2CC(NC(CS(C)(=O)=O)=O)C(F)(F)C2)=O)ccc2nc(Br)sc2c1 33618,S(=O)(=O)(c1ccc(Br)cc1Cl)NC(c1cn(CC(=O)N(C)C)nn1)=O 33619,N1(C(C(C)OCCCC)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33620,C1(NC(C(c2ccnn2C)NC(C2=C(C)CC2)=O)=O)CCCCCC1CO 33621,c1(CC)[nH]ccc1C(=O)NCC1(NC(=O)C(c2ccccc2)F)CCCC1 33622,N1(C(C(C2CCOC2)N(CC)CC)C(=O)NCC(C)C)CCC(S(N)(=O)=O)C1 33623,c1(NCC(=C)C)cc([N+](=O)[O-])cc(CN2C(=O)CN(CC)C2=O)c1O 33624,C1(C)(CNC(C(c2ccccc2)C)=O)CC(NC(=O)C(N2CCCC2)C2CC2)C1 33625,CCC(C(=O)NCC1(C)CN(C(c2[nH]c(=N)sc2CC)=O)CCO1)C(C)(F)F 33626,N1(C(c2ccc(F)c(C)n2)C(=O)NCC)CCOCC(C)(F)C1 33627,c1(C(N2CC(OCCNC(c3ccc(C#C)nc3)=O)C2)=O)cc(Cl)c(OC)cc1Cl 33628,C1(NC(=O)CCCF)CCC2(CCN(C(c3cnn4c3CC(F)(F)C4)=O)C2)C1 33629,c1(C(=O)NCC(CN(C(c2c(C(=O)OC)scc2)=O)C)C)ncc(Cl)nc1Cl 33630,Cc1nn(C(C)C)cc1C(=O)NC(C)(C)CNC(C1CCS1(=O)=O)=O 33631,O=C(CCS(=O)(=O)Nc1cccc(F)c1)N1C2CCCC1CC2 33632,Cc1cc(C(=O)N(C)CCNC(=O)CC(C(N)=O)NC(=O)C2CC2)ccc1O 33633,C(C)(C(CO)NC(c1ncoc1C(C)C)=O)NC(C(c1ccccc1)OC)=O 33634,C(=O)(C(F)(F)CC)N(CC(=O)NCCCN(CCC)CCC)C 33635,c1(C(=O)NC2C(C)=NN(C(=O)C(C)S(C)(=O)=O)C2)c(C)ccc(C)c1Cl 33636,c1(C(N2CCN(C(C=C(CC)CC)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33637,CC1CCN(C(=O)C=C(Cl)Cl)C1C(=O)NCc1ccc(Sc2ccccc2)o1 33638,N1(C(C(C2CC2)OC)=O)CC2CC3CC2C1C3NC(c1cnn2c1CCC2)=O 33639,CC1CCC(c2cn(CCCC(=O)OC(F)(F)F)nn2)CC1.C[Si](C)(C)C 33640,c1(C(N(CC)CC2CCOC2)=O)n[nH]cc1CNC(=O)C(C)=CC1CC1 33641,C(=O)(CCCCC(F)(F)F)NCCN(C(=O)CCc1ccc(CC(N)=O)cc1)C 33642,Cc1ccc(C=NOCC(N2CCN(C)CC2C2CC2)=O)cc1 33643,Cc1c(N)ccc(C(=O)NCCN(C(c2csc(Cl)n2)=O)C2CC2)c1C 33644,N1(CC)CC2CC1CN2C(C1CCCN(C(c2ccnnc2O)=O)C1)=O 33645,N1(C(C(CCC)CC)=O)CC2(CNC(=O)C(F)OC)CC1CCO2 33646,CC1CC(Br)CCN1c1ccccc1-c1csnn1 33647,c1(NC(c2ccc(CSC)o2)c2nnnn2C(C)(C)C)cncc(OC)c1 33648,C(c1ccc(OC)cn1)=CC(N1CCC(N(C(=O)CC2(C)CC2(Cl)Cl)CC)C1)=O 33649,CCCC(C(=O)N(CC(C)NC(C1(n2ccnc2)CCCC1)=O)C)C(C)C 33650,CCCC(C(=O)OC)C(=O)NC1CCC(CNC(=O)CC=CC(C)(C)C)CC1 33651,C1(CNC(c2c(C)oc(Cl)n2)=O)C2CCC(C2)N1C(C1CC1c1ccccn1)=O 33652,C1(N(C(=O)CCc2ccc(O)nc2)C)CCC2CN(C(C3CCC4CC34)=O)CC12 33653,N=c1[nH]cncc1C(=O)NCc1ccccc1CNC(=O)C1=COCC1 33654,Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(C(C)C)[nH]n3)=O)C2)c(=O)o1 33655,Cc1n[nH]c(C)c1C(C)CC(=O)NCC1(CO)CCN(C(C2(C)C=CCC2)=O)C1 33656,C(CC)(C(=O)NCc1ccc(C(=O)N(CC(C)C#N)C2CC2)s1)OCC 33657,C12CC3CCC1N3C2=O.c12sccc1C(=O)NC2.C1(OC)CC(C(=O)OC)C1 33658,C1(n2cc(CSC)nn2)CCN(C(=O)NNC(=O)c2n[nH]cc2C(F)(F)F)CC1 33659,C1(CCNC(CCN(C(=O)CC2CSCCO2)CC)=O)CC2CCC1O2 33660,CCC(CNC(C1(CC)CCN(C(C2CCOC(CC)C2)=O)CC1)=O)(CC)CC 33661,CCC(CC(=O)OCc1ccccc1)NC(=O)C(C)c1ccon1 33662,C(=O)(CCCCCNC(=O)Cc1cccc(C#N)c1)NC(c1c(C)cccn1)C 33663,C1(O)(CCNC(c2c(CC)occ2)=O)CCN(C(=O)CC2CCC(C)(C)O2)C1 33664,CC1(C)OCCOC(C(=O)NC2COCC2NC(c2cc(C3CCC3)[nH]n2)=O)C1 33665,C1(C(=O)NCCCC(C)NC(C2CCCOCC2)=O)C2CCCCCCC12 33666,c1(C(=O)OCc2ccc(C)c(C)c2C)cc2n(n1)CCN(C(=O)OC(C)(C)C)C2 33667,N1(C(c2c(OC)ccs2)C(=O)NCc2c(C)ncn2C)CC2CCCCC2C1C 33668,O=C1NCCc2cc(F)c(C(=O)NC(Cc3ccccc3)C3CC3)cc21 33669,c1(C(=O)NCC2CC(F)(CNC(=O)C=CC3CCOC3)C2)ccc2nc(S)oc2c1 33670,N1(C(C2CC(C)N(C)C2)=O)C(C)CC2CN(C(c3cocn3)=O)CC12 33671,N1(C(c2ccc(CCCCC)o2)=O)CC2C(CN(C(=O)CCn3cncn3)C)C2C1 33672,C1(NC(=O)Cn2nccn2)CC(O)CN(C(c2cccc(C=O)c2)=O)C1.C1CC1 33673,C1(CC)CN(C(c2ccc(OC)cc2)C(=O)NCCOCC2CC2)C(C)CO1 33674,Cc1nccc(C(=O)NCCCN(C)C(C2CNC(=O)N2C)=O)n1 33675,N12C(CCC13CC3)C(=O)N(C)CC2=O.C(CCC(=O)OC)OCCOC 33676,C(=O)(CCCC(=O)N1CCOCC(NC(=O)C(C)CCOC)C1)N(CC)CC 33677,C1(O)(C(N2CC(O)(CNC(C3(C)CCC(C)C3)=O)C2)=O)CCCC(C)(C)C1 33678,CC(C)C(C)C(CNC(=O)CCc1cscn1)NC(c1cnc[nH]c1=N)=O 33679,CC1OC(C)(C)OC1(C)C(N1CC2CC(NC(C3CC4(CC4)C3)=O)C1C2)=O 33680,C(CC(N)=O)(C(=O)NCC1CCC2(CC1)CC2)NC(c1cccc(C)n1)=O 33681,Cc1cc(Cl)c(CN(c2cc(F)ccc2Br)C(=O)NC(C)(C)C2CC2)cc1F 33682,C#CCC(C)(C(=O)NCC1COCC1(C)C)NC(C12CC(F)(C1)C2)=O 33683,c1(CSCC(=O)Nc2cc(OC)nc(C(F)(F)F)n2)cnc2ccc(Br)cn12 33684,c1(CC)nc(N(CC(C)SC)C)cc(=NC(C)c2cnn(C)c2)[nH]1 33685,N1(C(C2(CSC)CCC2)=O)CCC2(CCCN2C(c2cc(Cl)cs2)=O)CC1 33686,c1(N(CC(=O)N(CC)CC)C)[nH]c(=NC(C)c2ncccc2F)nc2sccc12 33687,N1(C(=O)CCCn2cc(-c3ocnc3C(=O)O)nn2)CCOC(CCO)C1 33688,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33689,c1(CNC(C2CC3(CCC3)C2)c2n(C3C(C)C3)nnn2)ccc(F)c(C)c1O 33690,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(COC)nn1)CC(F)(F)F 33691,c1(C(N2C(CNC(C3CCCN3C)=O)CC(COC)C2)=O)cc(=N)[nH]c(Cl)n1 33692,C=CCC(CC(=O)NCCC1CC(OC)C1)NC(=O)CN1CCNC1=O 33693,C(=O)(C#CC1CCCCC1)N(C)CC1COCCN1c1ncc2ccnc-2[nH]1 33694,N1(C(CC=CC)=O)Cc2ccccc2C(NC(C23CCC(CO)(CC2)CC3)=O)C1 33695,N1(C(C(CC)n2ccnc2)=O)CCN(C)C(CNC(=O)CC(C)N2CCCC2=O)C1 33696,Cc1nc(NC(C2C3CN(C(c4cnccc4N(C)C)=O)CC23)=O)ccc1[N+](=O)[O-] 33697,C1(CNC(=O)CCc2ccccc2O)CC(F)(F)CN1C(=O)Cc1c[nH]nc1O 33698,Cc1c(NCc2nnc(CO)s2)ncnc1N1C2CCC1COC2 33699,C1(OCCNC(CC=C)=O)CCN(C(=O)C(C)C=C)C1 33700,N#CCCCC(=O)NC1C=CCC(C(N2CCN(CC3CC3)CC2)=O)C1 33701,C1(CC)CCC(CNC(=O)CCN(C(=O)CC2(CSC)CC2)C)CC1 33702,C1(NC(C(C)N(C)C)=O)CC2(C1)CC(NC(c1cncc(-c3cnn(C)c3)c1)=O)C2 33703,CCC(CC(=O)N1CCN(C(=O)CCC(C)(C)OC)C(COC)C1)C(F)F 33704,C1(C(N(C)CC2CC2CF)=O)COCCN1C(c1cc(-n2cccn2)ccn1)=O 33705,N1(CC(=Cc2cnc[nH]2)C)CC2(CCC2)CC1C(=O)NC1CN(C(C)C)C1 33706,C1(OC)CC(CCNC(=O)C(F)C(C)C)N(C(C2CC(C)C2)=O)C1 33707,C1(NC(C(C)N(C)C)=O)CCCCN(C(=O)Cc2nc(C3CCCC3)n[nH]2)C1 33708,CC(C)C(C)(C)CNC(=O)C(c1ccccc1)NC(c1ncc(F)cn1)=O 33709,Cc1cncc(C(=O)NC2CCN(C(=O)C=CCN3CCOCC3)CC2O)c1C 33710,c1(OC)cccc2c1CC(C(N1CC(NC(=O)CSCC(N)=O)C(F)C1)=O)CO2 33711,C#CCC(O)C(=O)N(CC(C)O)CCNC(C1CC(=C2CCC2)C1)=O 33712,C1(NC(C(C(=O)OC)OC)=O)CC2CN(C(c3ccc(CO)nc3)=O)CC2C1 33713,N1(C(C=CC)=O)CCC2(CCN(C(c3cn(CCC#N)nc3C)=O)C2)C1 33714,N1(C(CCSCC(C)C)=O)CCC(C2(NC(c3c[nH]c(Br)c3)=O)CC2)CC1 33715,C(=O)(C(C)S(N)(=O)=O)NC1C2CN(C(c3c(C)cccn3)=O)C1C2 33716,c1(C(=O)O)ccccc1S(=O)(=O)NC1CN(c2ncnc3n[nH]c(Br)c23)CC1F 33717,C(C(C)CC(=O)N1CCOC(CN(C)C(c2c(C3CCCC3)cnn2C)=O)C1)OC 33718,C1(CNC(C2N(N=O)CCCC2)=O)CC2COCC2N1C(=O)CC1CCCC1O 33719,C(=O)(C1CCc2c[nH]nc21)NC1C(N(C(c2cncc(C#C)c2)=O)C)CCCC1 33720,N1(C(C2C(=C)CC2)=O)CCc2nc(CNC(C3CCC4C(C3)C4(F)F)=O)sc2C1 33721,C1(NC(Cc2n(C)ncc2)=O)CC2CC1CN2C(=O)Cc1ccncc1F 33722,c1(NC2(CNC(c3ccc(N)c4c3cncc4)=O)CC2)ccc(F)cc1[N+](=O)[O-] 33723,c1(C(=O)NCCN(CCC)C(c2cnc(C)cn2)=O)cc(C)nn1C1CCC1 33724,N1(C(C2C(OCC)C2)=O)CC(NC(=O)CC2CC2)CC12CCC2 33725,N1(C(C2SCCS2)=O)CCC2(CCCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)C1 33726,C1(NC(Cc2cc(C)c(F)cc2)=O)CCN(C(c2ccnn2C)=O)CC(O)C1 33727,C1(O)(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(c2cnn[nH]2)=O)C1 33728,c1(CN2C(C3(O)CN(C(=O)CC4(C5CCCO5)CC4)C3)CCC2)ccnc(Cl)c1 33729,C(=O)(C(CNC(=O)C(F)C(C)(C)O)CCC)N1CC(N(CC=C)C)C1 33730,c1(OCCN(c2ccc(-c3cn(CN)nc3)cc2)CC)c(C)cccc1F 33731,CC(C)CC(CC(=O)NC12CC(C1)N(C(C1C3COCC13)=O)C2)CC(N)=O 33732,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1C 33733,c1(C(N2CCC(COC)(CNC(=O)C(F)CC3CC3)C2)=O)cn2c(n1)CCC2 33734,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCN(C(C)=O)CC3)C2)[nH]c2c1COC2 33735,CP(C)(=O)CC(=O)NCCNC(c1cc(Cl)sc1Cl)=O 33736,N1(C(C=CC(=O)NCC(C2(O)CN(C(CCOC)=O)C2)(C)C)=O)CCCCCC1 33737,C1(N(C(=O)CSc2nnnn2C2CCCC2)C)CCC(NC(C2(C)CC2F)=O)CC1 33738,c1(-n2c(C(C)Nc3n(COC)nc(C4CCCC4)c3)nnn2)ccc(C)cc1C 33739,N1(C(CC(C)(C)OC)=O)CCC2(CNC(c3ccc(N(C)C)cn3)=O)CCCC12 33740,c1(-c2cc(C)c(O)c(C)c2)ccc2cc(C(=O)NC(C)C(F)(F)F)[nH]c2c1 33741,c1(C(N(C2CCCN(C(=O)COC(C)(C)C)C2)C)=O)cc2c(nc1N)CCC2 33742,N1(Cc2ccc(OCC)c(Br)c2)CCC2CN(c3ncc4sccc4n3)CCC12 33743,c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2)ccc(-n2cnnn2)c(OC)c1 33744,N1(C(=O)C(O)C2CCCC2)CC2(CCN(C(C3(CC4CC4)CCCO3)=O)CC2)C1 33745,C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(=O)C(c2ccccc2)O)CC1O 33746,C1(C(=O)NC2C(C)(CO)CCC2)CC1C1CN(C(=O)CNc2ncccn2)C1 33747,C(CO)(CCC(C)C)NC(C12CC(NC(C(C=C)OC)=O)(C1)C2)=O 33748,CC1CCC=C1C(=O)N1CCN(CCCNC(C2CC2Br)=O)CC1 33749,c1(CC(N2CC3(CCN3C(c3ccnc(CO)c3)=O)C2)=O)cccc([N+](=O)[O-])c1 33750,Cc1nc(O)c(C(=O)NC(C)CNC(c2ccccc2SCCO)=O)cc1Br 33751,c1(C(C)C)cc(I)ccc1NC(=O)CCn1nc(C(C)O)oc1=O 33752,N1(C(CCCC(C)=O)=O)CCN2C(=O)C(NC(=O)Cc3ccccc3F)CC2C1 33753,CC(C)(C)C(C)(O)C(=O)N1CCCN(CCNC(c2ccc([N+](=O)[O-])s2)=O)CC1 33754,c1(C(N(CCC(C)(C)NC(C(C2CC2)OC)=O)CC)=O)ccnc(OC)n1 33755,C1(NC(c2c(CCC)occ2)=O)CCCN(C(=O)COc2cnn(C)c2)CC1 33756,c1(C(N(CC(C)N(C(=O)Cn2ncc(O)nc2=O)C)C)=O)cc([N+](=O)[O-])nn1C 33757,C1(COC)(CNC(c2ccc(N)cn2)=O)CCN(C(=O)C(O)P(C)(C)=O)CC1 33758,C1(CNC(c2c(C)snn2)=O)CN(C(c2ccc(F)o2)=O)CCC12CCC2 33759,CC1(C)C2CCC(C(=O)NCc3cc(C(=O)NC4C5CCCCCC45)co3)C1C2 33760,C1(CNC(c2c(C)scc2)=O)CC(NC(c2nocc2Cl)=O)C1(C)C 33761,c1(OC)cc(NCC2CN(c3nnnn3C)CC2C)c(Br)cc1Br 33762,C(c1cccc(F)c1F)=CC(=O)N(CCC)CCNC(=O)CCC1CCCCO1 33763,CCC(C(C)C)C(C(=O)NC1CCC1)N1CCn2c(C(F)(F)F)nnc2C1 33764,C1(CCC)CN(C(=O)C(F)OC(F)(F)F)CC1CNC(=O)Cc1ccc(F)cc1 33765,C1(NC(C2CCC(C(N)=O)O2)=O)CCCN(C(=O)C=C2CCSCC2)CC1 33766,N1(C(CNC(C)=O)=O)CCN(CCN(C)C(C2CC2Cl)=O)CC1 33767,C1(C(N(CCC#C)CC)=O)CC(NC(c2coc(N(C)C)n2)=O)C12CCC2 33768,N1(C(c2cccc(C)c2)=O)CCN(C(=O)CCc2ccccc2F)CC(CO)C1 33769,C1(NC(c2ccc(SCC)cn2)=O)CCN(C(=O)COC2CC=CC2)CC1F 33770,N1(C(C=Cc2cn(C)nc2)=O)Cc2ccccc2C1CNC(c1cnnn1C)=O 33771,c1(SC)nc(N2CC3CC2CN3C(=O)C=Cc2ccccc2)c(Br)c(C)n1 33772,c1(NC(c2n(CCCSCC)nnn2)=O)cccc(Cc2ncc(Br)s2)c1C 33773,c1(OC)ccc(C(=O)NC2CC(NC(c3[nH]nnc3C)=O)C23CCC3)c(F)c1 33774,c1(C(N(CCCCCCO)CC2CC2)=O)cc2cc(Cl)cnc2[nH]1 33775,C1(CNC(CNC=O)=O)CC(O)CN1C(=O)CCN1CCOCC1 33776,n1(CCOCC)nc(COc2ccccc2C)nc1-c1occ(C)c1C 33777,N1(C(CN(CCC)C)=O)CC2CCCC2(C(=O)NC2(CC3CC3)CCC2)C1 33778,C1(C(=O)NC2CN(C(c3cc(OC)ns3)=O)CC2SC)CC(C)(C)OC1(C)C 33779,N1(C(C2CCCOCC2)=O)CCC(C2CCCN(C(C3CC(F)(F)C3)=O)C2)C1 33780,C12CCCN(C1)C(=O)C1CC1(Cl)C(=O)NCC2.c1(C(C)=O)[nH]nnc1C(=O)NC 33781,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 33782,C1(CCOC)(NC(c2ccon2)=O)CCN(C(C2CCOC2C)=O)C1 33783,C#CCCCC(C)C(=O)NC1CC(C)(CNC(c2cc(F)c(F)cc2F)=O)C1 33784,N1(C(CN(CC)Cc2ccccc2)=O)CCCCC1CN(c1cnccn1)C 33785,CCCCCC(O)CC(=O)NCCN(C(c1ccc(C)cc1F)=O)C1CC1 33786,N1(C(=O)CCC2(N3CCOCC3)CC2)CC2CCCC(N=c3cnc(F)c[nH]3)C2C1 33787,N1(C(c2cccc(N)n2)=O)CC2CCN(C(C3CCN(S(C)(=O)=O)CC3)=O)C2C1 33788,C12(CNC(c3c(C(C)C)ccs3)=O)CC1CN(C(c1cccc(F)c1)=O)C2 33789,N1(C(C2(OCC)CCC2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C2(CC2)C1 33790,N1(C(CCN2CCC(N(C)C)CC2)=O)CC2(CCCC2)C1 33791,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 33792,c1(N2CCC(CC(C)(C)C)C2)ccc(S(=O)(=O)NCc2cccc(CO)c2)cn1 33793,c1(N2CCC(COC)(OC)C2)nc(=NCCCC2CCOC2)[nH]c2ccsc12 33794,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 33795,C12(NC(CCOCCC)=O)CCCC1(F)CN(C(c1[nH]cnc1C#N)=O)C2 33796,N1(C(c2c(CC)nn[nH]2)=O)CCC(C)C(NC(=O)COCCOC)C1C 33797,c1(OC)cccc(C(N2CCC(N(C(=O)C=Cc3cnc[nH]3)CCO)C2)=O)c1F 33798,C1(C(=O)NCC2N(C(c3cccc(C#C)c3)=O)CCCC2)CC2CCC(C1)C2F 33799,CC1CN(C(=O)CCCOc2ccccc2)CCCN1C(=O)COCCOC 33800,C1(N(C)C)(C(=O)NCCCNC(C2(CO)CCCCC2)=O)CCCOC1 33801,C#CC1(NC(C2CN(C(C3CCCCC34CC4)=O)CC2C)=O)CCCCC1 33802,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C=CC(N)=O)C2)C1 33803,C=CC(C)(O)CC(=O)N(CC(C)O)CCNC(c1sc(C)cc1C)=O 33804,c1(OCCC)ccc(Cl)cc1C(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 33805,c1(OC(c2ccc(OC(F)(F)F)cc2Cl)=O)ccnc2cc(F)cnc12 33806,c1(OC)ccc(CNC(C(C)(C)OC)c2nnnn2CC(F)F)cc1C#N 33807,O=C1CCCC(NCC23CCC(CC2)O3)C1 33808,C1(NC(=O)NCc2cccc(-n3cc(CC(=O)O)nn3)c2)CC2(C1)CC(F)(F)C2 33809,c1(CNC(=O)NCCSC(C)C)ccc(C2COC2)cc1 33810,C1(C(N2C(C)CC(CNC(CCCNC(=O)OC)=O)C2)=O)Cc2cccnc2C1 33811,C(=O)(C(C(=O)Nc1cccc(CNC(=O)C(COC)OC)c1)C(C)C)OCC 33812,N1(C(CCC2CCCN(C(CC3C(C)(C)C3(C)C)=O)C2)=O)CCC2(CNC(=O)C2)C1 33813,C#Cc1ccc(C(=O)NCCCN(C(c2ccc(Cl)c(C)c2)=O)C2CC2)nc1 33814,c1(C(=O)NCCNC(C(F)OC)=O)c(Cl)c([N+](=O)[O-])nn1C 33815,N1(C(C2CC23CCC3)C(=O)NC(CC)C)CCc2ccc(F)c(F)c2C1 33816,C1(C(C)CNC(C2(F)CCC2)=O)CCN(C(c2ccc(O)nc2)=O)CC1 33817,C1(NC(c2c(CC=C)cccc2)=O)CCCN(Cc2cn(C)nn2)C1C 33818,CCC1=NOC(C(=O)NC2CC2NC(c2cn(CCO)nn2)=O)C1 33819,C1(NC(c2ncn(CC)n2)=O)CN(C(c2sccc2CC#N)=O)CC1C 33820,Nc1ccc(C(=O)NC(CNC(c2csc(Br)c2)=O)C2CC2)nc1F 33821,CCCCC(C(=O)NC1CC2CC1CC2C(N)=O)NC(C1CC(CCC)C1)=O 33822,c1(OC)ncnc(Cl)c1NC(C1CCCCN1C(c1ccc(C)cc1Cl)=O)=O 33823,C1(CNC(CCC(=C)C)=O)CN(C(C2CC(OC3CC3)C2)=O)CCC12CCC2 33824,C1(CNC(c2cnc(CCC)s2)=O)CC2CCC(C1)N2C(=O)CC1CCCOC1 33825,Cc1ccc(Cl)c(CNC(C23CC2CN(C(C)C)C3)=O)c1 33826,CC1(C)OCCC1(O)C(=O)NC1CCC(CNC(=O)COCC(F)(F)F)CC1 33827,c1(C2CN(C(c3c(C)csc3)=O)C(C(=O)N(C)C)C2)nc(C)n(C)n1 33828,N1(C(c2nc(C)oc2C)=O)CCCC2(C1)C(NC(=O)CCOC1CC1)CCN2C 33829,c1(C(N(C)CC2N(C(C3C(C)C3C)=O)CCCC2)=O)ccc(S(=O)CC#N)cc1 33830,CC1(NC(c2coc3c2CN(C(c2ncc[nH]2)=O)C3)=O)CN2CCC1CC2 33831,c1(CN(C(=O)C(CCc2ccccc2)C(=O)O)CC)cc(Cl)cc(Cl)c1 33832,C1(NC(C(C)OCCN(C)C)=O)CCSC12CN(C(=O)CCC1CC1(Cl)Cl)C2 33833,N1(C(C2C(C)C2C)=O)CC(CNC(c2cc(C(N)=O)c[nH]2)=O)(NS(C)(=O)=O)C1 33834,c1(C(=O)NCC(C)(C)CCNC(C2CCCC3CC23)=O)ccc2ccnn2c1 33835,Cc1c(CC(N2CCCC2C2(C(=O)NCC3CCOCC3)CC2)=O)cnn1C 33836,c1(OC)cnnc(C(=O)N(CC(O)CNC(=O)C(C)N(C)C)C)c1 33837,C1(NC(C2(CCF)CC2)=O)CCCN(C(C2(C(F)(F)F)CCOCC2)=O)CC1F 33838,N1(C(C(CC=C)C)=O)CCCC2(C1)CN(C(C1OCCOC1(C)C)=O)CCO2 33839,C(N=c1ccc(-c2ccccc2)c[nH]1)c1c(C)cc(Cl)cc1.[nH]1c(C)ncc1C 33840,C1(C(=O)NCC(C(=O)N(CC(=O)NCCC)C)(C)C)CCOC(CC)C1 33841,c1(C(=O)NC2CC(NC(CCOCCN(CC)CC)=O)C2)nn(C)cc1Br 33842,Cc1nsc(C(=O)NC(C2CCCN(C(=O)C(C)(C)c3ccsc3)C2)C)c1N 33843,CCC(C)CCC(=O)NCc1ccc(C(N2CC(OCCF)C2)=O)s1 33844,CCC1CC(=O)N1.c1(C(N2CC(CCCCO)C2)=O)ncccc1SC 33845,C1(CNC(C(C)OCC(C)C)=O)CCCN(C(c2ccc(SC3CC3)cc2)=O)C1 33846,N1(C(c2c(C)n[nH]c2)=O)CC(NC(=O)CCc2nnc(C(C)C)o2)C2CC12 33847,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CC(NC(=O)C(C)(C)CC3CCOCC3)C2)C1 33848,C=CC(C)(CC)NC(c1c[nH]nc1NC(C)=O)=O 33849,N1(C(C2(N(C(=O)CC3CCC=CCC3)C)CC2)=O)CCCC(C2CCC2)C1 33850,N1(C(CC2CC(=C)C2)=O)CC2CCC(NC(=O)Cc3cc(F)ccc3OC)(C2)C1 33851,C1(NC(C(=O)OC)=O)CCC2CCN(C(=O)Cc3ccccc3CC(C)C)C1C2 33852,c1(NC)cncc(C(=O)NCCN(C(=O)CCc2cc(Cl)no2)C2CC2)c1 33853,C1(C)(CNC(C2CC(CCC)C2)=O)CCN(C(=O)Cc2ncoc2C)CC1 33854,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(C=CC=CCC)=O)(COC)CCC1 33855,c1(N2CC3(CN(C(c4c(OC)nccc4)=O)C3)C2)ncnc2scc(C)c12 33856,C1(CNC(=O)CC2CNCCC2O)CCC=CCC1 33857,Nc1nc(Cl)ccc1C(N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1)=O 33858,N1(CC(=O)Nc2ccc(Cl)cc2)CCC2COCCC12 33859,CCC(C)(C)C(C)N(C(C)(C)C)C.C12CCCN1C(=O)OC2=O 33860,C#CCCCCCCC(=O)N(C1CC(C(=O)N(C(C)CC(C)CC)C)C1)C 33861,N1(C(c2ccc(CN(C)C)cc2)=O)C2CCC1CC(NC(c1occc1F)=O)C2 33862,C1(C(=O)NCC(=O)N(C(CCCC)C)C2CC2)CCC(C#N)CC1 33863,C1(C#N)(C(=O)NC(C)C(CO)NC(c2cccnc2CO)=O)CC1(C)C 33864,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CSc2ccncc2)CC1 33865,c1(CC(=O)NC2CC(CNC(CS(C)(=O)=O)=O)C2)ccc2nc[nH]c2c1 33866,Cc1c(C(=O)NCCC(C)(C)NC(C2CC2C(C)O)=O)cnc2ncnn12 33867,n1(C(C)C)cccc(CC(=O)NC2CN(C(=O)CCOCC3CC3)CC2C)c1=O 33868,c1(OC)ccccc1OCC(=O)NCC1CC(C)CO1.C(CSC)S 33869,O=C(C(c1cccs1)=Cc1ccc[nH]1)NCC1CCC(C(F)(F)F)O1 33870,C1(CC(=O)N(C(COC)C)C)CCN(C(=O)CC=C(Cl)Cl)C1(C)C 33871,C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NC1CCC(OC)C1 33872,c1(-c2n(-c3cn(CC)nc3)nc(CC3CC3)n2)ccc2ccccc2n1 33873,N1(C(C(C)SCC)=O)CCC2CCCC12C(=O)N(C)CC1CC(F)C1 33874,C(=O)(C(C)(CNC(=O)COCCOC)CC)N1CC(CC)OCC1 33875,N1(C(c2cnn(CCC)c2C)=O)CCC2C(C1)CN2C(C1CCC2(CC2)C1)=O 33876,c1(C(=O)NC2C(C)CCN(C(=O)C=Cc3ccccc3)C2)cc2occc2n1C 33877,CC1C(NC(C2CCCCS2(=O)=O)=O)CCCN1C(C1CCCC1)=O 33878,Cn1c(C(N2CC3CC2CN3C(=O)CCCF)=O)cc(=O)n(C)c1=O 33879,c1(C(=O)NCC2CCCN2C(C2CC(CCO)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 33880,c1(C(=O)NCC(COC)NC(c2cnnn2C(C)C)=O)cnc(Cl)n1C 33881,C(C)(C(C(C)C)NC(=O)CCCC1CC1)NC(c1n(CC#C)ccc1)=O 33882,N1(C(c2n(C)ccn2)=O)CC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 33883,C(=O)(CCC(C)CN(C)C)NCC(CO)NC(CSCC#C)=O 33884,C1(NC(C(C)OCCCCCC)=O)CCC2(CC1)CN(C(c1nccn1C)=O)C2 33885,C1(CNC(CC2(O)CN(C(c3cc(OCC)n[nH]3)=O)C2)=O)CCCCN1C 33886,C1(F)(CNC(CC(=C)C)=O)CCN(C(c2ccc(N(C)CC3CC3)cc2)=O)C1 33887,N1(C(C2(SC)CN(C(=O)CN3CC4CC4C3)C2)=O)CCc2oc(C)nc2C1 33888,c1(OC)c(C(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)ccc(Cl)c1Cl 33889,C1(C(=O)NCC(C)CN(C(=O)CC(C)C2CCCO2)C)CCC(F)(F)CO1 33890,c1(C(=O)NC(CCOC)CNC(c2cc(C)no2)=O)oc(C2CCC2)nc1C 33891,CC1CCCCN1CCNC(=O)C(CC1CC1)NC(c1ccc(CC#N)cc1)=O 33892,C1(=O)C(CC(C)C)O1.C1(C(=O)OCc2c(C)coc2C)CCC2CC2CC1 33893,N1(C(c2ccc(CCCC=C)cc2)=O)CCCC(C)(C(=O)N(C)C(C)C)C1 33894,C(=O)(C1OCCc2ccccc21)OCC(F)(F)F.C1(C)CCN1CC 33895,N1(C(CCOC(N2CCOCC2)=O)=O)CC(NC(C)C)C1(C)C 33896,c1(C(N2CC=CC(NC(c3cnc4sccn34)=O)C2)=O)c(F)ccc2n[nH]cc12 33897,N1(C(C(C)NC(CC)=O)=O)CC(N(C)C(c2n[nH]c(C)c2O)=O)C(C)(C)C1 33898,c1(CC(N2CC(N(C)C(C3CCSCC3)=O)C2)=O)noc2ccc(Br)cc12 33899,N1(C(C2N(C)CCN(C(CN(CC)CC)=O)C2)=O)CCCC(C)(C)CC1 33900,C1(CC(C)(C)C#N)C(=O)N1.N1(CCS(C)=O)CCC(SC(F)(F)F)CC1 33901,c1(-c2cn(CS(N)(=O)=O)nn2)ccn2cc(C(=O)O)nc2c1 33902,c1(-c2ccc(CC)o2)nc(C2CCC2)nn1C(C)(C)C 33903,C1(CNC(c2c(C)cccc2C(C)C)=O)CCN(C(C2CC2CF)=O)C12CCC2 33904,C(=O)(CCC=CBr)N(CC(C)NC(C1CC(=O)N(C)C1)=O)C 33905,C1(N2C(c3cn(CCOC)nn3)CCCC2)CCc2nc(O)c(C(=O)OC)cc2C1 33906,c1(NCCn2c(C(CC)(c3cncs3)NCC)nnn2)ccc(C(N)=O)cc1 33907,CC(C)C(C)C(C(=O)Nc1nccs1)N1CCN(C(c2cccnc2)=O)CC1 33908,CCCC(O)C(=O)NCCC1CCN(C(C2(C)CCNC2=O)=O)CC1 33909,N1(C(CCC(N)=O)=O)CC(N(C(=O)CC(O)CN(C)C)C2CC2)C2(CCC2)C1 33910,C1(NC(Cn2c(CCC)ncc2)=O)COC2CN(C(=O)C(F)C(=O)NCC)CC12 33911,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C2(CC(C)(C)C)CC2)=O)CCC1 33912,Cc1cc(C(=O)N(C2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)C)nc(C)c1 33913,C=CC(C)(CC)C(=O)NCCCNC(=O)CNC(=O)COc1ccc(F)cc1 33914,Cc1cncc(C(N2CCC(C)(CCNC(=O)C(c3cccnc3)O)C2)=O)c1 33915,c1(C(=O)NCC(C)(CO)NC(=O)C(F)CC2CCCCC2)cc(Cl)ccc1O 33916,C1(NC(C2N(CC)CCCC2)=O)CN(C(c2cc(F)n[nH]2)=O)CC(C)(C)C1 33917,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CCSCC2)CCC1 33918,CC1CC(NC(=O)Cc2ccn(C(F)F)n2)CN(Cc2ccc(O)c(Cl)c2)C1 33919,N1(C(=O)CCc2ccccc2)CCC2CCN(C(C3CCCCC3O)=O)CC2C1 33920,N1(C(C(=C(C)C2CC2)F)=O)CC(NC(=O)CC2CCC(C)CC2)C2CC12 33921,C1(NC(c2cnc(Br)s2)=O)CN(Cc2cn[nH]c2)CC1(F)F 33922,C1(NC(CN(C2CCCC2)C)=O)CC(F)CN(C(c2c[nH]nc2C(C)(C)C)=O)C1 33923,N1(C(CN(C(=O)OCC)C)=O)CCOC2(CCCN(C(=O)CC3(CO)CC3)C2)C1 33924,C(=O)(CCC(=O)NC1(c2cn(CC(C)C(N)=O)nn2)CCC1)NC1CN(C(N)=O)C1 33925,CC(C)CC(C)(O)C(=O)NCCC1(CNC(C2CC2c2ccccc2)=O)CC1 33926,C(=O)(C(C)(C)Cc1cnc[nH]1)N1CC(CNC(c2cc(COC)[nH]n2)=O)(OC)C1 33927,c1(C(=O)NC(C(C)NC(c2cc(C(=O)OC)cn2C)=O)C)ccn(C)c(=O)c1 33928,CC1=CC(O)CN(C(c2nc(CNC(=O)Cc3ccn(C)n3)oc2C)=O)C1 33929,C1(CCNC(C2(C)CCC2)=O)CC(F)(F)CN1C(c1n[nH]c(C2CCCC2)n1)=O 33930,c1(C(N2CCC(C(C)O)C2)=O)cc2ccc(Cl)cn2n1.N12CCN(CC1=O)CC2 33931,c1(CC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 33932,Cc1cc(C(N2CCCC2C(C)NC(C2CC(F)C(=O)N2C)=O)=O)cc(N)c1Cl 33933,C1(NC(CNS(N)(=O)=O)=O)CCCC1NC(c1[nH]nnc1-c1ccccc1)=O 33934,C(N=c1[nH]c(=NC2C=CCCC2)[nH]c2cc[nH]c12)c1c(OC)cccc1Cl 33935,c12cc(cnc1OC)C1CCN(CC1)C2=O.C(C(F)(F)F)(C1CC1)OC 33936,C1(C)CCC([SH](NC)(=S)NC(=O)OC(C)(C)C)CC1.C(=O)(C(C)N1CCC1)OCC 33937,c1(CC)noc(C(=O)N(C2CCN(C(C3(CO)CC3)=O)CC2)CC)c1C 33938,c1(C(=O)NC(C)CCNC(=O)Cn2cc(CO)nn2)cnc2c(c1)nc(O)n2C 33939,c1(C(=O)NCC(CC)(C)NC(c2cccc(OC)c2)=O)cn(CCOC)nc1C 33940,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 33941,c1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OCC)CC2)cc(C)nc(O)n1 33942,c1(C(=O)OC)cc(C(=O)Nc2cccc(SC(c3ccccc3)=O)c2)cc(Br)c1 33943,Cc1ccsc1C=CC(=O)NCC(CO)NC(c1cn(C2CCC2)cn1)=O 33944,C1(C(N2CCC(O)(C(=O)OCC)CC2)=O)CC2(CC(=O)CC(=O)N2)O1 33945,N1(C(C(C=C)(C)CC)=O)CCCCC12CN(C(c1ccc(C(=O)OC)s1)=O)C2 33946,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 33947,N#CC1(C(=O)NC2CC(CNC(C34CCOCC3C4)=O)C2)CCSCC1 33948,N1(C(c2c[nH]nc2C(=O)NCC)=O)CCC(NC(=O)COC2(C)CCCC2)CC1 33949,N1(C(c2sc(C)c(Br)c2)=O)CCN(Cc2ncccc2F)CC1C(F)(F)F 33950,c1(C(N2CCC(C(=O)NC)CC2)C(=O)NCCCCCC)nn(C(C)C)nc1Br 33951,Cc1ccc(C(=O)N(C)CC2CN(C(c3cocc3C)=O)CCO2)c(C)c1 33952,N1(C(C)C(=O)NC2CC(NC(=O)CC(C)(C)C)CC2O)CCCCC(C)C1 33953,C1(C)(C(N2CC(N(C(c3c(C)occ3C(F)(F)F)=O)C)C2)=O)OC(C)(C)OC1C 33954,C(=O)(C1CSc2ccccc21)NC1C(CNC(CC(C)(F)F)=O)CCC1 33955,C1(CNC(Cc2c(C)occ2)=O)CC12CCN(C(C1CC3CCC1C3)=O)CC2 33956,C1(C(N2CC(F)(CNC(C3N(CC)CCC3)=O)C2)=O)CCc2cn(C)nc2C1 33957,N1(C(CN=S(C)(C)=O)=O)CCCC2(C(=O)NCC(CO)C(F)(F)F)CCCC12 33958,N1(C(c2cc(C)sn2)=O)CC2(C1)SCCC2NC(=O)C(F)CC1CC1 33959,c1(SC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C4CC4)=O)CC23)c(O)n1 33960,CC1(C)CCCC(C(N2CC3(CC(CC(=O)NC(c4cn[nH]c4)(C)C)C3)C2)=O)C1 33961,C(C(=O)NC1CC(CSC)OCC1)(C(C)C)NC(c1ccc(OCCO)cc1)=O 33962,c1(C(=O)NCc2c(C(=O)NC(CC=C)CO)c[nH]n2)n[nH]c(C)c1Cl 33963,C1(OC)(CNC(c2cncn2C)=O)CCN(C(=O)C=C(C)C(C)(C)C)C1 33964,C(C1=NOC2COCC12)NC(=O)NC1CC(=O)N(Cc2ccccc2)C1 33965,C1(CNC(C(C)(C)OC)=O)CN(C(=O)C(C)NC(c2cccs2)=O)CC1C 33966,N1(C(=O)CO)CCCC(C)(NC(=O)COC(C2C(C)OCCO2)=O)C1 33967,CC1CC(NC(=O)CC(C)(C)F)CN(C(C2(CO)CC2)=O)C1 33968,c1(NC(=O)NC2C(C)(C(=O)NC3(C)CC3)CCC2)cnn2c1CCC2 33969,c1(NC(C(N2C(CSC)CC3CC32)=O)=O)cccc(C2CCCOC2)c1 33970,N1(C(CC=C=C)=O)CC2CC1C2NC(=O)Cc1ccccc1 33971,N1(C(c2n(CCOC)ncc2)=O)CCCC1(C)CCC(=O)N(CC(C)C#N)C 33972,c1(CNC(Cc2cc(C)on2)=O)nnn(C)c1C(=O)NC1C=CCCCC1 33973,c1(COC(c2ccc(OCc3cccnc3)cc2)=O)ccc(F)c2c1CCCC2 33974,c1(CNC(C(CC#C)C)=O)nnc2n1CCN(C(=O)CSc1n[nH]c(C)n1)C2 33975,C12C3CN(CC13)C2.Cc1nscc1C1CC1.C12(CC1)C(=O)N(C)NC2=O 33976,CCC(CCOC)C(=O)NCC1CN(C(=O)C(C)C(=O)OC)CC1(C)C 33977,C(=O)(C(C)(C)CC(F)(F)F)NC(CCC)CCCNC(=O)CO 33978,N1(C(C(c2ccccn2)C)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 33979,c1(C(=O)NCC2N(C(c3c(CC)nns3)=O)CC(O)C2)cnc(C)cc1Cl 33980,C1(CNC(=O)C(F)CC2CCOC2)COCCN1c1ccnc(C(F)(F)F)n1 33981,c1(CNC(C2N(C(C(C)OC)=O)C3CCC2C3)=O)cccc([N+](=O)[O-])c1 33982,c1(NC(CNC(CNC(c2c(OC)c(F)ccc2)=O)=O)=O)cc(F)c(F)cc1Cl 33983,c1(C(=O)NCCCN(C(CCC#C)=O)C2CC2)cc2nccnc2cc1C 33984,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cnnc2O)=O)c1 33985,N1(C(c2cncc(Cl)c2)=O)CCC2CCN(C(C34CCC(C3)C4)=O)C2C1 33986,c1(CSCC(=O)N(C2CCN(C(c3cscc3C#N)=O)CC2)C)ccc(Cl)cc1 33987,c1(N(CCCc2c(C)cccc2)C)nc(NCC2C3COCC23)c2ccsc2n1 33988,c1(OC)c(F)ccc(F)c1C(=O)NC(C1CCN(C(=O)C(C)NC(N)=O)C1)(C)C 33989,C1(C(=O)NCC2(C)CC(F)(F)CNC2)CCc2n[nH]cc2C1 33990,c1(CC(N2CC(C)CC(NC(CC=C(C)C)=O)C2)=O)coc2ccccc12 33991,C(=O)(C(F)(CNC(C1(C#N)CCCOC1)=O)C(C)C)NC(C(=O)N(CC)CC)C 33992,N1(C(c2c(C)con2)=O)CC(NC(=O)Cc2cccc3cn[nH]c23)C2(CCC2)C1 33993,C(C(CC(C)C)C(=O)Nc1cnc(C)c(C#N)c1)NC(C1(OC)CC1)=O 33994,N1(CC(=O)CC(c2c(C)cc(C)nc2C)=O)CCC2(CC1)OCCC2N(C)C 33995,c1(C(=O)NCC23OCCC(NC(c4c(C)n[nH]c4)=O)(C2)C3)ccc2nc[nH]c2c1 33996,c1(C(N(C(C)CN(C(=O)CCc2nc[nH]n2)C)C)=O)ccc2ccc(Cl)cc2n1 33997,N1(C(c2nnc(C)s2)=O)CCN2CCOCC2(CNC(=O)C(C)CCC(C)C)C1 33998,C(CC(C)(C)C(=O)NC1(C(C)O)CC1)NC(COC(CC)CC)=O 33999,CC(C)CCC(C)NC(=O)CCC(=O)NC(C(C)C)C1CC1 34000,Cc1cc(C(N2CCCC(N(C(=O)CCn3cnnn3)C)C2)=O)ncc1Cl 34001,CC1OC(=O)NC1C(=O)NC1CCCC(NC(c2cc(Br)sn2)=O)C1 34002,c1(SC)cc(NC2CCN(C(=O)C(C(C)C)c3cncnc3)CC2C)nc(SC)n1 34003,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34004,Cc1noc(C)c1C(C)C(=O)NCC(O)CNC(c1cnco1)=O 34005,c1(CNC(C2C(NC(=O)C=CCN3CCCCC3)C2)=O)cnncc1Cl 34006,N1(C(C(C)CNC(=O)C2CC2)=O)CC23CCC2(COC3)C1 34007,c1(C(N(C(C)CNC(=O)C(c2cncnc2)C)C)=O)cnc2cnn(C)c2c1 34008,CC(N=c1cc[nH]cc1S(=O)(=O)NCc1ccc2c(c1)OCO2)c1ncnn1C 34009,Cc1ccc2nc(C(=O)NC3COCCN(C(C4CC5(CCC5)C4)=O)C3)cn2c1 34010,C(=O)(CC(C)C1CC1)NCC1C(NC(COCC(C)C)=O)C1 34011,C1(N(c2c(CC)cccc2)c2cccc(C)c2)CCC2(CC1)CNC2 34012,N1(C(Cc2c(C)noc2)=O)CCC2C1CCCN2C(C1CCCCO1)=O 34013,C(CC(O)C(=O)NC1(c2ccccc2)CN(C(=O)C(O)c2ccsc2)C1)N(C)C 34014,c1(N(CCC2CCN(C(CCCNC(=O)OC)=O)C2)C)nc(Cl)ncc1C(C)=O 34015,C=CC(CC)C(=O)NCCC1(C(=O)N(C)CC2CC2C)CCC1 34016,C(CC(C(=O)NCC(=O)N(CC(F)F)CCO)NC(c1ccoc1C)=O)SC 34017,S(=O)(=O)(c1ccc2cccc(Cl)c2c1)N(CC1(C)CCCC1)CCO 34018,c1(SC)cccc(-c2cncc(CNCc3ncccc3Br)c2)c1 34019,c1(O)cccc(C#N)c1.CCC(CN1CCCC1)N(C)C(=O)NCCSCC 34020,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34021,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)CC3CCCNC3=O)CC12 34022,c1(C(N2CCC(C(=O)Nc3cc(Cl)ccc3F)C2)=O)nc2ccccc2o1 34023,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C(=O)Nc2c(OCC#N)cccc2)COC1 34024,C(=O)(C1CCc2c[nH]nc21)NC(C1CCCCC1)C(=O)NCC1(C)CC1 34025,C1(C(C)NC(=O)C(N2CCN(C)CC2)C2CC=CC2)CCCCCC1 34026,c1(NC(C(c2cccs2)NC(C(COCC)C)=O)=O)ccccc1Br 34027,N1(C(CC2(C=C)CCOC2)=O)CCC(F)(F)C(CNC(=O)C(C)NC(=O)C2CC2)C1 34028,C(N=c1ccn(C2CC2)[nH]1)(c1cc(C)ccc1C)c1n(CC(COCC)C)nnn1 34029,C(=O)(C(C#N)C(C)C)N1CCCC(NC(Cc2c(C)cnn2C)=O)C1 34030,C1(C(C)C)CN(C(C2(CO)CCCCC2)=O)CCN1C(c1csc(C2CC2)n1)=O 34031,c1(C(N(CC(CC)NC(C(CC=C)NC(C)=O)=O)CC)=O)cc(F)ccc1C 34032,N1(C(C(C=CC)O)=O)CC=C(C(C)(C)C(=O)NCC2CC(C3CC3)=NO2)C1 34033,C=CCC(CNC(=O)C(C)NC(C1(NC(=O)CSC)CCC1)=O)OC.C(CN(C)C)N 34034,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34035,N1(C(C(c2n(C)cnc2)O)=O)C2CCC1CN(C(=O)CC1(C#N)CC1)C2 34036,N1(C(CC2C=CC(NC(=O)CC3CCCOCC3)C2)=O)CCC12CCSCC2 34037,c1(CC(=O)N(CC(C)C)CCN(c2ccccc2)C)ccccc1-c1nn[nH]n1 34038,C1(C(=O)NC2(CC(C)C)CC2)CN(C)CCN1C(=O)Cc1cnccn1 34039,C(CCCCCCCO)=CC(N1CC2C(CNC(C3CC(C)OC3=O)=O)C2C1)=O 34040,c1(C(=O)NCC2CCN(C(c3n(C)ccc3)=O)C2)n[nH]c2ccc([N+](=O)[O-])cc12 34041,N1(C(c2c(C(=O)OC)cccc2)C(=O)NCCCF)CC2(C)CC1CCO2 34042,N1(C(C2C(C(=O)OC)CC2)=O)CCN(C(=O)CCC(C)C)CC12CC2 34043,NS(=O)(=O)CCCc1cn(Cc2cnco2)nn1 34044,C1(C(N(CCNC(C(C)OCCC#C)=O)CC)=O)CC2(CCOCC2)CO1 34045,Cc1nscc1C(=O)NCCCCNC(=O)CCC1CCC(C)O1 34046,C1(C(=O)NCCC(C)N(C)C(c2cn(C)nn2)=O)CCC(C)(C)C1 34047,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(=O)CC1OCCC1C)CC2 34048,N1(C(COCc2onc(C)n2)=O)CCN(C(c2cnc(O)n2C)=O)CC(O)C1 34049,Cc1cc(C(=O)NCC2CCC2C(=O)NCC2CCCCC2(C)C)cnc1C 34050,CCC(C(=O)NCC1(C)CCCN1C(=O)C1=NOC(C(C)(C)C)C1)C(C)C 34051,c1(CC(=O)NC(C2CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34052,CCCN=C(NCC1CC(OCC)C12CCC2)NCCS(N)(=O)=O 34053,C1(C(=O)NCCC2(C)CCN(C(C3C4C5CCC(C5)C34)=O)C2)C2CCC3C(C2)CC13 34054,C1(NC(CC(C)n2ccnc2)=O)CN(C(C2(F)CCS(=O)(=O)C2)=O)CC2(CCC2)C1 34055,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34056,c1(C(N2CC(C)C(NC(c3cccnn3)=O)C2)=O)cc(F)c2nc(O)ccc2c1 34057,C1(CCNC(CNC(CC)(C)C)=O)CCC(NC(=O)C(C)NS(C)(=O)=O)CC1 34058,C1(NC(c2c(CC)scc2)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CCC2)C1 34059,C(C(C)C(=O)NC(C(=O)NCC(F)F)C1CC1(C)Br)OC 34060,C1(C(N2CC(C(C)NC(C3CCCN3C)=O)C2)=O)CC12CCSCC2 34061,Cc1cc(Br)ccc1CC(=O)NC1CCC1NC(C1CCCCN1C)=O 34062,c1(CC)ncc(Br)cc1NC(=O)NCC1(OC)CC2CC1C2 34063,C1(C(=O)NC(CNC(c2c(C)cc(C)s2)=O)(C)C)CC12CCCOC2 34064,c1(OC)cc(C(N2CCC(CF)(NC(=O)C3CC3)C2)=O)cc(N)c1O 34065,C=CCC(O)C(=O)NC(C)C(C)NCCCCC 34066,C12CCCC1C(=O)N2C.CCC(CC)=CCNC 34067,c1(C(C(=O)NC)N(C(C)C)Cc2ccccc2)cc(F)c(Cl)c(F)c1 34068,C1(C(N(CC(=O)NCC)C)=O)CCCN(C(=O)COC2CC2)CC1 34069,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34070,CCCC(C(=O)NCCN(CCOC)C(C1CCc2nnnn2C1)=O)S(N)(=O)=O 34071,N1(C(C(F)=CCC)=O)CCCC(NC(=O)COCC2CCCO2)C1C 34072,N1(C(C(CCCC)O)=O)CC(C2(N=c3[nH]nc(-c4ccccc4)o3)CC2)C1 34073,C1(CC(=O)NCCC(C)(C)NC(C(C)OC)=O)COCCN1Cc1ccccc1 34074,C1(=O)C(CC(C)C)CN1C1CC1.C1(OC)CC(NC(=O)Cc2ccns2)C1 34075,N1(C(Cc2c(C)nn(C)c2)=O)CCCC(F)(CNC(=O)CC2CCOCC2)C1 34076,N1(C(c2c[nH]c3nccc-3c2)=O)CC2OCCN(C(=O)Cc3cc[nH]n3)C2C1 34077,C1(C(N2CCC(C3N(C(c4c(C)sc(O)n4)=O)CCC3)C2)=O)(CO)CC2CCC1C2 34078,CC(C)C(O)C(=O)NCc1ccc(C(=O)NCC2(C)CCOC2)o1 34079,N1(C(C(C2N(C(c3cnc(CC)o3)=O)CCC2)(C)C)=O)CC(=O)NC(C)C1 34080,c1(C(=O)NCC(CC)N(C)C(c2nn[nH]c2Cl)=O)ccnn1C(F)F 34081,N1(C(C(C(C)(C)C)SC)=O)CCCC(C2CN(C(=O)CN3CCC3)C2)C1 34082,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34083,Nc1cc(Cl)nc(Cl)c1C(N1C2CCC1CC(NC(=O)CC1CC1)C2)=O 34084,C(CC(C)C(=O)NC(C1CN(C(=O)CCc2conc2C)C1)C)=CC 34085,CC1CN(C(C2(C)CCCCO2)=O)CC1NC(C1(N(C)C)CCC1)=O 34086,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34087,C1(C(=O)Nc2nnc(SCC)o2)CCN(C2CC2)C1=O 34088,C1(OC)CCCN(CC(=O)NC(C2CCOCC2)c2nncs2)CC1 34089,c1(SC)ccccc1CNC(C1(C)CCCC1NC(=O)OC(C)(C)C)=O 34090,c1(C(N2CC(COC)N(C(C)C(=O)NC3CC3)CC2)=O)cc2sccc2n1C 34091,c1(NCCN(C)CCc2ccccn2)[nH]c(=NCc2cccnc2)nc2sccc12 34092,c1(C(N2C(C(=O)NCC(C)OCC#C)CCC2)=O)ccc(O)nn1 34093,c1(C(=O)NCCN(C(=O)C(F)C2CCCC2)CCC)ncc(Br)cc1C(F)F 34094,C(N=c1ccnc(CN2CCN(CCN3CC3)CC2)[nH]1)c1c(SC)cn(C)n1 34095,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34096,N1(C(C)(C)C)CCCN(C(=O)C(=O)Nc2ccc(N(C)C)cc2)CC1 34097,c1(OC)cc(NC(c2ccnn2C(C)C)c2nnnn2C2CC2)sn1 34098,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34099,c1(CC(=O)NC(C)CCCCNC(c2cc(C(N)=O)[nH]n2)=O)cccc(F)c1O 34100,C(=O)(CC(C)CC(F)(F)F)N(CC(C)CNC(c1cc2cc(Cl)ccn2n1)=O)C 34101,C1(CCC(=O)N(c2cccc(F)c2)C)CCCN(C(C2(N(C)C)CCC2)=O)C1 34102,N1(C(c2c(C)ocn2)=O)CC(C)CN(C(c2ccc(F)cc2F)=O)C(C)C1 34103,N1(C(C2(CC)CC2)=O)CCCC(C)(C(=O)N(CC(c2ccccc2)O)C)C1 34104,c1(C(N(C2CCC(NC(C3C(C)OCC3)=O)CC2)C)=O)ccc(S(N)(=O)=O)cc1 34105,c1(C(=O)NC2CN(C(Cn3c(C)nnn3)=O)C3C2C3)ccc2c(c1)C=CS2(=O)=O 34106,C1(CNC(C(CC=C)C)=O)CN(C(=O)Cc2ncccc2C)CCC12CCC2 34107,C1(CNC(CCC=C)=O)CN(C(C2CC(CF)C2)=O)CCC1C 34108,C(C(CC(=O)NCC1(CC)CCOC1)NC(=O)C(C)(C)CSC)OC 34109,C(=O)(CCCCCCNC(c1occc1CC)=O)N1C(C#C)CCC1 34110,N1(C(C2N(C(C)C)CCC2)=O)CCCC(C)(C(=O)NC(C)(C)C(O)C(F)F)C1 34111,c1(CC(=O)N(C2CCCN(C(c3cccnc3)=O)CC2)CC)c(F)cncc1Cl 34112,C1(C(=O)NCCCC)CCc2nc(C)cn2C1.C=CCCOCC(=O)N(CC)CC 34113,C(=O)(C(C(CC)CC)NC(=O)Cc1cnn(CC)c1C)N(CCC)CCC 34114,c1(C(=O)NC2CC(C)(NC(C(CCC)CC)=O)C2)cccc2oc(C)cc12 34115,c1(C(=O)NC2C(NC(c3oc(C)c(CO)c3)=O)C2)cnc2c(c1)CCOC2 34116,C1(NC(C(CC(C)C)NC(c2c(C)ccnc2C)=O)=O)CC(C2CCCC2)C1 34117,C1(c2nnnn2CCC2(C)CC2)(NC(CC)(C)CC)COC2(CCC2)C1 34118,C1(COC)(NC(=O)CCC=C(C)C)CCN(C(c2cocc2C)=O)C1 34119,c1(C(N2CC3C(CNC(c4ccncc4)=O)(C3)C2)=O)ccc(C2CC2)nc1O 34120,c1(C(=O)NCCOC2CCOC2)cnc(CNC(c2ccnn2C(F)F)=O)nc1 34121,N1(C(C(C2SC(=N)NC2=O)C)=O)CC2OCCN(C(c3cc(Cl)c[nH]3)=O)C2C1 34122,C(c1cccc(C)c1)=CC(N1CC(C(C(=O)N(C2(CC)CC2)C)O)C1)=O 34123,N1(C(c2cc(C(CC)C)no2)=O)CCN(C(C2CCC(=O)O2)=O)CC2(CC2)C1 34124,C1(NC(c2cc(OC)c(Cl)cc2)=O)CCN(CC#CC2CC2)CC(C)(C)C1.CCC(N)=O 34125,N1(C(C2CC(OC)C(OC)C2)=O)CC(NC(=O)C(C(C)C)NC=O)CC(C)C1 34126,c1(C(=O)NCC(CNC(C2(F)CCOCC2)=O)OC)nn(C)c(C)c1Br 34127,N1(C(c2nc(CCC)oc2)=O)CCC(CC)C1CNC(C1CCS1)=O 34128,N1(C(C2CCOC2CC)=O)CCCOC(CNC(c2cc(OCC)n[nH]2)=O)C1 34129,N1(C(C(C=C)c2ccccc2)=O)CCN(C(C2(CC3CC3)CCC2)=O)CC1CO 34130,n1(CC(=O)NC(CNC(C2CN(C)C2)=O)(C)C)nc2n(c1=O)CCCC2 34131,c12cccc(c1)NC(=O)C(C)O2.C(C)(C)(CO)N(C)C 34132,CCCCC(C)(F)C(=O)NCC(C1CC1)N(C(=O)CN1CCOCC1)C 34133,N1(C(C2(C)CSC2)=O)CCC2C(NC(=O)CSCC(F)(F)F)C2CC1 34134,N1(C(CC2C(C)CCC2)=O)CC2CCC(CNC(=O)C(C)(C)CNC(N)=O)(C2)C1 34135,C1(NC(c2ccc(CSC(C)C)cc2)=O)CC2CC1CN2C(=O)CNC(N)=O 34136,c1(C(=O)NCC(CNC(COCCN(C)C)=O)O)ccc(-n2cncn2)c(F)c1 34137,N1(C(CC2C(CC)C2(F)F)=O)CC2(CCCC2NC(c2sccc2CC#N)=O)C1 34138,N1(C(CC(=O)NCC)=O)CC2(CCC2CNC(=O)C(C)OCc2ccncc2)C1 34139,C(C(=O)NC(c1ccccc1)c1nn[nH]n1)(C(C)C)SC 34140,c1(CC(=O)N(CC(CC)NC(=O)COc2ccsn2)C)csc(C(C)O)n1 34141,CCCCC(=O)NCCOCC(=O)NCc1cnn[nH]1 34142,c1(C(N2C(C(C)NC(C3(C)CCOC(C)C3)=O)CCC2)=O)ccn2ccnc2n1 34143,c1(C(=O)NC2(COC)CCN(C(c3cnn(C)c3N)=O)C2)cc(C)cnc1C 34144,c1(C(N2C(CC)C(NC(c3ccc(C(N)=O)cn3)=O)CC2)=O)ccc(=N)[nH]c1Cl 34145,N1(C(c2cc(C(C)=O)oc2)=O)CCN(C(c2cnc(O)n2C)=O)C2CC12 34146,C1(CNC(=O)CC2(C(F)F)CC2)CCCCC1NC(c1nncn1C1CC1)=O 34147,N1(C(C(=O)NC(C)C)=O)CC2CC(NC(=O)CC3CC3)C1C2 34148,c1(C(=O)NCCC(=C)CNC(c2ncccc2C)=O)nn(C)nc1Br 34149,C1(CNC(c2ccn(CC)n2)=O)CCCCN(C(=O)CCn2nc(C)nc2C)C1 34150,c1(C(N(CCCNC(C23CSC(C2)C3)=O)CC)=O)ccncc1C 34151,C1(C(=O)NCC(N2CCN(C(C3CCC(C#C)C3)=O)CC2)=O)CCCCN1N=O 34152,CC(C)CCCCCCC(=O)N1CCC2CCCC12C(=O)NCC1(O)CC1 34153,c1(N2CC(C(C)(C)O)C2)ccc(S(=O)(=O)NCC2(c3cccs3)CCC2)c(Cl)c1 34154,C=CC(F)(F)C(=O)NCC1CCN(C(=O)CC2(O)CCC2)CC1 34155,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(=O)C(C#N)C1CC1 34156,CCC(C)CCC(=O)NCC(CC)(CC)NC(C12CC(C)(C1)OC2C)=O 34157,C(=O)(NNC(=O)C(O)C1CCCC1)CC(CN)O.Cc1cccc(Cl)c1 34158,C(=O)(C(CCSC)O)N1CC(=CCC)C1.c1(C(=O)NCC)cccs1 34159,C(=O)(CCCCC(=O)NCC1(C)CCN(C(c2cnccn2)=O)C1)OC 34160,c1(CN)ccncc1OC.C=C1CCN(C(=O)C(O)Cn2cncn2)C1 34161,N1(C(CSC)=O)CCN(CC2CCCN(C(=O)C(C)CF)C2)CC1 34162,CCC(CNC(=O)C(=O)Nc1cc(Cl)ccc1C(C)=O)CC(F)F 34163,C1(NC(C(C=C)O)=O)CN(C(c2nnsc2C)=O)CC1F 34164,N1(C(CC=C)=O)CC(C)(C)CCC1CNC(c1cccc(OCCOC)c1)=O 34165,c1(C(C)C)noc(CCC(=O)N(CC(C)CNC(C2CC2C)=O)C)n1 34166,CN1CCOCC(CNC(=O)CC2CCCN(C(C3COCCN3C)=O)C2)C1 34167,c1(CC)cncc(CNC(C2CCC(NC(C3CCCCS3)=O)C2)=O)c1 34168,C1(C(=O)NCC(C(C)C)NC(C=C(C)c2cccs2)=O)CCc2nncn2C1 34169,C1(C)(CNC(CN(C)CCO)=O)CCN(C(=O)CCc2cc(Cl)no2)C1 34170,C1(Oc2nc(Cl)c(OC)cc2C(F)(F)F)C2CCN(C(=O)C(Cl)(Cl)Cl)C2C1(C)C 34171,C12CCN(C1)C(=O)C1CC(C1)O2.c1(NC(=O)COC(F)F)ccns1 34172,C1(CCC)(NC(=O)CNC(=O)CC(C)CCC)CCCN(C(c2ccnn2C)=O)C1 34173,c1(C(C(=O)NCC2CC(Cn3cc(C(C)O)nn3)C2)(C)C)cccc(C#N)c1 34174,C12(C(=O)OC(C)C(=O)n3cccn3)CCN(C1)S(=O)(=O)C2 34175,c1(OC)cc(C)c(C(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34176,C1(F)(C(=O)NCCCN(C(C2(OC)CCC(C)C2)=O)C2CC2)CC2(CCC2)C1 34177,Cc1ccc(CO)c(NC(c2nc(Br)cs2)c2nnnn2C2CCOC2)c1 34178,c1(C(=O)NC(C(C)NC(CCOC)=O)(C)C)cc(F)c(F)c(O)c1F 34179,c1(C(=O)NC(C(=O)N(CC#C)CC=C)C2CCCO2)c[nH]c(=NC)s1 34180,c1(C(=O)NCC2(CC(=O)NCC(CCC)C)CC2)c(C)noc1C 34181,Cc1c(Cl)cnn1CC(=O)NCC1CCC(NC(=O)C=CC(F)(F)F)C1 34182,S(=O)(=O)(CC(=O)N1CC(NC(C2CCCN2C(=O)NC)=O)C(C)C1)N(C)CC 34183,N1(C(C(C(C)C)C)=O)CCC(CNC(=O)Cc2c(Br)cnn2C)C(C)C1 34184,c1(SC)c(C(=O)N(CCCOCCNC(=O)C=C2CCC2)C)cnn1C 34185,C(=O)(C(C)(CC)OC)NCC1C(C(=O)NCCC)C1(F)F 34186,C(=O)(C(O)CC1CC1)N(CC(C)NC(=O)Cc1csc(-c2ccccc2)n1)CC 34187,c1(CCC)cc(C(=O)NC(C)(C)C(C)NC(c2cccnc2F)=O)nn1C 34188,N12CCC(O)C(C1)C2=O.n1(CCCC2CCCN(C(C)=O)C2)cnc(C)c1C 34189,c1(C(N(C)CC2CCN(C(CNS(NC)(=O)=O)=O)C2)=O)cnc(O)c(C)c1 34190,N1(CC(=O)Nc2c(C)cccc2)CCCN(C2CCN(S(C)(=O)=O)C2)CC1 34191,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCCC2)C1 34192,Cc1ccc(N2CCCC2CCNC(c2nc(C3CC3)cs2)=O)c([N+](=O)[O-])c1 34193,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34194,CC(C)CC(F)(F)C(=O)N1CCCC1C1CCCN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 34195,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34196,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)nc(=O)n(C)[nH]1 34197,N1(c2cc(OC)ncn2)CCC(NC(c2ccccc2N(C)C)=O)C1(C)C 34198,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CC)=O)ncnc(O)c1F 34199,Cc1ccc(O)c(C(=O)NCCCCCCN(C(=O)Cc2ccoc2C)C)n1 34200,C1(NC(c2nccc(SC)n2)=O)CN(C(=O)CC2COCCO2)CCC1C 34201,C1(C)(CN(C)C)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O.CC1=CC(=O)NC1 34202,CC(C)CCCCCC(=O)NCC1(C(C)(C)O)CN(C(C2CC(C)N(C)C2)=O)C1 34203,c1(C(=O)NC(C2CC2C(=O)NCC2(CO)CCOCC2)=O)ccc2cnoc2c1 34204,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NCC2CC3C=CC2O3)CC1 34205,C(N=c1nc[nH]cc1C#N)C1(C(=O)Nc2cc(SC(F)(F)F)ccn2)COC1 34206,c1(C(N(CCNC(C(c2cn(C)nc2)O)=O)C2CC2)=O)c(Cl)ccc2c1OCO2 34207,c1(CC)cc(C(=O)NCC(O)CNC(=O)C=CC(=O)OC)ccc1Br 34208,C1(CC(=O)NC(c2cnn(C)c2)C)COCCN1C(c1ccc(CC#N)cc1)=O 34209,c1(C(=O)NC(C2CN(C(c3ccc(C)n3C)=O)C2)C)n[nH]c2ccc(Br)cc12 34210,c1(-n2cc(C3(NC(c4cncc(C)c4)=O)CC(F)(F)C3)nn2)cc(C)cnc1F 34211,C12(C(=O)NCC(C)NC(C(CC)(C)C(N)=O)=O)CCC(C)(C(=O)O1)C2(C)C 34212,C12(CNC(C3(C=C)CC3)=O)CCC1CN(C(c1cc(CC)n(C)n1)=O)C2 34213,c1(C(=O)NC2CN(C(c3c(C)nc(-c4nc[nH]n4)s3)=O)C2)cc([N+](=O)[O-])c[nH]1 34214,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)CC1CCCC2CC12 34215,N1(C(C2(CSC)CC2)=O)CCCC(C)(CC(=O)NC2CCC3CC23)C1 34216,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)C1CC1 34217,c1(NC(C)CCNC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34218,c1(CNc2cc(-c3cc(CC(F)F)cc(F)c3)ncc2)ccc2c(c1)CCN2 34219,Cc1cccc2nc(C(=O)NC(C)CNC(=O)C=Cc3nccs3)cn12 34220,N1(C(Cc2ncc(OCC)s2)=O)CCCC(CNC(=O)C(C)(C)OC(C)C)CC1 34221,C1(C2CCN(C)CC2)(C(=O)NC(C(C)NC(C=Cc2cccc(C)c2)=O)C)CC1 34222,C#CCCCCC(=O)NC(C1CCCN1C(=O)CCCCCSC)C 34223,Cc1cc(OCC(=O)NC2CC(C)(NC(=O)C(F)C3CCC3)C2)ccc1F 34224,c1(OCCCNC(C(=O)NC(c2cccc(C)c2)CO)=O)cc(C)ccc1C(N)=O 34225,Cc1oc(C(C)C)nc1NC(N1CCCC1c1ccc(F)cc1)=O 34226,C1(CC(=O)NCCOCCNC(CCc2ncc(C)[nH]2)=O)CCC2(CC2)C1 34227,N1(C(CCC#C)=O)CC(CNC(=O)CCC2CCC2)CCC1C 34228,c1(C(=O)NC2C(NC(C3N(C)CCC3)=O)C2)c(Br)ccc(Br)c1N 34229,C(C(C)(C(C)C)NC(=O)C(N)=O)NC(C(c1cccnc1)OC)=O 34230,CC1CC(C)(C)CCC1N(C1CCC(F)(F)CC1)C(C1CCC=CCC1)C(=O)NC 34231,c1(NC(C2CNCC2C)C)cncc(C(N)=O)c1 34232,c1(CCC(=O)N(C(=O)COCC(=O)OC(C2CCOC2)CC)C2CC2)cccnc1 34233,C12(C(N(CCNC(C=C(C)C)=O)CC3CC3)=O)CCCCC1C2.n12cncc1C2 34234,c1(C(N2CC(C)C(NC(=O)CCC3CC3(C)C)C2)=O)csc2c(O)ccnc12 34235,N1(C(C(CC)(F)F)=O)CC2CC(O)C1C2NC(c1ccnc(C(F)F)c1)=O 34236,c1(CC(=O)NCC2(CNC(CS(=O)(=O)NC)=O)CCCC2)ccc(F)cc1F 34237,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C#C)(C(=O)NC2CCN3CCC2C3)CC1 34238,C1(CNC(C2CCC(CC)O2)=O)COCCN(C(c2sccc2OC(F)F)=O)C1 34239,N1(C(=O)C=CC2CCOCC2)CC2CCN(C(=O)Cc3ccco3)CC2C1 34240,N1(c2cc(C)nc(C3CC3)n2)CCC2(CCCN(C(C3CCC(C)CC3)=O)C2)C1 34241,C1(F)(CNC(c2n[nH]c3c2CCC3)=O)CCN(C(C2CC3CC2CC3O)=O)CC1 34242,Cn1nc(C(F)(F)F)c(CN2CCC(F)(C(=O)NCCC#N)CC2)c1Cl 34243,CC(CN(C)C)C(=O)NCCN(CC(C)O)C(c1sccc1Cl)=O 34244,C#CCC(C)(C)C(=O)N1CCN(C)C(CNC(c2cncc(NC(C)=O)c2)=O)C1 34245,c1(OCC(=O)NCCN(C(=O)CC2CCC(=O)O2)C2CC2)ccc(Br)cn1 34246,c1(N2CCCC(C(C)NC(=O)C=CBr)C2)cc(Cl)nc(-c2ccccn2)n1 34247,N1(C(CCCC(C)=O)=O)CCC(CNC(=O)C=Cc2ccc(Cl)cc2)C12CCC2 34248,c1(C(=O)NC2CCN(Cc3c(C)cc(F)cc3)CC2)cc(Cl)cc(Br)c1F 34249,c1(N(C2CN(Cc3nnc(CC)o3)C2)C)ncnc2c(C)csc12 34250,Cn1cc(C(C(=O)NCC(CO)C2CC2)NC(=O)C(O)C2CCCC2)nn1 34251,c1(C(C)C)ccc(F)cc1NC(N1CCN(Cc2ccc(Cl)c(F)c2)C2CC12)=O 34252,C1(CC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C(C)(C)C2)CC2(CCCC2)CO1 34253,C1(F)(N(C)C(C2CN(C3COC3)C2)=O)CN(C(=O)COc2ccn(C)n2)C1 34254,N1(C(c2ccc(C)s2)=O)CCN(C(C2COCC2(C)C)=O)CC1 34255,c1(COC)ncc(C(F)(F)F)[nH]1.c12nnc(s1)CNC2 34256,c1(SCC(=O)NCC2CC2NC(=O)CO)nnc(-c2ccc(Cl)cc2)n1C1CC1 34257,c1(C(N(C(CNC(CCC(CC)C)=O)C)CC)=O)ccc2c(c1)CCN2C(C)=O 34258,N1(C(CCOCC#C)=O)CCC(C(=O)NCC(O)COCC)C12CC2 34259,C1(CC(N2C(C)CCC2C)C)CC2CC1CN2C(=O)C(C)(C)F 34260,CCCC(C(=O)N1CCC(NC(C)(C)C)C12CCC2)C(C)C.C1(=O)CS(=O)(=O)N1 34261,C1(CNC(C=CCCC=C(C)C)=O)CC(F)(F)CN1C(=O)C(c1ccc(Cl)s1)=O 34262,C(=O)(CC(CC)C(F)(F)F)N(C(CN(C(c1cccc(C#C)c1)=O)C)C)C 34263,CC1CN(C(=O)CSC(C)(C)C)CCC1NC(=O)Cc1ccc(Cl)nc1F 34264,N1(C(=O)C2CC2)CCC2(CCC(CNC(=O)CS)O2)CC1.CC(C1=CCCCC1)OC 34265,N1(C(C=CCOC)=O)CC2CCN(C(=O)C(F)(F)C3(O)CCC3)CCC2C1 34266,CC1C(NC(c2cccc(CC#N)c2)=O)CCCN1C(C1CC2(CCC2)CO1)=O 34267,C(=O)(C(C(C)(C)C)NC(=O)CN(C)C(=O)NCC)C1C(C(=O)NCC)CCCC1 34268,C(=O)(CC(C)(C)C1CCCCC1)N(CCNC(CCNC(=O)OCC)=O)CC1CC1 34269,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34270,C1(NC(CS(C)(=O)=O)=O)CCC2CCN(C(c3ccc(F)cc3O)=O)C1C2 34271,c1(CC(=O)NCC2N(C(C=CC3(C)COC3)=O)CC(O)C2)cc(F)ccc1F 34272,c1(OCC=C)ccc(Cl)c(CNc2cccc(C3CC(F)(F)C3)c2)n1 34273,C(CNC(=O)CSC1CCCCC1)(CCNC(=O)CN1CC=CC1)OC 34274,CC(O)C(F)(F)C(=O)NCc1ccoc1C(=O)NCCOCCCO 34275,N(C(=NCC1=CCOCC1)NC1CCN(C2CCCCC2)C1)C(C=C)C 34276,C(=O)(C(C)(C)C(C)O)NC(CC(C)NC(COCc1c(C)ncs1)=O)C 34277,N1(C(C(C)OCCC=C)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C 34278,N1(C(C2CCC(C)O2)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1c1cccnc1 34279,N1(C(CCCNC(c2c(CC)n[nH]c2)=O)=O)CC(N(C)C)C(C)C1 34280,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34281,C1(CC(N2CC(NC(C3CC4(CC(=C)C4)C3)=O)(CO)C2)=O)NC(=O)CN(C)C1=O 34282,c1(C(=O)NC2(C)CN(C(c3ccc(NC(C)=O)cc3)=O)C2)nn(C)cc1[N+](=O)[O-] 34283,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34284,N1(C(C2CC(C)(C)C(O)CC2)=O)CCC(S(=O)(=O)C(F)F)C1 34285,C(=O)(CCC(C)NC(c1c(N)sc(C)c1C)=O)OCCC 34286,c1(N(C(C2CCN(C(C)=O)CC2(C)C)=O)C)ccc(NNC(=O)OC)c(F)c1 34287,C1(C(=O)Nc2ccn3cncc3c2)CN2CC3CC2(CO1)C3 34288,n1(C(C)C)cncc1C(=O)N(CCCNC(=O)CC1CCCO1)C 34289,N1(C(c2ccc(OCCCC)cc2)C(=O)NCCCF)CC(C)OC(C)(C)C1C 34290,C1(O)(CC(N2CC(NC(C3(C(=O)OCC)CC34CC4)=O)C2)=O)CCCCC1 34291,c1(CNC2CC(OC)C(SC)C2)cnc2ncccn12 34292,N1(C(C2CCN(CC)C2)=O)CCCC(CNC(c2cc(F)ccc2F)=O)C1C 34293,[N-]=[N+]=NC1CCC2(C(=O)NC(CNC(=O)Cn3cnnn3)CO)CC12 34294,N1(C(c2cc(CC)n(C)n2)=O)CCCC(C2CC2NC(C2CCCCCO2)=O)C1 34295,C1(C(=O)NC2CCC(C(=O)OC)C2)CN(C(=O)C(CC(C)C)OC)CCCO1 34296,c1(C(=O)NC2C(NC(=O)CSc3ccncc3)CCC2)nnc(O)cc1O 34297,C1(C)(C(=O)NCCN(C(C(CSC)OC)=O)C2CCCC2)CCCC1C(C)C 34298,c1(C(=O)NC(CNC(CC(C)n2ccnc2)=O)C)cccnc1O 34299,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCC1)C 34300,c1(C(N2C(CNC(C3(C)COC(=O)C3)=O)CCC2)=O)cccc2ccccc12 34301,C(C(O)CC(=O)NCC1(CC2CC2)CCC1)NC(=O)CCc1ncccn1 34302,C1(C(NOCC)=O)CCC2(CC1)CCN2C(=O)Cc1csc(NC)n1 34303,c1(NC(C(Cn2cncn2)NC(Cn2c(C)nnn2)=O)=O)ccccc1CCO 34304,C1(NC(CC(c2ccc(C)cc2)C)=O)CCN(C(C2(C)C=CCC2)=O)C12CCC2 34305,CC1(C)NC(=O)CC1C(N1CCCC(NC(=O)C(c2ccc(F)cn2)(F)F)C1)=O 34306,CC(C)CC(CNC(=O)C(O)CN(C)C)C(=O)NC1CCCCCCC1 34307,CC(C)CC(C)CC(C)C(=O)NC1(CN(C(=O)CCc2cncc(F)c2)C)CC1 34308,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(CF)CCOCC1)=O 34309,C(=O)(CC(C)(C)C(F)(F)F)N(CC1CN(C(C(CC)(O)c2ccccc2)=O)C1)CC 34310,c1(C(N)=O)ccc(N2CCN(C(=O)Oc3cc(Cl)sc3Cl)CC2)nc1 34311,C1(CNC(C(CO)N(C)C)=O)CN(C(=O)CN2CCNC(=O)C2)CC(C)(C)O1 34312,c1(C(=O)NCCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34313,CCCN(N(CC1(C)CC(OC)C1)C)CCO.c1ccccc1 34314,C1(C(CC)C)CCCN1C(=O)C(C1CCN(C(C2C(C)C2C)=O)C1)C 34315,N1(C(C2CCC(C(C)(C)C)CC2)=O)CCCCCC1CNC(C1CCCSC1)=O 34316,c1(C2C(C(=O)NCCN(C(C3CCCSC3)=O)CC)CC2)ccccn1 34317,CC1(c2ccccc2)CCN1N1CC(C(N2CCOCC2)=O)C1CO 34318,Cn1ncc2ccc(CNC3CN(c4ccnc5cc(Br)nn45)CCC3F)cc12 34319,c1(C(=O)NC2CCC(CCNC(COCC#C)=O)C2)cc(N)cnc1C 34320,C1(NC(c2coc(C(F)F)n2)=O)COC2(C1)CN(C(=O)Cc1cc[nH]n1)C2 34321,C1(C(=O)NC(C2CCCN(C(c3cncc(Cl)c3)=O)C2)C)CC1C1CCCC1 34322,N1(C(c2cocn2)=O)CCCC(C2CCN(C(c3conc3C3CC3)=O)CC2)C1 34323,C(=O)(C#CC1(C)COC1)NCC1CN(C(Cn2ccc(C)cc2=O)=O)CC1O 34324,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34325,C1(NC(C2C(CNC(c3cccc(=O)o3)=O)C2)=O)C(O)C2CCOC12 34326,c1(OC)cc(OC)cc(C(N2CC3CC2CN3c2nccc(Br)n2)=O)c1 34327,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34328,C(=O)(CCCC(C)CC)N1C(C(N2CCCCC(CC)C2)=O)(C(C)C)CCC1 34329,c1(C(=O)NCC2(C)CCCN2C(C2CCC(O)C2)=O)n[nH]c2c1NCCC2 34330,c1(C(=O)NC(C)CCNC(C2CC3CC3C2)=O)cncc2n[nH]cc12 34331,C=C(F)C1(CC(=O)NCC(C2CCC2)NC(C2CSCN2C(C)=O)=O)CCOCC1 34332,C1(C#CC(=O)N2CC=C(CNC(C3CCC3c3nc(S)n[nH]3)=O)CC2)(CC)COC1 34333,C1(C2CC2)(NC(C(Cn2ccnn2)NC(c2nn(C)c(CO)c2)=O)=O)CCOC1 34334,c1(OC)cc(NC(=O)C(CCC2CCC2)NCC2CC=CC2)ccc1O 34335,CCC(CC)C(=O)NCC1CCCC1NC(C1(CC)CCCC1O)=O 34336,N1(C(CCOCC(=C)C)=O)CCC(n2cc(C(C)OC)nn2)CC1 34337,C1(N(C)Cc2ccn(CC)n2)CCCN(C(=O)CCC2CCCC(O)C2)C1 34338,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)CC12CCCC1C2 34339,C1(NC(c2c(C)ccn2C)=O)CC2(C1)CC(C(N1CCC(n3ccnc3)C1)=O)C2 34340,CC1(C)CCN(C(=O)CNc2cncnc2)C1CNC(c1c[nH]c(C(N)=O)c1)=O 34341,n1(COC)cc(CCO)nn1.C1(C(N2CC(C3C(=O)N3C)C2)=O)COCCO1 34342,C(=O)(CC(CC)CCCC)NC(CC#C)CC(=O)NCC1(C)CC(C)=NO1 34343,CCC(CC(=O)NCC1(C(=O)NCCCc2nncn2C)CCCO1)C1CC1 34344,Cc1nn2cc(CC(=O)N(C(C)CNC(=O)Cc3ccccc3F)C)nc2s1 34345,N1(C(C(=O)NCC(C2CC2)OCc2c(C)cccc2)C)C(=O)CN(C)CC1 34346,N1(C(C=CC=CC)=O)CCC2(CCC(NC(=O)CCc3ncc(F)cn3)CC2)C1 34347,CC1C(NC(C2CCC(C)(C)O2)=O)CCCN1C(=O)C(CO)NC(=O)C(F)(F)F 34348,n1(CC(=O)N(CCOCCSCCOC)CC)cc(CCC(C)(C)C)nn1 34349,C1(C(C)C)CCC(C(N2CCC2CC(=O)NCC(C)O)=O)CC1 34350,C(=O)(CCC(F)(F)C(F)(F)F)N1C(C)C(NC(=O)C(N2CCC(O)CC2)C)CC1 34351,Cc1ccc(C(N2CC=CC(NC(=O)C(c3ccccc3)O)C2)=O)cc1F 34352,Cc1ccc(Cl)cc1CN1CCOC(CNC(=O)C(C(C)C)c2ccccc2)C1 34353,N1(C(c2cc(C)c(C)s2)=O)CCC(CO)C(NC(c2csc(C(F)(F)F)c2)=O)C1 34354,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(N(C(C2CC(=O)N(O)C2)=O)CC)CC1 34355,c1(C(=O)OCC)cc(Cl)c(NC(=O)Cc2c(F)cc(F)cc2F)c(Cl)c1 34356,c1(C(C(=O)N(CC(C)O)CCNC(=O)COC2CCCCC2)C)ccc(F)c(F)c1 34357,N1(Cc2ccc(CC)s2)CCSC(C(=O)NC2CCS(=O)(=O)C2)C1 34358,C1(CN(C)C(N2CCC2CO)=O)CCC(F)C1 34359,N1(C(C)C(=O)N2CC(CCCCNC(C3CC3(C)C)=O)C2)CCN(C)CC1 34360,c1(NCc2c(C(N3CCC(C)(CN)C3)=O)c[nH]n2)cnc2ccccc2c1 34361,C1(n2cc(COCC(C)O)nn2)CCCN(C(=O)CC2COCCOC2)C1 34362,N1(C(n2ccc(C)n2)=O)CCCC(C)C1CCNC(=O)Cc1c(C)cnn1C 34363,c1(C(N(CCCNC(C2CC3CCC2C3)=O)C)=O)c[nH]c2c(F)cccc12 34364,N#Cc1ccnc(NC2CCC(C(=O)NCc3c(C4CC4)cccc3F)C2)n1 34365,c1(NC(=O)NC2CC(C=C)OCC2)cccc2cnccc12 34366,C=CCC(CNC(C1C2CCCC12)=O)C(=O)N1C2CCC1CC2 34367,c1(C(=O)NCC2C(NS(C)(=O)=O)CCCC2)ccc(Br)cc1C#N 34368,CCCCC(C(=O)NC1CCCC(CNC(c2cc(N)nc(Cl)c2)=O)C1)C(C)C 34369,NS(=O)(=O)N1CC(C(=O)NC2CN(C(=O)CCOCC3CC3)CCC2CO)C1 34370,C(=O)(CC(O)CCCCC)N1CCC(=C)CC1C(=O)NOCC1C2CCCC12 34371,C(C)(CNC(=O)CCc1cnc(C)s1)(CO)NC(C(c1ccccc1)SC)=O 34372,Cc1cc2cccnc2nc1C(N1CCC1CNC(c1cnc2[nH]nnc2c1)=O)=O 34373,C1(NC(Cc2c(C)ccs2)=O)CCCN(C(c2ccccc2CC(C)C)=O)C1C 34374,C1(NC(C2N(CC)CC2)=O)CCSC12CN(C(C1CCN(CC3CC3)CC1)=O)C2 34375,c1(-c2cn(CC3CN(C(c4nnn(C)n4)=O)C3)nn2)ccc([N+](=O)[O-])cc1 34376,N1(C(Cc2c(C)ccs2)=O)CCC2CN(C(C3CC3(F)F)=O)CCC12 34377,Cc1cc(NC(C2CN(C(=O)CCc3cnc(C)o3)CC2(F)F)=O)c(C)cc1O 34378,C1(NC(c2cccc(CSC)c2)=O)CC2(C1)CN(C(C1(C)CCCCO1)=O)C2 34379,N1(C(CC(C(C)C)C(C)C)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 34380,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34381,c1(C(N2C(C)CC(Nc3nccc(C(C)(C)C)n3)C2)=O)cn2ccccc2n1 34382,C(=O)(CC(F)(F)CC)NC(CCC)CNC(C1(C(=O)OCC)CCC1)=O 34383,Cc1cnc(N)c(C(=O)NC2CC(CNC(=O)Cc3occc3C)C2)c1 34384,Cc1nn2cc(C(=O)NCC(O)CNC(=O)C(C)NC(N)=O)nc2s1 34385,C#Cc1cccc(C(N2CCN(C(c3cc(C)nnc3O)=O)C(CC)C2)=O)c1Cl 34386,N1(C(C(CC)(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1cccc2c1CCC2 34387,CC1CCN(C(c2cn(C3CC3)nn2)=O)CC1NC(c1cnn[nH]1)=O 34388,N1(C(C(CC)(C)C)=O)CC2CCC1CN2C(=O)C(CCSC)NC=O 34389,C(=O)(C#CC1CCCCO1)NC1CN(C(c2cc(SC)c(F)cc2)=O)C(C)(C)C1 34390,N1(C(=O)OC(C)(C)C)CC2CCCN(Cc3cccc(C4=CCOCC4)c3)C2C1 34391,c1(COCCC(=O)NC(C2CCN(C(C3(C)CC3)=O)CC2)C)ccc(F)cc1 34392,C(=O)(C(C)(C)CCCOC)NC(CCC)CNC(=O)C(C)C1CCC1 34393,CCC(O)C(C)C(=O)NC1CCOCC1NC(c1cccn1CC(F)(F)F)=O 34394,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34395,C(CCCC(CO)NC(c1cc(C)nnc1C1CC1)=O)NC(C(N1CCNC1=O)C)=O 34396,c1(C2(C(N3CC(C)C(CN=c4[nH]nc(O)s4)C3)=O)CCC2)cccc(Cl)c1Cl 34397,c1(OC(C)C)cccc(C(N2CCC(C)C2CNC(C2(F)CC=CC2)=O)=O)c1F 34398,N1(C(c2cc(C)nnc2)=O)CCCC(C)(CNC(=O)Cc2cc(C)n(C)n2)C1 34399,c1(C(C)OC)ncc(C(=O)N(CC(CC)NC(c2ccc(C(F)(F)F)o2)=O)C)s1 34400,c12cc(C)ccc1OC2.C1(=O)C(C2(C)CC2)NC(=O)N1CCC.C1CC1.OC 34401,n1(CC(=O)OC)cnc(C)c1C(=O)NC1CCOCC1NC(c1ccncn1)=O 34402,N1(C(c2c(C(C)NC(=O)Cn3cncn3)noc2)=O)CCC2CC12 34403,C(CS(=O)(=O)C(C)C)NCCN1CCC(NC(C2C(C)CCC2)=O)CC1 34404,N1(C(C23CC(OC)C2C3)=O)CC(NC(=O)CCCSC)C(O)C1 34405,CC(=O)CCN=C(NCC1CCN(c2ccncn2)C1)N1CCC(S(C)(=O)=O)CC1 34406,N1(Cc2c(OC)cccn2)C2CCCC1CC(NC(c1ccc(C)cn1)=O)C2 34407,c1(OC)cc(C)c(C)cc1-c1ccc(CNC(c2ncc(C)s2)=O)nc1 34408,CC(C)(CCNC(C1CCC1C(C)(C)C)=O)NC(=O)OC(C)(C)C 34409,Cc1cc(-c2nsc(C3CC3)n2)ccc1O.N1CCC(C)C1c1cccc(F)c1 34410,C(C(C)(C)CCNC(C1(CF)CCOCC1)=O)NC(CC(C)n1ccnc1)=O 34411,C12CCCN(C1)C2.c1(CN(C)CC2CC2)cn(C)nc1C(F)(F)F 34412,N1(C(CCOCCOCC)=O)CC(O)CC1C(=O)NC1CCC(N(C)C)CC1 34413,c1(N(C)CCOCCOc2ccc(Cl)cc2)ccn2cncc2c1 34414,c1(CC(N2CC(C)(C(N3CCC=C(F)C3)=O)C2)=O)ccc2nc(O)[nH]c2c1 34415,N1(C(C(=O)NCCCC(=O)OCC)C2CC2C2OCCO2)CCOC(CN=[N+]=[N-])C1 34416,C1(C(=O)NCC2CC(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34417,CC(C)CC(F)C(=O)N(CCCCCNC(c1nn(C)cc1Br)=O)C 34418,Cn1cnc(C(N2CS(=O)(=O)CC2C(=O)NOCc2ccccc2)=O)cc1=O 34419,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34420,N1(C(CCC(C)C)=O)CCOC(C)(CNC(C2(CF)CCC2(F)F)=O)C1 34421,CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc(Cl)ns1)=O 34422,c1(NC(C2(OC)CCN(C(c3cocc3C)=O)C2)=O)ccc(O)c(Cl)c1 34423,C(=O)(C(CC)C1CCOCC1)NCC(c1cnn(C)c1)NC(CCSC)=O 34424,c1(-n2cc(SCCNC(c3nccc(OC)c3C)=O)nn2)ccc2[nH]ncc2c1 34425,N1(C(c2cccc(C)c2O)=O)CC2CCC1CN(C(=O)CN1CCCC1=O)C2 34426,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34427,c1(CC(=O)NC2CCCC(NC(C3CC(O)C3)=O)C2)c(F)c(F)c(F)c(F)c1F 34428,N1(C(C2CC(C)CN2C(c2cn(C)cn2)=O)=O)CCC2(CCSC2)C1 34429,Cc1cnc2cc(C(N3CCCC3C(C)NC(=O)CC(F)(F)F)=O)nn2c1 34430,N1(C(C2(CCCC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(CC)OC)C1 34431,C1(C2CC2)(c2scc(OC)n2)CCN(C(=O)NC2CN(C)COC2)C1 34432,C1(C(=O)NC2C3CN(C(C4(CC)CC4)=O)C2C3)CCc2nc(C(F)(F)F)[nH]c2C1 34433,C1(NC(COCCC)=O)CC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 34434,C1(NC(c2c(C)n[nH]c2)=O)CC2CCC1N2C(=O)C=CC1CCOC1 34435,C=CCC(CC(C)C)C(=O)NC1CCN(C(=O)CC2CCSC2)C1C 34436,N1(C(c2c(C)nns2)=O)CCN(CCCNC(=O)CC2CCOC2C)CC1 34437,CC(CCCC(=O)NCC1(CS(C)(=O)=O)CC1)NC(=O)CN1CCCCC1 34438,C1(NC(CCNC(C)=O)=O)CCN(C(=O)CC2CC3(COC3)C2)C1C 34439,C1(NC(Cc2cc(C(C)C)on2)=O)CCCCC1NC(=O)Cc1cncnc1O 34440,c1(CC)oc2ccccc2c1C(N1CC(NC(C2CCS2(=O)=O)=O)C(SC)C1)=O 34441,CC(Cc1ccc(Br)cn1)N=c1[nH]c(=NC(C)c2ccnn2C)[nH]c2ncn(C)c12 34442,Cc1nc(CC(=O)NC(C2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)C)co1 34443,C(=O)(CCCCBr)N1CC(C)(CC(=O)N(CC(C(C)C)n2cccn2)C2CC2)C1 34444,c1(OCCC(C)NC(=O)Nc2nn(C)cc2-c2cn[nH]c2)cccc(F)c1 34445,CCCC(C)CC(=O)NCc1nc(CCC(N2CCCC(O)(C(F)F)C2)=O)on1 34446,C(=O)(CCCCCCO)NCC1OCCCN(C(C(C)NC(C)(C)C)=O)C1 34447,c1(C(=O)NC2C(SC)CN(C(=O)CNC(N)=O)C2)cccc2cnnc(O)c12 34448,Cc1sc(Cl)nc1C(N1CCCCC1CNC(C1CC1C(F)F)=O)=O 34449,c1(N2CCN(c3nc(SC)c(F)cn3)C(C(C)C)C2)cc(=O)n(C(C)C)c(O)n1 34450,C1(CC(=O)O)CCC(C)C1.C(=O)(CC=CC)NC1(CCCOC)CC1 34451,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34452,Cc1cc(CNC(=O)C(C2CCCO2)NC(c2ccc(C)o2)=O)n(C)n1 34453,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34454,n1(CC)cc(Cl)c(C(=O)NC2CCC2NC(c2cnc[nH]2)=O)n1 34455,N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)(CNC(=O)CC2CC(C)(C)CCO2)C1 34456,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34457,S(=O)(=O)(c1c[nH]c2nc(Br)ccc12)NCC1CCC(CC)C1 34458,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34459,C1(NC(c2onc(CC)n2)=O)CC=C(C(=O)Nc2ccc(C(N)=O)cc2)C1 34460,O=S(=O)(c1ccncc1)NC1C2CCC1(c1ccccc1)C2 34461,C1(C(=O)NC2C=CC(CNC(c3c[nH]cc3C(F)(F)F)=O)C2)(CC)CC(F)(F)C1 34462,C1(NC(=O)C(C2(O)CCCC2)F)CCSC12CN(C(c1ccc(F)cc1Cl)=O)C2 34463,CC(CCC(C)(C)C)N=c1[nH]c(=N)[nH]c(=NCCc2c(N)cccc2F)[nH]1 34464,Cc1c(C(=O)N(CCC(C)NC(=O)CC2CC3(CC3)CO2)C)sc2nccn12 34465,c1(C(=O)NCC2C(CNC(C(CC)(C)OC)=O)C2)ccc2scc(C)c2c1 34466,c1(CCC)nnc(S)n1CC(=O)NC1CC(F)(CNC(c2cc(C#N)cs2)=O)C1 34467,CCCCC(CCCC)CC(CC)C(=O)NCC1=CCCOC1 34468,C=CCC(C)(C)C(=O)NCC(C1CCN(C(C2CCC(C(N)=O)C2)=O)CC1)O 34469,OC1COC2C(NC3CC(c4ccc(F)cc4)CC3O)COC12 34470,c1(CC(C(=O)NCC(N(C(=O)Cc2cc[nH]n2)C)C2CC2)=O)cc(Cl)cc(Cl)c1 34471,CC1CC2(CCO1)CC2C(=O)NC1CN(C(c2ccnn2CC(F)F)=O)C1 34472,N#Cc1ccc(CCNC(=O)CC2CCN(C(=O)CCc3ccc[nH]3)C2)cc1 34473,C(c1ccc(F)cc1)=C(C)C(=O)NCC1CC(F)(CNC(C2(F)CCOC2)=O)C1 34474,Nc1cnc(Cl)cc1C(N1CCCC(NC(=O)C=Cc2nnn(C)n2)C1)=O 34475,c1(C(CN(CC=C)CCc2cn(CCN3CCOCC3)nn2)O)ccc(Br)cc1 34476,N1(CC(=C)Cl)CCN(C2CCN(C(=O)CC(C)Oc3ccccc3)C2)CC1 34477,C1(N(C)C(=O)Nc2cccc(NC(C)=O)c2)CCCCC1S(C)(=O)=O 34478,N1(C(c2cc(C)ncc2C)=O)CCC(C)(C)C(CNC(=O)Cc2cnc(C)[nH]2)C1 34479,N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(Cc2cn(CC3CC3)nn2)C(F)(F)C1 34480,CN(C)N=Nc1ccccc1OCC(O)CNCc1ccc([N+](=O)[O-])cc1 34481,C1(C(NNC(=O)c2cc(C3CCOCC3)[nH]n2)=O)CCCN2CCSCC12 34482,N1(c2n(Cc3ccc(OC)c(I)c3)nnn2)CCOCC12CCC2 34483,C1(C(=O)NC(C2CCN(C(Cc3ncc(C)o3)=O)CC2)C)CCCC(C)(C)C1 34484,C(=O)(C1=CC2CCCCC12)Nc1cccc(OC)c1C(F)(F)F 34485,c1(C(=O)NCC23C(CN(C(C4CC(C)C4)=O)C2)C3)cccc2c1CCO2 34486,Cc1c[nH]c(C(=O)NCC(C2CC2)NC(c2cnc(C(N)=O)s2)=O)c1 34487,Clc1ccc(CNc2cnn(C3CCOC3)n2)c(I)c1 34488,N1(C(COC)=O)CCN(C(C2CCC(Oc3ccccc3)C2)=O)CC(O)C1 34489,C(C(O)C(=O)N1CC(C(O)C(=O)N(C)C(C)C)C1)SC 34490,CC1CCN(C(C2CCC(CO)CC2)=O)CC1NC(C1CCCN1C)=O 34491,C12(C(N3C(C)CC(NC(=O)CC4(CO)CC4)CC3)=O)CCCCC1CCCC2 34492,C#Cc1ccc(C(=O)NC2COCCC2C(=O)NC(C)(C)C#C)nc1 34493,c1(C(C(=O)NC2CN(C(C)=O)C2)N(CCSC2CCCO2)CC)cccc(C)c1 34494,c12cc[nH]c1c(=O)c2=O.C1CC(=O)N1CCCO.C(CCO)NC1CCC1 34495,c12nc(ccc1Br)N2.C1(O)(C(N)=O)CCN(C(C2CC2C(F)F)=O)C1 34496,n1(CC)cnc2c(N3CCC(CC#N)C3)[nH]c(=NCCCCCCSC)nc12 34497,c1(OC)nscc1C(C(=O)OC)N(C)Cc1occc1C 34498,C(CCOCCO)(C(=O)NC(C(N)=O)C1CC1)NOCC=CCC 34499,C1(CS(=O)(=O)N(CC(C)(C)CO)C)(C(=O)NC)CCCC1 34500,CCC(CC)(C(=O)OC)OC(=O)NC1C(C(=O)OC(C)(C)C)CN(C)C1 34501,Cn1c(Br)nc2c1CCN(c1ccnc3ncnn13)C2 34502,c1(OC)ccc2c(c1)CCC2(C)CNC(c1nc(-c2ccccn2)cs1)C 34503,C(=O)(C#CC1CCCCC1)N1CCC(C(C)NC(c2ccc(Cl)c(F)c2)=O)CC1 34504,c1(OC)ccccc1CCC(=O)NC(CNC(=O)C(CC)OC)C(C)(C)C 34505,Cn1cc(C(N2CCC(O)(CNC(C3CCC(F)C3)=O)C2)=O)c2cc(F)ccc12 34506,Cc1cc(C(N2CCC(C)(C(=O)NCC(C)(C)C3CC3)CC2)C)c(C)n1C 34507,C#CCC(CC(F)F)C(=O)NCCCOCC(N1CCN(C)C(=O)C1)=O 34508,N1(C(c2cc(OC)n[nH]2)=O)CCOCC1C(=O)NC1COCCOC1 34509,C(=O)(CCC(=O)NN(C)C)NC1CCN(C(COCCCC)=O)CC1OC 34510,c1(C(N2C3(CNC(c4cccc(Br)c4)=O)CCC3CC2)=O)cccc2cccn12 34511,c1(C(=O)NCC(C(C)C)NC(C2(F)CC2C)=O)ccc(SC(F)(F)F)nc1 34512,N1(C(CC=CC=C)=O)CC(NC(c2ccc(-c3cnn(C)c3)o2)=O)CC2(CC2)C1 34513,C1(NC(C=CSC)=O)C(C)CN(C(=O)CN2CCCNS2(=O)=O)CC1C 34514,c12ccccc1-n1nnnc1C2OC.C(C)(C)(CN(C)C)NC(C)CCO 34515,N1(C(CC2C(C)(C)CCO2)=O)CC=C(CNC(=O)C=CCn2cncn2)CC1 34516,c1(CC(=O)NCC2C(NC(C(CC)O)=O)CC2)c(C)nn(CC(C)C)c1C 34517,CC(C)C(CC(=O)NC1CC(n2cccn2)C1)NC(C1CC2CC(=O)C1O2)=O 34518,C(CCC(C)C(=O)NCC1(COC)CCOC1)OC 34519,c1(C(N2C(CNC(C3CC34CCCC4)=O)CC(O)C2)=O)cnn2c1CCC2 34520,CC1(CNC(=O)C=CCF)CC(F)(F)CN1C(C1CCC2(CC2)C1)=O 34521,C1(N(C2(CO)CCSC2)Cc2c(C)nns2)CNCCOC1 34522,C1(NC(c2n(C)nc(Cl)c2)=O)CN(C(c2nccnc2N)=O)C2(CCCOC2)C1 34523,c1(CC)nc(N(C(C)CNC(C2CC(F)(c3ccccc3)C2)=O)C)c(C)o1 34524,C(C)(C(=O)NC1(C)CCC(C2OCCO2)CC1)(C(C)C)OC 34525,c1(C(N2CCCC(N(C(CN3CC(C)C3)=O)CC3CC3)C2)=O)cc(Cl)ncc1F 34526,N1(C2CC2)CCOC(C)(CCCOCCOC)C1.c1(OCC)ncnc(NC)c1C 34527,c1(C)ncncc1Cl.C12CC(OC)CN1C2=O.C(F)(C(=O)NC)=CCC 34528,c1(C(N2CCC(C3CC3)(NC(C(F)=CC)=O)C2)=O)ccc2cnnc(O)c2c1 34529,C(CC(C(=O)NCc1cncs1)NC(=O)C=CC(F)F)=CC 34530,c1(C(N(CC(C)(C)CNC(=O)CC2CN(C)CC2O)CC)=O)cnc(N)c(N)c1 34531,Cc1ccc(Cc2ccco2)c(C(N2CCC(CNC(=O)CC(C)(C)C)C2)=O)c1 34532,N1(C(CC(C)SC)=O)C2COCC1CC(NC(=O)C(C)=NOCC#N)C2 34533,c1(C(CC#C)CC)nnc(N(C2CCOC2)C2CC2)n1Cc1ccccc1OCC 34534,C1(CC)CN(C(C2CCC(C3CC3)N2C(=O)CCC(=O)C2CC2)=O)CC1CC 34535,c1(N2CCC(n3cc(C(C(=O)OC)O)nn3)C2)ccccc1F 34536,C(N=c1cc(Cl)nc[nH]1)C1(O)CCCN(C(C(c2cc(F)c(F)c(F)c2)C)=O)C1 34537,C1(COCC(N2CCC(NC(C3(CCC#C)OCCO3)=O)C2)=O)CC2COCC12 34538,C1(CCCNC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCCc1ccccc1 34539,N1(C(C2C(NC(CCOC(C)=O)=O)CC2)=O)CCOC(C#N)C1 34540,c1(C(=O)NC(CNC(c2occ(C(=O)OC)c2)=O)(C)CO)cc(O)nc(C)n1 34541,CN=S(C)(=O)c1cccc(C(=O)NC2CCN(C(=O)COC3CC3)CCC2(F)F)c1 34542,C#Cc1ccc(C(=O)N(CC(O)CN(C)C(c2cn(C3CC3)nc2C)=O)C)cn1 34543,c1(C(N2CCC(C(CNC(C(C=CC)O)=O)(C)C)CC2)=O)ccc2ncsc2c1 34544,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34545,N1(CCc2c(C=C)cccc2)C(=O)CN(CC2CCC3CC23)C1=O 34546,C1(c2c(C(N(C)C)=O)con2)CCCN(C(c2ccccc2)=O)C1 34547,C1(NC(N(C)OC2CCCC2)=O)C2CCC(C2)N1CC(F)(F)F 34548,Cn1cnc(CNc2cccc(OC3CCC3)c2)cc1=O 34549,c1(C(CNC(=O)C(=O)NC2(C)CSCC2C)OC)ccccc1C(F)(F)F 34550,c1(C(=O)NCCCC(C)NC(=O)CC2CCCC(O)C2)cc(=O)n(C)cn1 34551,C1(C(C(=O)N(C(C)CN(C)C(c2cc(CO)[nH]n2)=O)C)F)CCC(=O)CC1 34552,C1(C2CCN(C(C3(C)CC3C)=O)C2)(NC(c2n[nH]c(C)c2C(F)(F)F)=O)CC1 34553,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34554,c1(CC)ccc(C)cc1C(=O)NCCCCCCOc1cncc(CC2CC2)c1 34555,C(=O)(C(CCC(C)C)NC(=O)Cc1c(C)n[nH]c1C)N1CCC(SC)C1 34556,N(C(=NCCC(=O)N1CCCC1)N1CCCC(F)(F)C1)CC(C)C(F)F 34557,C#CCCC(=O)N(CCC(C)(C)N(C)C)C.C12CC(C1)N(C(C)=O)C2=O 34558,c1(OC)ccc(S(=O)(=O)NC(C2(F)CCCN(C(=O)CSC)C2)=O)cn1 34559,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)CCCc1cc[nH]n1)OC 34560,c1(CC(=O)NCCCNC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34561,CC(C(=O)NCc1ccc(CNC(=O)C=CCN2CCCC2)cc1F)S(N)(=O)=O 34562,N1(C(c2c([N+](=O)[O-])cn(C)n2)=O)CCC2(CCOC2)C(CNC(C2CCC2)=O)C1 34563,N1(C(C(CC#C)C)=O)CC2CCC1C(CNC(C1(c3cccc(Cl)c3)CC1)=O)C2 34564,N1(C(=O)C(C2CCCCC2)F)CCCC(F)(C(=O)NC2C=CC(CC3CC3)C2)C1 34565,c1(CC)nonc1C(=O)N(C1CCCC1)CCNC(=O)CCC1(C)CC1 34566,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34567,c1(N(C)C)ncc(C(=O)NCC(O)CN(C)C(c2csc(C(F)(F)F)n2)=O)s1 34568,N(C1CC2(CCC2)Oc2ccccc21)C(=O)NCc1c(C)oc2ncnc(O)c21 34569,C1(C(N2CC(C(C)O)C2)=O)CN(C(=O)C(O)c2cnc[nH]2)CC2(CCC2)C1 34570,c1(C(=O)NCC(C)NC(=O)Cc2ccc(CO)cc2)nccc(C#N)c1F 34571,c1(C(=O)NCCNC(C2CCCC2)=O)c[nH]c2cccc(Br)c12 34572,c1(N(C)C)ccccc1NC(C1CCCN(CC2(C)CC2)C1)=O 34573,CCCCCCCCC(F)C(=O)N1CCN(C(c2c(C)nsc2N)=O)CCC1C 34574,c1(C(=O)NC2(C)CC(NC(CC3C(C)(C)C3)=O)C2)ccc2c(O)nncc2c1 34575,C=CC(C)CC(=O)NCC1(C)CCCC1C(N1CCCC1)C=CC(=O)N=CCSC 34576,N1(C(CCC(C)OC)=O)CCCC(F)(C(=O)NC2CC(C)C2)C1 34577,C1(CC#C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34578,N1(C(CC)=O)CCC2(CCC2)C(CNC(C2(c3ccno3)CCOCC2)=O)C1 34579,O=C(C#Cc1ccccc1)NC(=O)NCC1CCN(C2CC2)C1.c12cn-1nn2 34580,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)CC 34581,n1(CC)cccc1C(c1nnnn1C1CCC1)NCCC1CCC1 34582,c1(C(N(CCCNC(C(C(C)O)N(C)C)=O)C)=O)nnc2n1CCCCC2 34583,Cc1coc(C(C)(C)C)c1C(N1CC(NC(=O)C(F)C2CCOC2)C1)=O 34584,c1(C(=O)NCc2ccc(Cl)nc2Nc2ccnc(Cl)c2)cc(Cl)c(F)c(Cl)c1F 34585,N1(C(C2(C)N(C(CCc3c(C)noc3)=O)CCC2)=O)CCc2ncncc2C1 34586,C1(C(N(CC(C)NC(=O)CCc2cnc[nH]2)C)=O)CC2(C1)C(F)(F)C21CC1 34587,C(CO)(CCCCNC(C1(F)CCCCC1)=O)NC(C1(CC)CCC1)=O 34588,C(=O)(CC1=CCN(C(C23CCC(OC)C2C3)=O)CC1)NCC(C#C)OC 34589,C1(CNC(C2CC2c2ccco2)=O)CCCN(C(C2CCCCN2C2CC2)=O)C1 34590,N(C1CCOc2ccc(Cl)cc21)C(=O)NCc1ccc(F)cc1N1CCOCC1 34591,N1(C(c2c(OC)sc(Cl)c2)=O)Cc2cnc(C)nc2C1 34592,C#Cc1ccc(OCC(N2CCSCC2NC(=O)C=CS(C)=O)=O)cc1 34593,N1(C(c2n(COC)ncc2)=O)CCN(C(=O)CC(C)(C)c2cnsc2)CC1CF 34594,CC(C)S(=O)(=O)CCCNC1COC(C)C1.C1(C)(C)CNC(=O)N1 34595,CC(C)(Cc1cccc(Cl)c1)C(=O)NC1CC(NC(=O)C2=CCSC2)C1 34596,c1(SC)cc(C(c2nnnn2C(C)C)NC2(c3ccccn3)CC2)on1 34597,c1(SCC2(C(=O)NCC(CN(C(CC#C)=O)C)(C)C)CCC2)ccc(Cl)cc1 34598,S(=O)(=O)(c1ccncc1)NCCN(C(=O)Cc1cncnc1)CC 34599,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34600,N1(C(c2ccc(OC)cc2)=O)CCN(c2cc(C)nc(OC)n2)CC1CO 34601,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34602,c1(SCc2ccc(NC(C3C(=C)C3)=O)cc2)ccc(C#N)cc1 34603,C1(CC(N2CCC(O)(CNC(c3ccc(CC)s3)=O)C2)=O)OCCCC1(C)C 34604,c1(C(N2CCC(CNC(c3snc(Cl)c3Cl)=O)C2)=O)cccc2cnsc12 34605,C1(SC)CC2C=CC1O2.C12(C(=O)NC3COCC3CN(C)C)CN(C1)C2=O 34606,c1(C(=O)NC2C(SC)CN(C(=O)CN3CCSCC3)C2)nccn2nc(C)cc12 34607,N1(C(CSCC)=O)CCC(N(C(=O)CCc2ncccn2)C)CC1 34608,C1(C(N2CCN(CCN(C(=O)Cn3ccnn3)C)CC2)=O)CCCC12OCCO2 34609,C1(C(C(=O)N(CCO)CC2(O)CCC2)F)CCCCC1.C1CC(=O)N(C)CCN1C 34610,N1(C(CNC(CC)=O)=O)CC(NC(=O)Cc2ccccc2C)CCC1C 34611,N1(CC(=O)NC2(CO)CCN(C(C(C)(F)F)=O)C2)CCCCC(O)C1=O 34612,C1(C(=O)NC(C2CCN(C(c3cnc(C4CC4)o3)=O)C2)C)C=CC=CC=C1 34613,C(C(F)(C(=O)N1CCCC1CNC(N)=O)C(C)C)NC(c1cc(=NC)[nH]cc1)=O 34614,C(=O)(C(CCN(C)C)NC(c1cnnc(O)c1)=O)N1CCC(SC)C1 34615,c1(-n2cc(CC(C(=O)NS(=O)(=O)C3(c4ccccc4)CC3)O)nn2)ccc(O)cc1 34616,C1(C(N2CC(C)C(NC(C3(C(C)(F)F)CC3)=O)C2)=O)CC1C1CCOCC1 34617,CCC(CC1CCCC1)C(=O)NC(C)(Cn1cccn1)C1CNC1 34618,c1(CC)nc(C)c(C(=O)NC2CCC(N(C)C(c3cocc3C)=O)C2)o1 34619,N1(C(C2(CNC(C3CCC(C(=O)OC)C3)=O)CCCC2)=O)C2CCC1CC2 34620,C1(CN(C)C)CCCCN1C(C1CCCN1C(c1cnn(C)c1)=O)=O 34621,N1(C(C2C(=C)CC2)=O)CCN(C(C2CCCN(C(C3(C)CC3(Cl)Cl)=O)C2)=O)CC1 34622,Cc1nc(O)nc(C)c1C(=O)N(CC(C)NC(C1COCCC1(F)F)=O)C 34623,c1(CC)nc(C(C)C)ccc1C(=O)NCCCN(C)C(c1ccn(C2CCC2)n1)=O 34624,c1(OC)ccc2ncc(NC(N3CCCCCCC3c3ccccc3)=O)cc2c1 34625,c1(C(=O)NCC(CC)(C)NC(=O)CNC(=O)NCC2CCCC2)ncc[nH]c1=O 34626,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34627,c1(C(N(C2CCN(C(=O)C(C)(C)C)C2)CCC)=O)c2c(nn1CC)CCCC2 34628,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34629,C(CC(C(=O)NCCN1CC(CF)C1)NC(=O)C=Cc1cc[nH]n1)SC 34630,C1(C(=O)NCC(CN(C(C(C=C)CC)=O)C)O)CCC2(CC1)CNC(=O)C2 34631,CC1(C(=O)NC2CC(NC(=O)C(c3ccc(F)cc3)(F)F)C2)CCC(O)CC1 34632,N1(C(C=C(COC)C)=O)CCN(C(=O)CC2CCCCN2C(C)=O)CC1COC 34633,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34634,C(CCCCC(=O)NC1CCC(C(NC[Si](C)(C)C)=O)C1)OC 34635,Cn1ccc2nc(Nc3nc(CC(N4CCC(CO)C(F)(F)C4)=O)cs3)ncc12 34636,C1(OC)CC(C(=O)NCCCCC2CN(C(c3ccc(CO)cn3)=O)C2)C1(C)C 34637,c1(OC)cccc2c1nc(C(=O)NCC1CC3(C1)CS(=O)(=O)C3)n2C 34638,c1(C(=O)NCC(C)N(C(c2ccc(C)cc2C)=O)C)c(N)sc2ccccc12 34639,CC1=NOC(=O)C1CCC(=O)NCCOC1CCN(C(c2ocnc2C)=O)C1 34640,c1(COC)c(C(=O)N(c2nn(C)cc2C#N)C)oc2ccccc12 34641,C1(C(=O)NCCCc2scc(CC)n2)CCC2(CCCNC2)C1 34642,c1(C(=O)NCCC2CCC(NC(c3c(SC)cnn3C)=O)C2)cc(O)ccc1N 34643,CC1CN(C(C2(c3ccc(Br)nc3)CC2)=O)CCN1S(=O)(=O)c1cccs1 34644,C=CCN=C(NCCCOc1ccc(Cl)cc1)NCC1CC(=O)N(C(C)C)C1 34645,Cc1cccc2nc(C(=O)NC(C)(C)C(C)NC(C3CNC(=O)N3)=O)cn12 34646,c1(C(N2CC3(CCN(C(C4(OC)CCOC4)=O)C3)C2)=O)cnc2ncnn2c1O 34647,c1(C(=O)NCCCCNC(c2c(C)cc(CO)o2)=O)cc(C)c(O)c(N)c1 34648,CCC(CC)C(C)C(=O)N1CCC(C(=O)N(C)Cc2nnc(O)o2)(C(C)C)C1 34649,c1(C(=O)NC(C2CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C)cc(OC(F)F)n(C)n1 34650,C1(C(N(C2(C(N)=O)CC2)C)=O)C2CC3C(C2NC(=O)C(C)(C)Cl)C13 34651,c1(C(=O)NC2C(NC(c3n(CC)nnc3C)=O)CCC2)nsc2ccccc12 34652,N1(C(C2CC(NC(CCc3cc(C)sc3)=O)C2)=O)CCCCC1C 34653,Nc1c(C(=O)NCC(CO)NC(c2ccn(C(F)F)n2)=O)cc(Cl)cc1F 34654,O=C1CCCC(C(=O)NCC(CC(=O)N2CCC(CF)C2)C2CCC2)CC1 34655,C1(NC(CC2(C(=C)F)CCC2)=O)CN(C(=O)C(C)CC(C)C)C(C)(C)C1 34656,c1(C(=O)NCC(=O)NCC(=O)NC(CC)C(C)(C)O)cnc(C)nc1C.C(=O)C 34657,C1(CC#C)CN(C(=O)C(Cc2ccoc2)NC(c2cc(Cl)cn2CC)=O)CCO1 34658,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34659,Cc1c(C)c(C)c(C(=O)NC2C3CN(C(=O)CCSCC(N)=O)CC23)c(C)c1C 34660,c1(C(=O)NCC2N(C(CCCC#C)=O)CCC2)ccc(C(C)=O)c(C(F)(F)F)c1 34661,c1(C(=O)NC(C(=O)NCc2ncc(C)[nH]2)C2CC2)cncc(C#N)c1 34662,Cc1ccc(CC(C(=O)O)NC(C2CCOC2c2cnn(C)c2)=O)nc1 34663,c1(C(N2CC(CC)N(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)nccn2ccnc12 34664,C1(CCC(C)(C)NC(=O)C#CC2CC2)CCN(C(=O)CC23COC(C)(C2)C3)CC1 34665,C1(NC(C=CC)=O)CCN(C(C2CC2c2ccnn2C)=O)C1(C)C 34666,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34667,C(CCC(C(=O)N(C)Cc1cccc(C)n1)OC)NC(C1CC(=C)C1)=O 34668,n1(CC(=O)NCCOC2CCN(C(=O)C=Cc3cc[nH]n3)C2)cnnc1O 34669,Cc1cc(C(=O)NCC(C)(C)OCC(=O)N(C)CCC2CCC2)ccc1O 34670,C1(CC)CN(C(=O)Cc2cc(F)ccc2F)CCN1C(c1cc2n(c1)CCC2)=O 34671,C1(C(=O)NC(C(C)CNC(c2ccnnc2)=O)C2CC2)CC(C)(c2ccccc2)C1 34672,C1(CCC)CCCCC1NC(C1(CNC(c2csc(CC)c2)=O)CCCC1)=O 34673,CC1(C(N2CCCN(C(=O)CC3CCCC(F)(F)C3)CC2)=O)COCCC1(F)F 34674,c1(N2CC(NC(CC(C(C)C)C)=O)C(C)(C)C2)ccc2c(n1)CC(C)(C)CC2=O 34675,c1(C(=O)NCC(CNC(c2coc(CCC(F)(F)F)n2)=O)F)cnc(C2CC2)[nH]1 34676,C(=O)(C1=C(Cl)CCCC1)NCC1(COC)CCCN1C(C1CC12CCC2)=O 34677,c1(C(N2CCC(NC(C3CC(C)C3)=O)(CO)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34678,N1(C(c2c(C)snn2)=O)CCC(C2CC2)(NC(=O)CCCCc2cnc[nH]2)C1 34679,c1(OC)c(Cl)ccnc1NC(C1CN(Cc2ccc(F)c(F)c2)CC1O)=O 34680,N1(C(C2C3(CC(NC(C4C(C)CCOC4)=O)C3)C2)=O)CCC(O)(C(N)=O)CC1 34681,C(CC(C)(C)Cc1cn(C2CCCN(CCOC)C2)nn1)OC 34682,N1(C=O)CCN(C2CC2)C(C)C1.CC(C(=O)NC)N1CCCC1.C12(CC1C)C(=O)N2 34683,N1(C(CCN(C(=O)OCC)C)=O)CCN(C(=O)CCC(C)(C)C)CC(C)C1.C(C)(=O)N 34684,C1(OC)CC(C(=O)NCC(C)CNC(=O)C(C)OCC(C)C)N(S(C)(=O)=O)C1 34685,N1(C(C2(C)CNC(=O)C2)=O)CCCN(CCNC(=O)C=Cc2ccsc2)CC1 34686,CN1CCC(F)C(NC(=O)COC2(C)CN(C(=O)C3=CCCOC3)C2)C1 34687,C(C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(=O)CC2CCCCC2O)C1)OCC 34688,N1(C(c2ccnc(OC)n2)=O)CC2CC(NC(=O)CCn3cccc3)CC1C2 34689,Cc1cc(F)ccc1CC(=O)NC(CNC(C1CCCC(=O)N1)=O)CC(C)C 34690,C(C(O)CNC(=O)Cc1cn[nH]c1)N(C(=O)CSCC(F)(F)F)C 34691,C1(C)(CC(=O)NCCCC2(NC(C3(c4cccs4)C(C)C3)=O)CC2)CCCO1 34692,c1(C(N2CC(CC(C)NC(c3cncc(N)n3)=O)C2)=O)cccc(C(C)(C)C)c1 34693,N1(C(COC)=O)C2CCC1CC(O)(CNC(=O)C(C)OC1CCCC1)C2 34694,Cc1cc(C(=O)NC2CCN(C(C3CC4(CC4)C3)=O)CC(O)C2)cc(C)c1N 34695,N1(C(c2ccc(C)[nH]2)=O)CCOC2CN(C(C3CCC3C)=O)CCC12 34696,c1(C(N2C(C)CC(CNC(C(C)=C3CC3)=O)C2)=O)coc(S(C)(=O)=O)c1 34697,CCCCCC(C)CC(=O)NCC1(O)CCCN(C(C2(C(F)(F)F)CCC2)=O)C1 34698,C(CNC(C1(F)CC1)=O)(C(C)C(C)C)NC(Cc1c(C)cccc1)=O 34699,C=CC1(C(=O)NCC(C)(C)CNC(c2ccn(C3CC3)c2C)=O)CCCCC1 34700,C1(NC(C2CCCCC2)=O)C2CCC1N(C(c1ccc(C(F)F)cn1)=O)C2 34701,CC(C(CO)NC(=O)COCC(c1ccccc1)C)NC(=O)CCC1CCCO1 34702,CC(C(=O)N1CCN(C(=O)CN(C)C2CC2)C(c2ccncc2)C1)C(C)(C)C 34703,Cc1cccc(C(N2CC(C)(C(N3CCOC(C(C)(C)C)C3)=O)C2)=O)n1 34704,c1(C(=O)NCCCCC(CO)NC(C(C)SCC)=O)ncc2ccccn12 34705,N1(C(C2CCN(C)C2)=O)CCC2(CCCC2C(N2CCCC(F)C2)=O)C1 34706,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(CNC(C2CCC(OC)CC2)=O)C1 34707,C1(C(C)NC(C2CNC(=O)C2)=O)CN(C(c2ocnc2C2CCC2)=O)CCO1 34708,c1(C(N2C(CNC(CN3C(C)CC3)=O)C=CC2)=O)cn(C)nc1C1CC1 34709,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)[N+](C(C1CCCC1)=O)([O-])N 34710,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34711,N1(C(CCCOCCC)=O)CCC(NC(c2ccc(OC)cc2C)=O)CC1C 34712,c1(C(=O)NCCOC2CCN(C(=O)CC3C=CCC3)C2)n[nH]cc1[N+](=O)[O-] 34713,N1(C(Cn2c(C)ccc2C)=O)CC(C(=O)NCc2cccc(Cl)c2)CCC1(C)C 34714,C(CS)(C(=O)N=c1cc(C)n(CC)[nH]1)NC(C=CCC)=O 34715,C(=O)(C1=C(C)CCOC1)NCCN(C(C(C)NC(CC)=O)=O)CCOC 34716,c1(C(=O)NCC(CNC(c2onc(C)n2)=O)(C)C)cccc(C2CC2)c1Cl 34717,C1(NC(C(c2ccccc2)OCC)=O)(CO)CN(C(C2CCN(CC)C2)=O)C1 34718,c1(N(C(=O)CCCC(F)(F)F)C2CNCC2F)ncnc2n[nH]c(Br)c12 34719,Cc1cc(C(=O)NCCC2(O)CN(C(=O)CC3(C)CCCO3)C2)cc(F)c1C 34720,C#Cc1ccc(C(N2C(C(N3C(CO)CC3C)=O)CC3CC23)=O)o1 34721,N1(C(C(C)C(C)(F)F)=O)CC2(CCCC2CNC(=O)CCC2CCOCC2)C1 34722,C1(C(N2C(CCN(C(=O)C#CC3CCC3)C)CCCC2)=O)CC2(CCC2=O)C1 34723,CCC(CC(=O)NCCOCCC(=O)NC)OC.N12CC=CC1C2=O 34724,Cc1ccccc1CC(=O)NC1(CNC(=O)C(C)C#N)CCCC1 34725,CC(C)S(=O)(=O)C(C)C(=O)NC(C)(CNC(c1c(F)ccc(OC#N)c1F)=O)CO 34726,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34727,c1(OC)cc(Cl)ncc1C(=O)NC1CC1C(=O)Nc1cc(O)nc(Cl)c1 34728,CC1CC2CN(C(=O)C(C3CCCC3)NC(=O)CNc3nccs3)CCN2C1 34729,C1(C(C)C(=O)NCC=CCC(=O)NC2CC(C(F)(F)F)C2)CCC(=O)N1 34730,N1(C(Cc2cc(C)on2)=O)CCCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34731,c1(C(N2C(C3CN(C(=O)C=CC4CCOC4)C3)CCCC2)=O)ccc2ccnn2c1 34732,CCC(F)(F)CC(=O)NC1CC1NC(=O)C(c1ccnn1C)O 34733,c1(C(=O)NC2CCCC(C(=O)Nc3cncs3)CC2)cccn2nccc12 34734,C1(Cn2cc(C(C=C)(C)O)nn2)CCN(C(=O)C(c2ccccc2)F)CC1 34735,C(=O)(C(C)(C)C(F)(F)F)N1CC(O)(CN(c2ccc(Cl)c(C(F)(F)F)n2)CC)C1 34736,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34737,CCC(C)(CNC(=O)CCc1cnccn1)C(=O)NOCC(C)O 34738,c1(SC)ccc(NC(=O)NS(=O)(=O)CC2CCCC(C)O2)c(Cl)c1 34739,C1(CC)(CC)CC(C(=O)N(C)CCOCCC(=O)NC(C2CCCOC2)C)C1 34740,CCC(C)CCC(O)CC(=O)NCC1CCCN1C(C12CCC(CC1)C2(C)C)=O 34741,N1(C(c2nc(C(C)C)sc2)=O)CC(C)(C)CC1CNC(C1CCCCC1(C)C)=O 34742,C1(NCc2c(C)cc(C(=O)O)cc2)CCCCC1S(C)(=O)=O 34743,c1(COC)ccc(C(=O)N(C(C)CN(C)C(C2(C(C)C)COC2)=O)C)o1 34744,N1(CC(=O)N(CC)C(=O)CN2CCCCC2)CCN(C)CC1.Cc1conc1S 34745,Cc1nn(C)c(C)c1CC(=O)NC1CN(C(C2CC2F)=O)CC1C 34746,Cc1nc(=NC(=O)Nc2nn(-c3ccccc3)nc2C)n(C)[nH]1 34747,N1(C(COCCOC)=O)CCC1CC(=O)NCc1cnsc1 34748,N1(C(C2CN(C)C2)=O)CCC12CN(C(c1nc(O)[nH]c(=O)n1)=O)C2 34749,C(C(C)(C)CCC=C)NC(CCC=CCC)(C)c1nnnn1CC1CCOCC1 34750,C1(NC(C2(CC#C)CC2)=O)CC2(CCN(C(c3cn4ccccc4n3)=O)CC2)C1 34751,N1(C(CC(=C)Br)=O)CC(CNC(=O)CC(CC)C2CCC2)C(C)C1 34752,C1(NC(=O)CC2CCN2C(=O)CSc2ccccc2F)Cc2ccccc2C1 34753,O=C1CCN(C(C2(c3ccc(CCS(=O)(=O)C(F)F)cc3)CC2)=O)c2sccc2C1 34754,C1(C2CCN(C(=O)OC(C)(C)C)C2)(OC)CC1.C1(C)CCN1 34755,C=CC(C)(CC)C(=O)NCC1CC(NC(=O)C(C(=O)OC(C)(C)C)C2CC2)C1 34756,c1(C(N2C(C(=O)NCC#N)CC2)=O)cc(S(N)(=O)=O)c(F)c(F)c1F 34757,c1(C(=O)NCCCNCCC2CCC(C#N)C2)cc(F)cc([N+](=O)[O-])c1 34758,C1(C2CCN(C(C3(F)CC3C)=O)CC2)(NC(CN(CC(C)(C)C)C)=O)CCC1 34759,Cc1nc(Cl)[nH]c(=NC2CC(CNC(c3cncn(C)c3=O)=O)C2)c1F 34760,c1(C(N(CC(=O)Nc2cccc([N+](=O)[O-])c2)CC)=O)cnc2c(c1)c(C)nn2C 34761,C1(C(=O)NC23CC2CN(C(=O)CCc2ccsc2Cl)C3)CCCC1C1CC1 34762,Cc1[nH]nc(C(N2CCCC2C(=O)NCC2CCSCC2)=O)c1C 34763,C(=O)(CC(C)(C)OC)N(CCNC(=O)Cc1csc(-c2cn[nH]c2)n1)CC 34764,C(=O)(C(C1CC1)N(C(=O)CCc1ccsc1)C)N(CCCF)CC 34765,Cc1cc(=O)c(C(=O)NC2CC2CNC(c2cn(C)nc2C2CCC2)=O)cn1C 34766,CCCC(CNC(C1CCC2(CCC2)O1)=O)C(=O)N1CC2CCC2C1 34767,c1(C(C)NC(C2C=CC(NC(=O)NC3(c4cccs4)CC3)C2)=O)ccccc1 34768,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 34769,CCCC(C)CCCC(=O)NC(c1cnc(Br)c(OC)c1)C 34770,C1(C(=O)NCC2COCC(C)O2)(NC(c2cn(CC)nn2)=O)CCN(C)C1 34771,N1(C(=O)CC2CCC(F)(F)C2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC2C1 34772,c1(-c2cccc(OC)c2CO)ccc2oc(C(=O)NCCc3nccs3)cc2c1 34773,c1(CC)noc(CC)c1CC(N1CC(N(C)C(C2CCCCNC2)=O)C(O)C1)=O 34774,C1(NC(C2CCCCO2)=O)CCC2CC1CN2C(C1(C(F)(F)F)CCCCO1)=O 34775,Cc1nc(C2CC2)nc(N(C)C)c1N1CCCCC(CNC(C2CCN(C)C2)=O)C1 34776,C1(NC(=O)CC2CC23CC3)CCCC1NC(=O)Cn1ccc(Br)n1 34777,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(NC(=O)COC1CCCCC1)C2 34778,C#CCC(C)(C(=O)N(C)CC1CCCS1)NC(c1cc(C#N)cs1)=O 34779,C1(C(N2C(CNC(CNC3CCCC3)=O)CC2)=O)CCc2ncnc(C)c2C1.CO 34780,CCCCCCC(=O)N1CC(N(C)C(c2c[nH]nc2C(C)(C)C)=O)C(F)C1 34781,C(C1=CCN(C(C2CC(C)CN(C(C3C(C)(C)C3(C)C)=O)C2)=O)CC1)OC 34782,CC1=C(C(=O)N2CC3CCC3(CNC(C3CC3c3cncs3)=O)C2)CCCO1 34783,CC1C(NC(=O)CCC2CCC(=O)N2)CCCN1C(c1cn(C)c(=O)n1C)=O 34784,C(=O)(CC1c2ccccc2C(=O)N1C)NCCNC(Cc1cccc(OC)c1)=O 34785,Cc1ccc(C(F)(F)C(=O)NC2CC(C)N(C(c3cc(Br)c[nH]3)=O)C2)cc1 34786,S(=O)(=O)(c1ccc(=NCCS(=O)(=O)N2CCCC2)[nH]c1)N1CC(=O)N(CCO)CCC1 34787,c1(C(=O)NC2CN(Cc3cnc(CCCC)[nH]3)CC2O)cc(Cl)cc(F)c1Cl 34788,Cc1cc(C(N2CC(CNC(=O)CNC=O)CC(C)(C)C2)=O)c(C)nc1C 34789,C(C)(C(O)C(=O)N(C)Cc1nnc(-c2ccc(C(F)(F)F)cc2)o1)OC 34790,C(=O)(C1=CC(C)CC1)NC(C)CCNC(c1ccn(C2CCC2)n1)=O 34791,C12(CC)CC(CN(C(=O)CC3CCCCN3C(=O)COCC(C)C)C1)C2 34792,CC1CCN(C(C2(CCN(C)C)CC2)=O)CC1NC(C1CCN(C2CC2)CC1)=O 34793,CC1CN(C(c2cnc(Br)s2)=O)CC1NC(C12CC(C#N)(C1)C2)=O 34794,C12(COC)CC(OC(C)(C)C)(CN1C(=O)Nc1cccnc1SC(F)(F)F)C2 34795,C12(OC(COCC=C)C(=O)OC)CC3CC(C1)CC(O)(C3)C2 34796,CCCC(C(=O)O)N(C(=O)CC1CCN(C2CC2)CC1)CC 34797,c1(C(N2CCC(N(C)C(C3CCCCCCC3)=O)CC2)=O)c2c(nn1C)CCSC2 34798,c1(NC(CNC(c2ccn(C)c2)=O)(C)C)cc(C(C)(C)C)nc(Cl)n1 34799,c1(C(=O)NC(CN(C(C(C)SCCCC)=O)CC)C)cnc(CC)[nH]1 34800,c1(N(CC(F)F)C(C2(C)CC(=C)C2)=O)cc2cc[nH]c2cn1.C1(C(=O)N)CCC1 34801,Cc1cnc[nH]c1=NCCCC(C)NC(c1cnn(CCN(C)C)c1)=O 34802,c1(NC2C(C)CCN(C(C3CC3c3ccccc3)=O)C2)ncnc2sccc12 34803,C1(NC(COC)=O)CN(C(=O)Cc2scnc2C)CC1CC1CC1 34804,c1(C(=O)N(c2cccc(C(N)=O)n2)C2CC3CC2CN3)ccc(F)cc1Br 34805,N1(C(C2C(CN(C)C)C2)=O)CC2(C1)C(NC(=O)C=C1CCC1)CCS2(=O)=O 34806,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 34807,CCC(CC(=O)NC(CCOCCO)C(=O)NC1CCCC1CC)N(C)C 34808,c1(NC(c2cc(CC)sc2C(F)(F)F)c2n(CCC)nnn2)cc(Cl)ccc1CC 34809,C1(C(N(C)CC2CC(F)C2)=O)CCC(C2CC2)N1C(c1ccc(O)cc1)=O 34810,c1(-c2nc(C3C(C(N4CCC(C#N)CC4)=O)C3)[nH]n2)ccc2ccccc2n1 34811,CCCCCC(O)C(=O)N(C)CCc1cn(-c2ccc(C#N)cc2)nn1 34812,C1(CN(C)C(c2ccc(N3CCC(F)(F)C3)s2)=O)CCCCN1C(=O)C(N)=O 34813,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 34814,C1(C(CNC(CC(=O)NC)=O)C)CCN(C(=O)C(C)CN(C)C)CC1 34815,c1(CC(C)C)ccc(C(=O)Nc2cccc(NC(=O)CC3CSCC3)c2)cn1 34816,Cc1oc(-c2ccccc2)nc1CC(N1CC(CC(C)NC(C2CCC2)=O)C1)=O 34817,C(=O)(NNC(=O)C1CC1c1ccc(Cl)cc1)N1C(CN)CCC1 34818,Cc1c(C(=O)NC2CCCC23CN(C(C2CC4(CCC4)C2)=O)C3)sc2ccccc12 34819,N(C1CCCc2c1cnn2CCc1ccccc1)C(c1cc(C)c(O)c(C)c1)C 34820,C(=O)(C1CCSc2ccccc21)N1C(C)CCN(C(c2cnn[nH]2)=O)CC1 34821,c1(C(NNC(C2C(C)OCCO2)=O)=O)cc(=O)c2cc(Br)ccc2o1.C1COC1=O 34822,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 34823,C(CC(C)C(=O)NCc1ccnc(C(=O)NC2CC2)c1)=CC.C1CCOC1 34824,C(=O)(CC(C(F)(F)F)N1CCOCC1)OCCOC(C1(F)CCC(F)(F)CC1)=O 34825,O(NC(=O)C(C1CC=CCC1)NC(C1C2CCC(F)C12)=O)CC(C)(C)O 34826,c1(OC)cccnc1-c1cn(C2CCCC2NC(C2CC(=C3CC3)C2)=O)nn1 34827,N1(C(=O)C=Cc2ccccc2)CC2(CCC2)CC1C(N1CCC(CO)C1)=O 34828,c1(NCC2C(NC(c3nccc(Cl)c3F)=O)CCCC2)ncnc2cc(Br)sc12 34829,CCCC(C)CCCC(=O)NCC1CN(C(=O)Cc2cc(Cl)n(C)n2)CC1(C)C 34830,CC1CN(C(=O)CC2(O)CCOC2)CC(C)CN1C(C1CC12CC(O)C2)=O 34831,Cc1cc(C=CC(N2CCCC2(C)CNC(=O)C(C)NC(N)=O)=O)on1 34832,C(C(C)S(N)(=O)=O)NC(C1(NC(C(C)=CC=C)=O)CC1(C)C)=O 34833,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(C2C(C(=O)OC)C2)=O)C12CC2 34834,N1(C(CCCN(CC(F)(F)F)C)=O)CCN(C2CCCN(C(=O)C=CCF)C2)C(=O)C1 34835,C12(C(=O)NCCCCNC(C(c3cccnc3)C)=O)CCC(O1)c1ccccc12 34836,C1(NC(C=COCC)=O)CN(C(c2cnn(C(C)C)n2)=O)CCC1CO 34837,N1(Cc2nc(-c3ccc(CC)cc3)on2)CCC(CC(N)=O)C(F)(F)C1 34838,c1(C(C)C)cc(C(=O)NCCN(C)C(c2cnc(N)cn2)=O)cc(O)n1 34839,CCC(C)C(=O)C(=O)N(C)CC=CC(=O)NCC1OCCC1(C)C 34840,N1(C(C2(F)C(C)C2)=O)CCC(CO)(CNC(C2(c3ccno3)CC2)=O)C1 34841,c1(C(=O)NC2CN(C(C3N(C(CC)=O)CCCC3)=O)CC2C)c(Cl)ccnc1C 34842,S(=O)(=O)(c1c[nH]c(=NCCN(C)C2CC2)cc1C)NCC1CCN(CCC)C1 34843,C12(C(=O)NC(CC=C)CNC(C3CCC3)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 34844,Cc1cc(C(N2CC(CN(C(=O)CCN3CCCCC3)C)C2)=O)cc(C(F)F)c1 34845,c1(CC2N(C(=O)NC3CCCOC3)CCC2)c(F)ccc(F)c1Cl 34846,C1(O)(CN(C)C(C2(CO)CCCCC2)=O)CCCN(C(=O)COCCCF)C1 34847,c1(C(=O)NCC(CNC(C#CC(=O)N(C)C)=O)(C)F)ccc(F)cc1C 34848,c1(CC(=O)NCC=CCNC(C(C)CCN(C)C)=O)csc2ccccc12 34849,c1(C(=O)NCC2N(C(c3c(Cl)c(C)n(C)n3)=O)CC2)cncc2c1CCCC2 34850,N(C1CCOc2ccc(O)cc21)C(c1c(C)cc(CO)o1)=O 34851,Cc1ccc2c(c1)C(=O)N(CC(=O)NCC1COCCN1C(C1CC1C)=O)C2=O 34852,N1(C(C(C=C)C)=O)CC=C(C(=O)N2CCC(c3cccc(C#N)c3)C2)C1 34853,c1(SC)cccc(Cn2nc(C)cc2C)c1O.N12CCCC(C1)c1nc(cs1)C2 34854,N1(C(CC2C(C)CCO2)=O)CC(CNc2ncc([N+](=O)[O-])cn2)OC(C)(C)C1 34855,N1(C(C2(CO)CCN(C(C3CC(C)(C)C3)=O)C2)=O)CCCC(N=[N+]=[N-])CC1 34856,CCCCCCC(C)(CCC)C(=O)NC1(CNC(=O)CC(C)F)COC1 34857,C1(NC(Cc2nc(CC)sc2)=O)CN(C(=O)CC2C(=O)NN=C2C)C2(CCC2)C1 34858,Cc1noc(CN(C)C(=O)NCc2ccn(CC(F)(F)F)n2)n1 34859,C(CN=c1[nH]c(=NCCC2(CO)CCC2)c2ncccc2[nH]1)C1CC(C)OCC1 34860,C(CCCC(=O)N1CC(O)CC1C)NC(c1c(CCC)[nH]cc1)=O 34861,C1(C(N(C(CNC(COCCCC(C)C)=O)C2CC2)C)=O)CCCCC1(F)F 34862,N1(C2CCN(C(CC3C(C)C3)=O)CC2)CCC(NC(C2(CCN(C)C)CC2)=O)CC1 34863,N1(C(=O)NCC(C)SC)CCC(O)C(C)(O)C1 34864,c1(OC)nccc(COC(=O)N(C)C(c2nc(C)cs2)C)c1F 34865,CC1CC(NC(=O)Cc2c(F)cccc2Cl)CN(C(c2cccc(F)c2O)=O)C1 34866,N1(CC(=O)N(C(CC)(C)C)C)CCC(N(C)C)C(CO)C1 34867,C(=O)(CC(C)C(=O)OC)NC(c1ccc(CNC(c2ccc(CC)o2)=O)cc1)C 34868,c1(NC(c2nnnn2C(C2CC2)C2CC2)(C)CC2CCC2)ccccc1I 34869,c1(OC)cc(C(=O)NC2CC(NC(=O)C(C)N(CC(F)(F)F)C)C2)cc(C)c1 34870,C1(CNC(CCc2onc(C)n2)=O)CC(O)CN1C(c1cc(C(N)=O)cs1)=O 34871,C1(C)(NC(c2cn(CC#C)nc2)=O)CCCN1C(=O)CCOCC 34872,c1(C(=O)NCC2(F)CC(NC(c3cncc(NC)c3)=O)C2)c(F)ccc(C)c1F 34873,N1(C(CN(CCC)C)=O)CCC(C(=O)NCC(C)C2CCC2)C(O)C1 34874,c1(CC(=O)NCC(CNC(C(C)SCCCC)=O)C)ccc(-n2ccnn2)cc1 34875,c1(CC(=O)NCC2C3CCCC2N(c2nnco2)C3)cc2ccccc2o1 34876,CC1CCC=C1C(=O)N1CCC(C)(C)C1CC(=O)NOCCC(F)(F)F 34877,c1(CC(=O)OC)cccc(C(=O)NCC2CCCN2C(c2ccsc2Br)=O)c1O 34878,O=C(O)CCC(F)(F)C(=O)N1CC2CC1CN2C(=O)Cn1cc(F)ccc1=O 34879,c1(C(N(C(C)CNC(=O)C(C)N2CCCC2)C)=O)cc(Cl)cc(Cl)c1 34880,N1(C(c2cccc(SCCC)c2)=O)CCCC2CN(C(=O)COCC)CCC12 34881,C=CCC(C)C(=O)N(C1CCCN(C(=O)C=C(C)CCC)C1)CCO 34882,c1(OC)cc(N(C)C)ccc1C(=O)NC(C)CC(C)NC(=O)C(C1CCC1)OC 34883,C1(C)(OCC)CC(NC(C23CC(n4cc(C5(F)COC5)nn4)C2C3)=O)C1(C)C 34884,C1(C(=O)NCC2N(C(c3c(OC)nsc3)=O)C3C(C2)C3)Cc2ccccc2S1 34885,C1(NC(CC(C)OC)=O)C(C)(C)CN(C(=O)CN2CC3C=CC2C3)CC1(C)C 34886,CCCCC(F)C(=O)NCCOCCC(=O)NCC(CC)(CC)CO 34887,C(=O)(C(F)(F)C(C)O)N(C(C)CCNC(c1cc(F)cc(Cl)c1)=O)C 34888,c1(NC(c2n[nH]c(C3CC3)c2Br)=O)ccc(N2CCCS2(=O)=O)cn1 34889,C=C=C(C)CC(=O)NC1(CF)CCN(C(c2cnn(C(C)CC)c2C)=O)C1 34890,C(CC(C)(C)C(=O)N(CC(N1CCOCC1)=O)C)NC(=O)OC 34891,c1(C(N(CC(C)NC(C(C)=C2CCC2)=O)C)=O)c(F)c(Cl)cc(Cl)c1Cl 34892,N1(C(c2ccc(N3C(=O)OCC3)s2)=O)CCC2(NC(=O)Cc3cc[nH]c3)CC2C1 34893,c1(OC)ccc(C(=O)N(CCCN(C)C(c2c(F)cccc2F)=O)C)c(O)c1 34894,C1(C(=O)NCC2CCCN2C(=O)CN2CCSCC2)CCCCCC1(F)F 34895,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)C(c2cccc(O)c2)(C)C)CC1C1CC1 34896,c1(CC)[nH]c(=NCC2CCCC(C(=O)NCCOCCO)C2)sc1C 34897,c1(OCCCC)c(C(=O)N(CC(C)C)Cc2cnc(C)nc2C)cccc1Br 34898,CCCCCCCCC(=O)N1CC(CO)(NC(C2CCCCC2C(N)=O)=O)C1 34899,Cn1cncc1CCNC(C1(C)CCN1C(=O)COC(C)(C)C)=O 34900,C1(NC(C=CCCCCC)=O)CCN(C(=O)CN(C)C)C1C(C)C 34901,N1(C(C2CC23CCC3)=O)CCC(CNC(=O)C(F)(F)c2cnccn2)CC1 34902,CN1N=CC(CC(=O)N(CC(CO)(CO)NC(=O)CCc2cn(C)cn2)C)C1=O 34903,CCC(CC)CCCC(=O)N1Cc2[nH]nc(C(=O)NC3CCN(C)CC3)c2C1 34904,N1(C(=O)N(C(n2cc(SCC)nn2)C)CC)C(C)(C)C1(C)C 34905,Cc1ccc(CCCC(=O)NCC2CCN2C(C2CCCC2O)=O)s1 34906,C1(C)(CCNC(CCCC)=O)CCCN1C(=O)CCOCCOC(C)C 34907,N1(C(c2c(C)noc2)=O)CCN(C(=O)CCn2cccn2)CC1CO 34908,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(C(C2CC2)OCC)=O)CC1(C)C 34909,CCC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)CC2(CO)CC2)CC1 34910,c1(C(=O)Oc2cnn(CC(F)F)c2)noc2ccc(Cl)cc12 34911,N1CCCC1(C)C(=O)NCCSCCOC(C1(CC)CCC1)=O 34912,C12CC(F)(C1)CNC(=O)C1(CC1)C(C)ONC2=O.C1(NC(N)=O)CCCCC1 34913,c1(C(N(C(C)CNC(=O)Cc2cc(C)ns2)CC)=O)ccn(O)c(=O)c1 34914,C1(C)(c2cn(C(C)(C)CO)nn2)CCCN1C(C1CCC(C(=O)C2CC2)O1)=O 34915,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 34916,C1(NC(c2c(CC)n[nH]c2)=O)CCCN(C(c2ccsc2-n2cnnn2)=O)CC1 34917,c1(Nc2nnc(CSCC(=O)OC(C)(C)C)s2)cc(F)c(Br)c(Br)c1 34918,O=C(CCC(O)c1ccccc1)NC1C2CN(C(=O)C=CBr)CC12 34919,c1(CCN(CC(=O)NCCN(C)C)CC)c[nH]c(C(=O)NOCC2CCCC2)c1 34920,N1(C(C2(COC(C)C)CC2)=O)CC(C2CCCCN(C(C3COCCO3)=O)C2)C1 34921,c1(C(=O)NC2CCC(C)(CNC(c3cn(CC)nc3C)=O)C2)nnc(O)cc1O 34922,N1(Cc2c(N(C)C)ccc(Br)c2)CC2(CN(C(=O)Cn3ccnn3)CCO2)C1 34923,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 34924,N1(C(COCCNC(C(C2CCCCC2)C)=O)=O)CCC2(CC(F)C2)C1 34925,N1(C(C(CC)=CCCC)=O)CCC(O)(CNC(C2CC(O)C2)=O)CC1 34926,CC(C)CCCOCC(=O)N(CC(=O)N(C)CC1(C)CC1)C1CCC1 34927,N1(C(C(C)NC(=O)OCC)=O)CC(NC(c2nn(CC)cc2Cl)=O)C(C)(C)C1 34928,C12(C(=O)NC(CCN(C(C3(COC)CCOC3)=O)C)C)CC(CO)(C1)OC2C 34929,O=C(CCCC(F)(F)F)NC1CC(O)CN(C(=O)COC2CCOC2)C1 34930,c1(CC)oc2ccccc2c1C(=O)N(CC(CC)NC(C1CC2CC1CO2)=O)CC 34931,c1(-n2c(C3C(C)CC(C)C3O)nc(-c3cccnc3)n2)ccc2cccnc2c1 34932,CCCCCCC(C)C(=O)NCC1CC(F)(F)CN1C(=O)C(F)C1CC1 34933,C12(C(=O)NC(C)C(CO)NC(=O)C=CSc3nc[nH]n3)COCC1C2(F)F 34934,N1(C(C2(CC)CCC2)=O)CCCCC1CN(c1ccnc(SC2CC2)n1)C 34935,C(=O)(CCS(C)(=O)=O)NCC(=O)NCC1(C(C)OCC)CC1 34936,CN=c1ccc(C(=O)NCC(C2CCN(C(=O)CC3CCC(C)C3)CC2)C)c[nH]1 34937,c1(OC)cc(C(C)C(N2CCCC(C)(NC(=O)CCCC3CC3)C2)=O)ccc1C 34938,c1(C(N2CC(CC=C)(NC(c3ncc[nH]3)=O)C2)=O)cnn(C(C)C)c1C 34939,N1(C(c2cccc(Cl)c2)=O)CC(C2CCCN(C(C3CCCCS3)=O)C2)C1 34940,c1(N(OC(F)(F)F)C(c2cnc(C(C)C)s2)=O)ccc(Br)cc1N=[N+]=[N-] 34941,c1(CC)ccc(-n2nc(-c3ccc(OC)nc3)nc2-c2coc(SC)c2)cc1 34942,C1(F)(CS(=O)(=O)NCC2(O)CCCC2O)COCCOC1 34943,N1(C(c2cn(C(C)C)nn2)=O)CC2CCC(CNC(=O)CCC(F)(F)F)C2C1 34944,N1(C(c2c(C)nsc2)=O)CCCC2(NC(=O)CSC(C)(C)C)CCCC12 34945,N1(C(Cc2n[nH]c(=NC)s2)=O)CC=C(CNC(c2cc(OC)ccc2F)=O)CC1 34946,N1(C(CSC)=O)CC2CCC(C1Cc1ccccc1)N2C(=O)C(C)OC(C)C 34947,c1(CC)nc(-c2ccccc2)[nH]c1C(=O)NCCN(C(=O)Cc1nnc(O)s1)C 34948,[N-]=[N+]=NCC(C(=O)NC1(C2CC2)CCC1)NC(C1CS(=O)C1)=O 34949,C12(NC(=O)COC3CCCC3)CCN(C(c3cccc(O)c3Cl)=O)CC1C2 34950,C#CCCC(C(=O)N(C)CP(C)(C)=O)NC(=O)CCCCCN(C)C 34951,n1(CC)cnc2[nH]c(=NCCCN=c3cc[nH]cc3)nc(Cl)c12 34952,C1(C(N2CC3(CCNC3)C2)=O)CCCC12CCN(S(=O)(=O)CCCCCl)C2 34953,c1(NC)ccc(Br)c(C(N2CC(=O)NCC2C(N)=O)C(=O)NCC2CCOC2)c1 34954,O=S(=O)(c1cccc(F)c1F)N1CC2CN(Cc3ccc(F)cc3Cl)CC12 34955,c1(NC(=O)CCCC2CCN(C(=O)NC3C(C)CCC3)C2)c[nH]nc1[N+](=O)[O-] 34956,N1(C(c2cnn(CC)c2C)=O)CC2(C)CC1(C(=O)N(C)Cc1ccccc1C)C2 34957,N1(C(C=C(CC)CC)=O)CC2(CC2)CC1CNC(=O)C(C)OCC(F)(F)F 34958,C(=O)(C#CC1CCOC1)NC1(NC(CSC(C)(C)C)=O)CCOC1 34959,Cn1ccc(C(N2CC(NC(=O)CCC(=O)N(C)C)CC2CO)=O)cc1=O 34960,C1(NC(C2(F)CCN(C(c3cc(C)nc(C)c3)=O)C2)=O)CCOC2(CCC2)C1 34961,CC1(C)CC(O)(C(=O)NCC(C2CCCC2)NC(=O)CC2CCCOC2)C1 34962,C1(C(=O)NCc2cc(C(=O)N(C)CC3CCN(C)C3)n[nH]2)(OC)CCC(C)C1 34963,Cc1cc(F)c(C(N2CC3CN(C(=O)C(n4ccnc4C)C)CC23)=O)c(F)c1 34964,Cn1nc(C(=O)NC2CCCC2CNC(C2CC(=O)N2)=O)c2c1CCC(C)(C)C2 34965,N1(C(COCCCC)=O)CC2C(C(N3CCCC3C(=O)OC)=O)C2C1 34966,Cc1nccc(C(=O)NCC2(NC(=O)CNC(C3CCCCC3)=O)CCOC2)c1O 34967,N1(C(Cc2ccc(C)o2)=O)C2CCC1CC(CCNC(=O)C(C)CCO)C2 34968,c1(CC(=O)NC2C(NC(c3c(C)n[nH]c3C)=O)CC2)c(F)cccc1Cl 34969,S(C1CCc2c(F)cccc21)c1ncc(Br)c(N2C3COC(=O)C(C3)C2)c1F 34970,C1(OC)CC2(CCC(C(N3CC4CCN(C=O)CC4C3)=O)CC2)C1.C(C)(C)(C)NC 34971,C(CC(CC)C(=O)NCCN(CCCN(C)C)C(c1cc(F)n[nH]1)=O)=CC 34972,CCCCCC(C)CC(=O)NC(CN(C(=O)CN1C(=O)C(C)C(C)C1=O)C)CC 34973,CCC(C)C(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(N2CCC3CCCCC23)=O)C1 34974,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 34975,C1(CNC(C2CCC(CCCCC)O2)=O)CC(NC(C2CCCCC2)=O)CC1O 34976,N1(C(C2C(C)(C)CO2)=O)CC2CN(C(c3cccc4c3COC4)=O)CC2C1 34977,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 34978,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)Cc2cc[nH]n2)CC2(CC2)C1 34979,CCCCCCC(F)C(=O)NCC(F)CNC(=O)CC12COC(CF)(C1)C2 34980,c1(C(=O)NCC2N(C)CCN(C(=O)C=C3CCC3)C2)cnn2ccn(C)c12 34981,C=CCCCCC(=O)N1CCC(OCC(=O)NC(CCF)C(=O)OC)C1 34982,C=CCC(CC)C(=O)NC1CC(C(=O)N(C(C)C(N)=O)C)CC1O 34983,c1(-c2n(CCC=C)ccn2)cc(C2NC(=O)NC2=O)ccc1OC 34984,Cn1nccc1C(=O)NCCC(O)CNC(c1c[nH]c(Br)c1)=O 34985,CC1CCN(CCCC(=O)N(C2CCN(C(=O)COCC3CC3)C2)C)CC1 34986,CCC(CCCC(=O)N1CCCCC1CCO)NC(=O)C(C)(C)N(C)CC 34987,Cc1nn(C)c(C)c1-c1ncc[nH]1.c12nccc(n1)ON2C(C)C.c1(C)cnn[nH]1 34988,N(C(=S)N1CC(CO)CC(C)C1)c1ccc(OC)cc1Cl 34989,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NCC1(O)CN(C)C1 34990,S(=O)(=O)(c1cc(C(=O)NCC(C)N(C(=O)Cc2cn3ccsc3n2)C)co1)NC 34991,c1(C(=O)NC2(C(F)F)CC(NC(C3C(C(=O)OC)C3(F)F)=O)C2)nc(C)c(C)s1 34992,C1(CCN(C(C(C(=O)OCC)(C)CC)=O)C)CCc2ncnc(C)c2C1 34993,N1(C(C2CCC(CC)CC2)=O)CCC(C)(C)C(NC(c2sc(F)cc2C)=O)C1 34994,C(C1=NOC2COCC12)NC(CCN(C(=O)CCCC1CCCO1)CC1CC1)=O 34995,CC1CCC(CO)N(C(=O)C(=O)NN2CCC(c3nccn3C)CC2)C1 34996,c1(OC(CC)C(=O)NCC(C(C)C)NC(C2CC3(C2)CC3F)=O)cccc(F)c1 34997,c1(C(=O)NCCOCCCNC(C2C(C)C2C)=O)cc(C2CC2)cnc1Cl 34998,C12(CNC(c3c(CC)non3)=O)CCCN(C(c3c(C)n[nH]c3C)=O)C1C2 34999,c1(C(N2CC3(CCN3C(C3(F)CCNCC3)=O)C2)=O)ccc(Cl)c(F)c1F 35000,c1(OC(N2CC(OCCSCCC(F)(F)F)C2)=O)ccc(Br)cc1 35001,C1(CC(NCP(OCC)(C)=O)=O)CN(C(c2ccnc(COC)c2)=O)CC12CC2 35002,N1(C(c2n(C)c(S)nc2)=O)CC2CN(C(c3cc(Cl)no3)=O)CC2(C)C1 35003,N1(C(=O)CCC2CC2)CCC2(C1)CN(C(=O)CS(=O)c1ccc(Cl)cc1)CCO2 35004,N1(C(C(CC)(C)OC)=O)CC2=C(C1)CN(C(c1cnc(C(C)(C)C)[nH]1)=O)C2 35005,c1(OCC)cc(C(=O)NC2CN(C(=O)Cc3csnc3C)C2)[nH]n1 35006,N1(c2c(OC)cncn2)CCCC(N(C)C(c2cnc(Cl)cc2I)=O)CC1 35007,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35008,c1(N(CCN(C(=O)CNC(=O)OC(C)(C)C)C)C)cccc(Br)n1 35009,C(=O)(C(O)C(F)(F)F)N1CCC(CCC2N(C(CC3C(C)(C)C3)=O)CCC2)CC1 35010,c1(NC2C3(CC(NC(c4cnc(C)nc4)=O)C3)C2)ncnc2cccc(Br)c12 35011,c1(C(N2C(CNC(CSCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35012,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35013,C1(C(=O)OCC)CN(C(=O)C(C)N(C)C(c2occc2C)=O)C(C)(C)C1 35014,C1(C(N(CCCCC)CCO)=O)CN(C(=O)CCCOc2ccc(C)cc2)CCS1 35015,C(C1OCc2ccccc21)NC(=O)NC1(n2ccc(C(F)(F)F)n2)CC1 35016,C1(NC(CCCCNC(C)=O)=O)CC2(C1)CN(C(c1nccnc1Cl)=O)C2 35017,c1(OC)ccc(C)nc1C(=O)NCC1CC1NC(c1ccc(C(C)C)cc1C)=O 35018,C1(NC(C2C(C)CCC2)=O)CCC(NC(c2ncoc2C2CCC2)=O)CC1 35019,c1(OC)nccc(C(=O)NC2CC23CC(NC(=O)C#CC2CC2)C3)c1F 35020,N1(C(C(C)=CC2CC2)=O)CCCC(NC(=O)Cc2csc(S)n2)C(F)C1 35021,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1nc(O)ncc1C)=O)CCO2 35022,C(c1cccc(O)c1)=CC(=O)NCc1cccnc1CN1CCC=C(Cl)C1 35023,c1(CC2CCCO2)sccc1Cl.N12CCCC1Cc1cn(nn1)NC(=O)C2=O 35024,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35025,Cc1cc(C)n(CC(=O)NCCC2COCCN2C(=O)C(C2CCCCC2)O)n1 35026,c1(C(N2CC(CC(C)NC(C34CCC(C3)C4)=O)C2)=O)cnc2ncccn12 35027,c1(OCC(N2CC3(CN(C(Cn4ccc(C)n4)=O)C3)C2)=O)cc(N)cc(C)c1F 35028,c1(C(=O)NC2CCC(NC(CCCN=[N+]=[N-])=O)C2)cccc2ncsc12 35029,CCC(C(=O)NCC1CC(C)CN(C(=O)C(n2nccc2C)C)C1)C(F)(F)F 35030,CN1CCN(C(=O)COC2CN(C(=O)C(F)C(C)(F)F)C2)CC12CCC2 35031,N1(CCCOCC)CCC2(CCCCN(C(c3cncnc3)=O)C2)C1 35032,C1(C(N(C(CO)C2CC2)C)=O)CC12CCN(C(=O)CCC1(C)N=N1)C2 35033,c1(CC)nnc(C(=O)NCCNC(C2CCN2C(C2CCOCC2)=O)=O)s1 35034,C(=O)(C(CC(N)=O)N(C)C)N1CC(OCc2c(C)non2)C1.C1(=O)CO1 35035,c1(OCC)ccc(C(c2nnnn2C)NC(CCO)CC(C)C)cc1OCC 35036,C1N=C2C=C(N=CN2)NCCC12CC2.CC(C(C)(C)C)=C1CCC1 35037,C(=O)(CCC(C)(F)F)N1CCC(NC(C2(C=C)CC2)=O)CC1 35038,CCCC(CCC)CC(=O)NC(c1cccnc1)C(=O)Nc1cnc(C)c(C)c1 35039,N1(C(c2nc(C(C)C)oc2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC1C 35040,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35041,CC(C)(C(=O)NC1CC(OCC(=O)NC(c2ccco2)CO)C1)C(F)(F)F 35042,N1(C(CC2N(C(CC3CC(=O)NC3)=O)CC2)=O)CCOCC(CO)C1 35043,c1(NC(C2CC(n3cc(COC4C(C)CCCC4)nn3)C2)=O)cc2sccc2s1 35044,C(C)(C)(CCCC(=O)NC(CO)C1CC1)NC(c1ccc(OC)s1)=O 35045,c1(CNC(C(C2CCC(C)O2)N)=O)nc2cc(F)ccc2s1 35046,C1(C(NOCCOCC#C)=O)CCCCCCN1C(c1c(O)cccc1F)=O 35047,N1(C(C(c2ccccc2)C)=O)CC2CC(C1)N(C(c1cnc3n1CCC3)=O)C2 35048,C1(C(=O)NCCN(CCOC)Cc2cccc(OC)c2)CCCCC1O 35049,C12(CCNC(C3(C)COCCO3)=O)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35050,C12(NC(c3ccc(SC)s3)=O)CCC(C1)N(C(=O)CCCCNC(N)=O)C2 35051,c1(NCCC(=O)NC(C2(CCNC(C(C)NC(C)=O)=O)CC2)C)ccccn1 35052,C(CC(=O)N1CCC(C(C)(C)NC(c2nc(O)sc2C)=O)C1)(C(F)(F)F)OC 35053,Cc1cc(C(=O)NC(C)(C)CN(C(=O)C(c2ccc(Cl)cc2)CO)C)c(C)[nH]1 35054,C1(C(=O)NCC2(CO)CC23CCC3)C2CC3C(C2NC(c2csc(CO)c2)=O)C13 35055,N1(CCC(=O)N(CC(C)NC(c2cscc2C(F)(F)F)=O)C)CCCCCC1 35056,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(=O)Nc2nccs2)C(CCOC)CC1 35057,c1(CC(=O)NCCC(C(C)C)NC(=O)CC2CC(C)(C)C2)ccccc1[N+](=O)[O-] 35058,Cc1cc(Br)ccc1CC(=O)NCC1CC2CC2N1C(=O)CNC(=O)CC#N 35059,c1(C(N(CCCCN(C)C(c2cnc(Cl)cc2N)=O)C)=O)ccc(C(N)=O)c(F)c1 35060,c1(NCC2C3CN(C(C(c4c(F)cccc4F)C)=O)CC32)cccc2c1OCO2 35061,c1(C(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccnc(C(F)F)c1 35062,c1(OC)cc(C(=O)N(CC(C)N(C(=O)CN2CCCC2C)C)C)[nH]n1 35063,c1(N2C(CCC)SCC2)ccc(S(=O)(=O)NCC(C)(C)C)c(Br)c1 35064,C12(C(N3CC(C(=O)OC)(NC(c4nc(C)oc4C)=O)C3)=O)CC(C)(CN1CC)C2 35065,C1(C(=O)NCC23OCC(NC(C=CCOC)=O)C(C2)C3)COc2cc(Cl)ccc2C1 35066,CC1CNc2c(C(=O)NCC34CC(NC(c5ncccn5)=O)(C3)C4)cnn2C1 35067,C1(N2c3cccc(c3)C2=O)CCNCC12CC2.C1(NCC)CCOC1C 35068,C(C1CN(C(=O)CCN(C(=O)Nc2ccncc2)C)CC1C(C(C)(C)CS)=O)=CC 35069,c1(C(C(=O)NC(CC)(C)CNC(=O)Cn2nnc(C3CC3)n2)C)ccccc1F 35070,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35071,Cn1nc(C(=O)NCC2CCCN(C(=O)Cc3csc(C(=O)OC)n3)C2)cc1Cl 35072,c1(C(C)C)cc(C(=O)NC2CC(OC3CC3)C(n3cncn3)C2)n(C)n1 35073,C1(COC)(NC(C2CCOCC2)=O)CCN(C(=O)CCc2conc2C)C1 35074,N1(C(C(CC)F)=O)CC2CCOC2(CNC(c2cc(OC(C)C)ccc2Cl)=O)C1 35075,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(C(C)C)no2)=O)CC2CC12 35076,C(=O)(C1CCCc2cn(C(C)C)nc21)NCC(CNC(c1c(C)nns1)=O)F 35077,c1(OC)ccc(C=CC(=O)NCC(O)CNC(=O)C2=CCCOCC2)c(OC)c1 35078,CC(C)C(C(=O)NC1CN(C)CCC1(F)F)C(C)NC(c1ccnn1C)=O 35079,c1(CC(=O)NC2CCCCN(C(CCCCCC)=O)C2)csc2cccc(F)c12 35080,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2N)=O)CCCCC1C 35081,N1(C(C2CCCSC2)=O)CCCCC2(CCN(C(C3CC3C(F)F)=O)C2)C1 35082,c1(C(N2CC(OCC3(n4cc(CO)nn4)CC3)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 35083,c1(C(N(C2CCCN(C(c3noc(CC)c3C)=O)C2)C)=O)ccc(Cl)cc1OC 35084,Cc1ccc(S(=O)(=O)NC(Cn2ccnn2)C(=O)N2CCCCC2)cc1C 35085,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1C(C)(C)O 35086,CC1(C)C(CC(=O)NCCC2COCCO2)CCN1C(C1CCCCCC1)=O 35087,N1(C(CSCC(N)=O)=O)CC2CCN(C(c3ccnnc3O)=O)C2C1 35088,c1(C2CNC(=O)N2)ccc(-n2ccnc2)cc1.C1(C(=O)NCCOC)CCCO1 35089,c1(C(=O)NCC2(O)CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35090,c1(NCC2CN(C(c3[nH]cc(CC(C)C)c3)=O)CC2C)ncnc2c1nnn2C 35091,CON(CCC(=O)NCC(c1cnc[nH]1)C)C(=O)C1CC1Cl 35092,N1(CC2N(CCC)CCC2)CCOC(C(=O)NC(C)COC(C)C)C1 35093,c1(C(N(CC(CC)NC(C2(c3cccs3)CC2)=O)C)=O)cnc(O)n(C)c1=O 35094,O(NC(=O)CC(C)(C)CNC(=O)C(O)CCl)CC(C(N)=O)O 35095,C12(C(=O)NCCCN(C(=O)C(C)C(C)O)C(C)C)CC3CC(C1)CC(F)(C3)C2 35096,Cc1c(C(=O)NCCC2CCCCN2C(=O)C2=COCC2)cccc1CO 35097,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35098,C(CC(=O)NC(C1(NC(C2CCCC2)=O)CC1)C)OC(C)C 35099,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(CC)n1 35100,c1(NC(=O)NC(c2ccc(C#N)s2)C)cn(CCO)nc1C1CC1 35101,C12(C(N(CC)Cc3cnoc3)=O)CC(n3cc(CCCCO)nn3)C1C2 35102,C(=O)(C1CCCc2ncccc21)N1CCC(NC(CCSC)=O)C(C)C1 35103,Cc1ccc(NNC(=O)CNC(C2CCC(C(F)(F)F)CC2)=O)cn1 35104,N1(C(c2c(C)n(CCO)nc2)=O)C2CCC1CN(C(C1CC3CCCC13)=O)CC2 35105,c1(C(c2c(C)oc(Cl)n2)NC(=O)NC2CCCCC2C(F)(F)F)ccc(F)c(F)c1 35106,C=CC(C)(O)CC(=O)NC1CN(C(c2ccc(N(C)C)cn2)=O)C(C)(C)C1 35107,C1(CC)CCCCN1C(=O)C(N1CCC(OC(C(C(C)C)NC(C)(C)C)=O)CC1)=O 35108,c1(C(=O)NCCCCCCN(C(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35109,C1(C(=O)NCCCCCCC)CC12CCN(C(c1ccc(CC)o1)=O)C2 35110,c1(C(N2CCCC(CN(c3ncncc3Br)C)C2)=O)cncc2c[nH]nc12 35111,C(CN=c1cnc(C)c[nH]1)NC(C(C=C)(C)C)=O 35112,CC1CC(C(N2CCCC(C3CCCN3C(=O)CCCF)C2)=O)CCO1 35113,CC1(C)CCC(NC(C2CCC(c3ccc(Cl)cc3Cl)C2)=O)C1CO 35114,c1(C(N2CC(SC)OCC2C)C(=O)NCCOCC)cccc(F)c1C 35115,CC(C)(C)C(O)C(=O)NCC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC1(C)C 35116,Cn1nc(C(=O)NC2CCC(NC(c3coc(N(C)C)n3)=O)C2)cc1C#N 35117,c1(OC)ccc(S(=O)(=O)N2CC3CC2CN3C(c2ccc(Br)c(F)c2)=O)cn1 35118,N#Cc1cccnc1NS(=O)(=O)CC1CCC2(CCC2)O1 35119,CC(C(=O)Nc1cncc(C(F)(F)F)c1)(C(F)F)c1ccccc1 35120,Cc1cc(C(=O)NC2C3CC2CN(C(c2csnc2Cl)=O)C3)nc(O)n1 35121,CSC1=C(C(=O)N(CCNC(=O)C(CO)c2ccccc2)C(C)C)CCCC1 35122,C1(C(=O)NCc2cc(C(=O)N(CC(=O)N)C)no2)(CC)CC1(F)F.C(=O)N(C)C 35123,C1(NC(N2CC=C(C(=O)OC)CC2)=O)CCN(C)C2(CC2)C1 35124,C1(NC(C(CC)NS(CCC)(=O)=O)=O)CCN(C(=O)CC2(CSC)CC2)C1C 35125,c1(C(=O)OCC)c(OCC)cc(NC2C3CN(c4ncc(F)cn4)CC23)cc1I 35126,c1(CN(C(=O)NC(c2csc(C)n2)(CC)C)CCO)cc(C(C)(C)C)n[nH]1 35127,C1(CNC(c2cnc(C(C)OCC)s2)=O)C2CCC(C2)N1C(C1(CF)CC1)=O 35128,c1(CCC)onc(C)c1C(=O)NCCC1CN(C(=O)C(C)OC(C)(C)C)C1 35129,C12(C(=O)NCC(C)(C)C(=O)NC3CC(CF)C3)CC=CC(C1)OC2 35130,C(C(CC(F)(F)F)NC(=O)CC=Cc1ccc(F)cc1)NC(C1N(C=O)CCC1)=O 35131,c1(C)ccccc1O.O=C(O)CC(C)C1CCCCC1.c12nc(no1)CC(=O)N2 35132,Cc1ncncc1C(=O)NCCOCCn1cc(COC(C)C)nn1 35133,N1(CCNC(c2c(C)onc2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35134,C1(NC(C(C)C2(O)CCC2)=O)CCCCCC1NC(c1cc(F)ccc1F)=O 35135,CC1CC(C(=O)NC2C3CCC2N(C(c2ccon2)=O)C3)=NO1 35136,C1(C(=O)N(C)C)CCCCC(=O)NC(C)C(=O)N1.C(C(=O)OCC#C)C1CC1 35137,C1(C(N(CC(C)NC(C(c2cc(C)sc2)(C)C)=O)C)=O)C2CCCCC12 35138,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35139,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(F)F)=O)NC1C(C)COC1 35140,CCCN=c1[nH]c2c(c(=NC(C)c3ccc(Cl)cc3Cl)[nH]1)CSC2 35141,c1(C(=O)NC2C(NC(=O)Cc3ccnnc3O)CCCC2)ccc([N+](=O)[O-])o1 35142,N1(C(c2cn(CC)nc2C)=O)CCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC(O)C1 35143,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)C(C)Sc1nnnn1C1CC1)CO2 35144,CCC(C)(CCNC(=O)C(F)C1CCOC1)NC(c1cc(OC)ns1)=O 35145,C(=O)(C(C(C)OC)N(C)C)N(CCC(N1CC(CC#C)C1)=O)CC 35146,C(C(C)(CNCc1cnc(SC)n1C)CO)SC 35147,c1(C2C(CNC(C(N3C(CC)CC3)=O)=O)C2)ccc(Cl)cc1Cl 35148,C1(C(N2CCC(CNC(CCC(=C)C)=O)C23CC3)=O)COc2cc(F)ccc2C1 35149,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)Cc3ccsc3)CO2)C1 35150,c1(C(N2CCC(N(C(=O)CS(=O)(=O)NC)CC)CC2)=O)ccc2nccn2c1 35151,C1(C(N)=O)CC(C(C)(C)C)CN(C(c2ccc(Br)o2)C(=O)NCc2ccccc2)C1 35152,c1(C(N2CC(CN(C(C(CN(C)C)O)=O)C)C2)=O)cccc2c1CNC2=O 35153,c1(C(N2C(CNC(c3cc4cccnc4s3)=O)CCC2)=O)ncn2ccccc12 35154,CC1CCn2cc(C(=O)NCC(CO)C(C)(C)C)nc2C1 35155,c1(-n2c(C(C=C)O)nc(COc3ccc(CO)cc3)n2)cccc(Cl)c1C 35156,C1(CNC(=O)CCCC2CC2)CC2COCC2N1c1nc2cccnc2s1 35157,C(=O)(C1=CC2CCCCC12)N(C)CC1CN(C(=O)CCn2cccn2)CCO1 35158,c1(CNc2c(C)cc[nH]2)ccc(-c2ccc(F)cc2)c(F)c1.N12CCC(O)C1C2=O 35159,N1(C(c2cc(C)ncc2C)=O)CC2CCCC(C1)N2C(c1cccc(N)c1O)=O 35160,C1(C(N2CCCC(C(=O)NC3(COCC)CCCC3)C2)=O)CCC12CCOCC2 35161,C(=O)(C(F)CC(CC)CC)N1CCC(N(CC#C)C(c2cc(CF)on2)=O)C1 35162,C(=O)(C1CCCc2sccc21)NCC(CNC(c1c(CC)cccc1CC)=O)C 35163,N1(C(C(C)SCCCC)=O)CC(O)CC1CNC(=O)C(N1CCSCC1)C 35164,N1(C(c2ccc(C#N)cc2)=O)CC(NC(C2CCCCS2)=O)C2(CCOCC2)C1 35165,C1(CC(N2C(CNC(c3ncoc3-c3ccco3)=O)CCC2)=O)CCCS1(=O)=O 35166,C1(NC(C2(OC)CC2)=O)CCCN(C(c2ccc(C(C)O)cc2)=O)CC1 35167,c1(C(=O)NC2COCC2NC(C23COCC2C3)=O)n[nH]c2cccnc12 35168,N1(C(c2ncc(CC)s2)=O)CC(CCNC(c2cncnc2)=O)OC(C)C1 35169,C(C(C(F)(F)F)N1CCN(C(=O)CC2CSCCS2)CC1)NC(CCOCC)=O 35170,c1(C(N2CC(N(C(=O)CC3CC(C(F)F)C3)C)C2)=O)coc(Cl)c1 35171,C1(C(N(C)CCC2CCN(C(=O)CN3CCCCC3)CC2)=O)CCCCC12CC2 35172,c1(NC(Cn2ncc(C)cc2=O)=O)oc2ccccc2c1OC(F)F 35173,C(=O)(CCCCCNC(C12CC1CNC2=O)=O)NCc1c(C)cc(C)s1 35174,C1(C(=O)NCC(C(C)C)NC(c2cn3c(n2)SCC3)=O)CCC(S(C)(=O)=O)CC1 35175,C(=O)(C(F)CCC(C)C)NCCN(C(CN(C1CC1)CC)=O)C(C)C 35176,c1(C(C)C)ccc(C(=O)NC2COCCC2NC(C2CC(F)C2)=O)cc1[N+](=O)[O-] 35177,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(C2(C)CC=CC2)=O)CC1 35178,CCCCC(C(=O)NCC=CCSC)NC(=O)CCC(N)=O 35179,c12nnc(n1C)-c1n[nH]c(n1)S2.N1(CC)CC=CC1(C)C(=O)OCC 35180,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35181,c1(CC(N2CC(NC(=O)CC3(O)CCOC3)C(O)C2)=O)cc(F)cc(Cl)c1 35182,N1(C(C(C)(C)SC)=O)CCN(CCN(C(=O)C=Cc2cocn2)C)CC1 35183,c1(C(N2CCOCC(NC(C(CC)O)=O)C2)=O)cccc2ncnc(O)c12 35184,C(=O)(C1=C(Cl)CCC1)NCc1c(C(=O)NC(C)C(C)CO)nco1 35185,c1(NC(c2n(C(C)C)nnn2)CC(C)N(C)C)ccc2c(c1)COCO2 35186,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NC(c1ccccc1)CF 35187,N1(C(C(C)(C)C(N)=O)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35188,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CCC3)=O)C2)[nH]1 35189,C(C(CC(C)(C)C(=O)OC)Nc1ccc(Cc2cc(C)cc(C)c2)cc1)OC 35190,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCc3ccnn3C)C1)C2 35191,Cc1[nH]c(C#N)cc1C(=O)NCCCNC(=O)CC1COCC(C)O1 35192,C1(CNC(=O)CCCn2cncn2)CC2CCC1N2C(c1cnc(O)[nH]1)=O 35193,c1(OC)cnc(F)cc1C(=O)NC(CNC(=O)C=Cc1cccnc1)CO 35194,Cc1cccc(CC(N2CCC(CNC(C3(C)CCCCO3)=O)C2)=O)c1Cl 35195,C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(c2cc(OC)nn2C)=O)C1 35196,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CCC2)C(CCO)C1 35197,c1(C(N2CCC(N(C)Cc3ccc(F)nc3)C2)=O)cncc2cccnc12 35198,C1(C(=O)NCC2(NC(=O)Cc3cccs3)CCC2)CC12CCSCC2 35199,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(O)CCC2)=O)CC1)CCC 35200,c1(C(=O)NC2CC3CN(C(CC#N)=O)C2C3)ccc(S(=O)(=O)NC2CC2)o1 35201,C#CC1(O)CN(C(c2ncoc2CNC(C2CC3(CCC3)C2)=O)=O)C1 35202,C1(CC)C(C(=O)NCC2(O)CCN(C(c3ccc(C(F)F)cn3)=O)C2)CCN1C 35203,c1(C(N)=O)ccc(C(N2CCC(C3CCCN3Cc3nc(C(F)F)no3)C2)=O)o1 35204,c1(CC)nn[nH]c1C(=O)NCCC1(NC(=O)C(COC)OC)CC1 35205,c1(NC(CN2CCN(C)CC2)=O)ccc([N+](=O)[O-])cn1.C12CC13CCN(C3)C2=O 35206,C(=O)(CCCS(C)(=O)=O)NC(CC=C)CNC(=O)C=C1CCC(C)CC1 35207,C(=O)(C1=NNC(=O)C1)NCC(CC(=O)N(C(CC(CC)C)C)C)O 35208,c1(NC(C(C(C)O)NC(=O)CCCCN(C)C)=O)ccc(C#N)cc1 35209,c1(C(N2CCC(NC(c3c(C)ccs3)=O)CC2C)=O)cncc2sccc12 35210,c1(C(=O)NCC(CC2CN(C(C3C(C)CCCC3)=O)C2)(C)C)nsc2ccccc12 35211,CC1(C)CC2(CC2C(N2CCC(O)(CNC(c3nc(C(C)(F)F)cs3)=O)C2)=O)C1 35212,C(=O)(CCC(C)(C)F)N1CCCC(OCC(=O)N(C2CCC23CCC3)C)C1 35213,C1(CNC(=O)CC2(O)CC2)CCN(C(=O)CSc2ccsc2[N+](=O)[O-])C12CCC2 35214,c1(CC(=O)NC(C2CCCN(C(=O)CC3CC3)C2)C)ccc(F)c(F)c1 35215,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35216,CC1(C)CCCC(n2cc(CCCCNC3CCCC34CCC4)nn2)CC1 35217,CC(C)(CCC(=O)NCc1nc(=O)o[nH]1)NC(=O)CCc1nccs1 35218,c1(SCC2(NC(C3CCN(OC)C3)=O)COC2)ccc(F)cc1.C1(=O)C(C)C1=O 35219,N1(C(C=CCOC)=O)CCC(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)CC1 35220,N1(CC)C(=O)CCC1CC(=O)NCCOCCCNC(=O)CN1C(=O)CNC1=O 35221,C1(C)(CCC(=O)NCC(=O)N(C2CCCCC2)CC)CCC(=O)N1.CCCC=O 35222,n1(CC(=O)NC2(C)CC(NC(C3(CC)CCNC3=O)=O)C2)c([N+](=O)[O-])cnc1C 35223,O=C(CCC(=O)N1CCC(F)C1)NC(=O)CCc1cnc[nH]1.N1CCC(O)CC1 35224,C12(C(N3CCCC(NC(CSCC)=O)C3C)=O)CC3CC(CC(C3)O1)C2 35225,Cn1cc(CNC(=O)CSn2cc(-c3cnn(C)c3)nn2)nn1 35226,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)cc2c(s1)CCC2 35227,CC(C)S(=O)(=O)CCCN1CC(NC(C2CC3(CCC3)CO2)=O)C(C)(C)C1 35228,C(=O)(CC(C)(C)N(C(=O)C(F)CC1CCCC1)C)NC(n1ccnc1C)CC 35229,C=CC1CN(C(=O)Cn2cc(C3CC3)nn2)CC1NC(c1cc(C)c(C)[nH]1)=O 35230,N1(C(Cc2ccc3c(c2)CCC3)=O)CCC2C1CCCN2C(=O)C(C)OC(C)C.CS 35231,C=C(Cl)CC(C(=O)NCC1CCOC1(C)C)NC(=O)CCOCCOC 35232,C1(CC=C)(C(=O)NCCC(O)C2CCCC2)CCN(C(=O)C=Cc2cocn2)C1 35233,Cc1ccc2n[nH]cc2c1C(N1CC(C)(NC(c2cnc(O)c(Br)c2)=O)C1)=O 35234,N1(C(C2(CCC)CC2)=O)CC2CCC(N=c3ccc(C(=O)OC)c(OC)[nH]3)CC2C1 35235,C1(NC(=O)CC2COCCCO2)CCN(C(c2cc3ccsc3s2)=O)CC12CCC2 35236,C(=O)(C1CCCc2c[nH]nc21)NCC1CC(NC(C23CCC(C)(OC2)C3)=O)C1 35237,c1(C(N(C(C)CCNC(C2C(C)C2C)=O)C)=O)ccc2nccnc2c1 35238,C1(NC(C(COC)(C)OC)=O)CC2CC(C1)CN(C(=O)C(C)CSC)C2 35239,C1(C(=O)NC(C)CCOC)(CC)CCCN(C(c2cc(CO)nn2C)=O)C1 35240,c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc([N+](=O)[O-])c(C)cc1Cl 35241,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35242,c1(C(=O)NC2CC(NC(C(N)=O)=O)C23CCC3)nc2ncc(CCO)cn2n1 35243,C(C(=O)OC)=CCN(C)OCCCN(CCNCC=O)CC.CC=C 35244,N1(C(C2OCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1sccc1F)=O 35245,N1(C(C2C(C)(COC)C2)=O)CC2(COC(CNC(=O)Cn3nc(C)nc3C)C2)C1 35246,N1(C(C(C)(C)c2ccccc2)=O)CCCC(NCCc2ccccc2)C1 35247,CCC(CC(C)C)C(=O)NCCC1(O)CN(C(=O)Cc2ccn(CC)n2)C1 35248,O=C1CCc2cccc(C(=O)NC3CC3C(=O)Nc3ncccc3CO)c2N1 35249,C1(C)(NC(C2(C)CN(C(C=C(C)C(F)F)=O)C2)=O)CCC(=O)NC1=O 35250,C1(N(C)C(C2(C(C)(C)C)CCC2)=O)CCN(C(=O)COc2ccsn2)C1 35251,c1(C(=O)NCC2CN(C(c3c(C)nccn3)=O)CC2C)ccn(C)c(=O)c1 35252,C1(C(N(CC(=O)N(CC(C)C)CC=C)C)=O)CC2CC1CC2N(C)C 35253,N1(C(CSCC(=O)NCC(=O)NC(CC2CCCC2)CO)=O)CCC(O)CC1 35254,C=C1CCN(C(=O)CC2CCCN2C(=O)Cc2ccc(Br)cn2)CC1 35255,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)COCC(=O)NC 35256,C(=O)(C(F)CCC(C)(C)C)N(CC(C)CNC(=O)CCCCCF)C 35257,c1(C(=O)NCCC2(NC(C(CSC)O)=O)CCCC2)cncc(N(C)C)n1 35258,N1(CCC(=O)NC2CCCCC2NC(=O)CCc2cnoc2)CCC(O)CC1 35259,N1(C(C(CCOC)OC)=O)CCN(C(=O)CCCSC)C(C)C1 35260,CC1CS(=O)CCN1C(C1(F)CCN(C(=O)C#CC(C)(C)C)C1)=O 35261,C12(C(N(C)Cc3ccco3)=O)COCC1CN(C(c1cc3ncccn3n1)=O)C2 35262,C(CNC(C1(O)CCC1)=O)(CC(F)(F)F)NC(c1cccc(OC)n1)=O 35263,c1(C(C(=O)NCC(F)F)N(CCNC(C)=O)CC)ccc(C)nn1 35264,Cc1ncc(C#N)cc1NC(C1(O)CCN(Cc2ccon2)C1)=O 35265,N1(C(C(C)=C(C)C)=O)CCC2CN(C(C3(C)C=CCC3)=O)CC2CC1 35266,C1(=O)C(C)(C)C(=O)N1.C1(CCCn2c(C)ncc2)CCNCCC1C 35267,C(=O)(CC(C)CNC(=O)C(C)c1ccco1)NCc1n(C(C)C)cnn1 35268,C(CC(C)C(=O)N1CCN(CCN(C(=O)Cc2n[nH]c(=NC)s2)C)CC1)=CC 35269,CC(C)CCC(F)C(=O)NC1(CCC(=O)N(C)Cc2ccsc2)CCCC1 35270,c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC(=O)CC3)=O)C2)c1F 35271,N1(C(C2C(NC(CCc3cnc(C)o3)=O)CCCC2)=O)CCCC2OCCC2C1 35272,CCC(Cc1ccccc1)C(=O)NCC1(F)CN(C(=O)C(c2cnccn2)C)C1 35273,CCCC(CC)C(=O)NC(C)CCCNC(c1cc(=O)c(Br)c[nH]1)=O 35274,N1(C(Cn2ncc(C)c2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35275,CC(CC(C)N(C)C)N=c1[nH]c(=NC2CN(c3ccccc3)C2)c2[nH]ccc2[nH]1 35276,CC1(C(=O)NCC2CC(NC(C3CC(=O)N(O)C3)=O)C2)CS(=O)(=O)C1 35277,C1(C(=O)NC2CC(NC(C)=O)C2)CN(C(=O)CCC(=O)N(CC(N)=O)C)CCO1 35278,C(CC(=O)NCCCC(F)F)(C1CC1)NC(C(C)c1cc[nH]n1)=O 35279,CCCC(C)(CCCOC)NC(=O)Nc1nc2c(o1)CCSC2 35280,N1(C(c2cn(C)nn2)=O)CCCCC1CCNC(c1cncn1C(N)=O)=O 35281,c1(C(=O)NC2CN(C(c3c4c(n[nH]3)C(C)(C)OC4)=O)C2)ccc2cccc(F)c2c1 35282,C(C)(CCCNC(=O)C(F)n1cccn1)NC(CC1(OC)CCC1)=O 35283,C(=O)(NNc1cccc2cc[nH]c12)C1N(C(=O)OC(C)(C)C)C2C(C1)C2 35284,N1(Cc2nc(-c3ccc(C)cc3)on2)CC2CCCCN2c2ccccc21 35285,c1(C(=O)NC2C(C)CCN(C(c3csc4cncn34)=O)C2)cc2occc2n1C 35286,N1(C(C(C)=CC)=O)CCC2(CCC(CNC(C3COCC3(C)C)=O)O2)CC1 35287,N#CC1(C(=O)NCC2CCC(C(=O)N3CCCCCO3)CC2)CC2CC2C1 35288,N1(C(C2CCCC(C)O2)=O)CCN(C(=O)Cc2cc(O)nnc2O)CC1C1CC1 35289,Cc1cc2[nH]c(C(=O)NC3CC(C)CN(C(c4cc5c(s4)CCC5)=O)C3)cc2o1 35290,CC(=O)CCCCC(=O)NC(C(=O)N(C)CC1(O)CCCC1)C(C)(C)O 35291,C1(C(N2CCC(C(C)OC)CC2)=O)CC2CCC1N2C(c1csc(C)c1)=O 35292,CN=c1[nH]c(=NCCCc2ccccc2)[nH]c(=NC2CCOC3(CCC3)C2)[nH]1 35293,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35294,c1(C(=O)NCC2CC(F)(CNC(C3CC(=O)NCC3)=O)C2)cc2ccncc2o1 35295,N1(C(C(c2c(C)ccnc2)(C)C)=O)CCCC(C)C1CNC(c1nccn1C)=O 35296,c1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)C3C2C3)=O)c[nH]c2ccccc12 35297,N1(C(CCN(C(COc2cc(C)on2)=O)CC(C)O)=O)CC2(CCC2)C12CCC2 35298,C1(CN(C(C2CC(C)C2c2ccc(Cl)cc2)=O)C)CCCN(C(=O)CSC2CC2)C1 35299,N1(C(CC)=O)CCC(C)(CNC(=O)C(C(C)C)NC(C)=O)C1 35300,C(=O)(C(C)CCCC(C)=O)NCC1=CCN(C(C2CC(SC)C2)=O)CC1 35301,c1(OC)ccc(CC(=O)NCCC(O)CNC(C2CNC(=O)N2)=O)cc1O 35302,C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(c1cc(C2CC(F)(F)C2)[nH]n1)=O 35303,C=CCC(CC(=O)NC(c1nc(C)no1)C)NC(c1ccc(C2CC2)cc1)=O 35304,C1(NC(C(CC)CO)=O)C2CC3CN(C(=O)Cc4c[nH]c5ccccc45)C1C3C2 35305,Cc1ccc(C(=O)N(CC(C)(C)NC(=O)CC2C=CCC2)C)c(O)n1 35306,c1(CO)c(CNCC(O)CN2CCCCC2)ccc(Cl)c1Cl 35307,c1(NC)cc(C(N2CCC(=CCNC(C3CCCC3F)=O)CC2)=O)cc(F)c1 35308,Cc1ccc(Cl)c(C(=O)NCC(C)(C)NC(=O)Cc2ccc(F)cn2)c1N 35309,N1(C(COC(CC)C)=O)CCC(NC(c2nc3ccccc3[nH]2)=O)C(C)(C)C1 35310,C1(NC(C2C(C)CCN2C(=O)C(C)CCN(C)C)=O)(CO)CC2CCCC12 35311,CCCCCC(O)CC(=O)NCC1CC2(CC2)CN1C(=O)C(O)CC1CC1 35312,N1(CCNC(c2nc(C(C)C)oc2)=O)CCCN(C(C2CC2F)=O)CC1 35313,CC1CC(C(F)(F)F)n2nc(C(=O)NCC3CC4(CC4)CO3)cc2N1 35314,n1(CCC)nnnc1C(c1cc(COC)on1)NCCn1ccnn1 35315,Cc1nc([N+](=O)[O-])cn1CCC(=O)N1CC(CS(N)=O)C1 35316,C1(CN=C(NC(CC)C(C)C)NCC(F)F)COC2(CCC2)CO1 35317,c1(C(=O)NC2C(NC(C(C)(C)OC(C)C)=O)C2)ccc(Cl)c(F)c1O 35318,O(C1CCCc2ccccc21)CC(=O)OC.c1(CN2CC2)n[nH]c2c1CCCC2 35319,C(=O)(C(O)CCCc1cn[nH]c1)NCC1C(NC(CN2CCN(C)CC2)=O)CC1 35320,N1(C(c2nc(C(N)=O)sc2)=O)CC2C(NC(=O)CC(=O)NC3CC3)C2C1 35321,c1(N(CCNCC2N(CC)CCC2)C)ccc(C)c(F)c1F 35322,C1(NC(C2C(NC(CS(CC)=O)=O)C3CCC2C3)=O)(CO)CC2CCCC12 35323,c1(C(=O)NC(C)C(C)C(=O)N(C)CC2(C)CCCC2)cc2occc2[nH]1 35324,C1(CNC(c2ccc(N)c(O)c2)=O)CCC2(CCC2)C1NC(=O)C=C1CC1 35325,N12CC(CC(=O)N(CCn3ccnc(O)c3=O)C(=O)C1)c1ccccc12.COC 35326,Cc1cn2cccc(C(N3CCCC4(NC(=O)Cn5ccnn5)CC4C3)=O)c2n1 35327,C1(CN(C(=O)C=Cc2ccccc2)C)CCCN(C(c2nc(Cl)sc2Cl)=O)C1 35328,n1(CC#C)cccc1C(=O)NCCCNC(=O)C(C)OCc1ccccc1 35329,C1(C(N(CCCNC(C2CC2CC)=O)CC)=O)CC2CCCC(C1)C2 35330,N1(C(C(CC=C)NC(C)=O)=O)CCC(C)N(C(=O)CSC(C)(C)C)CC1 35331,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C(N)=O)C1 35332,c1(OCC(C)NC(=O)C(O)C2CCC2)ccc([N+](=O)[O-])cc1-n1cc(CO)nn1 35333,c1(CN2CCCC(C)(CCOC)C2)ccccc1P(C)(C)=O 35334,N1(C(c2c(OC)ccnc2)=O)CCCC(NC(=O)CC(C)(C)C#N)C1C 35335,N(C(=NCCCNC1CC2CCC2C1)NCCF)CCOC 35336,CCCCCCCCOCCC(=O)NCC1C2CN(CC3COCCN3C)CC12 35337,c1(OC)ccc(C(c2nnnn2CC2CC2)NCCS(C)=O)cc1C 35338,Cc1ccc(Cl)c(C(=O)NC23CC(C(N4CCC(C)C(C)C4)=O)(C2)C3)c1 35339,CC1CN(C(=O)CC2(NC(C3CCCCC(=O)C3)=O)CCCCC2)CC(C)(C)C1 35340,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35341,C1(CNC(C(c2ccc(C)o2)C)=O)CN(C(=O)C=Cc2cccs2)C(C)(C)C1 35342,C1(NC(C(CC)C)=O)CN(C(C2CC(O)(C(F)(F)F)C2)=O)Cc2ccnn2C1 35343,c1(C(N2CCC(C(N(CCC(=O)OC)C)=O)C2)=O)ncc(F)cc1F 35344,C(N=c1nc(N2CCCC(CCO)C2)cc(C)[nH]1)C1CC(N2CCC(OC)C2)C1 35345,N1(C(c2scc(OC)c2OC)=O)CCN(C(C2(CSC)CC2)=O)CC2(CC2)C1 35346,c1(C(=O)NC(CC(C)NC(Cc2c(C)n[nH]c2C)=O)C)cc2c(cnn2C)nc1C 35347,C1(CC)CN(C(=O)C(=O)NC23CC(C(F)F)(C2)C3)CCN1C(C)=O 35348,N1(C(c2c(OC)cc(C)cc2)=O)CC(NC(C2COC(C)C2)=O)CC(C)(C)C1 35349,C=Cc1cnc(NC(N2CC=CC(O)C2)=O)nc1 35350,N1(C(c2c(C)con2)=O)CC(CNC(c2cccc(C(F)(F)F)n2)=O)CCC1C 35351,c1(C(N(C(CC(=O)OCCOC)c2ccccc2)CCC)=O)ccc(CC)o1 35352,c1(C(=O)N(Cc2c(C(=O)NCC(C(CC)C)C)con2)CC)ccnc(C)c1N 35353,c1(C(=O)NCC2N(C(CCCCCCCC=C)=O)CC=C2)cc(N)c(F)c(F)c1Cl 35354,c1(-c2c(C)cc(OCC)c(C)c2)cnc2ccc(C(N3CCC(F)C3)=O)cn12 35355,C(c1cn(C2c3csc2n3)nn1)=CC.C1(C(=O)OC)CCN(C2CCCCC2)CC1 35356,C1(NC(C2CCC(NC(Cc3cn(CC)nn3)=O)C2)=O)CCC(F)CC1 35357,C12(C(=O)NC(c3c(C)cc(N(C)C)cc3)CNC(N)=O)CCC(C)(CC1)OC2 35358,N1(C(Cn2cccc(N)c2=O)=O)CCC2CCN(C(=O)CNc3nccs3)C2C1 35359,C1(C(=O)NC23CC(C2)C3)CC(F)CN(C(c2cncc(-c3ccncc3)c2)=O)C1 35360,Cc1ccc2sc(C(=O)NCC3(O)CCN(C(=O)CCCCC(N)=O)C3)cc2c1 35361,N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCCC(C1)N2C(=O)C(=Cc1cscn1)F 35362,c1(C(=O)NCC2CC(C)C2)cncc(CNC(C2CC(C)(C)CO2)=O)c1 35363,C(=O)(CCC(=O)NC1(C(=O)Nc2ccsc2C)CCC1)Nc1nnc(CC(C)C)s1 35364,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35365,CC1(C)CC(NC(=O)Nc2ccnc(I)n2)C(=O)O1 35366,C1(NC(=O)CC2=CCCC2)CCCC2CN(C(=O)Cc3ccc(O)c(F)c3)CC12 35367,C1(Nc2ccc(CC)nc2)CC2c3ccccc3C1c1ccccc12 35368,Cn1nnc(CNC(=O)C(C2(C)CC2)NC(c2ccn(CC(F)F)n2)=O)n1 35369,N1(C(Cc2c(C)ocn2)=O)CCC2CC(CNC(C3CCC(C)CC3)=O)CCC2C1 35370,CC(C)CC(C(=O)N(C(C)CC(F)(F)F)C)ONC=Cc1cocn1 35371,C1(C(=O)NC(C(C)NC(CCC=CC(C)C)=O)(C)C)(CC2CC2)CCNC1=O 35372,C1(CC)CN(C(=O)OC(C)(C)C)CCC1CNCc1coc(C)n1 35373,c1(C(CC)C)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35374,N1(C(CCCCOCC)=O)CCN(C(c2ccnc(OCCO)c2)=O)C(C)C1C 35375,C1(F)(C(=O)NC(CCC)C(=O)OC)CCCN(C(C2CCC(C)CC2)=O)C1 35376,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35377,c1(C(=O)NC(CN(C(C(C(C)C)N2CCCC2)=O)C)C)ccc2c(c1)CCCC2 35378,c1(OC)ccc(F)cc1C(=O)C(=O)NC1CCN(C(c2ccc(C)o2)=O)C12CC2 35379,N1(C(C(=O)C(C)=O)=O)CCOCC(CN)C1.c1(NC(=O)N)ccc(C)[nH]1 35380,C1(C(=O)NCC(CC=C)NC(c2cc(CC3CC3)oc2C)=O)CC2C=CC1C2 35381,C(=O)(CC(C)P(C)(C)=O)Nc1c(CC(=O)NCC(CC=C)OC)nccc1 35382,Cc1cc(O)nnc1C(=O)NC(CNC(=O)C(C)(C)c1nccs1)C1CCC1 35383,c1(CC)c(N(C2CCCN(C(=O)CCC3CC3(F)F)CC2)C)nc(C)nc1Cl 35384,N1(C(c2nnn(CC)c2C)=O)CCC(C2(NC(=O)C3=C(C)CC3)CC2)CC1 35385,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35386,c1(C(N(CCOCCN(C(c2cc(C)c(C)[nH]2)=O)C)C)=O)cc2ncccc2o1 35387,C1(SC)CCCN1N(C)CC.C1(C=O)CCCN1C(=O)C(O)CSC 35388,N1(C(CC(C(C)C)OCC)=O)CCC2(CCCN2C(=O)CS(=O)(=O)CC)CC1 35389,c1(N2CC(CNC(C(C(=O)OCC)(C)C)=O)OCC2)ncnc2c1CCCC2 35390,C1(CC)CCN(C(c2ccc(SC)s2)=O)C1C(=O)Nc1cnn(C)c1SC 35391,N1(C(c2ncncc2Cl)=O)CCC(CC(=O)NC2C(C)(C(F)(F)F)C2)C(O)C1 35392,N1(C(c2c(C)nc(C)o2)=O)CC2(COC(CNC(c3csc(S)n3)=O)C2)C1 35393,N1(C(c2cnn(C(C)C)n2)=O)CCC2CN(C(c3cc(CO)on3)=O)CCC2C1 35394,C(=O)(CCS(=O)(=O)C1CCCC1)NC(CN(C)C(C1CC1C(F)(F)F)=O)(C)C 35395,C=CCC(C)C(=O)N1CCC(CNC(=O)CC2(COC)CCCC2)C1 35396,CC(C)(C(=O)NC1(c2ccccc2)CN(C(c2cc(F)cc(F)c2)=O)C1)C(N)=O 35397,Cc1c(F)ccc(C(=O)N(C2CCC(NC(c3cncs3)=O)C2)C)c1C 35398,C1(COC)C=CCCN1C(C1CCC(CNC(=O)CCc2cncnc2)C1)=O 35399,Cc1cc(C)c(C=CC(=O)NC2(CO)CCN(C(=O)C#CC3CC3)CC2)cc1C 35400,C(=O)(CC1=CCCC1)N(CC(=O)NCC(C(=O)NC)C)C 35401,C1(CCNC(Cc2cc(OC)no2)=O)COCCN1C(c1coc(SC)c1)=O 35402,N1(CC(=O)NCCOC2CN(C(c3ncsc3Br)=O)C2)CC2CC2C1 35403,c1(C(=O)OC)ccc(S(=O)(=O)NCc2cc(C(=O)O)no2)cc1.C1CN1 35404,CCC(CC)CCC(=O)N1CC2CCC1CC2NC(C1C=CC=CC=C1)=O 35405,N1(C(c2cc(CC)no2)=O)CCc2nc(CNC(c3cc(CC)[nH]n3)=O)sc2C1 35406,CC(=O)CCN=C(NCCC1COC(C)(C)C1)NCCN1CCCNC1=O 35407,C12(C(=O)NCCCOC3CCN(C(=O)C=Cc4nccs4)CC3)CCC(CC1)O2 35408,C(N=c1nc(C(=O)NC)c(Cl)c[nH]1)C1C(CNC(C(CCC)OC)=O)C1 35409,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35410,C(=O)(C(C)C(O)CC)N(CCCCCCNC(C=CCOC)=O)C 35411,C1(CNC(c2nc(OCC)oc2)=O)CCCCN(C(=O)CN(C)C(C)=O)C1 35412,c1(C(=O)NC2CN(C(c3c(COC)ccs3)=O)C3C2C3)cc2sccc2[nH]1 35413,c1(C(N2CC(NC(CC(COC)C)=O)(COC)C2)=O)c([N+](=O)[O-])cnn1C 35414,C1(CNC(c2cc(CC)[nH]n2)=O)CN(C(c2cocc2C)=O)CCC1C 35415,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCCC3)=O)C2)=O)cc(C)c1F 35416,C1(NC(C2(C)CCN(C)C2)=O)CS(=O)(=O)C2CN(C(=O)CSCCN(C)C)CC12 35417,C1(C(=O)NC2CC(NC(C3CC4(CC4)C3)=O)C2)CCC12CCCO2 35418,c1(C(=O)NC2C(NC(c3nncc(OC)c3)=O)COCC2)cc(C)c(Cl)cn1 35419,S(=O)(=O)(c1ccnc(CC)c1)NC1C(C(=O)OCC)=CC=C(C(F)(F)F)NCC1 35420,C1(N(C)C2CC2)CCC(n2cc(C(C)(C)N(C(=O)NC3(F)CC3)C3CC3)nn2)C1 35421,N1(C(c2c(C)coc2)=O)CCC2(CC1)CN(C(c1csc3nccn13)=O)CCO2 35422,c1(C(N(C2C3CN(C(Cn4nc(C)oc4=O)=O)CC32)C)=O)ccc2c(c1)COC2 35423,C1(c2cn(C(C)CNC(N)=O)nn2)(C(=O)NCc2cn(CC)nc2)CC(C)(C)C1 35424,CC1CC(CNC(=NCCN2CCCCC2)NCc2ccsc2)CC(C)O1 35425,N#Cc1ccncc1NC(C1CCC(NCc2ccc(Br)c(C(=O)O)c2)CC1)=O 35426,C1(CC)(NC(C2CN(C(C)C)CCO2)=O)CCN(C(c2cc(F)n(C)n2)=O)CC1 35427,C(C(C(=O)NCCNC(=O)C(C)(C)n1cccn1)C(C)(C)C)OC(C)(C)C 35428,C1(=O)CCCC(=O)NCCCCN1CC.c1(C(=O)NN(C)C)ccc(CO)cn1 35429,Cc1c(CC(=O)NCC2(O)CC(NC(=O)CCCc3cnn[nH]3)C2)ncn1C 35430,C(=O)(CCCCCC#N)NCC1(C(=O)NCC2(C)CCN(C)C2)CC1 35431,c1(C(=O)NCCCC(C)NC(c2ccncc2Cl)=O)cccn(C)c1=O 35432,c1(C)oc2ccccc2c1C.C12CN(CC1O)C2.CCS(=O)(=O)N(CC(=O)N)C 35433,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35434,c1(C(N2C(CN(C(C3C(C=C)C3)=O)C3CC3)CCC2)=O)nc2cccnc2s1 35435,CCC(CCC(=O)N(CCO)C)NC(=O)CSCC(C)(C)C 35436,C1(C(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35437,c1(C(N2C(CNC(C(N3CCC(O)CC3)C)=O)COCC2)=O)ccc(C#N)n1C 35438,C(=O)(N1CC(C)(O)CO1)C1(CCNC(C2(C3(C)CC3)CC2)=O)CCC1 35439,c1(CCCC)[nH]c(C)c(C(N2CC(C(=O)Nc3cc(C(C)=O)on3)C2)=O)c1C 35440,c1(CC)cc[nH]c1C(=O)NCC(C)NC(=O)C=C(C)C 35441,N1(C(C(CN=[N+]=[N-])NC(=O)CCCn2cncn2)=O)CC2CCC(O)C2C1 35442,c1(CC)ncc(C(=O)NC(c2cccnc2)C2CCCCC2)c(C)n1 35443,c1(OC)nccc(C(=O)NCCc2ocnc2CNC(C2CC2C)=O)n1 35444,C1(F)(CNC(COCCCOC)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 35445,c1(C(N2CCC(N(C(c3cncn3C)=O)CC)C2)=O)cccc2ccnn12 35446,c1(CN2CCN(CC)CC2)ccc(C(F)(F)F)c(F)c1.c12cc(ncn1)S2.C1CC1 35447,C1(COC)(CO)CN(C(C2CC(NC(=O)C(n3ccc(C)n3)C)C2)=O)C1 35448,N1(C(c2cc(CCC)ncc2)C(=O)NCCC2CC2)CCCC(C)(C)CC1 35449,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35450,C(=O)(CCCCCn1cc(CNC=O)nn1)N(c1ccccc1C)C(CC)C 35451,c1(CC(=O)N(CCOC)CCNC(C2CCC2)=O)cccc2cccnc12 35452,NC(=O)C1CN(C(c2ccnc(Br)c2)C(=O)NCC2CCCO2)c2ccccc21 35453,C(C)(CCC(=O)N1CCN(C2CN(C(=O)CN3CCCNC3=O)C2)CC1)OC 35454,c1(C(=O)NC(C)CNC(c2cc(C(N)=O)ccn2)=O)cc(Br)c(Cl)nc1N 35455,C1(C(=O)NC(C)C)CCCCCC1NC(C1CC1(F)F)=O 35456,C(CP(C)(C)=O)(C(=O)OC(C)(C)C)C(=O)NC(C)Cc1cccs1 35457,c1(CNC2C(NC(=O)OC(C)(C)C)CCCC2)cc(N)ccc1Cl 35458,N1(C(CCSc2cn(C)nc2)=O)CCC(C(=O)NCCSCCCO)C(C)(C)C1 35459,C1(CNC2CCC(CC)CC2)CCN(C(C2CC(=C3CC3)C2)=O)CCC1(F)F 35460,N1(C(CC(=O)NC)=O)CC2CCCC(C1)N2C(=O)Cc1ccnnc1O 35461,N1(c2nc(N(C)Cc3cnc(C)o3)cc(C)n2)CCC(=O)N(C)CC1 35462,c1(OC)cc(C(N2CC(C(C)NC(=O)C=Cc3ccccc3)C2)=O)cc(N)c1N 35463,C(=O)(CC(C(C)C)NC(C1CN(CC)CCO1)=O)NC(c1ccccc1)C#C 35464,C1(SCC)CC(=O)N(c2cnn(C)c2)C1.N12CC(C1)N(C)C(=O)C1CC1CC2=O 35465,C1(C)(NC(C2C(NC(C(CO)OC)=O)CCO2)=O)CC2(CCC2)C1 35466,C(=O)(C#CC1CC(F)(F)C1)NCC(C)(C1CCC1)NC(C1C2CCC1CC2)=O 35467,C1(N(C(=O)CN2CCSCC2)C)CCCC(NC(=O)C=CC2CCCC2)C1 35468,N1(C(C2(C3CC3C)CCC2)=O)CCCN(C(C)C)CC1.Cc1ccc(CC(=O)N)o1 35469,C12(C(=O)NCC(C)(C)OCCNC(C3(C=C)CC3)=O)CCC(CO)(CC1)C2 35470,N(C(=NCCCF)NC1CCC2CC12)CC1CCN(CCC)C1 35471,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35472,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35473,Cc1nc(N2CCC(NC(c3ccc(O)nc3)=O)C2)c2c(n1)COC2 35474,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCNC2=O)o1 35475,C1(CC(=O)N(C(C)Cc2cnc[nH]2)NC(=O)CCC2CCCO2)CC2(CC2)CO1 35476,CC1=CC(NC(=O)CCOCCNC(C2CCC=CCC2)=O)CCC1 35477,CC1CC(C(N2CCC(N(C(=O)COCC3CCC3)C)CC2)=O)CC(C)C1 35478,NS(=O)(=O)c1cccc(NC(=O)CN2CC3(CCN3C(=O)CCc3ccc[nH]3)C2)c1 35479,N(C1CN(C(c2cnn(C3CC3)c2)=O)Cc2ccccc21)C(C1CC(=O)NCC1)=O 35480,C(=O)(CCC1CCc2ccccc21)NCc1c(N(C)C)cc(C(=O)O)nn1 35481,C1(NC(=O)C=CC2CCCC2)CCN(C(C2CCCS2)=O)CC1F 35482,c1(N(CCCC(C2CC2)OC)C)[nH]c(=NCCc2nc(=N)[nH][nH]2)nc2scnc12 35483,n1(CNC(CSCCC#N)=O)cnc(C(=O)NCC(=O)OC2CC2)c1 35484,N1(C(c2cc(CC)on2)=O)CCCN(C(=O)CN2CCN(C)CC2)C(C)C1 35485,C(=O)(CC1=CCOCC1)N1CCC(C(C)(C)NC(=O)Cc2cccc(C#N)c2)C1 35486,C(N=c1cc(NCCCc2ncc[nH]2)nc(C(F)(F)F)[nH]1)C1(F)CCOC1 35487,Cc1ccc2cc(C(N3CCC4CCC(C3)N4C(=O)CSC(C)C)=O)ccc2c1 35488,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(OC)c3)=O)COC1C2 35489,C12CCN(CC1)C2=O.Cn1nnc(C(=O)NCC(C)(C)NC(=O)CO)n1 35490,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35491,c1(C(C(N2CC(N(C(C(C)=CC)=O)C)C2)=O)OCC)ccc2ncccc2c1 35492,N1(C(c2cnc(CNC(c3ccc(CO)o3)=O)nc2)=O)CC2C3C=CC(O3)C2C1 35493,c1(C(C(=O)NCCC)N(c2ccccc2)CC2CCOCC2)ccc(CC)cc1 35494,C1(CCC)(C(=O)NC2CCC(NC(=O)C(C)(C)C3CCC3)C2)CCNC1=O 35495,N1(C(CSCC(N)=O)=O)CC2ON=C(CNC(c3cccc4c3OCO4)=O)C2C1 35496,CCCC(C)CC(=O)NCCC(C)NC(=O)CSc1cc(F)ccc1F 35497,c1(C(=O)NCC2N(C(CCCC(=C)C)=O)CCC2)ccc2cc[nH]c2n1 35498,c1(CN2C(COC)CN(C(=O)CC(C)(C)C)CC2)ccc(F)c(C)c1F 35499,n1(CC(=O)N(CC(C)NC(c2ccc(-c3ccccn3)o2)=O)C2CC2)cnc(=N)[nH]1 35500,CN=c1[nH]c(=NCc2cnc(Br)c(C)c2)[nH]c(=NCCc2cc(C3CC3)no2)[nH]1 35501,N1(C(C(C)=C2CC2)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 35502,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)Cc2ccnc(C)c2)C1 35503,C1(CC=C)(NC(=O)Cn2nc(C)nc2C)CCN(C(=O)COCC2CCC2)C1 35504,N#Cc1cncc(NC(C2CN(C(c3cnc(Cl)s3)=O)CC2(F)F)=O)n1 35505,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35506,N1(c2[nH]c(N3CC(CO)C(C=C)C3)nc(=NC)n2)CCCC2CN(C)CCC12 35507,C1(NC(C2C(CC)CCO2)=O)CC12CCC(NC(=O)CC1OCCCO1)CC2 35508,C(C(C(=O)N(C)CC1CCCCN1C(C1CCOC(=O)CC1)=O)C(F)(F)F)OC 35509,Cc1cncc(C(N2CCC(C)C2C(=O)NCCNC(N)=O)=O)n1 35510,c1(OC)ncc(Cl)cc1C(N1CCCC(C(=O)NCc2cc(C#N)ccn2)C1)=O 35511,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35512,N1(c2n(CCC#C)c(-c3nc(C)c[nH]3)nn2)Cc2ccccc2C(C)C1 35513,CC1CC(NC(=O)CC(C)(C)C)CN(C(C2(N(C)C)CC(CF)C2)=O)C1 35514,c1(C(=O)NCC2(CO)CCO2)cccnc1.c12nocc1C(=O)NOC2 35515,c1(C(=O)NC(CCCC)CNc2ncc(C#N)cc2F)cnc2c(c1)ncn2C 35516,c1(N2CCC(C(C)OC)C(C)C2)cccc2nc(-c3cn(CCF)nn3)cn12 35517,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35518,N1(C(=O)CC2CCCCC2F)Cc2[nH]nc(C(N3CCCC3CCCO)=O)c2C1 35519,N1(C(C2(C)CCC2)=O)CC2COCCC2(NC(=O)CC2CCNC2=O)C1 35520,C1(C(N(CCCC)CCO)=O)CCN(C(=O)CC2CCCCN2C)O1 35521,c1(C(N(C2CCN(C(c3cncn3C)=O)CC2)C)=O)ccc(O)nc1 35522,c1(C(=O)NCCN(C(=O)C=CC2CCCN2C)C)cnc2[nH]ncc2c1 35523,Cc1c(CC(=O)NC(C)CN(C(=O)CCC2CC2(C)C)C)ncn1C 35524,CC(C)C(CC(=O)N1CCC1NC(=O)CNC(=O)C1CC1)Nc1ccc(C#N)cn1 35525,N1(C(C(CCC)O)=O)CCC2(CC1)CC2C(=O)NCCSc1ccc(Cl)cc1 35526,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35527,c1(CC(=O)NC(C2CC=CCC2)C(=O)NC2CC(CCOC)C2)c(C)n[nH]c1C 35528,C(C(C(=O)NCCCOC1CCCC1)C(C)(C)C)N(C)C(C1(C2CCC2)CC1)=O 35529,c1(C(=O)NC(CC)C)ccc2c(-c3cscn3)nn(C)c2c1 35530,N1(C(CC2CC(=O)C2)=O)CC=CC(NC(C23CSCC2C3)=O)C1 35531,C1(NC(Cc2cccc(CCS(N)(=O)=O)c2)=O)CC2CC1N(C(C1(F)CC1)=O)C2 35532,Cn1cc(C(=O)NC2CCC(NC(C3(C)COC3)=O)CC2)c(C(F)F)n1 35533,C#CC1CN(C(=O)CCC2CCCCN2C(c2cc(Cl)no2)=O)CCO1 35534,C1(C(=O)NC2CC(C(C(=O)NC(C#C)CC3CCC3)F)C2)Cc2ccccc2C1 35535,C(=O)(C(C)(C)F)N(CCCN(C(CC1CC(OC)C1)=O)C)C 35536,N1(CCC2CC(N(C(CC3(C)CC3)=O)C(=O)Cc3cccs3)C2)CC1CO 35537,c1(CCC=C)ccc(C(=O)NCC2(CO)CN(C(=O)CSC)C2)cc1 35538,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)CC(C)O1)=O)C2 35539,CCC(C)(C)C(=O)N(C)CC1(C(=O)NC2(C3CCCO3)CC2)CC1 35540,c1(C(N2CC(N(C(C3(CC)CC3(F)F)=O)C)C2)=O)ccccc1S(C)(=O)=O 35541,CCCC(C)CC(=O)N(C)CCN(C(=O)CCCc1ccncc1)C(C)C 35542,c1(C(=O)NCCC2CN(C(C3CCC(=O)NC3)=O)C2)[nH]cc2c1CCC2 35543,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35544,C(=O)(CCCCC(F)(F)F)N1C(C2(O)CN(C(CC(C=C)C)=O)C2)CCC1 35545,C(CC(C(C)(C)C)NC(=O)CC1CN(C)C1)N(C(c1c(C)c[nH]c1)=O)C 35546,CCCCCCCNC(c1nnnn1Cc1nnn(C)n1)(C1CCCOC1)C 35547,Cc1cnc(F)c(C(N2CCC(NC(c3cc(C(N)=O)ccn3)=O)C2C)=O)c1 35548,Cc1nnsc1C(=O)NC1CCN(C(=O)C(C)(C)c2ncco2)C1 35549,CN1C(=O)OCC1C(=O)NC(CNC(c1cccc(=O)o1)=O)C1CC1 35550,c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)C2CC2)cc2n(n1)CC(F)C2 35551,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35552,c1(C(=O)NC2(C)CCC(C)C2)coc2c1CN(C(=O)Cc1cscn1)C2 35553,C1(CC(N2CCCC(O)C2)C(=O)NCCCSC)CCC(F)(F)CC1 35554,N1(C(CSCc2ccc(C)cc2)=O)CCC(C2CCCN(C(=O)C(C)O)C2)C1 35555,c1(OC)n[nH]c(C)c1C(N1CCC(CNC(c2cc(CC3CC3)[nH]n2)=O)C1)=O 35556,C(=O)(CCCCCCSC)NC1CN(C(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 35557,n1(CC)nccc1C(=O)NCCc1cc(C(=O)N(C)CC2COC(=O)N2)no1 35558,CC1=C(C(=O)C(=O)CCCCCC#N)COCC1.C1(N)CC2CCC1N(C(=O)N)C2 35559,CCCC(C)CC(=O)NCC(O)CN(C(=O)COc1ccc(CC(N)=O)cc1)C 35560,N1(C(c2[nH]cc(C(=O)OC)c2C)=O)CC2CC(OC)CC2C1.C1(=O)CCCN1C 35561,C1(NC(=O)CC2CC(C3CCC3)C2)CN(C(c2cncs2)=O)CC1C1CC1 35562,N1(C(C(=Cc2ccco2)C)=O)C(C)CN(C(c2cc3ccccc3[nH]2)=O)CC1C 35563,Cc1ccc(S(=O)(=O)N2CC3(CC3)CC2C(=O)NCC2CCCO2)cc1Br 35564,c1(C(=O)NCCC(=O)NCC(C)CNC(C2CC(F)C2)=O)ccccc1 35565,c1(C(=O)NCC2(NC(c3noc(CC)c3C)=O)CCC2)ccc(C(C)=O)cn1 35566,N1(C(CC(CC)SC)=O)CC(NC(=O)Cc2cnn3ccccc23)C2(CCC2)C1 35567,C1(NC(C(=Cc2ccco2)C)=O)CCC(CNC(=O)C(c2cccs2)SC)CC1 35568,C1(C)(OC)CCN(C(=O)C(O)CCCNC(=O)COc2ncccc2F)CC1 35569,C1(C(=O)OC)CC(C2CC2)=NO1.C(C)(COC)(C(=O)N)NC(C1C(OCC)CC1)=O 35570,CC#CCC(C(=O)N(C)CCC)NC(=O)OC(C)(C)C.C12(CCC1)C(=O)NC2 35571,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC1N2C(C1CCC1)=O 35572,c1(NC(C(CCN(C)C)NC(C(CC)C)=O)=O)ccnc2cc[nH]c12 35573,c1(C(N(CCNC(CN2C(C)CCC2C)=O)C)=O)cccc([N+](=O)[O-])c1Cl 35574,c1(C(=O)NCC2CCN(C(c3ccc(C)c(C)c3)=O)CC2)c(C)c(C)n(C)c1C 35575,C#CC1(C(=O)NC2CN3CCCC2C3)CCN(C(c2cn(C)nn2)=O)CC1 35576,c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NCCCN(C(=O)C(CC)C(C)O)CCO 35577,C1(C(=O)NC(CC)CN(C)C(c2cnnc(C)c2)=O)CCCCN1N=O 35578,c1(COC)nnc(N(CCC(C)NC(=O)CC2(C(F)(F)F)CC2)C)o1 35579,c1(C(=O)NC2CC(NC(C3CCCO3)=O)C2)c[nH]cc(F)c1=O 35580,N1(C(C(CC#C)C2CC2)=O)CCC2CCC(NC(c3conc3C3CC3)=O)C12 35581,CC1(C)CCC(C(N2CC3CC2C3C(=O)NC2C3COCC23)=O)O1 35582,N1(C(C)=O)CC(O)CC1C(=O)NCc1csc(NC(N2CCCC2)=O)n1 35583,c1(NCCc2cncc(F)c2)cc(S(=O)(=O)NC(C(C(C)C)O)C)ccc1C#N 35584,CCC1=NOC(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)C1 35585,CC1CCN(C(=O)Cc2cnns2)C(C)C1NC(=O)CC1C=CS(=O)(=O)C1 35586,c1(CC)ccc(C(N2CC(CF)(NC(=O)C=Cc3cncn3C)C2)=O)cc1CC 35587,N1(C(C(CC#C)C)=O)CCN(C(c2cc(Cl)c(O)c(Cl)c2)=O)C2CCC12 35588,C1(NS(CC)(=O)=O)CCCCN(C(C23CCC(OC)C2C3)C(=O)NC)C1 35589,CCCCCCCCCC(=O)NC1COCCN(C(=O)CC2CCCCCO2)C1 35590,C(=O)(CCCCCNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35591,C12(C(=O)NC(C3(O)CN(C(C4CC5CC5C4)=O)C3)C)CC(C)(C1)OC21CCC1 35592,C(=O)(C(CO)C(F)(F)F)N(CC(C)C)C(C1CC(C)CCC1O)=O 35593,C(=O)(C(F)C(F)(F)F)Nc1c(C(=O)NCC2CCCN(c3nccs3)C2)cccc1 35594,C1(NC(CCC(C)SC)=O)CCCCN(C(=O)CSc2n[nH]c(=N)s2)C1 35595,CC1CC(=O)NC(C(=O)N(C)CCN(C)C(c2cn(CCC(C)(C)C)nn2)=O)C1 35596,c1(C(N2CCOCC(CO)C2)C(=O)NCC(C)C)ccn(CC(F)F)c(=O)c1 35597,c1(CC)ccc(S(=O)(=O)NC(C2CN(C)CCN2C)C)cc1 35598,c1(CN(C(C#C)COC)C=O)ccc(C#N)cc1Cl 35599,CCC(C)C(C(=O)NCC#CCCO)N(C(C1(F)CC1)=O)C 35600,Cc1cc(C)c(C(=O)N(C)CC2CCN(C(=O)C=Cc3cncn3C)C2)[nH]1 35601,C(C(=O)NC(c1cc(C)on1)C)(C(C1CCOC1)O)N(C(C)(C)C)C.C1CC1 35602,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35603,c1(C(=O)NC(CNC(C(CC)n2nccc2C)=O)C2CC2)cc2cccnn2n1 35604,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C2CCC2)nc1O 35605,CCCC(C(=O)NC)NC(=O)CC1(NC(=O)C(C)(C)n2cnnn2)CC1 35606,N1(C(CCNC(=O)C=CCl)=O)C(CNC(=O)C(O)c2cnc[nH]2)CC2CCCC12 35607,c1(C(CN(c2ccccc2)C)NCC2CCN(CC)C2)nccc(C)n1 35608,C1(CCN(C(=O)CCC2CC2(C)C)C)CCCCN1C(=O)COC1CCC1 35609,N1(C(c2cc(CC)no2)=O)CC(NC(C2CC(O)C2)=O)C(C2CC2)C1 35610,C(C(C)C(F)C(=O)N1CC2CSCC2C1)NC(C(C(C)C)F)=O 35611,C1(N)C(F)(F)C12CC2.CC(C)(COC)CNC(=O)COCc1ccccc1 35612,CCC(Cc1cccc(C)c1)C(=O)N(CCCCNC(C1C(Cl)(Cl)C12CC2)=O)C 35613,C1(C(N2CC(C#N)(CCOC)C2)=O)CCN(C(=O)C(C)SC)O1 35614,c1(C(=O)NC2CCC2NC(C2CCCOC2)=O)cc(F)c(O)c(Cl)c1 35615,C1(CC=C)(NC(c2ocnc2C)=O)CCN(C(C2CCC(=O)N2C)=O)C1 35616,C1(C(=O)Nc2nccc(N(c3ccccc3)C3CC3)n2)CN2CCN1CC2 35617,N1(C(C2N(C(Cc3c(C)ocn3)=O)CC(O)C2)=O)CCC(N=[N+]=[N-])C1 35618,N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(CNC(c2cncs2)=O)C1 35619,C(=O)(C(C)(C)CCCO)N1C(OCC2CCN(C(C(C(C)(C)C)O)=O)CC2)CCC1 35620,Cc1nocc1NC(=O)CNC(=O)CNC(c1ccc(F)s1)=O 35621,N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(=O)CCCn2cncn2)C)C1 35622,C1(C(=O)NC(C)CNC(C2CC(=O)N(c3nccs3)C2)=O)C2C3CCC(C3)C12 35623,N1(C(c2c(C#C)cn(C)n2)=O)CC2(COCC(=O)N2)C1.C12(OC)CCN(C1)C2=O 35624,N1(N2CCCC(NC)C2)CC2CCCC(N)C2C1.C(=O)CSC(=N)N 35625,c1(C(=O)NCC(C)N(c2nc(COC)nc(Cl)c2)C)ccc2c(c1)nc(O)n2C 35626,c1(OC)cc(NC(C2CC(NC(c3ccc(C)c(F)c3)=O)C2)=O)nc(OC)n1 35627,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35628,C1(CNC(CCC(C)OC)=O)CN(C(C2CCC(N(C)C)CC2)=O)CC(C)(C)C1 35629,N1(C(CC(C)OC)=O)CC2CCN(C(c3nccc4[nH]ccc34)=O)C(C2)C1 35630,c1(CNC(C(C)OCCOCC)=O)cccc(F)c1CC(C(=O)NC(C)=O)C 35631,c1(C(N2CCC(N(CCC)C(C3C=CCC3)=O)C2)=O)c(CC)nn2ccccc12 35632,c1(OC)cccc(CC(=O)NC2CCC(NC(c3cocn3)=O)C2)c1F 35633,N1(C(CCc2cc(C)nn2C)=O)CC(NC(=O)C=Cc2ccn(C)c2)CC(C)C1 35634,C1(C(=O)NCC2(F)CCN(C(=O)C(O)C3CC3)C2)C2CCC1(c1ccccn1)C2 35635,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35636,n1(CCOC)cncc1C(c1cc(C)on1)OC 35637,c1(COC)c(C(=O)NC2CCNC(C(=O)O)C2)oc2ccccc12 35638,c1(CC(N2CCCC(N3CCN(C(CC)=O)CC3)C2)=O)c(F)cc(F)cc1Br 35639,CC1CCCCC1C(=O)NCC(C)(C1CC1)NC(c1cnn(C2CC2)c1)=O 35640,CC(C)(CC1CCOC1)C(=O)NCC(=O)NCC1CCN1CC1CCOCC1 35641,N1(C(CCC(C)SC)=O)CCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CC1C 35642,C1(C(=O)NC(c2onc(C)n2)C)COCCN(C(C2(N(C)C)CCCCC2)=O)C1 35643,N1(C(=O)CCc2cc[nH]c2)CCC2(CCCN2C(=O)C(c2ccccc2Cl)=O)C1 35644,O=C(CC1=CCCC1)NC1COCCN(C(c2cc3n(c2)CCC3)=O)C1 35645,N(C1=NC2=NC(=O)CCN2N1)CC(=O)NC(=O)CCOc1cc(Cl)cc(Cl)c1.CN 35646,C(C(C)(C)CNC(=O)C(COC(C)C)NC(=O)CC(C)c1ccco1)OC(C)=O 35647,c1(C(=O)NC2CC(NC(C3(O)CCCC3)=O)C23CCC3)nnn2c1CSCC2 35648,C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(n2cc(-c3ccc(C#N)nc3)nn2)C1 35649,C#CCC(CC(=O)N(C)Cc1cccc(C)c1)NC(c1ccc(O)nc1)=O 35650,c1(OCC2(c3cn(Cc4cnc(C)s4)nn3)CCCOC2)ccc(F)cc1Cl 35651,Cc1nn(CC(N2CCCCC2C(C)NC(c2oncc2C)=O)=O)c(=O)o1 35652,C1(NC(CNC(CC)=O)=O)CC2C=CC1N(C(=O)CCNC(N)=O)C2 35653,N1(C(c2cc(CC)no2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35654,C12C3CN(CC13)C(=O)OC2.c1(OC(C(C)=C(F)Cl)=O)ccccc1 35655,N1(C(CC=C=C)=O)CCC2(NC(=O)Cc3cccc(C)c3C)CCCCC12 35656,c1(C(N2CCCC(C(C)(C)C(=O)Nc3cnc(Cl)nc3)C2)=O)cnc2ccccn12 35657,N(C1CCc2ccc(F)c(C)c21)C(=O)NCCc1c(OC)ccc(C)c1 35658,c1(C(N2CCCC(OC)C2)=O)cc2ccc(-c3ccc(C#N)c(F)c3)cc2[nH]1 35659,c1(C(=O)NC2CCN(c3nc(COC)nc(C)c3)C(C)C2)ccc2ncsc2c1 35660,C1(F)(NC(C2CC(=C3CC3)C2)=O)CCC(NC(C2CN(C(C)=O)C2)=O)C1 35661,C1(CC(=O)NCCC2COCCN2C(=O)Cn2ccc(N)n2)(OC)CCOCC1 35662,C=CCCCC(C(=O)NC(C)Cc1cnn(C)c1)NC(=O)CCCCC(C)C 35663,C(CC)(CC(=O)N(C)CC1CCOC1=O)NC(CC=C)=O 35664,S(=O)(=O)(c1ccc(CNC(C)=O)cc1)N(CCCC[Si](C)(C)C)CC 35665,Cc1cc(F)ccc1C(=O)NC1CCCN(Cc2scnc2C)C1 35666,Cc1cc(C(N2C3CCC2C(CNC(=O)C(C)CF)C3)=O)c(Cl)cc1N 35667,N1(C(=O)CC2CC(O)CN2Cc2cccnc2)CC2(CO)CC2(CO)C1 35668,C(CC(=O)N(CCNC(=O)CC1CCCC1O)C1CC1)(C(C)C)OCC 35669,CC(=O)n1cnc(-c2nnc(N3CC4C(CF)C4C3)n2CCCC#N)c1 35670,c1(NC)nccc(C(=O)NC2CCN(CCNC(C3CCCCO3)=O)C2)n1 35671,c1(NC(C2C(NC(c3c(CC)cccc3)=O)CC=CC2)=O)cccc2c1OCO2 35672,C(c1cnn(C)c1)=CC(=O)NCC(COC)NC(c1csnn1)=O 35673,c1(C(=O)NC(C)C(CO)NC(c2cnc3ccccn23)=O)cccc2nn[nH]c12 35674,c1(N(C)C)ncccc1C(=O)NCC=CCNCCC(=O)NC1(c2cccs2)CC1 35675,N1(C(C(CC)(F)F)=O)CCN2C(=O)C(NC(=O)Cn3ccnc3C(C)C)CC2C1 35676,CC1CN(C(=O)Cc2cn(C)cn2)CCC1NC(C1(c2ccncc2)CCC1)=O 35677,C(=O)(CC(C)COC)N(C(C1(CN(C)C2CC2)CN(C(=O)COC(F)F)C1)C)C 35678,c1(N2CCC(NC(CC3CCCC(CC)C3)=O)CC2C)nc2nc(C)ccc2s1 35679,c1(C(=O)NC2CCC(N(C(CCC=C=C)=O)C)C2)cc(C2CC2)cc(SC)c1 35680,c1(OC)ccc(F)c(NC(C2CCC(NS(=O)(=O)CC#N)CC2)=O)c1 35681,CCC(CC(=O)NCc1ncc(C(=O)NC23CCCC2C3)cn1)C(C)(C)C 35682,CCC(C)(C)OCC(=O)N(CC(CC)NC(=O)Cc1ccsn1)C 35683,N1(C(CCCC(C)=O)=O)CCN(C(=O)CCN(C2CCOCC2)C)C(C)C1C 35684,C1(NC(CCC(N)=O)=O)CC2CC1CN(C(c1cccc(-n3cccc3)c1)=O)C2 35685,N1(C(c2cc(C)sc2)=O)CC2CCC1CN2C(=O)C(C)SCc1c(C)noc1C 35686,C1(N(C(c2cscc2Br)=O)CCF)CCCN(C(C2CCCC(O)C2)=O)C1 35687,C1(C2CN(C(=O)CSc3nncs3)C2)(NC(C2CC(C)OC2=O)=O)CC1 35688,CC1(CCNC(C2CC(CCO)C2)=O)CCN(C(C2(O)CC(F)(F)C2)=O)C1 35689,Cc1ncc2n1CCC(C(=O)NC1CC3CCC1N3C(=O)CCC1CC1)C2 35690,C#CCCCCCC(=O)N1CCC2CN(C(=O)COCC)CC12 35691,CCCCC(C)CCC(=O)N(CC(=O)NC1CCOCC1)CCCOCCF 35692,c1(C(N2C3C(NC(C4CC(OCC)C4)=O)CC(C3)C2)=O)sc2ccccc2c1Cl 35693,c1(OC)cccc(C(O)C(=O)NC2(C)CCOC2)c1OC 35694,c1(NC(C2(CC)CCOC2)=O)ccc(C(N2CCC2CC(C)(C)C)=O)cc1C 35695,C12(CNC(C3CCOC3)=O)COCCN1CCN(C(C13CCCN1CCC3)=O)C2 35696,CS(=O)CCCNC(=O)C(CC1CCC1)NC(C1CN(C(=O)N(C)C)C1)=O 35697,c1(CC)noc(C)c1C(=O)NC1(CC(N2CC(N3CC(F)C3)C2)=O)CC1 35698,N1(C(Cc2cn(C)nc2)=O)CC(NC(C2CC3CCC3C2)=O)C2(CC2)C1 35699,C1(C(=O)NC23C(CN(C(COC4(C)CCCC4)=O)C2)C3)CNc2ccnn2C1 35700,C1(CC)CCN2C1C(=O)NCCCCOC1(C)CN(C1)CC2=O.C(C)(=O)OC 35701,C1(NC(C=CC(CC)C)=O)C2CCC1CN(C(=O)C#CC1CCCC1)C2 35702,c1(C(C(=O)O)NC2CN(C(=O)OCC(F)(F)F)C2)ncccn1 35703,C1(CNC(C2(CC(=O)OC)CC2)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35704,c1(OC)ncnc(OC)c1N1CC2C(NC3CCC(F)(F)CC3)C2C1 35705,CCCCCCCCC(CO)NC(c1cc2nc(Br)sc2[nH]1)=O 35706,N1(C(CC2(COC)CC2)=O)CCC2(CC1)CC2CNC(=O)C(C)C(O)C(C)C 35707,Cc1nc(N2CC3(CNC(c4cc5c(s4)CCC5)=O)CC2CO3)c2cc[nH]c2n1 35708,Cc1c(C(=O)NC2CC23CC(NC(C2CCC4CC24)=O)C3)oc2ccc(F)cc12 35709,c1(-c2ccc(NC(C(C)NC=O)=O)cn2)ccc2c(c1)OCCN2C 35710,C1(NC(c2c(CC)con2)=O)CC(CNC(c2cc(C(C)C)nn2C)=O)C1(C)C 35711,c1(CC)cc(C(=O)N(CC(=O)NCCCC(C)(F)F)C(C)C)ncn1 35712,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35713,C1(CNC(CC(C)OC)=O)Cc2ccccc2CN1C(C1(C2CC2)CCCO1)=O 35714,N1(C(C2C(C)CCO2)=O)CCCCC2(C1)CN(C(c1coc(C3CC3)n1)=O)C2 35715,C1(NC(=O)CC2CC2C(F)(F)F)CCCCN(C(=O)C=Cc2ccccc2)C1 35716,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(O)CN(C)C)N(C)C 35717,C(CC)(CCC(C)C)(c1cccc(C(N(C)Cc2cn(CC(=O)O)nn2)=O)c1)OC 35718,S(=O)(=O)(c1c[nH]ccc1=NCC(C)(C)C(O)C(C)C)N(CCC(=C)C)C 35719,CCCC(C)(O)CC(=O)N1CC(CNC(c2cc(CC3CC3)on2)=O)C(C)(C)C1 35720,N1(C(C(C)=CC2CC2)=O)C2CCC1C(C(=O)N(C1CC(CO)C1)C)C2 35721,c1(OC)cnccc1C(=O)NCCC1(NC(=O)CC2CC3(CC3)CO2)CC1 35722,N1(C(C2CC(=C)C2)=O)CCN(C(=O)CC2CCS(=O)(=O)CC2)C2CC12 35723,N1(C(c2c(C)n3c(n2)scc3)=O)CCC(C2CC(NC(C3SCCCS3)=O)C2)C1 35724,c1(C(=O)NCCC(C)NC(C2C=CCC2)=O)coc2c(Cl)cccc12 35725,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35726,c1(CC)cc(C(N2CCC(CC(=O)N(CC(C)C#N)C)C2)=O)on1 35727,N1(C(c2c(Br)cn(C)n2)=O)CC2CC(NC(c3ccc(CO)cn3)=O)C2C1 35728,C1(COC)CN(C(c2cc(Br)c(C)cn2)=O)CCN1C(c1cnc(O)o1)=O 35729,c1(CCN(C(c2onc(C)n2)C)CC(=CCCC(C)N)C)c(C)cccc1C 35730,Cc1c(C(=O)N(C)CCOCCNC(=O)C(C)CC2CCCO2)cccc1Cl 35731,Cc1ccc(C(N2CCCC(C)(NC(c3cscc3F)=O)C2)=O)c(Cl)c1 35732,C1(NC(CSCC(=O)NCCCC)=O)(CC2CC2)CCCCC1C.c1(C=O)cc[nH]n1 35733,N1(CC)CCOC(C(N2CCCC(C(=O)Nc3c[nH]ccc3=O)C2)=O)C1 35734,C(=O)(C1CCc2nccn21)NCC1CCN(C(c2cccc(C(N)=O)c2)=O)C1 35735,n1(CC(CC)NCC(C)(C)C)cc(Br)cn1 35736,N1(C(c2c(CC)c3c(o2)cccc3)=O)CCOC2(CCC(C)CC2)C1 35737,N1(CC(C)C)CCCC1C(=O)NC1CC(CNC(C2CC3CC3C2)=O)C1 35738,C1(CNC(=O)CC2OCCO2)COCCN1C(c1cncn1-c1ccncc1)=O 35739,c1(C(C(=O)NC(CC(C)NC(c2c(C)cn(C)c2)=O)C)(C)C)ccc(Cl)cc1F 35740,[N-]=[N+]=NC1CN(C(=O)COC2CCCCC2)CC1NC(c1ccc(OC)cc1)=O 35741,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2C)c1C 35742,c1(CC)onc(C)c1NC1CCCN(C(=O)CN(CCCCC)C(C)=O)C1 35743,Cc1ncc(Cl)cc1C(N1CC(CCNC(c2cncc(F)c2Cl)=O)C1)=O 35744,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35745,c1(NC(C(=O)NC2(CCNC(C(C=C=C)C)=O)CC2)CC)ccc2sccc2c1 35746,c1(C(=O)NCCC2CCN(C(C3(C)CC=CC3)=O)C2)ncnc2sccc12 35747,C1(CC)(CO)CCN(C(=O)C(CNC(=O)CC2(OC)CC2)CC2CC2)C1 35748,c1(C(=O)OC)cc2c(N3C4CN(C(=O)C(COC)OC)CC34)[nH]cnc-2n1 35749,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 35750,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(=O)CC2CCC(=O)NC2)C1 35751,C1(C(N)=O)CCCC(C(=O)N(CCNC(=O)C=C(Cl)Cl)C2CC2)C1 35752,O=C1NC(=O)C2C3CCC(CC3)C12C(N1CCC(O)(Cc2ccccc2)C1)=O 35753,CC(C)=C=CC(=O)N1CC(CNC(=O)Cc2ccc(SC(C)C)cc2)C1 35754,C(C(C(=O)N1CC(N(C)C)C2(CC2)C1)C(C)C)NC(c1c(CCC)nco1)=O 35755,C1(CNC(=O)Cn2cnnc2)(NC(c2cc(Br)no2)=O)CCCC1 35756,C1(SC)CN(C(=O)C#CC2CC2)CC1NC(=O)CN1CCCS1(=O)=O 35757,C1(NC(c2[nH]cc(C(=O)OC)c2)=O)CN(C(=O)CCC(C)N(C)C(C)=O)CC1F 35758,C1(NC(CN(CC(=O)NCCC)C)=O)CCCCN(C(=O)CC2CCOCC2)C1 35759,CC(CC(=O)NCCOC1CN(C(=O)CC2CC2)C1)C1CCCO1 35760,c1(OC)cc(C#N)ccc1C(=O)NC1CS(=O)(=O)CC1NC(=O)CCP(C)(C)=O 35761,C#CCCCCCC(=O)NC(C)(C)CN1CCN(C(=O)CC2CSCCS2)CC1 35762,c1(C(=O)NCCCCNC(C2CCCN(C(C)=O)C2)=O)cc(F)c(F)c(F)c1 35763,C1(C(=O)NCC(CCC)C)CC2CC(=O)C1O2 35764,C1(COCC)CCCN(C(=O)C(C2CCC2)NC(=O)CC2(C)CCC2)C1 35765,C(=O)(CCCCC(C)(C)C)C1CC2C3C(NC)C1C3C2C(N1CCCC1CO)=O 35766,Cc1nc(C2CCCCC2)nc(O)c1CC(=O)NCC(C)(C)CN1CCOCC1 35767,c1(C(=O)NCC(CO)NC(CSc2n(C)ccn2)=O)c(Cl)ccc(F)c1F 35768,N1(C(CCOC)=O)CCC(C)C1C(=O)NCCn1cnnc1C 35769,C1(C(=O)NC2(COC)CN(C(=O)CSCCC(F)(F)F)C2)COCCC1C 35770,N1(C(C(CN(CC)CC)F)=O)CCC(F)(NC(=O)CC2CCOC2C)CC1 35771,C12CCCN(CC1)N2C.c1(NC(C(=O)N(C)C)=O)coc2c1COC2 35772,n1(CC(=O)NCCC(=O)NC(C)CCc2cn[nH]c2)ccccc1=O 35773,N1(C(CC(CC)SC)=O)C2CCC(C(=O)NC34CC(C)(CCO3)C4)C1CC2 35774,N1(C(CCCN(C)C)=O)CC(F)(F)CC1CNC(=O)C1CC1.C1(C=O)CC1 35775,Cn1nc(C(=O)NCCC2CCC(NC(C3(CF)COC3)=O)C2)cc1Cl 35776,C1(NC(C(C2CN(C(c3c(OC)cccn3)=O)C2)OC)=O)CC2(CCC2)C1O 35777,c1(OC)cc(C(=O)NC(C)(C)CNC(c2cccc(OC(F)F)c2)=O)cc(Cl)n1 35778,C1(CC)CCCCC1C(=O)NC1(CN(C(=O)C(C)(C)C2CC2)C)CC1 35779,C1(C(=O)NC(C)CN(C(=O)C(C)OC2CCCCC2)C)CC2(CCO2)C1 35780,Cc1cccc2c1CC(C(N1CCC(NC(c3occc3Cl)=O)C1)=O)O2 35781,Cc1c(C(N)C(=O)Nc2ccc(CCNC(N)=O)cc2)cccc1F 35782,c1(C(N(C2CN(C(C=CC)=O)CC23CC3)C)=O)cnc2c(C)cccn12 35783,N1(C(C(=O)N)=O)CCCC(N(CC2=CCCCC2)C)C1.Cc1nccn1CC 35784,c1(C(CO)NC(C23C(CN(c4ncc(C(=O)OCC)cn4)C2)C3)=O)ccc(Cl)cc1 35785,N1(C(=O)NC(c2cccnc2)CO)CCCC1CCn1ccnn1 35786,CN1CCC(C)(C(N2CCC2CNC(=O)C=Cc2ccccc2)=O)C1=O 35787,C1(NC(c2cc(OC)ncc2)=O)CN(C(c2nc(C)ncc2Cl)=O)CC2(CC2)C1 35788,C(=O)(CCCC(F)(F)F)NCC1(OC)CCCCC1C.c1(C2C(=O)N2)cnn(C)c1 35789,c1(CCC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 35790,N1(C(C2(SC)CC2)=O)CCCN(C(c2cnn(C3CC3)c2C)=O)CCC1 35791,C1(CNC(=O)Cc2ccc(Cl)s2)CN(C(C2CC3(CCCO3)C2)=O)CC12CCC2 35792,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 35793,[N-]=[N+]=NC1COCC1NC(=O)Cn1cc(CON2CC3CC3C2)nn1 35794,C1(C(=O)NC(CC=C)CNC(=O)COC2CCCC2)CC2(COC(=O)N2)C1 35795,n1(CC)cc([N+](=O)[O-])c(C(=O)NCC(C)(C)OCCNC(=O)CN(C)C)n1 35796,N1(C(c2cc(OC)c(C#N)cc2)=O)CCC2CCC(C1)N2C(C1(C#N)CCC1)=O 35797,C1(C(=O)NC(CCC)C(=O)N2CCOC3CC23)CCCCC1(C)C 35798,CC(CC(C)NC(c1cc(C(F)F)no1)=O)NC(=O)C=CCn1cc(Cl)cn1 35799,N1(CCC(=O)NC(CNC(CC2CN(C(=O)NC)C2)=O)(C)C2CC2)CCCCC1 35800,C1(CCC)(NC(c2ccc(F)c(Cl)c2)=O)CCCN(C(=O)C(=O)NCC2CC2)C1 35801,c1(CC)cc(C(N2CCC(C(=O)NCC=Cc3ccncc3)C2)=O)nn1C 35802,C(=O)(C(C)C(F)F)NCCC1CC(NC(C(C2CCCC2)OCC)=O)C1 35803,CC(O)C(C(=O)N1CC(Cc2n(CCOc3cccnc3)ccn2)C1)NC(N)=O 35804,c1(NC(=O)C(c2ccccc2)O)nccc(N2CCOCC2)n1.C12CNCC1C2 35805,N1(C(c2c(CCC)n[nH]c2)=O)CC(NC(c2cc[nH]c2)=O)C2CC2C1 35806,c1(C(=O)NCC2(CN(C(=O)CC)C)CC2)ccc(Cn2cnnc2)o1 35807,N1(C(Cc2ccc(C(C)=O)cc2)=O)CCC(CO)C(NC(c2cc(C)[nH]n2)=O)C1 35808,S(=O)(=O)(c1cccc(Cl)c1)N1CCC(NC(=O)NC(CC)CN2CCCC2)C1 35809,Cc1ccc(C)c(OC(c2ccc(N3CCC(CN4CCCS4(=O)=O)C3)cc2)=O)c1 35810,N1(C(CSC)=O)CC(C)(C)OCC1CNC(=O)CP(C)(C)=O 35811,C(=O)(C(F)C1=CCCCC1)NC(C)CCNC(=O)CCc1cnn[nH]1 35812,N1(C(c2nc(C)sc2)=O)CC2CC1CN2c1cc(-c2ccc(F)cc2)nc(Cl)n1 35813,c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC1CCN1C(C1CC12CC2)=O 35814,c1(C(=O)NCCC2C(C)CN(C(=O)CN(C)C)C2)nn(C)c(=O)c2ccccc12 35815,Cc1nn(C)c(NC(=O)OC(C)(C)C)c1C(=O)NCCC12CCC(CC1)O2 35816,C(=O)(C(CCCC(=O)OC(C)(C)C)OC(C)=O)N(CC=C)CCC1CC1 35817,C(=O)(CC(C(F)F)NC(=O)Cc1ncn(C)c1C)N(C1CCCC1)CCOC 35818,c1(CNC(C2CN(C(c3cnc(N(C)C)o3)=O)C2)=O)ccc(F)c2ccccc12 35819,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 35820,Cc1c(C(=O)NCC(CC2CCCC2)C(=O)N(CCCCCO)C)ncn1C 35821,C=CCC(C)(C)CC(=O)N(CCCOCCN(C)C(c1c(C)coc1C)=O)C 35822,N1(C(C2C(CCOC)C2)=O)CC2(CC(NC(=O)C=CCOC)CO2)C1 35823,n1(C(c2ccccc2)(C2CC2)NCC(CC)(C)OC)c(-c2ccccn2)nnc1S 35824,C(c1ccc(C)cc1)=C(C(=O)N(CCCNC(C(C(C)SC)O)=O)CCO)C 35825,c1(C(=O)OCC)cccnc1N1CCC(NC(c2conc2CC)=O)CC1 35826,Cc1nc(O)nc(C)c1C(N1CC2(CCN(C(=O)CC3CCSCC3)C2)C1)=O 35827,Cc1ccc(F)cc1C(N1CCC(C(F)F)(CNC(=O)Cn2cncn2)C1)=O 35828,CCCN=C(NCC1CCOC1)NC1CCN(C2CC2)C(C)C1 35829,CC1CCN(C(=O)CCn2cccc2)CC1NC(c1ccnc(OC(F)F)c1)=O 35830,Cc1cc(C(=O)NCC2(O)CCCN(C(=O)C=C(Cl)Cl)C2)c(C)n1C1CCOC1 35831,C12(NC(c3n(C=C)nnc3)=O)CCN(C(c3c(Cl)cnn3C3CCCC3)=O)CC1C2 35832,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 35833,c1(C(=O)NCCN(C(=O)C(O)CC(C)C)CC)cnn2cc(C(F)(F)F)nc2n1 35834,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 35835,C1(NC(C2ON=C(CC)C2)=O)CCCC(F)(F)CC1 35836,C1(C(=O)NCCC(C)NC(c2sc(F)cc2Cl)=O)CC2(CCOCC2)C1 35837,C1(N(C(=O)C(F)Cc2ccccc2)C)CCCN(C(=O)OC(C)(C)C)CC1 35838,C1(CNC(C2C(C(C)O)C2)=O)CCCCC12OCCO2 35839,c1(C(=O)NCC(CNC(C2(C)CCC2)=O)O)ccc(-c2cnc[nH]2)cc1 35840,C12(CNC(=O)COC3CCC3)CCC(C1)N(C(C1CC(=C3CCC3)C1)=O)C2 35841,N1(C(C(CCC)C)=O)CCC2(CC(C(=O)Nc3cc(SC)cc(Cl)c3)=NO2)C1 35842,c1(SCCC)cccc(C(=O)NCC(O)CN(C(=O)CCN2CC(C)C2)C)c1 35843,CCCCC(F)C(=O)NC1(CC)C2CCCN(C2)C(=O)C2C1C2(C)C.C(C)(=O)O 35844,c1(C(=O)NC2CCCN(C(c3ccc(CO)o3)=O)CC2)cn2c(Cl)cccc2n1 35845,c1(N(C)C)cnc(C(N2CCC(NC(c3ccncc3C(F)(F)F)=O)C2)=O)nc1 35846,C1(NC(CCOC)=O)CC2CCC(C1)N2C(c1cnc(O)c2ccsc12)=O 35847,N1(C(c2c(C)nc(=N)[nH]c2C)=O)CCC2CCN(C(=O)Cc3ccno3)CC2C1 35848,CC1C(NC(C2C=CCC2)=O)CCN1C(=O)Cc1cn(C)nc1Cl 35849,C=CC(C)(CC)C(=O)NCC(C)(C1CC1)NC(=O)CCc1nc(N(C)C)no1 35850,C(=O)(CCCc1cccnc1)NCCN(CCC)C(c1cnnn1C1CC1)=O 35851,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 35852,c1(C(=O)NCC2CCCN2C(C2CC2C2CCCCC2)=O)nc2cnccc2s1 35853,c1(CN(C)C(C2CCCC2CNC(=O)CCc2cnco2)=O)nncn1C 35854,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 35855,C1(C(=O)NCC(=O)NCCC(CN(C)C)O)OCCCC1(C)C.c1(C)nc[nH]n1 35856,CCCCC(O)C(=O)NCC1CN(C(=O)CC2=CCCC2)CCO1 35857,N1(C(C(Cc2cc[nH]n2)NC(c2c(C)snc2)=O)=O)CCOC2CCCC12 35858,C(=O)(CN=c1[nH]c(C)cs1)N1CCC(CNC(c2c(OC)nccc2)=O)C1(C)C 35859,C1(COC)CC(C)(C)CN1C(CC)C(=O)NC1CCOC1 35860,N1(C(C(C(C)C)n2cccc2)=O)C2CCC1C(C(=O)NC1CCC(N(C)C)C1)C2 35861,C(CCCCOCc1cc(C(=O)OC)no1)OC 35862,c1(C(C(=O)NCCC(C)NC(c2c(C)nn(CCO)c2)=O)O)cc(Cl)ccc1F 35863,c1(C(=O)NC(C2CCCCCC2)CNC(CCOCC#C)=O)nnc(O)cc1O 35864,N1(C(CNC2CCCCC2)=O)CC2CC3CC2C1C3.c1(C=O)n[nH]c2c1CCC2 35865,C1(NC(CN(C)CC)=O)(CC)CN(C(=O)CC(C)c2ccccc2)C1 35866,CCC(C)(CNC(c1cccc(F)c1C)=O)C(=O)N(C)CC1(OC)CCC1 35867,CC1Oc2ccc(C(N3CCC3CNC(C3(C)CCCS3)=O)=O)cc2NC1=O 35868,N1(C(C2C(C)(C)OCC2)=O)CCC2CN(C(c3ccnc4ccnn34)=O)CC12 35869,c1(C(N(CC(C)NC(c2c(C(C)C)nco2)=O)C)=O)ccnc(S)c1 35870,c1(OC)ccc(Cl)c(C(=O)NC(C)CCNC(C2CC(C3CCC3)C2)=O)c1 35871,c1(C(N2CC3CN(C(c4n[nH]c(CC)c4F)=O)CC32)=O)cc2ccc(Cl)cc2[nH]1 35872,c1(C(C)C(N2CCCC2CN(C(=O)Cn2cccc2)C)=O)ccc(F)cc1 35873,c1(N(C)CC2CC2(C)C)ccc(S(=O)(=O)N2CCN(C)CC2CCO)cc1Cl 35874,N1(C(CSCC)=O)CCC(NC(=O)C(c2ccc3c(c2)OCO3)C)C(F)(F)CC1 35875,n1(CC)ncc(C(=O)NCC(n2cc(CNC(c3c[nH]c(=N)o3)=O)nn2)C)n1 35876,CCC(C)CC(C)N(C(=O)CCNC(c1cn(C)cc1C)=O)C 35877,c1(C(N2C(Cn3cc(CCS(C)(=O)=O)nn3)CC2)=O)cc2ccsc2c(=O)[nH]1 35878,c1(OCCCC(C(=O)NCCF)NC(c2cc(C)c(C)s2)=O)nn(C)cc1[N+](=O)[O-] 35879,N1(C(=O)OCC)CCCCC1c1ncc(C(F)(F)F)[nH]1.C1C(=O)N1C 35880,c1(CC(N2CCN(C)C(=O)C2)=O)ccc2n[nH]cc2c1.C1(=O)CC(C)O1.N(C)C 35881,C1(NC(C2CC(C)(CC)C2)=O)C2CC3C(C2)C13C(=O)Nc1cccc(C(C)C)c1 35882,c1(C(=O)NCCN(C(=O)C(C)C(C)O)C(C)C)cc[nH]c2nccc1-2 35883,C(=O)(CC(C)C(F)F)N(C1CCCN(C(=O)CC(Cl)Cl)C1)CC 35884,CC1(C)CCC(C(=O)NC2CCc3n[nH]cc3C2)CN1C(C1CS(=O)C1)=O 35885,Cc1ccc(F)c(C(N2CCC(C)(NC(c3ncsc3S(N)(=O)=O)=O)C2)=O)c1F 35886,C1(CN=C(NCC2(NC)CC2)NCC(C)(C)C)CC(O)C12CCC2.CO 35887,CC(CC(=O)NCC(=O)Nc1ccccc1)c1ccco1.C12CCN(C1)CCN2 35888,C=C(Cl)CCC(=O)N1CCC(C(C)(O)CNC(c2ccn(CCOC)n2)=O)CC1 35889,C(=O)(C(F)(F)c1nccs1)NC(C1CCOC1)CNC(CNC=O)=O 35890,O(C1CCCc2ccccc21)CC(=O)NC1CN(C(=O)COCC2CC2)C2CC12 35891,Fc1cc(CO)cc(C(CN2CCC(C(F)(F)F)C2)NCc2ccc(Br)cc2)c1 35892,c1(NC(c2cncc(-c3cc(Cl)ncc3CO)n2)=O)ccc(F)cc1I 35893,C1(NC(C(=O)NCC)=O)CN(C(c2c(O)ncc(Br)c2C)=O)CC(C)(C)C1 35894,N1(C(C2CCC(CC)CC2)=O)CCCC2CN(C(=O)Cc3ccsn3)CCC12 35895,c1(CCC(N2CCC(n3cc(CNc4cccs4)nn3)C2)=O)ccccc1 35896,C1(NC(CCC(=O)NCCC)=O)CC2CN(C(C3CCCC3C)=O)CC12 35897,C1(C)(NC(CNC(=O)OCC)=O)CCCN(C(C2C=CC=CC=C2)=O)C1 35898,c1(C(=O)NCC2C=CC(NC(C3(COCC)CC3)=O)C2)ccc(Cl)cn1 35899,CC(C)=C=CC(=O)NC(C(=O)NOCC1CCCC1)C1CC=CCC1 35900,C12(CNC(c3n(COC)ncc3)=O)CCC(NC(c3cncn3C)=O)(CO1)C2 35901,N1(C(COCC#C)=O)CC2CCC1C2CNc1ccnc(N(C)CCO)n1 35902,N1(C(C2C(C(=O)O)C2)=O)CCc2[nH]nc(-c3cccc4ccsc34)c2C1 35903,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 35904,c1(C(N2CC(CNC(=O)C3=CCCOC3)C2)=O)cccc(S(=O)(=O)C2CC2)c1 35905,C12(NC(N(C)CC3CCCO3)=O)CNC(c3ccccc3)C1C2 35906,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3ccnc3)C2)o1 35907,C1(C(=O)OCCN(C)C)CN(C(=O)OC(C)(C)C)C(C)(C)C1.C1CCO1 35908,c1(C(=O)NC2C(CNC(c3cscc3F)=O)C2)cc(F)cnc1O 35909,CCC(C(=O)NCC1CCN1C(C1CCOCC1)=O)C(F)(F)F 35910,C1(CNC(C2(C(=O)NC)CC2)=O)CN(C(c2nn(C)cc2C(F)(F)F)=O)CCO1 35911,N1(CC(C)NC(CCCOC)=O)CCN(C(=O)CCCC2CCCO2)CC1 35912,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1cc(C(C)C)no1 35913,N12CCCC(C)(C1)C(=O)NOC(CO)C2=O.c1(OC)cn(C)nc1C(N)=O 35914,C1(NC(C(COCC)NC(=O)CS(=O)CC)=O)COCC(C)(C)C1 35915,CCCC(C)CC(=O)N1CCC(N(C(=O)C(=O)NCC2CC2)CCO)CC1 35916,c1(C(=O)NC2C(NC(C(C(C)C)N(CC)CC)=O)CC2)c(F)cccc1Cl 35917,n1(CCC(=O)NC2C(C(=O)NCCC)C2)sc2ccccc2c1=O 35918,C(=O)(CCCC(C)CC)N(CCC)CCNC(c1[nH]c(=N)sc1CC)=O 35919,N1(C(CCCOC)=O)CCC2CN(C(C3(C)CC4CC4C3)=O)CC2C1 35920,C1(C(=O)NC2(CCC=C)CC2)C2CCC(C2)N1C(=O)C(C1CC1)C1CC1 35921,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 35922,N1(C(c2c(N)cn(C)n2)=O)CC(NC(=O)Cc2cc(Cl)n(C)n2)CC2(CC2)C1 35923,N1(C(CC2CCN(C(c3c(C)coc3)=O)C2)=O)CCC(Cc2ccccc2)CC1 35924,C12C(C3CCCC13)C(=O)N2.c1(NCC=CCOCC)nnnn1C(C)C 35925,N1(C(c2cccc(OC(F)F)n2)=O)CC2CCC(C1)N2CC1CCCO1 35926,c1(C(N(CCCCNC(CN(CCC)C)=O)C)=O)cc(C#N)ccc1Br 35927,c1(SC)ccc([N+](=O)[O-])c(C(=O)NCC2CC2NC(=O)CC(C)C(C)C)c1 35928,C(=O)(CCC(C)(C)NC(=O)CC1(O)CCOCC1)NC(C)Cn1cnnc1 35929,C1(NC(c2cccc(=S)n2O)=O)CCN(C(c2cnn(CC3CC3)c2)=O)CC1F 35930,C1(NC(C(C)NC(CC)=O)=O)CCCCN(Cc2cc(Br)ccc2C)C1 35931,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 35932,CN1C2CCC1CN(C(C1CCCCN1Cc1ccc(O)c(C#N)c1)=O)C2 35933,Cc1cc(CNC(=O)CC2C=CC(NC(c3ncc[nH]3)=O)C2)n(C)n1 35934,C1(CCNS(NCC)(=O)=O)(NC(=O)OC(C)(C)C)CCC(C)CC1 35935,Cn1ncc(Cl)c1C(=O)NCCn1cc(-c2nn[nH]n2)cn1 35936,C1(OC)C(NC(=O)CC(C)C(C)(C)NC(c2cnnn2C(C)C)=O)CC12CCC2 35937,c1(CCC)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 35938,c1(OC)cc(CC(N2CCC(C)(NC(c3cc(C(F)F)on3)=O)C2)=O)cc(Cl)c1 35939,N1(C(CC2(C=C)CN(C(c3cnn(C(C)C)c3N)=O)C2)=O)CC2(CC(O)C2)C1 35940,N(C1CCCn2cnnc21)Cc1ccc(OC)cn1 35941,Cc1ccc(CCC(=O)NCC2CC(NC(c3cccnc3)=O)C2(C)C)cc1Cl 35942,Cc1ccc(S(=O)(=O)N2CC(C)NC(C)C2)cc1NC(=O)C(N)C1(F)CCC1 35943,c1(C(C)N)nn(C)c2ccccc12.C(=O)(CO)NCCSCN 35944,C1(OCCNC(=O)Cc2ccon2)CCN(C(=O)CCC2CC2(Cl)Cl)C1 35945,C(=O)(CC(CNC(=O)CN1CCC(=O)CC1)C1CCC1)N(C)CC1CCC1(C)C 35946,C(=O)(CC(c1ccccc1)C1CC1)NCCCNC(C(=O)NCC(F)F)=O 35947,c1(CC(=O)NC2CCN(C(c3cc[nH]n3)=O)C23CC3)ccc([N+](=O)[O-])cc1 35948,C(=O)(CCS(=O)(=O)c1ccccc1)NC1C(CNC(C=CCOCCOC)=O)COC1 35949,CCCC(CC)CC(=O)NC1CN(C(=O)CNc2cccc(C#N)c2)CC1O 35950,C1(F)(C(=O)NCC(C)N(C(C2(C(C)C)CC2)=O)C)CC1C 35951,C(=O)(CCCC(=O)N1CCC1CNC(=O)C=CCF)N(c1ccc(O)cc1)CCC 35952,C(=O)(CCCCN=[N+]=[N-])NC(CN(C(C1(C2(C)CC2)CC1)=O)CC)C 35953,N1(C(CN(C(=O)Cc2nccn2C)C)=O)CCN(C(C2(C)CCCS2)=O)CC1 35954,C(=O)(C(F)(F)F)N(C(=O)C=Cc1cscn1)CCF.C12COCC1NC(=O)CS2 35955,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 35956,C#CCCC(CC)NC(=O)CC(C)CNC(=O)CS(=O)CC 35957,N1(c2cc(NCC(F)(F)Br)nc(C)n2)Cc2cccc(C)c2C1 35958,Nc1nccnc1C(N1CCC(O)(CNC(c2nc(Cl)cs2)=O)C1)=O 35959,c1(C(=O)NC(C2CCCN2C(c2sccc2Br)=O)C)cccc(=O)n1C 35960,CCCC(C(=O)NCC1(F)CC(CNC(C2(COC)C=CCC2)=O)C1)N(C)C 35961,N1(C(CCC(=O)NC)=O)CCN(C(c2coc(C(C)=O)c2)=O)C(C)C1 35962,C1(C(=O)NCCCNC(C2(S(N)(=O)=O)CCC2)=O)CCc2nccn2CC1 35963,Cc1cc(C(N2CC(C)(NC(=O)CC3CCCOCC3)C2)=O)cc(N)c1 35964,C(=O)(C1CCCn2c(C)cnc21)NCC1CCCN(C(CC(C)F)=O)CC1 35965,N1(C(C2(C(N(C)C)=O)CC2)=O)CC(NC(C2OCCCO2)=O)C(C(F)F)C1 35966,c1(NC(C(=O)N(C)C)=O)cccc(CC(N2CCCC2C2CCCC2=O)=O)c1 35967,C1(N(C(=O)CC2(N3CCOCC3)CC2)CC)CCN(C(C2CC(F)C(=O)N2)=O)CC1 35968,CC1CC=C(C(=O)N2CCCC(CC(=O)NC3(CO)CCCCC3)C2)CC1 35969,c1(C(=O)NC2CC(OC)C(O)C2)ccc(C(N2CCCCC2CO)=O)c(C)c1 35970,N1(C(C2C(C)(C)C2)=O)CC2(CC(C(=O)NC(C(N)=O)C3CC3)CO2)C1 35971,C1(CC)CC(C(=O)NC(c2ccnn2C)C(=O)NCCSCCOC)CCO1 35972,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)Cc2cnoc2)CC1)C)C 35973,c1(C(=O)NCCOCCCN(C(C2(CC)CC2)=O)C)cc2c(cc1Cl)CCCC2 35974,c1(C(=O)NC2CCC(CCNC(c3c(OC)csc3)=O)C2)cn(C)c(=O)cc1C 35975,Cc1ccc2c(c1)CCC2=O.N1CC(F)CC1CNC(=O)CCC1CCOC1 35976,C=CCC(C)(C)CC(=O)NCC1C(CNC(C2CCOC2C)=O)C1(F)F 35977,c1(C(C)CC)nc(C)c(C(=O)NCc2nc(CO)sc2)s1.C(=O)(C(F)C1CC1)C 35978,C12(CNC(C3CC4CCC4C3)=O)CCC(NCCCCC3CC(F)C3)(CC1)CO2 35979,c1(C(=O)OC)cnc2n1CCN(C(=O)Nc1cccc(Br)c1N)C2 35980,C1(CNC(c2ccnc(CO)c2)=O)CC2CC2N1C(=O)COCC1CCOCC1 35981,C1(NC(C=Cc2cc(OC)ns2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 35982,c1(CC(C)NC(c2ccc(C#N)[nH]2)=O)ccc(CNC(C2CN(C)C2)=O)cc1 35983,N1(C(c2cccc(OC)n2)=O)CCC2(CCCN(Cc3ccc(I)cc3)C2)CC1 35984,N1(C(C2(CC=C)CCC2)=O)CC(CNC(=O)C(n2cc(C)cn2)C)C(O)C1 35985,c1(C(=O)NC2C(CNC(c3ncc(F)s3)=O)CCCC2)cnn2c1C(=O)NCC2 35986,C1(C(=O)NCc2ccc(C(N(C3CCCC3)CCC#C)=O)s2)CC(C)(C)CN1C 35987,C(=O)(CCCCC#N)NCC(C)(CO)NC(=O)CCC1CCC(=O)NC1 35988,C1(CNC(C(C#C)(C)C)=O)CCCC2(CCN(C(c3nc(C)oc3C)=O)CC2)O1 35989,c1(CC(=O)NCC(CNC(CN(C2CCCCC2)C)=O)O)cc(F)ccc1O 35990,N1(C(C(C)OCC#C)=O)CC(NC(=O)CCn2cc(C)cn2)C(C)C1 35991,n1(CC#C)cccc1C(=O)NC(C)CNC(c1cc(C2CCC2)no1)=O 35992,c1(CC(=O)NCCC(C)NC(CC(CC)OC)=O)cccc(F)c1F 35993,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CNC(=O)C2)c1 35994,C1(NC(C(C)(C)NC(C2CNC(=O)N2)=O)=O)CCCCC1CO 35995,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 35996,C(=O)(C(O)CCSC)NC1(CCC(=O)NCCCC=CC)CCCC1 35997,C=CC1CN(C(=O)C=CC(CC)=CC)CC1N(C(=O)CCc1ccccn1)CC 35998,C1(c2n(C)ncc2)CN(C(C2CCC(C(F)(F)F)N2)=O)CCO1 35999,C=C(C)CC(=O)NCCCN(C(=O)C(C1CCC(C)O1)SC)CC1CCCCC1 36000,N1(C(C2CCCOC2)=O)CC2CCN(C(C3(O)CCSCC3)=O)CC12 36001,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36002,N1(C(C(c2ccccc2F)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36003,N1(C(C2(CC)CCCC2O)=O)CCC12CN(C(=O)C(C)(C)C1CCOC1)C2 36004,CCCCCC(C)(C)C(=O)N(C)CCN(C(=O)Cn1cc([N+](=O)[O-])cn1)C 36005,C(CCCCCCCO)=CC(=O)NC1COCC1CNC(=O)CCCCCC#N 36006,C#CCC(CC(=O)NC1CC(CNC(=O)Cc2cc(C)no2)C1)c1ccccc1 36007,C(=O)(CC(C)C(C)C)NC1CC(C)(C(=O)NCCC2(OC)CCCC2)C1 36008,c1(C(=O)NCC(N2CC=CC(NC(C=CC)=O)C2)=O)cc[nH]c2nccc1-2 36009,C(c1cccc(C)c1)=CC(N1CC(N(C(=O)COc2ccccc2Cl)C)C(F)C1)=O 36010,C1(C(=O)Nc2cccc(NC(c3cnn(C)n3)=O)c2)CC2(C1)CC2(F)F 36011,C1(C(N(C2(COC)CC2)C)=O)CC12CC(NC(=O)CCc1cscn1)C2 36012,c1(OCC)ccccc1OC.N12CC3CC1(C3)COC(=O)C2C1CCCC1 36013,C1(C(=O)NC(C)C(=O)NC(C)(C)C)C(C2CC2)CCN1C(C12CCCN1CCC2)=O 36014,C(CC(CC)C(=O)NCC(=O)NC(COC)C(C)C)=CC.C1C(=O)N1 36015,Cc1ccc(CC(=O)NCCNC(C2(n3ccnn3)CC2)=O)cc1 36016,CCCCC(CC(=O)NCC1=C(C)CCC1)NC(C1CC2(CC2)CO1)=O 36017,n1(CC(=O)NCCCCN(C)C(c2cnc[nH]2)=O)nnc(-c2ccco2)n1 36018,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36019,N1(C(Cn2nnc(C)n2)=O)CCCCC(N(C)C(c2nn(C)cc2Cl)=O)C1 36020,C(=O)(C1CCCc2ncc(C)n21)N1CCC(NC(CCc2nnc(CC)o2)=O)C1 36021,c1(OC)ccc(-n2cc(CC3CCOC3)nn2)cc1.c12ccc(nc1)N(C)C2 36022,CC1CC(F)(F)CN1C(=O)C=CC(C)(C)NC(=O)C=CC1CCC1 36023,CCCC(C(=O)OC)C(=O)N1CCC(C)(C(=O)NC(c2cncnc2)C)C1 36024,C(C1CCOCC1)=CC(=O)NC1CC(NC(C2(C(N)=O)CCC2)=O)C1 36025,c1(C(=O)NC(CNC(c2cnn(C(C)C)n2)=O)C(C)(C)C)ncnc2sccc12 36026,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36027,C(=O)(C(C)(C)CC#N)NC1C(NC(c2c(SC)cn(C)n2)=O)COCC1 36028,N1(C(C(N2CCC(O)CC2)C)=O)CCCC(CC(=O)NCCn2cncn2)C1 36029,c1(C(N(CCCOCCNC(C(C)=C2CC2)=O)C)=O)cc2oc(C)c(C)c2[nH]1 36030,c1(OCC)ccccc1C(=O)NC(c1cnc[nH]1)C 36031,C1(C(N2CC(OC)C(NC(c3ccnc(N(C)C)c3)=O)C2)=O)CCCC(=O)N1C 36032,c1(CN(C(CCNC(=O)OC)=O)C)nnc(CNC(C2CC2C(N)=O)=O)s1 36033,C1(C(=O)NC2CCC(NC(=O)Cc3ccccc3F)CC2)(COC)CCOCC1 36034,C=CC(CCC)CC(=O)NCC1CCN1C(c1cc(F)c(N)c(F)c1)=O 36035,N1(C(=O)OC(C)(C)C)CCC(N=[N+]=[N-])(C(=O)OCC(C2CCCC23CCC3)=O)C1 36036,C1(C(=O)NC(C2(CCOC)CC2)=O)CCCCC1O.C1(=O)CC2(CC2)CN1C 36037,N1(Cc2cccs2)CCN(NC(=O)NC(C)(C)CNC(=O)CN2CCCC2)CC1 36038,C1(c2cn(C3CC(NC(=O)NCCc4ccc(C)o4)C3)nn2)CC12CCCCC2 36039,c1(C(=O)NCC2N(C(c3cc(COC)no3)=O)CC2)ccc([N+](=O)[O-])cn1 36040,C(=O)(C(CO)C(F)(F)F)N1CCN(C)CC1C(=O)NC1(C)CCCC1(C)C 36041,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CC3CC=CCC3)CC2)c(O)n1 36042,N1(C(CC=C)=O)CC(NC(C2CCC(CN(C)C)O2)=O)C(SC)C1 36043,C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(=O)C(C(C)C)c1cccnc1 36044,C12(C(=O)NCC(CNC(C(N3CCOCC3)C)=O)C)CCCCC1C2(F)F 36045,Cc1ncnc(N2CCOC(CNC(=O)CSc3cccc(Cl)c3)C2)c1Br 36046,C12CCCN(C1)c1nnc(o1)CC(=O)N2C.c1(C(OC)OC)ccccc1Cl 36047,c1(CNc2c(C(=O)Nc3c(C)cnc(O)c3)nccc2)c(Br)ccc(Cl)c1F 36048,C(Cc1cnc[nH]1)(C(=O)N1CC(C)(CN(C)C)C1)NC(CN(C(C)=O)C)=O 36049,c1(C(=O)NCC(CC)(C)NC(c2[nH]ncc2C#N)=O)cc2c(F)cc(F)cc2[nH]1 36050,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36051,C1(C(=O)NCCN(CCCCCC)C(=O)C=Cc2cn(C)nn2)CCCCN1C 36052,C(=O)(C1=CCCSC1)N(CC(C)NC(=O)CCC(=O)N(C)C)CC 36053,c1(C(=O)NCC2(NC(C3N(CC)CC3)=O)CCC2)cc2nc[nH]c2cc1N 36054,N1(CC2(c3cn(C(C)C(=O)NCC4(Br)CC4)nn3)CCC2)CCN(C)CC1 36055,CC1(C(=O)NC(CCF)C(=O)NC2CC(N3CCCC3)C2)CCC(=O)NC1 36056,C1(NC(CSCC=C)=O)CC(C)CN(C(=O)Cc2c[nH]nc2O)C1 36057,c1(CNC(NCCOC)=NCCc2cn3c(n2)SCC3)ccc(C#N)c(F)c1 36058,c1(OC(C)C)ccccc1C(=O)NC(c1cnn(C2CCOC2)c1)C 36059,C=C=CC(C)C(=O)NCCCCN(C)C(c1cc(C)n(CC(F)(F)F)n1)=O 36060,c1(OCC)cncc(C(=O)NCC2(C(N)=O)CN(C(=O)C(C(C)O)N(C)C)C2)n1 36061,C1(NC(c2cncc(OC)n2)=O)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 36062,C(=O)(C#CC(C)(C)C)N(CC(=O)NCCNC(=O)CN1CCNC(=O)C1)C 36063,CC1(CNC(C2CC3(C2)CC32CC2)=O)CCCN(C(=O)CC2CC(=O)NC2=O)C1 36064,c1(N2CC(C)C(CO)CC2)ccc(S(=O)(=O)NC=O)cn1.c1(C)ccnc(Cl)c1 36065,C(CCCCCC(=O)NC1CC2(CCC2)C1)NC(C1N(C=O)CCC1)=O 36066,Cc1cc2cc(F)cc(CNC(c3cccc(C(F)C(F)(F)F)n3)=O)c2nc1Cl 36067,CC(C)CC(O)CC(=O)N1CC(C)C(C)(C(=O)NCC2(C)CCCC2O)C1 36068,Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccnc(F)c3F)=O)C2)cc1N 36069,c1(OCC)ccc(C(=O)NC2CCN(C(=O)C(c3cnn(C)c3)C)C2)cn1 36070,C1(NC(c2cnc(C)s2)=O)(CNC(=O)Cc2cccc(F)c2)CCCCC1C 36071,N1(C(c2cc[nH]c2)C)CC2C(C(=O)NCc3ccc(Cl)cc3)C2C1 36072,c1(CCN(CCC=C)C(C)=O)c(C)nn(C2CCCCO2)c1C 36073,CC1CCCN(C(=O)CC(C)(C)C#N)C1CNC(=O)CCc1cc(Cl)no1 36074,C1(C(N2CCC(C)(C)C2)=O)CCC2(CC1)NC(=O)c1ccccc1NC2=O 36075,C=CCC(CC(F)F)C(=O)NCCCN(C(c1n[nH]cc1[N+](=O)[O-])=O)C(C)C 36076,c1(OC)cc(CC(N2CCC(NC(C3CCCOCC3)=O)C2(C)C)=O)ccc1C 36077,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36078,CCC1=NOC(CC(=O)N(CCC)CCNC(c2ccc(CC(N)=O)cc2)=O)C1 36079,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36080,CC(C)C(CNC(C1CCC(N(C)C)C1)=O)C(=O)N1CCCC(C)C1 36081,C1(C(N(C(C)C(=O)NOCC(=O)OC)C(CC)(C)C)=O)CC(F)(F)C1(C)C 36082,N1(C(=O)NC2N(C(C(C)NC(CC)=O)=O)CCCC2)CCN(C)CC1C 36083,C1(CNC(CC=C)=O)CC(C)N(C(c2cccc(CNCC#N)c2)=O)C1 36084,N1(S(C)(=O)=O)CC2CCC1C2CC(=O)NNC(=O)c1ccc(Cl)cc1 36085,Cc1cc(C(N2CC(N(C)C(c3cc(C4CC4)no3)=O)C3(CC3)C2)=O)c(C)cn1 36086,C(=O)(C(CNC(=O)Cc1cncnc1O)CC(C)C)N1C(C=C)CCC1 36087,C(=O)(C(CNC(c1oncc1CC)=O)CC(C)C)NC1(CC)CCC1 36088,C1(N(C(=O)CC2CCC3CC23)CC)CCN(C(=O)Cc2ccccc2F)CC1 36089,CC1CN(C(c2cc(C(C)(C)C)on2)=O)CC(C)C1NC(c1n[nH]c(C2CC2)n1)=O 36090,N1(C(C2CCOC2)=O)CCCC(Cn2cc(C3CC=CCC3)nn2)C1 36091,C1(NC(CCCC=C)=O)CC2CC1N(C(c1ccsc1SC)=O)C2 36092,N1(C(C(C(C)(C)C)n2cc(CN3CCSCC3)nn2)=O)C2CCC1CC(F)C2 36093,c1(NC2C(C)(C)SC2)c(C(=O)O)nc2ccccn12 36094,c1(C(N(CC(=O)NCC(F)(F)C(F)(F)F)C)=O)ccnc2ccccc12 36095,c1(C(N2CCN(C(c3cn(CC)nc3)=O)C(CO)C2)=O)cccn2c(O)nnc12 36096,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36097,CCC(CCC(=O)N1CCC(C(C)(F)F)CC1)OC 36098,C(C(=O)NNC(=O)c1ccc(Cn2cccn2)o1)Oc1cccc(CC#N)c1 36099,C1(C(NOCCOC(C)C)=O)CC(NC(=O)CCC2CCCN2C)C1(C)C 36100,C1(COC)COC(C)(C)CN1C(c1cc(C)nc(OC)n1)=O.CCC1CNC1=O 36101,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(F)F)N1CCCC(C(C)C)CC1 36102,c1(NC(C2N(C(COCCCCC)=O)CCC2C)=O)cnc(F)cc1C 36103,C1(NC(C2N(C)CC(C)(C)C2)=O)C2CCC1CN(C(c1ccc(F)c(F)c1)=O)C2 36104,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36105,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)C=C2CC2)C1 36106,C#CC1CN(C(c2cc(CC)[nH]c2C)=O)CCN1C(=O)CCc1ccc(Cl)s1 36107,C#CC1(C(=O)NCCC(=C)CNC(C2(N3CCCC3)CC2)=O)CCCCC1 36108,Fc1cc(F)c(CN2CCCC2CSc2ccc3c[nH]nc3c2)c(F)c1 36109,C(CCCC(C)(C)C)c1nnc(C(c2cncnc2)C)o1 36110,c1(C(C(=O)N(CCC(C)NC(CC(C)N2CCCC2=O)=O)C)O)ccc(O)cc1 36111,C1(NC(CCOC)=O)CC=C(C(=O)NCC2CC3C=CC2O3)C1 36112,N1(C(c2nnc(C(C)(C)C)s2)=O)CCC2(CC1)CCN(C(=O)C=CS(C)(=O)=O)C2 36113,N1(c2snc(C(C)C)n2)CC2(COC(CNC(c3cnc(O)nc3O)=O)C2)C1 36114,c1(C(=O)NCC(C)NC(=O)Cc2ncn(C)n2)ccc(-c2ccco2)nc1C 36115,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36116,Cc1nc(N)c2c(C)c(C(=O)NCc3ccc(CO)cc3)sc2n1.C12CCN1C2=O 36117,N1(C(C2CC(C)(C)OC2)=O)CCc2sc(CNC(=O)COCC(F)(F)F)nc2C1 36118,c1(CC)ncc(C(=O)NC2COCC2NC(=O)CCC2CC2(F)F)c(C)n1 36119,C1(C(=O)Nc2scc(C3C(CC)C3)n2)C(C2CC2)CCN1C(=O)OC(C)(C)C 36120,C(C)(C)(C(=O)NC1CCC1CNC(=O)CN1CCCC1C)SC 36121,C(C(=O)NNc1ccc(Br)cc1F)c1nc(C)sc1 36122,N1(CCC)CCC(N=c2[nH]c(N3CC4COCC(C4)C3)nc(=NC)[nH]2)C1 36123,c1(C(N2CCC(N3CCC(N(C)C)CC3)CC2)=O)ccnc2ncccc12 36124,C1(CC)CN(C(=O)C(C2CCC2)NC(c2ccnnc2C)=O)CCO1 36125,N1(C(C=CC)=O)CCC2CCN(C(=O)Cn3ccc(C(=O)OC)cc3=O)CC2C1 36126,c1(C(=O)OCC)nccn1CCNCc1cc(-c2ccccc2)no1 36127,C#CCN(OC)C(=O)C(C)NC(=O)C(CC(=C)C)SC 36128,CCC(O)C(C)C(=O)NCCCC1CCN(C(=O)COCCO)CC1 36129,Cc1c(C(=O)N(CC(O)CN(C)C(C2COC(=O)N2)=O)C)[nH]c2c(C)cccc12 36130,C1(NC(C2ON=C(CC)C2)=O)CN(C(=O)COc2c(F)cccc2Cl)C(C)(C)C1 36131,CC1(C)C(CNC(C2CCCC2)=O)CCN1C(=O)CC1COC(=O)C1 36132,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36133,C#Cc1cnn(C)c1C(N1CCC(NC(=O)C(CC)SC)C12CC2)=O 36134,C1(C2(NC(C(C)=C3CCC3)=O)CC2)CCCCN1C(=O)CCc1conc1C 36135,N1(C(C#CC2(C)CC2)=O)CC2CCCCC2(CNC(C2(C)CCS(=O)(=O)CC2)=O)C1 36136,c1(-c2n(CCC)ccn2)ccc(C)cc1SC 36137,O=C1CCC(CNC(C2C=CC(c3ccccc3)C2)c2cn(C3CC3)nn2)CCO1 36138,C(=O)(CS(=O)(=O)CCO)N1C(CCCNC(c2cccc(OC)n2)=O)CCC1 36139,C#Cc1ccc(C(N2CC(C)CC2C(=O)N(c2cnn(C)c2)C)=O)cc1C 36140,Cc1nc[nH]c1CC(O)CN(CCCNC(=O)OC(C)(C)C)CCCO 36141,C(C)(N=c1[nH]c(=NCC(CO)C2CCCCC2)c2c(ncn2C)[nH]1)c1ncc(C)s1 36142,C1(C(=O)NC(CC)CNC(c2snnc2C)=O)CCN(S(=O)(=O)NC)CC1 36143,C(=O)(C1=CC2C=CC1C2)NC(CC1CCN(C(c2c(C)c[nH]n2)=O)CC1)C 36144,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)n1)=O 36145,C1(C(N2CCC(CN(C(=O)C(=O)NCC3CC3)C)C2)=O)CCc2n[nH]cc2C1 36146,n1(CC)ccnc1C=CC(=O)NCC1CCC(NC(C2(C(F)F)CCCO2)=O)C1 36147,C(CCCCN(C(=O)CSc1nncs1)C)NC(C(c1ccnn1C)OC)=O 36148,Cn1cc(C(=O)NC2CC(C)(NC(=O)C(C)(F)C(F)(F)F)C2)c(O)nc1=O 36149,NS(=O)(=O)CCCCCC(=O)NC1(CNC(=O)Cc2ccccc2F)CCCCC1 36150,N1(C(CC(CC)C)=O)CC(CNC(c2sccc2C#N)=O)OC(C)(C)C1 36151,Cc1cc(N2CCCC(CNC(=O)C(C)C(F)F)C2)ccc1[N+](=O)[O-] 36152,C(=O)(CN1C(=S)N(C)C(C)(C2CC3CCC2C3)C1)Nc1ccc(OC)cc1 36153,N1(C(C(C)N(C)CC)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36154,c1(NC(C)=O)cnc(C)c(C(N2CCCC2CN(C)C(C2CCCS2)=O)=O)c1 36155,C(N=c1[nH]c(=NC2CCN(C3CC3)C2)[nH]c2ccsc12)c1c(Cl)cccc1Br 36156,c1(OC)cc(F)c(NC(C2CCCN2S(=O)(=O)C(F)(F)F)=O)cc1F 36157,Cc1sccc1C(=O)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C 36158,CC1CN(C(=O)Cc2ccc3sccc3c2)CC(C)CN1C(c1csc(F)c1)=O 36159,CC1CC=C(C(=O)N2C(CNC(c3coc(Br)c3)=O)CC3CCCC23)CC1 36160,c1(OCC(=O)NC2CCC(NC(C(C(C)C)SC)=O)CC2)cc(C)ccc1F 36161,c1(C(N(C2CN(C(c3ccc(CC)nc3C)=O)C2)C)=O)cc2sc(NC)nc2s1 36162,c1(CC)cc(N(C(C)C)CC2CCS(=O)(=O)C2)ccc1OC 36163,c1(SC)nc(NCC2CCCN2C(=O)CCc2cccc(F)c2)cc(Cl)n1 36164,CCC(CC(C)C)C(=O)N1CCC1CC(=O)NCC(=O)NC 36165,c1(C(C(N2CC(C3CC3)C2C2CCNCC2)=O)NC)c[nH]c2ccccc12 36166,C1(O)(CNC(C(C)C(F)F)=O)CCCN(C(C23CCC(C(F)F)(CC2)C3)=O)CC1 36167,c1(C(c2n(CC(=C)C)nnn2)NCCc2cccc(F)c2)cc(F)c(F)cc1F 36168,S(=O)(=O)(C1CCN(Cc2ccccc2)CC1)N1C(C(=O)O)CCS(=O)(=O)C1 36169,c1(C(N2CCOC3CN(C(COC)=O)CC32)=O)cnc2c(C)cccc2c1 36170,C1(CCNC(c2cn(CC3CC3)nn2)=O)CCCN(C(C2(CC=C)COC2)=O)C1 36171,N1(C(c2coc(C(F)F)c2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C(CO)C1 36172,c1(CCC)cc(NC(=O)N(C(CO)CCC)CC)c(C)o1 36173,Cc1nccc(N2CCC2)n1.C12(CCCC1)CC(=O)N(C)CC(C)N(C)C2=O 36174,C1(O)(CNCC(=O)NS(C)(=O)=O)CCCN(C(=O)CC2CC3CCC2C3)C1 36175,N1(C(C(CC)OCC)=O)CCC(O)(C(C)NC(=O)CCC2(C)CC2)C1 36176,c1(C(N2CCN(C(C)=O)C(CO)C2)=O)cc2ccc(C(=O)O)cc2n(C)c1=O 36177,C1(NC(C2(N)CC2)=O)CCC(CC(C)C)CC1.C1(CCC)(C(=O)NCC)CC1 36178,c1(-c2ccc(NC(C)=O)cc2)c(C)ccnc1F 36179,c1(OC)ccc(Cl)c(OC)c1C(N1CC(F)(NC(c2c(C)cccc2C)=O)C1)=O 36180,N1(C(CN(CC#C)C(c2ccsc2Cl)=O)=O)CCCC1C 36181,c1(CC)cncc(C(=O)NCC(C2CCC2)O)c1.c12conc1C(=O)NC2 36182,Cc1cncc(C(N2CCOC(CN(C)C(c3cc(Br)oc3C)=O)C2)=O)n1 36183,C1(CC(=O)NC2CCC(CN=c3ncc(Br)c[nH]3)C2)CCCC12NC(=O)NC2=O 36184,N1(C(=O)Cc2cscn2)CCCN(C(C2CCOC2)=O)C(c2ccccc2)C1 36185,C1(CC=C)(C(=O)NCCCC(C)(C)NC(=O)C(C)NCC(F)(F)F)CCCCC1 36186,C(CC(O)CC(=O)NC1CCCN(C(=O)CC2(O)CCC2)CC1)SC 36187,C1(NC(C(C)NC=O)=O)CC2CCC1(C(N1CCCC1C)=O)C2 36188,c1(C(N2CC(C)(CNC(C(C(=O)NC)(C)C)=O)OCC2)=O)csc2ccccc12 36189,c1(C(N2C(C(N3CCC(CCO)CC3)=O)CC(F)C2)=O)ccc2cccnc2c1 36190,c1(C(C)(C)C(N(C(C)C)Cc2cccc(F)c2)=O)cc(F)c(Cl)cc1Cl 36191,Cc1cc(C)c(C(N2CCOC(C(C)NC(=O)C=CC(F)(F)F)C2)=O)c(O)n1 36192,C(c1ccc(Br)cc1)=CCC(N1CCC(C)(CCNC(=O)C(F)F)C1)=O 36193,CC1(C)CN(C(C2(c3ccno3)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)C1 36194,c1(CNC(C2(COC)CN(C(C34CCC(CO3)C4)=O)C2)=O)cc(OC)ncc1F 36195,C#CCCCCC(=O)NCC1(C(=O)NC(C2CCCO2)CO)CC(=C)C1 36196,N1(C(CCS(C)=O)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36197,C1(OC)CC(NC(=O)C(C)Cn2ccnc2)CN(C(C2(n3nccn3)CC2)=O)C1 36198,c1(C(=O)NC2C(NC(C3(CCN(C)C)CC3)=O)CC2)cccnc1C(F)(F)F 36199,c1(NCC2C(C)CN(C(c3ccc(=O)n(C)c3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36200,c1(CC)ccc(C(=O)N(CC(=O)NC2CSCC2C)C(C)C)o1 36201,N(C(=NCc1cc(C)nn1C)N1CCc2ccc(Cl)cc2C1)CC(C=C)(F)F 36202,Cc1cccc(CO)c1NC(=O)C(N1CCCC(N(C)C)C1)C.C1(=O)CO1 36203,N1(C(CN(C(C2C(CC)OCC2)=O)C(C)C)=O)CC(C)CC(C)(C)C1 36204,Cc1nc(NC(=O)NC(C2CCOC2)CO)sc1C 36205,C12(NC(c3nocc3Cl)=O)CCCC1N(C(c1ccc(OC(F)F)cc1)=O)CC2 36206,C1(CNC(C(C)(C)OCCC)=O)CCN(C(c2coc3c2COC3)=O)CC1O 36207,C1(C(C)C)C(NC(C2CCC(C(N)=O)CC2)=O)CCN1C(=O)CC(F)(F)Cl 36208,c1(NC(=O)NC(C)CCc2ccccc2)cc(P(C)(C)=O)ccn1 36209,Cc1cc(F)c(C(=O)NCC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)cc1F 36210,Cc1cccc(-c2cncc(C(=O)OC(C)C(N)=O)c2)n1 36211,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(C)O)C2)=O)c1C 36212,c1(NC(C(N2CCN(C3(C)CC3)CC2)CN(C(C)=O)C)=O)cc(S(N)(=O)=O)c[nH]1 36213,C1(CNC(c2ccc(C)cc2)=O)CCCN(C(c2cc[nH]c2C2CC2)=O)CC1 36214,C(=O)(C(C(=O)N(C)C)c1ccccc1)NCC(C)(C)NC(=O)C(F)n1cccn1 36215,C1(CNC(C(OC)OC)=O)CN(C(c2ccc(OC3CCC3)nc2)=O)CC12CC2 36216,C#CC1(S(=O)(=O)NC(c2nn(CC(F)(F)F)cc2Br)=O)CC1 36217,N1(C(c2c(C(C)C)noc2)=O)CCN(C)CC1CNC(=O)Cn1nccc1N 36218,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36219,c1(C(=O)NCC2(CNC(C(CCOC)OC)=O)CC2)cnc2[nH]c(O)nc2c1 36220,C(C(C(=O)NCC1CC(C)(NC(=O)C(C)Sc2nncn2C)C1)NC(C)=O)OC 36221,C1(NC(c2n(C)cc(C(N)=O)c2)=O)COC2CN(C(=O)CN3CC=CC3)CC12 36222,NC(=O)CCC(C(=O)O)NC(=O)CC(n1ccnn1)C1CC1 36223,c1(OCC(=O)NC(CC=C)CNC(C2CCCC2(F)F)=O)ccccc1C(F)F 36224,C(=O)(N=c1[nH]c(Cl)nc(O)c1Cl)c1c(OCC)nc2sc(C)cn21 36225,C1(C)(C(=O)NC2CC(C)(NC(C3CC4C(C3)C4(C)C)=O)C2)C2CC3CC(C2)CC1C3 36226,C1(COC)C(C(=O)NCCCCCNC(=O)C(C2CCOCC2)OCC)C1(C)C 36227,C(=O)(C(C)(C)c1cccs1)NC(C1CC(NC(=O)Cc2cnc[nH]2)C1)C 36228,C1(NC(CC(=O)OC)=O)CN(C(c2ncc(Br)cn2)=O)CC1O 36229,c1(C(N2C3C(CNC(C4CC(C)(C)C4)=O)C(C3)C2)=O)ccc2ncc(=O)[nH]c2c1 36230,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36231,CC1CCN(CC(=O)NCC2CCC(N(C)C(C3(C4CCC4)CC3)=O)CC2)CC1 36232,C(=O)(C(C(C)C)N(C)C)N1CC(=C(CNC(CNC(CCCC)=O)=O)F)C1 36233,CC1CN(C(C2CCCC2CNC(C23C(=O)C4CC2C3C4)=O)=O)CC(C)S1 36234,N1(C(C(OC)OC)=O)CCC2(CCC2)C(C(=O)NCC(CO)OC)C1 36235,C1(O)(C(C(=O)NC2CC(NC(c3c(C)snn3)=O)C2)(F)F)CCOCC1 36236,N1(C(c2nc(CNC(C(CCC)NC(N)=O)=O)oc2)=O)CCC2(CCCN2C)C1 36237,c1(C(N2CCC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36238,c1(C(N(C(CN(C(C(C(C)C)F)=O)C)C)C)=O)nc(S(C)(=O)=O)n2ccccc12 36239,C1(C)(NC(C#CC(=O)NS(C)(=O)=O)=O)CCCC1(F)F 36240,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36241,C1(CC(=O)NC2(CC)CCCOC2)CC2(C1)CN(C(c1ncc(F)cc1N)=O)C2 36242,c1(C(N2CC(C)C(CC(=O)NC3(C4CCCO4)CC3)C2)=O)cc2ncccc2[nH]1 36243,C(CC(O)C(F)(F)F)NC(C1N(C(c2cc(C(C)=O)[nH]n2)=O)CC1)=O 36244,Cc1nn2c(c1CNC(=O)C(C)c1ccco1)CN(C(C1CCC(C)O1)=O)CC2 36245,c1(CNC(c2c(C)coc2)=O)nn(C)c2c1CN(C(C1CC1C(F)F)=O)CC2 36246,C1(C(C)NC(C2(COC)CCCCC2)=O)CCN(N2CCC2C(=O)OCC)CC1 36247,CC1CC(=O)NC(C(=O)NCc2ncoc2CCNC(C2CCCOC2)=O)C1 36248,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36249,C1(CC)COCCN(C(=O)C(C)N(C(c2cc(C(=O)N(C)C)on2)=O)CC)C1 36250,C1(C)(C(=O)OC)CCN(C(c2ccc(C)c(I)c2)C(=O)NC2CC2)CC1 36251,c1(C(=O)NC(CC)(C)CCNC(c2sccc2CO)=O)c(O)cc(F)cc1F 36252,C(=O)(C(O)Cc1ccccc1)NCCCN(C(=O)CC1CCCO1)C(C)C 36253,c1(-n2c(C(CC)CO)nc(CO)n2)ccc(S(=O)(=O)CC)cc1 36254,C1(NC(CC(C)(C)SC)=O)CN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(C)(C)C1 36255,C1(NC(CN(CCOC)C)=O)CN(C(c2c(F)ccc(F)c2F)=O)CC(C)(C)C1 36256,c1(N(C)C(C)C)[nH]c(=NC2CC2c2n(-c3c(C)cccc3)ccn2)nc2scnc12 36257,Cc1ccc(C)c(C(=O)NC2CC(C)N(C(C3CC(O)(C(F)(F)F)C3)=O)C2)c1 36258,c1(CC(=O)NC(C)C(c2cnn(C(C)(C)C)c2)O)ccc(F)cc1F 36259,C=CC(CC)C(=O)NC(c1cccc(C)c1)CNC(=O)C(CC)SC 36260,c1(OC)nc(C(N2CCC2CNC(=O)CCCSc2ccco2)=O)cc(O)n1 36261,NS(=O)(=O)c1cc(C(=O)NC2CC23CC(NC(=O)CN2CCCC2CO)C3)co1 36262,C(C(C)NC(=O)Cc1cc(C)cs1)(C(C)C)NC(C1(CCC=C)CC1)=O 36263,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36264,C1(F)(CNC(CCC=C)=O)CCCN(C(=O)C(N2CCCCC2=O)C)CC1 36265,c1(C(N(CCCCN(C(C(CSC)O)=O)C)C)=O)ccc2nnnn2c1 36266,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36267,CN1CCC(C(=O)NCC2(O)CN(C(C3CCCC34CCC4)=O)C2)S1(=O)=O 36268,Cc1cc(C)n(C(C)CNC(N2CCCC2C(c2ccncc2)(C)C)=O)n1 36269,c1(OC)cc(F)c(F)cc1NNC(=O)C(c1cnn(C)c1C)OC 36270,c1(C(=O)NC(CC(=O)N(CCN(C)C)C)C2CC2)ncncc1Cl 36271,C(CCCCC(=O)NCC1(CC(N)=O)CC1)N(C(c1ccc(CC)cc1)=O)C 36272,C12CCCC(C1)C(=O)N2.C1(NC(C2(SC)CC2(C)C)=O)CCOC(C)C1 36273,c1(CC(=O)NCCC(C)N(C(CC(C=C)C)=O)C)cc(Cl)cc2c1OCC2 36274,C(=O)(C(O)C(C)(C)C)N1CCC(n2cc(CNC(C3CC(C)OCC3)=O)nn2)C1 36275,Cn1nnnc1SC(c1nccn1C(F)(F)F)c1ccccc1 36276,c1(CC)c(C(N2CCCCC2CNC(=O)CCc2nncn2C)=O)ccn1C 36277,C1(C)(CC)CC(NC(=O)CNC(C2CCC2)=O)CN1C(=O)C=CC(F)(F)F 36278,C(CCCCC(=O)N(C1CC1)CC1CC(O)CN1C)OCC.C1(C)C(=O)N1 36279,C(=O)(C(C)(C)CCSC)N1CC(O)(CNC(C(CC)C)=O)C1 36280,C1(NC(C(C)NC(C2CCCC2)=O)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1F 36281,N(C1CCCc2ccoc21)C(C1N(C(=O)COC2CC2)CCN(C)C1)=O 36282,C1(CN(C(C2(CC)CC2)=O)C)CN(C(c2snnc2C2CC2)=O)CC12CC2 36283,C(C(C)C(C)C)N(CCC(=O)N(C1CC(NC(C(C)N(C(C)=O)C)=O)C1)C)C 36284,N1(CC=C)CCCN(C(=O)CC2CCCN2C(=O)C2=CCOCC2)CC1 36285,CC1=CCSC1C(=O)NCc1ccsc1C(=O)NCCc1nnc(O)o1 36286,C(=O)(CC1=NNC(=O)C1)NC(C1N(C(c2c(C)cc[nH]c2=N)=O)CCCC1)C 36287,C1(O)(CN(C(=O)CSc2nc[nH]n2)C)CCCN(C(=O)CCC2CC2(F)F)C1 36288,c1(NC2CCCC(CNC(Cc3c(C)cco3)=O)C2)ccc([N+](=O)[O-])cc1C#N 36289,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36290,c1(C(N(CC)CC2CCCN2C(=O)C(F)(F)COC)=O)cc2ncccc2s1 36291,C1(c2cn(C3(OC(C)C)CC3)nn2)CCCN(C(=O)COc2ccccc2Cl)C1 36292,c1(C(N2CCCCC2c2ncc[nH]2)C(=O)NCC2C(COC)C2)cc(Br)ncc1F 36293,c1(CC)cccc2[nH]c(C(N3CCC(CNC(=O)CNC=O)C34CCC4)=O)cc12 36294,CC1=CCC(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)(C)C)C2)=O)CC1 36295,c1(C(N2C3CC(C(=O)NCC4CC(C)OC4=O)(OC3)C2)=O)cc2ccccn2n1 36296,C1(NC(C=C(COCC)C)=O)CC(OC)CN(C(c2cccc(C(F)(F)F)n2)=O)C1 36297,c1(C(C)(C)C)nccc(N2CC(C)(C)C2C2CCN(C(c3cncs3)=O)CC2)n1 36298,C1(NC(COc2ccc(OC)cc2)=O)CCN(C(C2COCC2O)=O)C12CCC2 36299,c1(C(=O)NCCCN(C(c2cccc(CN(C)C)c2)=O)C)coc2ccccc12 36300,N1(C(CCC(C)OC)=O)CCC(C=CC(=O)NCCc2cnco2)CC1 36301,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)F)c2)=O)CC1(C)C 36302,C(CC(C(=O)N(C1CCOCC1C)C)NC(c1ccc(Cl)cc1)=O)OC 36303,C1(NC(c2cccnc2C(F)(F)F)=O)CN(C(c2ccc(F)s2)=O)CC1F 36304,C1(CNC(c2ccsc2)=O)CN(C(=O)CC2CCC3(CCC3)O2)C2(CCC2)C1 36305,C1(C(=O)NCC(C)CNC(C2C3CCN2CC3)=O)CCC(C)(C)CC1 36306,C(=O)(CCCCCCCCC)NCC(CN(C(C1C(=C)CC1)=O)C)(C)C 36307,c1(C(=O)NCC2C3(CCN(C(CC4(C)CC4)=O)CC3)C2)cnc2ncnn2c1O 36308,CCC(C)CC(CO)NC(C1CCN(C(=O)Cn2cnc(C)c2C)C12CC2)=O 36309,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CC1 36310,C1(O)(C(C)N(C(=O)CSC(F)(F)F)C2CC2)CN(C(c2cn(C3CC3)nn2)=O)C1 36311,C1(CNC(c2c(C)scc2)=O)C(C2CC2)CCN1C(c1coc(C(C)C)n1)=O 36312,C1(NC(c2n(C)ccc2)=O)CC2CC1CN(C(=O)C(C1CCS(=O)(=O)CC1)O)C2 36313,CC1CCC(NC(=O)Cc2nccs2)CN1C(=O)Cc1cnn(C(C)(C)C)c1 36314,C(CC)(C(C)N(C(=O)C=CC(F)(F)F)CC)NC(C1(C(=O)OCC)CCO1)=O 36315,C1(CNC(C2CCCS2)=O)CC2(CC2)CN1C(=O)COCC1CCCO1 36316,N1(C(C=Cc2cnc(C)s2)=O)CCCC2C1CCCN2C(=O)C#CC1(C)CC1 36317,CCC(C)(C)CC(=O)NCC1CN(C)CCN1C(c1cc(C(N)=O)ncn1)=O 36318,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36319,C#CCC(CC#C)NC(=O)C(CNC(=O)C=CC1CCOC1)N(C)C 36320,C1(CCC)CC(CC(C(=O)N(CCC(=O)NC(=O)C2CC2)CC2CC2)C)C1 36321,C1(CC)(NC(=O)C(c2ccc(F)c(Cl)c2)C)CCN(C(=O)C2=NNC(=O)C2)CC1 36322,CC(CC(F)F)C(=O)NC1CCC(NC(=O)C(Cc2ccsc2)N(C)C)CC1 36323,N1(C(CCCCC)=O)CC2CCC(C1)C2NC(=O)COC1CCCC1 36324,C1(Cc2n(CC)cnn2)CCCCN1C(N1CCC(C)CC1)=O 36325,C1(NCc2c(C(C)(F)F)nsc2)CCc2nncn2C1 36326,c1(CNC(C(CC)CC)=O)nnc2n1CCN(C(C1(C(F)F)CCCC1)=O)C2 36327,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(c2cnn(-c3nccs3)c2)=O)C1 36328,N1(C(C(CC2CN(C(C(CCN(C)C)O)=O)C2)F)=O)CC2(C1)CC(C)(F)C2 36329,N1(C(CC)=O)CCC2(CC1)C(C(=O)N(c1ccccc1COC)C)CCS2(=O)=O 36330,C1(NC(=O)Cn2cnnn2)CCCCC1NC(c1coc(Br)c1)=O 36331,CCCC(C(=O)N1CC(CNC(c2coc(Cl)n2)=O)(COC)C1)C(C)C 36332,C1(NC(=O)CC2CCCCC2)CC(F)CN(C(=O)C(F)F)C1 36333,C1(OC2CN(C(c3c(CCC)nns3)=O)C2)CCN(C(c2ncoc2C)=O)CC1 36334,N(C(=NCCC(=O)NC)NCC1CCCCC1O)C(CC)C 36335,C(CCN=c1cc(C)nc(CO)[nH]1)N1CCN(C(c2ccc(OC)cc2)=O)CC1 36336,C1(NC(c2cscc2C2CC2)=O)CC2CCC(C1)N2C(c1ccns1)=O 36337,N1(C(C(=O)NCC)=O)CCC2(CC1)COC(CNC(c1c(Cl)nn(C)c1C)=O)C2 36338,Cc1c(Cl)ccc(C(=O)N(C2CCCN(C(c3cccc(=O)n3C)=O)C2)C)c1O 36339,C1(C(=O)OC)CCN(C(C2CN(C(c3ncc(N)cc3Cl)=O)CC2(C)C)=O)C(C)C1 36340,Cc1nc(Cl)nc(N2CC3CCC2CN3C(=O)Cc2ccn(C)n2)c1F 36341,C(=O)(C(C)(C)C1=CCN(C(=O)COCCCC(C)C)C1)N1CCCC(C#C)C1 36342,Cc1nnccc1CN(C)Cc1cccnc1N1CCN(C)CC1 36343,c1(C(=O)OC)nnc(C(C)NC(=O)OCc2nnc(C)o2)s1 36344,n1(CCOC)nnnc1C(c1cncs1)Nc1cnn(C(C)C)c1 36345,CC1CN(C(c2scnc2C(F)(F)F)=O)CCN1C(C1CC2(CCOC2)C1)=O 36346,c1(OC)cc(C)c(-c2ccc(C(=O)Nc3cccc(F)n3)nc2)cc1C 36347,c1(C(N2CCC(C)(C3OCCO3)CC2)C(=O)NC(C)C)cc(S(N)(=O)=O)cs1 36348,Cc1ccc2c(C(=O)NCC(C)NC(C3CCN4CCOCC34)=O)ccnc2c1 36349,c1(Cn2c(NC(N3CC(CS(C)(=O)=O)C3)=O)ccn2)ccc(Br)cc1F 36350,CC1CCC(=CC(=O)N(CCCNC(=O)C=Cc2cccs2)C2CC2)CC1 36351,C1(CN(C)C(c2c[nH]nc2C2CCOC2)=O)CCN(C(C2(C(N)=O)CC2)=O)C1 36352,C1(C(N(C2CCN(C(c3coc(Cl)n3)=O)C2)C)=O)COC(=O)N1 36353,c1(C(N(CCN(C(=O)Cn2ccc(C)n2)CC)CC)=O)ccnc(F)c1OC 36354,c1(C(N(C)CC2CCN(C(C3(C(=O)OC)CC3)=O)C2)=O)cc(N(C)C)cnc1OC 36355,N#Cc1c(C(=O)NCCN2CCN(C(c3n[nH]c4c3COC4)=O)CC2)cccc1F 36356,N1(C(C(C)NC2CCCCC2)=O)CCCC(C)C1C(=O)C(C)(C)F 36357,C1(n2cc(C(C)(C)SCC)nn2)CN(C(c2nc(C)n(C)n2)=O)CC1O 36358,c1(OCC)ccccc1C(c1cccc(Cl)c1)NC(C)C(=O)OC(C)(C)C 36359,c1(CNC2CCC(C(=O)NCc3ccc(C)o3)CC2)cccc2cnccc12 36360,Cc1cc(NC(c2cc(CCNC(=O)CSCC(F)F)on2)=O)cc(C#N)c1 36361,N1(C(Cn2cc(CNC(C=Cc3occ(C)n3)=O)nn2)=O)CCCC(O)(CO)C1 36362,N1(C(c2c(CC)ocn2)=O)CCCC(C)C1CNC(=O)Cn1nc(C)n(C)c1=O 36363,C1(C(N2CCN(C(=O)C=Cc3ccccn3)C(C3CC3)C2)=O)CC2CCC1CC2 36364,C(CN=C(NCc1cc(C)ccn1)NCc1cc(O)cc(O)c1)N(CC)CC 36365,c1(C(C(=O)NCC2(C(=O)NCC(C)Cn3cccn3)CCC2)=O)cccn1C 36366,c1(CN(C(=O)COC(C)(C)CNC(=O)CC2COC(=O)C2)C)c(Cl)cnn1C 36367,c1(C(=O)NC2C(CNC(=O)COCC3CCCO3)CC2)cc(Br)ccn1 36368,C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2CCC(=O)N2C2CC2)=O)C1 36369,C1(C(=O)NC2CCC(NC(c3ccncc3O)=O)C2)CCCC1(F)F 36370,Cc1nn(C2CC2)cc1C(=O)NCC(C1CC1)NC(=O)CNc1ccccn1 36371,N12CC3CCN(CC13)C(=O)c1cc(on1)CC2=O.C1(N(C)C)CC(CN(C)C)C1 36372,c1(C(=O)NC(CC)CNC(=O)C(C)(CC)C(F)F)ccnc2ccc(Cl)cc12 36373,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2cccc3nonc23)C(C)C1 36374,C(CCC(N)=O)(C(=O)NCCC1CN(C(=O)CCN2CCCCCC2)C1)N(C)C 36375,C(C(C(=O)Nc1ccccc1OC(c1ncc(C)s1)C)C(C)C)OCC 36376,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2cc(O)no2)=O)C1 36377,c1(CC)nc(C)c(C(N2CC(C(=O)NC(C)(CO)C3CC3)(CC)C2)=O)o1 36378,C1(C(=O)CC2(CC3CC3)CC2)CCCN(C(=O)C(=O)COC(C)=O)C1C 36379,N1(C(c2c(NCC)scn2)=O)CC2CCCC(NC(C3OCCC3(C)C)=O)C2C1 36380,c1(C(=O)NCC2C(NC(COC(C)C)=O)COC2)c(F)cccc1[N+](=O)[O-] 36381,N1(C(c2c(OC)n(C)nc2)=O)CCN(C(c2cc(O)cs2)=O)CC1C 36382,c1(C(N2CCC(c3c(NC(=O)OC(C)(C)C)c[nH]n3)C2)=O)cc(C)n(C)c(=O)c1 36383,C(=O)(C(C)(O)CC(C)C)NC1C(CCC)CN(C(=O)CCS(=O)(=O)NC)C1 36384,C(=O)(C#CC1CCOCC1)NC1CCC(CC(=O)NCC(C)O)CC1 36385,C(CC(C)C)(C(=O)N(CC(=O)NCC1CCC(C)(C)CO1)C)NC(C)=O 36386,C1(CN(C(=O)Cc2cn(C)nn2)C)COCCN1C(=O)CN1CSCC1=O 36387,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1(C)Br)=O 36388,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36389,CCC(C)C(O)C(=O)NCC1CCCN(C(c2ccn(C)c2C)=O)C1 36390,C1(C(c2n(CCSC)nnn2)NCCc2ccncc2)CC2CCC1CC2 36391,c1(OC)ccc(C)cc1CNCC(O)CNC1(C#N)CCCC1 36392,Cc1ccc(S(=O)(=O)Nc2cc(C)cnc2OC(F)F)c(F)c1 36393,N1(CC(=O)N(c2ncccn2)C)CC2C3CCC(C2C1)N(C(C1CCC1)=O)C3 36394,c1(C(N2C(CN(C(c3cnc(C)[nH]3)=O)C)CCCC2)=O)ccc2nc(O)cn2c1 36395,C1(CC(=O)NCCC(C)(C)NC(CC(C)SC)=O)CCOC(C)(C)C1 36396,C1(NC(C(C)NS(CCC)(=O)=O)=O)CCC(C)(CNC(C2(CO)CC2)=O)CC1 36397,C1(C#CC(=O)NC(CNC(=O)C=C(C)c2cccnc2)C(C)(C)C)(CC)COC1 36398,C12(C(N3C(C(C)NC(C4(COCC)CC4)=O)CCC3)=O)CCC(CO)C1CC2 36399,c1(C(N(C(C(C)O)(C)C2CCOCC2)C)C)ccc(Br)cc1OC(F)F 36400,N1(C(C=CCCC)=O)CCC(CC(F)(F)F)C(NC(c2cc(C)nn2C)=O)C1 36401,C(=O)(NNC(=O)C1CC(Cl)=NO1)NC(CCC)c1cccs1 36402,Cn1c(F)nc(Cl)c1N1CCCC(CN2CCCCC2COCC(F)(F)F)C1 36403,CC(C)C(O)C(=O)N1CCSCC1CCNc1cc(Oc2ccccc2)ncn1 36404,c12ccc(C)c(c1)COC(=O)C(C)CS2.C1(N(C)CC)CCCOC1 36405,CC1CCc2nc(NCCNC(=O)OC(C)(C)C)ccc2C1 36406,C1(C(=O)O)(NC(=O)NCc2onc(-c3c(C)cccc3)n2)CC2CCC1C2 36407,Cc1ccc(F)cc1CC(=O)NCC(C)N(C)C(C1CC2(CCC2)CO1)=O 36408,n1(C(C)C)nccc1CNC(=O)CC1CCCN1C(C1CCOCC1)=O 36409,c1(C(N2CCC(NC(c3ccc(S(C)(=O)=O)s3)=O)C2)=O)cccc2nc(Cl)cn12 36410,C(=O)(N=c1[nH]nc(C2CC2)s1)N(C)CCc1c(OC(C)(C)C)cccc1 36411,C1(COC)(NC(=O)Cn2cnc([N+](=O)[O-])c2)CCN(C(C2(C)CCCO2)=O)CC1 36412,Cc1nc(F)ccc1CNC(C1CCN(C(=O)C2CC3CCCC3C2)O1)=O 36413,CCCCCC(O)CC(=O)N(CCCNC(=O)CC=Cc1ccccc1F)CC 36414,N1(C(CC=CC)=O)CC(NC(=O)C=Cc2ccoc2)CC(F)(F)C1 36415,CCCCCCCCC(C)C(=O)NC(C1CCN(C(C2(C)CCC(=O)C2)=O)C1)C 36416,N1(C(c2ccc(Cl)s2)=O)CC(=O)N2CCOCC2(CNC(C2(O)CCOC2)=O)C1 36417,N1(C(CC2(OCC)CC2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccc(F)cc1 36418,c1(C(C)NC(N2CCC(N(C)C(=O)OC(C)(C)C#N)C2)=O)cn2ncsc2n1 36419,C1(CC(N2CC(OC(=O)OC)C2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)C1 36420,c1(N2CC(C(=O)NCc3cc(C)nn3C)C(F)(F)CC2)ncnc2scc(C)c12 36421,c1(N2CCCC(CCNC(C3C(C)CC(C)O3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 36422,C1(C(=O)OCC(C)C(=O)N(CCCCN(CCCCl)C)C)COCCN1C 36423,N1(C(c2ccn(C)c2)=O)CCC(C(C)(C)CNC(=O)Cc2ccncc2F)CC1 36424,CC(C)C(C)CC(=O)NCC1CC(C(=O)NCC2(F)CCCC2)CO1 36425,C1(NC(c2ccc(OC)c(I)n2)=O)CCc2ncc(Br)n2C1 36426,c1(C(N(C)CC2CN(C(c3c(CC)nccn3)=O)C2)=O)cc2c(=O)[nH]ccn2c1 36427,n1(CC)cnc(C(=O)NC(CO)C(C)NC(C2CN(C3CCOC3)C2)=O)c1 36428,C(=O)(C(C(C)C)C(C)C)NCCC1N(C(Cc2cc(C)c(O)cc2)=O)CCOC1 36429,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36430,CN=c1[nH]cc(C(N2CC(CCCC(=O)NCC3(C(N)=O)CCCO3)C2)=O)o1 36431,C(c1ccc(F)cc1F)=CC(=O)NC1C2CN(C(CC=CC=C)=O)CC1C2 36432,C1(N(CCCC)C(=O)C=Cc2cscn2)CCN(C(c2cc(C)cs2)=O)CC1 36433,c1(OCC(=O)NCCc2ccc(-n3cncn3)cc2)ccc(Cl)cc1[N+](=O)[O-] 36434,C1(N(C(c2c(OC)nsc2)=O)CCO)CCN(C(C2CC(C)(C)CC=N2)=O)CC1 36435,N1(Cc2ccc(CCOCC)o2)C2CCC1CN(CC#N)C2 36436,C1(C2CCOCC2)(NC(CC2CC(NC(C(C)n3cncn3)=O)C2)=O)CC1 36437,C1(CNC(c2scc(CNC(C(CC=CCC)C)=O)n2)=O)OC(=O)CC1(C)C 36438,Cc1cc(C)c(C(=O)NC(C)CNC(C2(O)CC2(C)C)=O)c(=O)o1 36439,C(=O)(C1=CC2(CN(C(=O)Cn3cnnc3O)C2)OC1)N(C)CC1(CO)CCC1 36440,C1(CCC(=O)NC(CNC(CCC=CC)=O)C)CCCC(O)C1 36441,C1C(F)(F)Cn2cc(nn2)C1.C1(C(N2CC(N3CCC3)C2)=O)CC(C(=O)O)C1 36442,C1(CC(=O)NCCC(CC)CO)CCN(C(C2OC3CCC2C3)=O)C1(C)C 36443,c1(C(=O)NCC(C)CNC(c2cccc(I)c2)=O)ccc2cnccc2c1 36444,c1(C(C)C)cccc(OCC(=O)NCCCCC(C)NC(=O)C=CCO)c1 36445,c1(NC(c2c(-c3ccc(C(C)(C)C)cc3)ncs2)=O)cc(Cl)cnc1O 36446,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36447,C(=O)(C1=CCCCO1)NCCCCN(C)C(C1CC1(C)C(F)F)=O 36448,CCCCCCC(=O)NC1CC(CNC(=O)C(CC(F)F)NC(=O)OC(C)(C)C)C1 36449,c1(C(N2CC(O)(CNC(CN3CC(CC)C3)=O)C2)=O)sc(C)nc1C 36450,N1(C(CC2(OC)CCC2)=O)CCN(C(c2ncnc(C)c2C)=O)CC(C)C1 36451,c1(C(N2CC(CN(C(C(CC)SC)=O)C)OCC2)=O)c(C)ccc(OC)c1N 36452,c1(N(C)CCC2CCCCC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)COC2 36453,CCC(C)C(=O)NCC(=O)NCC1CC(NC(C2(C3CC3)CCCO2)=O)C1 36454,N1(C(CC=C)=O)C2CCC1C(C(=O)NCc1c(C)cccc1Br)C2 36455,CC1(NC(c2c[nH]nc2-c2ccn[nH]2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 36456,C1(C(=O)Nc2cccc(CNC(CC3(COC)CC3)=O)c2)CC(C)(C)C1C(C)C 36457,N1(C(c2n(C=C)nnc2)=O)CCC2CCCC12C(N1CC(OC)CC2(CC2)C1)=O 36458,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)NS(=O)(=O)CC)C(C)C1 36459,C(=O)(C1=C(F)CN(C(=O)C(C)N(C)C)CC1)Nc1ccc(C)c(CO)c1 36460,C(CC(CC(=O)NC12CC(C1)C2)Nc1ccccc1)NC(=O)CCn1ccnn1 36461,N1(CC(=O)NCc2c(OC)cncc2)C(=O)NC(C)(c2ccc(F)cc2C)C1=O 36462,c1(-c2c(C(N3CC(CC(C)(C)C)C3)=O)c[nH]n2)ccc2c(c1)CCCO2 36463,c1(C(N2CCC(N(C(c3c(C)nccc3)=O)C)C2)=O)ccc(C(F)(F)F)c(Cl)c1 36464,c1(C2C(=O)NN2C2CC2)ccc(Br)c(OC(F)F)c1F.C(COC)NCCO.C(C)C.O 36465,C1(NC(C2C(CC)CCN2C(C2CC3CC(=O)C2C3)=O)=O)CC(C)OC(C)C1 36466,C(=O)(C#CC1CCCCC1)NC1CC2CN(C(C(CCCOC)C)=O)CC21 36467,C1(CC)CNC(=O)CN1C(=O)CC=CCNC(C1(CC(=O)OC)CC1)=O 36468,C1(C(=O)NC(C)CNC(C2(CC3CCCC3)CCCC2)=O)CC2C=CC1C2 36469,c1(C(=O)NC2CCC(C)(CNC(=O)C(Cl)=CCl)C2)cccn2cncc12 36470,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C)CC3C)=O)CC12)=O 36471,c1(C(=O)NCC2(C(N(CC(C)O)C)=O)CCCC2)nccc2cc[nH]c12 36472,CCCCC(F)F.C(=O)(C(CCC1CCCOC1)NC(=O)OC)OC(C)(C)C 36473,N1(C(CC(C)OC)=O)CCC(NC(=O)CCC(C)OC)C1(C)C 36474,C1(CCC(N2CCN(C(C=CCC)=O)C(C)C2)=O)CCc2ccccc2C1=O 36475,C(c1ccc(C)cc1C)=CC(=O)NC1CCCC(CNC(CN(C)CC)=O)C1 36476,Cc1ncccc1COC(c1ccc(-c2ccc(N(C)C)cc2)cc1)=O 36477,C=CCC1CN(C2CCCC2)C1=O.c1(COC(C(=O)NCC)C)ccccc1 36478,N1(C(C(C)SCC)=O)CCC(CNC(c2cnccn2)C2CCCC2)C12CCC2 36479,N1(C(c2cc(CC)nc(O)c2)=O)CC2CCC(NC(=O)C3=C(C)OCCC3)C2C1 36480,c1(C(N2C(C)(C(N3C(CC)(CC)CC3)=O)CC(O)C2)=O)nccc2[nH]ccc12 36481,C(CNC(=O)Cc1ccccc1)(C(C)(C)C)NC(CCN(C)CCO)=O 36482,C1(C(=O)NC(C)CN2CCCC2)CCC(O)CN1C(c1cc(C(N)=O)[nH]n1)=O 36483,N(C1=NCC2C(N1)C2)CC(c1ccc(C)cc1)OC.C1(SC)CCC1 36484,c1(NS(C)(=O)=O)ccnc(C(=O)NCC(C2CC2)NC(c2cncc(F)n2)=O)n1 36485,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cn(C(C)C)nn2)=O)C1 36486,CC1CC2(CCN(CCNC(C3CC3C(F)(F)F)=O)CC2)C(=O)N1 36487,c1(NC(=O)CC2CN(CCCNS(=O)(=O)NCCO)C2)cccnc1N1CCCC1 36488,N1(C(C(C)NC(C(CC)C)=O)=O)CCC2(CC1)CC(NC(=O)CC(C)O)C2 36489,c1(C(=O)N)cc(CC)[nH]n1.C(=O)(C(CC)OCC)N(CCCN)CCC 36490,N1(C(C(Cc2cccs2)NC(=O)OC)=O)CCC(F)(F)C(C(=O)NC2(F)CC2)C1 36491,C1(NC(c2ccnc(F)c2Cl)=O)CC2CC1CN2C(=O)Cc1cccnc1 36492,C#CCCCCCC(=O)N(CC(C)C(=O)N1CCC1(C)C(=O)OC)C 36493,C1(=O)CC(C2CCC2)CN1.CCC(C)C(=O)NCC.c12cc(cs1)NC2=O 36494,C(=O)(C(C)(C)CCCF)NCC(C(=O)NCc1c(C)cc(O)cc1)CC1CC1 36495,N1(C(CCOCC(C)(C)C)=O)CCCC(F)(C(=O)NCC23CCCC2CCC3)C1 36496,C1(C2(C)CC2)COCCN1C(=O)NC1CC2(C1)CC2C(N)=O 36497,CC1CN(C(=O)Cc2coc3cc(Cl)ccc23)CC2(CCN(C(=O)C3CC3)C2)O1 36498,c1(C(=O)NC(C2OCCN(C(Cc3c(C)nn(C)c3)=O)C2)C)cc(Cl)cc(Cl)c1 36499,CC(=O)C(C)(C)CC(=O)NC1C(c2ccccc2)(C(F)(F)F)C1 36500,C(C)(CCC(=O)N1CCCCC1C1(NC(c2ocnc2C(F)F)=O)CC1)SC 36501,N1(C(c2ccc(SC)cc2)=O)CCC(CNC(=O)Cc2cnc[nH]2)C12CC2 36502,C1(C(C)C)CCC(C(=O)N(C)Cc2cn[nH]c2)N1C(c1cnnn1C)=O 36503,C1(CNC(CC(C)SC)=O)CN(C(c2ccc(Cl)c(C)c2N)=O)CC12CCC2 36504,C(=O)(CCCCCNC(C1CC(CC2CC2)C1)=O)N(CCOCC#C)C 36505,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(C(F)(F)F)c1)CC 36506,c1(C2CC2)ccncc1NC(=O)CCN(C(c1cc(CCO)on1)=O)CC 36507,c1(CC)ccc(F)c(C(=O)NCC2CC(F)CN2C(C2CCCC(=O)N2)=O)c1F 36508,C1(CNC(c2c(C)cncc2)=O)COC(C)(C)CN1C(c1cc(Cl)c[nH]1)=O 36509,N1(C(CSCC(C)C)=O)CC2CC1CN(C(c1cc(C3CCCN3C)[nH]n1)=O)C2 36510,C1(NC(CCCC=C)=O)C2CCC1N(C(C1(CC=C)CC1)=O)C2 36511,C1(C2CC2)(C(=O)NCC(c2ccccc2)CNC(C)=O)CC1 36512,CCCC(C)CC(=O)NCCCC(O)C(=O)NC(c1cnccc1C)C 36513,C(CCCCCC(=O)N1CC2(CO)CC2(CO)C1)NC(Cc1c(CC)n[nH]c1)=O 36514,c1(C(=O)NCC(C(C)C)NC(c2occc2Br)=O)ccc2cccnc2n1 36515,Cc1c(NCC(N2CCOCC2)(C)C)nc[nH]c1=NCC1(C)CC1(Cl)Cl 36516,N1(C(C=CC)=O)CCC(CNC(=O)CC2CCNC2=O)C1C(C)(C)C 36517,c1(OC)ccc(CC(N2CCCN(C(C3CC4(C3)CC4F)=O)CC2)=O)c(C)c1 36518,C1(C)(COC(C(C(C)C)n2cncn2)=O)CCCN(C(=O)OC(C)(C)C)C1 36519,c1(NCCCCC(N)=O)[nH]c(=NCCCC2CCCCC2)nc2scnc12 36520,c1(C(=O)NC(CCC)CNC(c2cnc(C)s2)=O)c(OC)nsc1OC 36521,C#CCCCC(C)C(=O)N1CCOC(C(=O)NCCCc2n[nH]c(C)n2)C1 36522,C1(C(=O)Nc2cc(OC)ncc2Cl)CC12CCN(C(C1COCCO1)=O)CC2 36523,CCS(=O)(=O)CCN=c1[nH]c(N2CC3CCCCC23)nc2c1CCC2 36524,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36525,C1(O)(CNC(C2C(OCC)C2)=O)CCN(C(=O)C(c2cccc(O)c2)(C)C)C1 36526,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(c2n(CCC)ccc2)=O)CC1O 36527,CC1CC(C(=O)NC2(CCNC(=O)Cc3ccc(Br)nc3)CCCC2)=NO1 36528,C(=O)(C1CCS(=O)(=O)c2ccccc21)N(CC(C)C)CC(C)NOCC(=O)NC.N 36529,c1(C(N(CC(C)CNC(=O)CSC2CC2)C)=O)c[nH]c2ccc(Cl)cc12 36530,N1(C(c2c(CC)c[nH]c2)=O)CCC(CNC(C2CCC(=C)CC2)=O)C(C)C1 36531,CC(CCCCNC(c1cnn(C2CC2(F)F)c1)=O)NC(C1CCCCC1O)=O 36532,c1(-n2c(C(N3CCC(N(C)C(c4sccc4Cl)=O)C3)=O)ccc2)ccccc1Cl 36533,c1(CNC(c2cc(C)ns2)=O)nc(C)c(C(=O)N(CCF)C2CC2)o1 36534,CC1=NOC(C)(C(=O)NC(CO)C(=O)NCCn2nc(C)nc2C)C1 36535,C(C1=CCSC1)N(C)C(C1(F)CN(C(c2ccccn2)=O)C1)=O 36536,C(CCC(=O)NNC(=O)Nc1ccc(C(=O)NC2CC2)cc1)OC(C)C 36537,C(c1c(C)noc1C)=CC(N1CCC(N(C(C2CCCN2C=O)=O)CC)C1)=O 36538,N1(C(COC(CC)(C)C)=O)CCN(C2CCN(C(=O)Cc3csnn3)C2)CC1 36539,N1(C(CN2CCCC(C(=O)NC)C2)=O)CCCN(C(C2CCSC2)=O)CCC1 36540,Cc1cc(C(N2CCCCC2CNC(=O)C2=NOC(C)C2)=O)cc(C(F)F)c1 36541,N1(C(C2(SC)CN(C(=O)C(C3CCOCC3)O)C2)=O)CC(C#N)(CCF)C1 36542,CC(CN=[N+]=[N-])N(C(C1(NC(=O)CCN)CCC1)=O)C 36543,C12(C(N(C)OCc3ccccc3)=O)CC(C)(CN1C(=O)CCc1ccccc1)C2 36544,Cc1ccc(C(c2nnnn2Cc2nnn(C)n2)NCC=CCl)c(F)c1 36545,c1(OC)ccc(NC(C2CC3(CC3)CN2S(=O)(=O)CC#N)=O)c([N+](=O)[O-])c1 36546,C1(CNC(c2c(C)coc2)=O)CN(C)CCN1C(c1ccncc1NC(N)=O)=O 36547,N1(C(c2n(CCC)ccc2)=O)CC2CC(C1)CN(C(C1CC1C(C)(C)C)=O)C2 36548,CC(C)(CCCO)C(=O)NC1CCCCC1NC(c1c[nH]nc1[N+](=O)[O-])=O 36549,C(=O)(C(CNC(C1(C)CC(F)(F)C1)=O)CC=C)N(CC#C)CCOC 36550,Cc1nc(NC2(CO)CCN(C(=O)C(O)Cc3cnc[nH]3)CC2)c2cc[nH]c2n1 36551,c1(CC)ccc(F)cc1C(=O)N(CCNC(c1nn(C)cc1Cl)=O)CC1CC1 36552,N1(C(C(C(C)C)OCC)=O)CC(NC(c2cnn(C)c2N)=O)CC12CCOCC2 36553,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36554,N1(C(C(=O)NC)=O)CCC(CC(C)(C)NC(=O)CCc2ccc(CO)cc2)CC1 36555,C(=O)(CC(C)c1ccco1)N(CCCOC)CCO 36556,C=C(CNC(=O)CN1CC(C)C1)CCNC(c1csnc1OC)=O 36557,C1(NC(CC(C)C2CCCO2)=O)CCCCN(C(c2ccn(O)c(=O)c2)=O)C1 36558,Nc1ccnc2c(C(=O)NC(C(=O)NC3CCOC(CSC)C3)C3CC3)cnn12 36559,C1(OC)CCC(CC(=O)NC2CCN(C(c3ccn(C)c3)=O)C2C(C)C)CC1 36560,c1(CC(N2CCOCCC2C2CC2)C(=O)OC)ccc(S(=O)(=O)C(C)(C)C)cc1 36561,c1(C(N2CC(CCNC(c3scc(OC)c3)=O)(OC)C2)=O)cnc(N)c(Cl)c1 36562,N1(C(c2c(CCCC)ocn2)=O)CCN(C(=O)Cc2ccns2)CC1CCC 36563,C(C(C)(C)C(=O)N1CCCC1CC(C1C(C)C1C)=O)N(C(CNC(=O)OC)=O)C 36564,Cc1c(C(=O)NCC2CCCN2C(=O)Cc2cn(C)nc2Cl)sc2nccn12 36565,c1(C(N2C(COC)CN(C(c3nc(Cl)ccc3N)=O)CC2)=O)cc(C)cc(C)c1O 36566,O(C=CC(=O)N1CCCC1C1CCN(C(=O)C(F)CN(CC)CC)C1)CC 36567,c1(C(=O)NCC2(O)CCN(C(CC)=O)C2)ccc(C#N)cc1C 36568,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36569,CN=c1[nH]cc(C(=O)NCC2CCCN(C(c3[nH]nnc3C3CC3)=O)C2)o1 36570,c1(SC)ncc(C)c(N2CCCC(C(C)(C)O)C2)n1.N12CCCC(C1)C2 36571,c12n[nH]cc1C(=O)NCC2.N1(C(COCC#C)=O)CCC(OCC=C)C1 36572,C1(CC(C)C)C(=O)N2CCC(C)C(C2)C(=O)NO1.C(C=O)N(CCOC)C 36573,C=CCC(C(=O)N(C(C)CNC(=O)C(C)N(C)C)C)NC(C)=O 36574,N1(C(C2CC2(Cl)Cl)=O)CC2(CCN2C(c2cc(-c3ccoc3)on2)=O)C1 36575,C1(C(N2CC(CNC(c3cccc(SC)c3)=O)C(C)C2)=O)CCC2(CCC2)CO1 36576,CCCC(CCNC(=O)C(C)(C1CC1)N(C(=O)COCCF)C)C1CC1 36577,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CC2CCC(C)O2)CC1 36578,Cc1nn(C(C)CN)c(C)c1C(=O)N(c1ncncc1Cl)CCC1CCNCC1 36579,CC(CC(F)F)C(=O)NCCC1CCCCN1C(=O)C(O)Cc1cnc[nH]1 36580,N1(C(C2CC(=O)NC(=O)N2)=O)CCC(CNC(=O)Cn2cc(Cl)cn2)C(F)(F)C1 36581,c1(CNCC(=O)N(CC(C)(C)NC(=O)CCC2CCCOC2)C)ccnc(O)c1 36582,C1(C(=O)NC2C(NC(c3ccc(C(=O)OC)cn3)=O)C2)CCc2nc[nH]c2C1 36583,N1(C(C2CC(=O)NC2)=O)CC2(C1)CN(Cc1cc(Cl)ccn1)C2 36584,N1(C(C2(C)C=CCCC2)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(CO)C1 36585,c1(C(C(c2nnnn2CCCF)NCC(C(C)C)OC)(C)C)ccc(F)cc1 36586,CC1(CO)CC2(CCN2C(C2C=CCCN2C(c2cc[nH]n2)=O)=O)C1 36587,C1(NCC(=O)Nc2ccncc2)CC2CCC1N2C(=O)CC1CCC(F)(F)CC1 36588,N1(C(C2(C)CC(=O)C2)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36589,N1(C(CC(CC)SC)=O)CC2CCC(C1)N2C(=O)C(C)C(=O)OC 36590,N1(C(=O)NCc2cc(F)c(C(C)C)c(Br)c2)CCN(S(=O)(=O)N(C)C)CC1 36591,N1(C(C(CC)N(C)C)=O)CC=C(CCNC(C2CN3CCN2CC3C)=O)CC1 36592,c1(C(=O)NC(C)C(CO)NC(C2(O)CCCCCC2)=O)cn2ccc(F)cc2n1 36593,C1(C(=O)NC(C2N(C(CC3(CC)CCOCC3)=O)CCC2)C)CCC(C)(C)CC1 36594,C1(C(C)C)CCN(C(=O)C(n2cc(CN3CCSCC3)nn2)C)C1 36595,CC(C)CC(C)CC(=O)NCCCCN(C)C(c1nncn1C1CC1)=O 36596,N1(C(C(C)Cc2ccncc2)=O)CC2(CC(NC(C3CC34CCOC4)=O)C2)C1 36597,C1(C)(CNC(C(CCC)O)=O)CCCN(C(c2nn(C)c(N)c2C)=O)C1 36598,c12ccc(cn1)S(=O)(=O)N2.C(C(C)(C)CN1CCC(CS(C)(=O)=O)C1)N(C)C 36599,N1(CCCNC(C2CCC(C)C2)=O)CCN(C(C2CCSCC2)=O)CC1 36600,c1(C(N(C)CC2N(c3cc(C)ncn3)CCOC2)=O)cnc(F)c(F)c1 36601,c1(C(N2CC3CN(Cc4c(OC)c(Cl)ccc4)C3C2)=O)ccc2c(C)[nH]nc2c1 36602,c1(OC)cc(C2CC2)ccc1CN(c1cnc(C(F)(F)F)[nH]c1=O)C 36603,C1(CC)CCC(CNC(=O)C=CC(C)(C)NC(=O)CCc2ccn(C)c2)CC1 36604,C1(CNC(c2c(CC)con2)=O)CN(C(=O)C(C#N)C(C)C)CCCO1 36605,C1(NC(C(C)SCC)=O)CC(OC)CN(C(c2cc(C)nc(C)n2)=O)C1 36606,c1(C(=O)NCC2(F)CCC(NC(C3CCCC3F)=O)C2)n[nH]c2cccnc12 36607,N1(C(CCCCCOC)=O)CC2CCCN(C(=O)CCC(C)(C)C)C(C2)C1 36608,C1(NC(c2cnc(C)nc2)=O)CC2CC1N(C(=O)C(C(C)(C)C)n1ccnn1)C2 36609,C1(C(=O)NCC(=O)N(C)OC(C(C)C)=O)CCC(SCc2ccccc2)O1 36610,N1(C(C(F)OC)=O)CC2(CCC(CNC(c3ccc[nH]3)=O)O2)C1 36611,c1(OC)ncc(Cl)cc1C(N1CCC(C)C(N(C(=O)CC23CC(C2)C3)C)C1)=O 36612,CC(C)CC(F)(F)C(=O)NC1CN(C(c2nc(C(F)(F)F)cn2C)=O)CC2(CC2)C1 36613,C(=O)(CC(C)CC(=O)NCCC(C)NC(c1ncc2ccccn12)=O)OC 36614,N1(C(c2cc(C)oc2C)=O)CCCC(NC(=O)C(c2c(F)cccc2F)C)C1C 36615,N1(C(C(C=C)(C)C)=O)CCCC2(C1)C(=O)N2C.C1(C#N)(COC)CCC1 36616,c1(C(N(C2CCN(C(c3c[nH]nc3SC)=O)C2)CC)=O)cn2ccc(C)cc2n1 36617,C1(C(N2C(CNC(CCOCC)=O)CC(COC)C2)=O)CC(CO)C12CCC2 36618,C1(C(=O)NC(c2nccs2)C)CCCC12CCN(C(c1ccc[nH]1)=O)C2 36619,c1(C(N2CC(C)C(CNC(c3cn[nH]c3)=O)C2)=O)nc(Br)c2ccccn12 36620,N1(C(C)=O)CCN(C(C2COC(=O)N2C)=O)C(c2cccc(Cl)c2)C1 36621,Cc1ccc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(C)C(N)=O)c(C)c1Br 36622,c1(-c2nn(-c3ccc(C)cc3)c(-c3c[nH]nc3F)n2)ccc(C(F)(F)F)c(F)c1 36623,C(=O)(C(F)CC1CN(C(C2(C)COC2)=O)C1)N(CC)Cc1ccccc1 36624,C12(CNC(Cc3cc(OC)c(C)cc3)=O)COCCN1C(=O)CN(C(=O)C1CC1)C2 36625,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36626,CC1CN(C(=O)Cc2ccccc2)CCC1NC(c1ccnc(O)c1)=O 36627,N1(C(C(c2ccnn2C)C)=O)CCC=CC1C(N1CCC1C(C)O)=O 36628,C1(NC(CCC#C)=O)CC2CC1CN(C(c1cc(C(F)F)no1)=O)C2 36629,c1(CC(=O)NS(Cc2cccc(NC)c2)(=O)=O)ccc2c(c1)Cc1ccccc1-2 36630,c1(C(N2CC3CCC2CN3C(C2CC(O)C2)=O)=O)cc2oc(Br)cc2[nH]1 36631,CCC(C)CC(=O)N1CCC(C(=O)NC2CCCC2c2ccccc2Cl)CC1 36632,c1(C(CC)N(c2cc(C)nc(C)n2)C(=O)CC2CCC2)c[nH]c2cc(F)ccc12 36633,c1(SCCCC(=O)NCC(CC=C)NC(=O)C(CSC)OCC)ccc(O)cc1 36634,c1(C(C(=O)NCCC#N)N(C)CC2CC(=C)C2)cc2sccc2s1 36635,N1(C(C(CC)(C)NC(C2CN(c3ncco3)C2)=O)=O)CC2(CC(CO)CO2)C1 36636,S(=O)(=O)(c1cnc(NCC2(C)CC2)c(Cl)c1)N1CCCC(CC)C1 36637,CC1(C)CN(C(C2CCN(C(C3CC(O)C3)=O)C2)=O)CC1O 36638,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36639,c1(SC)ncc(C(=O)NC(C)CNC(=O)C(C(C)C)SC)cn1 36640,c1(CCC(=O)NC(CNC(C(CSC)O)=O)C(C)(C)C)ccccc1[N+](=O)[O-] 36641,c1(CC(=O)NC(CNC(c2c(C)n[nH]c2)=O)(C)C)cccc(OC(F)(F)F)c1 36642,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC(C)(O)C2)=O)C12CC2 36643,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36644,N(C(=NCC1CCC1)N1Cc2ccccc2C2(CC2)C1)Cc1cc(CC)ncc1 36645,N1(C(Cc2cncc(C)c2)=O)CC2CC3CC2C1C3NC(C12CCCC1C2)=O 36646,c1(C(=O)NCCCC(C)NC(CCCCC)=O)ccccc1C#N 36647,CC1CN(Cc2ccc(=O)n(C)c2)CCCN1C(c1ccc(F)nc1C)=O 36648,c1(NCC2CCCN(C(Cn3cc[n+](C)c3)=O)C2)ncc(C#N)cc1F 36649,N1(C(c2sc(C(F)F)nc2Br)C(=O)NCCCC)CC2(CCC2)CC1CO 36650,C(C(C)(C)CNC(=O)Cn1cnnn1)N(C(=O)CN(C1CCCC1)CCO)C 36651,C1(C(N(C)CCOCCCO)=O)CCN(C(C2(OC)CCCCC2)=O)CC1(C)C 36652,C1(NC(C2(C(N(CC=CCl)C)=O)CCCO2)=O)CCC(C#N)CC1 36653,Cc1c[nH]nc1C(=O)N(CCC(C)NC(=O)C(Cc1ccccc1)N(C)C)C 36654,C1(OCC)CN(C(c2nnn(C)c2CC)=O)CC1CNC(c1cccnn1)=O 36655,C(CCCC(=O)N1CCC(N(C(=O)C(c2nc(C)cs2)C)C)C1)(OC)OC 36656,N1(C(C(CC)N(C)C)=O)CCSCC1CNC(=O)C(O)c1cnc[nH]1 36657,C(=O)(C1CCC(=O)c2cccn21)N1CCCC(NC(CC2(OC)CCC2)=O)C1C 36658,c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC23CCC3)nn(C)c2ccccc12 36659,c1(C(N2C(CNC(C3OCCN(CC)C3)=O)CCCC2)=O)cc2ncccc2[nH]1 36660,c1(SC)cc(C(=O)N(CCCCCNC(=O)CCc2cnco2)CCO)co1 36661,c1(C(C(=O)NCCC(C)(C)NC(Cc2nnc(C)s2)=O)N(C)C)cccc(Cl)c1 36662,C1(OC)CC(NC(c2cc(C)nc(O)c2)=O)CN(C(=O)C(C)Cc2cnc[nH]2)C1 36663,C(=O)(CC(O)C(C)C)NC(C1CCN(C(c2c(OC)noc2C)=O)CC1)C 36664,N1(C(Cc2cn(CC)nn2)=O)CC(CNC(=O)C(c2cncnc2)C)C(C)C1 36665,N1(C(C2(OC)CCSC2)=O)C2CCC(C2)C1CNC(c1cc(C)c(C)[nH]1)=O 36666,C(=O)(CC(F)(F)F)NC1(N(C)C(C2CCC(C(F)(F)F)C2)=O)CN(C(=O)C2CC2)C1 36667,c1(C(N2C(C)CCC(NC(c3coc(O)n3)=O)C2)=O)ccc2cncn2c1 36668,Cc1cccc(CC(N2CC(F)CC2CC(=O)NCCOC2CCC2)=O)c1F 36669,c1(N2CC(C(C)NC(c3n(COC)ncc3)=O)C2)cc(C(F)F)nc2ncnn12 36670,C1(N(C)C)CN(C(C23CC2CCN3C(C2COCCN2C)=O)=O)CC1(C)C 36671,N1(C(c2n(CC)ncc2)=O)CCOC(CNC(=O)CCCc2nc(CC)no2)C1 36672,c1(C(N(C2CC(C)(C)O2)CCNC(C2CC(C)C2)=O)=O)ncoc1C1CCC1 36673,Cc1cc(O)ccc1C(N1CC=CC(NC(=O)CCn2cccnc2=O)C1)=O 36674,c1(C(=O)NC2C3(CC(NC(c4c(C)cc(Br)o4)=O)C3)C2)cc[nH]c2nccc1-2 36675,C(=O)(CCC(=O)N(CCCCCNC(c1c(C)nsc1N)=O)C)NC 36676,c1(C(N2CCC(N(C(=O)CNC(N)=O)CC)C2)=O)cc(OC)c2c(c1)CCO2 36677,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)=O)N(C1CCCC(C)C1C)C 36678,C(C(C)(C(C)C)NC(=O)C(c1cccc(F)c1)F)NC(C=C(C)C(C)C)=O 36679,c1(C(N2CCC(NC(C(CCSC)OC)=O)C(F)C2)=O)cc2oc(C)c(C)c2[nH]1 36680,c1(CC(=O)OCC2(C)CCOC2)cccc(Cc2ccccc2O)c1 36681,CC1CCN(C(=O)C(O)CCCNC(C2CC(C)(C)CCO2)=O)CC(C)O1 36682,CCCC(C)(C)C(=O)NC12CC(C(N3CC(=O)NC(CC)C3)=O)(C1)C2 36683,C(=O)(C(C)(CCC#N)N(C(=O)C(=O)NC)C)N(C(C)C=O)C.C(C(F)F)N 36684,CC1(c2ccc(NCCCc3nnc(-c4cccnc4)o3)cc2)NC(=O)NC1=O 36685,c1(C(C(=O)NCC2CCOC2)N(C)Cc2cnc(CC)s2)ccc(C)cc1Cl 36686,C1(C)(CN(CCC)C(C2CCN(C(=O)NC)CC2)=O)CCCC1C.C1(=O)CCN1 36687,C(=O)(CCC(F)F)N(CCN(C(c1cc(O)cs1)=O)CC)CC 36688,C(N=c1[nH]c(=NCCS(=O)(=O)c2ccccc2)[nH]c2c1CCCC2)C1(CCC)CC1 36689,c1(C(=O)NCC2CCCN(C(C3CNC(=O)N3)=O)C2)cc2cc(F)cc(F)c2[nH]1 36690,C1(=CC(=O)NC2(CC=C)CN(C(c3ccsc3CSC)=O)C2)CCC(C)CC1 36691,C1(O)(C(=O)OC)CC(NCCSCCc2ccccc2)C1 36692,C1(O)(CNC(C(C)=C2CCCC2)=O)CCN(C(=O)C(O)C2CCCC2)CC1 36693,CC(=O)C(C)(C)CC(=O)N1CC=CC(C(=O)NC(C)(CN(C)C)CO)C1 36694,CCC(C)CCN=c1[nH]c(=NCC2CC23CCC3)c2ncccc2[nH]1 36695,CC1(C(=O)NCCNC(C2CCN(C3CCC3)C2)=O)CCC2CC2C1 36696,c1(CC(N2C(C)(CNC(=O)CO)CCC2)=O)cccc2ccccc12 36697,c1(CNC=O)ccc(OCCC2CCC2)nc1.C1(CC(=O)C)(SC)CC1.C1CC1 36698,C(=O)(C1=COCCC1)NCC1N(C(C(C)CN(C)C)=O)CC1 36699,C1(C(N2CC(=CCC)C2)=O)CN(C(C2CC(N(C)C)C2)=O)CC1F 36700,Cc1cc(C2(C(=O)NC3CCCN(C(C4CCCCC4)=O)C3)CC2)cc(C)c1 36701,Cc1ccnc(C(=O)N(CCCC(=O)N(C)CCN2CCCC2)C)n1 36702,c1(C(=O)NCCC2(O)CN(C(CC=C(C)C)=O)C2)cnc(N(C)C)nc1 36703,N1(C(C2C(OCC)CC2)=O)CCCC(O)(CCOC(=O)C(C(C)C)N(C)C)C1 36704,N1(C(c2c(C#N)nc[nH]2)=O)CC(NC(c2c[nH]c(=O)cn2)=O)CC12CCCOC2 36705,C(CN=C(NCC(c1cccc2c1CCCC2)O)N1CC(O)C(C)(C)C1)SC 36706,c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)C2CC2)scc(C)c1C 36707,CCCCC(O)C(=O)N(CC(=O)NC1(CC)CCCC1)C1CC1 36708,Cn1cnc2c(NCC(C(C)(C)C)C3CC3)[nH]c(=NCCOCCC(F)F)nc12 36709,C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NCC(CC)C(C)C)CC(O)C1 36710,c1(CNC(c2nnnn2CC(F)F)CCOC)cc(OC)c(OC)cc1O 36711,C1(O)(CC)CCN(C(=O)C=CC(C)NC(C2CCCC2O)=O)C1 36712,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36713,c1(OC)ccc(F)c(C(=O)N(C2CCN(C(C3SCC=C3C)=O)C2)CCO)c1 36714,C1(C(=O)NCCCOCC#C)CCC2(CCC2)CN1C(=O)C(C)C(C)COC 36715,c1(N(CC(C(=O)NC2CC2)NC(=O)C(O)CN2CCCC2)C)ccc(Cl)cc1Cl 36716,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36717,C1(NC(C(C)(C)SC)c2nnnn2CCC2(C)CC2)CCC(C)C(C)C1 36718,c1(C(=O)NC2CCCC(NC(C3C(C#N)C3)=O)CC2)cnc2c[nH]nc2c1 36719,N1(C(C=CC(CC)=CC)=O)CC(NC(c2nccnc2C)=O)CC1CO 36720,Cc1c(N(C(C)C)CC2(F)CC2)ncnc1N1CCC(OC2CC2)CC1 36721,n1(CCC(=O)NCCCCCN(C(=O)CC2CC23CC3)C)ccc(O)nc1=O 36722,c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2)cncc(F)c1C 36723,c1(CCC(=O)NC2CC2NC(c2cc(Cl)ns2)=O)ccc(OC(F)F)cc1 36724,CCCC(C)(CC)C(=O)NCc1cccc(N(C(C2CC23CCSCC3)=O)CCCC)c1 36725,C1(C(N(C2CN(C(C(c3cccnc3)C)=O)C2)C)=O)C(C)(C)C1(C)C 36726,C1(NC(CCCCCC)=O)CC2CN(C(=O)C(=Cc3cccs3)C)CCN2C1=O 36727,CCC(CC)C(=O)NCC1CCCCC1O 36728,c1(CS(=O)(=O)N(C)C(c2cc(C(=O)O)[nH]n2)=O)ccc2ccccc2c1 36729,c1(CC(=O)OCC2C(C)CCCC2)cc(Br)ccc1Cl 36730,Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)CCc2cc(Cl)no2)cc(N)c1 36731,N1(C(C2(C)CC2c2ccccc2)=O)CCC(CC(=O)NC(C)(C)C(C)(C)O)CC1 36732,c1(C(=O)NC2(C)C(NC(CC3(COC)CCCC3)=O)CCC2)ncc(Cl)cc1Cl 36733,c1(OC)ccccc1CC(C)CC(=O)NCCC(C)(C)NC(=O)C(F)C(C)C 36734,N1(C(c2cc(C)no2)=O)CCC2CCCN(C(=O)CCc3cn(C)nc3C)C2C1 36735,C1(COC(c2nc(OC)c(C)s2)=O)C2CC1N(C(=O)OC(C)(C)C)C2C(F)(F)F 36736,C1(C(=O)NC(c2ccc(OC)nc2)C)CC2CCC1N2C(c1cncc(C)c1)=O 36737,c1(COC)ncc(C(=O)NC2CC(CNC(=O)C(C)OCC3CC3)C2)c(O)n1 36738,c1(C(=O)Nc2ncccn2)cc(NC(=O)C2CC2)ccc1F.C12CN(C3CC13)C2=O 36739,c1(C(=O)NC(C2N(C(c3c(C(C)C)ncs3)=O)CCC2)C)cc2n(n1)CCC2 36740,c1(OC)ccc(Br)c(C(=O)NCC2CC2CNC(=O)CS(C)(=O)=O)c1 36741,c1(OC)c(C)cc(NC(C2CC23CN(C(=O)CCc2ccco2)C3)=O)cc1C 36742,C1(C(=O)NCC2(F)CCC(CNC(Cn3ccc(C)n3)=O)C2)CC(C2CCC2)C1 36743,C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccn(C)c2)(COC)CCCC1 36744,c1(C(N(C)CCF)=O)ccc(Cn2cc(CCN3CCCC3)nn2)o1 36745,c1(Cn2c(-c3n(CC)ccn3)ncc2)ccccc1Oc1csc(C)n1 36746,c1(C(=O)NSc2nccc(C)n2)cc(Cl)ccc1Cl 36747,C1(N(C(=O)CCN2CCOC2=O)C)CCCC(NC(=O)Cc2cc(Cl)n(C)n2)C1 36748,c1(C(N2CC3CC2CN3C(c2nc3ccccc3o2)=O)=O)cccn2ncnc12 36749,CC1CCC(C)(NC(C2CCCN2C(c2cc(CO)on2)=O)=O)C1 36750,C1(N(C(CCc2nc(C)sc2)=O)C)CCN(CC(O)C(C)c2ccccc2)CC1 36751,c1(C(=O)NCC(CN(C(C2(OCC)CCC2)=O)C)O)c(C)nn(C)c1N 36752,CC(C)C(CC(=O)N1CCC(O)CC1)NC(c1cocn1)=O 36753,CCC(CC(=O)NC(C(=O)NCC1(CC)CCCO1)C(C)OC)OC 36754,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(C23CC(C)(CO2)C3)=O)C1 36755,CCC(C)C(O)C(=O)N1CCCN(C2CC2)CC1.c12ccc(cc1)OCCO2 36756,c1(C(=O)NC2C(CNC(C(C)NC=O)=O)C2)ncc(F)cn1 36757,c1(N(C)CCn2cc(Br)cn2)cc(S(=O)(=O)NC)ccc1Cl 36758,N1(C(c2ccc(C)n2C)=O)CCCCC2(CCN(C(c3cncc(N)n3)=O)C2)C1 36759,CC1(C)CCCCCC1NC(=O)CC1CCCNC1=O 36760,Cc1ccc(I)c(C(=O)NC2CN(C(=O)C(c3ccc(F)cc3)F)CC23CC3)c1 36761,C1(NC(C2C(C(C)C)CN(C(=O)CC3CSCCO3)C2)=O)CCNC(=O)CC1 36762,CP(C)(=O)C(O)C(=O)NCCOC1CN(C(=O)CCC2CCCC2)C1 36763,CC1CNc2cc(C(=O)NC3CCC(N(C)C(C4CC(F)C4)=O)CC3)ccc2O1 36764,C(C(C(=O)NOCCC1CC1)C(C)(C)C)NC(CSCCCC)=O 36765,N1(C(CC(=O)NCC#C)=O)CC(CNC(c2ncc(C)cc2OC)=O)C2(CC2)C1 36766,C1(C(=O)NCCN2CCCOC2=O)Cc2ccc(Br)cc2N1 36767,c1(C(N(CC(O)OC)Cc2ccccc2)C)nc2ccc(Cl)cc2[nH]1 36768,C=C(C)C(CC(=O)NCC1CCC1NC(=O)COc1ccc(F)cc1F)OCC 36769,C1(NC(C2CCCC(F)C2)=O)CCN(C(c2cnccn2)=O)CC12CCC2 36770,C1(COC)(NC(=O)C(C)=CC(C)(C)C)CCN(C(=O)CCC=C(C)C)C1 36771,c1(C(=O)NC2CC(NC(CCC=CCC=C)=O)C23CCC3)cc2ccccn2n1 36772,C(=O)(CCC1CC1(F)F)N(C)CCOCCN(C)C(C1CC1C(F)(F)F)=O 36773,C1(C(=O)NCCCOCCCNC(C(C)(C)CC2CCC2)=O)CCCCC(=O)N1 36774,Cc1nn[nH]c1C(N1CCCC1C(=O)NCC1(C)CCC1)=O 36775,c1(NCc2c(C)cccc2Cl)cn2cnnc2cn1.C12(OC)CN(C1)C2=O 36776,C12(C(=O)NCC(O)CNC(C3CC(OC(F)F)C3)=O)CC3CC(C1)CC(O)(C3)C2 36777,c1(OCC)c(C(N2CCN(C(=O)CC(CC)SC)C(CF)C2)=O)cccc1Cl 36778,N1(C(C(Cc2cn[nH]c2)NC(C2C(C)CC2)=O)=O)CCOC(C)(C)C1C 36779,c1(C(N(C)CC2CN(C(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 36780,C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(c1ncccc1OC)=O)C2 36781,C(=O)(C(C)(C)CCCO)N1CCCC(N(C)C(c2cnn[nH]2)=O)C1 36782,N1(C(C(CC)CN(C)C)=O)CC2CCCC(C1)N2C(=O)CCC(C)OC 36783,C1(CC(=O)N(C(c2ncc[nH]2)C)C2CC2)(NC(=O)CC2(N(C)C)CC2)CCC1 36784,c1(C(=O)NC(C2CN(C(c3cc(OC)no3)=O)C2)C)cnc(C2CC2)nc1O 36785,C1(CC(=O)NC2(CF)CN(C(CCC#C)=O)C2)CCCC1O 36786,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 36787,C1(CNC(Cc2c(C)con2)=O)CCCN(C(c2ccnn2C(C)C)=O)C1 36788,C1(NC(c2c(OC)cnc(Br)c2)=O)CC2(CCN(C(=O)CC3CCCC3)CC2)C1 36789,N1(C(CS(=O)(=O)NC)=O)CC(NC(=O)Cc2ccc(O)cn2)CC12CCC2 36790,c1(C(N2CCC(Br)C2)=O)cnn2c1CN(Cc1ccc(F)cn1)CC2 36791,C1(C(N2CC(OCCNC(c3c(C(C)C)c[nH]c3)=O)C2)=O)CC(=O)NC(C)C1 36792,c1(C(NOCC(C)CC2CC2)=O)cc(OC#N)cc(Cl)c1 36793,CC1CN(C(C2CN(C(C3(Cc4ccccc4)COC3)=O)C2)=O)CC1 36794,Cc1cc(=O)c(C(=O)NCC2CN(C(=O)CCc3nc(O)n[nH]3)CCC2C)cn1C 36795,N1(C(C(N(C(CC(CN(C)C)O)=O)C)C2CC2)=O)CC2CCC(O)C2C1 36796,c1(NC(C(=O)NC(C(CC)C)CO)=O)c(I)cnc(Cl)c1F 36797,c1(CC)cc(C(=O)NCC2CC(CNC(=O)CN(c3ccccc3)C)CO2)on1 36798,c1(C2(NC(C3CN(C(C4CCC(OC)C4)=O)CC3O)=O)CC2)ccc(F)cc1F 36799,N1(C(C(C2CCC2)NCc2[nH]nnc2C2CC2)=O)CC2(C=C(C(=O)OC)CO2)C1 36800,c1(-c2n(C)ncc2)ccn2cc(-c3cccc4c3OCO4)nc2c1 36801,N1(C(CN(c2ccccc2)C)=O)CC2CCCN(C(=O)CC3(C#N)CC3)C2C1 36802,Cc1ccc(OCC(N2CC(C)(NC(c3c(C)coc3C)=O)C2)=O)c(C)c1 36803,c1(CC(N2CC(OCCNC(C(C=CC)O)=O)C2)=O)cc(F)ncc1Br 36804,Cc1cccc(C(=O)NCC(=O)NC2CCC(Cn3cc(C(C)O)nn3)CC2)n1 36805,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 36806,C=CC(CC)CC(=O)NCC=CCNC(=O)C(c1cccc(Cl)c1)O 36807,c1(C(C)C)cc(C(=O)N(CCC(C)NC(C2CNC(=O)C2)=O)C)ccc1F 36808,c1(C(N(CCC)CCN2CCN(CC)CC2)=O)c[nH]c2cc(F)c(F)cc12 36809,c1(C(=O)NC2(COC)CN(C(C3C(C=C)OCC3)=O)C2)cc2ncccc2o1 36810,C1(NC(C=C(C)Cl)=O)CCC(O)CN(C(C2CC2CF)=O)C1 36811,c1(C(=O)NC2CCC(NC(c3c(CC)nccn3)=O)C2)cc(C(=O)OC)ccc1O 36812,N1(C(C2CC23CC(O)C3)=O)CC2(C(=O)NCCOCCO)CCC1CC2 36813,c12cccc(c1)C(=O)N2.C1(C(=O)NC(C)CN2CCCCC2)NC(=O)OC1C 36814,c1(C(=O)NCC2C(C(=O)OC)C2)cn2cc[nH]c(=O)c2n1.C12COCCN1C2=O 36815,n1(CC(C2CCCS2)=O)cc(CCN2CCOCC2)nn1 36816,C(=O)(C1=CCCOCC1)NCC1(C)CCC(NC(=O)Cn2ccccc2=O)CC1 36817,c1(N(C2CCCC2)C(=O)NCCNC(=O)CCn2cncn2)ccc(Cl)cc1Cl 36818,Cn1ccc(CC(N2CC(F)(CNC(C3(C(c4ccccc4)=O)CC3)=O)C2)=O)n1 36819,c1(NC(=O)CC2COCCN2C(C2CC3CCCC3C2)=O)ccc2nc(O)[nH]c2c1 36820,c1(CCNC2CN(C(c3cnn(-c4ccccc4)n3)=O)C2)ccccc1CSC 36821,N1(C(C2N(C(C)=O)CSC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 36822,c1(C(N(CCN(C(CN(CCC)C)=O)C(C)C)C)=O)cc(C)c(Cl)cc1C 36823,N1(C(CC2CC(SC)C2)=O)CCCC(C)C1CNC(=O)C(C)n1ccnc1 36824,C(=O)(CCCN=[N+]=[N-])NCc1nn(CC(C)C)c(-c2cn(C3CCOC3)nn2)n1 36825,N1(C(c2c(CC)non2)=O)CCC(CCCCNC(C2CC(C)C2)=O)CC1 36826,c1(N2CCC3(CC(OC)C3)C2)nc(=NCc2cc(C)cs2)[nH]c2c1CCC2 36827,N1(C(C(CC)O)=O)CC2CCCC(CNC(c3cc(O)cc(=O)o3)=O)(C2)C1 36828,c1(OC)ccc(C)c(C(F)(F)F)c1.c12nc(n(C(C)C(F)(F)F)n1)C1CC21 36829,C1(NC(=O)CC2(O)CCCCC2)CCC2CN(C(=O)CC3(CO)CC3)CC2C1 36830,c1(C(=O)NCCC2CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 36831,C1(CC)(NC(C2(CC(C)C)CC2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 36832,C1(NC(Cc2c(C)n[nH]c2C)=O)CCCN(C(=O)CNC=O)CC1F 36833,c1(CC(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)C)ccc(F)c(F)c1 36834,CCCCC(C)C(=O)N1CC(F)CC1CN(C)C(C1(CO)CCCC1)=O 36835,C1(C)(C(c2n(CC=C)nnn2)NCCC(=O)N(C)C)CCOCC1.C(CN)S 36836,C(C(C)(C)CNC(c1nonc1N)=O)N(C)C(C1C=CCCC1)=O 36837,C1(N(C(C(C2CC(C)(C)C2)OC)=O)C)C2CN(C(=O)CC(C)(F)F)CC12 36838,C(=O)(C1=CC2C=CC(C1)C2)NCCN(C(CC)CC)C(=O)CC1(n2cccn2)CC1 36839,c1(C(N2C3CC(CNC(C(C)C(C)(C)O)=O)C2CC3)=O)ccccc1[N+](=O)[O-] 36840,c1(C)ccccc1CNC(CC(C)C1CC1)=O.C1(C(NC)=O)C(F)(F)C12CC2 36841,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)C(C)CC1 36842,c1(NC(=O)C(=O)NC(C)CC2(Br)CCC2)ccccc1CC(C)N(C)C 36843,c1(CC(=O)N(CCCCCCNC(=O)CC2CCSCC2)C)ncnc2[nH]cnc12 36844,Cc1ccc2oc(C(=O)NC3CN(C(=O)CCNC(=O)CO)C4CC34)cc2n1 36845,C(CC(C(C)(C)C)NC(=O)C1=CCCCC1)N(C(C1(C)C(C)C1)=O)C 36846,CCCCC(C(=O)NC1CC(F)C1)NC(=O)C(C)OCC 36847,C1(CN(C(C(CC)C)=O)C)CCCCN1C(=O)C(C)(C)NC(C1CCCC1)=O 36848,c1(C(=O)NCC2(CF)CCC2)cc(Br)cnc1N1CCCC1 36849,CCC(C)(C(=O)NC(CNC(=O)C=Cc1cccc(F)c1F)C(C)C)C(F)F 36850,C(=O)(C(CC)C(C)O)N1CC(C(C)(C)O)(CNC(C(CC)CC)=O)C1 36851,c1(C(=O)NC(=O)Nc2cnn(CO)c2)scnc1CC1CC(c2ccccc2)C1 36852,N1(C(Cc2cc(CC)no2)=O)CCC2CC12C(=O)NCC12CCC(OCCC)C1C2 36853,N1(C(C2(CC)CC2)=O)C(C(=O)NCc2ccc3nc[nH]c3c2)CC2CCCCC12 36854,c1(NC(C(C2CCCN(C(=O)C(=O)NCP(C)(C)=O)C2)(C)C)=O)ccccc1F 36855,C1(NC(CCOCC)=O)CCC(CC(=O)NCCCC2CCCC2)C1 36856,C(=O)(C(O)P(C)(C)=O)N1CCC(C(=O)NC2C(N(C)C)CC2)C1 36857,C1(NC(C(C)CC2CCC2)=O)CCS(=O)(=O)C12CN(C(C1CN(C)CCO1)=O)C2 36858,c1(C(=O)NC2C(NC(c3cc(CCC)nn3C)=O)CCC2)nc(C)c(C)[nH]c1=O 36859,c1(CCC(=O)NCC(C)N(C2C(CC)CC2)CC)nc(-c2cccs2)no1 36860,C1(c2nnnn2Cc2ccnn2C)(NC(COC)(C)C2CC2)CN2CCCC2C1 36861,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 36862,Cc1cnc(C(=O)NCC2C(C)CCN2C(c2cnn(C3CCC3)c2)=O)cc1C 36863,c1(OC)ccc([N+](=O)[O-])cc1CNC(N1CCC1C1CCCC1)=O 36864,c1(C(=O)NC(CN(C(C(CC)n2cncn2)=O)C)C)ccccc1C(N)=O 36865,N1(C(C(Br)=C(C)C)=O)CC(C)OC2(CCN(c3ncc([N+](=O)[O-])cc3Br)C2)C1 36866,CCCCC(C(=O)NC1CCN(C(C2(CF)CC(F)(F)C2)=O)CC1)N(C)C 36867,N1(C(CC(COC)(C)O)=O)CC(CO)C2(C1)CN(c1ncnc3cnn(C)c13)C2 36868,C1(CNC(C2CN(CC)C(=O)C2)=O)C(C)CCCN1C(=O)CCc1cncn1C 36869,c1(C(=O)NC2(C)CN(C(C(CC)OC)=O)C2)ncc(OC)nc1OC 36870,C1(NC(C2CC(CC)(CC)C2)=O)CN(C(=O)CC2COC(=O)C2)CC1S(C)(=O)=O 36871,c1(SCC(=O)N(CCN(C(C(C2CCCCC2)NC(C)=O)=O)C)C)n[nH]c(O)n1 36872,Cn1nc(C(=O)NCCN2CCCS2(=O)=O)c(C2CCCO2)n1 36873,C(N=c1[nH]nco1)c1cnn(C(N2CC(O)(C(F)CO)C2)=O)c1 36874,Cn1c(C(=O)NCCNC(c2c(F)cc([N+](=O)[O-])cc2F)=O)cc2c1CCOC2 36875,C(=O)(CCCCO)N.N1(C(C(C2CCCC2)OCC)=O)CCC(OC(C)C)C1 36876,Cc1ccnc(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)c1F 36877,c1(C(C)C)ccc(C(N2CCN(C(c3ccnc(Cl)c3)=O)CC2CO)=O)c(O)c1 36878,c1(C(=O)NC2CCCC(NC(C3CC(CC4CC4)C3)=O)C2)cccc2ccsc12 36879,CC(CC(=O)N(C)CCc1ccc(Cl)c(C(F)(F)F)c1)C(C)(C)C 36880,N1(C(C(CC)NC(N)=O)=O)CCCC(N(C)Cc2ccc(F)c(Cl)c2)CC1 36881,C1(OC(C)(C)C)CC(N(C)C)CN(C(=O)OC2CN(C(C)=O)C2)C1 36882,C1(C)(NC(c2c(CC)c[nH]c2)=O)CCCN(C(c2nn(C)cc2N)=O)C1 36883,CN1CCCC(N2CC=CC(NC(c3cc(C4CCCN4C)[nH]n3)=O)C2)C1=O 36884,Cn1c(Cl)nc2cc(C(=O)OCC(c3ccc(Br)cc3)F)c(O)nc12 36885,CCC(C)(CO)C(=O)N1CC(C(N2CC(OCCOC)C2)=O)C(F)C1 36886,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)N(C(=O)COC1CCC1)C1CC1 36887,C#Cc1cn(C)nc1C(=O)NCCN1CCN(C(=O)C(C)=CC2CC2)CC1 36888,c1(C(N2CC(CNC(Cc3c(CC)c[nH]n3)=O)C(O)C2)=O)cc(F)cc(F)c1 36889,C(=O)(CCC(N)Cc1ccccc1)N(C(CCC)C)C 36890,C(=O)(CCC(=O)NCC(C(=O)OCC)NC(C1CC(O)(CCC)C1)=O)OC 36891,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 36892,C1(C(N2CC(C#N)(SC)C2)=O)(CC)CCCN1C(=O)C=CC1CCCN1C 36893,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccnn1CC(F)F)=O 36894,C1(C(N(C(C#C)C)CCCC)=O)CC12CC(NC(c1cnncc1C)=O)C2 36895,N1(C(C(C)=CC)=O)CCC2CC2(NC(c2ccn(C3CCCCC3)n2)=O)CC1 36896,c1(C(N(C(c2cn(CCC)nc2)C(=O)NC(C)C)CCC#N)C)ccc(F)cc1 36897,c1(OC)c(Br)ccc(F)c1-c1cnc(CC(=O)N(CCCCO)CCO)nc1 36898,c1(CC)nc(C)cc(=NCC(O)CNC(=O)C(C)CSC2CCCC2)[nH]1 36899,N1(C(CC(c2cccc(F)n2)NC(=O)C(Cl)Cl)=O)CC2(CCCO2)C1 36900,c1(C(=O)Nc2cncc(-c3cnc(-n4ccnc4)cc3C)c2)ccc(C#N)cc1 36901,C1(OC)C=CCN(C(=O)C(C)(CO)NC(c2ccncc2F)=O)C1 36902,N1(C(C(C)=CC)=O)CCC(CCNC(c2cc(COC)n(C)n2)=O)CC1C 36903,c1(N2CCC(N(CCNC(=O)C(C)COC)CC)C2=O)c(F)cccc1F 36904,C1(NC(=O)CC2CCN2C(=O)CSC2CC2)CC2C(C1)C2(F)F 36905,c1(C(CCCOC)C)nc(C2CCCN(C)C2)nn1-c1ccc(F)cc1 36906,n1(CC)ncc(CCNC(=O)NOC(CC)CCCO)c1C 36907,C1(C(N(CCCC)CCCC)=O)CC(COC)CN1C(=O)Cc1cncn1C 36908,C1(C(=O)NCC(C)(C2CCC2)NC(C2C3COCC23)=O)C2CC3C(C2=O)C13 36909,CCC(O)C(=O)NC1CC(c2ccccc2)(CNC(c2ncoc2C(C)C)=O)C1 36910,C12(C(N3CCN(C(CCCNC(=O)OCC)=O)C4C3C4)=O)CCC(C)(CC1)OC2 36911,C1(NC(=O)NCC(N2CC(C(CO)NC(=O)C3CC3)C2)=O)C2CCCCCCC12 36912,c1(NC)ccccc1C(=O)NC1CC1NC(c1cnc(Br)s1)=O 36913,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 36914,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 36915,C(=O)(CC(CC)CC)NC(C1CC(CCC2CC(NS(=O)(=O)CC)C2)C1)CC 36916,N1(C(CC)NC(c2cnc(NC(=O)OC(C)(C)C)s2)=O)C(=O)CCC1=O 36917,c1(OC)nc(C)ccc1C(N1CCC(C)C1CNC(C1(C)CC(=O)N(C)C1)=O)=O 36918,C1(C(N(C2CC(SC)C2)C)=O)CCCCN(C(C2CCOC2(C)C)=O)C1 36919,C1(Cc2cn(C)nn2)CCN(C(c2cnc3sccn23)=O)CCC1C1(CO)CC1 36920,Cc1sncc1C(=O)NC(C(=O)N(CCO)CCc1ccccc1)C1CC1 36921,C1(NC(C2CCCN2CC2CC2)=O)CCN(C(C2(CF)COC2)=O)CC1F 36922,c1(C2C(CC3(N(C)C(C)=O)CN(OC(=O)OC(C)(C)C)C3)C2)ccc(C)c(F)c1 36923,c1(C(N(CCNC(=O)C(O)C2CCCC2)CC)=O)ccc(Br)c([N+](=O)[O-])c1 36924,C1(C(N(C2CCC(OC(C)C)C2)C)=O)OCCCC1(C)C 36925,Cc1cc(NC(=O)NC2CCN(C(=O)CN3CCOC3=O)C2)cc(C)c1Cl 36926,c1(C(=O)NC2CC(F)(CNC(C(CC)O)=O)C2)cc(OC)c(OC)c([N+](=O)[O-])c1 36927,C1(C(=O)NCC2CCC(NC(c3n(CC)ccc3)=O)C2)CCc2nc(O)[nH]c2C1 36928,S(=O)(=O)(c1ccc(C(=O)O)c(C)c1)NCC1=C(C)C(=O)c2c(cccc2)C1=O 36929,Cc1nnc(CCC(=O)N2CCC2CNc2csc(-c3ccc(F)cc3)n2)n1C 36930,CC1CCC1C(C)NC(C1CC1(F)F)C1CC1 36931,c1(CC(=O)NC2CC(F)(CNC(CCC(C)SC)=O)C2)ccc(C)c(F)c1F 36932,C(C)(C)(C(C)NC(=O)CC(C)C1CCCO1)NC(CC)=O 36933,C1(C(=O)NC2(CC(=O)N(CC(C)C#N)C)CC2)CCNC(=O)C1 36934,CN1C(=O)OCC1C(=O)NCC1(NC(C2CCCCC2c2nnc(S)n2C)=O)CC1 36935,C1(CNC(CCc2c(C)ncs2)=O)CN(C(c2cccnn2)=O)C2CCN1C2 36936,C1(CNC(C(C)Oc2ccccn2)=O)CN(C)CCN1C(c1cncc(Cl)c1)=O 36937,N1(C(c2ccnc(C(C)C)n2)C(=O)NCc2ccco2)CCC(C2(O)CC2)CC1 36938,CCC(O)C(=O)N1CCCC1C(=O)NC(C)Cc1cn[nH]c1 36939,CC1(C)CCC(C)(NC(=O)CCNC(c2ccc(F)cn2)=O)C1 36940,c1(NC)nc(C)ccc1C(=O)NCC1CCCC(NC(=O)Cc2ccsc2)C1 36941,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 36942,C12(NC(c3nc(CCCCC)sc3)=O)CC1CN(C(c1sc(C)nc1C)=O)C2 36943,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 36944,N1(C(C2(C=C)CC2)=O)CCCC(C2CN(C(=O)C3CCc4scnc43)C2)C1 36945,Cc1ccnc(C(N2CCC(C(=O)NOC3CCOC3)(C(C)C)CC2)=O)c1N 36946,CCC(C(=O)OC)C(=O)NC1CN(C(c2ccc(OC)cn2)=O)C1 36947,c1(CC(=O)NCC(C)N(C(c2ccc(SCCC)o2)=O)CC)ccc(F)cc1C 36948,Cc1ccc2ncc(C(=O)NCC3CC3CNC(=O)Cc3cnnn3C)n2c1 36949,C(=O)(CN=c1cc[nH]cc1)N(CCNC(=O)C1=C(C)OCCS1)CC 36950,N1(C(C(=O)Nc2c(C(=O)OC)nn(C)c2Br)=O)CCC2(CNC(=O)C2)C1 36951,N1(C(CCc2cnc(C)s2)=O)CCC(NC(=O)C=CC(=O)N(C)C)C1C 36952,C(=O)(C1=C(SC)CCCC1)NCC(C)CN(C)C(c1ccc(Br)o1)=O 36953,C1(NC(C2(CC#C)CCCO2)=O)CCC2CC1CN2C(=O)CC(=O)OCC 36954,CC1(C)C2CCC1(CC(=O)NC1(CF)CCN(C(=O)CCC3CCCO3)C1)CC2 36955,C#Cc1ccccc1CC(=O)NC(C)CNC(c1cc(C2CC2)on1)=O 36956,C1(NC(CCOCC)=O)CC2(CCN(C(c3cnn(CC)c3Cl)=O)C2)C1 36957,c1(C(CN(C)Cc2ncoc2CCCN)=O)cccc(C(N)=O)c1 36958,c1(N2CCC(CCCC)C2)nc2cccnc2c(=NC2CCCC2N(C)C)[nH]1 36959,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)C(C)(O)C1CCOC1)CC2 36960,C1(CCOC)(NC(COCC=C)=O)CCN(C(=O)C(C)=CC2CC2)C1 36961,c1(OC)cc(CC(=O)NC2CCC(NCc3cc(C(=O)O)n[nH]3)C2)ccn1 36962,N#Cc1ccc(C(=O)NCC(CC2CCCC2)C(=O)NCCC(F)F)o1 36963,C12(C(N(C(CC)CC)C3CC3)=O)CC(NC(=O)C(F)n3ccnc3)(C1)C2 36964,N1(Cc2c(Br)ccc(C)n2)CC2C(C1C(N1CC(n3cccn3)C1)=O)C2(C)C 36965,C1(C(N2C3C(NC(C(CCC)=CCC)=O)C(C3)C2)=O)CCC([N+](=O)[O-])CC1 36966,c12c(Br)ccc(c1C)NC1C3CCN(CCC31)C2=O.N1(CCO)CCOC1=O.CSC 36967,c1(C(=O)NC2OCCN(C(C=CC(C)C)=O)C2)cc(N(C)C)ccc1Br 36968,c1(N2CC(C)OCC2)nc(=NCCOc2ncccc2F)[nH]c2c1SCC2 36969,C(c1ccc(C)cc1)=C(C(N1C(CC)C(NC(COCCCCC)=O)CC1)=O)C 36970,c1(CC(CNC(=NCC2CC(OC)C2)NC2CC2)OC)cc2occc2[nH]1 36971,c1(CN(C(C(=O)OC)C(C2CCCCC2)OC)CCOC)ccnc2[nH]ncc12 36972,c1(SCC)cnccc1C(=O)NC(CNC(=O)Cc1nccn1C)CC 36973,c1(C(C)C(=O)N(C2CCCC2)Cc2ccc(Cl)cc2)ccc2c(c1)OCO2 36974,C1(NC(C=C(CC)C)=O)CC(C2CCN(C(c3ccc([N+](=O)[O-])c(C)c3)=O)C2)C1 36975,C1(NC(C(C)=C2CCCC2)=O)CCC2CN(CCc3ccc(CO)cc3)CC2C1 36976,Cc1ncc(C(N2CCC(C)C2CNC(C2CCCSS2)=O)=O)c(O)n1 36977,c1(COc2ccc(-c3nn(C(C)(C)C)c(=S)s3)cc2)cc2nc[nH]c2cc1F 36978,N(C1CCCc2cc(OC)ccc21)C1c2n(nnn2)C(C=C)C(CC)c2c1c[nH]n2 36979,Cn1cc(I)cc1C(=O)Nc1nc(CN2CC(O)CC2c2ccc(Br)cc2)cs1 36980,C1(C(=O)NC(CCC)c2ccco2)CCCCN(C(=O)CC2CN(C(C)=O)C2)C1 36981,C(=O)(C(C)(C)CCCC(=O)NCC(C)(C)CNC(c1sc(C)nc1C)=O)OC 36982,C(C)(N=c1nc(N2CC=CC(N(C)C)C2)c2c([nH]1)CCC2)c1ccc(C)c(C)c1 36983,C(=O)(CCC(C)(C)C)N1CCC(C)(CCNC(CN2C(C)CCCC2)=O)C1 36984,c1(C(=O)NC(CC2CCN(C(C(C=C)O)=O)CC2)C)cnc2c(c1)NC(=O)CO2 36985,c1(N(CCN(C(c2c(C)n(CC(C)C)nc2)=O)C)C)nc2ncc(Cl)cc2o1 36986,CCC(CC(C)C)C(=O)N(CC(O)CNC(c1ccc(Br)c(Cl)c1)=O)C 36987,c1(CC(=O)OCC2C(OC)CCC2)ccc(C(F)F)cn1 36988,C12(C(N3CCCCC(N(C)C(c4csc(O)n4)=O)C3)=O)CC1Cc1c[nH]nc12 36989,c1(C(N2CCC(NC(CC3(C)CCCO3)=O)C2)=O)nccc(Cl)c1F 36990,N(C1CCCc2n[nH]cc21)C(C(CO)NC(CCC(C)(F)F)=O)=O 36991,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 36992,C=CCN=C(NCC1CCCC2(CCC2)O1)N1CCN(c2cc(COC)[nH]n2)CC1 36993,Cc1c(C(=O)N(CCCNC(=O)C=CCO)CCO)c(C(F)F)nn1C 36994,N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(O)CO)C1CC1 36995,C1(C(=O)NC(CNC(Cc2c(C)cnn2C)=O)C2CCC2)CCC(C)(C)CO1 36996,c1(C(=O)NC2C(NC(c3c(CC)nc(C)o3)=O)COCC2)cc(C)nc(C)c1 36997,c1(C(N2CCC(F)(C(N3CCC(OC(F)F)C3)=O)C2)=O)ncccc1Br 36998,C#CCC(C(=O)N1CC(=C)CO1)NC(c1ccc(C)n1C)=O 36999,C1(NC(=O)C(C2CCCCC2)O)CC1C1CCN(C(c2nnc(O)cc2O)=O)CC1 37000,C1(C(N(C2CCC(O)C2)C)=O)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 37001,CC1CN(C(C(=O)NCC2CCOC2)c2ccon2)CC(c2ccco2)O1 37002,CCC(N=c1nc(N2CCC3NC(=O)NCC3C2)c2[nH]ccc2[nH]1)C1CCC1 37003,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37004,N1(C(c2n(C)nnc2CNC(C2(Cl)CC2(F)F)=O)=O)CC12CCC1(CC1)CC2 37005,c1(C(N2CC(C)(C)C(CO)C(C)(C)C2)C(=O)NCC)ccc2c(c1)OCC2(C)C 37006,N1(C(C2C(C)(C)C(=O)C2)=O)CC=C(CC(=O)NC2CCC23CCC3)CC1 37007,c1(CC(=O)N(CCNC(C(COC)OC)=O)C2CC2)ncn2c1CCCC2 37008,C(=O)(C(C)(C)CCCC(=O)NC1CCCCC1CNC(=O)C#CC1CC1)OC 37009,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(CC)=CC)=O)C1)CCO 37010,C1(C(=O)NCC(C)OCC=C)CCC(CNC(c2ccccc2O)=O)CC1 37011,CC1(C)CC(O)(C(=O)NC2CCCN(C(=O)CSc3ccccc3F)C2)C1 37012,Cc1cccc(C)c1CNC(C1CCCC1NC(c1ccncc1)=O)=O 37013,c1(C(=O)NCC(=O)N(C(C)C)Cc2onc(CC)n2)ccc(C)cc1 37014,N12CCCCC13CC(C3)C2=O.C1(C(N(CCOC)CCF)=O)C2CCCCC12 37015,C1(C(=O)Nc2nccnc2F)CC2CC1CC2C(=O)O 37016,N1(C(c2n(C(C)C)nnc2)=O)CC2CCC2(CNC(C2CCS(=O)(=O)C2)=O)C1 37017,N1(C(c2ccc(SC)cc2)=O)CC=C(CNC(=O)C(C2CCOCC2)O)CC1 37018,CCCCCC(=O)NC1CCOC(CNC(=O)C(C)(C)c2cnc[nH]2)C1 37019,CC(CN(C(C)(C)C)C)C(C)(C)C.C1(C)(C)C(=O)O1 37020,C1(C(N2CCN(CC=C)CC2)=O)CNC(=O)CN1C(C1(CC2CC2)CCC1)=O 37021,C1(C(N2C(CNC(CC3(N(C)C)COC3)=O)CCCC2)=O)CC2C=CC1C21CC1 37022,C1(C(=O)NC(C)C(C)S(C)(=O)=O)(OC)CCS(=O)(=O)CC1 37023,C1(CCC)CN(C(c2scnc2C(C)(C)C)=O)CC1NC(C1C=CCC1)=O 37024,N1(CC)CC(C(=O)NCCCC2(NC(=O)C=CC=C(Cl)Cl)CC2)c2ccccc21 37025,C(=O)(CC1=NN(C)C(=O)C1)N1C(C(N2C(COC)C=CCC2)=O)CC(O)C1 37026,C#Cc1ccc(Cl)c(C(N2CCCC2C(C)NC(=O)C=CCn2cncn2)=O)c1 37027,N1(CC)CCCN(C(N2CCC(NC(CC(C)C)C(=O)OC)C2)=O)CC1=O 37028,CCCCCCOC(C)C(=O)NCCCN(C(=O)CCC1CC(F)(F)C1)C1CC1 37029,Oc1c(F)ccc(CN=c2ccnc(N3CCN(c4ccncc4)CC3)[nH]2)c1F 37030,Cn1nc2ccccc2c1C(N1CCCN(C(=O)Cc2ccns2)C(CO)C1)=O 37031,N1(C(C(CC)C)=O)CCC2CN(C(=O)CCc3nc[nH]n3)CCC12 37032,c1(C(=O)NCCOCCNC(CCC#C)=O)ccc(F)c(F)c1F 37033,C1(CNC(c2cc(CC)nn2C)=O)CC2(CCN(C(=O)C=CC3CC3)C2)CO1 37034,c1(SC(C)C(=O)NCC2COC(=O)N2C)nc2ccccc2n1C(F)F 37035,C1(CNC(C(COC)O)=O)CCC(C)(C)CN1Cc1ccc(C#N)cc1Cl 37036,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1conc1C 37037,c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)C(C(C)O)N(C)C)C2)c(F)cn1 37038,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37039,C12(CNC(C3N(C)CCC3)=O)CC(CO1)N(C(C1CCN(CCO)C(=O)C1)=O)C2 37040,Cc1nn(C)c2ncc(C(N3CCC4(NC(c5n[nH]cc5Cl)=O)CC4C3)=O)cc12 37041,N1(C(=O)NC2C(C)=CCS2)CCCC(C(N2CC=CC2CF)=O)C1 37042,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(c1cnn(CCF)c1)=O)OC 37043,C(=O)(CCCC(C)(F)F)N(C(C)CNC(=O)CCc1ccco1)CC 37044,CC1(C)CC(NC(=O)COC2CC2)CN(C(c2ccns2)=O)C1 37045,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCC(CC)NC(=O)C1=NN(C)C(=O)CC1 37046,Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C(C)C 37047,C12(C(N(C(CN(C(C)=O)C)C)C)=O)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37048,c1(C(N(C)CC2N(C(C3(C=C)CCCCC3)=O)CCC2)=O)cc2cn[nH]c2cn1 37049,N1(C(CC(CC)C)C)CCCOC(CNC(=O)CNC(=O)C(F)(F)F)C1 37050,C1(CC(=O)NC(CC(=O)OCC)C)CN(C(=O)CC(C)C)CC12CC2 37051,c1(C(N2CC3N(C(C4N(CC)CCOC4)=O)C(CC3)C2)=O)c[nH]c2nccc-2c1 37052,C1(C(=O)NCc2c(C(=O)NCCC#N)scc2)CCn2cnnc2C1 37053,CC(C)C(CO)C(=O)N1CCC(NC(=O)Cn2nnc(C3CC3)n2)C1C 37054,C(=O)(C#CC1CC1)NCC(=CC(=O)N(CCC=C)CC)C 37055,C1(C(=O)NCCCC)CCCC(NC(=O)COCC2CCCC2)C1 37056,C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 37057,c1(C(N2C(c3cn(C(C)C)nc3)CCC2)=O)cncnc1C1CC1 37058,Cc1nc(Cl)nc(N2C3CCC2CC(NC(C2(C)CCC2)=O)C3)c1C#N 37059,C1(NC(C2(F)CCCCC2)=O)CC2CCC1(NC(C1(C(O)C(F)(F)F)CCC1)=O)C2 37060,c1(S)nccc(C(F)(F)F)n1.C(=O)(CCC1CC(C(C2CC2)NC(=O)N)C1)OCC 37061,C1(NC(C=CSC)=O)CC2(C1)CC(CNC(c1cc(C3CC3)nc(O)c1)=O)C2 37062,C1(CC(=O)NCC2(C)CC(NC(=O)CN3CC4CC4C3)C2)CCCCC1(F)F 37063,C1(CNC(C(=O)NCC(F)(F)F)=O)CC2COCC2N1C(c1ccc(CO)[nH]1)=O 37064,C1(C(N2C(C)(C(=O)NC)CC2)=O)CCN(C(C2(CC(=O)OC)CCC2)=O)CC1(C)C 37065,C1(C(N(OC)CC2CCCC2)=O)CCN(C(=O)Cc2ccsc2)CCO1 37066,C(CC(O)C(=O)NCC(C1CCC1)NC(c1ccc(-n2ccnc2)nc1)=O)SC 37067,C1(CC(=O)NCCN(C(c2cncn2C)=O)CC)CC(C)(C)CCO1 37068,c1(C(N2CC3C(NC(C4CCN(C5CC5)CC4)=O)C3C2)=O)ccc2nnnn2c1 37069,c1(SC)cc(-c2c[nH]c(=NCc3cccc(C=O)c3O)s2)nc2ccccc12 37070,C1(C(=O)NC2CC(NC(C3CCOCC3)=O)C2)CCCCCC1(F)F 37071,C1(C)(C(=O)NCC2C(NC(C=CC=CC)=O)COC2)CC2CCC(C1)S2 37072,N1(C(C2(CNC(c3c[nH]c4cccnc34)=O)CC=CC2)=O)CCc2cnccc2C1 37073,c1(N2CCC(NC(C(c3ccc(Cl)cc3)N(C)C)=O)C2=O)cc(F)c(F)c(F)c1 37074,C1(O)(CNC(C=CC(CC)=CC)=O)CCN(C(C2CNC(=O)C2)=O)C1 37075,c1(C(=O)NCC2CCCC2NC(c2ccnc(CO)c2)=O)cncc(Cl)c1Cl 37076,c1(CCCN(C)C(=O)NC(C2CCCCC2)C2CC2)ccc(C#N)cc1 37077,c1(CNc2cccc(C(=O)NCc3n(CC)ccc3)c2)cc(F)ncc1C 37078,C1(OC)CCC(C(=O)N(CC(n2cc(-c3c(C)cnn3C)nn2)C)CCO)CC1 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37131,C(=O)(C(CC(C)(C)C)N)N1CCC(C(CC)=O)CC1.C1OCCOC1C 37132,C1(C(=O)NCC=CCNC(C2C(OCC)C2)=O)CCC(C2CCC2)CC1 37133,C1(C(=O)NC2(CC(C)C)CCC2)C=CCN1C(C1CC1C(C)(F)F)=O 37134,c1(CC)cc(F)ccc1C(=O)NC1CC(NC(c2nc(C)ncc2Cl)=O)C1 37135,S(=O)(=O)(c1ccc(Cl)nc1)N1CC2(CC(NC(c3nc(C)sc3)=O)C2)C1 37136,C1(c2ccccc2)(C(C2CC2)NC(C23CC2CNC3)=O)CC2(CC2)C1 37137,C1(N(C(COCCC#C)=O)C)CC2CC1N(C(c1cnn(C3CC3)c1C)=O)C2 37138,Cc1cc(=O)oc(C)c1C(=O)NC(C)CN(C(=O)C(C)CC(C)(C)C)C 37139,c1(-c2ccc(NC(=O)CCc3ccncc3)cn2)cccc2ccccc12 37140,c1(C(=O)NCC(C)NC(C2(C(=O)OC)COC2)=O)cc2c(cc1Cl)NC(=O)C2 37141,c1(Cn2c(-c3c(OC)ccs3)nc(Cc3ccc(Cl)cc3)n2)nc2ccccc2s1 37142,N1(C(C(CC=C)CC)=O)CCC2(CCC2NC(c2nncn2CC)=O)CC1 37143,N1(C(c2c(C)ccs2)=O)CCCC(CN(C(=O)Cn2nnc(=O)[nH]2)C)C1 37144,N1(C(=O)CCc2ncccn2)CCN(C(=O)CC2CCCC2(F)F)CC1 37145,C12(C(=O)NC(CNC(C3CC(C)(CC)C3)=O)C3CC3)CCCCC(=O)N1CCC2 37146,c1(C(N(CCC(C)NC(=O)Cc2c[nH]nc2O)C)=O)cc(F)c(Cl)cc1F 37147,c1(N2CCC(C)(NC(c3ccc(C)cn3)=O)C2)ccc([N+](=O)[O-])c(OC(F)F)c1 37148,Cc1ccc(C(=O)N(C)CCNC(=O)CC2CCOC2=O)cc1OC(F)(F)F 37149,C1(CCC)(C(=O)OC)CCCN1C(COC)COC 37150,c1(NC(C)=O)cnccc1C(=O)NC1(C)CC(C(N2CCC2CO)=O)C1 37151,c1(CC(=O)N(CCN(C(C2C(C(=O)OC)CCO2)=O)C)C)ccccc1CO 37152,Cn1c(CCc2cn(CC(F)(F)CNC(=O)CC3CC3(Cl)Cl)nn2)nnc1S 37153,C(=O)(C(CCC1CC1)NC(=O)OC(C)(C)C)NC(C)CCC1CCCC1 37154,N1(C(CSCCC)=O)CC(COCc2cn(C3CCCCC3)nn2)OC(C)(C)C1 37155,N1(C(C=C(C)C)=O)CCCOC(CNC(=O)CC2COC(=O)C2)C1 37156,c1(NC(C(N2C(C)CC2)=O)=O)ccc(C(=O)OC(C2COCCO2)C2CC2)cc1 37157,C1(C(N2CCC(CCN(C(COC(C)=O)=O)C)CC2)=O)CCC(C)=C(C)C1 37158,c1(C(=O)NCC(CNC(C2C(C)=CCS2)=O)(C)F)cc(N)c(O)c(F)c1 37159,c1(OC)ccc2ccccc2c1C(=O)Nc1cc(-c2ccnc(F)c2)ccc1Cl 37160,C(CCCC(=O)NC1CCC(CNC(=O)CCNC(=O)CO)CC1)N(C(C)=O)C 37161,CC(C)CC(CNC(=O)CC1CC2(CC2)C1)NC(C1CCCCC2CC12)=O 37162,C(CCCCCC(=O)NOCCC(F)(F)F)NC(c1c(C)nccc1)=O 37163,O=C1CC(C(N2CCC(OCCO)C2)=O)N(C(C2CCCC2F)=O)C1 37164,N1(C(Cc2cn(CC)nn2)=O)CC(NC(=O)CSC(C)(C)C)C(C(=O)OC)C1 37165,C(N=c1nc(C)cn[nH]1)C1(O)CN(C(C(C(CC)O)C)=O)C1 37166,c1(NCC)cncc(NC(=O)C(F)CC2CN(c3cc(OCC)ncn3)C2)c1 37167,C1(OCC)CCCN(C(=O)CN(C(c2cnn(C)c2N)=O)CC2CC2)C1 37168,c1(C(=O)NC2(CC(=O)NCC3N=C(C)SC3)CCC2)cc(C#N)ccc1C 37169,c1(COc2cccc(CCNC3C(C)CCC3C)c2)cc(F)cc(F)c1 37170,Cc1ncnc(NCCCCNC(=O)CCCC2CCCCC2)c1C#N 37171,C(=O)(C(CC(C)C)NC(C)=O)NC1(CO)CN(C(c2ccc(OC)nc2)=O)C1 37172,N1(C(C(C)OC)=O)CC2(CCC(CNC(=O)CCCNC(c3ccco3)=O)O2)C1 37173,N1(C(c2cc3cc[nH]c3cn2)=O)CC2CN(C(C3CCCCCC3)=O)CC2C1 37174,C1(C(=O)NCC=C(C)C)CN(OC(=O)Cc2[nH]cc(C)c(=O)c2C)C2(CCOC2)C1 37175,N1(C(C2ON=C(CC)C2)=O)CCC2(CC1)CN(C(=O)CN(C(=O)C(C)C)C)CCO2 37176,C(=O)(C1=CCCC1(C)C)NCCOC1CCN(C(C2CCN(OC)CC2)=O)C1 37177,C1(C(N(CC(C)(C)NC(c2cc(OCC)n[nH]2)=O)C)=O)C(O)C(=O)N(C)C1C 37178,C1(C)(C(=O)NC2C(OC)CN(C(C3CSCCS3)=O)C2)Cc2ccccc2N1 37179,c1(C(N2C3CCC2CN(C(C2CC(O)C2)=O)C3)=O)cccc(S(=O)(=O)CF)c1 37180,c1(C(=O)NC(C(C)NC(C2(F)CC(C(=O)OCC)C2)=O)C)ccc(F)cc1 37181,CC(C)CC(O)C(=O)NCCC(C)N(C(=O)CCc1nc(C2CCCC2)no1)C 37182,N1(C(CCCOC(C)=O)=O)CCCC(C2CCN(C(=O)CC(C)F)CC2)CCC1 37183,Cc1nc(C(N2CC(O)(C(C)NC(C3(Br)CC3(F)F)=O)C2)=O)c(C)n1C 37184,N1(C(c2c(Cl)ccc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C(N)=O 37185,C1(C(=O)NC2C(CC(=O)N(CCOCCCOC)C)CCC2)NC(=O)OC1(C)C 37186,N1(C(C(c2cc(C)on2)(C)NC(C2CCS2(=O)=O)=O)=O)CCC(N)C(C)(C)C1 37187,C1(C(=O)NC2CC(=O)N(c3ccccc3OC)C2)(COC)CCN(C(C)=O)CC1 37188,C1(N(C(C=C(C)C)=O)C)CCC(N(C)C(C2CCCN2CCC(C)C)=O)CC1 37189,C1(NC(c2cncc(-c3ccc(Cl)cc3)c2)=O)CCC(O)(c2cnc[nH]2)CC1 37190,N(C1c2ccccc2OCC1F)C(CC1N(C)CCOC1)=O 37191,CCCCCCCN=c1nc(N2CCC(C(N)=O)(OC)C2)c2c([nH]1)COC2 37192,C12(C(N(C)CC3CN(c4cc(C(F)F)ncn4)C3)=O)CCC(O)(CC1)CC2 37193,N1(C(C23CC(NCc4ccn(-c5ccccc5)n4)(C2)C3)=O)CCc2n[nH]cc2C1 37194,C(C(CNC(c1cc(O)cs1)=O)C(F)(F)F)NC(c1ccc(CCO)cc1)=O 37195,N1(C(c2cc(C)cc(N)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37196,N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC1C(C)(C)C1 37197,c1(CN(CC(=O)O)C)cccc(NC(Cn2cc(C(C)OCC)nn2)=O)c1 37198,C1(OC)CN(C(c2cn(C)nc2C)=O)CC1NC(c1ccccc1O)=O 37199,C1(NC(C2CC3(CCC3)CO2)=O)CCC2CN(C(=O)CCN3CCCC3=O)CC12 37200,CC1CN(C(C2CCC(N(C)C)CC2)=O)CCN1Cc1cccc(C#N)n1 37201,Cc1ccc(C(=O)NCC2CC(NC(=O)CC3COCCO3)C2)cc1C 37202,N1(C(C(C2CCCC2N(C)C)C)=O)CCC(NC(C2CCOCC2)=O)C(C)(C)C1 37203,C1(NC(c2cncc(OC(C)C)c2)=O)CC2CCC1CN(C(=O)COCC(F)F)C2 37204,N1(C(c2n(C)c(Cl)cn2)=O)CCCOC(CCNC(C2CC(=O)C2)=O)C1 37205,N1(C(C2CCCC(C(=O)OC)C2)=O)CCCC12CCN(C(C1CCCSC1)=O)C2 37206,c1(OC)c(C(=O)NC(C2CCCN2C(c2ncccc2O)=O)C)c(C)nn1C 37207,c1(C(N2CC(CCNC(C3(OC)CC3)=O)(OC)C2)=O)cn2ccnc2s1 37208,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37209,C1(CNC(CC=C=C)=O)CCN(C(C2(C(C)C)CC2)=O)CC1(F)F 37210,C(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1C(NC(c2c(OC)nn(C)c2)=O)CCC1 37211,CCCCC(O)C(=O)N1CCCC(NC(c2ccc(C3CC3)cn2)=O)CC1 37212,N1(C(C(c2ccc(C)o2)C)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 37213,C12CCOCCN1N1CC(OC1)O2.C1CC1 37214,C=CCC(CC)C(=O)N1CCC(n2cccn2)(C(=O)Nc2csc(C#N)c2)CC1 37215,CCC(C)C=CC(=O)N(CC(=O)NCCCNC(=O)C1CC1)C(C)(C)C 37216,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC1CN(C(C2(C3CC(F)(F)C3)CCC2)=O)C1 37217,Cc1nc(C(=O)NC(C(=O)NOC(C)C(F)(F)F)c2ccco2)ccc1C#N 37218,c1(CC)ccc2ccccc2c1CNC(=S)NCC1CCCO1 37219,CCCCC(COC)(c1nnnn1-c1cccc(F)c1)NCc1cncc(C)c1 37220,N1(C(C2C(CNC(c3ccoc3C3CC3)=O)C2)=O)CC(F)(F)C(F)(F)C1 37221,C1(NC(C=CC(CC)=CC)=O)COCC1NC(c1n[nH]cc1Cl)=O 37222,CC(C)C1=NOC(C)(C(N2CCC(C)(CNC(=O)C=C(C3CC3)C3CC3)C2)=O)C1 37223,N1(C(C2(CSC)CCC2)=O)CC(OC)C(NC(C2CCCS2)=O)C1 37224,c1(CCC(N2CCC(CO)(NC(C3CC(O)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 37225,C(=O)(CC(F)(F)C(F)F)NCC1C(NC(C(C)(C)C(F)F)=O)COC1 37226,C1(NC(COc2ccn(C)n2)=O)CC(F)CN(C(=O)Cn2cnc(=N)[nH]2)C1 37227,N1(C(c2cccc(SC)c2)=O)CCCC(NC(C2C3CCC2CC3)=O)CC1 37228,C(C(C(=O)NCC1CC(F)(F)C1)C(C)(C)C)NC(C1C(C(=O)OC)C=C1)=O 37229,CN1CCN(C(=O)CC2CN(C(=O)CC3COCC(C)(C)O3)CCO2)C(CO)C1 37230,c1(Cc2occ(CNC(C(C3CCCO3)N(CC)CC)=O)n2)ccc(Cl)cc1 37231,C1(C(=O)NC(C(=O)NCCC)CC)CC(C)(C)CCN1C(=O)Cn1cnnn1 37232,C(=O)(CCCc1cncs1)N(CC(CC)NC(=O)Cc1cscn1)CC 37233,C1(C)(CC)CN(C(c2ccccc2C#N)=O)CCO1 37234,c1(C(=O)NCC2N(C(CN3C(C)CC3)=O)CC(O)C2O)cn2c(n1)COCC2 37235,C1(CNC(=O)Cc2ccco2)CC(C(F)(F)F)CN1C(C1CC(C2CC2)C1)=O 37236,c1(-c2cc(C(N3CC(NC(C(CC)F)=O)C3)=O)on2)c(F)cccc1F 37237,Cc1nccc(C(N2CCCC2C2CCCN(C(=O)CC3(CO)CC3)C2)=O)c1C 37238,N1(C(CN(CC(=O)NCC2CC2)C)=O)CC(C)(C(=O)NCCN=[N+]=[N-])CC1(C)C 37239,c1(C(=O)NC(CCNC(c2c(C)c(CO)ccc2)=O)C)noc2ncccc12 37240,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37241,c1(C(=O)NC2(C(=O)NC(c3ccnc(C)n3)C)CCOCC2)cc(O)nc(C)n1 37242,c1(CCC(=O)NCCCN(C(c2sccc2C)=O)CC)ccccc1Br 37243,CC(C(=O)N1CC(O)(CNC(C2CCC(=O)NC2)=O)C1)S(=O)(=O)C1CCOCC1 37244,C(C(C(C)(C)C)NC(=O)C(O)C1CCC1)NC(C=C(C)C(F)F)=O 37245,c1(C(C(=O)N(CC(C)C)C)NC(=O)CC2CC2(C)C)cccnc1 37246,CCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(c1c(C)nn(C)c1C)C)C1CC1 37247,CC1(CC(N2CCOC(CNC(=O)CSCc3ncc[nH]3)C2)=O)CCS(=O)(=O)N1 37248,O=C(C1CCc2nccn21)NCCC1CN(C(c2ncc3c(F)cccn23)=O)C1 37249,c1(N2CC(C)CC(C)(C)C2)nc(Cl)nc2cc(C(C)(C)C)sc12 37250,c1(C(C(=O)NC2COC2)N(CC(=O)OCC)Cc2ccccc2C)cc(F)cc(F)c1 37251,c1(C(COC)NC2CCNC2=O)cccc(Cl)c1Br 37252,C(=O)(CCCCCS(N)(=O)=O)NC1CCCCN(C(CCc2c[nH]c(=N)s2)=O)C1 37253,c1(C(=O)NC(C(CC)C)CO)cc(C#N)ccc1NC(=O)Nc1cnn(C)c1 37254,CCCC(C(=O)NCC1(O)CCCN(C(=O)C#CC2CCC2)CC1)S(N)(=O)=O 37255,C(C(CCC(=O)N1CCC(N(C(=O)CCS(N)(=O)=O)C)C1)OC)OCC 37256,c1(CCNC(c2n(C(C)C)nnn2)c2csc(-c3ccsc3)n2)ncccc1F 37257,c1(CC(=O)NCC2C(NC(C(C)OCCC=C)=O)CCC2)cn2ccccc2n1 37258,c1(NC(=O)NC2CN(c3cccc(CC)c3)C(=O)C2)nc2c(O)ncnc2s1 37259,c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)nc2ccccc2o1 37260,N1(C(c2c(OC)cncn2)=O)CCC2(CC1)CN(C(=O)CC(C)(C)O)C2 37261,N1(C(CC(C)SC)=O)CCOCC(CNC(c2coc(N(C)C)n2)=O)C1 37262,N1(C(CCC(C)=O)=O)CCC(O)C(C(=O)Nc2cc(CO)cc(F)c2)C1 37263,N1(C(C(C)O)=O)C2CCC1CC(NC(C13CC4CC1C3C4O)=O)C2 37264,c1(COC)nccc(=NC2(C)CC(NC(c3cccn4c(O)nnc34)=O)C2)[nH]1 37265,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)CC3CCCC3C)(C1)C2 37266,C(C(CNC(=O)CCc1ccon1)C(F)(F)F)NC(C1C=CC=CC=C1)=O 37267,C(C(=O)N=S(C)(=O)c1cnn2c1CN(C(C1CCC(CC)C1)=O)CC2)=CC 37268,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)(C)CC(F)(F)F)C2)n1 37269,N1(C(C(CC)OC)=O)CCCC(CC(=O)NC(C2(OC(C)C)CCC2)C)CC1 37270,CN=S(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2cnco2)=O)cc1 37271,CC1CN(C(C2(F)CCN(C(=O)CN(C)C)C2)=O)CC2(CCC2)O1 37272,Cc1cnc(F)cc1C(N1CC(NC(=O)C(F)CC2CCOC2)C(O)C1)=O 37273,N1(C(c2cccc(C)n2)=O)CCC(C)(C)C(NC(=O)C(C)NC(c2ccco2)=O)C1 37274,C1(C(=O)NCCNC(C)(C)C)CC2C(C(=O)NC3(C(CCC)=O)CC3)C2C1 37275,CC1(C)CC(NS(=O)(=O)N2CCCC2c2ccccc2)CN(S(N)(=O)=O)C1 37276,c1(CC)c(NC(=O)C(CCNC(c2cncn2C)=O)OC)cnn1CC 37277,C1(N(C2CC3(CNC3)C2)C(c2ccc(C(F)(F)F)cc2)=O)CCCCCC1O 37278,N(C1CCCc2cc(F)ccc21)Cc1ccc(O)c(Br)c1.N12CCC(F)(C1)C2 37279,c1(C(=O)NC(CNC(c2c(C)cc(F)s2)=O)(C)CC)cccc(F)c1N 37280,C1(CNC(c2c(C)scc2)=O)CCC(C)(C)CN1C(C1CN(C(C)C)C1)=O 37281,C1(C)CCC2CN(C(=O)COC(F)F)CCC2C1.C1CC1C(=O)OCC 37282,c1(C(=O)NC2C(CNC(C(C)CN3CCCC3)=O)C2)ccc(C(F)(F)F)cn1 37283,C1(C(=O)NC(CNC(C2C(CCC)C2)=O)C)OCC2CCCC12 37284,CCC(CCOC)C(=O)NCCCOCCN(C(=O)C(C)(C)n1cccn1)C 37285,CC1(C)CCCC(N2CCCC(Oc3ccc(C#N)cc3)C2)C1 37286,CCC(CC1CCCC1)C(=O)NCC1CN(C(C2CC2C(C)(C)C)=O)C1 37287,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37288,C1(C(=O)NCCNC(CCCSC)=O)CCCN(C(c2cnnc(Cl)c2)=O)C1 37289,N1(C(c2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc[nH]c2)CC12CCCCCC2 37290,CCC(C)(CN)C(=O)NC1CCN(C(c2cc(-c3cc(F)ccc3F)on2)=O)C1 37291,C(=O)(C(CN(C)C)C(C)C)NC(CC1CN(C(c2nc(CC)sc2)=O)C1)C 37292,C12(C(N3CC(C(C)NC(C(CC)(C)OC)=O)C3)=O)CCCC1C2(F)F 37293,CC1(C)CCCC(CC(=O)NCCC2=CCN(CCOCC3CC3)CC2)CC1 37294,c1(C(=O)NCC2(F)CC(NC(C(C)C(C)O)=O)C2)cnc(O)c2ncccc12 37295,c1(NC2CC(NC(=O)NCCC3CCC(C)O3)C2)ncccc1Cl 37296,CCCC(CCCNC(=O)COCCF)NC(=O)CCCN(CCO)C.[SH](=O)(=O)CC 37297,C(CS(=O)(=O)c1cccs1)NC(=O)NC(CC=CC)C(=O)OC(C)(C)C 37298,c1(C(N2C3CC(NC(C(C)CN(C)C)=O)C3CC2)=O)cccc2c1nnn2C 37299,N1(C(C=CC(C)(C)C)=O)CCC1CNC(C1(C2CC2)CC1)=O 37300,C(C(CCCC)NC(C12COC(CF)(C1)C2)=O)NC(CSCC=C)=O 37301,C=CCC(F)(F)C(=O)NC1CCCC(N(C)C(c2ncncc2N)=O)C1 37302,CCC(C)C(C(=O)NC1CC(C(N)=O)(CC)C1)NC(=O)CC1(OC)CCC1 37303,C1(C(=O)OC)C(NCC(O)S(=O)(=O)C2CC2)C2(C)CCCCC12 37304,c1(C(N(C)CC2(NC(CSCCC)=O)CC2)=O)cc(C2CC2)on1 37305,c1(C(N(C2CCN(C(=O)CCC(C)(F)F)C2)CC)=O)c(C)cc(O)nc1C 37306,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C)ccccc1C1(C#N)CC1 37307,C=CC1CCN(C(C2(CNC(=O)C(F)F)CC(=C)C2)=O)C1 37308,C1(O)(CC(=O)NCC2C3CN(C(CCC(=C)Cl)=O)CC32)CCCCCC1 37309,C1(NC(c2cncc(CC)c2)=O)CN(C(=O)C=C(C)C)CC12CCC2 37310,C1(OC)CC(CNC(c2cc(C)nn2C2CC2)=O)N(C(c2cc(C)ccn2)=O)C1 37311,c1(OC)ccc(C(=O)OC2CC23CC(OCc2ccccc2)C3)c(Cl)n1 37312,c1(C(N(C2CCN(C(c3c(CC)scn3)=O)C2)CC)=O)cc2c(cc1N)OCO2 37313,c1(CC(N2CCC(CC=C)(NC(=O)C(O)CF)C2)=O)cn2cc(F)ccc2n1 37314,c1(CC(=O)OCCN(C(=O)C(CCN(C)C)SC)CCC)ccc(OC)cc1C 37315,C1(C(=O)NCC2OCCCN(C(CC3CNC(=O)N3)=O)C2)Cc2cncn2C(=O)N1 37316,C#Cc1ccc(C(=O)N(CCC(N2CC3CC(O)C3C2)=O)CC(=C)C)cc1 37317,C(=O)(C(C)(CC)CC)N(CC(CNC(C(CCC)=CCC)=O)O)C 37318,C(=O)(C(F)C(F)(F)F)NC(C(n1cc(-c2c(OC)nn(C)c2)nn1)C)=O 37319,FC1(F)C2CCC1(n1cc(N3CC4CC3C4c3cccc(Br)c3)nn1)CC2 37320,CC1CN(C(=NCCCOc2ccc(C#N)cc2)NCCCCl)CC1(C)C1CC1 37321,C1(F)(CNC(C(C)OC(C)C)=O)CCC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 37322,c1(CNC(C(=O)OC(C)(C)C)CCc2ccncc2)cnc2cccc(Br)n12 37323,CC1OC23CC1(C2)NC3.C1(C)(CNC(c2cncc(F)c2)=O)CCCC(=O)N1 37324,N1(C(CCOCCOC)=O)CCCC(CCNC(=O)CC2CCC(=O)N2)C1 37325,c1(OC)ccc(C(=O)C(N2CC3CC3C2c2cccs2)C)cc1OC 37326,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)NCCN1CCOC1 37327,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37328,C(=O)(CS(=O)(=O)C1CCCC1)NCCOCCN(C(C(C)CF)=O)C 37329,Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CC(NC(c2c(C)sc(C)c2C#N)=O)C1 37330,N1(C(C=Cc2n(C)ncc2)=O)CCC2(CC1)CCN(C(c1cncnc1)=O)C2 37331,c1(C(=O)NC2CN(C(C(C(=O)OCC)CC)=O)C2)cc(=O)n(C)c2ccccc12 37332,c1(CNC(c2ccc(F)nc2F)=O)c(Cl)cncc1Cl.C12CC3(C1)CN(C3)C2=O 37333,C1(CNC(C(N2CC(O)(SC)C2)=O)=O)CC(Cl)=CC=N1 37334,Cc1cc(C(=O)N(CC(C)N(C)C(c2cnsc2)=O)C)nc(C)c1 37335,C1(C(N2CC(OC(=O)NCC)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1(F)F 37336,C(=O)(C1=CC2C=CC1C2)NCC(CNC(=O)C(C)(C)C1(O)CCC1)OC 37337,Cc1cc(C(=O)NCCN(C(=O)C(F)C(C)C)C(C)C)cc(C)c1Cl 37338,c1(OC)nccc(C(=O)NCC2(NC(C3OCCC3(C)C)=O)CCCCC2)n1 37339,C1(C(N(C2CCN(C(c3nc(Cl)cs3)=O)C2)CC)=O)CCC(C)(C)O1 37340,CCC(C(=O)NC1CC(CNC(c2c[nH]nc2C(C)C)=O)C(O)C1)C(C)C 37341,C1(C(N2CC(CC)(OC)C2)=O)CN(C(=O)CC(O)C2CCCC2)CC1(F)F 37342,c1(C(C(=O)NC(C)C)N(CCCC2CCCO2)C2CCC2)ccc(Br)s1 37343,C1(CNC(C2N(CC)CCC2)=O)CN(C(c2ccn(C)n2)=O)CCC12CCC2 37344,c1(CC(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)cnc2ccccc2c1 37345,c1(OC)cc(C)c(F)cc1-c1cnc(C(=O)Nc2c(Cl)c(C)nn2C)cc1C 37346,c1(C2NC(c3n(C(CC)CC)ncn3)C2)ccc(C#N)cc1F.C1(N)CC1 37347,Cc1nc(=N)[nH]c(C)c1C(=O)NCCCNC(C1OC(C)CC1C)=O 37348,N1(C(C2N(C(=O)C=CCN3CCCC3)CCC(=C)C2)=O)CCC(C)C(C)(C)C1 37349,CC1=C(C(=O)NC2CC3CC2CN3C(C2CC2C)=O)CCCO1 37350,C(CN=c1[nH]c(=NC2CC3CCCCC23)c2ncccc2[nH]1)N1CCC(C)C1 37351,N1(C(C2CC3(CC(=C)C3)C2)=O)CC2CCCC(C1)N2C(C1(C)CCC12CCC2)=O 37352,c1(C(N(CCNC(C(C=C)O)=O)CC2CC2)=O)cc(C)sc1Br 37353,C=CC1(CO)CCN(c2ncnc(NCC(c3cc(C)ccc3C)O)c2C)CC1 37354,c1(OC(C)C)nccc(C(=O)NC2CCCCN(C(C3(CF)CCC3)=O)C2)c1F 37355,c1(C(=O)NCC2CC(CNC(c3ccn(C(C)(C)C)n3)=O)C2)cc(CO)ccn1 37356,C(=O)(CCCCCn1cnnn1)NC1CCCN(Cc2nc(C)[nH]n2)C1 37357,c1(C(=O)NC(C)CN(C)C(c2ccncn2)=O)cnccc1N1CCCC1 37358,c1(C(=O)NC2C=CC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37359,c1(C(N2CC(C#C)(CNC(C3(C(=O)NC(C)C)CC3)=O)C2)=O)ccc2ccoc2c1 37360,c1(OC)ccc(C(C)N(C(=O)C(COC)N(C)C)C)c(C)c1.N12CCCC1C2=O 37361,c1(CN(N2CCC(C(CC)C)CC2)C)ccc(Br)c(OC)c1 37362,N1(C(C(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cc3cc[nH]c(=O)c3o2)=O)C1 37363,O=C(CCN=c1[nH]c(=NCCF)[nH]c2c1COC2)N1CCOCC1 37364,C(=O)(C1CCC(N)c2ccccc21)N(C)CC1CCCN(Cc2ccccc2)C1 37365,C1(C(=O)NC2CC(C(=O)NCc3c(C)occ3)C2)CCC2(CCC2)C1 37366,N1(C(CCN(CC)CC)=O)CCN(C(=O)CSCc2ccccc2)C2CC12 37367,N1(C(C(=O)Nc2ccc(C)cc2Br)C)CCC(C2CC(O)C2)CC1 37368,N1(C(CC(C)N(C)C)=O)CCC2(CCCN2C(C2CCOC2)=O)C1 37369,C1(N(C(=O)C=CC2CC2)C)CN(C(C2CCN(CC(F)F)C2)=O)CC12CC2 37370,CC1(C)CCC=C(C(=O)NCCC2CN(C(C3CCCS3)=O)C2)C1 37371,c1(CC(N2CC3CC3(CNC(C3CCC(C(F)(F)F)C3)=O)C2)=O)cccc(F)c1O 37372,N1(C(c2cncc(NC(CC)=O)c2)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37373,c1(COC)nccc(CNC(=O)NC2(CO)CCCOC2)n1 37374,C(=O)(C#CC1CCOCC1)NC(CNC(c1cc(C)n(C)c(=O)c1)=O)C1CCC1 37375,CCCCC(O)C(=O)N1CCC(C)(C(=O)Nc2nc(F)ccc2Br)C1 37376,N1(C(CC2(C)CC2(F)F)=O)CC2(CCN(C(C3(C)CNC(=O)C3)=O)C2)C1 37377,c1(NC(c2cccs2)C)[nH]c(=NCC2CC2C2CCOCC2)nc2scnc12 37378,N1(C(c2ccc(OC)nc2)=O)CCC2(COC(CNC(=O)CC(C)C3CC3)C2)C1 37379,C1(C)(CC(=O)NC2C(CC)N(C(=O)CN3C(=O)CNC3=O)CC2)CCS(=O)(=O)N1 37380,C#CCCCCCCC(=O)N(CCCCCC(=O)NCc1cn(C)cn1)C 37381,c1(C(C(N2CCCC(Cc3ccnn3C)C2)C)=O)ccc(F)c(F)c1 37382,c1(COCC)cccc(F)c1NC(=O)NCC1(C)CCCC(OC)C1 37383,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37384,N1(C(C(c2ccccc2F)C)=O)CCCC(C2CN(C(C3CC34CCC4)=O)C2)C1 37385,c1(C(=O)NCc2c(C(=O)NCc3n(C)ccn3)nco2)ccc(I)c(O)c1 37386,C1(NCc2ncc(C)cc2Br)C2CCC1CN(C(c1nc(CC)c(Br)s1)=O)C2 37387,C(CC(F)F)(C(=O)NOCCSCCC=C)NC(=O)CC(C)(C)C 37388,c1(C(=O)NC2CC(SCC)C2)cccc2occc12 37389,N1(C(CCC2(C)CCCN2C(c2ccsn2)=O)=O)CC(O)C(O)CC12CCC2 37390,c1(OCC(CC)OC)cc(OCCOC)ccc1C(C)(C)C 37391,c1(CCC(=O)NCC2CCCC2NC(C2CCOCC2)=O)c[nH]c2ccccc12 37392,C1(CC(=O)N(CCCOC)CC(C)C)CCCN(Cc2cccc(CO)n2)CC1 37393,c1(OCC)ccc(C(N2CCOC(CCNC(=O)C=CCOC)C2)=O)cc1OC 37394,c1(C(=O)NCC2(C)CN(C(C3CN(C)C(=O)CC3)=O)C2)cc(Cl)c(N)c(Cl)c1 37395,C(=O)(CCCN=c1nccc[nH]1)NCCC(C)NC(=O)C1=CCOCC1 37396,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(O)C(C)(C)C)CC2)cc1F 37397,n1(C(C)C)cc(Sc2cc(C3N(C(=O)N(C)C)CCC3)n[nH]2)c(I)n1 37398,N1(C(=O)NC)CCN(C(c2ccc(Oc3nc(C(C)(C)C)cs3)o2)=O)CC1 37399,O=C1OCc2cc(C(=O)NCC3CC34CC4(F)F)ccc21 37400,N1(C(c2cccc(F)c2)=O)CCN(C(=O)CC2OCCCO2)C2CC12 37401,n1(CC=CC)c(C(=O)CC)nc2ccccc12.C12CCCC1n1cc(nn1)CN2 37402,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)C(=O)NCC1CC1)CC2CO 37403,c1(S)cccc2ccccc12.C=CCC(C)(C)C(=O)NCCN1C(=O)C(C)S1 37404,CS(=O)(=O)c1nccc(N2CCCCC2CNc2cc3ccccc3s2)n1 37405,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37406,Cc1ccc([N+](=O)[O-])c(CN=C(NCC(c2cccs2)OC)NCC2CC2(C)C)c1 37407,c1(CC)c(C(N2CCC(C)C2C(=O)NC2(C)CC(C(N)=O)C2)=O)ccn1C 37408,c1(Nc2cc(OCCOC)cc(Br)c2)ncc2ccccc2n1 37409,N(C1CCCn2ccnc21)C(C1(C)CCCN1C(=O)Cc1ccc(O)cn1)=O 37410,c1(C(=O)NC2C(CNC(C(CC)(C)CO)=O)CCC2)noc(C)c1[N+](=O)[O-] 37411,C1(NC(C2(CN(C)CC)COC2)=O)CCC(CCNC(c2cc(CO)on2)=O)C1 37412,C(=O)(CCCC(=O)c1ccccc1N)NCC(CCCCN)OC 37413,CCCC(O)CC(=O)N1CC(CNC(c2ccn(C)c2C2CCC2)=O)C(C)(C)C1 37414,O=C1NCCn2ncc(C(N3CC(C(=O)NCC4CC4)CC(F)C3)=O)c21 37415,C1(NC(C2(c3ccccc3)CC2)=O)CC2(C1)CC(NCc1ccnn1CCCO)C2 37416,S(=O)(=O)(c1ccc(N2CCSC2)c(F)c1)N1C(C)SC(C)C2=C(C1)CC(=O)N2C 37417,C12(CNC(CC(CCC)O)=O)CCCCC1CN(C(c1cnn(CC)c1C)=O)C2 37418,C1(C(=O)O)(OC)CCC(C)C1.c12nc(co1)C(=O)NC1CC(C1)C(=O)NC2 37419,c1(C(C)NC(c2cn(CCCF)nn2)=O)c(Cl)ccc2ccccc12 37420,C(C1CNC1=O)C(C1COCC1O)=O.C(C(=O)NCCl)N(C)C(N)=O 37421,Nc1cc(F)cnc1C(=O)NCCC1CN(C(=O)CC2CCCNC2=O)C1 37422,C(=O)(CC(CC#N)c1ccccc1)NC1C2CN(C(c3n(CC)cc(Cl)c3)=O)CC21 37423,c1(C(=O)NC(c2ccc(C)cn2)C(C)C)cc2c(C)sc(C)c2s1 37424,C1(n2cc(C(=O)OC)nn2)CCC(C(=O)NCCCOC(C)(C)C)CC1 37425,CCC(C)(C(=O)N1CC(NC(=O)Cc2ncc(C)s2)C(F)C1)C(F)F 37426,c1(C(=O)NC2C(C)CCN(C(=O)CC3CCCS3(=O)=O)C2)ccc(N=[N+]=[N-])cc1 37427,C1(C(=O)N)COC2(CCC2)CO1.N1(C(C2C(C)C2)=O)CCC(OCCOC)CC1 37428,c1(C(N2CC(O)(CNCc3cncc(C(=O)O)c3)C2)=O)cnn2ccncc12 37429,c1(C(N2CCC(NC(C3(Cl)C(C)(C)C3)=O)C2)=O)cnc(S)nc1 37430,c1(C(=O)NCC(CNC(=O)C(C)(CO)N(C)C)OC)cc(Cl)nnc1O 37431,C(C(C(C)C)NC(C12CC(CO1)C2)=O)NC(C)=O 37432,c1(OC)cc(C)c(OCCNC(=O)Cn2cc(Cl)c(C)n2)c(C)c1 37433,c1(CNC(C2CC(CC)C2)=O)nc(C(=O)N(CCCN=[N+]=[N-])C)c(C)o1 37434,c1(CC)ccc2cc(NC(N3CCC(SC)CC3C)=O)ccc2c1 37435,CC(CN=C1NCC2CN(N1)CCC2O)C(F)(F)F.[SH](C)(=O)=O 37436,c1(C(C(=O)NC(C)Cn2cc(-c3sccc3Cl)nn2)=O)ccc(O)cc1 37437,C(=O)(CCC(C)(C)NC(=O)Cn1cc(Cl)cn1)NC(c1nc(C)[nH]n1)CO 37438,c1(C(N2CCN(C(CSCCOC)=O)C3C2C3)=O)ccc2occc2c1 37439,N1(C(c2c(F)ncc(-c3cccc(C#N)c3)c2)=O)CCC2(CC1)CC(=O)NC2=O 37440,Cc1cscc1C(N1CCC(C(C)NC(C2(C)CC2C)=O)C1)=O 37441,N1(C(c2c(C)onc2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37442,c1([SH](CC(=O)NCCN(C(c2nncn2C2CC2)=O)CC)C(C)(C)C)ccccc1 37443,c1(OC)nc(N2CCCC(C)(NC(=O)CCCCCCBr)C2)nc2[nH]cnc12 37444,C1(C(N2CC(OCCO)C2)=O)COCCN(C(c2cccc(O)n2)=O)C1 37445,C1(C(N2CC(N3CCN(C(c4nn(C)c(O)c4)=O)CC3)C2)=O)CC2(CCCC2)C1 37446,c1(CNC(C2CC(C)(C(C)(C)C)C2)=O)ccc(Br)cc1N1CCNCC1 37447,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37448,C1(NC(CN(CCC)C)=O)CCCC(CNC(=O)C(C(C)CC)OC)CC1 37449,C(C(C)(F)CNC(=O)C(c1cccnc1)O)NC(CC1C(C)(C)C1)=O 37450,C1(NC(C=CC)=O)CS(=O)(=O)CC1N(C(c1cnc(-c2cccc(Br)c2)s1)=O)CC 37451,c1(C(=O)NC(C2CN(C(c3ccnn3C3CC3)=O)C2)C)conc1C1CC1 37452,c1(C(=O)NCC(C2CC2)NC(C2CC(C)(F)C2)=O)cc(F)cc2cc[nH]c12 37453,O=C(C#CC1CCCC1)N(CCNC(C12CCCC1(C(N)=O)C2)=O)CC1CC1 37454,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(CNC(c1cc(C(N)=O)[nH]n1)=O)C2 37455,C(C(O)CNC(=O)CCN1C(=O)CC1)SC.c1(NC(C2CC2)=O)scnc1C 37456,n1(CCOC(N(CC(C(C)C)C(=O)NC(C)(C)C)C)=O)cc(-c2cc[nH]n2)nn1 37457,O=C(C1CSc2ccccc21)NC1CCN(c2nccc(-c3ccncc3)n2)C1 37458,C(C#Cc1cn(CCCCF)nn1)NC(C1C(COC)CC1)=O 37459,N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(C)C2CC2)CCC1C.n1(C)nnnc1C 37460,C(=O)(C(C)C(C)(C)C)NCC1(OC)CN(C(c2n(CC)c(O)nc2)=O)C1 37461,N1(C(CC(C)CF)=O)CC2CCC1C1CN(C(c3c(N)ccc(F)c3F)=O)CC21 37462,C1(N(C(C=NOC)=O)C)CCCC(NC(=O)CCc2cc[nH]n2)C1 37463,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(c1cnccn1)=O 37464,C1(NC(c2c(C)c(Br)ccc2F)=O)CCN(C(C)C(=O)N(C)C)CC12CCC2 37465,c1(C(=O)NC(CNC(CSCc2cccc(OC)c2)=O)(C)C)cc2[nH]ccc2s1 37466,C(C(=O)N)(C(C(C)C)OC)OC.C(C)(C(=O)N)N(CCCOCCOC)CC 37467,C1(C(=O)NCC(C)NC(C2CNC(=O)C2)=O)CS(=O)(=O)CC(=O)N1 37468,C(=O)(CC(C)CC(C)(C)C)NC(c1ccccc1)C(=O)NCCn1ncc(C)c1 37469,c1(OCC(F)(F)F)cccc(C(F)(F)F)c1-c1nc(CCCO)no1 37470,Cc1cccc2c(CCC(=O)N(C3CC(NC(=O)C(F)F)C3)C)c[nH]c12 37471,Cn1c(C(=O)NC(CNC(C2CCC(C(N)=O)O2)=O)C2CCC2)cccc1=O 37472,c1(C(=O)NCC2CN(C(CC(CC)C)=O)C(C)C2)cccc2nn(C)nc12 37473,C1(C(=O)NCC(CN(C(=O)C(C)CC(F)F)CC)(C)C)CCOC(=O)CC1 37474,N1(C(C(CCC)NC(C2CCOC2CC)=O)=O)CCC(C)(CC)CC1 37475,C1(C(N(C(CNC(=O)CC2CC2)C2CC2)C)=O)CCC(O)C1 37476,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37477,CC1(C)CC(C(=O)N2CC(CNC(CCC3CCC(C(=O)N(C)C)O3)=O)C2)=NO1 37478,C1(C(=O)NCC2CN(CC)C(=O)O2)CC(NC(=O)CC2CC(=O)C2)C12CCC2 37479,c1(C(N2CC(C(F)(F)F)C2)=O)cc(CCNC(C2CC2C(F)(F)F)=O)ncn1 37480,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37481,CCCCN=C(NCc1cc(OC)ccc1F)N1CCC(OC)C(C)(C)C1 37482,C1(S(N)(=O)=O)(C(N2CC(CC)C(NC(c3[nH]c(O)nc3C)=O)CC2)=O)CCCC1 37483,C=CCC(CNC(=O)CC=CCCCCC)C(=O)NC1(CCC)CCCCC1 37484,c1(NC(=O)COC(C2(c3cccs3)CC2C)=O)ccc(N2CCOCC2)cc1 37485,c1(C(=O)NC(CNC(c2ccc(C(C)O)cc2)=O)CO)c(Cl)cccc1[N+](=O)[O-] 37486,C(=O)(C1CSc2ccccc21)NC(C(C)NC(=O)CC(C)(C)C(F)(F)F)(C)C 37487,C(C)(N=c1[nH]c(=N)[nH]c(=NCc2nc(CO)cs2)[nH]1)C1(C)CC1Br 37488,N1(C(CSC)COc2ccccc2)CCOCC(C(=O)On2nc(C)cc2C)C1 37489,c1(C(=O)OCC(N2CC(C=CC)C2)=O)ccc2nc(O)n(C)c2c1.c12nscc1N2 37490,CN1CCN(C(c2ccccn2)=O)CC1C(=O)NCCC1CCOC1(C)C 37491,C(=O)(C(O)CC[S+](C)C)NCC1(F)CN(C(C(C)(C)OC(C)C)=O)C1 37492,CN=c1nc(C(N2CCCC(CNC(=O)CSc3ccccn3)C2)=O)cc(C)[nH]1 37493,C1(CNC(C2(SC)CC(F)C2)=O)CN(C)CCN1C(c1ccc(C)nc1N)=O 37494,Cc1oc(C(N2CC3(CC3C(=O)Nc3ccccc3)C2)=O)cc1C(N)=O 37495,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(C(n1cnnc1O)C)=O 37496,C1(NC(C(C)(CO)OC)=O)C2CC3C1C3C2C(N1CC(N2CCCCC2)C1)=O 37497,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37498,c1(C(N2C3CN(C(C(C)OC)=O)C(CC3)C2)=O)ccc(S(C)=O)cc1[N+](=O)[O-] 37499,C(=O)(C(O)C(F)(F)F)N1C(C2CCN(C(Cn3cc(C(C)=O)nn3)=O)C2)CCC1 37500,C(c1ccc(F)cc1)=C(C)C(N1CCCN(C(=O)CC(O)C2CCCC2)CC1)=O 37501,c1(-c2c(CNC(C3CCCCC3C#N)=O)cn(C)n2)cccc(S(N)(=O)=O)c1 37502,C1(CNC(c2c(OC)c(Cl)c(Cl)s2)=O)CCN(C(C2CC2F)=O)C12CCC2 37503,C12CCCC13CCN(C3)C2=O.c1(SCc2ccc(C)nc2)cc(Cl)c(F)cc1F 37504,Cc1nc(C2CC2)sc1CC(=O)NC1CCCN(C(c2ocnc2C2CC2)=O)C1 37505,N1(C(CC=C)=O)CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C(C2CC2)C1 37506,C1(CNC(C2CN(C(C)=O)C2)=O)CCN(C(c2ncsc2-c2ccccn2)=O)C1 37507,N12CCC(CO)(C1)CNC2=O.c1(C(C)(C)C)cc(Cn2cccn2)cs1 37508,c1(C(C(=O)NCC2C(NC(c3cc(CO)[nH]n3)=O)C2)O)ccc(F)cc1 37509,C1(O)(c2cn(C(C(N3CC4(C(C(C)=O)CCS4)C3)=O)C)nn2)CCC(F)(F)CC1 37510,c1(C(N(CCN(C)C(c2cccnn2)=O)C)=O)c[nH]c2cc(Br)ccc12 37511,c1(OCC)nc(C(=O)NCC(C2CC2)NC(C2CCCO2)=O)co1 37512,c1(C(N(CCCNC(C2CC2C)=O)CCC)=O)cc2n(n1)CCN(C)C2 37513,c1(N2CCC(C#N)C2)nc(N2CCC(C3CCCCO3)CC2)c2c(n1)CCS2 37514,c1(C(C(=O)Nc2ccccc2)N(C(C)C)C)cccc(Cl)c1Br 37515,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37516,c1(C(N2CC(NC(C3(F)CCCC=C3F)=O)C2)=O)ccc2cc[nH]c2c1 37517,CCCC(CNC(=O)CC1CCCN1C)C(=O)NC(C)CSCC(=O)N(C)C 37518,Cc1ccc(CC(N2CCC(C)C(CNC(=O)C(C)(C)N(C)C)C2)=O)cc1O 37519,c1(NC(C2CCN(C(C3CCN(C)C3)=O)C2)=O)cc2c(F)cccc2[nH]1 37520,N1(C(C(C)=C2CC2)=O)CCC(CC(C)NC(=O)C(c2ncccc2F)(F)F)CC1 37521,c1(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)nccn2cnnc12 37522,N1(C(c2cc3ncc(C)n3cc2)=O)CC(C2CCCCN(C(=O)C3=CCC3)C2)C1 37523,C1(C(=O)NCCC2N(C(CCC(C)SC)=O)CCCC2)CCC(C)(O)CC1 37524,C1(C(N(CCOCCN(C(CCCCC#C)=O)C)C)=O)COC2(CCC2)CO1 37525,C1(C(=O)O)COC2(CCN(C(=O)Cc3cnc4n3CCNC4)CC2)C1 37526,Cn1nc(C2CC2)cc1C(F)(F)F.C12CCCC(C1)C(=O)OC2.c1(=O)c(=O)[nH]1 37527,c1(CC2(C(=O)NCC3(CNC(C4CCC(=O)N4)=O)CCCC3)CC2)cccc(C)c1 37528,CCC(C)(C)CC(C(=O)NCCOC)N(C1(C)CC1)C 37529,c1(C(C(=O)NC(CC)C)N(C)CC2(C)CC2)csnc1OC 37530,CC(C)CC(C(=O)N1CC2CC(NC(=O)CCC(C)(C)O)CC1C2)C(N)=O 37531,C1(CC)(CC)CC(NC(c2cnccn2)=O)CN1C(C12COCC1C2(F)F)=O 37532,C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(C3CC3C(F)F)=O)CC(C2)C1 37533,C1(S(N)(=O)=O)(C(=O)NC(C)CCNC(c2cn(CCN(C)C)cn2)=O)CCC1 37534,C1(C(N(C)CC2CCCN(C(C34CC(C3)C4)=O)C2)=O)C(O)C(=O)N(C)C1C 37535,N1(C(C2CC(F)(F)C2)=O)CCC(CCNC(C2COCCO2)=O)CC1 37536,CCCCCC(CC)C(=O)NCCOCCC(N1CCN(C(C)C)C(=O)C1)=O 37537,Cc1ccccc1CCC(=O)NC1CCC(NC(=O)CC2CCCCN2C)C1 37538,C12CCCN(C1)C(=O)CN1CCC(C1)NC(=O)C2.c1(COC)nccn1CCF 37539,N1(C(CCCO)=O)CCCC(O)(N(C(=O)Cc2nc(C)sc2C)CCOC)C1.OC 37540,c1(C(=O)OC)ccnc(C(=O)N(c2cccnc2)C(=O)CN(C)C(C)C)c1 37541,C1(C(C)NC(=O)C=CCN(C)C)CCN(C(c2csc(C#N)c2)=O)CC1 37542,C(=O)(CC(C)(C)N(C(=O)C(C)c1cccs1)C)N(CC#C)CC=C 37543,C=CCC(F)(F)C(=O)N1CC(O)(C(F)C(=O)NCC(C)(C)CC)C1 37544,N1(C(CSCC)=O)CCC2(CCC(C(=O)Nc3ccc(OC)c(OC)c3)O2)CC1 37545,C1(O)(CNC(c2c(OCC)scc2)=O)CCN(C(c2nnn3c2CCC3)=O)CC1 37546,C1(NC(Cc2ccc(C)cc2)=O)CC(F)CN(C(=O)COc2ccccc2)C1 37547,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37548,Cc1cc(OCCOC(=O)C(n2nc(-c3ccccc3)ccc2=O)C)ccc1Cl 37549,c1(C(N2CC(CC(=O)Nc3n(C)ncc3Br)C2)=O)cc2ccoc2cn1 37550,c1(C(=O)NCC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)F)ccc(OCC(F)F)nc1 37551,c1(CC(=O)NCCN(C(C2(CCO)CC2)=O)C2CC2)c(F)cc(F)cc1F 37552,Cn1cncc(C(=O)NCC(N2CCN(C(=O)CC3CCCCO3)CC2)C)c1=O 37553,CC1(OCCC(=O)N(CC(=O)NC(CCO)c2cccs2)CC2CC2)CCC1 37554,c1(C(N2CCC(NC(c3cccn(C4CC4)c3=O)=O)C2)=O)ccn2ncccc12 37555,c1(C(=O)NC(CCN(C(COCC(=O)NC)=O)C)C)cnc(Cl)s1 37556,C(C(=O)NCCC1(NC(C2CCCC(C)O2)=O)CC1)(C(C)C)OC 37557,C1(N(C)C(C2CC2(F)Cl)=O)CCC2CN(C(=O)Cn3cnnc3)CC12 37558,C12(NC(c3cnn(CC)c3Cl)=O)CCCC1N(C(=O)C(COC)OC)CC2 37559,C(CC(C)CN=C(NC1CCC1)NC1CCN(S(=O)(=O)CCOC)CC1)OC 37560,c1(C(N2CCC(C)(CCNC(=O)C3CC3)CC2)=O)cc(F)cc(F)c1O 37561,O=C1C(C(=O)N(O)Cc2cncn2-c2ccccc2)CCN1c1ccccc1F 37562,N1(CC(=O)NC(CC)C)CCN(CCCCCc2ccc(Cl)cc2)CC1 37563,C1(NC(C(F)=CC)=O)CC(F)(F)CC1C(=O)NC1CC1.c12ccc(cc1)[nH]c2=O 37564,c1(CC(=O)NC2CCCN(c3ccnc(Br)n3)C2)cnn2c1CCCC2 37565,N#CC1CCCCN1C(C1C2CCC(C2)N1C(=O)CC1CC2C=CC1C2)=O 37566,c1(OC)ccc(C(=O)NCC2CCN(C(=O)Cc3cc[nH]c3)CC2C)c(Cl)c1 37567,C123C4C5C1C1C2C4C51C(=O)N1CCN(CC1)C3=O.c1(N(C)C)ccn(C)n1 37568,c1(C(=O)NC2(CCNC(C(c3ccc(Cl)s3)C)=O)CCC2)n[nH]c2c1COC2 37569,C1(CCC=C)(NC(=O)CC2CCCC2O)CN(C(C2CCC(C)O2)=O)C1 37570,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)Cc1ccc(Cl)cc1 37571,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37572,Cc1ccc(CN(C(C2CCCC2C)C(=O)O)CCO)c(N)c1C 37573,c1(NC(=O)NC2CC2C2CCCC2)ccnn1C(C)(C)OC 37574,N1(C(=O)CCC2CCCO2)CC2CCC(C1)N2C(=O)CC1CC2CC2C1 37575,N1(C(c2ccsn2)=O)CC2(C1)CN(C(=O)CCc1ccnc(Cl)c1)CCO2 37576,C1(NC(Cc2ccc(NC)cc2)=O)C2CC(O)C1N(C(c1cnc(S)nc1)=O)C2 37577,CC1C2C(CCN2C(=O)Cc2ccc(O)cn2)CN1C(C12CCC(C1)OC2C)=O 37578,C1(CNC(C2C(COC)C2)=O)CN(C)CCN1C(c1cc(N)ccc1SC)=O 37579,c1(C(=O)NCC(CCCC)NC(=O)CCC(F)F)cc([N+](=O)[O-])ccc1O 37580,C1(OC)CC(NC(=O)C=Cc2cnc[nH]2)C12CCN(C(c1cncc(F)c1)=O)CC2 37581,N1(C(C(=O)NC)=O)CCN(C(=O)C(N2CCOC2=O)C)C(CCC(C)(C)C)C1 37582,c1(C(=O)NCC2C(NC(c3c(C)ncc(C)c3)=O)C2)cc(Cl)cc2c1OCC2 37583,CS(=O)(=O)c1ccc(CN2CC(O)CC2C(N2CCC(F)(F)CC2)=O)cc1Br 37584,c1(NC(c2cccnc2)=O)cnc(Br)nc1.c12ccncc1-c1ccc(nc1)N2 37585,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37586,c1(C(C(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)O)ccc(Cl)cc1F 37587,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37588,CCCCCCNC(C1COC(CNC(=O)C(C)SCC)C1)=O 37589,CC1CN(C(=O)CC2NC(=O)NC2=O)CC(C)CN1c1nccc(C(C)(C)C)n1 37590,Cc1c(C(=O)NC(C)C(C)NC(c2c(Cl)ccc(Cl)c2O)=O)sc2ccccc12 37591,C(CC(=O)NCCOC1CCCCC1)(C(F)F)NC(c1c(NC)cccc1)=O 37592,Cc1cc(C(=O)NC23CC(NC(=O)C(C)OCCC(C)C)(C2)C3)cc(C)c1N 37593,C1(CNC(CC(C)(C)SC)=O)CC12CCN(C(=O)Cc1cccnc1Cl)CC2 37594,c1(CC(N2CC(CNC(C3(OC)CCC3)=O)C(O)C2)=O)cccnc1Br 37595,C(=O)(C(C)C1=CCCC1)NC1CN(C(C2C(OC)CCCC2)=O)CC1O 37596,c1(C(N2CCC(N(C(C(CC)=CC)=O)CCC)CC2)=O)cc2c(s1)CN(C)CC2 37597,N1(C(CCCC(=C)C)=O)CCCC2(C1)CN(C(C1CCCN(CCC)C1)=O)C2 37598,c1(C(=O)NC(CC=C)CNC(=O)C(C)Cc2ccnn2C)ccc(Cl)cc1F 37599,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)CC1C 37600,c1(C2(NC(c3ccc(C4CCCCC4)o3)=O)CC2)ccc([N+](=O)[O-])[nH]1 37601,N1(C(CCC#C)=O)CCC(F)(F)C(C(=O)NC(C)(C)C#CCCC)C1 37602,c1(OC(C)C)ccc(Cl)cc1C(=O)N(CCC(C)NC(=O)CC1CC(=O)C1)C 37603,C1(C(=O)NCc2c(C)nc(CC)o2)CN(C(C2CCCC2CC)=O)CCC1(C)C 37604,N1(C(C2CC(C)NCC2)=O)CCCCC2(CCOCC2)C1 37605,C1(NC(N(C(C)C)CCO)=O)CCC(NC2CC2(F)Cl)CC1 37606,c1(-c2cn(CC3CCC(CNC(C4(CF)CC4)=O)CC3)nn2)cc(F)c(F)c(F)c1 37607,c1(C(N2CC(CNC(c3nc(C(C)=O)sc3)=O)C(C)C2)=O)c(C)nc(C)nc1C 37608,CCCCC(=O)N1CC(F)(NC(c2cnc(-c3ccco3)s2)=O)C1.C(N)(=O)NC 37609,C1(COC)(NC(=O)OCCC(=O)OC)CCN(C(=O)CN(c2ccccc2)C)C1 37610,c1(C(=O)NC2CC(NC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37611,Cc1cnn(C)c1CC(=O)NCCC(C)CCNC(c1ccnn1C1CC1(F)F)=O 37612,C1(CNC(C=C(CC)CC)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37613,C#CCC(C)C(=O)NCCC1CCCN(C(=O)C(C)(C)Oc2ccccc2)C1 37614,N1(c2cc(C)c(C#N)cn2)C2CCC1C(C)C(NC(=O)Cn1ccnc1C)C2 37615,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37616,N1(C(C)=O)CCCCC1CC(=O)NCC1CC1NC(C1CC1c1ccccc1)=O 37617,N1(C(=O)Nc2ccccc2)CCN(C2CCC(C(c3ccc(Cl)cc3)O)C2)CC1 37618,c1(C(=O)NC(C(C)NC(C=CC=CC)=O)CO)ccccc1OC1CCCC1 37619,N1(C(CCSCCC)=O)CCC2(CCC2CNC(=O)CN2CC=CC2)CC1 37620,C1(NC(C(C)C(C)(F)F)=O)CN(C(=O)CCc2nc[nH]n2)CC2(CCC2)C1 37621,c1(C(N2CCC(CO)C2(C)C)C(=O)NC(CC)C)cc(Cl)c(Cl)c(Cl)c1 37622,C(=O)(C(C)(C)N1CCCC1)NCC(C)N(C(=O)CCNC(N)=O)C 37623,C1(C)(C(=O)NCC(CC)NC(c2coc(C(C)C)n2)=O)CC(C(F)(F)F)=NO1 37624,c1(OC(C)C)cc(C(=O)NC(CO)C(C)NC(=O)C=Cc2ccncn2)ccn1 37625,C1(NC(C(CCC)OCC)=O)CCN(C)C12CCCN(C(C1(F)CCOC1)=O)C2 37626,c1(CC)ccc(C=CC(=O)NCCC(C)(CC)NC(c2cnnn2CC)=O)o1 37627,N1(C(c2c(C)cc(Br)cc2)=O)CCC2CN(C(c3conc3C)=O)CC2C1 37628,CCCS(=O)(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CCC1OCCO1)CC2 37629,C1(Cn2cc(CC(C)(C)CO)nn2)CN(C(=O)CC2CCOC(=O)CC2)C(C)(C)C1 37630,c1(CNC(C(N2CC(C)C(C)C2)CCc2ccccn2)=O)cccc2ccccc12 37631,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37632,C1(O)(C(CCOCCN(C(C2C(C(=O)OC)CCC2)=O)C)=O)CCC(C)(C)CC1 37633,C1(C(=O)NC(c2cnn[nH]2)C)CCCN1NC(=O)c1c(Cl)cnn1C 37634,CCCC(C)(O)C(=O)NC1CC(O)CN(C(c2ncoc2C(C)(C)C)=O)C1 37635,C1(C(=O)NC2C(CCOC)C2)C2CCC(C2)N1C(C1CC2C=CC1C2)=O 37636,C(CS(=O)(=O)C1CCOC1)NC(CO)Cc1ccccc1F 37637,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCCCN(C(C1CCC(C)CC1)=O)C 37638,N1(C(CCC(C)=O)=O)CCN(C(=O)CSCC)CCC1C 37639,c1(C(=O)NCC2CCN2C(c2ccnc(C3CC3)c2)=O)ccn2ncnc2c1 37640,C1(C(=O)NCC2(O)CN(C(c3ccc(CC)o3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37641,N1(C(c2c(CNC(c3cncc(OC)c3)=O)c[nH]n2)=O)CC2(CCC2)OCC1C 37642,C(C)(c1cccs1)=CC(=O)NCC(CC)NC(=O)C(c1cccnc1)O 37643,C(=O)(CC(F)(F)F)NCCC1CCC(NC(COCCC)=O)C1.C1(=O)CCN1 37644,c1(C(c2n(CC)nnn2)NCc2cncc(Br)c2C)cccc2c1OC(F)(F)O2 37645,C1(NC(c2ccc3ccoc3c2)=O)CCN(C(C2CCCSC2)=O)C12CCC2 37646,C1(C2CCC2)(CNC(C(C)=C(C)C)=O)CCN(C(c2cccc(Cl)c2C)=O)CC1 37647,CC1CC(CCNC(C2(C)CC2)=O)CCN1C(=O)Cn1ncnn1 37648,CCC(CC(=O)N1CCCC(CCNC(C2(C3CC3)CCCO2)=O)C1)C(C)C 37649,N1(C(C(C(C)C)CNC(=O)CNC=O)=O)CCOCC(C)(F)C1 37650,N12CCOC(C1)C(=O)OC2=O.CCCCN(CC(F)(F)F)CCCN(C)C 37651,c1(CC(=O)N(C2CCN(C(C(CC#C)C3CC3)=O)C2)C)cn2cc(F)ccc2n1 37652,C(=O)(C(O)C(F)F)NCCCNC(C1CC(C(C)C)C1)=O 37653,c1(C(=O)NCCC2CC(NC(c3cc(Cl)no3)=O)C2)sc(F)cc1Cl 37654,C1(C(=O)NOCCOCCCC(=O)NC(CO)C(C)C)(CC)CCCC1 37655,c1(CNCC2C(C(=O)NCC3C(C(=O)OC)CCC3)CCC2)cccc(C#N)c1C 37656,C1(C(=O)NCC2CC2(Cl)Cl)(COC)CN(C(=O)CC2(O)CCC2)C1 37657,c1(C(N2CC(NC(c3cc(COC)[nH]n3)=O)C(F)CC2)=O)ccc2c(c1)CCC2 37658,c1(NC)c(C(N2CC(CN(C)C(c3ccc(Cl)o3)=O)C2)=O)sc2cccnc12 37659,c1(C(=O)NC(C(=O)NCCCC=C)C2(O)CCC2)nccnc1N 37660,c1(NC(C2CCCC(C(N3CC(C(=O)OC)C3)=O)C2)=O)ncnc(C)c1C 37661,CC(C)(C)CC(O)C(=O)NCCC1CC(C)C1.c1(CNC(=O)C)nccs1 37662,C(=O)(C1COc2ccccc21)NC(C)CC1CCN(C(=O)C(C)(C)N(C)C)CC1 37663,c12nn(c(=O)n1C)C(=O)NCC(=O)NCCNC(=O)C2.Cn1cncc1CO.CC 37664,c1(C(N2CC(C(C)NC(C(CC)OC)=O)C2)=O)ccc(OC)cn1 37665,Cc1ccc(C(N)=O)cc1C(N1CC2CC1C2CNC(C1CN(C(N)=O)C1)=O)=O 37666,CC1(CNC(=O)CCN2CCCCC2=O)CCCN(C(=O)Cn2cncn2)C1 37667,C(C)(CN=c1[nH]nc(CC(F)(F)F)o1)Oc1c(OC)ccc(CNC2CC2)c1 37668,n1(C(C(=O)NC(CCCC)CNC(=O)Cc2cccs2)C)nc(C)n(C)c1=O 37669,C(C)(CC(C)C(F)F)NC(CCN(CC#C)C(c1nn(C)cc1C)=O)=O 37670,c1(C(=O)NC2CCCCN(C(=O)C(=O)C3CCCC3)C2)ccc2occc2c1 37671,c1(C(C(=O)NCCNC(CC(=O)OCC)=O)C)ccccc1Cl.c12cccn1C2 37672,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37673,C1(CCNC(c2cc(OCC)n[nH]2)=O)CSCCN1C(=O)CS(=O)CC 37674,c1(C(=O)NCC(CC)(C)NC(=O)Cc2cccc(F)c2)ncc[nH]c1=O 37675,c1(NC(c2n(CC)ncc2)CSC)ccc2c(c1)CCC(C)C2 37676,Cc1cc(C(=O)OCCSC2(c3ccccc3)COC2)c2c(Br)cnn2c1 37677,C1(CNC(CCOC2CCCC2OC)=O)CCC(CNC(COC)=O)CC1 37678,c1cc2[nH]c(=NCC3SCCS3)nc(-c3ccccc3)c2[nH]1 37679,c1(NC(C2CC(NC(c3cnc[nH]3)=O)C2)=O)ccc(I)cc1[N+](=O)[O-] 37680,c1(OC(C)C)ccc(C(=O)NC2CC2CNC(=O)CN2CCS(=O)CC2)c(Cl)c1 37681,N1(C(C)=O)CCN(C2CCCC2NC(c2cscc2C)=O)CC1 37682,Cc1cc(C(N2CCOCC2C(N2CCOCC(O)C2)=O)=O)cnc1C 37683,c1(CC(=O)NCC2(CN(C(=O)C(CC3CC3)SCC)C)CC2)c(C)nn(C)c1C 37684,c1(C(N2CC(CNC(C(CSC)(C)C)=O)OCC2)=O)cn(C2CC2)c(C)cc1=O 37685,CC(C)(C)C(C(=O)N1CC(OCC(=O)NCC23CCN(CC2)C3)C1)N1CCNC1=O 37686,CC#CCCCC(=O)N(CC(C)CNC(=O)C(C1CCOCC1)C)C 37687,C(C)(C(=O)N1CC(NC(c2ccc(CSC)o2)=O)C2(CC2)C1)(C(C)C)OC 37688,C(=O)(CCC(=O)N1CCN(c2ccnc(SC)n2)CC1)NCCC.N(C(C)=O)CC 37689,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)N(C(C)C(F)F)C)C(C)(C)C1 37690,N1(C(CC(COC)C)=O)CC(C)(CNC(=O)CSS(C)(=O)=O)CC1(C)C 37691,CC(C)CCC(O)C(=O)NC(C)C(=O)NOCCC1CC2C=CC1C2 37692,S(=O)(=O)(c1ccc(NC2CC2)c(Cl)c1)N(CC(C)C1CCC1)CC1CCC1 37693,c1(C(C2C(C)OCC2)C(N2CCC2)=O)ccc(=O)n(-c2ccccc2)n1.N(C)C 37694,Cc1ccc(NC(C2(CNC(=O)CCCC3CC3)CCCCC2)=O)cc1C 37695,c1(C(=O)NCCNC(=O)CCCn2c(O)nnc2O)ccc2ccccc2n1 37696,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)CC1O 37697,c1(N(C)C(C2CC2)C2CC2)nnc(-c2cc(Br)no2)n1CC1CCOC1 37698,C(=O)(C#CC1CCOC1)NC1CCC(NC(CN(c2ccccc2)CC)=O)CC1 37699,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37700,c1(C(=O)NC2C3(CC(NC(C(CCSC)O)=O)C3)C2)cc(Cl)ccc1O 37701,Cc1cnc(N2CCN(C(=O)C(C)(C)CF)CC2)nc1-c1noc(-c2cccc(Cl)n2)n1 37702,C(=O)(CC(CNC(=O)CCC1CCCCC1)CC)N(CC=C)CC1CC1 37703,c1(CCOC)nc(N2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)cc(Cl)n1 37704,C(=O)(CN=c1cc[nH]cc1)N1CC(C(N2Cc3c[nH]nc3C2)=O)SCC1 37705,N1(c2ncc(C(=O)OC)c(C)n2)CCC2(CCCN(C(c3ccc(Cl)s3)=O)C2)C1 37706,CCCCC(CNC(=O)COCCCOC)NC(=O)CC1CCS(=O)(=O)C1 37707,CCC(CN(C)C)CC(=O)N1CC(NC(c2cn(CC(N)=O)nn2)=O)CCC1C 37708,c1(C(N2CCC(O)(CC(C)NC(c3cncs3)=O)C2)=O)[nH]c2ccccc2c1Cl 37709,C=CC1(C(=O)NOCc2ccc(C)cc2)CCN(C(=O)Cc2ccccc2)CC1 37710,C12(C(N3CCOCC(CNC(c4c(C)ncs4)=O)C3)=O)CC1Cc1c[nH]nc12 37711,CC1(C)CCOC(C(=O)NCC2CCCCC2C(=O)NCc2ccc(O)cc2)C1 37712,C1(CC)CN(C(=O)CC2(N3CCCC3)CC2)CC1C(=O)NC1CCCN(C)C1 37713,N(C(=NCCc1nnc(CO)s1)NC1CCN(CC2CCCCO2)C1)C(=O)OC 37714,c1(N(C)C)cccc(C(=O)NCC2CN(C(=O)C3=CCC3)CCO2)c1.C1CCO1 37715,CCCCCC(C)NC(=O)CC1CN(C(=O)CCCOC)C1 37716,C(=O)(CC(F)(F)C(F)F)NC(C(C)C)(C)CNC(=O)CCOCC1CCCO1 37717,c1(C(N2CC(NC(c3ccc(SC)cc3)=O)C(O)C2)=O)cccc2nccnc12 37718,C(=O)(C1CC(=O)c2ccccc21)N1CCC(C)(NC(C=C(COC)C)=O)C1 37719,c1(C(N2C(C(=O)O)C3CC2C3)=O)cc2ncc(Br)cn2n1 37720,N1(C(C2(C=C)CCCC2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1C 37721,c1(-c2occ(CN(C(C(=O)Nc3c(C)n(C)nc3)=O)C(C)C)n2)ccc(F)cc1F 37722,C1(C(N(C)Cc2ccc(C)o2)=O)CCn2nncc2C1.C1(C)CN1 37723,c1(CNC(C2COCCN2CC(F)F)C)cc(C)c2c(c1)CCC2 37724,CN1CCc2[nH]nc(C(N3CC4C(NC(=O)CNS(N)(=O)=O)C4C3)=O)c2C1 37725,c1(C(=O)NC23COC(CNC(C4(CF)CC4(F)F)=O)(C2)C3)cn2c(n1)CCCC2 37726,N1(C(CCC2C(C)C2)=O)CCC(CCOc2ccsn2)(OCC(=O)NC)C1 37727,c1(CC)ccc(C(=O)NCC(C)(C)NC(=O)CC2CCCCO2)cc1S(C)(=O)=O 37728,c1(NC2CCN(C(CN(C(=O)OC(C)(C)C)CC)=O)C2)cccc(Br)c1 37729,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(CNC(c2ccc(C=C)cc2)=O)C1 37730,c1(C(=O)OC)cc(C(=O)O)n(C)n1.n12nnnc1C(C1CC1)NCCC2 37731,C(=O)(C(CCC)C(=O)OC)N1CCC(C)(C(N2CCC(N(CCC)CC)C2)=O)C1 37732,N1(C(C(C)OCCC)=O)CCN(C(=O)C(c2ccccc2)O)CC12CCC2 37733,N1(C(C(CC)C(C)O)=O)CC2(CCC(NC(C3CCC(OC(F)(F)F)C3)=O)CC2)C1 37734,c1(C2C(C(=O)NCC3CCCN3C(C3(O)CCOCC3)=O)C2)c(F)cccc1F 37735,c1(CC(=O)NC2CCCC(CNC(C3CCOCC3)=O)C2)ccc2c(c1)CCCS2 37736,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 37737,c1(COC)nc(C(=O)NCCC2CCN(C(=O)C=Cc3nccs3)C2)n[nH]1 37738,C1(c2ncc(C)[nH]2)(NC(=O)NCC2CON(C)C2=O)CCCCC1 37739,c1(OCC)cc2c(C(=O)N(CC(O)CNC(=O)CNC(C)=O)C)c[nH]c2cc1Cl 37740,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1CCC(CNC(c2ccccn2)=O)CC1 37741,N1(C(C(CSCC)NC(=O)CCC2CCCOC2)=O)CC(N=[N+]=[N-])C1 37742,c1(C(N(C)CCNC(C2(COC)CC2(F)F)=O)=O)nccc2ccsc12 37743,Cc1cc(Cl)c(C(=O)NNC(=O)C2CCC3CC3C2)c(Cl)c1 37744,C(=O)(C(C)(C)CO)N1C(c2n(C)ccn2)CC1 37745,CC(C(=O)NCCC1CCN(C(c2ccc(Cl)cc2)=O)C1)C(F)F 37746,C=CCC(CC(=O)NC(CC)CC(=O)NC(C)CC)NC(c1cc(F)ccc1C)=O 37747,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 37748,c1(-c2cn(CCCNC(C3CCCSCC3)=O)nn2)cnc2c(Cl)cnn2c1 37749,N1(C(CCCOC)=O)CCC(C)(C)C(C(=O)NC(C)COC(C)C)C1 37750,Cc1cc(C2CC2)n(CC(N2CCCCC2CN(C(=O)C(C)(C)CO)C)=O)n1 37751,N1(C(CC2(C)CC2)=O)CCC2CCCC12CNC(c1ccnc(Cl)c1N)=O 37752,c1(C(=O)NCCN(C(c2cc(CC)c(CC)o2)=O)C)ccc(N)c(Cl)c1O 37753,C(CC(C(=O)NC(C1CCCC1)C)NC(c1ccc(OC)s1)=O)OC 37754,c1(CNC(c2n(C)ncc2)=O)ncccc1C(=O)Nc1cnn(CC(F)(F)F)c1 37755,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 37756,C1(C(C)C)CCC(C(=O)NC(C2CN(C(c3ccc(C4CC4)o3)=O)C2)C)CC1 37757,c1(C(=O)NCC2(O)CCN(C(C3(COC)CC3)=O)C2)c[nH]c2cc(C#N)ccc12 37758,C1(NC(C(C(CC)C)O)=O)CN(C(c2conc2C)=O)C2(CCCC2)C1 37759,C1(C)(CC)CC(C(=O)NC(Cc2ccoc2)CO)CCO1 37760,C1(CC)CN(C(c2ccnc(I)c2F)=O)C(C)CO1 37761,CC(C)(C)C(C(=O)NCC1CC(NC(=O)CC2CCOC2)C1)C1CCCC1 37762,C12(C(=O)NC(C)CSC(F)F)CC(CO1)C2.C12CCCC1CC(=O)N2 37763,c1(C(=O)NCC2N(C(c3cccn(C)c3=O)=O)CCC2)cnn(C)c1S(C)(=O)=O 37764,N1(C(C(CC)OCC)=O)CC23CCCCC2(C1)CN(C(c1ccncc1F)=O)C3 37765,c1(NCC)cccnc1C(N1CC(OC)C1)=O.C12(CC(F)(F)C1)C(=O)N2 37766,c1(N2CCC(NC(C(C)OCCOC)=O)C(C)(C)C2)nc2cc(Br)ccc2o1 37767,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC1CCCN(C(C23CCC(CO2)C3)=O)CC1 37768,C1(CC)CCCCC1C(N1CC(CNC(c2ccn(CC#N)n2)=O)C1)=O 37769,c1(CC)c(C)nn(C)c1NC(=O)NC1CC2CC(NC)CC12 37770,C=CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(=O)CNC(=O)CCC 37771,N1(C(C2CN=C(C#N)CC2)=O)CCC(NC(=O)Cn2cnnn2)C(CO)CC1 37772,C(CCCCC(F)(F)F)NC(NC(C)C)=NCCN(S(=O)(=O)c1cccs1)C 37773,N1(C(C2N(C(CC3COCC(C)O3)=O)CCC2(C)C)=O)CCC(N=[N+]=[N-])CC1 37774,N1(C(c2cnc(Cl)s2)=O)CCC2CN(C(C3Cc4nncn4C3)=O)C2C1 37775,N1(C(CNC)=O)CC(F)CC1CNC(=O)COC1CC1.c1nc[nH]n1.C1(=O)CN1 37776,N1(C(C2CC(C)N2C(C2CCOC(C)C2)=O)=O)CCC(C)(C#N)CC1 37777,c1(C(=O)NCCCCNC(C(CCOC)C)=O)cc2c(s1)CCCNC2=O 37778,N#CC1(c2nn[nH]n2)CCN(C(C2CCN(CC(F)(F)F)CC2)=O)C1.n1(CC)cnnc1 37779,C12(C(N(C3CCN(C(c4c(C)sc(O)n4)=O)C3)CCO)=O)CC(C1)C(C)(C)O2 37780,N1(C(C(CCOCC(=O)N(C)C)c2ccccc2)=O)CCC(N)C(C)(C)C1 37781,c1(C(=O)NCC2CN(CC)C(=O)C2)ccc2c(c1)CCN(C(n1cc(Br)cn1)=O)C2 37782,c1(CN2C(NC(C(C)OCc3ccccn3)=O)CCC2)cc(Cl)cc(Br)c1O 37783,N#Cc1cccc(CCC(=O)NC23CC2CN(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1 37784,c1(CN2C(C)(C(N3CCC(N(C)CC)C3)=O)CCC2)c(F)cc(Cl)cc1Cl 37785,c1(N2C3(CNC(C4C(C(C)O)C4)=O)CC(C2)C3)ncc(Br)cc1C#N 37786,N1(C(C2C(C=C)OCC2)=O)CC2CCC(NC(c3ccoc3CCC)=O)(C2)C1 37787,Cc1cc(Cl)cc(C(N2CCCCC2CNC(=O)CC2CCCOCC2)=O)c1N 37788,c1(-n2cc(C3CC(NC(=O)Nc4coc(Br)n4)C3)nn2)ncccc1Cl 37789,C1(CNC(C2CCC(C3CCCC3)O2)=O)CCCCC1N1CCCC1=O 37790,CCC(C)C(C)CN=c1[nH]ccc(=NCCOc2ccc(F)c(F)c2)[nH]1 37791,c1(C(=O)NCC(CC(C)C)NC(C2(CC)CCCCC2)=O)ccoc1S(C)(=O)=O 37792,C1(OC)(CONC(c2ccc(SCc3cncn3C)cc2)=O)CCC(C)C1 37793,C1(C)(NC(C(=O)Nc2nc(C)c(Cl)cc2)=O)CCCC(C)(C)C1 37794,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 37795,c1(C(N2C(C(N)=O)CCC(C)C2)=O)cc(C#N)ccc1Br.C(COCCOC)N 37796,CCCCCC(O)CC(=O)NC1CCC(NC(=O)CCCN(C)C(=O)OCC)C1 37797,CC(C)(C)C(C(F)F)NC(C1CCN(C(=O)CCN2CCCCC2)C12CC2)=O 37798,C1(NC(c2c(C)cco2)=O)Cc2ccccc2C1NC(=O)CC(F)(F)Cl 37799,CCCN=C(NCCN1CCN(C)C(=O)C1)NC(c1cncc(C(F)(F)F)c1)C 37800,n1(CC)cc(C(=O)NC2CC(CCNC(C3CC3(C)CC)=O)C2)c(C(C)C)n1 37801,C(=O)(C1=CCCC1(C)C)NC(C(C)(C)NC(CC1(C=C)CCC1)=O)C 37802,N1(C(CCC=C)=O)CCC2CCN(C(C3CCCCN3S(C)(=O)=O)=O)C2C1 37803,N1(C(c2cnn[nH]2)=O)CCN(C(c2coc(CC3CC3)n2)=O)C2CCCCC12 37804,N1(C(CSC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 37805,Cc1nc(-c2cccc(Oc3ccc(C(F)(F)F)cc3)c2)n(CCC#N)c1C 37806,CCC(CC)(C(=O)NCC(C(C)(C)C)NC(=O)CCc1ncccn1)C(C)C 37807,C1(C(C)C)CN(C(=O)C(C)(C)C(=O)N(C)C)CCC1NC(=O)C1=CCSC1 37808,c1(OC(CC=C)=O)cccc(C(C)Oc2cnc(C(C)=O)s2)c1 37809,c1(N2CC(C)C(N(C)C(C)=O)C2)nc(C(=O)NC(C)(C)C)nc2sccc12.CCO 37810,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(=O)CC2CCC(C3CC3)O2)C1 37811,C#CCCCCCCCNC(=O)CC(CC)NC(c1cc(C)cc(C)c1)=O 37812,Cc1ccnc(F)c1NC(=O)Nc1ccc(Br)cc1C(=O)N(C)C 37813,C12(C(CNC(c3cn(C(C)(C)C)cn3)=O)NC(C=CC(C)C)=O)CCC(CC1)C2 37814,O=C(C(CO)OC1CCCC1)N1CCC1C(=O)NCC(F)Cl 37815,N1(CCc2c(C)cccc2)C2CCCC1CN(C(C1CCC(C)(C)C1)=O)C2 37816,N#Cc1c(C(N2CCC(F)(C(=O)NC3CCCCC3(F)F)C2)=O)cccc1Cl 37817,N1(C(c2ccc(CC)cc2I)C(=O)NCC)CCC(C2(O)CN(CC3CC3)C2)CC1 37818,CCCCC(C)CCC(=O)NCCN(CC(C)O)C(c1cccc(C)c1N)=O 37819,c1(C(N2CCC(NC(C3CC(CC)(CC)C3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 37820,Cc1c(C(=O)NC2(C)CCN(C(=O)C(C)O)CC2)sc2[nH]cnc(=O)c12 37821,C1(NC(C2C(OCC)C2C)=O)CCS(=O)(=O)C12CN(C(=O)Cn1cc(CO)nn1)C2 37822,C(C)(C(C(=O)N(C1CC(O)C1CCO)C)NC(C1OCCC1(C)C)=O)OC 37823,C1(NC(C2C(C)N(C(=O)Cc3cccs3)CC2)=O)CCn2nnnc2C1 37824,N1(C(C2CC(C(C)(C)C)C2)=O)CCCC2(NC(C3CCCOC3)=O)CCCC12 37825,Cc1nn(C)nc1C(=O)NC(C)Cn1cc(COC2CCCCO2)nn1 37826,O=S(=O)(c1cnc(Cl)c(C(F)(F)F)c1)N1CCCC(CN2CCOCC2)C1 37827,c1(N(C)C)cccc(-c2cc(N(C(=O)Cn3cc(Cl)cn3)CCO)ncn2)c1 37828,CCC(C)CC(C)C(=O)NCC1CC12CCN(C(C1CN(C)C1)=O)CC2 37829,C1(CNc2[nH]c(=N)sc2)CCN(S(=O)(=O)CC2CCO2)CC1(F)F 37830,N1(C(CNc2c(C)onc2)=O)CCC(NC(=O)CC(C)(C)C)C1C 37831,N1(C(CC(C(=O)O)OCC)=O)CCC(C)N(C(=O)C(c2ccccc2)C)CC1 37832,C1(OCCNC(C(=O)NS(=O)(=O)c2cccs2)=O)CC2CCC1CC2 37833,C(C)(C(=O)NC1CCCC1NC(=O)Cc1ccoc1)(C1CCOC1)NC(C)=O 37834,C1(C(=O)NC(CC)C2CCC2)(NC(=O)Cc2cccs2)CSC1 37835,c1(CC)c(NC(c2ccccn2)Cc2ccc(F)cc2)cnn1C(C)(C)C 37836,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)c(F)c1 37837,C1(C(=O)Oc2ccc(C(C)=O)cn2)CCN(C(=O)C=CC(CC)=C(C)C)C(C)C1 37838,C#Cc1ccc(C(=O)NC2CCCC2NC(C2CCC(=O)N(C)C2)=O)nc1 37839,C(=O)(CCCCCCn1cc(-c2ccc(N)cn2)nn1)N1CCCC(C)(CO)C1 37840,C1(C(N2C(C(=O)NCC(C)(C)CO)COCC2)=O)CCc2nc[nH]c2C1 37841,c1(C(N(CC(=O)Nc2nc(C(C)C)no2)CC)=O)cncc(Cl)c1 37842,c1(C(=O)NC2CC(C)(NC(COCCCC)=O)C2)ccc(C)c(C)c1 37843,C(=O)(CCCS(N)(=O)=O)NC(c1ccccc1)C(C)NC(=O)COCCN(C)C 37844,c1(C(C(=O)NC2CC(CC3CC(C)=NO3)C2)N(C)CC)cccc(F)c1F 37845,c1(C(=O)NCCN(C(C(C)C2CCCO2)=O)C2CC2)cnc2sccc2c1 37846,C1(CNC(C2(CC#C)CCCO2)=O)CC(C)CN(C(=O)C(C)(C)OC(C)C)C1 37847,c1(OC)ccccc1C(CNC(C1CC1F)=O)NC(=O)C(C#N)CC1CC1 37848,C(CCC(CO)N(c1nc(C)co1)C(=O)C1CC1)NC(C=CCOC)=O 37849,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)C2CCC2)c(Cl)ccc(F)c1C 37850,C1(NC(c2n[nH]c(O)n2)=O)CC2CN(C(c3ccnnc3Cl)=O)CC12 37851,C(=O)(C(O)CC(C)(C)C)NCCCC(CCC)NC(C1CN(C)CCN1C)=O 37852,C(N=c1cc2c(c[nH]1)CCCC2)c1cc(C(=O)OCC)c(OC2CC2)cc1 37853,c1(C(=O)NCC(C)(C)NC(C(CCSC)O)=O)ccc(C2=NOC(=O)C2)cc1 37854,CCCCC(CCC)N=c1nc(N(C)Cc2ccncc2Br)c2[nH]ccc2[nH]1 37855,c1(C(N2CC3CN(Cc4c(OC)nccc4)C3C2)=O)cc(C)c(Cl)cc1Cl 37856,C(=O)(C1CCCc2n[nH]cc21)NC1CC(OCC)C12CCC2 37857,c1(C(N(C2CCN(C(c3cncs3)=O)C2)CC)=O)cc2cccc(F)c2o1 37858,c1(C(=O)NCC2(F)CC(CNC(C(CC)O)=O)C2)cccc(CCO)c1 37859,C1(NC(c2cc(-c3ccco3)no2)=O)CC(F)CN(C(=O)CC2CCCSC2)C1 37860,CS(=O)(=O)c1cccnc1NC1CCCN(C(C2(O)CC3CC2C3)=O)C1 37861,N1(C(c2c(C)cc(SC)s2)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 37862,c1(NC(=O)NC(C2CN3CCCC3CO2)C)nc2ccc(Cl)cc2[nH]1 37863,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCN(C(C2CCCS2)=O)C2(CC2)C1 37864,c1(CC(=O)N(CCCNC(=O)Cc2n[nH]c(=N)s2)C)ccc(Cl)nc1F 37865,CCCC(C)(O)CC(=O)NC1COCCC1NC(c1cc(OC)ns1)=O 37866,Cn1nc2c(c1CNc1cc(N3CCOCC3)ccc1C(F)F)CCC2 37867,C1(CN=C(NC2CCC2)NC2CCCCC2)(C(F)(F)F)CC2(CC(F)C2)C1 37868,CCCCC(F)C(=O)NCC1CCCC1C(N1CCC(OC)C(C)C1)=O 37869,Cc1ccnc2c(C(=O)NCCCN(C)C(C34CC(C)(CCO3)C4)=O)cnn12 37870,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)CO)C3)sc2c1F 37871,Cn1cc2c(n1)CC(CNc1cscc1CNC(=O)C(=O)NC1CC1)CC2 37872,c1(N2CCC(CC)CC2)ncnc(NCCC2CC(O)C2)c1C 37873,c1(CC(=O)NC(CCOC)CNC(c2nn(C)cc2N)=O)c(C)ncnc1C 37874,C(=O)(C1=NN2CCC(C)N=C2N1)NCC(CC=C)NC(=O)CC1(C)CCCC1 37875,C1(C(=O)NC(C)(C)CCNC(=O)CC2C=CCC2)CC2(CCCC2)CO1 37876,c1(C(=O)NCC2C=CC(NC(c3c(Cl)nc(OC)s3)=O)C2)n[nH]c2c1COCC2 37877,C1(C(C)(C)C)C(NC(=O)Cn2cnc(CO)n2)CCN1C(=O)C=C1CCSCC1 37878,N1(C(c2c(CC)c(C)sc2)=O)CC2CC(NC(c3sc(OC(C)=O)nc3C)=O)C1C2 37879,N1(C(C2C=CC(NC(c3ccc(C#N)cn3)=O)C2)=O)CCc2cncnc2C1 37880,C1(C(=O)NCCC2(NC(C(CSC)O)=O)CCC2)CCN(CCO)C(=O)C1 37881,c1(C(=O)NCC2(C)CCN(C(c3ncccc3F)=O)C2)cccc(F)c1F 37882,N1(C(C(C=C)O)=O)CC2(CC2)CC1CNC(=O)C(=Cc1cccnc1)C 37883,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(C)n2)=O)CC1 37884,c1(-c2sc(C(=O)NC3C(NC(C=C(C)C4CC4)=O)CC3)c(C)n2)c(C)nn(C)c1C 37885,c1(SCC)ccc(-c2nc(-c3cnn(C)c3)nn2-c2ccnc(O)c2)cc1 37886,C1(C(=O)NC2CC(NC(c3c(C)ocn3)=O)C2)CCCCC1n1cccc1 37887,c1(C(=O)NCCCCCNC(=O)COC2CCOC2)cc(O)cc(Cl)c1 37888,C1(CC)COCCN1N1CCN(C(=O)CO)C(c2ccccn2)C1 37889,CN1CCC(n2nc(-c3ccc(C(F)(F)F)nc3)nc2-c2cc(Cl)n[nH]2)CC1 37890,Cc1ccc(C(CO)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 37891,c1(CN2C(CC)CN(C(c3c(Cl)ccnc3Cl)=O)CC2)ccc2nc(O)[nH]c2c1 37892,C1(C)(C(N(CC(CNC(CCc2c(C)noc2Cl)=O)C)C)=O)CCCCC1C 37893,C(C(=O)N(CCCNC(=O)C=C1CC1)C)(C1CCCC1)OC 37894,c1(C(=O)NC2CCCC(N(C(CCC(=O)NC)=O)C)C2)oc2ccccc2c1C 37895,c1(C(=O)NC2CC(NCc3ccc(F)c(C(F)(F)F)c3)C2)c(Br)cc(F)c(F)c1F 37896,CC(N=c1[nH]c(=NCCSCC2CCCO2)[nH]c2c1COC2)c1ccco1 37897,CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CCN(C(=O)C=CC2CC2)CC(O)C1 37898,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 37899,Cc1ccc2c(c1)CC(C(=O)NC1COCCN(C(=O)C(C)(C)O)C1)S2 37900,C(=O)(CCCC(=O)NC1CC(NC(C2CC2c2cccnc2)=O)C1)OCC 37901,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 37902,Cc1cn2c(C(=O)NCC3CCCCN3C(=O)CCC(C)C)cnc2s1 37903,c1(CNC(=O)Nc2c(C)cncn2)ccnc2ccccc12 37904,Cc1ccc(N(C)C)c(C(=O)NC2CCC2NC(=O)C(C)n2cnnn2)c1 37905,N(C1CCc2sc(Br)cc21)C(=O)OC(C)(C)C.c12cccc(c1)CNC(=O)N2 37906,C1(CC)CCCCC1N(C)C(c1cncc(C(F)F)c1)=O.C12(CCC1)C(=O)NC2 37907,C1(N(C)C)CCC(C(=O)NCCCN2CCCC2)CC1.C12CC(C1)NC2=O 37908,C1(CNC(=O)COc2nccc(-c3ccccn3)n2)CC2(CCC2O)C1 37909,C1(O)(CN(C(CC(=O)NCC)=O)C)CCN(C(=O)C(c2ccccn2)C)C1 37910,C1(NC(C2C(C(=O)OC)CC=CC2)=O)CN(Cc2nc(CO)cs2)CC(F)(F)C1 37911,C1(CNC(c2ccc(SC)s2)=O)CC2CN(C(=O)CN3CC(C)(C)C3)CC12 37912,C(=O)(C(C(C)(C)CC)OC)N(CCN(C(=O)C(CC)OC(C)C)CC)CC 37913,CCC(CC(=O)N1CC(CN(C(=O)CC2(O)CCC2)CC)C1)C(C)(C)C 37914,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1F)=O 37915,N1(C(c2ccc(C)nc2N)=O)CC2CCN(C(=O)C3=NOC4COCC34)CC2C1 37916,C1(C(N2CC(CCNC(c3ocnc3C3CC3)=O)OCC2)=O)CC(=O)C12CCC2 37917,N1(C(CCC)=O)C(C(=O)Nc2ncn(CC)n2)CC2CCCCC12 37918,CC(C)(C)CCC(F)C(=O)N1CCCC(O)(CNC(c2nn[nH]c2Cl)=O)C1 37919,C12CCCC1NC(=O)C2.C1(NC(c2ccsn2)=O)(CO)CCC1.CCC 37920,C12(CNC(=O)CN3CCC3)CCCC1CCN2C(c1cc(F)ccc1Cl)=O 37921,C1(Cn2cc(C(C)(C)C)nn2)CCCN(C(=O)CC2(n3ccnc3)CC2)C1 37922,C1(C(N2CCC(SC)C2)=O)CC2CC2N1C(=O)CC1(C)CC1 37923,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 37924,N1(CCC)CCCC(C(N2CCC(CC)C2CNC(=O)CN2CC=CC2)=O)C1 37925,c1(C(=O)NCC2CC(CNC(c3cc(F)c[nH]3)=O)OC2)cnc2ccccn12 37926,c1(C(N(CC(CN(C(C(C)SC(C)C)=O)C)O)C)=O)cccc(=O)o1 37927,c1(CSCC(=O)NCC2(NC(=O)CCC3CC3(F)F)CC2)nnnn1C1CC1 37928,C1(C(=O)NC2(CO)CN(C(=O)CC3C=CCC3)C2)CC2CC(=O)C1C2 37929,C(=O)(C(CO)NC(=O)C=CC1CC1)NCC(C)(O)C1CC1 37930,c1(C(C)C)cc(C(=O)NC23CC(CNC(C4CCC(O)C4)=O)(C2)C3)n[nH]1 37931,c1(C(=O)NCC(C)NC(=O)CC2CC=CCN2C)ccc2c(c1)CCC(C)(C)O2 37932,C1(C(=O)NC(C2CCN(C(=O)Cn3nccn3)CC2)C)(OCCO)CCOCC1 37933,CCCCC(CC)CC(=O)NCC(C)(C)C(=O)NCCS(=O)(=O)NCC 37934,C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(C2CN3CCN2CC3)=O)C1 37935,Cn1nc(-c2ccccc2)c([N+](=O)[O-])c1N1C2CCC1C(NC(C1CC1(C)C)=O)C2 37936,c1(C(=O)NC(CCN(C)C(c2cnc(Cl)s2)=O)(C)C)ccc2ccncc2c1 37937,N1(C(=O)Cc2ccnn2C2CCOCC2)CCCC(CO)(CO)C1 37938,c1(C(c2n(CCC)nnn2)Nc2cccc(N(C)C)c2)c(F)ccc(Br)c1C 37939,N1(C(C)=O)CCCC(O)(C(=O)NC2CC(NC(=O)CC3CCN(C)CC3)C2)C1 37940,C(=O)(CC(C)(C)C)NC(C)CN(C(=O)CC1CCC(C)O1)C 37941,C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CSC(C)(C)C)CCC1C 37942,c1(CC(C)C)cccc(C(=O)NCC(O)CNC(=O)C(C)SCc2cccs2)c1 37943,c1(C(=O)NCCC2CCN(C(C(C)C#N)=O)CC2)ccn2cncc2c1 37944,C1(F)(CNC(C2CCc3nncn3C2)=O)CCCN(C(C2CCCC2O)=O)CC1 37945,CC(C)(C#N)CCC(=O)N1CCC(NC(=O)CSc2nc[nH]n2)C(F)C1 37946,CC1(C)CCCN(C(c2ccc(Cl)c(F)c2)=O)C1CNC(=O)Cc1ccco1 37947,C1(NC(C(CC)n2ccnc2)=O)CCC(CNC(=O)C(c2cccnc2)F)CC1 37948,Cn1cc(C#CC(=O)NCC2CCCOC2c2ncc[nH]2)cn1 37949,CC1CCCCC1OCCCC(=O)NCC1CC(c2ccccc2)(NC(N)=O)C1 37950,c1(CNC(CSCC(C)=O)=O)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 37951,C1(Nc2ccc(C3COCCN3)cc2)CCCOC12CCCC2 37952,C1(N(C)C)(NC(N(C(C2CCOC2)CO)C)=O)COc2ccccc2C1 37953,c1(CC)ccc2c(c1)C(CCNC(c1cc(C)nn1Cc1ccco1)=O)C(=O)N2 37954,c1(N(CCOCC(=O)NCCc2cn(CC)nc2)C2CC2)ncccc1C#N 37955,CC1CN(C(=O)CNc2ccccn2)CCC1CNC(=O)C=Cc1cc[nH]c1 37956,c1(C(N2CCC(C)CC2CNC(c2cn(C)cn2)=O)=O)cc2cc[nH]c(=O)c2s1 37957,c12cc(S(N)(=O)=O)cnc1N2.C1(C(N2CC(C(=O)OC)C2)=O)Cc2nccn2C1 37958,C12(CC)CCCN1C2=O.C1(C(NC[Si](C)(C)C)=O)CCC(F)CC1 37959,c1(C(N(CCC(C(C)C)NC(=O)C=CBr)C)=O)ccc2c(n1)CCO2 37960,CCC(CC)CC(C(=O)NCCOC)N1CCC2CCCC2C1 37961,c1(S)ccccc1.CC(C(=O)NC1(CCNC(C2CC2C(F)(F)F)=O)CCC1)C1CC1 37962,N1(C(C(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccn(CC)n3)C2)C1 37963,C(=O)(CCc1cncs1)N(C(C)CNC(=O)C(C1CCC1)OC(C)C)CC 37964,C(=O)(C(O)C(C)(C)C)NCC1CCN(C(c2ccc(C(C)C)cc2)=O)C1 37965,N1(C(C(c2ccc(F)cc2)C)=O)CCC(C(=O)NCc2occc2C(=O)O)CC1 37966,C1(C(=O)NCCC2N(C)CCC2)COCCC1NC(=O)CP(C)(C)=O 37967,CCC(O)C(C)C(=O)N1CCN(C(=O)C(N2CCOCC2)(C)OC(C)=O)CC1 37968,c1(C(N2C(C)(CNC(=O)C(F)=C3CCCC3)CCC2)=O)occ2c1CCOC2 37969,c1(C(N2CCC(CC(N3CC4C(C(=O)O)(C4)C3)=O)CC2)=O)cncc(F)c1I 37970,c1(C(N(CCCCNC(c2ccc(CF)cc2)=O)C)=O)cccnc1NC(N)=O 37971,C=C(C)C1OCCC1C(=O)NC1C=CC(CNC(C2C=CCC2)=O)C1 37972,CCC(C(=O)NCC1CN(C(C2(C#N)CCC2)=O)C1)OC1CCCCC1 37973,c1(-c2cn(C3CN(C(C(C)c4ccco4)=O)CC3O)nn2)nsc2ccccc12 37974,c1(CC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(CC)c1 37975,C1(CC(=O)NC(CC)CSC)CN(C(=O)OC(C)(C)C)CC1OC1C=CCC1 37976,C1(C(N2C(CNC(c3cncc(C#C)c3)=O)C=CC2)=O)CC2(C1)CC1(CC1)C2 37977,c1(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C(C)C)C)coc2ccccc12 37978,c1(CN2CCC(C)(C(=O)NCCC)C2)cc2ccccc2s1 37979,N1(C(CN(C(CNC(C(c2ccccc2)C)=O)=O)C)=O)CC2CCC(CO)(C2)C1 37980,c1(CNC(CCCNC(N)=O)=O)cncc(C(=O)NC2COC(C(F)F)C2)c1 37981,c1(C(C)=O)cccc(CC(=O)NC(C2CCN(C(=O)C=C3CCC(C)C3)C2)C)c1 37982,C(=O)(CCCNC(C)=O)OC(C(=O)N(CCOC)CCF)CC1CC1 37983,c1(NCC(c2cn(C)nc2)O)nc(NC2CC3CC(CO)CC23)c2ccsc2n1 37984,C(=O)(CC(C)C(C)C(C)C)NCC1(F)CC(NC(c2nnc(C)s2)=O)C1 37985,C1(C(=O)NCC(C)OCCO)CN(C(=O)CC2(O)CCOCC2)CCC1(C)C 37986,N1(C(=O)CCCSCc2ccc(Cl)cc2)CCC2CN(C(=O)CNC3CC3)C2C1 37987,C1(C(=O)NC2(CO)CC(C)C2)CCN(C(C2CCC(=O)N2C)=O)CC1 37988,N1(C(C2C(C(C)C)C2)=O)CCC(F)(F)C(CNC(=O)Cc2ccsc2)C1 37989,N1(C(C=CC)=O)CCOC2(CCC(NC(C3CCCC(C(C)(C)C)C3)=O)CC2)C1 37990,c1(C(=O)NCC2N(C(CC(=O)NC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 37991,C1(C(N2C(CCNC(C3CC=CCO3)=O)CCC2)=O)CCc2nnnn2C1 37992,CC(CC(=O)NCC1CCN1C(=O)CC1CCCC1)c1cnn(C)c1 37993,C(C(=O)NCCCCC(C)NC(C1(C(F)(F)F)CC1)=O)(C(C)C)c1cc(C)no1 37994,c1(CC(=O)NCC2N(C)CCN(C(c3cn(C)nn3)=O)C2)ccn2cncc2c1 37995,N1(C(CCCC=C)=O)CCN(C(C2CC3CCC3C2)=O)C(c2ccccc2)C1 37996,C12(C(=O)NC(CC)CNC(C3COC(=O)N3C)=O)CC(CO)(C1)OC2(C)C 37997,C1(C(N2CCC(CN(C(=O)CN=S(C)(C)=O)CC)CC2)=O)COC2(CCC2)C1 37998,c1(C(N(CCNC(C(CC)CC(F)F)=O)C2CC2)=O)ccc2c(c1)CCCC2=O 37999,c1(COC)c(C(=O)NC2(CO)CN(C(=O)C(F)(F)c3nccn3C)C2)cnn1C 38000,N1(C(C2CCCC(=O)C2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccsc1)C2 38001,CC1CCN(C(=O)CC(=O)Nc2nccs2)CC1NC(C1CCS(=O)(=O)CC1)=O 38002,C(=O)(C1CCc2cccc(=O)n21)N.N1(C(CCNC(=O)NC)=O)CC(OC)C(OC)C1 38003,C(=O)(CS(=O)(=O)C1CC1)NCC1(NC(c2ccc(SCCO)cc2)=O)CCOC1 38004,c1(C(=O)OC(C)(C)C)cccc(CN(C)C)n1.C12(C)CCN1C2=O 38005,C(=O)(C(C(C)(C)C)OCCOC)NCc1cc(C(N2CCC(CC=C)C2)=O)sc1 38006,N1(C(C)C)C(=O)CCC1C(=O)NCC(C)N.C1(=CC(N2CCOCC2)=O)CCCCC1 38007,C(C1CCN(C(C2CCC3(CCC3)C2)=O)CC1)=CC(=O)NC(CCC=C)CO 38008,N1(C(CC2CCC(C)C2)=O)CC2(CCN(C(c3ccccc3SC(F)F)=O)C2)C1 38009,c1(C(=O)NC(C)C(CO)NC(c2cc3n(n2)CC(F)C3)=O)cccn2nccc12 38010,C1(CC(=O)NCc2ncc(C)o2)CC(NC(=O)C(C)OCOC)C12CCC2 38011,Cn1cc(C(=O)NCC2COCCN(C(C3CCOC(C)(C)C3)=O)C2)ncc1=O 38012,CCC(C)CCCCC(=O)N1CCCC1CNC(=O)CCCCc1ccccc1 38013,C1(NC(C(CCC)CC2CCCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 38014,Cc1cc(C(=O)N(CCCNC(=O)C=Cc2ccco2)C(C)C)c2c(c1)CCC2 38015,Cc1cc(F)ccc1CC(N1CCC(C)(NC(=O)C(=O)NC2CC2)CC1)=O 38016,Cc1ccnc(O)c1C(=O)NC1CC(O)CN(C(c2snnc2C2CC2)=O)C1 38017,C(=O)(C(CC)(CC)CC)N(C1CCC2C(=O)C(C(C)C)C(=O)N(C2)C1)OCC 38018,C1(NC(=O)CCCc2ccccc2)CN(C(=O)CN2CCCCC2=O)CC12CC2 38019,N1(C(CC2N(CC)CCC2)=O)CCN(C(=O)C=C2CCOCC2)C2CS(=O)(=O)CC12 38020,c1(NC(=O)NC)ccc(Cl)c(C(=O)NC2CC2NC(=O)CSc2ccncc2)c1 38021,C1(CNC(CCC(C)SC)=O)CN(C(=O)C(C)(C)N2CCCCC2)CCCO1 38022,c1(N2CCC(N(CC(=O)NC)C)CC2)nc(=NCC2CC2)[nH]c2c1SCC2 38023,CCC(C(=O)NC(C)CNC(=O)Cc1cccc(OC)n1)C(F)(F)F 38024,C(=O)(CC(C)(C)CCC1(O)CCC(C)C1)NCC1CC1.C1(=O)CCN1 38025,CC1(C)CC(C(N2CC(CCCCNC(c3ccnn3C(C)(C)C)=O)C2)=O)C1 38026,CCCCCS(=O)(=O)CC(=O)N1CCC(C)(NC(c2cc(F)c(N)c(F)c2)=O)C1 38027,CCC(C(=O)NC(CO)C(=O)NCCCCO)n1ccnc1 38028,Cc1cc(O)c(C(N2CC(NC(=O)C=CC3CCCC3)C(C)(C)C2)=O)nn1 38029,c1(NC2CCC(NC(c3c(C)cc(F)c(Cl)c3)=O)CC2)ncccc1S(C)(=O)=O 38030,c1(C(=O)NCCNC(=O)CC2CC(F)C2)c[nH]nc1Cl 38031,C1(NC(CCC(=O)NC)=O)CC(F)CN(C(=O)Cn2cccc(O)c2=O)C1 38032,C#CCC(C)(C(=O)Nc1ncnc(C)c1CC)NC(=O)C(CC)(C1CC1)SC 38033,N1(C(C(CC#CC)C)=O)CC2(CCC2)C1c1ccncc1 38034,C1(NC(C2CCC(CC)O2)=O)CCN(C(=O)CC2C=CCC2)CC1O 38035,c1(C(=O)NC2CCC(CCNC(c3nc(COC)sc3)=O)C2)sc(C)c(C)c1C 38036,c1(CC(C)C(=O)NC(C)(C)CNC(C2(C)CCCS2(=O)=O)=O)ccc(F)c(F)c1 38037,C=CC1OCCC1C(N1CCC(C(C)NC(=O)CC(O)CN(C)C)CC1)=O 38038,N1(C(CC2C(C)C2)=O)CCC(O)(C(C)NC(c2cn3ccsc3n2)=O)CC1 38039,C12(NC(c3cnc(C(C)C)[nH]3)=O)CCCC1CN(C(=O)CN(C)C(C)C)C2 38040,c1(C(=O)NCCC(C)(C)NC(=O)C(O)CCS(C)=O)nnc(O)c2ccccc12 38041,C1(C(=O)Nc2c(OCC)cccc2Cl)=CNC(C)=CC1=C1CCCCO1 38042,Cc1cc(F)nc(N2CCC(N(C)C(=O)NC34CCCCC3C4)C2)n1 38043,N1(C(C2(CC=C)CCC2)=O)CC2CC1CN2C(C1CC1(F)Cl)=O 38044,N1(C(c2c(C)cn(C(C)C)c2)=O)CC2(CC2)CC1CNC(c1cncs1)=O 38045,CC1CCN(C(=O)C2=CCCC2)CCN1C(c1noc2c1CCCC2)=O 38046,n1(CCC(=O)N(C(C)CNC(C2(C)CC2C)=O)C)c(C)nc2ccccc2c1=O 38047,Cc1ccc(C(=O)NC2CCC(NC(c3cnn4cccnc34)=O)C2)c(C)c1Br 38048,c1(CCC(=O)NCCCNC(c2nc(OC)oc2)=O)ccc(O)nc1 38049,Cc1oc2ccccc2c1C(N1CCN(C(=O)CCC2CCCCC2)C(C)C1)=O 38050,C1(CC(=O)NCC2CCN(C(C3C(C=C)C3)=O)CC2)CCCC2(CCC2)O1 38051,N1(C(C2CN(C(C)=O)C2)=O)CCC2CCCN(C(c3csc4cncn34)=O)C2C1 38052,N1(C(C(C)NC(=O)OC)=O)CCOCC(F)(CNC(C2(C3CC3)CCC2)=O)C1 38053,C(=O)(C1=CCCCC1C)NC(CC=CC)C(=O)Nc1cc(Cl)ccc1C 38054,CCCC(C)(CCC)C(=O)NCCNC(=O)COCC1CCCCO1 38055,C1(CC=C)(NC(=O)C(F)=C(C)C)CCCN(C(c2cn3c(n2)SCC3)=O)C1 38056,c1(C(=O)NCC2CC(NC(C3(SC)CC3)=O)C2)ccc2c(c1)OCO2 38057,c1(CC(N2CC(OCCNC(C(CN(C)C)O)=O)C2)=O)ccc(Cl)cc1C 38058,N1(C(C(CC)O)=O)CC2CCC1C1CN(C(c3cccc4c3NCCC4)=O)CC21 38059,c1(C(=O)NC(C2N(C(C(CC)n3ccnc3)=O)CCC2)C)ccc2c(c1)OCO2 38060,Cc1conc1C(=O)NC(C1CN(C(c2cnn(C(C)C)n2)=O)C1)C 38061,C1(C(=O)NCC2(C(C)(C)O)CN(C(CSC(C)C)=O)C2)CCCCCC1(F)F 38062,CC(C(C)(C)C(=O)NCC1CC1)NC(c1cnc(CC2(CF)CC2)o1)=O 38063,C1(C(=O)NC(c2cnccc2C2CC2)C)CCCN1NC(=O)C(F)C(F)(F)F 38064,C1(C)(NC(c2cc(C)oc2C)=O)CCC(C(C)(C)C)CC1.C12(C)CCN(C1)C2=O 38065,C(C(F)(F)C(F)(F)F)CCNC(C1C(NC(=O)OC(C)(C)C)CC1)=O 38066,CON(Cc1ccccc1)C(=O)C(CNC(c1cnn(C)n1)=O)C(C)C 38067,n1(CC)ccc2cc(OCCNC(=O)Oc3ncnc(Cl)c3C)ccc12 38068,C1(C(=O)NCCc2ccc(OC)cc2)CC2CCC1N2C(=O)CC1CCCSC1 38069,C#CC(C)(C)C(=O)NC1CC(OCC)C1.C1(C)C(C)(C)OCC(=O)N1 38070,n1(CC(=O)OC)nnnc1C(c1nocc1C)NCCOCC1CCCO1 38071,C1(C(N(CC(=O)NC(C)C)C)=O)CN(C(c2cccn2C)=O)CC1(F)F 38072,c1(CNCC(C(C)C)O)nc(Br)sc1Br 38073,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38074,C#Cc1ccc(OCCC(=O)NCCNC(c2ccc(Cl)cn2)=O)cc1 38075,C1(C(=O)NCCCN(C2CCCC2)C(=O)C2CC2)CCS(=O)(=O)C1 38076,C1(OC)CN(C(=O)CCN2C(=O)CCC2=O)CC1NC(=O)CCC1CCCC1 38077,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38078,N1(C(C(C=C)CC)=O)CC(CNC(=O)CCC(C)C)C(F)(F)C1 38079,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38080,C1(CNC(CC=C)=O)(CO)CCCN(C(C2CCCO2)=O)C1 38081,C1(CNC(C(=O)N(C)Cc2ccn(CC)n2)=O)C2CCCCCC12 38082,N1(C(CN(CCC#C)C)=O)CC2CC(C1)CN(C(=O)CC1CC(OC)C1)C2 38083,C1(NC(c2ccn(C3(C)CC3)n2)=O)CC2CC(C1)CN(C(C1CCOC1)=O)C2 38084,N1(C(C(=O)NC)C2CC(OCOC)C2)CCN(S(=O)(=O)N(C)CCO)CC1 38085,C1(C(=O)NCC(CN(C)C(C2(CCF)CC2)=O)O)CCC=CCCC1 38086,C12C(O)C(O)CCN1C2=O.C1CCCN(C(=O)OC(C)(C)C)C1.CN 38087,CC1CC(NC(c2cccc(C3SCCS3)c2)=O)CCN1C(C1CCCS1)=O 38088,c1(C(N2CC=CC2)=O)ccc(F)cc1OC(F)(F)F.C12CC(C1)NC2=O 38089,Cc1cc(C)c(C(=O)NCc2n[nH]cc2C(=O)NC2CCC(COC)CC2)cn1 38090,c1(NC(=O)NCC(CC)Oc2ccc(OC)cc2)nc(C(F)(F)F)oc1C 38091,c1(C(c2nnnn2C)(Nc2ccc(C(CC)C)cc2)CC)c(C)oc2ccccc12 38092,c1(C(=O)NCC2C(NC(CC(c3cccc(F)c3)C)=O)C2)ncnc2ccsc12 38093,n1(CC(N2CC(CCNC(c3n(C=C)nnc3)=O)C2)=O)nnc2ccccc12 38094,C(CCCCC(=O)N1CC=CC1C(=O)NCCN1CCCCCC1)=CC 38095,CCCC(C(=O)N1CCOCC1CNC(=O)C(C)OCCN(C)C)N(C)C 38096,C(=O)(CC(C)CNC(C1(CO)COC1)=O)N1C(C(CC)O)CCC1 38097,N#Cc1n[nH]c(=NC2CCCC23CN(C(=O)C2CCc4c[nH]nc42)C3)s1 38098,CC1CC=C(C(=O)NCc2cncc(C(=O)NC3CCCC3(C)CO)c2)CC1 38099,C1(C(N2CCC(OC)C2C(=O)O)=O)COC2(C1)CN(C(c1cccc(F)c1)=O)C2 38100,C(=O)(C(C)CCCC(C)=O)N(C1CCN(C(C2CCC(C)(C)O2)=O)CC1)CC 38101,N1(C(C2COC(=O)O2)=O)CC23CCCC2(C1)CN(C(c1cnc(O)s1)=O)C3 38102,C1(CNC(c2cc(NC(C)=O)c(C)cc2)=O)CCN(C(=O)C(C)S)CCC1(F)F 38103,N(C1COc2ccccc21)C(C(C(C)(C)C)NC(C(C)C(F)F)=O)=O 38104,C12(NC(C3(C#N)CC(C)C3)=O)CCCC1N(C(=O)CCOCC(F)(F)F)CCC2 38105,c1(CC(C(=O)OC)NC(=O)CCc2cn(C)nn2)cn(C)c2ccccc12 38106,CC1CN2CCN1C(C(N1CC(NC(c3ncc(F)cc3Cl)=O)C(C)(C)C1)=O)C2 38107,CC1(C)CCN2CC1C2=O.C1(CNC(C2CCC2(F)F)=O)CC(O)C(O)C1 38108,C1(NC(Cc2cn(CC)nn2)=O)CCCN(C(c2sccc2-n2cnnn2)=O)C1 38109,C1(C(N)=O)(CNC(=O)CSc2cccs2)CN(C(=O)CSC2CCCCO2)C1 38110,N1(CC)C(=O)CCC1CC(=O)N(C1CCCN(C(C23CSCC2C3)=O)C1)C 38111,C1(C(=O)NCC2N(C(CN(CCC)C)=O)CCCC2)CCCN(C(C)(C)C)C1=O 38112,N1(C(C(C)C2CCCO2)=O)CCSCC1CCNC(=O)C(C)OC=CCl 38113,c1(C(=O)NCC2C(C)CCN2C(C2CC(F)(F)C2)=O)nc(Cl)ccc1F 38114,C(C(C)C(F)C(=O)NCc1ncc[nH]c1=O)NC(c1cc(C)sc1)=O 38115,C1(CC)(CNC(=O)C(c2ccccc2)F)CCN(C(C2CC23CC3)=O)CC1 38116,C(=O)(NNC(=O)C(CC1CCCCC1)C(C)(C)C)C1(C)CC(C)NC1 38117,N1(C(C(CC(C)(C)C)NC(c2cnn(CC)c2C)=O)=O)CC(C)C12CCOCC2 38118,C(CS(=O)(=O)NCC(=O)NCC1(O)CN(C(=O)C(C)Cn2ccnc2)C1)OCC 38119,c1(CC(=O)NCCN(C(C)C)C(C2CN(CC(F)(F)F)C2)=O)ccc(F)c(F)c1 38120,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)CNC3=O)CC2)=O)O1 38121,C1(C(CNC(c2ccsc2)=O)CO)CC(F)(F)C1 38122,c1(-c2onc(C)n2)ccccc1CC(=O)NCC1CCN1C(=O)CCCN(C)C 38123,C1(CC)CC(C(=O)NCC#CCOC)CCN1C(=O)CN1CC=CC1 38124,c1(-n2c(N(C3CCCCC3)C(C(=O)OCC(C(C)O)O)=O)cnc2)ccccc1F 38125,C(=O)(C(C)C(O)CC)N1CCC(N(C(CC2(C=C)CCC2)=O)C)CC1 38126,c1(C(N2C(C(=O)NC3CC(C#C)C3)C=CC2)=O)ccc(O)nc1 38127,C(C1=CCN(C(=O)Cc2ccsc2)CC1)NC(c1cn(C2CCC2O)nn1)=O 38128,C1(C(N2CCCN(C(CCSc3n(C)nnn3)=O)CC2)=O)CC2CCCCCC12 38129,C1(NC(c2cc(C(C)C)ncc2)=O)CCN(C(c2sccc2F)=O)CC1CO 38130,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(F)n3)=O)C2)C1=O 38131,c1(C(=O)OC)cccc2c1[nH]c(=O)[nH]2.c1(C(CC2CC2)=O)ccncc1O 38132,C=CCN=C(NCCN=c1cc(C)nc(C2CC2)[nH]1)N1CCC(F)(F)CC1 38133,C1(CNC(C2CC(CC)C2)=O)CC2CCC(C1)N2C(=O)C#CC1CCCO1 38134,c1(C(N(C2CCCCC2NC(C2(C)COC2)=O)C)=O)ccc2c(c1)OC(C)(C)C2 38135,N1(C(c2cc(C3CC3)cc(F)c2)=O)CC2CCC2(CNC(C23COCC(C2)C3)=O)C1 38136,c1(C2C3(CC(C(=O)OC)C3)C2)ccc(NC(c2cc(OC)cc(Cl)c2)=O)c(O)c1 38137,C1(NC(c2c(CC)ncs2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38138,C(=O)(C(CNC(=O)C(Cl)Cl)CC(C)C)N1CC(O)(CC=C)C1 38139,C1(C)(C(=O)NCCCNC(c2c(COC)cco2)=O)CCOC1C 38140,c1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)(C)C)cc(C)c(C)c(C)c1 38141,C1(NC(CC2C(C)(C)CCO2)=O)CN(C(=O)CC2=CCOCC2)C2(CCC2)C1 38142,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38143,Cn1c(C(=O)NCC2C=CCN2C(C2CCNC(=O)C2)=O)cc2ccccc12 38144,N1(C(c2ccc(O)nn2)=O)CCC(C2CN(C(C3CN(C4CCOC4)C3)=O)C2)C1 38145,c1(C(=O)NC2CC(CNC(C(N3CCN(C)CC3)C)=O)C2)cc2c(ccn2C)[nH]1 38146,C1(C(C)(C)C)CCN(CC(O)COc2ccc(Cl)c(F)c2)C1(C)C 38147,c1(NC(N2CCN(Cc3c(C)nc(CC)o3)CC2)=O)cnc2ncccc2c1 38148,C12CCN(CC1)C(=O)CCCN2C.c1(C(C)OCC)noc(-c2cccs2)n1 38149,N1(C(=O)CSCC(F)(F)F)CCN(C(=O)Cc2ccc(Cl)nc2)CC1CF 38150,N1(C(CSCC#C)=O)CCC(NC(c2ccc(OC(F)F)c(Cl)n2)=O)C(C)C1 38151,c1(C(N2CC(C)(C(=O)Nc3cncc(C(F)(F)F)c3)C2)=O)ccc(Br)nc1Br 38152,c1(C(=O)OCC)n[nH]c(C)c1[N+](=O)[O-].C1(N)CCCN(C(C2(C)CCC2)=O)C1 38153,c1(C(N2C3CC(NC(c4n(CC)nnc4)=O)C2CC3)=O)cccc2c1OCCO2 38154,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38155,CCCCCCCCC(C)CC(=O)NC1CC(CNC(=O)C(F)(F)C(F)(F)F)C1 38156,C1(CNC(C=CCC)=O)CN(C(=O)CC2CC(SC3CC3)C2)C2CCCC2O1 38157,N1(C(C2C(NC(c3ccc(F)c(O)c3)=O)CCCC2)=O)CCCC(F)CC1 38158,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(F)C3)=O)C2)=O)n1 38159,Cc1ccc(-c2nc(CC(n3cc(CCC4CC4)nn3)C)n(C3CC3)n2)cc1Br.C 38160,c1(C(=O)NCCC(C)N(C(=O)C(O)CC(F)F)C)cccc(S(=O)(=O)C2CC2)c1 38161,c1(CC)ncoc1C(=O)NC(CNC(c1cnoc1-c1ccoc1)=O)C1CCC1 38162,C1(CNC(c2nc(CCC)sc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38163,C1(NC(c2cn3c(n2)CCC3)=O)CCN(C(=O)Nc2ccc(CO)cc2)CC1F 38164,c1(C(=O)NC(C)C(CO)NC(=O)CCCC2CCOCC2)cccc(F)c1Cl 38165,C1(C(=O)NC(C#C)(C)C)(NC(=O)C=CCCC)CCN(C)C1 38166,C(=O)(CC(c1cccs1)n1cccc1)NCC(CN(C(C(=O)N(C)C)=O)C)O 38167,CC1(CNC(c2cc3cn[nH]c3cn2)=O)COCCN(C(C2CCCCS2)=O)C1 38168,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38169,c1(C(=O)Nc2cc(O)n[nH]2)cnc2n[nH]c(-c3cccnc3C(F)F)c2c1 38170,N1(C(C(CSC)(C)C)=O)CC2CCC2(CC(=O)NCCOC2CCOC2)C1 38171,c1(NCC2C(C)(C)CCCO2)ncc(S(=O)(=O)NCCNC=O)cc1Cl 38172,Cc1c(C(=O)NCC2(C)CCN(C(=O)CCCNS(C)(=O)=O)CC2)cncc1Cl 38173,C=CCC(CC(=O)NCc1nc(C#N)cs1)NC(=O)C(CCC)N(C)C 38174,C1(NC(c2cc(OC)nn2C)=O)CN(C(=O)CCCCSC)C(C)(C)C1 38175,c1(C(=O)OC(C)C)cccc(S(=O)(=O)NC2(C)CCC(=O)NC2=O)c1 38176,c1(C(N2CCN(C(C(C(CC)C)O)=O)C(CO)C2)=O)cc(C)c2[nH]nnc2c1 38177,c1(CC(=O)NCC(CNC(c2c(COC)cco2)=O)F)ccc2nn[nH]c2c1 38178,C1(C(C)NC(=O)CC2(C(F)F)CC2)CCCCN1C(c1nc(C(C)(C)C)cs1)=O 38179,N1(c2nc(C#N)cc(C)n2)CCCC2(CCN(C(=O)CNS(=O)(=O)CC)C2)C1 38180,c1(C(=O)NCc2cc(C(N(C)CC3CCSC3)=O)n[nH]2)ccc2c(c1)CCN2 38181,C1(NC(C(C)N2CCCC2)=O)CC2CCC1CN2C(=O)CCCCN(C)C 38182,C1(CC(=O)NCc2cncc(O)c2)C2CCCC2N1C(=O)CC1CC2(CCC2)C1 38183,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(C2CCC2)cnn1C)=O 38184,n1(CC(=O)OC)cc(Cl)cn1.C1(C(C2CN(C=O)C2)C)CCN(C(C2(O)CCOC2)=O)C1 38185,C1(C(N(C)CC2(C)CCC2)=O)CC(O)CN1C(=O)COC1CCOC1 38186,C=C(C)CCC(C(=O)OC(c1ccc2c(c1)OCO2)=O)N1C2CCC1CC(O)C2 38187,CC1COCc2c(NC(=O)NCCCC3CCS(=O)(=O)C3)cccc21 38188,CCN=c1ccc(C(=O)NCC2(F)CCCN(C(c3ccc(SC)o3)=O)C2)c[nH]1 38189,c1(OC)ccc(CN2CCN(C(C3CCCCN3C)=O)CC2C)cc1F 38190,c1(C(N2C(CNC(C3CC34CC4)=O)CCC2)=O)c[nH]c2c(F)ccc(F)c2c1=O 38191,O=S(=O)(CCCCC1CC1)NC1(C2CC2)CCOC1 38192,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38193,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38194,c1(C(N(C(C2CCOCC2)C)C)=O)ccc(CNC(C2CC3(CC3)CO2)=O)cn1 38195,c1(CC)oc(C(=O)NCCC2(O)CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38196,c1(C(N2CC(O)(C(C)NC(c3n(CC)nc(C)c3)=O)C2)=O)c[nH]cc(C)c1=O 38197,Cc1cc(F)ccc1-n1nc(C(=O)NC(C)(C)CNC(=O)CC#N)cc1C 38198,c1(OCC(=O)NC(CN(C(C(C)=CC)=O)C)C)ccc(C#N)cc1Cl 38199,CC1CCC(C)(C(=O)NC2CCCC2NC(=O)CCC2OCCO2)C1(C)C 38200,c1(CNC(C2CCC3(CN(C(CCC(C)C)=O)C3)O2)=O)ccc2ncccc2c1 38201,c1(C(=O)NCC2CC(NC(C3(S(N)(=O)=O)CC3)=O)C2)cn2cc(Cl)cnc2n1 38202,C1(CC(=O)N(C)CC2CN(C(=O)Cc3cnsc3)C2)OCCC1(C)C 38203,C12(C(=O)NC3CCCC(N(C(C(CC#C)O)=O)C)C3)CCOC(C)(C1)C2 38204,CN=c1[nH]cc(C(=O)NCC2CCN2C(C23CCC(CC2)C3)=O)s1 38205,C(CC(=O)N=c1cc(C(=O)O)n(C)[nH]1)N(C(C)C)Cc1scc(C(C)C)n1 38206,N1(C(C(c2nc(CC)sc2)N(C)C(C)=O)=O)CC(C2CCC2)CCC1NC(C)C 38207,C(=O)(CC(NC(=O)COCc1ccon1)NC1CCCO1)NCC(N)=O 38208,c1(C(=O)NC(C(C)C)c2nc[nH]n2)conc1C(C)N(C(=O)CCC1CC1)CCO 38209,C1(C(N2C(CNC(C3CCCO3)=O)CC3CC32)=O)CCc2nc(O)[nH]c2C1 38210,C1(CC(=O)NCCCCCNC(C(CSC)OC)=O)CCCCC12CC2 38211,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38212,N1(Oc2cc(OCC)ncc2)CCC(NC(c2ccc(CO)cc2)=O)C(F)C1 38213,N1(C(CC2CN(C)CC2O)=O)CCC(NC(c2ccc(Cl)cn2)=O)CC(C)(C)C1 38214,N1(C(Cc2n(C)cnc2)=O)CC2CC1CN2C(c1[nH]ncc1C#N)=O 38215,c1(C(=O)NCC(CO)NC(C2C(C3C(C)C3)C2)=O)coc(C#Cc2ccccc2)c1 38216,c1(COC)cnc([N+](=O)[O-])cc1N1CCCC(c2ccccc2)(OCC)C1 38217,O=C(CCCC(c1ccccc1)NC1(F)CCC1)NCc1cccc(F)c1F 38218,N1(C(c2cc(OC)ncn2)=O)CCCN(C(=O)CC2(O)CCCO2)CC1C.C1CC1 38219,C1(NC(c2c(C)oc(-c3ccccc3)n2)=O)C2CC3C1C3C2F 38220,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(C2CCCN(CC(C)C)C2)=O)CC1 38221,C(C(C)CC(=O)NCCN(C(=O)Cn1nc(C(F)(F)F)cc1C)C)OC 38222,C1(NC(CC2(C)CC2)=O)CCC(NC(c2ncoc2CCC(F)(F)F)=O)CC1 38223,C(=O)(CC(O)CNC(=O)CCc1nccs1)N(C)CC1CCCC1 38224,c1(CC(=O)NCCC2CCC(NC(c3nc(CC)oc3)=O)C2)c[nH]ccc1=O 38225,CCCC(C)(O)CC(=O)NCC1(C)CN(C(=O)Cc2nc(C)c(C)s2)CC1C 38226,N1(C(C2C(C)CC2)=O)CCOC(CCCNC(c2cc(C(F)F)on2)=O)C1 38227,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38228,C(=O)(C(CCC)OCC)N(C(C(=O)N(CC=C)CCOC)C)C 38229,Cc1ccc(C(N2CCC3CN(C(C4CCCCC4F)=O)CC23)=O)cc1C#N 38230,CC(CN1CCN(C)CC1)N=c1[nH]c(N2CCSCC2)nc2c(F)cccc12 38231,Cc1nc(O)nc(O)c1CCC(=O)NCC1(O)CCN(C(C2(CCF)CCC2)=O)C1 38232,C(CNC(c1cc(Br)no1)=O)(C(C)(C)C)NC(c1ccc(C(=O)OC)s1)=O 38233,N1(C(c2cnc(-c3ccccc3)o2)C(=O)NCC=C)CC(=O)N2CCCCC2C1 38234,C(=O)(CCCC(C)C)NC1C(NC(CCCc2ccc(C)s2)=O)CCCC1 38235,C(C(C)(CNC(=O)CC1(C)OCCO1)CO)NC(C(N1CC(C)C1)C)=O 38236,C1(NC(c2n[nH]c(C)c2O)=O)(CNC(=O)CC2(C)CCCC2)CCC(C)(C)CC1 38237,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1C#N 38238,c1(OC)ccc2oc(C(=O)NC3CCCCC3NC(=O)C=C3CCC3)cc2c1 38239,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38240,c1(OC)cc(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(C)c2Cl)ccc1F 38241,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38242,Cc1cc(=O)c(C(N2CCOC(CNC(=O)Cn3nccn3)C2)=O)cn1C 38243,C(=O)(C(C)C(O)C(C)C)NC(C(N1CCCC(C)(CC)C1)=O)(C)CO 38244,C1(C(N2CC=CC2Cn2cc(CCN3CCCCC3)nn2)=O)C2COCC12 38245,C1(NC(C(=O)OCC)Cc2cc(F)ccc2Br)CC2(CCC(N)CC2)C1 38246,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)N1CCN(C)C2(C1)CC2 38247,c1(OC)ccc(C)cc1-c1cc(NC(c2cccc(-c3ccccc3)c2)=O)no1 38248,Cc1nnccc1C(=O)NCCn1cc(C(=O)NCC(O)CC2CCCC2)cn1 38249,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38250,c1(-c2cccc(S(N)=O)c2)cnc2[nH]cc(C(=O)Nc3cc(Cl)ccn3)c2c1 38251,N1(C(C(=C(C)C2CC2)F)=O)CCC(N(C(C2C(C)C2(F)F)=O)CC2CC2)CC1 38252,CC1(C2CCN(CC(N)Cc3ccccc3Cl)CC2)CC1 38253,C1(C(N(CC(C)(C)N(C)C)C)=O)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38254,N1(C(C(=O)N2CCC(C)(n3nnc(SCC)n3)C2)(CC)CC)CCc2sccc2C1 38255,N1(CCCc2ccc(OC)cc2)C(=O)CN(Cc2ccc(Br)c(F)c2)C1=O 38256,C1(C(N2CCC(C(C)NC(C(C)CN(C)C)=O)C2)=O)CC(O)CN1C 38257,N1(CC(=O)NC2CN(C(COCCCC)=O)CC2C)CCCc2sccc2C1 38258,c1(C(N2C(c3nc(C)sc3C)CCC2)=O)cc2c(=O)[nH]ccn2n1 38259,S(=O)(=O)(C1CC2(CCCC2)C1)NCC(C1(N)CC1)O 38260,c1(N2CCC(CCC)C2)nc(N2CCN(C3(C)CC3)CC2)c2sccc2n1 38261,C(CCCCNC(=O)C(=O)NCC(F)F)NC(C(C1CCOCC1)OC)=O.C1CN1 38262,C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCN(C(=O)COCC2CC2)CC1F 38263,N12CCC(O)(CC1)CNC(=O)c1ccc(o1)C2=O.C1CCNC1=O.CO 38264,C1(N(C(C(C)OCCC=C)=O)C)CCCN(C(C23CC(C(C)(C)C)(C2)C3)=O)C1 38265,N1(C(C=C2CCC(C)CC2)=O)CCC2CN(C(c3cccc4nonc34)=O)C2C1 38266,CC1CN(C)CC1C(=O)N(C)Cc1ccc(C(F)(F)F)nc1.C12(CC1)C(=O)N2 38267,c12cncc(c1)C(=O)NCC(C)(O)CN(C)C2=O.c1(Cc2ccoc2)cnc[nH]1 38268,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CN(CCCN(C)C(C)=O)C)C1 38269,c1(C(N(CC(CN(C(=O)COCCOCCO)C)O)C)=O)c(N)cccc1Cl 38270,c1(-c2ccc(C(C)OC)cc2)cc(CN(CCO)CC2CCCO2)nc2ccccc12 38271,C=CC1(C(=O)NCC2CCN(C(C3(N(C)C)CCCC3)=O)CC2)CCCCC1 38272,N1(C(CCN(C(C2CN(C(C)C)C2)=O)C(C)C)=O)CCC(O)CC(C)C1 38273,C(C(C)(C)C(=O)NOCc1ccccc1Br)NC(C1COCC(C)O1)=O 38274,N1(C(CC(=O)NC)=O)CCCC(CC(=O)NCC(C)COC)CC1 38275,N1(C(c2c(CCC)n(C)nc2)=O)CCC2(CCN(C(=O)C(C)(CC)OC)CC2)C1 38276,N1(C(C2(CCOCC)CCC2)=O)CCN(C(=O)CCc2cncs2)CCC1C 38277,CCC(CC(=O)N1CCC(C#N)(c2ccccc2)CC1)CC(C)C 38278,N1(C(C(CSC)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38279,c1(C(N(CCC(C)NC(c2cn3ccncc3n2)=O)C)=O)cccc2c[nH]nc12 38280,Cc1csc2c(C(=O)NC3(CNC(=O)C=Cc4ccoc4)CCC3)cccc12 38281,N1(C(COCCCC)=O)C2CCC1CC(O)(CNC(=O)C(F)Cc1ccccn1)C2 38282,C1(CNC(C2C3CCC(F)(F)C23)=O)CCC2CN(C(=O)CC3CC4CCC3C4)CC12 38283,C(C(=O)NCCn1cc(C(=O)NCCC2CCCCC2O)nn1)(C(C)C)OCC 38284,N1(C(C(CC2CCC2)OC)=O)CC(n2cc(Cn3ccnc3)nn2)C(F)(F)C1 38285,c1(C(=O)NC2C(OC)CN(C(=O)C(N3CCC4(CSC4)C3)=O)C2)c(C)cccc1C 38286,C1(C(F)(F)F)(C(=O)NC2CC(F)(C(C)(C)C)C2)OC2CCC1CC2 38287,C1(C(C)NC(=O)CN(C)C(=O)C2CC2)(CO)CCN(C(C2C(C)C2(F)F)=O)C1 38288,c1(OCCC)cccc(C(=O)NC2CC3(C2)CC3NC(=O)COCC(F)F)c1 38289,c1(CC(=O)NC2CCC(CNC(C(F)=C(C)C)=O)C2)nc(C)sc1Br 38290,S(=O)(=O)(c1ccsc1)NC(C1(C)CCN(CC2CC=CCC2)C1)=O 38291,C1(C(C(CC(CC)C)=O)NC(C)C)CC12CCC(F)(F)CC2.c1ccccc1Cl 38292,CC(CCCCNC(C1(N(C)C)CCOCC1)=O)NC(C12COCC1C2)=O 38293,C1(NC(c2n(CCSC)nnn2)Cc2cc(Br)cn2C)CCC2(CC1)CSC2 38294,c1(C(=O)NC2C(NC(C(C3CC3)SC)=O)C2)ccc2cccc(Br)c2n1 38295,c1(OC)nscc1CO.C1(=O)C(COC(C)C)N1.C12CC(F)(C1)C(=O)N2 38296,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38297,C(=O)(CCCNC(c1ccco1)=O)NCC(CNC(c1cnc(Cl)[nH]1)=O)OC 38298,CC(CS(C)(=O)=O)C(=O)NC1CCN(C(C2(c3ccccc3Br)CC2)=O)CC1 38299,C1(C(=O)NCC2CN(C(CC(=O)OC)=O)C(C)CC2)CN2CCN1C(C)C2 38300,c1(N2CC(C)(C)C(CO)C2)nc(NCCN2CCOCC2)c2ncsc2n1 38301,CC1CCN(C(C2(F)CC=CC2)=O)CC1NC(=O)CCc1ccc(O)nn1 38302,c1(C(=O)NC2(C3CCCCN3C(=O)C(F)=CC3CC3)CC2)cc(Cl)c(F)c(Cl)c1 38303,c1(C(N2CCC(NC(c3ncc(CC)nc3)=O)C2C)=O)c(C)oc(C)c1C 38304,C1(NC(C(CC)(F)F)=O)C2CC3C1C3C2C(=O)NCC(C(F)(F)F)OC 38305,c1(N(CCN(C(C(CSC)NC(C)=O)=O)C)C)ncnc2sc(C(F)(F)F)nc12 38306,N1(C(C(C(C)(C)C)OC)=O)CCC(C2(NC(c3scc4c3OCCO4)=O)CC2)C1 38307,c1(C2C(C)C2)ncc(C(=O)NCC2(N(C(=O)Cc3c[nH]nc3O)CCCC)CCC2)[nH]1 38308,C1(c2n(CCOC)nnn2)(NC(C2CCOC2)C)CC2(C1)CC(F)(F)C2 38309,Cc1cc(=NCC2CCC(NC(=O)C(C)OCC3CCCO3)CC2)[nH]c(Cl)n1 38310,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(F)F 38311,C1(C(C)(C)NC(=O)CC2CC2(C)C)CCN(C(=O)CC2COCCO2)CC1 38312,c1(CC(=O)N(C(C)C(=O)NC2CCN(C(C)C)C2)CCC)c(SC)cnn1C 38313,N1(C(c2cc(C)c(C)nc2C)=O)CC(CO)C2(CCN(CCCC#N)CC2)C1 38314,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38315,C1(c2n(C(c3ccccc3C)C)nnn2)(NCCCOC2CCOC2)CSC(C)C1 38316,c1(NC(CC2N(C(c3c(C)nco3)=O)CCC2)=O)cccc(NC=O)c1 38317,N1Cc2cc(Br)ccc2C2CC1C2.N1(c2nc(C)nc(NC)c2)CCc2c(Br)cccc2C1 38318,c1(CCC(=O)N(C(C)C)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38319,c1(N(C2CC2)CC)nc(NC)cs1.C1(=O)C(C)O1 38320,CC1(C)Cc2cccc(NC(NC(=NCCCCl)NC3CC34CC4)=O)c2O1 38321,N1(C(C2C(OC)CCC2)=O)CC2(CC2)CC1CNC(=O)CC1CCNC1=O 38322,C#CCC(C(=O)NC1CCN(C(N)=O)C1)NC(=O)CC1CC1 38323,N1(C(CC(C)F)=O)CC2C(C(=O)NC3CCN(c4ccc(Cl)cn4)C3)C2C1 38324,C=CC(C)(CC)C(=O)N1CCN(C2CN(C(c3sc(C)cc3Cl)=O)C2)CC1 38325,C1(NC(COCCNC(COCCC=C)=O)=O)CCC(C(C)O)CC1 38326,C1(C)CN(C(=O)C(c2nc(C)cs2)C)CCO1.n12ccc(n1)CC(=O)N2.CC 38327,Cc1cccc(CC(=O)NCC2CN(C(c3ncnn3C(C)C)=O)C2)c1 38328,C1(C(=O)NC(c2ccccn2)C)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38329,C(C(C)(CC(C)C)NC(=O)CCc1ccsc1)NC(c1sn(CCC)c(=O)c1)=O 38330,CCC(C)CCCC(=O)NCCCC(C)(C)C(=O)N1CCC1CC(=O)OC 38331,c1(N2CCC(C(C)NC(C3CC3C(N)=O)=O)CC2)nc(Cl)ncc1C1CC1 38332,N1(C(c2c(C)ccs2)=O)CCCCC1C(=O)Nc1ccccc1C(N)=O 38333,c1(C(N2CC(NC(CC3(C)CC3)=O)C2)=O)ccc(-n2cnnc2)cc1 38334,N1(C(CCN2CCN(CC)CC2)=O)CCCN(C(C2(O)CC2(C)C)=O)C(C)C1 38335,c1(C(=O)NCC(C)N(C)C(c2cc(-c3cccs3)on2)=O)csnc1Br 38336,C1(CCN(C(CC#C)=O)C)CCCCN1C(=O)CC1CC1C 38337,Cc1csc2ncc(C(N3CC(F)(CNC(C45CCCC4CC(=O)C5)=O)C3)=O)n12 38338,C1(CN(C(C2CCCC(=O)N2)=O)CC)CCN(C(=O)CC2OCCCO2)CC1 38339,n1(C(C)C)nccc1C(C(=O)NCC1CC=CCC1)N(C)C(c1ccccc1)C 38340,Cc1ccc(C)c(OCC(=O)Nc2ncoc2CNC(=O)CC2CC=CCC2)c1 38341,c1(C(N2CC(C(N3CCC(F)(F)C3)=O)SCC2)=O)c(O)cccc1O 38342,C1(OCCC)CCC(C(=O)NCC(C)NC(c2cnccc2C(F)(F)F)=O)CC1 38343,C1(C)(C(=O)NCCCCN(C)C(C2(C)CC2c2ccccc2)=O)CC(C2CC2)=NO1 38344,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C=CC1CCCCC1 38345,c1(C(=O)NC(CN(C(=O)Cn2nnc(C3CC3)n2)C)(C)C)ccc2nccn2c1 38346,Cc1c(Cl)cc(NC(=O)Nc2ccc(=O)n(CCOC(C)C)c2)cc1Br 38347,C(CC(C)(C)C)(C(=O)N1CCC(CO)(NC(=O)CSC(F)(F)F)C1)OC 38348,C1(CNC(C(CCC)=CCC)=O)COCCN(C(C2(C)CC=C(C)CC2)=O)C1 38349,C(=O)(C1=COCCC1)NCC1CC(NC(C(CCOC)OC)=O)C1 38350,Cc1ccc(CC(N2CCC(CNC(=O)C(C)CCO)C2)=O)cc1 38351,c1(OC)nc(Cl)c(C(N2CC=CC(NC(=O)CNCC3CC3)C2)=O)s1 38352,c1(NC)cccc(OC)c1C(N1CCCCC1CNC(C(COC)(F)F)=O)=O 38353,C1(CN(C(=O)CCCc2ccsc2)CC)CCCN1C(=O)CCCC1OCCO1 38354,Cc1nn(C(C)C)c(C)c1C(=O)NCC(C(C)C)NC(=O)Cc1ccccc1F 38355,C12(C(=O)NC(C3CCN(C(=O)Cc4ccccc4)C3)(C)C)CCC(N=[N+]=[N-])C1C2 38356,N1(C(C(=Cc2cnc[nH]2)C)=O)CC(C(F)(F)F)C(CNC(C2CC23CC(O)C3)=O)C1 38357,c1(CC)cccnc1C(=O)NC1CCC1CNC(c1ccn(C(C)(C)C)c1)=O 38358,Fc1cc(C2(NC(=O)CCN(CC(F)F)CCO)CC2)ccc1Br 38359,CCCCC(O)C(=O)NCC(C(C)C)NC(=O)COCc1cnn(C)c1 38360,c1(OCC)ccc(NC(=O)NC2CC2Br)cc1C 38361,c1(OC)cc(C(=O)NCC2(NC(C3CCN(C)C3C)=O)CCOC2)ncn1 38362,C1(C)(NC(C(C2CCOCC2)OC)=O)CCCN(C(=O)Cc2cccnc2C)C1 38363,C(C(=O)Nn1ccnn1)C1N(C(c2cc(C)[nH]n2)=O)CC1 38364,c1(CC)onc(C)c1C(=O)NC(c1ccc(Br)nc1)CO 38365,CCCC(C#N)C(=O)NCC(CNC(=O)C(CSC)OC)OC 38366,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2ccccc2Cl)C1 38367,N1(CC)CCC(C(=O)NC2CC2CNC(c2sncc2C)=O)C1 38368,C1(NC(C(=C(C)C=O)CC)=O)CC(C(=O)NCCN2CCCNC2=O)C1(C)C 38369,c1(C(N2CC3CC(C2)N(C(C2CC(O)C2)=O)C3)=O)ncn2c1COCC2 38370,c1(OCC)ccsc1C(=O)N(CCNC(=O)CC1C(C)C1(F)F)CC 38371,C=CCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38372,c1(C(N2C3CC(NC(CN(C)S(N)(=O)=O)=O)C2C3)=O)cn2cccnc2n1 38373,c1(NC(=O)C(F)(F)c2cncs2)cc(Cl)cc([N+](=O)[O-])c1O 38374,CC1CC2(CCN(C(=O)CC3CCCCO3)CC2)CN1C(c1nn[nH]c1Cl)=O 38375,c1(C(C)(C)NC(c2ccco2)=O)cn(C2CCC(C(N3CC(C#N)C3)=O)C2)nn1 38376,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38377,C(N=c1[nH]c(N2CCCC(C)C2)nc2c1COC2)c1c(F)cc(C)c(Cl)n1 38378,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38379,N1(CC(=O)NCC(CNC(=O)CN2CCOC2=O)OC)CC2CC2C1 38380,N1(C(C(CC)F)=O)CCC2(CCCN(C(=O)CNc3ccc(Cl)cc3Cl)C2)CC1 38381,N1(C(C(C2CC2)OCC)=O)CC2(CCCC2NC(=O)CC2CCOC2)C1 38382,N1(C(c2c(C)cc(N)cn2)=O)CC2COCC2(C(=O)NC2CCNC(=O)C2)C1 38383,c1(OC)cc(OC)c(C(=O)NCC2CN(C(=O)C(C)C(C)O)C(C)(C)C2)cc1N 38384,CCC(CC(F)F)C(=O)N1CC(N(C)C(C2CCSCC2)=O)C1 38385,CCCCC(C(=O)NCC1CC(OC)C1)NC(c1ccoc1COC)=O 38386,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(c1c[nH]nc1C)=O 38387,N1(C(=O)CC2=CCCC2)CCC2C(CCCN2C(c2noc(C3CCC3)n2)=O)C1 38388,c1(C(N2CCC(N(C)C(C3CC(C(C)(C)C)=NO3)=O)C2)=O)ccc2n[nH]cc2n1 38389,C(c1cnc(C)nc1O)=CC(N1CC(C(N)=O)(CNC(CCC=C(C)C)=O)C1)=O 38390,c1(C(=O)NC2CCN(Cc3c(C)ccs3)CC2)cc(F)cc(Cl)c1 38391,c1(CC(N2CCC(C(=O)NC(C(=O)OC)C3CCC3)C2)=O)ccnc(O)c1 38392,C12(OC)CCCCC(C(=O)NCC(C3CC3)NC(=O)CCn3ccccc3=O)(C1)C2 38393,C1(C)(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C(C)C)n2cnnc2)CC1 38394,c1(OCCc2cccc(CC)n2)cc(Br)c(F)cc1F 38395,c1(CC2CCN(C(C(=O)Nc3nnn(C)n3)c3ccco3)C2)cccc(OC)c1 38396,c1(C(N2C(C3CCN(C(C(CC=C)C)=O)C3)CCC2)=O)ccc(C)c2cccnc12 38397,N1(C(CC2C(C)(C)C2)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38398,C1(F)(C(N(C2CCN(C(C(C)(C)C)=O)C2)CCO)=O)CCCOC1 38399,CN1CCC2CCN(C(=O)CSCCNC(=O)C=CC3CCCC3)CC12 38400,c1(CC)ccccc1CCC(N1CC=CC(NC(C2(C)CC2Br)=O)C1)=O 38401,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(C3(CO)CCC3)=O)C2)c1Cl 38402,C1(NC(C2C(C(=O)OC)CC2)=O)CC2(CCC(NC(=O)CC(C)F)CC2)C1 38403,c1(C(=O)NC(CN(C(c2c(C)snn2)=O)CCO)C)csc2cc(Cl)cnc12 38404,C(CN=c1[nH]cnc2c(Cl)cc([N+](=O)[O-])cc12)NC(N1CCC(C(=O)OC)C1)=O 38405,c1(CCC)cc(C(N2CCC(CN(C)C(c3cc(O)ncn3)=O)C2)=O)ccn1 38406,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)NC.C1(C(=O)O)(O)CC2(C1)OCCO2 38407,n1(CCC)cc(Cl)c(C(=O)NCC23CC2CN(C(=O)Cc2conc2C)C3)n1 38408,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4C)=O)CC23)[nH]1 38409,Cc1nnc2n1CC(C(=O)NCC1CCC13CN(C(C1CC(O)C1)=O)C3)C2 38410,C(=O)(CCCC(C)(C)NC(c1n[nH]c(C)c1O)=O)N1CCC(OC)C(C)C1 38411,C(=O)(C(C)CCCC(C)C)NCC1(C)CCCCN(C(c2cc(C)ncc2)=O)C1 38412,N(C1CCCn2cnnc21)C(CC(C)NC(C(=C1CCCCC1)C)=O)=O 38413,c1(OC)ccc(N(S(C)(=O)=O)CC(C)C)cn1.C1(CC2CCCCC2)C(=O)N1 38414,N1(c2nccc(NC)n2)CC2CCC(NC3CCOCC3)C2C1 38415,C(=O)(C1COc2ccc(F)cc21)N(C1CCN(c2nncs2)CC12CCC2)C=O 38416,N1(C(c2nncc(NCC)c2)=O)CCC(NC(C2CC(OCC)C2)=O)C(F)(F)CC1 38417,C12(C)CCCN(C1)C(=O)C2.C1(C#N)(C(N(C)CC2(COC)CCC2)=O)CC1C 38418,C1(CN(C(CNC(C)=O)=O)C)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38419,C(=O)(CCCCC(C)(C)C)N1CCC(NC(c2c(C(C)C)onc2)=O)C1 38420,c1(OC)cc(C(=O)NCC(C)(C)CC2CN(C(=O)CS(C)(=O)=O)C2)c(C(C)=O)cn1 38421,N1(C(=O)NCC(CC=C)c2ccccc2)CCCC(CCCO)C1 38422,C(CCCCCC(=O)NCCC1CCCC12CC2)c1ccc(OC)cc1 38423,C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(CNC(CCNS(CC)(=O)=O)=O)C(O)C1 38424,N1(C(C2(SC)CC2)=O)CCC2(CCCCN(C(=O)CSC(F)F)C2)C1 38425,N1(C(c2n(C)cnc2C#N)=O)CC(C(=O)NCC(CO)C(C)(C)C)CCC1(C)C 38426,N1(C(C2C3CC4C(C3)C24)=O)CCC(C2CCCN(C(=O)CNC(N)=O)CC2)CC1 38427,N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(=O)C(C)CF)c3nccn32)C1 38428,C(=O)(C#CC(C)(C)C)N1CC(OC)C(NC(c2ccccc2SC(C)C)=O)C1 38429,c12nn(C)c(c1Cl)CC(=O)NCCCC(=O)NC(C)C(CO)NC2=O.CC 38430,N#Cc1c[nH]c(=NC(=O)N(C(Cc2cccc(F)c2)C(N)=O)CCO)cc1Cl 38431,C(N=c1[nH]cncc1C)C1(N(C(CC(n2c(C)ncc2)C)=O)CC)CCC1 38432,c1(C(N2CCN(CCCNC(C3C(=C)C3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 38433,C1(C2(O)CN(C(=O)CC(O)C3CC3)C2)(CNC(Cc2c(C)ccnc2)=O)CC1 38434,C12(CNC(CC)=O)CCCC1N(C(=O)Cc1c(OC)cccc1F)CCC2 38435,N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CN(C(=O)C3=CCC(C)CC3)C2)C1 38436,Cn1cc(C(c2nnnn2C2CCC2)NCC2(CF)CC2(F)F)cn1 38437,c1(C(C)C)conc1CC(N1CC(CC(C)NC(c2c[nH]nc2C2CC2)=O)C1)=O 38438,C1(CC)CN(C(C2CCOC2C)=O)CCN1C(=O)C=Cc1ccc(SC)cc1 38439,N1(C(Cc2c(OC)cccc2Cl)=O)CCC2(CCC2)C(NC(=O)CC(C)F)C1 38440,N1(C(CCCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CCCCC2)C1C 38441,c1(CN(c2n(CCC#C)c(-c3cc4sccc4s3)nn2)C)ccc2c(c1)OCO2 38442,C(=O)(C1CC(=O)Nc2ncn(C)c21)NCCCC(C)NC(C1C2CNC(=O)C12)=O 38443,CCCC(CCC)CC(=O)NC(CC(=O)N1CCN(CC)C(C)C1)C(C)OC 38444,N1(C(c2cc(C)c(F)cc2)=O)CCC2CCN(C(C3CCCC3(C)C)=O)C2C1 38445,c1(CCC)ccc(C(=O)NC2CC(C)(NC(=O)CC3CC3CC3CC3)C2)cc1 38446,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(C(F)(F)F)c2)=O)C1 38447,c1(C(CNC(=O)Nc2ccc(OCC(C)C)nc2)C(F)F)ccc2cc[nH]c2c1 38448,C(C)(CO)(C(=O)NCCCCNC(=O)CCN1CCCCC1)NC(C)=O 38449,C(=O)(C(C)(C)CCCn1cc(CO)nn1)NC(CC)COC(F)F 38450,N1(C(C2CN(C(C(CC)(C)COC)=O)CC2CC)=O)CCOC2C(O)CC12 38451,CC(CO)CCCNC(C1CCCN1C(=O)CC(=O)N(C)C)=O 38452,C(=O)(CCCCC(C)C)N1CCC(NC(C2C(CC)CCC2)=O)(CC)CC1 38453,C1(C(N(C(CNC(C2N(CC)CCC2)=O)C)C)=O)CCc2nncn2CC1 38454,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(C(CC)(C)C)=O)C(C2CC2)C1 38455,c1(C(=O)OC)cncc(-c2cccc(CCNC(C3CCCC3)=O)n2)n1 38456,C(Cn1cccn1)(C(=O)N(C)C(C1CCOCC1)C)NC(C=CC)=O 38457,N1(C(C2CN(C(c3nccc(OC)c3)=O)C2)=O)CCCN(CCCCOC)CC1 38458,C1(CC(=O)NCC(C)N(C(=O)CC(C)=C(C)C)CC)OCCC1(C)C 38459,N12CCC(C(C(=O)NO)C1)C2=O.c1(OC)cc(C(=O)Oc2ccccc2)ncn1 38460,C=CCC(CNC(=O)Cn1cc(C(=O)NC)cn1)NC(C1(CC)CCOC1)=O 38461,C12(C)CCCC1NC(=O)N2.c1(SC(C)C2CC2)cccc(C2CC2)c1 38462,C1(C)(C2CC(CNC(=O)NC(c3nn[nH]n3)C)C2)CCCO1 38463,Cc1ccc(C(=O)NC2(C3CCCN3C(=O)C3=NNC(=O)CC3)CC2)c(Cl)c1C 38464,C1(N(C(CC(=O)OC)=O)CCc2ccccc2)C2CN(C(C3CCCS3)=O)CC12 38465,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C(C)C)cc(C2CC2)n(C)c1C 38466,Cc1nnc(N(C)CCc2ccc(Cl)cc2)n1CC1CCOCC1C 38467,c1(C(=O)N(C2(CNC(=O)COC3CC3)CC2)C2CC2)cncc([N+](=O)[O-])c1 38468,O(NC(=O)C(NC1CC1)OC(C)(C)C)CCOCCOCC 38469,N1(C(c2n(CC)nnc2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38470,c1(OC)c[nH]c(C(=O)NCCC2CCN(C(C3CN4CCC3C4)=O)CC2)cc1=O 38471,c1(CNC(c2cc(NCC3CC(O)C3)ccn2)=O)ccc(F)cc1F 38472,C(CC(O)C(=O)NC1CCCC1NC(c1ccn(C2CC2)n1)=O)N(C)C 38473,c1(C(=O)NCCCCNC(CCC#CC)=O)cc2ccc(C(C)C)cc2[nH]1 38474,N1(C(COCCCC#C)=O)CCCCCC1CNC(C1CC12CC(F)(F)C2)=O 38475,c1(OC)cccc(C(CF)NC(=O)Nc2cnc(C3(C)OCCO3)s2)c1 38476,C1(CC(=O)NCCN(C)C(c2ncc(F)cc2N)=O)CCCC(F)(F)C1 38477,C(=O)(CC(C(C)OC)NC(=O)CCCCn1cccc1)NC(COC)CO 38478,C(=O)(N=c1[nH][nH]c(C)c1Cl)c1cnc(C(c2scc(C)n2)=O)c(Br)c1 38479,c1(C(C)C)ccc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)cc1 38480,C1(c2nnnn2-c2cccc(CC)c2)(NCC=CC)CCCC(F)(F)CC1 38481,C(=O)(CC(=O)NCCCC(C)NC(c1[nH]nnc1Br)=O)NCC#C 38482,N1(C(c2ccc(C#C)o2)=O)CC2CCC1CC2NC(=O)CNc1ccccn1 38483,C1(CNC(CCc2cn(C)nn2)=O)CCCCCN1C(C1CCC(C)(C)CC1)=O 38484,c1(C(=O)NCC2N(C(C(C3CCOC3)OCC)=O)CC(F)C2)cc(N)c(Cl)cn1 38485,c1(NC(C(C2CC2(Br)Br)N(CCOC)CC)=O)ccc(N)cc1.C1(O)CCOCC1 38486,CC1CCN(C(C2CCCCC2(C)C)=O)CC1CNC(c1ccccc1O)=O 38487,C1(NC(C(C)=CC)=O)CC2(CCCN(C(=O)CC3(CSC)CC3)C2)C1 38488,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38489,Cc1ccc2sc(NC(C)CC(C)NC(c3cc4n(n3)CCC4)=O)nc2c1 38490,C1(C(=O)NCCCOCCNC(=O)C=CC2CCCO2)CC(C2CCCC2)C1 38491,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38492,C(=O)(CCS(C)(=O)=O)N(C1CCN(c2ncc(Cl)c(SC)n2)C(C)C1)CCC 38493,N1(C(C(CCF)NC(C(OC)OC)=O)=O)CCC2CN(C)CC12 38494,N1(C(C2(N(C)C)CC2)=O)CCCOC(CCNC(=O)CC2CNC(=O)C2)C1 38495,C1(C(N2C(C(N3CCC(c4ccccc4)C3)=O)CCC2)=O)CC(=O)N(O)C1 38496,c1(C(=O)NC2(CNC(CCC(C)(C)C)=O)CCOCC2)n[nH]c2cnccc12 38497,CC1(C)NC(=O)C2=C1N(c1ccc(Cl)cc1F)C(=S)NC2c1cc(F)cc(Br)c1Cl 38498,C(=O)(CCC(C)CN(C)C)N1CCC(O)(CCNC(C(CC=C)C)=O)C1 38499,N12CCC(C)(C)CC1C(=O)OC1CCN(C1)CC2=O.C1(NC)CCC(COC)CC1 38500,CC1(c2cn(CCCCCC3COCCN3)nn2)CCCC(F)(F)C1 38501,n1(CC)cc(NC(=O)C(c2cccs2)NC(c2cncc(C#N)c2)=O)ccc1=O 38502,C(C(=O)N=c1ccn(C2CCCCC2)[nH]1)=CC(C)NC(C(C)N(C)C)=O 38503,Cn1ncc(C(=O)NC(CNC(c2csc(=N)[nH]2)=O)C2CC2)c1S(N)(=O)=O 38504,c1(OCC(=O)OC)cccc(OC)c1.C(=O)(C(O)C(C)C)NC1CNC12CC2 38505,Cc1c(Cl)c(C(N2CCN(C(=O)C(C)(C)CO)CC2c2cccc(F)c2)=O)nn1C 38506,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)NC(c1conc1OC(C)(C)C)=O 38507,O=C1Nc2ccc(C(N3CC4CN(C(=O)CC5(O)CCC5)C4C3)=O)cc2C1=O 38508,N1(C(C(CC)N(C)C)=O)CCN(C(=O)CC2(C)CC2)C(C(C)C)C1 38509,C1(C2CCN(C(=O)CN3CCCC3C)CC2)(NC(CC(CC=C)(C)C)=O)CCC1 38510,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)N(C(C)COC)C)SCC 38511,CCC(O)C(F)(F)C(=O)N1CCC(NC(c2coc(C(C)(C)C)n2)=O)CC(O)C1 38512,N1(C(CSC2CCCCC2C)=O)CC(C)(C)OC2(C1)CN(C(c1nc(C)[nH]n1)=O)C2 38513,C1(NC(C2C(N)CC2)=O)CCC2(CCOCC2)C1 38514,Cc1ncc2ccc(C(N3CCC(CNC(C4(C5CC5)CC4)=O)C3)=O)cn12 38515,C1(NC(c2nnn(CC)c2N)=O)COCCN(C(=O)COCOc2ccsn2)C1 38516,CCCC(C(=O)Oc1c(C(=O)O)cncc1)NC(=O)OC(C)(C)C 38517,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)Cc3ccnnc3O)C2C1 38518,C1(C(=O)NCCN(C(=O)CCOCCN(C)C)C)OCCC1(C)C 38519,n1(CC)nncc1C(=O)NCC(C1CCCC1)NC(C1CNC(=O)N1)=O 38520,c1(C2(C(N(C(C)(C)CCNC(C3COCCO3)=O)C)=O)CC2)c(F)cccc1F 38521,CCC(CCCC(=O)NCCn1ccccc1=O)NC(c1cn(CCO)nn1)=O 38522,c1(C(C)NC(=O)Nc2ccnc(C(=O)NCCOC3CC3)c2)nnc2n1CCC2 38523,C1(CCN)(OCC)CN(C(=O)C(C)=C(C)C)C1.C1(=O)CC1=O.C1(N)CC1 38524,c1(C(N(CC(CNC(Cn2c(C)nnn2)=O)O)C)=O)ccc(NC=O)cc1 38525,C(=O)(CCCCC(N)=O)N1CCC(C2N(C(C)=O)CC2(C)C)CC1 38526,Cc1[nH]c2ccccc2c1C(=O)NCC1CN(C(C2C3(CC3)C23CC3)=O)CCN1C 38527,N1(C(Cn2nnc(C)n2)=O)CCC2(CCCCC2NC(C2CCC(=O)N2C)=O)C1 38528,O=C(NN1CCCC1C(N)=O)C(O)CCCNC(=O)CCCn1cccc1 38529,C1(C(C2C(C)(C)C2)=O)CC2(CCN(c3cc(C#N)nc(-c4ccccc4)n3)C2)C1 38530,C(=O)(CC(C)CC(C)(C)C)NCC1C(NC(c2cnn(CC)n2)=O)CCCC1 38531,N1(CC(N2CC(F)(CNC(COCc3onc(CC)n3)=O)C2)=O)CC2C=CC1C2 38532,Cc1ccc(F)cc1-c1cn(CCN(C(=O)COc2ccsc2)C2CC2)nn1 38533,c1(CC)ccc(C(N2CC(COC)(NC(c3cc(C)on3)=O)C2)=O)cn1 38534,C1(C(=O)N(C)CC2CCN(C(C3COCOC3)=O)C2)(NC(C)=O)CCOC1 38535,c1(COC)nc(C)c(C(=O)NC(C)(C)CCCNC(=O)CSC(C)C)s1 38536,c1(C(=O)NC2(C)CCN(c3cc(C(F)(F)F)ncn3)C2)ccc2c(c1)CC2 38537,c1(-c2c(C(N(CCNC(=O)Cc3ccsc3)CC)=O)occ2)cccc(C#N)c1 38538,CCC(N=c1[nH]c(N2CCC(CCO)CC2)nc2cc(OC)ccc12)C1CSC1 38539,C(CC(CNC(=O)COC1CC=CC1)NC(c1scnc1C1CC1)=O)OC 38540,C(=O)(C(C)C(O)C(C)CC)N1C(C(N2CCC(C(=O)OC)O2)=O)COCCC1 38541,C1(CNC(C=C=C(C)C)=O)CC2CCC1N(C(c1cc3cc[nH]c3cn1)=O)C2 38542,c1(C(=O)NC2CCC(CCN(C)C)C2)ccc(-c2ccc(Cl)cc2)nc1O 38543,C(=O)(C(F)(F)C(C)(C)O)NCC1CC(NC(CNC(=O)OCC)=O)C1 38544,C1(CNC(C2CC2C(=O)N(C)CC2CCN(C(C)=O)C2)=O)CCC(C)CC1 38545,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38546,N1(C(C(CC(C)C)F)=O)CC2C3CCC(C2C1)N(C(c1cscn1)=O)C3 38547,CC1CCC(NC(=O)CCc2ccc(F)nc2)CN1C(C12CCC(CC1)OC2)=O 38548,c1(CCC(=O)NCCC2CC(OC)CN2C(=O)C(N)=O)cc(F)c(F)c(F)c1 38549,c1(C(N2CC3C(C(=O)NC(C)CS(C)(=O)=O)C3C2)=O)cn(C)c(=O)cn1 38550,n1(CC(=O)NC(CC)CNC(c2cnccc2C(F)F)=O)cnc2ccccc12 38551,c1(C(=O)NC2CN(C(c3c(Cl)cc(C)s3)=O)CC2C)cc2c(Cl)nccc2o1 38552,C1(NC(C(c2ccc(Br)cc2)(C)C)=O)CCC(NC(C2CC2F)=O)CC1 38553,CC1CC(C(=O)NC2(CNC(C3CCS(=O)(=O)CC3)=O)CCC2)CCC1=O 38554,Cc1ccc(C=CC(=O)NCC2(CNC(C3CCS(=O)CC3)=O)CCC2)cc1C 38555,CCCC(C)CC(=O)N1CCC(C(C)C(=O)NC(c2nc[nH]n2)C2CC2)CC1 38556,c1(C2C(F)(C(=O)NCCC3(O)CN(C(c4ccsc4)=O)C3)C2)ccc(F)cc1 38557,N1(C(C(c2ccoc2)NC(CCCC(OC)OC)=O)=O)CC2(CC(CO)CO2)C1 38558,c1(NCCC(=O)NC)nc(N2CCN(C3CCSC3)CC2)cc(C)n1 38559,c1(NCc2ccc(OCC)nc2)ccc(F)cc1C(=O)NC1CNC(=O)C1 38560,c1(CNC(C(C2CCCN(C(C3CCN(C)C3)=O)C2)C)=O)cc(F)ccc1F 38561,C(=O)(C1=CCCCC1)NCC(CN(C(CC1CCN(C(C)=O)CC1)=O)C)C 38562,C1(COC)CCN(C(c2nc[nH]n2)=O)C(C(=O)NCC(C2CCC2)OC)C1 38563,C1(C(=O)NCCNC(COC)=O)COCCC1NC(C1CN(C)CCO1)=O 38564,C1(CC(=O)NCC2N(C(C(C3CCC3)N(C)C)=O)CC2)CCOCC1 38565,c1(-c2n(C(C(=O)NC(C=C)C)C)nnn2)ccc(Cl)cc1 38566,C(C(COC)CC(=O)NCn1cc(CC2CN(C(=O)CC(C)(C)O)C2)nn1)OC 38567,C(CC(F)F)(C(=O)NC1CC2C(C1)C2(F)F)NC(C1(OCC)CC1)=O 38568,c1(C(N2C(CN(C(C(CC=CC)C)=O)CC)CCC2)=O)cc(C)cc([N+](=O)[O-])c1 38569,Cc1cc(C(N2CCC(C)(CNC(=O)Cc3ccnn3C(C)C)C2)=O)cc(C)c1 38570,c1(OCCC(=O)NC(C(C)NC(=O)Cc2ccncc2)C)ccc(C(N)=O)cc1 38571,C1(C)(NC(CC2CC(CC)OCC2)=O)CCN(C(c2sncc2C)=O)CC1 38572,c1(CC)cc(NC(c2coc(CNC(=O)C=C3CCC3)n2)=O)cc(O)c1 38573,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)ccc(N)c(Cl)c1O 38574,c1(N2CC(C(C)NC(=O)CCC3(C)CC3)OCC2)cc(-n2ccnc2)ncn1 38575,c1(C(=O)OC)ccc(-c2nccs2)nc1NC(C1CC(=O)N(C)C1)=O 38576,c1(C2CC(NC(c3c(C)c4c(s3)cccc4)C)C2)ccc2c(c1)OC(C)(C)O2 38577,C1(CC)CN(C(C2CC3CC3C2)=O)CCN1C(C)=O.c12ccnc(Cl)c1NC2=O 38578,C(C(F)(C(=O)NCc1coc(C)n1)C(C)C)NC(C(CC#C)O)=O 38579,c1(CC)cc(CC(=O)NC2CCN(Cc3sccc3Br)C2)n(C)n1 38580,Cc1cccc(N(Cc2cnc[nH]2)CCc2cncc(OC(C)C)c2)c1 38581,C(C(=O)NCC1CCCC(CNC(c2ccc(C#N)cn2)=O)C1)(C(C)(C)C)SC 38582,C(=O)(C(C(C)C)N(c1ccccc1)Cc1c(C)nn[nH]1)NC(c1ccccc1)=O 38583,c1(SCC)conc1C(=O)NCC1CCC(NC(C2(n3cccn3)CCC2)=O)C1 38584,Cc1c(C(=O)NC2CC(C)N(C(c3cccc(N(C)C)n3)=O)C2)noc1C1CC1 38585,Cc1c(C(C)NC(c2cnn(C)c2)C(=O)OC)cccc1Cl 38586,N1(C(C2(CC#C)CCCO2)=O)CCC(C)N(C(=O)CC2(C)CCC2)CC1 38587,C1(OCCNC(C2CC2(F)Cl)=O)CCN(C(C2(Cl)CC2)=O)CC1 38588,N1(C(=O)NC(C)CCn2cncn2)CC(F)(CF)C1 38589,C(=O)(C(CCC1(NC(=O)CO)CCC1)N(C)C)NC1CC(CC(C)(C)C)C1 38590,CCCCC(CNC(=O)C(C)N1CCC1)NC(=O)CC(O)CN(C)C 38591,N1(C(C=CCC)=O)CCC2CN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2CC1 38592,Cc1cc(C(=O)N(CC(C)CNC(=O)C(C)Cc2ccc(F)cc2)C)ccc1N 38593,N1(C(C2CC(COC)C3CC23)=O)CCC(O)(C2(C(=O)O)CCC2)CC1 38594,C(C(C(=O)N(CC(=O)NC(C)C)C)C(C)C)NC(C1(CC=C)CCC1)=O 38595,Cc1ccc(C(N2CCN(C(=O)CC3=NNC(=O)C3)C3CC23)=O)c(F)c1F 38596,S(=O)(=O)(CCC(=O)NC1CCC12CN(C(C1CCC1OC)=O)C2)NC 38597,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38598,Cc1cnc(-n2nnc(CC(=O)NCC3CCCC3C)c2C)c(C)c1 38599,c1(C(=O)NC)cn(CC(=O)NCCCC(C)NC(=O)C(C)n2cncn2)nn1 38600,c1(CC(N2CC(CC(C)NC(c3ccc(C(N)=O)s3)=O)C2)=O)ccccc1O 38601,c1(C(c2nnnn2CC2CCCO2)NCC=CCCC)ccc(OC)cc1 38602,c1(CC)cnc2cc(C(=O)NC3(CCC(=O)OC)CCCC3)[nH]c2c1 38603,c1(OCCC(C)C)ccc(C(=O)NCC(O)CNC(C2CCCN2C=O)=O)cc1 38604,c1(C(=O)NC2CC(C)N(C(=O)CC3(O)CCCC3)CC2)noc2cc(F)ccc12 38605,n1(CC(=O)NCCCCN(C(=O)CCC2(C)CC2)C)cc(N)cn1 38606,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38607,C(=O)(CC(C)F)NC(CNC(CC=CCC)=O)(C)C1CC1 38608,C1(NC(=O)CCc2cncnc2)CCCC12CCN(C(c1ccc(Cl)c(Cl)c1)=O)C2 38609,c1(CCNC2CC(C(C)OC)C2)cccc2c1CCC2 38610,c1(C(=O)NCCN(C(C2C(F)(F)C23CCC3)=O)CC)scc2c1OCCO2 38611,C1(CC=C)OCCC1(c1nnnn1CCC1(C)CC1)N(CC=CBr)CC 38612,c1(C(N2CCN(C(c3coc(O)n3)=O)C3CC23)=O)cc2ncc(Br)cc2o1 38613,Cc1[nH]c(=N)[nH]c(=NCC2CCN(C3CCCCC3)CC2)c1Cl 38614,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38615,C(=O)(CCCCC(=O)OC(C)(C)C)NC1CN(C(C(CC)C(C)O)=O)C(C)C1 38616,C1(CC)(NC(=O)C(C)CF)CN(C(=O)COC(C)C)C1 38617,C(=O)(CCC(CF)CF)N1CCC(CC)(NC(=O)C(CC(C)C)n2ccnc2)C1 38618,c1(C(N(CCC2CCCC2)OC(COCCC)=O)=O)cnccc1Cl 38619,N1(C(Cc2c(F)ccc(C)c2)=O)CCCN(C(c2nc(C)ncc2Cl)=O)CC1C 38620,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38621,N1(C(Cc2ccn(C)n2)=O)CCC2(CCC2)C(NC(c2cn(C)c(=O)n2C)=O)C1 38622,N1(C(c2c(CC)cncc2)=O)CC(NC(c2[nH]nnc2C)=O)CCC(O)C1 38623,CCCS(=O)(=O)C(C)C(=O)NC(C)(C)C(C)NC(=O)C=Cc1ccc(F)cc1 38624,c1(C(=O)NC2(C(=O)NCC(C(CC)C)OC)CC(F)C2)c[nH]c2ccccc12 38625,CC(c1ccco1)=CC(=O)NCC1C2CC1N(C(=O)C(F)(F)c1ncccn1)C2 38626,C=C(C)CC(C(=O)NCCn1ccccc1=O)NC(=O)CC(C)n1cccc1 38627,Cn1ncc(C(F)(F)F)c1CC(=O)CC1(O)CCOCC1.C12CC1C(=O)N2.CN 38628,c1(C(N(C(Cc2c(OC)cccc2)=O)C2CC2)C)ccc(C#N)cc1 38629,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(CC#N)c2)=O)C1 38630,c1(-c2cn(CC3N(C(C4CCC(C)O4)=O)CCC3)nn2)cc(=O)cc[nH]1 38631,Cc1ncc(Cl)cc1NC(c1c(C)[nH]c(C(=O)N(C2CCSCC2)C(C)C)c1C)=O 38632,c1(C(N2CCC(CF)C2)C(=O)OC)cccc(S(N)(=O)=O)c1 38633,C=CCCCCCC(=O)NC(C)(CC)CCNC(C1COCCN1CC)=O 38634,N1(C(C2COCO2)=O)CC2(CCN(C(C3(F)CCCCC3)=O)C2)C1 38635,c1(OCC)ccc(C(N2CCN(C(=O)C(C)C)CC2)C(=O)NC2CCOC2)cc1 38636,N1(C(c2cc(CCC)ncc2)=O)CCC(C2CCN(C(=O)C3=CCCOC3)C2)C1 38637,CS(=O)(=O)C1CCN(C(C2CN(Cc3ccccc3)CC3(CCC3)O2)=O)CC1 38638,c1(CNC(c2c(OC)csc2)=O)ccc(CNC(c2ccncc2)=O)cc1 38639,CSC1=C(C(=O)NC2CCN(C(=O)Cn3ccnn3)C(C)C2)CCCC1 38640,CC(C)(C)C(C)(O)CNC(C1CC1CNC(c1csnn1)=O)=O 38641,c1(CC)nonc1C(=O)NCCCC(c1ccccc1)NC(=O)C=CC(C)C 38642,CC1(C(=O)NC2CCCC2(C)C)C=CCN1C(c1cc(CO)on1)=O 38643,N1(C(c2cc(C)oc2)=O)CC(CNC(=O)Cc2ccsc2Br)C(C)(C)C1 38644,c1(OC)c(F)ccc(F)c1C(=O)NCC1CC(C)N(C(=O)CC2CS(=O)(=O)C2)C1 38645,C=CC1(C(N2CCC(C)(C(=O)NCc3cncc(Cl)c3)C2)=O)CCCCC1 38646,C(=O)(CC1CCOc2ccccc21)NCC1N(C(C2CC(OC)C2)=O)CC(F)C1 38647,c1(C(=O)NC2CC3CN(C(C(C)C#N)=O)CC32)cc2ncccn2n1 38648,Cc1cc(Cl)cc2cc(C(=O)NC3CC3NC(c3cnn4ncccc34)=O)[nH]c12 38649,C1(NC(CC(C)SC)=O)CN(C(=O)Cc2cc(Cl)ccc2O)C(C)(C)C1 38650,C1(NC(CN(C2CCCC2)C)=O)CC=CCC1C(=O)NCC1(CO)CC12CCC2 38651,c1(OC)c(F)ccc(F)c1C(N1CC2CC(NC(=O)C(F)C3CCCC3)C1C2)=O 38652,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(=O)Cc2cccc(C3CC3)c2)C1 38653,c1(OC)cccc(C(N2CCC(C(=O)N(c3ccc(C)o3)C(C)C)C2)=O)c1O 38654,C1(N(C)C)CCCN(C(=O)C(CC2CC2)NC(=O)CCc2ncnn2C)CC1 38655,CC1(C)C2CCC1(C(N1CCC(C(=O)NOCCO)C1)=O)C2 38656,N1(C(C(C)(C)CO)=O)CCC(NC(C2(C(F)F)CC(O)C2)=O)C(F)C1 38657,N1(C(C(C)OCCC(C)C)=O)CC2CC3CC2C1C3NC(=O)CCCCC(C)C 38658,c1(CSC)cccnc1C(=O)N(C(C)CCNC(=O)Cc1nnc(C)s1)C 38659,Cc1cccc2c1CC(C(=O)NC1CCN(C(C3CC(Cl)(Cl)C3)=O)C1)N2 38660,N1(C(C(CC)F)=O)CCCC(CNC(=O)CC2(Oc3ccccc3)CC2)C1 38661,C(c1cncnc1O)=CC(=O)NCC1N(C(c2c(C(C)C)ccs2)=O)CCC1C 38662,c12ccc(c(C(C)(C)C)c1)N(C)c1nnc(CC)n1CCN2.C(=O)(C(F)(F)F)OC 38663,CCCC(CCC)=CC(=O)NCCOC1CN(C(c2c(C)cnn2C(C)C)=O)C1 38664,C(=O)(C#CC1CCCCC1)N1C(C)(C(=O)NC2CC(SC)C2)CCC1 38665,O=C1CCC2(CN(Cc3cc(Cl)ccc3Cl)C2)N1 38666,N1(C(c2cccnc2)=O)CC23CCCCC2(C1)CN(C(C1C2CC2C2CC12)=O)C3 38667,CCC(C)CCC(=O)N1CCCOC(C2CN(C(=O)C(CSC)OC)C2)C1 38668,CC(CC(N)=O)N(C(=O)C(=O)NC1C(c2ccccc2)C1(C)C)C 38669,CN1CCN(CC(=O)NC2CCCCC2NC(=O)C(O)C(F)F)CC1 38670,c1(CNC(c2ccc(C(C)C)nc2)=O)cncc(C#N)c1.C1(C)(C)C(=O)NC1 38671,CCC(CC)C(=O)NCCC(O)CNC(C1CCCC(C(=O)N(C)C)C1)=O 38672,C12(NC(CCC#C)=O)COC(C1)C(NC(c1cc(CSCC)cs1)=O)C2 38673,N1(C(CCOC)=O)CCC2C(CCN2C(c2cnc(F)cc2C)=O)C1 38674,N#Cc1csc(CNC(=O)CN(C(=O)C(O)C2CC2)C2CCC2)n1 38675,C1(CC=C)(NC(c2cncc(OC)n2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38676,c1(NC(C2C(CC)CN(C(=O)Cn3cccc3)C2)=O)cc(CO)ccc1C 38677,C1(NC(C2C(C=C)OCC2)=O)CC2(CCN(C(=O)C=C(C)COC)C2)C1 38678,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(NC(C2CC(O)CN2C)=O)CC(O)C1 38679,C(=O)(C(F)(F)CCn1ccnn1)N(CCCNC(C(N)=O)=O)CC1CCCC1 38680,c1(C(=O)NC2CC(C(=O)OC(C)(C)C)OCC2)ccc(Br)c(C2CC2)c1 38681,c1(CC)ncc(C(=O)NC2(C(=O)N(C)CCC3CCCN3C)CCSC2)cn1 38682,c1(C(C(=O)NC2CCOC2)N(C(C2(C)CC2)C)CC)snc(OC)c1F 38683,N1(C(CCOC)=O)CCCC2(C1)CN(C(=O)C=C1CCOCC1)C2 38684,C1(F)(CNC(C2CCN(CC)C2)=O)CCC(NC(=O)Cc2c[nH]nc2C)C1 38685,Cc1nn2c(c1CNC(=O)C(O)C1CCC1)CN(C(C1CCCSC1)=O)CC2 38686,c1(C(=O)NCCNC(C(C)C)=O)cc(CNC(C2CCCC2O)=O)cs1 38687,CCC(C(=O)NCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38688,N1(C(C2CN(C(C(C)=CC=C)=O)CC2COC)=O)CCCOCC1C 38689,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38690,C1(C(=O)NCC(CNC(=O)CSc2nc[nH]n2)CO)CCCC1C1CC1 38691,N1(C(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)Cc3nccn3C)CC2C1 38692,Cc1cc(C(N2CCC(NC(c3nc(Cl)oc3C3CC3)=O)CC2)=O)ccc1CO 38693,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3F)=O)CC2)C1 38694,N1(C(=O)NC(COC)C(C)C)CC2CS(=N)(=O)CC2C1 38695,C1(OC(C)C(=O)NC(C2CCCN2C(C23CC(C(F)F)(C2)C3)=O)C)CCCCC1 38696,C1(C(=O)NCCC2CC(NC(C=CCOC)=O)C2)Cc2nccn2C1 38697,c1(C(=O)NC(C(C)NC(=O)C(O)C2CC2)C)ccc(Br)c(F)c1F 38698,CCC(C)CC(CO)NC(=O)CCN1CCCC(N(C)C)C1 38699,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2C1 38700,C1(NC(c2c(C)ccnc2C)=O)CC2CCC1C(NC(C1CCC(=O)N1C)=O)C2 38701,c1(C(N2CC(NC(c3c(C#C)cnn3C)=O)C2)=O)cc(C)n(NC(N)=O)c1C 38702,C1(O)(CNC(c2ccc(CNC(c3cnc(=N)[nH]c3)=O)nc2)=O)CCCCCC1 38703,C1(CC(=O)N(C(c2cccnc2)C)C)CN(C(=O)C(N)=O)C(C)(C)C1 38704,c1(C(=O)NC2CCN(C(CCCC(=C)C)=O)CC2CC)nc2ccccc2s1 38705,C1(C(=O)NC2CN(C(CCc3ccc(N(C)C)nc3)=O)C2)CCC(C)NC1=O 38706,CC1=CC(NC(C23CC(CN2C(=O)C(=O)NC(C)(C)C)C3)=O)=C(C)S1=O 38707,C1(C(=O)NC(CC=CC)C(=O)NCC2(CCC)CC2)CCC2CC1CO2 38708,C1(=O)N=C2C=CN(N2)C2CCN1CC2.c1(OC)cc(C)ncc1C#N 38709,Cc1cc(C(=O)NCC(C(N2CCOC3CC23)=O)N(C)C)c(N)c(F)c1 38710,C1(C(N(C2CCN(C(C3CCN(CC4CC4)C3)=O)C2)C)=O)CCCCC12CCC2 38711,n1(CC(N2C3(CN(C(C(C)(C4CC4)OC)=O)C3)CC2)=O)ncc2ncccc12 38712,Cc1ncc2n1CCN(C(=O)C(CO)NC(c1ccc(Cl)cc1)=O)C2 38713,C1(O)(C(=O)OC)CCN(C(=O)CC2CCCNC2)CC1.c12nc(no1)CNC2=O 38714,N1(C(c2cc(CC)c(O)cc2)=O)CC2CCN(C(c3cn(C)cn3)=O)CCC2C1 38715,O=S(=O)(c1ccc(Br)cc1Cl)NCc1ccc(F)cc1OC(F)(F)F 38716,c1(NC(C(n2ccc(C)n2)C)=O)ccc(NC(=O)CSc2nncs2)c(C)c1 38717,N1(C(COCC)=O)CCC2(CC1)CN(C(c1scc(C)c1Br)=O)CC2CO 38718,c1(C(=O)NCCN(C(=O)Cc2nncs2)CC)cnn(CC(C)C)c1 38719,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 38720,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(Cc2ccoc2)C1)C 38721,CCCC(C)(O)C(=O)NCCC1CN(C(=O)C(C)(C)C(=O)N(C)C)CCCO1 38722,N1(C(C)=O)CCCCC1C(N1CCN(c2cc(C(F)(F)F)ncn2)CC1)=O 38723,C1(C)(C(=O)NCC2CN(C(c3ccc(NC)nn3)=O)CC2C)CC(C)OC(C)C1 38724,c1(-c2c(C)n(C)cn2)cnc2ncc(C(N3CC(N4CCC(C)(C)C4)C3)=O)n2c1 38725,c1(NC(CCCC#C)=O)nc(F)ccc1C(=O)Nc1cc(C2CCCCC2)no1 38726,C#CCCC(O)C(=O)NCC=CCNC(c1cccc(-c2ccoc2)c1)=O 38727,N1(C(CCC(=C)C)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 38728,C(C)(C(C)NC(=O)C=CC(C)(C)NC(=O)C=C)(C1CC1)OC.c1(C)ncoc1C 38729,c1(C(=O)NCC(C)(CNC(C2(C#N)CC2C)=O)OC)nn(C)cc1C 38730,C1(C(=O)NC(C(=O)OCCC)(C)C)CC2C=CC1N(C(C1(C(N)=O)CC1)=O)C2 38731,C1(C(=O)NCC2(CC)CCOC2)CN(C(=O)CN2CCNC2=O)C(C)(C)C1 38732,CCC(C#N)C(=O)N(C)CC1CCCC(NC(C2(C(F)(F)F)CCC2)=O)C1 38733,Cc1cn2c(n1)CC(C(=O)NC(C1CCCCN1C(c1csnc1Cl)=O)C)CC2 38734,C1(C2CCN(C(=O)COC(=O)CO)C2)(NC(CC(CCC)C)=O)CC1 38735,c1(C(=O)NC(C)C(C)NC(C2(CCF)CC2)=O)ccc(CN2CCCCC2)cc1 38736,C1(C)(CNC(C2N(C(COC3(C#C)COC3)=O)C(C)CC2)=O)CCC(=O)NC1 38737,c1(C(=O)NC2CC3CN(C(C(COC)NC(C)=O)=O)C2C3)ccsc1S(C)(=O)=O 38738,C(=O)(C(C)(C)CCNC(C1CC12CC2)=O)NCC1CCC(N(C)C)C1 38739,c1(C(=O)NC(C2(O)CN(C(C3(O)CC3)=O)C2)C)ccc(-c2ccsc2)nc1 38740,C1(NC(C2C(NC(C(C)C3(O)CCC3)=O)CCCC2)=O)CC2C(C1)C2(F)F 38741,N1(C(c2cncc(C)c2)=O)CCC(C2(NC(C3CC4(CCCC4)CO3)=O)CC2)C1 38742,c1(C(=O)NCC(CC)NC(=O)CSC)cccc2oncc12 38743,O=C1CCCc2cc(C(=O)NC3CN(Cc4cc(F)cc(F)c4)CC3F)ccc21 38744,c1(NC(C(=O)N(c2ccc(Cl)cc2)CC(C)O)=O)ccc(S(C)=O)c(F)c1 38745,c1(C(N2CCN(CCCNC(CCC=C(C)C)=O)CC2)=O)ccc2nnnn2c1 38746,C1(NC(C2(C#C)CN(C(C3C4CC5C(C4=O)C35)=O)C2)=O)CC2CCC(C1)N2C 38747,S(=O)(=O)(c1cccnc1NCc1ccc(C)cc1)NC(CC)CS(C)(=O)=O 38748,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 38749,C1(C)(CNC(c2c(C)cn(C)c2)=O)CCCN(C(c2ccc(CO)cc2F)=O)C1 38750,c1(CC)cccc(C)c1CN1CCC(C(C)C(=O)NC2CC(F)(F)C2)CC1 38751,C=C(C)C(C)(C)C(=O)N1CCC(OCC2CCN(C(c3n[nH]c(C)n3)=O)CC2)C1 38752,C1(C(C)C)CCN(C(C2CN(C(=O)CC(C3CC3)N(C)C)C2)=O)C(CO)C1 38753,Cc1ccc(-n2nc(CSc3ccccc3)nc2CC2CC=CCO2)cc1 38754,N1(C(C(CC2CCC2)NC(C2(Cl)CC2)=O)=O)CCCCC1C1CC1 38755,N1(CC2CCCN(C)C2)CCC2(CC1)CC2NC(C1CCC(=O)N1)=O 38756,c1(C(N2CC(O)(CNC(C3C(C(=O)OC)C3)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O 38757,C12C3CCCC1CC(C3)N2.c1(C(=O)O)[nH]cc2c1CCCC2 38758,C(=O)(CC(C)F)N(C(C(=O)NC1(CC#C)CCC1)C)C 38759,C1(C(=O)NCC2(C)CCN(C(C3N(CC)CC3)=O)CC2)CCc2cc(F)ccc2O1 38760,C1(N(C(C(C2CCCO2)OC)=O)CC)CCC(C)(C)CC1.C1(NC(=O)NC)CCCC1 38761,C(=O)(CC(C)C(F)F)N(CC(CN(C(c1ccc(C)cc1)=O)C)O)C 38762,C(CCN=[N+]=[N-])N(CC(N1CCCC1CCC1CC1)=O)C 38763,C(=O)(C1=CCN(C(=O)CC(C)(C)COCC)CC1)N1CCCC(CCCC)C1 38764,c12ncccc1C(=O)N2CCC.C(=O)(COC)NCC1(CC(C)C)CC1 38765,C(C)(C(C(=O)NCc1ncc(F)cc1F)C(C)C)NC(C(F)=CCC)=O 38766,C(=O)(CC(C)(C(F)(F)F)NC(c1cn(C)c(=O)n(C)c1=O)=O)NC1(CSC)CC1 38767,N1(C(Cn2cc(C(N(C)C)=O)nn2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 38768,CC1CCC(C(N2CC(CCCCNC(=O)CN3CCOCC3)C2)=O)S1 38769,c1(C(C)=O)ccc(C(=O)NCC(CO)NC(c2ncnc(C)c2C)=O)c(F)c1 38770,N1(C(CCNC(=O)NC)=O)CC2C(CC(=O)NCc3cccc(C(C)C)n3)C2C1 38771,c1(CN(c2cccnc2-c2cccc(Br)c2)C(=O)NC2(F)CCC2)ccc(Cl)cn1 38772,N1(C(=O)Nc2cc(OC)nc(C)c2)Cc2cccn2C(C)C1 38773,c1(C(N2CC(CC=C)(NC(=O)C(C)N(C)C)C2)=O)cc(C(C)(C)C)nn1C 38774,CCC(F)(F)CC(=O)N1CCC(F)CC1C(=O)NOCCCCCC1CC1 38775,C1(n2c(-c3cc(OC)c(Cl)cc3)nc(-c3ccc(CO)o3)n2)CCN2CCCCC12 38776,N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCOC(CNC(=O)CSC2CC2)C1 38777,C(C)(C)(CCCCC(=O)N(C)CC1CN(C(C2CCO2)=O)C1)OC 38778,CCCCC(C(=O)O)OC(C1COC(c2ccccc2OC)C1)=O 38779,C(C(C)(C)C(=O)N(C1CCC(C(F)(F)F)O1)CC(F)(F)F)OC(C)=O 38780,CC(C)(CC1CC1)C(=O)NC(C(=O)Nc1cccc(SCCO)c1)C1CCOC1 38781,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)CC)=O)CCc2nc(C)nn2C1 38782,N1(C(c2c(C)cno2)=O)CCCC2CN(C(=O)C(c3ccc(Cl)s3)C)CCC12 38783,c1(NC)ccc(C(N2CC3CC2C3CNC(c2ccc(OC)nn2)=O)=O)cc1 38784,c1(N(C(C(=O)N(C2C=CCCC2)CC2(C)CC=CCC2)=O)C2CC2)ccccc1C#N 38785,c1(C(N2CCC(CC=C)(CNC(=O)CC(C)CC)C2)=O)cc2[nH]nc(C)c2cn1 38786,c1(OC)ccc2[nH]c(=NCCS(C)=O)[nH]c(=NCCc3cccnn3)c2c1 38787,c1(C(N2CCC(NC(C3(Br)CCC3)=O)CC2)=O)ccc(Cl)c(F)c1F 38788,c1(C(=O)NC2C(C)C2C)cc(C#N)ccc1N 38789,Cc1ccc(CCN(C(=O)CN2CCC(CSc3ccccc3)C2)C(C)C)s1 38790,C#Cc1ccc(OC(C)C(=O)NCC2(NC(C3CCN(C)S3(=O)=O)=O)CCC2)cc1 38791,c1(CN2CC(NC(=O)CC3CCCC3)C(C(F)(F)F)C2)cc(=O)n2nccc2[nH]1 38792,c1(C(=O)NC2C=CC(CNC(C(C)(C3CC3)OC)=O)C2)nc(Cl)oc1C 38793,N1(C(CC(CC)OC)=O)CCOCC(C)(CNC(c2ccc(C)cc2[N+](=O)[O-])=O)C1 38794,CCCC(CCC)=CC(=O)NC(C)CC(C)NC(=O)CCc1nccn1C 38795,c1(C(=O)Nc2ncccc2OCF)ccc2nc(O)n(C3CC3)c2c1.C(CO)O 38796,c1(C(N(CC(CC)NC(c2cc(C)[nH]n2)=O)C)=O)cc(C#N)on1 38797,C1(NC(c2n[nH]cc2I)=O)CC12CCN(C(c1c(Cl)cc(F)cc1Cl)=O)CC2 38798,N(C1CCc2c(Cl)ccnc21)C(c1ccc(N2CC(C)OC(C)C2)nc1)=O 38799,c1(CC)cc(C(=O)NCC2(C)CCC(NC(=O)CC3CCCO3)CC2)ccc1O 38800,C(=O)(CN=c1[nH]c(C)cs1)N(CCCNC(C(CC)c1cccnc1)=O)C1CC1 38801,C1(C)(CC(=O)OC2CCC2)CCN1C(=O)COCCCN=[N+]=[N-].CC1CO1 38802,Cc1cn2c(C(=O)NCCN(C(=O)C(c3ccc(F)cc3)C)CC)c(Cl)nc2s1 38803,C1(CC(C)(C)C)CCN(C(C2(NC(COCCOCC)=O)CCC2)=O)C1 38804,C(=O)(CS(C)(=O)=O)NCCC1CN(C(CN(C2(CO)CC2)C)=O)C1 38805,N1(C(c2n(CCC)ccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1 38806,n1(CC(=O)Nc2scc(C(=O)NCc3cc(C)ncc3)n2)nc(C)c(O)c1C 38807,c1(C(c2cccs2)NC(C2(C(F)F)CC2)C)nnnn1C1COC1 38808,c1(C(=O)NC(CCNC(c2c(CC)nc(C)o2)=O)C)nc(C(C)C)ncc1Br 38809,C(=O)(CCC(=O)N1CC(O)(CCNC(C2C(Cl)(Cl)C23CC3)=O)C1)OC(C)(C)C 38810,C1(CCNC(C(c2ccc(F)cc2)OC)=O)CCCCN1C(c1c[nH]nc1F)=O 38811,c1(OC)ccnc(C(=O)NC(c2cccnc2)CNC(=O)COCCCF)c1O 38812,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 38813,c1(CC(C)C(=O)N2CC(O)(CCNC(=O)C(C)C(F)(F)F)C2)cccc(C#N)c1 38814,C12CCCCC1Nc1cccc(c1)CNC2=O.C=CCCOCCCOC 38815,N1(C(CCCCCC=C)=O)CCC(C2CC2)C1C(N1CC(C#C)C1)=O 38816,c1(CC(=O)NCCCNC(c2c(C)n(C3CC3)nc2)=O)cn2cccc(C)c2n1 38817,N1(C(c2ccc(-c3n(CC)c(C)nc3)cc2)=O)CC2CCC2(C)C1 38818,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC(CC)NC(c1ccc2c(O)n[nH]c2c1)=O 38819,C(N=c1[nH]c2c(c(=NC3CCC4NC(=O)CC34)[nH]1)CC(C)CC2)c1nc(C)[nH]n1 38820,c1(C(N(c2nc(OC)c(F)cn2)C2CCCNC2)=O)cc(O)ccc1[N+](=O)[O-] 38821,c1(C(=O)NCC2CC(CNC(c3c(C)nc(CC)o3)=O)C2)cc2n(n1)CCOC2 38822,c1(CCNC(=NCCC)NCC2(C)CCC2)nc2nc(C)cc(C)n2n1 38823,c1(C(=O)NCC2(O)CN(C(=O)CC3CCCC3(F)F)C2)ccc(C(F)F)nc1O 38824,c1(C(=O)NCC2(O)CCN(C(C(C)OCCC#C)=O)C2)ccc(C)c(CC)c1 38825,C(=O)(C(C)(C)CCCO)NCC1CC2CN(C(c3cccc(OC)n3)=O)CC21 38826,C1(C(=O)NCc2c(C)n[nH]c2)CN(C(=O)CCC(=O)C2CC2)CC12CC2 38827,C(=O)(C1=CC2CCC=CCCC12)NCC1C(C)CCN(C(C2(O)COC2)=O)C1 38828,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 38829,C(CC(C)(C)CC(=O)NCCCCC(C)NC(c1cc(C2CC2)n(C)n1)=O)OC 38830,Cc1ccnc(C)c1NCC12CC=C(CN1C(C)C)C2 38831,C12(CCOCC1)NC(=O)NC2.c1(CC2CC2)ccccc1C1CC1(F)F 38832,CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCN1C(c1cccnc1C1CC1)=O 38833,c1(CC(=O)NCC2C(NC(=O)C=CC3CCC3)C2)nc([N+](=O)[O-])n[nH]1 38834,C(=O)(CCCCCCC)N1CCN(CC(=O)NC2CC(=C)C2)CC1 38835,N1(C(=O)NCC2=CC=C(SC)S2(CC)c2cnn(C)c2)CC2CC1CCC2O 38836,CC(C)CN=C(NCCn1ccnn1)NC(c1ccccc1-n1cccn1)C 38837,C1(CNC(=O)NCc2cc(CC(C)C)[nH]n2)CCNC(=O)C1 38838,Cc1scc(C(=O)NC2CC(CNC(c3cccn3C(C)C)=O)C2)c1Br 38839,c1(C(=O)NC2CCC(CNC(c3ccn(CO)n3)=O)C2)ccc(C2CCC2)cc1 38840,C1(C(N(C)CC2CCN(CC)C2)=O)CC2CCC1N2C(C1COC(=O)N1C)=O 38841,CC(C)C(C(=O)N1CC2CC1(CNC(=O)OC(C)(C)C)C2)C(=O)OC(=O)C(N)=O 38842,C1(NC(CCC)=O)CC2CN(C(c3cn(C)c(OC)n3)=O)CC2C1 38843,Cc1cnc(C#N)nc1C(=O)NC1CN(C(N)=O)C1.C1CCCN1 38844,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 38845,N1(C(c2scc(C)c2)=O)CCN(C2CCCN(C(c3c[nH]cc(Cl)c3=O)=O)C2)CC1 38846,CC1(C(=O)NCC2CN(C(=O)Cn3cc(C(F)F)cn3)CC2O)CC=CCO1 38847,c1(CNC(=O)CC2CC=CCC2)ccc(C(N2CCC(c3cnn[nH]3)C2)=O)cc1 38848,C1(C)(CNC(c2nccc(C)c2Br)C)CC(C2CC2)=NO1 38849,c1(SC)ncccc1NC(=O)CCC1CCCN(C)C1 38850,C1(NC(C2CC2)=O)CCN(CC(=O)NC)C1.N(C1CC1)C1CC1 38851,c1(C(N2CCC(C)(CNC(C3CS(=O)C3)=O)C2)=O)c(F)ccc(Cl)c1N 38852,c1(C(=O)NCCCN(C(C(C)SCC)=O)C2CC2)cc(O)c2[nH]c(C)nc2c1 38853,C12(O)CCCN(C1)C(=O)C1CCC(n3cc2nn3)C1.C1(O)(CCOCC)CCC1 38854,c1(C(N2CCN(CCCCO)CC2)C(=O)NCCCOC)ccccc1OC 38855,C1(NC(C=C(C)C)=O)C2CC(CN(C(C3CCn4cncc4C3)=O)C2)C1CO 38856,C1(NC(c2cc(CC)[nH]n2)=O)CCCCC1CNC(c1cn(C)nc1C)=O 38857,c1(CNC(c2nnc(C)s2)=O)cc2n(n1)CCN(C(C13CCCN1CCC3)=O)C2 38858,N1(C(C2(C)CCCO2)=O)C2CCC1CC(NC(=O)C(CO)NC(N)=O)C2 38859,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 38860,N1(C(c2ncn(C(C)C)c2)=O)CCC2(CCN(C(=O)CSc3cnn(C)c3)C2)C1 38861,C1(OC(C)C)CCCCCC1.C1C(O)C(=O)N2CC(O)(C2)c2cn(nn2)C1C 38862,c1(C(N2C(C)(C(=O)NCc3noc(C)c3C)CCC2)=O)ccc([N+](=O)[O-])[nH]1 38863,C1(C(=O)NCC(C)(CO)NC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 38864,c1(C(CC)(C)C)cn(CC2CC(NC(=O)C(F)OC(F)(F)F)C2)nn1 38865,C1(C(N2CC(C)C(CCNC(C3(C(F)(F)F)CC3)=O)C2)=O)Cc2nccnc2C1 38866,CC1=NNC(=O)C1CC(=O)NCC(N1CCCCC1C(=O)NCc1ncco1)=O 38867,CS(=O)(=O)c1ccnc(N2CC3CC(NC(c4cnc5[nH]cncc4-5)=O)C3C2)n1 38868,C(=O)(CC(CC)N(C(=O)C(C)NC(N)=O)C)N1C(CCC#C)CCC1 38869,CC1CC(C(=O)NOCC(F)F)CCN1C(C1CCCC1F)=O 38870,n1(CC(N2CC(NC(=O)COc3ccon3)C(C(F)F)C2)=O)ccc([N+](=O)[O-])n1 38871,c1(C(=O)OC)cccc(C(=O)NC(CO)C(C)NC(C2CCS(=O)(=O)N2)=O)c1 38872,C(=O)(CCS(=O)(=O)NC(C)C)NCC1(OC)CN(C(c2ccc(OC)o2)=O)C1 38873,C1(C(=O)NCCCC(C)NC(c2sccc2CO)=O)CC2CC1CC2O 38874,C1(CNC(Cn2c(C)cc(C)n2)=O)(NC(C2(O)CCC2)=O)CC2CCC1CC2 38875,Cn1nnc2c1CCC(C(=O)NC1CCN(C(C3(C)CCCC3)=O)CC1F)C2 38876,CC(C)CC(CC(C)C)NC(=O)CC(O)CNC(=O)Cc1ccc[nH]1 38877,N1(C(C2C(C)OCCN2C(C2CCCS2)=O)=O)CC2(CCNC(=O)O2)C1 38878,Cc1cc(C(N2CC(CC(F)C(=O)NC3COCC3CO)C2)=O)sn1 38879,c1(CN(C2CCN(C(CCCCC)=O)C2)C(=O)CSC)cc(=O)c(OC)c[nH]1 38880,c1(C(N2CCC(OCCNC(CCC#C)=O)C2)=O)ccnc(C(N)=O)c1 38881,c1(CNCC(C(C)(C)C)OC)nc2ccccc2o1 38882,C1(C(=O)NC2CN(C(c3ccn(CC)c3C)=O)C(C)(C)C2)CNC(=O)CC1(C)C 38883,N1(CCC(=O)NCC(CC)(C)NC(c2cnc(SC)s2)=O)CCCCC1=O 38884,c1(C(CN2CCOCC2)NCC2(C)C=CCC2)cc(F)cc(Cl)c1 38885,C1(NC(C(=O)NC(COCC)(C)CO)=O)CCCN(C(=O)C=CCF)C1 38886,N1(C(C(Cn2ccnn2)NC(C)=O)=O)CCCN(C(C2(O)CC2)=O)CC1 38887,Cc1cc(C(=O)NC(CNC(c2nc(C(F)(F)F)sc2C)=O)CO)c(N)c(C)c1 38888,N1(C(c2cnc(C)[nH]2)=O)CCN2C(=O)C(NC(=O)CSCCC(C)C)CC2C1 38889,C1(C(N(CCN(C(=O)Cc2ccc(N)cc2)C)C)=O)CC1C1CCCC1 38890,Cc1cccc(CN(C(c2ncccc2C)C(=O)NCC2CCOC2)C)c1Br 38891,Cc1nc(C)n(CC(=O)NC(CNC(c2sc(N(C)C)nc2C)=O)C(C)C)n1 38892,c1(C(=O)NC2CCC(NC(C34CC(C)(C3)C4)=O)C2)nc(C(F)(F)F)oc1Br 38893,C1(NC(C(CC(C)C)C)=O)CCC(O)CN(C(=O)Cn2nnnc2C(C)C)C1 38894,S(=O)(=O)(c1cccc(Br)c1)N1CCC(C#N)(NC(c2c(F)ccc(Cl)c2F)=O)C1 38895,CC1C(NC(=O)C=Cc2ccccc2)C(C)CCN1C(C1CCC=CO1)=O 38896,Cc1nc2ccc(-c3cncc(NS(C)(=O)=O)c3)cc2n1C 38897,N1(C(C2(CC)CC=CC2)=O)CC2CCC(C1)C2C(=O)NCc1ncc(C)o1 38898,c1(C(N2C(CC)CN(C(=O)C(SC)SC)CC2)=O)cc(O)cc(C#N)c1 38899,Cc1c(NC(=O)CNC(=O)C(C)(C)COC2CCOCC2)cccc1Cl 38900,N1(C(CCOCC)=O)CC2C(CN(C)C(C3(CF)CC(F)(F)C3)=O)C2C1 38901,N1(C(C(C(CC)C)N(C)C)=O)CCC2CN(c3ccccc3OC)CC2CC1 38902,c1(C(=O)NCC2CN(C(CCCCSC)=O)CC2O)cc2cc(Cl)ccc2[nH]1 38903,C1(CNC(C(=O)NC2CC2)=O)CN(C(=O)CCC2OCCO2)CC12CCOCC2 38904,C(=O)(C(CC(F)F)NC(C1CC2CC1CC2O)=O)NC1CCN(CCC)C1 38905,O=C1NC(=O)C(CC(=O)NC23CC(C2)N(C(c2ccncc2Br)=O)C3)S1 38906,N1(C(CCc2ccc(N)c(F)c2)=O)CC2ON=C(CNC(=O)C3=CCSC3)C2C1 38907,C(C(=O)NC1CC(N2CCCCC2)C1)(C(C)C)C1CN(C(C(N2CC(C)C2)C)=O)C1 38908,O=C1CN(C(=O)Cc2ccccc2)C(C(N2CCC(O)C(CO)C2)=O)CN1 38909,C1(C2CCN(C(=O)Cc3cnsc3)C2)(NC(C2C3COCC23)=O)CC1 38910,Cc1scc(C(=O)NCC2(O)CN(C(=O)CCc3ccon3)C2)c1C 38911,c1(CNC(c2c(OC)n(C)nc2C)=O)nc2cc(C#N)ccc2[nH]1 38912,CC1CCCc2ncc(C(=O)NC3CN(C(C4(c5cccs5)CC4)=O)CC3C)n21 38913,N1(C(CC(CC)C)=O)CCC(C(=O)NCCCSC(F)F)C(C)(C)C1 38914,Cc1ccc(C=CC(N2CCCC(NC(=O)C=C3CCC(C)C3)C2C)=O)nc1 38915,C1(NC(C(C=C)(C)C)=O)CC1C1CCN(C(c2c[nH]c3cc(C)ccc23)=O)CC1 38916,c1(C(=O)OC)sc(Br)cc1NC(c1coc(CCOC2CCCC2)n1)=O 38917,C1(C(=O)OCC)CC(ONC(C2CCCN2C)=O)C12CCC2 38918,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1(n3cccn3)CCC1)=O)CC(C)O2 38919,C1(NC(C(C)n2ccnc2)=O)CC(NC(C2COCCN2C)=O)C12CCC2 38920,C1(F)(CNC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)CC(C)(C)SCC)C1 38921,c1(OC(C)C(=O)NCC(O)CNC(=O)C=Cc2ccccn2)c(F)cccc1Cl 38922,C1(CNC(C=CC(=O)OCCCC)=O)CN(C(=O)CC)C2CCN1C2 38923,C1(CC)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 38924,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 38925,CC1CCC(C(=O)NCC2(C#N)CCC2)CN1C(=O)C(F)C1CCCC1 38926,C1(CC(=O)N(CC(C)N(C(=O)CCCc2cccs2)C)C)CCC2CC2C1 38927,c1(C(=O)NCCC2CCN(C(c3c(COC)noc3)=O)CC2)cncc(Cl)c1C 38928,N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C=CC2CCCO2)C2(CC2)C1 38929,c1(OC(C)=O)ccccc1C(N1CC2(CC2NC(C2CCCC(OC)C2)=O)C1)=O 38930,Cc1cc(=NCCCS(=O)(=O)C(C)(C)C)[nH]c(NC(c2ncccn2)C)n1 38931,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 38932,C1(NCCOC)CC(NC(=O)C(N2CCN(CCS(N)(=O)=O)CC2)=O)C12CCC2 38933,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1COCCN(C(c2cc(C)no2)=O)C1 38934,C(=O)(CCCC(=O)NCC(O)CNC(=O)Cc1cnn(C2CC2)c1)N(C)C 38935,c1(OC)cncnc1C(=O)NCCSCC(N1CCC2CCC12)=O 38936,c1(CC)cc(C(=O)NC2CCCN(C(=O)C(C)n3cncn3)CC2)ccc1OC 38937,CCC(C)CCCC(=O)NCC(CNC(=O)Cc1cc(O)nnc1O)OC 38938,N1(C(C2(CNC(C3ON=C(C)C3)=O)CCCC2)=O)CCC2(CC1)CSC2 38939,c1(C(N2CCC(C)(NC(COC(C)=O)=O)C2)=O)nn(C)c(C)c1N 38940,c1(C(=O)NC2C(C(=O)NCCC(CC)CO)COCC2)cccc2ccoc12 38941,C(=O)(CC1=Cc2ccccc2C1)NCC(CC)(C)NC(=O)CCCc1cnn[nH]1 38942,Cc1nc2cc(C(N3CCCC3CNC(C3CCN(C)C3)=O)=O)ccc2s1 38943,C1(CC)CCCCC1CNC(=O)CNC(=O)CCOCCOC 38944,C1(CN(C)C(C2CCC(C)(C)O2)=O)COCCN1C(C1CCSC1)=O 38945,C1(NC(c2c(C)cn(C)n2)=O)C(C)(C)C(NC(=O)CS(=O)C(F)(F)F)C1(C)C 38946,C1(C#N)(CC(=O)NC2CCN(C(CCOC(C)C)=O)C2C)CCCCC1 38947,c1(C(Cn2c(C(F)(F)F)ccn2)N)cnc(-c2cnccn2)s1.N1(CC)CCCC1 38948,C1(CCC(=O)NC2CCN(C(CC3C(C)CCO3)=O)C2)CCCN(C)C1 38949,CC1(C)CC(NC(C2(C)CCCC2)=O)CN1C(=O)CC1C=CS(=O)(=O)C1 38950,N1(C(Cc2ccc(C#C)cc2)=O)CC2(C1)CN(C(=O)CCC(=C)C)CCO2 38951,c1(-c2cn(CC(NOCC(Cc3ccccc3)OC)=O)nn2)cc[nH]c(=N)c1 38952,c1(CCC(=O)NC2C(NC(C=Cc3nnc(C(C)C)o3)=O)C2)nnc(O)nc1O 38953,C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1(O)CN(C(C(CC#C)O)=O)C1 38954,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 38955,CC1(C)CN(C(=O)CSc2ccccc2Cl)CC1NC(c1csnc1Cl)=O 38956,c1(C(c2n(CCCSC)nnn2)NCC2CC2)onc(Br)c1C 38957,C1(CNC(C2(SC)CC2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 38958,c1(C(=O)NCC2CCC(NC(C(C)OC3COC3)=O)C2)cnc(C2CC2)nc1O 38959,C(CCN=c1nc2scnc2c(NC(c2nccs2)CC)[nH]1)N(C(C)C)C(C)C 38960,C(=O)(CC1=CCN(C)CC1)N1CCN(C(C2(CCC=C)CC2)=O)C(C2CC2)C1 38961,C(C(N=c1nc(-c2cc(F)cc(F)c2)[nH]s1)C1CC1)NC(C1C(OC)CCCC1)=O 38962,N1(CCC(=O)N2CCC2CNC(c2ccc(Cl)s2)=O)CCCCCC1 38963,c1(OCC(=O)NCCNC(=O)NCc2ncc(Cl)s2)ccc(F)c(Br)c1 38964,N1(C(CN(CC)CC)=O)CC(CNC(=O)C(C)N2CCCC2)C2(CC2)C1 38965,c1(C(N2CC(O)(C(C)NC(=O)CC3CC4COCC34)C2)=O)cc(Cl)c(F)cc1Cl 38966,Cc1nc(NC(C23CC(C(N4CCOC(CCN(C)C)C4)=O)(C2)C3)=O)nc(Cl)c1Br 38967,N1(C(C(=O)NCCCOC)C2=NOCC2)CCC(C2CCN(C)CC2)C1 38968,C1(CC(=O)NC2(CNC(C(CCOC)OC)=O)CCCCC2)CCC(F)(F)CC1 38969,C#CCC(C)(CC)C(=O)NC1C2CC3C1C3C2C(=O)N(CC#CC)C 38970,C1(N=c2[nH]n(C)cc2[N+](=O)[O-])(CNC(C2N(C)CC(C)(C)C2)=O)CCOCC1 38971,N1(C(CC2CCN(OC)CC2)=O)CCC2CC(NC(=O)C(F)=C(C)C)CCC2C1 38972,CCCCCCCCCC(O)CC(=O)N(CC(=O)Nc1cncc(Cl)c1)CCC 38973,CC1CC(C(=O)NC(C)(C)CCCNC(=O)Cc2cnc[nH]2)CCS1(=O)=O 38974,CC1CC(NC(=O)CCC2(C)CC2(F)F)CN(C(C2(C(F)(F)F)CCC2)=O)C1 38975,CC(CF)CC(=O)N1CCCC(CCNC(c2ccc(C(F)(F)F)o2)=O)C1 38976,N1(C(c2c[nH]c(=NCC)s2)=O)CCC2CN(C(c3cnn[nH]3)=O)CCC2C1 38977,CCC(C)(CC)C(=O)NC(C1(O)CN(C(c2cccc(C#N)c2)=O)C1)C 38978,c1(OC)ccnc(O)c1C(N1CC(CNC(=O)C=Cc2ccnn2C)C1)=O 38979,N1(CC(CC)=O)CCN(CC2CCN(C(c3ncc[nH]3)=O)C2)CC1 38980,c1(OC)cnc(C(=O)N(C2CCCN(C(=O)CC3CC(SC)C3)C2)C)c(F)c1 38981,N1(C(c2c(C(C)C)cnn2C)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 38982,C1(CNC(C(OC)OC)=O)(COC)CCN(C(c2c(Br)ncn2C)=O)CC1 38983,C1(C(=O)NC(C(C)NC(C2CC3CC2C3)=O)CO)CC(C)(C)CO1 38984,C(c1cccc(C#N)c1)=NC(N1CCN(C)C(C(F)F)C1)=O 38985,NC1(CN2CCN(C(=O)Nc3ccc(-c4cccc(F)c4)o3)CC2)CCSCC1 38986,C1(NC(C2CCC=CCC2)=O)C=CCN(C(=O)COc2ccc(Cl)nc2)C1 38987,C1(C(C(=O)N(C2CSC2)CC)C)CCN(C(=O)COC2CCCC2)C1 38988,CC(C)(CCNC(=O)Cc1cocn1)NC(=O)CSC(F)F 38989,CC1CC(NC(C23CC2CCN3)=O)CCO1 38990,C1(C(N2CC3C(CNC(CN4CCCC(CC)C4)=O)(C3)C2)=O)CC(C2CC2)=NO1 38991,c1(OC)ccc2c(C(N3CC(CNC(=O)Cc4cnoc4)C(O)C3)=O)cnn2c1 38992,C(C(C)(C)C(=O)NCCC1CCCN(C(=O)CCc2ccccc2C)C1)SC 38993,n1(CC)cccc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C 38994,C1(CNC(c2c(C)snc2)=O)CC2(CCC2)CN1C(=O)Cc1cn(C)nn1 38995,C(=O)(C1=COCCO1)N(C)CCOCCCNC(c1ccc(C(C)(C)C)cn1)=O 38996,c1(C(=O)NC(C(C)NC(=O)CCC(=O)N(C)C)C)nnc2ccccc2n1 38997,N1(C(C(C)OCCOC)=O)CCN(C)C(C(=O)NC2CC(CC)(CO)C2)C1 38998,C1(CC=C)(C(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CSC 38999,Nc1cncc(C(=O)NC2CCCCC2CNC(c2cc(Br)no2)=O)c1 39000,S(=O)(=O)(c1cccc(Cl)c1)NC(CC)C(N1CCN(C(=O)CN(C)C)CC1C)=O 39001,N1(C(C(C(C)C)OC)=O)CC2(NC(=O)C(CO)NC(N)=O)CCC1CC2 39002,CC1CCCN1CC(=O)N(CC(=O)NC(c1cccnc1)CO)C1CC1 39003,N12CCN(C(C3CC3)C1)C(=O)C(C)c1ccc(cn1)C1(CC1)C2=O.C(C)(C)OC 39004,C1(C(=O)NCCNC(=O)C(O)C2CN(C(c3nc[nH]n3)=O)C2)CCOC1 39005,N1(C(C(C=C=C)C)=O)CCCC(CC)(NC(c2cc(Cl)ccc2Cl)=O)C1 39006,C1(NC(C=C(C)C(C)C)=O)CCC(CNC(=O)CCc2ncc(F)cn2)CC1 39007,C1(C)(NC(CC2N(C(C(C)CC#N)=O)CCC2)=O)CCCNC1=O 39008,CC1CCN(C(C2C=CCS2)=O)CCN1C(=O)CCC(C)(C)C#N 39009,c1(N(C2CCC23CCNCC3)Cc2nc(C)sc2)ncc2c(Br)cccc2n1 39010,c1(C(=O)N(CCCC)CCCO)ccc(CNC(C2(C)CC2)=O)cc1 39011,c1(-c2nc(-c3ccc(C(=O)C4CC4)s3)on2)cccc(F)c1 39012,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(C)O)CCNC(=O)COC1CCOC1 39013,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(CNC(COCC(C)C)=O)CC1 39014,N1(C(C=Cc2n(C)ncc2)=O)CCCC2(CCN(C(C3CS(=O)C3)=O)C2)C1 39015,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)N(C)Cc1nnnn1C 39016,C1(C(=O)NCC2N(C(CN3C(C)CCC3)=O)CCC2)CC(S(C)(=O)=O)C1 39017,CC1CN(C(C2COC(C)(C)O2)=O)CC2(CCN(C(=O)CN3CCC3)C2)O1 39018,CC(C)CC(O)CC(=O)N(CC(N1CC(C(N)=O)CC(C)C1)=O)C1CC1 39019,N1(C(c2cncc(OC)c2)=O)CCN(C(=O)CC(C)(F)F)C(C(C)C)C1 39020,C1(C)(C(=O)NCC(CNC(C=C(CC)CC)=O)O)CCCC1O 39021,N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(NC(c2ccn(CC(C)C)n2)=O)C(F)C1 39022,N1(c2cc(NC3CC4CC5C(C4)C35)nc(C)n2)CCc2cc(C)ccc2C1C 39023,N1(C(c2ccccc2)C(=O)Nc2cccc(F)c2)CCc2cc(F)cc(Cl)c2C1 39024,N1(CC)CCCC(CN(C(C2CC(F)C(=O)N2)=O)Cc2sccc2C)C1 39025,CN1N=C(C(=O)N2CC=C(C(=O)NCc3ncc[nH]c3=O)CC2)CCC1=O 39026,N1(C(CC)=O)CC=CCC1CNC(=O)C(c1ccn(C)n1)C 39027,CC(C)(C(=O)N1CCCC(C)(CNC(c2ocnc2C2CCC2)=O)C1)C(N)=O 39028,N1(C(c2ccc(CNC(C3(O)CCCC3)=O)[nH]2)=O)CC2CC(CO)C2C1 39029,C1(N(C(C2CCN(C3CC3)CC2)=O)Cc2nc(CC(C)C)sc2)CCS(=O)(=O)C1 39030,C(=O)(C(C)(C(C)C)N(C)C)NC1(C(=O)NCCN(C)C(=O)OC(C)(C)C)CCC1 39031,N(C1CCCn2ccnc21)C(C(CO)NC(C(C)n1cccc1)=O)=O 39032,c1(C(=O)NCCCCC2CN(C(C(C)NC3CCCC3)=O)C2)ccc(C(N)=O)o1 39033,N=c1ccn(CC(=O)NCC(C2CCCC2)NC(=O)Cc2cnn(C3CC3)c2)[nH]1 39034,c1(C(=O)NC2C(C)CN(C(C3CCCCC3)=O)C2)cc(=O)cc(Cl)[nH]1 39035,c12ccc(F)cc1C(=O)N2.N1(C(=O)OC(C)(C)C)CCC(CCNC=O)CC1 39036,N1(C(c2c(NC)nccc2)=O)CCCN(C(C2OC3CCC2CC3)=O)CC1 39037,C(c1ccc(OC(C)C)cc1)=CC(=O)NC(CNC(c1c(C)coc1)=O)C 39038,c1(C(N2CCC(C3C(C)(C)CN3C(C3CC3CF)=O)CC2)=O)cnn2ccsc12 39039,N1(Cc2ncc(C)c(C(C)C)n2)CC(C)OC2(CCN(C(=O)CSC(C)C)C2)C1 39040,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)Cc2cc(CO)on2)CC(O)C1 39041,C(=O)(NNc1c(C#N)c(C)nn1C)N1CCC(CCCC)C1 39042,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39043,c1(CCCN2CCN(C(C3(CC(C)C)CC(=O)C3)=O)CC2)nc2ccccc2o1 39044,c1(C(=O)NCC2N(C(C(C)OCCC#C)=O)CCC2)ccc(OC(F)(F)F)cn1 39045,Cc1noc(C)c1CC(=O)NCCOCC1CCCC(C(=O)NC2CCC2)C1 39046,c1(CN(C)C(C2CNC(=O)N2)=O)cnn2c1CN(C(c1cnnn1C)=O)CC2 39047,C(=O)(C(O)C(F)(F)F)NCC1(CNC(C(COC)(C)OC)=O)CCCC1 39048,C(=O)(C1=CCC(C)(C)CC1)N1C(C(=O)Nc2cnc(OCC)nc2)CCC(C)C1 39049,c1(C(=O)OC)ccc2c(c1)SCCN(C(=O)Cn1cc(CN3CCCC3)nn1)C2 39050,C1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)C)CCCCN1N=O 39051,C(=O)(C(CC1CCC1)NC(c1cc(C2CC2)[nH]n1)=O)N(CCCOCC)C 39052,c1(-c2nc(CC(C(CC)O)C)nn2CCOC)csc2cc(C)ccc12 39053,c1(C(=O)NC2CCC(NC(c3ccncc3)=O)C2)ccc([N+](=O)[O-])o1 39054,C1(O)(CC(N2C(CN(C(C(C=C)(C)C)=O)CC)CCC2)=O)CCN(C)CC1 39055,C1(OC)CC2(C1)CC1(CN(C(=O)NC3Cc4ccccc4CO3)C1)C2 39056,C(c1cccnc1)=CC(=O)N(CCN(C(CN(CCC#C)C)=O)C)C 39057,C=C(C)CC(C(=O)N(CC1CCC1)OC)NC(=O)CN1CC2CC2C1 39058,N1(C(c2ccc(OC)cc2O)=O)CCC(C)C(NC(=O)CSCC(C)C)C1C 39059,N1(C(CCCNC(C2(CC=C)CC2)=O)=O)CCC12CCCCC2 39060,CCCCCCC(F)C(=O)N1CCC(CNC(c2ccc(O)c(N)n2)=O)C1 39061,c1(C(=O)NC2CC(CNC(C3(C=C)CC3)=O)C2)cccc(C(N)=O)c1N 39062,c1(C(N2C(C)CC(CNC(=O)CNC=O)C2)=O)cncc2[nH]ccc12 39063,n1(CCC)nc(C)cc1C(=O)NCCOC1CN(C(=O)C(N2CCOCC2)C)C1 39064,c1(C(CNC(c2c(COC)nn(C)c2)=O)NC(c2ccc[nH]2)=O)c(C)cccc1C 39065,C=CC1(C(=O)NCc2coc(CC)n2)CCN(C(=O)CC2C3CN(CC)CC23)C1 39066,Cc1cccc(NC(=NCCc2c(F)cccc2Cl)NCCO)c1C(C)(C)C 39067,c1(NCNc2c(C)nsc2)nc(N2CCC3(CCCN3C)CC2)c2c(n1)CCC(C)C2 39068,C1(C(=O)NCC(C)N(C(C(C(=O)OCC)CC)=O)C)CC2(C1)CC(F)(F)C2 39069,C=CCC(F)(F)C(=O)NCC1CCN(C(c2ccc(C3(C)CC3)cc2)=O)CC1O 39070,C(=O)(C(CC(C)(C)C)OC)NC1CC(C)(C(=O)NC(C#C)CC2CCCC2)C1 39071,C1(C(=O)OC)CCCC2CN(C(c3nc(C(F)(F)F)cn3C)=O)CC12 39072,n1(CC(N2CCN(C(CSCC#C)=O)C(C(F)F)C2)=O)c(=O)oc2ccccc12 39073,c1(OC)nc(Br)ccc1NC(C1(F)CCN(C(=O)Cc2cc(F)ccc2Cl)C1)=O 39074,c1(C(=O)NC2CN(C(C3CCC(=O)N3)=O)CC(F)C2)cccc2nccn12 39075,Cc1cccc(OCC(N2CC(NC(c3nnc(S)n3C)=O)CCC2C)=O)c1C 39076,C(=O)(CCN=c1[nH]ccs1)NC1C(NC(C2C3CC(C)(C3)OC2)=O)CC1 39077,n1(CC(=O)N(CCNC(C(N2C(=O)CCC2=O)CC)=O)C)cc(S(N)(=O)=O)cn1 39078,N1(C(c2ccc(C)nc2C)=O)CC2COCCC2(NC(C2SCCS2)=O)C1 39079,C(C)(CO)(C(=O)NC1CCN(C(c2ncoc2-c2ccccc2)=O)C1)NC(C)=O 39080,C(=O)(C(F)C(C)CNC(=O)Cn1ccnn1)NCC1(C)C(=O)N1.C(C)(=O)OCC 39081,C1(NC(C2(S(N)(=O)=O)CC2)=O)CN(C(C2CCCC(C3CC3)O2)=O)CCC1CO 39082,c1(OC)ncc(C(N2CC(C)(NC(C3CCC(OC)C3)=O)C2)=O)c(C(F)F)n1 39083,CC1(C)OCC2(CCN(C(C3CN(c4c(F)cccc4F)C(=O)C3)=O)C2)CO1 39084,C(=O)(CC(C)(C)CC(F)(F)F)NC(C(C)C)CNC(=O)Cc1cnc[nH]1 39085,CC(C)S(=O)(=O)c1ccc(C(N2CC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cc1 39086,CC(C)(C)C(O)C(=O)N1CCC(C(C)(O)CNC(C2CCC(CO)CC2)=O)CC1 39087,N1(C(CSC(C)(C)C)=O)CCC2CCN(C(C3CC4(C3)CC43CCC3)=O)CC12 39088,CCCC(CCC)CC(=O)NC1(C(=O)NCC(C)(COC)CC)CC(F)(F)C1 39089,c1(C(C)=O)ccc(C(=O)NC2CCC(CNC(c3ccc(Br)s3)=O)C2)o1 39090,C1(CNC(Cc2cc(C)[nH]n2)=O)COCCN(C(=O)Cc2ccccc2F)C1 39091,C1(NC(C(CC)OCC)=O)CN(C(c2cn(C(C)(C)C)nc2C)=O)CC12CC2 39092,C1(C(N2CCC(CC(=O)OC)C2)=O)N(C(=O)Cc2ccn(C)n2)CCC1(C)C 39093,c1(C(=O)NC2CCC(CNC(c3c(C)nc(C(C)C)o3)=O)C2)cccc(N)c1O 39094,C=CC#CC(C)(C)NC(=O)C(C)NCC=CCC(=O)OC 39095,N1(C(C2(C)CCNC2=O)=O)CC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(C)(C)C1 39096,C1(=CC(=O)NCc2cn(CC(=O)NCCCCC3CC3)nc2)CCCCCC1(F)F 39097,C1(CNC(c2c(CC)ncs2)=O)CCC(C)CN1C(c1cc(C2CC2)nn1C)=O 39098,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)CSC(F)F)C(CC)C1)=O 39099,n1(CCC)ncc(C(=O)NCCN(C(=O)CCC2CCC(O)CC2)C)c1C1CC1 39100,N1(C(c2ccc(C(C)=O)cc2)=O)CCC2(CCC(NC(=O)OC(C)(C)C)CC2)C1 39101,C1(C(=O)OCC)C=CC(C(=O)NC2CC(NC(=O)CCN3CCOC3=O)C2)C1 39102,C1(C(=O)NCC2(CNC(CC=CC)=O)CCCC2)CCC(C)(O)CC1 39103,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39104,CCCCS(=O)(=O)NCC(N1CCC(CCOC)(NC(=O)Cn2ncnn2)C1)=O 39105,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39106,N1(CC(=O)NCC(C)C)CCN(C(=O)CCC(=O)C2CNCCO2)CC1 39107,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)CCNC(=O)OC)CCO2 39108,C1(NC(C2CCC(CC)CC2)=O)C2CC3C1C3C2C(=O)N(C1CCCC1C#N)C 39109,C1(NC(C2C(C(C)C)CCCC2)=O)CC(N=c2[nH]c(C(F)F)nc(=N)[nH]2)C1 39110,N1(C(=O)COCC2CCOC2)CC=C(CCNC(C2(n3cccn3)CCC2)=O)CC1 39111,C(=O)(C(CCc1ccccc1)C(C)(C)C)NC(CC1CN(C(CCC)=O)C1)C 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39148,N1(C(C2C(C)C2C)=O)CC(CNC(=O)CC2CC(C)OC2C)OC(C)(C)C1 39149,N1(C(c2cc(C)c(C)o2)=O)CCC(C2CC2NC(C2CCC3CC23)=O)CC1 39150,c1(CC)ccc(CNC(=O)C(N)Cc2ccc(F)cc2)cc1C 39151,N1(C(CCC(C(C)C)NC(=O)C(C)(C)CO)=O)CCC(C2CCOC2)C1 39152,N1(C(C=C(C)CNC(=O)C(C#N)C(C)C)=O)CC(=O)NCC12CC2 39153,c1(CN2CC(C)C(N3CCOCC3)C2)cc2c(Cl)nccc2s1 39154,C1(CCNC(CCOC)=O)CCCCN1C(=O)C(N1CCC(C)CC1)=O 39155,C1(C(N2CCC(=CCNC(c3c(CC)nns3)=O)CC2)=O)CN(CP(C)(C)=O)C1 39156,C1(CC(=O)NCC2(C(C)(C)C)CCC2)CCN(C(c2cnn[nH]2)=O)C12CCC2 39157,N1(C(CCOCCC)=O)CCCC1C1CCCCN1C(=O)C(=O)NCC(F)(F)F 39158,c1(OC)ccc(OCCC(=O)OCc2ccc(SC)cc2)c(Cl)c1C#N 39159,c1(CNC(c2n(CCOCC)nnn2)(CC)CC)cc(OC)c(C)cc1OC 39160,CC(C)CCC(C)OC(C1C=CCCC1CC(=O)OCc1ccccc1)=O 39161,C1(N(C(Cn2ncc(C)c2)=O)C)CCC(CNC(=O)CC2CCC(=O)O2)CC1 39162,c1(C(=O)NCC2CN(C(C(C(C)C)SCC)=O)CC2(C)C)cc2n(n1)CCCC2 39163,c1(C(=O)OCC)cccc(COC(=O)CCN(C)CCO)c1 39164,CCC(C)CCC(=O)NC(c1ccc(F)cc1)CNC(=O)C=Cc1cc[nH]c1 39165,C1(NC(C(=O)NC(C)C)=O)CCOC(C(=O)NCC2COCC(C)O2)C1 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39202,c1(C(C#C)NC(=O)Cc2cccc(N3CCCC3=O)c2)cccnc1OCCO 39203,c1(NC(=O)CCC2CCN(C(c3ccc(C(F)F)o3)=O)C2)ccc2ncnn2c1 39204,C(=O)(CCCC(OC)OC)NCCCOCCCNC(CC(CC)C1CCC1)=O 39205,Cn1cc(NC(c2ccn(C)n2)c2nnnn2C2COC2)c(C(N)=O)n1 39206,c1(C(=O)NC(CCC)C(=O)N2CC3(CCC3)C2)cc(C#N)cn1C 39207,C(=O)(C(CC)CC(F)F)NCC(=C)CCNC(=O)CSc1nnc(S)s1 39208,CN=c1[nH]cc(C(=O)NC2(C(=O)NC34CC(C3)C4)CCCC2)s1 39209,N1(C(CCc2c(C)nn(C)c2)=O)CC(NC(c2c(C)nc(C)n2O)=O)CCC1C 39210,CCCCC(O)C(=O)NCCc1cc(C(N2CCCC(C)C2CO)=O)no1 39211,C1(C(=O)NCCc2n(C)c(=O)on2)C2CC3C(C2NC(=O)CC2CCC(=O)C2)C13 39212,C1(c2ccc(OC)nc2C)NC(=O)N(CCF)C2=C1C(=O)N(C)C2C 39213,c1(C(N2C(C(C)(C)NC(C(=O)OC3CC3)=O)CCC2)=O)ccnc2ccccc12 39214,C1(N(C(c2nc(CC)oc2)=O)C)CCN(C(=O)C(C2CCC2)C2CCC2)CC1C 39215,CC1(C)CCCC1C(N1CCCC(c2cn(-c3cncc(Br)c3)n[n+]2[O-])C1)=O 39216,c1(C(N2CC3C(CNC(CS(=O)(=O)NC)=O)(C3)C2)=O)c[nH]c2cc(N)ccc12 39217,N1(C(C)=O)CC(F)CC1C(N1CCC(C(C)NC(=O)Cc2ccon2)C1)=O 39218,N1(C2CCN(C(C)C)C2=O)CC2CN(C(=O)CCCN=[N+]=[N-])CC2C1 39219,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(C(=O)Cc3ccc(C#N)cc3)CC12 39220,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39221,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)NCCOCC(F)F 39222,C=CC(C)(O)C(=O)NCC1CC1NC(=O)CCn1ccnc1-c1ccccc1 39223,c1(NC(c2ccc(C)cc2)C2CC2)n[nH]c2c(C)cccc12 39224,Cc1cccc2c1CCN2CCc1ncnc(NCCOC2CCC2)c1C 39225,Cc1ccc(C2=NOC(C(=O)NCC3CC(NC(C4CC4C4CC4)=O)C3)C2)cc1 39226,S(=O)(=O)(c1ncc(F)cn1)NCC(C)(CO)CO 39227,c1(CSC)noc(C)c1CN=C(NCC1CCC1)NC1CC1(C)C(F)(F)F 39228,C(C)(C)(C(C)NC(=O)CCCc1cc(C)no1)NC(CSCC)=O 39229,C1(Cn2c(-c3cc[nH]n3)nc(-c3ccsn3)n2)CCC12CC(F)(F)C2 39230,c1(C(=O)OCC)ccc2c(c1)CCN(N1CC(OC(F)F)C1)C2 39231,N1(C(C2CC(C#N)C2)=O)CCC(O)(CCNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 39232,c1(NC(C2(C)N(C(c3c(OC)n[nH]c3)=O)CC2)=O)cc(C#N)cn1C(C)(C)C 39233,c1(C(=O)NCC(C)N(C(=O)CC=CC(C)(C)C)C)ccc2nc(=N)[nH]n2c1 39234,N1(CCC(CC2CCN(c3nc(C)cc(C)n3)C2)=O)CCCC2CNCC12 39235,Cc1cc(-c2cnn3c2CCC3)c2cc(C(=O)N)ccc2n1.c1(C(N)=O)cn(C)nn1 39236,CCC(CC)C(O)CNC(=O)CC1CN(C(=O)CCc2ccco2)CC1C 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39307,C1(SC)CN(C(=O)CCn2cc(Cl)cn2)CC1NC(C1CCNC1=O)=O 39308,C(C)(N=c1cc[nH]cc1S(=O)(=O)N1CCC(C2(C)CCCO2)C1)c1n(CC)ncc1 39309,c1(NC(C2CCCC(NC(C(C=C)(F)F)=O)C2)=O)cccc(F)c1C 39310,CC1CCOC(C(=O)NCC(F)CNC(c2cncc(-c3ccncc3)c2)=O)C1 39311,c1(C(=O)NCCN(C(c2c[nH]c3nccc-3c2)=O)CC)sc2cncn2c1C 39312,c1(NC(C2(NC(c3nc(C)sc3)=O)CCCCC2C)=O)cnc2c(c1)COCC2 39313,N1(C(N(C)CC2CC2)=O)CCC(Cc2c(CC)nn(CC)c2)C(O)CC1 39314,c1(CC(=O)NC(C2CCN(C(C34CSC(C3)C4)=O)CC2)C)c(F)cncc1Cl 39315,N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 39316,c1(NCC(C)NC(C2(c3ccc(Cl)cc3)CC(F)(F)C2)=O)ncn(C)c(=O)c1Br 39317,c1(CN(C)CCN(C)C)cccc(-c2cc(OC(F)F)ncn2)c1 39318,C1(C(=O)NC(COC)CC(C)C)CCN(C(=O)OC(C)(C)C)CCO1 39319,C1(CNC(c2n(C)cnc2)=O)CCCN(C(=O)Cc2ccn(CCF)n2)CC1 39320,C(CCCCC(=O)NCc1nc(C(=O)NCC2COC(C)(C)C2)co1)=CC 39321,C(C1=NOC2CCCC12)NC(CCCCc1ccccc1)c1n(C(C)C)nnn1 39322,C1(C)(C(=O)NCc2cccc(CN(C(CNC(=O)NC)=O)C)c2)CCCS1(=O)=O 39323,C1(NCC2CCCN(C(C3(CS(C)(=O)=O)COC3)=O)C2)OCCOC12CCC2 39324,c1(OCC)ccc(C(N2CCN(C(=O)NCC3CCOCO3)CC2)=O)cc1.CC 39325,Cc1cc(C)n2ncc(C(N3CC(n4cc(CCCCO)nn4)C(C)C3)=O)c2n1 39326,c1(C(=O)NCC2(F)CCCN(C(c3c(SC)snn3)=O)C2)ccc2[nH]ccc2n1 39327,N(C1CC(C)(C)CCc2ccc(Br)cc21)C(c1ccc(CSC)o1)=O 39328,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC)C1 39329,Cc1cc(NC(N2CC(n3cc(C(F)(F)F)c(C)n3)C2)=O)ccc1I 39330,CCCC(C(=O)N1CCC(N(C)C(c2cn(CCC3CC3)nn2)=O)C1)C(C)C 39331,c1(C(=O)NC2C(NC(=O)Cc3ccncc3Cl)C2)ccn2cccnc12 39332,N1(C(C(c2ccc(C)cc2)=O)=O)CC(NC(C2CC2C(F)(F)F)=O)CC(C)(C)C1 39333,C(C(C)CC(=O)N1CCC(C)(C(N)=O)C1)NC(C(OCC)OCC)=O 39334,c1(NC(=O)C=Cc2cnccn2)ccc2c(c1)CN(C(=O)C1=CCSC1)C2 39335,Cn1c(I)cc2c(N(C(c3cnnc(Cl)c3)=O)CC3(O)CNC3)ncnc12 39336,N1(C(c2cccc(C(N)=O)n2)=O)CCCC12CCN(C(c1cnc(O)[nH]1)=O)CC2 39337,C1(c2onc(C(C)N)n2)CCN(C(=N)NCCF)CC1 39338,C12(C(=O)NCCCOCCCNC(c3c(C)nc(C4CC4)[nH]3)=O)COC(CCO1)C2 39339,c1(C(=O)NCC(C)(S(C)(=O)=O)NC(=O)OC(C)(C)C)nnc2ccccc2c1O 39340,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)C=CCl 39341,C(CCNC(=O)C(=O)Nc1c(C)csc1C)(C(C)C)NC(C(C)OCCC=C)=O 39342,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)c3)=O)C2)C1 39343,C1(CC)(CNC(=O)C(c2cncnc2)C)CN(C(C2CCC2C(=O)OC)=O)C1 39344,C(=O)(C(C)(O)CCc1ccccc1)NCCC(C)NC(CCCOC)=O 39345,c1(C(c2nnnn2C2COC2)Cc2c(COC(C)C)ocn2)ccc(Br)cc1Cl 39346,C1(NC(CCC#C)=O)CC(CNC(=O)CCc2nc(-c3ccoc3)no2)C(O)C1 39347,N1(C(CC2C(CC)C2)=O)CCC(F)(F)C(CNC(C2(C(F)(F)F)CCCC2)=O)C1 39348,N1(C(COCc2ccc(C)cn2)=O)CCCC(NC(=O)Cc2ccsc2C)CC1 39349,C1(C(=O)NC2CCC(NC(C(CC)OCC)=O)CC2)CCC2CC2CC1 39350,c1(OC(C)C)ccc(C(=O)NCCCCN(C)C(C2CCC2C)=O)cc1 39351,C1(n2cc(C(C(C)C)N(C)C)nn2)CCCCN(C(C2CN3CCCC2C3)=O)C1 39352,c1(CC(=O)NC)cc(CC(=O)NCC(=O)NCCNCCOC)on1 39353,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39354,c1(CC)ncc(Cl)c(C(=O)N(C)CC2CCCCN2C(c2cnoc2)=O)n1 39355,Cc1nsc2ncc(C(=O)NC(C3CCCN(C(=O)C(F)CC4CC4)C3)C)cc12 39356,C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CC1N(C(C1(C(N)=O)CCCO1)=O)C2 39357,CC(C)(CCCCNC(C1CC=CC(O)C1)=O)NC(C1CC1C1CCC1)=O 39358,C(=O)(C(CCSC)NC(=O)CC1CC(NC(C)=O)C1)NC(C(=O)OCC)C 39359,c1(C(N2C(C)CC(CNC(=O)Cc3cncn3C)C2)=O)cnc2ncc(Cl)cn12 39360,CC1(C(=O)NCC2COCCN2C(C2COCCN2C=O)=O)CCCNC1=O 39361,N1(C(C=Cc2scc(C)n2)=O)CCC(C)C(CNC(=O)C(c2cccnc2)C)C1 39362,C1(CNC(c2nnn(CC)c2C)=O)CN(C(c2nn(C)cc2N)=O)CCC1C 39363,C1(O)(C(COC(C)C(=O)NCC2CC2)(C)C)CN(C(c2csc(C(F)F)n2)=O)C1 39364,C(C1CN(C(=O)C2=CCCCC2)CC1C(=O)NCC(C)(C)CC)=CC 39365,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncn1C 39366,C1(C(=O)NC(C)Cc2nc[nH]n2)CN(C(=O)CCCc2ccccc2)C(C)(C)C1 39367,CC1CCCc2ncc(C(N3CCCC(C)(NC(=O)C4=C(Cl)CC4)C3)=O)n21 39368,CCCCCCC(C(=O)NCC1CN(C(c2scnc2C)=O)CC1O)NC(C)=O 39369,c1(NCCOC)cc(=NCC(N)CCSC)[nH]c(CSc2ccc(F)cc2)n1 39370,C(=O)(C(CC1CC1)OCC(=O)N(C(C)C)CCOCCCN(C)C)N.C(C)(C)C 39371,N1(C(CCC=C(C)C)=O)CCc2ccccc2C1CNC(=O)CC1COCC1O 39372,C(=O)(C(CNC(c1cnsn1)=O)CC(C)C)NCc1nc(COC)on1 39373,C1(NC(c2cc(CO)ccn2)=O)C2CCC(C2)C1C(=O)NC1CC2CC3C(C2)C13 39374,c1(OC)cc(C)ccc1CNC(=O)NCCC(C(=O)N(C)C)OC(C)(C)C 39375,CCC(C)(CCC(C)C)C(=O)N(CC(C)(C)NC(c1n[nH]c2c1CC1CC21)=O)C 39376,Cc1cn2cccc(C(=O)NC3CCSC34CN(C(c3ccc(C)o3)=O)C4)c2n1 39377,c1(C(=O)NC(CC(C)NC(CC2(OC)CC2)=O)C)c(C)ccnc1O 39378,C1(C)(C(=O)NC2(COC)CC2)CN(C(C2CCC2)=O)C1 39379,C(=O)(C#CC1CCOCC1)NCc1c(C(=O)NCC2CCCN(C)C2)n[nH]c1 39380,c1(C(N(C)CC2CCN(c3c(F)cnc(OC)n3)C2)=O)cccc2c1CCC2 39381,N1(C(C(COC)C)=O)CCC2(CCCN2C(=O)CCN(c2ccccc2)C)CC1 39382,c1(C(C(=O)NCCCN(C(C2CCC(F)C2)=O)CC)(C)C)cccc(Cl)c1 39383,C1(C)(CNC(Cc2c(C)occ2)=O)CC(F)(F)CN1C(c1ccc(C)nn1)=O 39384,C1(C2(O)CN(C(=O)CCC(F)(F)F)C2)(CNC(c2ccn3c2CCCC3)=O)CC1 39385,Cc1nc(=NN2CCC(C#N)CC2)c(C#N)c[nH]1 39386,c1(NC(c2cccc(COC)c2)=O)ccc2c(-c3ccsc3C#N)cccc2n1 39387,c1(C(=O)Nc2cc(Cl)ccn2)n[nH]c2cc(-c3cccc4cccnc34)ccc12 39388,c1(OC)nn(C)cc1C(=O)NC1CCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 39389,c1(OCCC(=O)NC2CC(N(C)C(C3CCNC3=O)=O)C2)ccc(Cl)cc1 39390,c1(C(=O)NC23C(CN(C(C4C(C)C4)=O)C2)C3)nccc2ccccc12 39391,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39392,C1(C(N2CCCCC2)=O)(CO)CCN(CC=CC2CCCC2)C1 39393,Cc1nc(C(C(=O)NCc2ccco2)N(CC(F)(F)F)C)nn1C 39394,C#CC1COCCN1C(c1ccc(OCOC)c(F)c1)C(=O)NCCC1(C)CC1 39395,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39396,NC(=O)CC(O)C(=O)NC1CN(C(=O)CCSC(F)(F)F)CCC1O 39397,CN1CC2CC2(NC(C2CCC(CNC(=O)CCC3CCCN3C)C2)=O)C1 39398,C1(C(=O)NCC2CCC(C)O2)CC2(CCN(Cc3cccc(Cl)c3)CC2)CO1 39399,C=Cn1nccc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1CC(F)(F)C1 39400,c1(OC)ccc(CC(N2CCC3CC23C(=O)N(C)CC2CCCCO2)=O)cc1 39401,C1(C(=O)NCC2COCC2NC(C2(n3cccn3)CC2)=O)CCCCO1 39402,C1(C(=O)NC(C2CCN(C(=O)CN3CC4CC4C3)CC2)CO)C2CCN1CC2 39403,Cc1cccc(-n2nc(Cn3nccn3)nc2-c2cnn3c2OCC3)c1C 39404,C1(NC(c2cccnc2C)=O)CCCN(CC)C1C.C12CC3(C1)CC3C(=O)N2 39405,c1(N(C)COc2cccc(OC)c2)nccc(=NC(C)CN2CCCCCC2=O)[nH]1 39406,C1(C(=O)NC2CC(C)C2)(NC(=O)CC2(O)CCCC2)CCCC1C 39407,CC1(C)CCCC(NC(=O)CSCCNC(=O)CC2CC=CCC2)C1 39408,C(=O)(C#CC1CCOCC1)N1CC(C)C(CNC(=O)CCCCC2CC2)C1 39409,c1(CC(=O)N(CCC(=O)NCc2c(C(C)C)con2)C)ccc(O)cc1 39410,N1(C(CC2C(C)(C)C2(C)C)=O)CCC(C2CC2)(CNC(=O)CC2CC3CC3C2)C1 39411,N1(C(c2c(NC)scn2)=O)C2CCC(C(=O)NC3CCCC(C)CC3)C1CC2 39412,c1(C(N2CCC3(C(C(=O)NCC4CCC(F)(F)C4)C3)C2)=O)cc(F)c(F)cc1Br 39413,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39414,C1(CC(=O)NCC(CNC(C(COCC)C)=O)F)CCCCC1(C)C 39415,c1(C(=O)NC(C)CNC(c2coc3c2COC3)=O)ccc(NC2CC2)cc1F 39416,C12(C(=O)NCCC3(O)CN(C(C(C)SCC)=O)C3)CC(C)(C1)OC21COC1 39417,N1(C(c2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CC1)=O 39418,C1(CCNC(=O)NC(c2nc(C)[nH]n2)C)CCCC2CC12 39419,C1(C(N2CCCC(CNC(=O)COCC3CCC3)CC2)=O)CCc2ncsc2C1 39420,C1(F)(CNC(C(F)=CCC)=O)COCCN(C(C2OCC2(C)C)=O)C1 39421,CCCC(C)(O)CC(=O)N1CC(NC(c2cnc(C(C)C)s2)=O)C(CC2CC2)C1 39422,c1(OCC)ccc(C(=O)NCCCC(C)NC(c2oncc2C)=O)cn1 39423,c1(C(N2C(CNC(C(CC)(CC)CO)=O)CCC2)=O)cn2nccc2nc1C 39424,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(c1cc(OCC(F)F)ccn1)=O 39425,N1(C2CN(C(c3cc(CNC(c4coc(CO)c4)=O)[nH]n3)=O)C2)CCCOCC1 39426,C12(NC(c3c(CC)c[nH]c3)=O)CCN(C(C3(CC4CC4)CC3)=O)CC1C2 39427,N#CC1(NC(=O)CN2CCCCC2=O)CCN(C(c2ccncc2)=O)C1 39428,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(CO)CC1 39429,C=CCC(F)(F)C(=O)NCC(O)C(=O)NC1CC2CCC(C1)O2 39430,C(=O)(C(F)CC(C)(C)C)N1C(C(C)C)C(NC(C2(Br)CC2)=O)CC1 39431,C(=O)(C(F)CC(C)(C)NC(C1(C)CCCCC1C)=O)NC(c1nncs1)C 39432,c1(CC)c[nH]c(C)cc1=NC1CCc2cc(Br)ccc2C1 39433,c1(OC)ccc(CNC(=O)C(C)(O)Cc2cc(Cl)ccc2Cl)c(F)c1F 39434,CCC(CC(=O)N1CCC(CF)(NC(c2c[nH]nc2C2CC2)=O)C1)C(C)(C)C 39435,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)Cc1cnc[nH]1 39436,C1(CNC(c2c(SC(C)C)cccc2)=O)CCN(C(=O)CCc2ccc[nH]2)CC1F 39437,N1(C(c2cc(OC)ns2)=O)CCC12CCN(C(c1cccc(OC)c1C)=O)CC2 39438,c1(C(C)C)cc(Cl)nc(NC(N2CCCC(Oc3cccc(C(N)=O)c3)CC2)=O)n1 39439,C(CNC(C1(C)CC1(F)F)=O)(CCNC(c1[nH]cnc1C)=O)OC 39440,C1(NC(c2ccc(C)n2C)=O)CCC12CN(C(=O)CN1CCOCC1)C2 39441,N1(C(C)CNC(C2CCN(C(=O)CC3CC3)C2)=O)CCN(C(=O)CC(C)CF)CC1 39442,C=CCC(C)C(=O)NC(c1ccccc1CC)CNC(C1(Cl)CC1)=O 39443,N#CC1CC2(CC(NC(C3CC(NC(=O)Cn4cccn4)CCO3)=O)C2)C1 39444,c1(CNC(=O)Nc2ccccc2)cc[nH]c1C(N1CC2CC2C1)=O 39445,CCCC(O)(CCC)CC(=O)N1CCN(c2cc(C(=O)N(CC)CC)ccn2)CC1 39446,CC1CCN(C(C2CCC2)=O)CC1CNC(c1cccc(F)c1OC(F)(F)F)=O 39447,C1(C(=O)NC2CCC(CCNC(C(C3CC3)SC)=O)C2)C2CC3C(C2)C13 39448,C1(NC(c2cncc(OCC)c2)=O)CC2CN(C(=O)COC3CCCOC3)CC12 39449,N1(CC)CCC(N(C(=O)C(C2CCOC2)NC(=O)C=CC(C)(C)C)C)C1 39450,CC(C1C(=O)C2CC(C2)C(=O)N1)NC(=O)OC1CC1.c1ccoc1.C(C)(C)(C)OC 39451,N1(C(=O)CC2=CCCC2)CC2=C(C1)CN(C(c1cccc(C(F)F)n1)=O)C2 39452,Cn1nc2c(c1C(=O)OCc1ccc3cnccc3c1)S(=O)(=O)NCCC2 39453,C1(C(=O)NCC23C(CN(C(C4N(CC)CC4)=O)C2)C3)CCCN2CCCCC12 39454,C1(N(C(=O)C(C)OCc2ccccc2)CC)CCCN(C(c2ncn(C)n2)=O)C1 39455,c1(COCCN(C(CCNC(C(N2C(CC(C)C)CC2)=O)=O)O)C)ccccc1 39456,c1(C(N(C2CCN(C(C3CCOC3C(F)(F)F)=O)CC2)C)=O)cnnc(O)c1 39457,C(C1=CCN(C(C2CCC(=O)NC2)=O)CC1)NC(=O)CCCc1ccccc1F 39458,C(CCCCC(=O)N1CCC(CC(=O)NCC2(O)CCC(C)C2)C1(C)C)OC 39459,Cc1ncc(C=CC(N2CC=CC(NC(C3(C)CCCOC3)=O)C2)=O)s1 39460,c1(C(C(=O)NC2CC(NC(c3cn(CC=C)nn3)=O)C2)(C)OC)ccccc1F 39461,C1(CC)CCCCC1C(=O)NC1(C(=O)NCC23CCN(CC2)C3)CC(C)C1 39462,Cc1[nH]c2ccccc2c1C(N1CCCCC1CCN(C)C(c1cnns1)=O)=O 39463,C1(NC(CNC(C)=O)=O)CC1C1CCN(C(=O)C2=CCOCC2)CC1 39464,N1(Cc2cc(C)ns2)CCC(C)(NC(=O)CC2CCC(=O)N2)CC1 39465,C1(CNC(CCC(=O)OC)=O)COC(C)(C)CN1C(C1CC2CCC(C1)N2C)=O 39466,N1(C(c2nnn(C)c2C2CC2)=O)CCC2CCN(C(c3cccc(Cl)c3)=O)CC12 39467,c1(C(=O)NCCNC(CC(C=C)(C)C)=O)nc(C(F)(F)F)n2ccccc12 39468,N1(C(C(CC)=CC)=O)CCC2(CCCCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 39469,C(=O)(CCCC(C)NC(=O)C1=CCSC1)N(C)Cc1n(CC)cnn1 39470,C12(C(=O)OC)CN(C(=O)OC(C)(C)C)CC1(CNCC1CCC(F)C1)C2 39471,C1(C(=O)NC2CCN(C(C)=O)C2)CN(C(=O)CC2CCSC2)CC1N(C)C 39472,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1ncn(C(C)C)n1)=O 39473,c1(C(=O)NCCCCNC(CC2CCC(C)C2(C)C)=O)c2ccccc2nn1C 39474,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39475,O=C1COc2cc(C(N3C4CCC3CN(C(C3CCC5CC35)=O)C4)=O)ncc2N1 39476,N1(C(C2(CC)CC2)=O)CCC(SCC)CC1.c12cn(nn1)C1COCC1NC2=O 39477,C1(C(N2CCC(C)(C(=O)NCC3N(C)CCC3)CC2)=O)Cc2ccccc2C1(C)C 39478,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39479,CC(C)CCCC(C)C(=O)NC1(C(N2CCc3nc[nH]c3C2)=O)CC1 39480,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1ns[nH]c1=O)=O 39481,c1(CC)nc(C(=O)NCc2ccc(C(N3CCOCC3C(N)=O)=O)cc2)c(C)o1 39482,c1(C(=O)NCCC(C)N(C(=O)CNc2ccccn2)C)occc1C1CC1 39483,C1(C)(NC(C(F)OC)=O)CCN(C(=O)CSc2cc(SC(F)(F)F)oc2C)C1 39484,C1(C(N2C(CCNC(Cc3c(C)cnn3C)=O)COCC2)=O)Cc2cscc2C1 39485,C1(C(=O)NCCOC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39486,C(c1cc(C)ccc1OC)=CC(=O)NCC1C(NC(C(COC)(F)F)=O)CC1 39487,N1(C(C(C(C)C)SC)=O)CCCCC(NC(=O)COc2cc(C)on2)C1 39488,Cc1ccc(C(N2CCCC2CCCNC(=O)CN(C)C)=O)n1C 39489,c1(C(=O)N(C)CCNC(=O)NCCNC(C)=O)ccccc1SC.CO 39490,c1(C(=O)NC(C)CCNC(C2(C(N)=O)CC2)=O)ccn(C(C)(C)C)c1 39491,c1(CNCCC(OC)OC)cnn(C)c1CC1CC1 39492,C(C)(CCCCNC(=O)CCc1nnc(C2CCCC2)o1)NC(C1C(C)C1C)=O 39493,C=CCCCCCCC(=O)NC1CCC(CNC(C2NC(=O)C3CCC23)=O)C1 39494,c1(CC)ccc(C(=O)N(C2(CC(=O)N(CCC(F)(F)F)CC)CC2)C)[nH]1 39495,C1(O)(CNC(COCCOC)=O)CN(CC(=O)Nc2cnn(C3CC3(F)F)c2)C1 39496,c1(C(=O)OC)cncc(NC(C(CO)NC(C2(C)CCNC2=O)=O)C2CC2)c1 39497,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(=O)C(C2CC2)N(C)C)C1 39498,c1(CCC)c(C(N2CCCC(CCc3ccccc3Cl)C2)=O)nnn1CC 39499,c1(C(=O)NC(C)C(CO)NC(c2cn3ccsc3n2)=O)ccc(Cl)nc1O 39500,c1(CCNC(C2N(C(C3N(C)CCC3)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39501,C(C1=CCN(C)CC1)NC(C1(NC(=O)CC2C(C)(C)C2(C)C)C(C)C1)=O 39502,N1(C(c2cnc(CC(C)C)s2)=O)CCC(C)C(CNC(=O)C(C)(C)C(C)O)C1 39503,N1(C(CN(C(CC)CC)C(=O)C(c2ccn(C)c2)C)=O)CC(O)CC1CC 39504,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)N2CCn3ncc(CO)c3C2)c(Br)c1 39505,c1(OCC)ccc2c(c1)OCCN(C(=O)OCC(C)C#N)C2 39506,n1(CC(=O)N(CC(C)NC(C2CCC(OC)CC2)=O)C)ccc(C)cc1=O 39507,c1(OC)ccccc1C(=O)NC(c1cccnc1OC)C(=O)NCc1cccs1 39508,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(=O)COC(F)F 39509,C1(Nc2ncccn2)CCc2nncn2CC1.c12cn(nn1)C1CCN(C1)C2=O 39510,Cc1ccn(C)c1C(=O)NCC1CC(F)(CNC(C2(F)CC=CC2)=O)C1 39511,C1(C(=O)NC(C=C)C)CC12CC(NC(c1c[nH]nc1C1CC1)=O)C2 39512,CC(C)CC(C(=O)NC1CCCC(NC(c2cnc[nH]c2=N)=O)C1)C(N)=O 39513,c1(OC(C)C)cccc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2Cl)c1 39514,C1(CNC(C2(c3n(C)ccn3)CC2)=O)CCCCN1C(c1cnsn1)=O 39515,N1(C(C2CCC(=O)N2)=O)C2CCC1(CNC(c1cnn(CC(F)(F)F)c1)=O)CC2 39516,c1(C(CN(C)C)N(C)C)nnnn1C(=O)CCCc1ccc(Br)s1 39517,N1(C(=O)OCc2cccc(Cl)c2)CCC2(CSC2)C1 39518,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCc2cscn2)C1 39519,N1(C(CCCC[SH]=C)=O)CCC(C)(C)C(NC(=O)C(C(C)CC)NS(C)(=O)=O)C1 39520,C1(NC(CCC#C)=O)CCCC(N(C(=O)CCc2ccco2)C)C1 39521,C1(C2(C(N(C(CC)CC)C)=O)CC2)CCCN1C(=O)CC1CCOC1=O 39522,Cc1cc(C(C)NCC(C)CCCO)ccc1[N+](=O)[O-] 39523,c1(NC(C(C)NC=O)=O)cccc(F)c1.c1(C2C(=O)N2)cscn1 39524,C1(CC(=O)NCCC2CCC2)CCCCCC(=O)N1.CC1(C)CC=CC(=O)N1 39525,C1(CC(N2CC(CCO)(NC(CCCC#C)=O)C2)=O)NC(=O)CN(C)C1=O 39526,C1(C(=O)N)CC2CCC1O2.C(CC(O)CNC(C1(C(=O)NC)CCC1)=O)CC 39527,C(CCCCC(=O)N(C)CCN(C)C(c1c(C)ccn1C)=O)=CC 39528,C(=O)(C(C)(C)CCC#N)NCCCCC(C)NC(C1OCCN(C)C1=O)=O 39529,C(C)(CCCC(=O)N1CCOCC1C1CC1)NC(COCCCC(C)C)=O 39530,Cc1cncc(C(N2CC(NC(=O)C(C)NC=O)CC2C)=O)n1 39531,c1(C(=O)NC(C(CO)NC(CCN(C)CCO)=O)C)cc(Cl)c(Cl)cc1N 39532,C=CCCCCCC(=O)NC(C(=O)NC1CC(C)(C)OC1(C)C)C1CC1 39533,Cc1ccc2n[nH]cc2c1C(c1ccc(Br)c(F)c1F)NC(N1CCC(F)C1)=O 39534,N1(C(=O)C2=CCCCCCC2)CCCC2C(CCCN2C(=O)CSc2cccs2)C1 39535,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39536,C1(F)(C(=O)NC2C(CC(=O)NC(C)C3CC3)CCC2)C(C)(C)C1(C)C 39537,CC1CCCC(NC(C2CC(c3ccccc3)(NC(=O)OC(C)(C)C)C2)=O)C1 39538,c1(CNC(C)C[SH](C)O)cc2cc(F)ccc2cn1 39539,C12(C(=O)NCCOCCCC)CCC(CC1NC(c1cncc(O)c1)=O)C2 39540,CC1OC(C)C(C(=O)NCC2CCN(C(C3CCCS(=O)(=O)C3)=O)CC2)C1C 39541,Cc1cc(N(C2CCN(C(=O)C(C3(O)CCOCC3)(F)F)C2)C)c(C#N)cn1 39542,C(=O)(C(F)CC(C)(C)C)N1C(CC(N2CC(SCC)C2)=O)CCC1 39543,c1(C(=O)NCC(C2CCCCC2)NC(Cc2c(C)noc2)=O)cc(Cl)nn1C 39544,C(=O)(C1=NN(C)C(=O)CC1)NC1C2N(C(C=NOC)=O)CC(CC2)C1 39545,c1(OC)c(NC(=O)NNC(C2COC(C)(C)O2)=O)ccc([N+](=O)[O-])c1F 39546,N1(C(=O)NCCC(O)C(F)(F)F)CCC(C=CC(=O)Nc2c(C)cc[nH]2)CC1 39547,Cc1cc(C(=O)NC(C)(C)CNC(C2CN(C3CCOC3)C2)=O)ns1 39548,c1(C(=O)NC23CC2CN(C(C2CC4C=CC2C4)=O)C3)cncc(Cl)c1Cl 39549,O=C1NN2CCCC2C(=O)OC2CC1C2.c1(CCC(F)F)nc[nH]n1 39550,N1(C(C(=O)Nc2cn(CC)nc2)c2nc[nH]n2)CCCCC1c1cccc(Cl)c1 39551,c12cc(nn1C)C(=O)N2.C1(OC)CCN(CC(N2CCC(CC3CC3)C2)=O)C1 39552,C#Cc1cn(C)nc1C(=O)N(C(CC(C)C)C(=O)N1CC(C(=O)OC)C1)C 39553,C1(CC(=O)NCCCNC(C(C)c2ccco2)=O)CSc2ccccc2O1 39554,N1(C(c2ncn(CC)n2)=O)CC(NC(C2(C(F)F)CCCO2)=O)C(C)C1 39555,C(=O)(C(F)(F)C(F)F)NCC1(NC(C(C(C)C)F)=O)CCCCC1 39556,C(=O)(C(F)CC(C)(C)NC(c1ccc(F)cc1)=O)NC(C1CCCO1)C 39557,CN1CCN(C(c2cnn[nH]2)=O)C(CNC(C2CCOC(C)(C)C2)=O)C1 39558,c1(-c2cc(C)c(F)c(C)c2)cc(Nc2ncn(C)c2Br)cc2[nH]ccc12 39559,C(CCC(=O)NCC1CC(CNC(C2(C)CCCC2)=O)CO1)SC 39560,c1(C(N2C(C(=O)Nc3cccc(Br)c3I)CCCC2)=O)cc(CO)ccc1O 39561,c1(OCC)cc(C=CC(=O)NC2CC(F)(CNC(=O)C(C)(C)C)C2)ccc1OF 39562,C=C=CCCC(=O)OCC(=O)N(C1CCCC1)C.c12noc-1n2 39563,c1(CC)[nH]nc(C(=O)NC2(C(=O)N(CCCN=[N+]=[N-])C)CCCC2C)c1C 39564,N1(C(C2C(CNC(C3CCC4(CC4)C3)=O)CC2)=O)CCC2(C=CCO2)CC1 39565,c1(C(CN(C=O)CCc2ccccc2)(F)F)c(F)cccc1F 39566,c1(CCC(=O)NC(CCCNC(c2c(C)n[nH]c2C)=O)C)ccc(Cl)cc1Cl 39567,n1(CC(=O)NC2(C3CN(C(C4(C)CC4)=O)C3)CC2)ncc2ccccc12 39568,C1(C(=O)NC2CON(CC)C2=O)CN(C(C2CC3(CC3)CO2)=O)CC1(C)C 39569,N1(C(c2cc(C)n(CCO)n2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 39570,NS(=O)(=O)C1(CNC(=O)NC2CC3CCC2C3)CCCC1 39571,c1(OCCC#C)cc2oc(=O)[nH]c2cc1OC 39572,Cc1cccc(C(=O)NCC2CC(C)N(C(c3c(F)cccc3F)=O)C2)c1C 39573,c1(C(=O)NC(CC2CN(C(Cc3cccc(C)c3)=O)C2)C)cnc(N)c(N)c1 39574,C(=O)(C(C)(C)CS(C)(=O)=O)NCC(CN(C(=O)CCCc1ncco1)C)C(F)(F)F 39575,n1(CC)nccc1C=CC(=O)NC(C)(CNC(c1ccc(C2CC2)s1)=O)C(C)C 39576,Cc1ccn2c(C(=O)NCC3(CNC(=O)CC4CC5CC45)CCC3)c(C)nc2c1 39577,c1(C(=O)NCCOCCOCCO)cccc(Cl)c1Cl.n12cc(nn1)CC2 39578,c1(CNC(C(=O)NCc2ccc(OC)c(OC)c2)=O)cc2c(s1)CCOC2 39579,C1(C(N(C2CC(C)C2)C)=O)C=CCCN1C(=O)CC(O)CN(C)C 39580,C1(N(C(C2(C#C)CCCC2)=O)C)CC2CC1N(C(=O)C(CC)=CC)C2 39581,C(CN=C(NCC)NCc1cc(-c2ccccc2)n(C)n1)NC(=O)NCC 39582,CC1N(C(=O)Cn2cc(CNC(=O)C(=O)NCC(F)F)nn2)CCCC1(C)C 39583,Cc1nc(C2CC2)ncc1C(N1CCC(N(CCO)C(c2nccn2C)=O)CC1)=O 39584,Cc1cc(NC23CCCC2CN(C(=O)CO)C3)n2ncnc2n1 39585,N1(C(C2N(C(C(C=C)(F)F)=O)CC3(CC3)C2)=O)CC2(CC(CO)CO2)C1 39586,N#Cc1ccc(C(=O)NC2CCCN(C(=O)CCNC(C3C=CCC3)=O)C2)s1 39587,C1(C(=O)NC2CC(CCNC(C3(OC)CCC3)=O)C2)CCCCC(=O)C1 39588,c1(NC(C)=O)ccc(N2CCC(C)(C(=O)NOCCOC(C)C)C2)nc1 39589,c1(OCC(=O)NCCOCCOCCCNC(=O)CCC2CCOC2)ccncc1 39590,N1(C(C2C(C(=O)OCC)C2)=O)CC2(CCC2)OCC1C.C1C(=O)O1 39591,C(Cn1cncn1)(C(=O)OC)NC(COCC)=O.C1CC(=O)NCCO1.OC 39592,N1(C(C(C2CC2)OC)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39593,N1(C(CCCOC)=O)CCCC(CO)(CNC(c2cc[nH]n2)=O)C1 39594,c1(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCOCC2)cc(F)ccc1N 39595,N1(C(=O)CCC2CCC2)CCC(n2cc(CC(N3CCCC(Br)C3)=O)nn2)CC1 39596,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C=CC=CCC)=O)CCC1CO 39597,c1(CC)ccc(F)cc1C(=O)NC1CC1.C1(C(=O)NC2CC2N)CCCOC1.COC 39598,N1(C(CCc2n[nH]c(=N)s2)=O)CCN(C(C2CC3C=CC2CC3)=O)C2CCCC12 39599,C(=O)(C(=O)CC(C)CC)N1C(CC)CCCC1.C1(=O)CN1CC(C)(C)C 39600,c1(C(=O)NC2CCC(NC(c3c(CC)nns3)=O)CC2)cc2c[nH]cnc-2n1 39601,n1(CC)c(=O)c(C)nc2cc(C(=O)NC3CN(C(=O)CN(C)CC)C3)ccc12 39602,Cc1cc(CCCC(=O)N(CC(C)N(C(=O)C=Cc2ccccn2)C)C)c(C)s1 39603,CC1(C)CCC2(CN(C(c3cn(CC(F)(F)F)nn3)=O)C2)O1 39604,C(=O)(C1OCCc2ccccc21)N1CCC(CN(C(=O)C2=C(Cl)CCC2)C)CC1 39605,S(=O)(=O)(c1[nH]c(=NC(C)Cn2ccnc2C)ccc1Br)NCc1c(C)cccc1 39606,c1(C(N2C(CNC(C(C)(C)Br)=O)CCC2)=O)cccc2cc[nH]c12 39607,CCC(C)(C#N)C(=O)N1CCCC(O)(CCNC(c2ccc(O)nn2)=O)C1 39608,C(=O)(C(C(C)C)NC(C1CCC2(CC2)C1)=O)N(CCOCC)C(C)C 39609,c1(C(C)=O)cc(C(=O)NCC(n2cc(-c3cccnc3F)nn2)C)c(C)o1 39610,C1(C2CCOCC2)(C(=O)NC(c2ccccc2)CNC(COCCC=C)=O)CC1 39611,C1(C(=O)NCc2nc(CNC(C3(C)ON=C(C)C3)=O)sc2)CCc2nnnn2C1 39612,C(=O)(C1=NOC(C)C1C)NCC(CC)(C)NC(c1ccncc1OC)=O 39613,N1(C(CC=CC=C)=O)CCC2(NC(c3cn(C(C)(C)C)nn3)=O)CCCCC12 39614,c1(N(CCOC)CCNC(=O)CSc2ccccn2)cc2nnc(C)n2cn1 39615,C1(NC(Cc2cc(C)on2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39616,C(=O)(C(F)C(=O)NCC1(F)CC(NC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C1)OCC 39617,Cc1ccc(CCNCC2(CCNC(C3(c4cc[nH]n4)CC3)=O)CCC2)cn1 39618,N1(C(c2ccnc(OC)n2)=O)CCC2(CNC(=O)CCC3(C)N=N3)CCCCC12 39619,C1(C(N2CC(OCc3c(OCC)oc(C)n3)C(C)(C)C2)=O)CC12CCCCCC2 39620,C(=O)(CCCCC(F)F)N1CC2C(NC(c3ccc(N)cc3F)=O)C(C2)C1 39621,n1(CC)cc(Br)cc1C(=O)N(CC(C)O)CCNC(C1(CCOC)CC1)=O 39622,C1(CC=C)CCCCC1NC1C(C(=O)OCc2ccccc2)CCC1O 39623,C=C=CCCOC(=O)C(C)c1cccs1.C1(=O)C(C)O1 39624,Cc1cc(C(=O)NC2CC2NC(c2c[nH]c(=O)cn2)=O)c(O)c(Br)c1 39625,c1(C(=O)NCC2(N3CCCCCC3)CC2)cccnc1C(=O)NC(C#C)C(C)OC 39626,c1(NC(CC(=O)NCC2C(SC)CCCC2)=O)ccc2nc(N(C)C)sc2c1 39627,C1(NC(Cc2c(C)scc2)=O)CCCC(NC(=O)C=CBr)C1 39628,c1(C(=O)NC2CC(C)(NC(=O)CCn3cncn3)C2)cc(N)c(F)cn1 39629,C(=O)(CC(F)(F)F)N(CC(C)NC(=O)C(C)(C)C1CCCC1)CCOC 39630,CC1=C(C(=O)N2CCN(C(=O)CCSC(F)(F)F)C(CC(C)(C)C)C2)CCO1 39631,C1(C(=O)NCCn2c(C)ncc2)CCCN(C(=O)CC2COCC2O)CC1 39632,N1(CC(=O)NC(C(C)(C)NC(C2C(SC)CCC2)=O)C)CCNC(=O)C1 39633,c1(C(N2C(C)CCC(CNC(CC(C)(C)OC)=O)C2)=O)cccc2ccsc12 39634,N1(C(c2c(-c3ccc(OC)nc3Cl)ncs2)=O)CCc2[nH]ccc2C1 39635,C(=O)(C(CCCCCO)N1CCC(n2cnnn2)C1)NC(C1CCC1)C.N(C)C 39636,c1(OC)ncc(C(c2c(F)cccc2Br)NC(=O)OC(C)(C)C)cc1F.C1C(=O)N1 39637,c1(-c2ccn(C)c(=O)c2)nc2ccc(C#N)cc2[nH]1 39638,N1(C(Cc2ncc(C)[nH]2)=O)CCN2CCOCC2(CNC(=O)C=C2CCSCC2)C1 39639,c1(C(=O)NCCC(CC)(C)NC(=O)C(F)CC(C)C)snc2ccccc12 39640,C1(C(N2CCC(c3cc(C)no3)C2)=O)CN(C)CCN1C(C1CCCC(C#N)C1)=O 39641,c1(C(=O)NC(C)C=CC(=O)N(CCCO)CCO)cccc(=O)n1C 39642,Cn1cnc2[nH]c(C(=O)Nc3ccc(Cc4nc(=O)o[nH]4)cc3)nc2c1=O 39643,N1(C(C2(C)C=CCCC2)=O)CC2CC1CC2CNC(=O)CCc1ccc(Cl)nc1 39644,N1(c2nnn(C)n2)CCCC12CCN(C(c1cccc3c1CCO3)=O)C2 39645,C1(C(N2C(C(C)C)CN(C(C34CCC(C3)C4)=O)CC2)=O)Cc2cccnc2C1 39646,N1(C(=O)C(=O)OC)Cc2ccccc2CC1C(=O)Nc1csc(OCC)c1OC 39647,C(c1ccccc1F)=CCC(=O)NCCN(C(=O)CC1CCOC1)C 39648,C1(CNC(=O)NCC(C2CCCCC2)C)CCN(C(C)(C)C)C1 39649,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39650,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(COC)CCOCC1 39651,N1(C(c2nc(CC(C)C)sc2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 39652,C1(C(N(CCCCNC(=O)C(C2CCCCCC2)O)C)=O)CCC2(CCC2)OC1 39653,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)Cn2nc(C)n(C)c2=O)C1 39654,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39655,N1(C(c2n(CC)ccc2)=O)CC(NC(c2c(C)ncn2OC)=O)CC12CCCCC2 39656,CC(CCC(=O)NCC1CCN1C(c1cnc(N(C)C)s1)=O)c1ccccc1 39657,c1(OC)c(C(N2CC(N(C)C(c3ccnnc3O)=O)C2)=O)oc2ccccc12 39658,C1(CC)COC(C)CN1C(C1CC(C)CN(C(=O)CN2C(=O)CNC2=O)C1)=O 39659,N1(C(CCC(=O)OCC)=O)CCC(C2CC2)C1CNC(c1cnc(C)c(C#N)c1)=O 39660,c1(OC)ccc(C#N)cc1NC(c1cccc(N(C)C)c1)c1nnnn1C 39661,N1(C(c2cccc(CNC(CCCCC#C)=O)n2)=O)CCC2C(CCN2C)C1 39662,c1(C(=O)NC2C(NC(c3cncc(NCC)c3)=O)CCO2)nc[nH]c2nccc1-2 39663,c1(C(C)(C)NCc2ccncc2)ccnc(Cl)c1F 39664,C(=O)(C1CCc2cccc(F)c21)N1CC(COC)OC(C)C1 39665,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)cn1)=O)=O 39666,C1(NC(c2cc(Cl)no2)=O)CCC12CCN(C(=O)CCC1CC1)CC2 39667,N1(C(C(CC)(C)C)=O)CCCN(C(=O)CC2CCCCC23CC3)C(CO)C1 39668,N1C(=NCCCN(C)C)NCc2nc(no2)C1.c1(C2C(C)C2)cccc(Br)c1 39669,C1(C(=O)NCC2(F)CN(C(C(C(C)C)(F)F)=O)C2)CCC2(CCOCC2)C1 39670,Cc1ccc(CC(=O)NCC(C(C)(C)C)NC(=O)CC2(O)CCOCC2)c(C)c1 39671,N1(C(Cc2scc(C)c2)=O)CC(C)CN(C(=O)CN2CCCCC2)C(C)C1 39672,C(C)(C)(CC(=O)NC(c1cn(C)nn1)C)NC(C=CCCC)=O 39673,c1(C(=O)NCC(C2CCC2)NC(C2(C)CCC(=O)N2)=O)cc2cc(Cl)ccc2o1 39674,C(=O)(CC(C)C(C)(C)NC(c1cc(=O)cc[nH]1)=O)N1CCC(C)(CSC)C1 39675,c1(C(=O)NCC2C3CN(C(C4(C)CC=CCC4)=O)CC32)csc2cccnc12 39676,c1(-c2cccc(OC(C)C)c2)ccn2nc(C(N3CCOCC3C)=O)cc2c1 39677,c1(C(=O)NC2CCN(C(C(C)N(C3CCCCC3)C)=O)C2)cn2cnnc2cn1 39678,C1(NC(c2ccn(CC(C)C)n2)=O)CCN(C(=O)CC2(C)CC2)C1C1CC1 39679,CCC(C(=O)NC(CNC(=O)CNS(N)(=O)=O)CC(C)C)C(C)(C)CC 39680,C(=O)(CCC(C)(F)F)N(CC(CC)NC(c1c(Cl)cnn1C)=O)CC 39681,CC1Cc2ccccc2N1C(C1CN(C(=O)CCn2cccc2)CCC1O)=O 39682,CC(C)(CC(=O)N1CC2(NC(C3CCOCC3)=O)CCC1C2)C(F)F 39683,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39684,C1(C(N2CCC(OCC(C)C)C2)=O)CCC(C)(C)N(C(C2CC2(Cl)Cl)=O)C1 39685,c1(CC(=O)N(C2CC2)CC2CCCN2C(C2CC(F)C2)=O)cc(Cl)sc1Cl 39686,CC(Cl)(Cl)C(=O)N1CCC(CC(=O)NCC2CCC(C3CC3)O2)C1 39687,N1(C(C(CC#C)C)=O)CCN(C(C2(c3cc(C)on3)CCC2)=O)CC1CF 39688,C1(OC)(CNC(C2C3CN(C)CC23)=O)CCN(C(c2c[nH]c(C#N)c2)=O)C1 39689,C#CCCC(C(=O)NC(C1CCOC1)CC)NC(=O)C=C1CCCCC1 39690,c1(C(N2CC(CNC(c3c(NC)snc3C)=O)OCC2)=O)cn2ccccc2n1 39691,c1(C(=O)OC(c2cccc(-n3ccnn3)c2)C)ccc(C#N)c(Cl)c1 39692,C(=O)(C(F)C(F)(F)F)NCC1CC(F)(CNC(C(C)Cc2cccnc2)=O)C1 39693,C1(C(N2CC(OCC(=O)NC3CC(C#N)C3)C2)=O)C2(CC2)C12CC2 39694,N1(C(C(C(COC)C)C)=O)CCCC2(NC(C3CCCCC3C)=O)CCCC12 39695,O=C(C1=C(Cl)CCOC1)NC1CC(NC(c2cc(CO)nn2-c2ccccc2)=O)C1 39696,c1(CCC)ccccc1CNC(C1CCOCC1NC(=O)CCC1CC(C)C1)=O 39697,N1(C(c2c(C)scc2)=O)CC2CN(C(=O)CSC(F)F)CCC2(CO)C1 39698,C(=O)(C1CCCc2ncnn21)NC1CCN(C(c2cccc(OC)c2)CO)CC1 39699,C12(NC(c3c(OCC)ccs3)=O)CCCCC1CN(C(=O)C#CC1CC1)C2 39700,C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(Cc2c(C)nc[nH]2)=O)C)CC(F)C1 39701,C1(C#CC(=O)NCC2CN(C(C34CC5CC3C4C5O)=O)CC2(C)C)(CC)CC1 39702,C(CC)(C(=O)N(C1(C(=O)N(C)CCC)CC1)C)=CC 39703,O=C(CC1=CCCCC1)N1CCC2(CC2C(N2CCC(CO)CC2)=O)C1 39704,N1(C(c2ccc(C)s2)=O)CC2CCCCC2(NC(c2occ(C)c2C)=O)C1 39705,C1(CC(=O)OCC)CCCN(C(C23CCC(C2)OC3C)=O)CC1 39706,C(=O)(C(F)(CNC(=O)C=CC(F)F)C(C)C)N1CC(C(C)C)N(C)CC1 39707,N1(C(C2CCC(OC)C2)=O)CC2CN(C(c3ccc4nc[nH]c4n3)=O)CC(C1)O2 39708,N1(C(c2c(CC)nc(CC(C)C)s2)=O)CC2CC1CN2C(C1CC12CC2)=O 39709,C1(C(=O)Nc2cn(CC)nc2)CC12CCN(C(=O)COC(C)=O)CC2 39710,C1(CNC(C2N=C(C)SC2)=O)Cc2ccccc2CN1C(=O)C(C)c1ccco1 39711,N1(C(C2C=CCS2)=O)CC2CN(C(C3CCCC3C3CC3)=O)CC2C1 39712,Cc1ccnc(O)c1C(=O)NCCOCC(=O)NCC1(n2ccnc2)CCCC1 39713,c1(OCC)ccc(CC(=O)NC(C2CCN(C(C)=O)CC2)C2CC2)cc1 39714,CC1CCCN(CCNCc2c(C(=O)NC3CN(C4CCC4)C3)nccc2)C1 39715,C12(C(=O)NCC3C(Cn4cc(-c5cn(C)nc5)nn4)C3)CC3CC(CC(C3)O1)C2 39716,c1(C(=O)NCC(C)NC(CCN(CCC)C)=O)noc2c1CCCCC2 39717,C1(C)(C(N2CC(O)(COC)C2)=O)C=CCCC1.N(CCN)C1CC1 39718,C(=O)(CCCN(C)C(C1CC1)=O)NC(CNC(C1(C#C)CC1)=O)C1CC1 39719,c1(C(N2CC(S(=O)(=O)N(C)C)C2)C(=O)NCC(=C)C)cc2ccsc2c(O)n1 39720,C1(NC(=O)CCCC2CC2)CCCC12CN(C(C1(c3cccs3)CCOCC1)=O)C2 39721,C1(C)(CNC(c2c(C)cno2)=O)CCCN1C(=O)CCSCC(N)=O 39722,Cc1noc(C)c1CSCC(=O)N(C1CCC(NC(C2CC=CC2)=O)C1)C 39723,Cc1cncc(NC(=O)CC(C)(C)NC(=O)C(C)CC2CCC2)c1 39724,C(C)(CN=c1nc(C2CC2)[nH]s1)N(C(Cn1ncc(C)c1)=O)C.C1CNC1 39725,C1(C(N2CCC(C)(C(N(C)CC3CCN(C)CC3)=O)C2)=O)CCC2(CCC2)O1 39726,C1(Cn2cc(C(C)(C)C)nn2)CC2CCC(C1)N2C(c1cc(F)cc(Br)c1)=O 39727,N1(C(CCCCCOC)=O)CC(C)N(C(c2ccc(C(F)(F)F)cn2)=O)CC1C 39728,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)Cn2ncnn2)C1)SC 39729,N(C1CCCc2c(F)cccc21)CC(CC=C)(C)CO 39730,N1(C(C2CCC(C#N)C2)=O)CC(=CC(N2CCC3(CCCO3)C2)=O)C2(CCC2)C1 39731,N1(C(C(C=CCCC)O)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)C(C)(C)C1 39732,N1(C(=O)Nc2c(C#C)cccc2)CCC2CN(CC(C)C)C(=O)C2C1 39733,N1(C(CC(=C)Br)=O)CCC2(C=CC(NC(=O)CCN3CCC3)C2)CC1 39734,C1(CNC(c2n(CC)cnc2)=O)CC(NC(=O)COC)C12CCC2 39735,Cc1c(C(=O)NC2CC2CNC(=O)CC2COCCO2)cc(Br)cc1N 39736,S(=O)(=O)(c1ccc(NCC(C)(O)CCO)c(F)c1)N1C(C)CCCCC1 39737,c1(CNC(c2c(CC)noc2)=O)ccc(CN(C(=O)CC2CC3CC3C2)C)cc1 39738,Cc1ccc(C(=O)NC2CCC(CNC(c3ccn(C4CC4)c3C)=O)C2)nc1O 39739,c1(C(C2CCOCC2)NC(=O)Nc2cncc(F)c2)ccc(F)cc1F 39740,N1(C(=O)NC2CCN(C(C)=O)CC2)CC2CCN(C(=O)Cc3cnccn3)C2C1 39741,N1(CCONC(=O)NCC2C=CCCC2)C(=O)c2ccccc2C1=O 39742,N1(C(C2=C(C)OCC2)=O)CC2CC(NC(c3nccc4n[nH]cc34)=O)C(C2)C1 39743,c12cc(ccc1C)OCCN(C(C(CCC)OC)=O)CCNC2=O.C1CC1.OCC 39744,c1(C(N2CC(C)CC(NC(CC=CCC)=O)C2)=O)ncc(P(C)(C)=O)cn1 39745,c1(OC)ccc(C(=O)NCC(C)NC(C2CCCCN2C(C)=O)=O)c(O)c1 39746,C1(NC(c2oc(CC)c(C)c2)=O)CCN(C(C2CC3CCC2O3)=O)C(C)C1 39747,C(CCCCCNC(=O)CCS(C)=O)N(C(c1c(CC)c[nH]n1)=O)CC 39748,O=C1NCC2CN(C(=O)CC3CCCN3C(=O)C(Cl)(Cl)Cl)CC12.c1ccc(F)nc1 39749,c1(C(N2CC3(CCN3C(C3CCN4CCOCC34)=O)C2)=O)cnc2[nH]cnc2c1 39750,Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1CCN(C(C2(Br)CCC2)=O)C2CC12 39751,N1(C(c2noc(CC)c2C)=O)CC(NC(c2ccc(Cl)cn2)=O)CC(O)C1 39752,C12(NC(CS(c3c(C(N)=O)cccc3)(=O)=O)=O)CCOCC1CN(C(=O)CCF)C2 39753,c1(NC(C)C(C)n2cccn2)cccc2cccnc12 39754,C1(C(=O)NCC2CCC(C)C2)C2CCC(C2)C1NC(C1CCC(=O)O1)=O 39755,c1(CCCCCNC(c2c(C)cccc2)c2nnnn2C2CC2)ccccc1Br 39756,Cc1ccccc1N1CCC(NC(c2cccnc2)C(c2ccccc2)C)CC1 39757,c1(OC)ccccc1.C12CCCC1C(=O)OC2.c1(C(=O)NC2CC2)c[nH]c(C)c1 39758,C1(NC(c2c(C)[nH]nc2Cl)=O)CN(C(=O)CCCC(C)SC(C)(C)C)CC1(C)C 39759,CC(CC(=O)N1CC(O)(C(F)C(N2CCCC(NC(N)=O)C2)=O)C1)C(F)F 39760,c1(C(C(=O)NCc2ccco2)N(CC)Cc2ccccc2)c2c(nn1C)CCSC2 39761,c1(C(=O)NC(C)CCCNC(c2csc(=N)[nH]2)=O)nccn2nccc12 39762,N1(C(C=C)=O)CC(C)(C)OC2(C1)CN(c1nnc(-c3cccc4ccccc34)s1)C2 39763,CC1(C(=O)NCCOCCCNC(=O)CC2(C)CCC2)CS(=O)(=O)C1 39764,C1(NC(CSCC)=O)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 39765,O=C1CNC(=O)C(CC(=O)NC2CCCCN(C(=O)C=CC3CCOCC3)C2)N1 39766,CCCCCC(CC)C(=O)N1CCCC1CN(C(=O)CCC(=O)NCCC)CC 39767,C(=O)(CCCCCC#N)N1C(C(C)C)CN(C(=O)C(C2CCCCC2)F)CC1 39768,N1(C(C=CCOC)=O)CC(C2CN(C(=O)C(CO)NC(c3ccccc3)=O)C2)C1 39769,CCCCCC(C)(CC)C(=O)NCC1CC2(CC2)CN1c1ccnc2ncnn12 39770,c1(C(C(=O)NCCCF)N(C)CC2(c3ccccc3)CC2)ccc(F)c(Cl)c1 39771,N1(C(CNC)=O)CC2CC2(CNC(c2nnsc2NC(=O)OC)=O)C1 39772,c1(NCC)cnccc1C(=O)NCCCN(C(C1CCOC1C)=O)CC 39773,N1(C(CCOC(C)=O)=O)CCCC2CCN(C(c3ccncc3)=O)CC12 39774,N1(C(c2cncc(-c3ccc(F)c(C)c3N)n2)=O)CC2CCN(C)C(=O)C2C1 39775,c1(C(=O)NC2CCC(NC(C(CCOC)C)=O)CC2)cc(OC)c(O)c(N)c1 39776,N1(C(C(C)SC)=O)CCC2CN(C(c3cc(Br)c(C)o3)=O)CC2C1 39777,S(=O)(=O)(c1ccc(NC2CC(C(N)=O)C2)c(Cl)c1)N1CC(C)(C)OCCC1 39778,C1(CNC(c2cn(CCC)nn2)=O)C(C)CCCN1C(C1CCC(CO)CC1)=O 39779,CCC(C)CCC(=O)N1CCOCCC1C(=O)NC1CCN(C)CC1 39780,c1(CC(=O)NC2CC3(NC(=O)C4=CCSC4)COC2C3)c[nH]c2ccncc12 39781,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 39782,c1(CCC(=O)N(C2CCCN(C(C3CN(C(C)=O)C3)=O)C2)CCC)cccnc1F 39783,N1(OC(=O)C=CC(N2CCCC2)=O)C(C(=O)NC2CCCC2(F)F)C2CC(O)C1C2 39784,N1(C(=O)OC)CCC(CNC(C2CSCC2NC(=O)CC2CC=CC2)=O)C1 39785,C(C)(C1CCCc2ccccc21)NC(c1ccc(Cl)cc1F)C 39786,c1(N2CCCC(C(C)NC(c3ccc(C)nc3)=O)C2)ncnc2sc(C)nc12 39787,C1(C(=O)NCc2cc(CC)no2)C2CCN(C(C3COCC(C)O3)=O)CC12 39788,CCCCC(CNC(=O)C=CC1CC1)NC(C1CSCN1C(=O)OC)=O 39789,c1(CC(=O)NC(CN(C(CN(CCOC)C)=O)C)C)ccc(Br)c(F)c1 39790,c1(C(C)C(=O)NCCN(C(=O)Cc2ccc(CO)cc2)C)c[nH]c2ccccc12 39791,C(CCN(C)C(c1ncc(C)cc1Br)=O)(C(C)(C)C)NC(CC(COC)C)=O 39792,C1(COC)(CN(C(=O)C(c2ccc(C#N)cc2)(C)C)CC)CCN(CCCF)CC1 39793,C=C(C)C(O)CC(=O)N(C1(NC(=O)Cc2cnn(C3CCCC3)c2)CC1)C 39794,C12(CC(=O)NCc3cccc(C)n3)CCC1CN(C(C1CCCCNC1=O)=O)C2 39795,CC(C)C(O)C(C)(C)C(=O)N1CC(C(=O)NCCC(C)C(C)(C)C)C(F)C1 39796,C(CNC(=O)C(C)(C)C(C)C)(C(C)C(C)C)NC(c1c(C)noc1)=O 39797,C(=O)(C#CC1CCCOC1)Nc1cccc(CNC(C2CC(C)C2)=O)c1 39798,N1(C(CCC)=O)CCC(CF)(NC(C2CC(F)C2)=O)C1 39799,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(C(F)F)nn2)=O)CCC1C 39800,C=CCC(C)(C(F)F)NC(=O)CCNC(=O)CC(C)CNC(=O)CO 39801,Cc1nc(C)c(CCC(=O)NCCC2CN(C(=O)CCOC3CCC3)C2)c(O)n1 39802,CCCCCCCC(=O)NCC(C)NC(=O)CN1CC(=O)N(C)C1=O 39803,C1(CNC(c2cc(C)ns2)=O)(CO)CCN(C(=O)C(C)C2CCOC2)CC1 39804,C1(C(N2CCC(CN(C)C(c3cc(Cl)nc(=N)[nH]3)=O)CC2)=O)CCOCC1(C)C 39805,C(=O)(C(F)CC(C)(C)C)NC(C(=O)Nc1c(C)ncc(Cl)c1)C1CCC1 39806,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 39807,C=C(C)C(CC(=O)N(CCC(C)C)CCOC1(OC)CC1)OCCCO 39808,N1(C(c2nc(C)n(C)c2)=O)C2CCC(C(=O)NC3(C(C)(F)F)CC3)C1CC2 39809,C1(COC)CCCN(C(c2cc(C(=O)OC)ns2)C(=O)NC2CCOC2)C1 39810,c1(CC)nc(N2CCC(CNC(=O)CN(CC(C)(C)C)C)C2)c(C)c(C)n1 39811,N1(C(c2ccccc2)C2CCC2)CCCCC12CNC2 39812,C1(CNC(c2ncoc2C2CCNCC2)=O)CCC(=O)N1 39813,C12(NCC)CCN(C1)C2=O.C1(C(N(CCC(=O)OC)CC)=O)CCC(O)C1 39814,C1(C(N2CC3C(CNC(C(c4cccnc4)C)=O)C3C2)=O)CCCCC12CCC2 39815,CS(=O)(=O)c1cc(CN2CCN(Cc3cnc(Cl)s3)CC2)ccc1Br 39816,C12(C(=O)NCC(c3n(C)ncc3)O)CCN(C1)C(=O)CO2.c1(CO)nc[nH]n1 39817,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 39818,C1(NC(=O)N(C2CCCC2)CCN2CCCCC2)CCS(=O)(=O)C1 39819,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 39820,C1(NC(=O)CC2COCCO2)CC(O)CN(C(c2ccc(N3CCC3)cc2)=O)C1 39821,C(CCCCC(=O)N1CC2CC1(CNC(C)=O)C2)OCC 39822,c1(C(=O)NC2CCCN(C(C3C4COCC34)=O)C2)cc2oc(Br)cc2s1 39823,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)c[nH]3)=O)C2)cnccc1Cl 39824,C(=O)(C(C)(CC)CC)NCC(C)(O)CSC.N1(CC)CCC(N(C(C)=O)C)CC1 39825,C1(C(N(CC)Cc2[nH]nnc2CC)=O)CCCN(C(C2CCN(C)CC2)=O)C1 39826,c1(CNC(CCN2CCCC(C(=O)NC)C2)=O)cccc(OC)c1CC 39827,O=S1(=O)c2cccnc2CN1.c1(CN)cc(C(F)(F)F)on1.C1(CCO)CCCC1 39828,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 39829,C=CCCC(C)(C)CN=c1nc(N2CC(CCO)OC(C)(C)C2)cc(C)[nH]1 39830,C(CCCC(C)NC(=O)C(N1CCCCC1)C)NC(CC1N(CC)CCC1)=O 39831,C(C(C)(F)F)N(C(C=CC(C)NC(=O)C1CC1)=O)C1(Cl)CC1 39832,c1(NC(=O)NCc2cnc(CO)s2)cc(Cl)n[nH]1.C12CC1C2 39833,c1(C(C)NC(=O)CSC(C)(C)C)ccc(CNC(C2(F)CC2)=O)cc1 39834,N1(CC(N2C(c3ccc(OC)cc3)CNCC2)=O)CCSC2CCNCCC12 39835,C1(NCc2c(C)nn(C3CCOC3)c2)C2CCCC1CC2 39836,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 39837,N1(CCNc2n(C)ccn2)CCCC2(CCN2C(=O)CCS(C)(=O)=O)C1 39838,CC1OC2(CO)CC1(C(N1CC3CC3(CNC(=O)Cn3ccccc3=O)C1)=O)C2 39839,C1(CN(C)C)(CO)CCCN(C(C2SCCS2)=O)C1.C12(CCCC1)C(=O)N2 39840,c1(C(=O)NCCCC(C)NC(c2cc(C3CC3)cs2)=O)ncsc1S(N)(=O)=O 39841,C1(C)(C(=O)NCC(C)CN(C(=O)CCCCN2CCOCC2)C)CCC12CCC2 39842,c1(C(=O)NCCCN(C(C2CCCC(OC)C2)=O)CCO)cc(Cl)ccc1N 39843,N1(C(C=CC(C)(C)SC)=O)CC2CN(C(C3CSCN3C(=O)OC)=O)CC2C1 39844,N1(C(c2ccn(CC)n2)=O)CC2CC(C1)N(C(=O)CCC(C)C#N)C2 39845,C1(NC(Cc2cnc(C)s2)=O)CC(N=c2[nH]c3cccc(F)c3s2)C1 39846,C1(N(C(C(C)N(CC(F)(F)F)C)=O)C)CN(C(=O)CCc2nccs2)CC1(C)C 39847,c1(CC(=O)NC2CC(C(=O)OCC)NCC2)cccc(OCCF)c1 39848,C1(C(=O)NC2(CF)CCN(C(=O)C(C3CCOCC3)O)C2)COC2(CCC2)CO1 39849,c1(C(N(C(C)CNC(=O)CC2CCCCC2)C)=O)ccc(Cl)c(N)c1Cl 39850,N1(C(Cc2c(C)nccc2)=O)CC(NC(=O)CSc2ccccc2)CC2(CC2)C1 39851,C(C)(CCC(=O)NC(CSC)C(=O)N(CC(C1CC1)OC)C)OCC 39852,c1(C(=O)NCC2(F)CN(C(CNC(=O)OC)=O)C2)ccc(C)cc1C 39853,C12CN(CC1(F)F)C(=O)N1CCCC1CNC2=O.C1(CC#N)(CO)CCCC1 39854,c1(C(=O)NC(CNC(CC(C)OC)=O)C2CC2)cnc2ncnn2c1C(C)C 39855,C1(CNC(CCC=CCC=C)=O)CC(NC(c2coc(Br)n2)=O)C12CCC2 39856,C1(C(=O)NC(C)CCN(C)C(C2(CC(F)F)CCC2)=O)(COC)CCOC1 39857,c1(C(N(CCCOCCN(C(C(CC=C)C)=O)C)C)=O)c(C)cc(C)nc1O 39858,CCC(C(=O)NCc1cn(CCNC(=O)C(C)OCC(F)(F)F)nn1)N(C)C 39859,N1(C(C(C(C)(C)C)NC(=O)C(F)OC(F)(F)F)=O)CC2C3CCC(O3)C2C1 39860,C(C(C(=O)N1CCN(CCC)C(=O)C1)C(C)(C)C)NC(CCC=C)=O 39861,CN(S(=O)(=O)NCC1CCCCCC1)CCCc1ccc(-c2ccncc2)cc1 39862,c1(NC(CC2CC(CNC(C3C(C(C)C)(CC)C3)=O)C2)=O)cc(C(N)=O)n[nH]1 39863,Cc1cc(C(N2CC3C(C2)N3C(=O)C(C)Sc2ccccc2)=O)c2cc[nH]c2c1 39864,c1(C(N2CCC(NC(Cc3c(C)scc3)=O)C2)=O)cccnc1-n1nccn1 39865,C=C(C)CC1C(=O)N1.C(C)(=O)NCCNCCOC 39866,N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)C1C 39867,c1(CN(C(CCC2(NC(C(C3CC3)OCC)=O)CCC2)=O)C)nnnn1C 39868,Cn1cncc1C(c1nnnn1Cc1cccs1)NCCC(=O)NO 39869,c1(C(N2C(CNC(c3c(C#N)cn[nH]3)=O)CCCCC2)=O)noc2cc(F)ccc12 39870,O=C(N=c1[nH]c(Cl)nc2cc(Cl)ccc12)C1CCN1Cc1ccc(CO)cc1 39871,C1(N=[N+]=[N-])(C(N(CC(C(=O)NC)C)C)=O)CCN(C(C2CCCC2C(C)C)=O)C1 39872,N1(C(CC(C)N2CCCC2=O)=O)CCC(C(F)F)(CNC(C2(Cl)CC2)=O)C1 39873,c1(C(=O)NCC(CO)NC(c2ccc(N(C)C)nn2)=O)cnc2n1CCC2 39874,C#CC1CCN(C(=O)C(CCC=C)NC(C2CCS2(=O)=O)=O)CC1 39875,c1(C(=O)NCC2CN(C(CC(C)(C)C)=O)CC2O)c(N)c(F)cc(F)c1F 39876,CCC(Cc1ccccc1)C(=O)NC(C)CNC(c1cc(C(F)(F)F)no1)=O 39877,S(=O)(=O)(c1ccoc1)Nc1cccc(C(C)(F)F)c1 39878,C(=O)(CCCC(F)F)NCCN(CCC)C(C1CCC2CC1C2(C)C)=O 39879,C=C(C)C(C)(C)C(=O)NCC1CCN(C(C2CC3CC3C2)=O)C(C(=O)OC)C1 39880,c1(C(N2CCC(O)(C(C)CNC(=O)C(O)CF)C2)=O)ncc2ccccn12 39881,C(=O)(NN1CCCC1NC(C1CCC1O)=O)c1c(C)ocn1 39882,N1(C(C)=O)CCC(CC(=O)NC2(CF)CN(C(C3SCC=C3C)=O)C2)C1 39883,c1(C(=O)NCC(CNC(Cn2nnc(C)n2)=O)C)cc(C)c(C)c2ncsc12 39884,N1(C(C(=O)N(c2ccccc2)C(c2n[nH]cc2Cl)=O)C)CCCOCC1.CCO 39885,N12CCC(C1)CN(C(=O)Cc1cnnn1C)CCC2=O.Cc1cocn1 39886,S(=O)(=O)(c1cnc(NCCc2cccc(Cl)c2C)c(Cl)c1)NC(COC)C1CC1 39887,n1(CC)nc(C)c(C(=O)NCC2CCN(C(=O)CC(C)OC)C2)c1Cl 39888,C1(Cl)(C(=O)OC)CC12CCN(Cc1ccncc1)CC2.c12cnn(c1)CCC2 39889,CCC(O)C(C)C(=O)N1CC(CCn2cc(-c3ccc(C)cc3C)nn2)C1 39890,C(=O)(C(O)CCCNC(=O)C(O)COC)NCCC(CC)C 39891,C(C(CNC(=O)CC1(C)CC1)NC(=O)C=C1CCC1)OC 39892,CC1(C)C(NC(c2cc(C3CCC3)no2)=O)CCN1C(=O)Cn1cccc1 39893,C=CC(C)C(C)C(=O)NCCCCCNC(=O)CCCc1sccc1C 39894,C=C=CC(C)C(=O)N1CC=CCC1C(=O)NCCc1scnc1C 39895,C(=O)(CCN(OC)C(=O)C(C)(O)C(F)(F)F)NCCCCCCC#C 39896,C1(S(C)(=O)=O)(C(N(C)CCNC(C2CCC2C(F)F)=O)=O)CC(O)C1 39897,C1(NC(Cc2cncc(C)c2)=O)CC2CCC(C1F)N2C(c1csc(=N)[nH]1)=O 39898,N1(C(c2occ(C)c2)=O)CCC(N=[N+]=[N-])(C(N2CCC(CN=[N+]=[N-])CC2)=O)C1 39899,C(=O)(C(O)CC(N)=O)N1CCC(C)(CC(=O)NC(CCOC)C(C)C)C1 39900,c1(C(C(N2CC3C(CN(C4CCCC4)C(=O)NC)(C3)C2)=O)=O)cccc(OC)c1O 39901,N1(C(C2CCC3CC3C2)=O)CCC(NC(c2ccccn2)=O)C12CCC2 39902,N1(C(C(C)Oc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 39903,c1(NC(N2C(C)CCCC2C2CCNCC2)=O)cccc(S(C)=O)c1 39904,c1(-n2c(C(C)NC(c3c(OCC)nccn3)=O)nnn2)ccc2c(c1)OCCO2 39905,c1(C(N2CCCC(CCNC(C(F)OC)=O)C2)=O)cc2cccc(Cl)c2o1 39906,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 39907,C1(NC(c2csc(-c3ccsc3)n2)=O)CC(O)CN(C(c2cnc(S)[nH]2)=O)C1 39908,C(C(C(=O)NC(c1ncc[nH]1)COC)N1CCC(OCC)C1)OCC 39909,C(=O)(CCC(=O)NN(C)C)NC1C2(CC(NC(CC(C(C)OCC)C)=O)C2)C1 39910,c1(C(N2CC(OC)(CNC(=O)CCOCCF)C2)=O)cc(Br)ccc1Cl 39911,c1(C(N2CCC(Oc3ccccn3)C2)=O)cc(C(F)F)cnc1O 39912,C1(CCC)CN(C(=O)C=C(C)c2cccs2)CC1NC(C1(CC(C)C)CC1)=O 39913,c1(OC)cc(N)c(Cl)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)C1 39914,CC1(O)CCN(C(C2(F)CCN(C(=O)CCc3cnoc3)CC2)=O)CC1 39915,C1(C(=O)NC(C)C(C)(C)C)CN(C(C2(c3ccccc3)CC2)=O)CCC1(C)C 39916,c1(CNC(=O)OC)cc(Cl)cc(C)c1SC.n1(CC)nnnc1C1C2CC(C2)N1 39917,c1(C(C(C)NC(=O)C2CC2)N(C(=O)COC2CCCC2)CCO)ccccc1 39918,C1(C(=O)Nc2cncc(C(=O)OC)c2)CC12CCN(C(=O)COC1CCCC1)C2 39919,N1(CC(CC)O)CCC(F)C(NC(C2(F)CC2c2ccccc2)=O)C1 39920,c1(C(N(C)Cc2nc(-c3cccc(CC#N)c3)no2)=O)cc([N+](=O)[O-])ccc1I 39921,CC1OCCC1(F)C(=O)NCC(C1CCCCC1)NC(=O)CN(C)CCO 39922,C12(CCNC(C(C)=C(CC)C)=O)CCC(C1)N(C(=O)NC1CC1c1ccsc1)C2 39923,c1(C(=O)NC2C(CNC(c3ccc(C4CC4)o3)=O)C2)cc2c(s1)CCCC2 39924,C(CC(CNC(C1(CCF)CCC1)=O)NC(C1(CCF)CCC1)=O)OC 39925,n1(C(C)C)nccc1NC(CC(C)C)c1nnnn1C1CCC1 39926,C1(C2CCCN(C(=O)Cc3ccc4n[nH]cc4c3)C2)(NC(C=CSC)=O)CC1 39927,C1(CC(N2CCOCC(O)C2)C(=O)NCc2ccco2)CC2(CCC2)CO1 39928,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CC2(COC(C)C2)C1 39929,N1(C(c2c(C)onc2)=O)CCN(C(C2C(C)C2C)=O)C2(CCC2)C1 39930,c1(CC(N2CCC3CC23C(=O)NCC23CC(F)(C2)C3)=O)cccc(Br)c1 39931,c1(CC)ccc(CNC(=O)NC2CCC(CC)CC2)nc1O 39932,C(=O)(C(O)CC[S+](C)C)NCC1(F)CCN(C(c2cc(OCC)n[nH]2)=O)CC1 39933,c1(N(C)C)nccc(C(=O)NC2CCN(C(=O)C(C)Br)CC2O)c1Cl 39934,[N-]=[N+]=NCCC(=O)N(CCC(F)Cn1cc(CCOC(=N)O)nn1)C(C)=O 39935,C(=O)(C(F)C(CC)CC)N1C(C(=O)NC(CN(CCCC)C)C)CC(OC)C1 39936,N1(C(C(CC)N(C)C)=O)CC2(CC(N(C(=O)CC(C)COC)C)C2)C1 39937,Cc1ncc(C#N)cc1NC(C1(F)CCN(C(=O)C=Cc2ccsc2)CC1)=O 39938,C(CN=c1ccnc(NC(c2cccc(F)c2)CC(N)=O)[nH]1)C1C(C)(C)NC(=O)O1 39939,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 39940,c1(CNC2CC(C)(C)CN(C(=O)C#CC3(C)COC3)C2)c[nH]c2ccncc2c1=O 39941,C12CN(CCC1O)C(=O)C(C)(C)C(=O)N2C.CC(CF)CC(=O)OC(C)(C)C 39942,CC(C)C(CC(=O)Nn1cncn1)NC(=O)C(C)(C)c1ccno1 39943,c1(C(=O)NC2C3CN(C(C4CCC(=O)N4)=O)C2C3)c[nH]nc1[N+](=O)[O-] 39944,N1(C(C(C)(C)C#N)=O)CC=C(CCNC(C2(CO)CC2(F)F)=O)CC1 39945,c1(C(=O)NCC(CC=C)NC(CCC#C)=O)ccc(OCC)nn1 39946,C1(C(=O)NC(CCNC(c2c(C)ncnc2)=O)C)COc2ccc(F)cc2C1 39947,c1(N2C(C)CC(NC(=O)CCCc3cnccn3)CC2)ncc([N+](=O)[O-])cc1Cl 39948,OC1CCCN(C(=NCc2c(F)cc(Cl)cc2F)NC2CCS(=O)(=O)C2)CC1 39949,c1(C(=O)NCCC2(OC)CN(C(C(CC)N(C)C)=O)C2)c(Cl)ccc2c1OCO2 39950,c1(C(=O)NCC(C2CCC2)NC(=O)Cn2cncn2)cccn2cnnc12 39951,C12(C(=O)NCc3ccnc(C)n3)CCC1CN(C(C1CCCC1F)=O)C2 39952,C(=O)(CCS(=O)(=O)NC1CC(C(=O)OC)(CN)C1)OC 39953,C(C(C(C)C)NC(=O)C(F)=C(C)C)(c1ccccc1)NC(c1n(CC)cnn1)=O 39954,c1(C(=O)NC2C(NC(=O)CC3CCC(O)C3)CC2)cccc2c1CCC2=O 39955,C(C(COC)C(=O)NC1CCC(CNC(=O)C(F)(F)c2cnn(C)c2)CC1)OC 39956,C#Cc1c[nH]nc1C(N1C(C(=O)NC)CC1C)=O 39957,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2cc(Cl)cn2)C1 39958,C(=O)(C1=CCCCCC1)N(C(C)C(=O)NCC1CC(=O)NC(C)C1)CC 39959,C1(CNC(c2cnc(CC)s2)=O)(OC)CCN(C(=O)C(F)(F)c2nccs2)C1 39960,c1(C(N2C(CNC(C3CCN(OC)CC3)=O)CC2)=O)cnc(O)c2c1NCCC2 39961,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(CC(C)C)NC(C1CC(C)=NO1)=O 39962,N1(C(C(C2CCOC2)NC(c2ccc(C#C)o2)=O)=O)CC(C2CCCCC2)C1 39963,C12(C(N(C3CCCN(C(c4c(CC)c[nH]n4)=O)CC3)C)=O)CC3CC(CC1C3)C2 39964,C12(NC(c3c(C)ncs3)=O)CCC(CN(C(c3ccc(F)cc3Cl)=O)C1)C2 39965,C(C1CN(C(C2(C)CCCCO2)=O)CC1C(N1CC(COCC)C1)=O)=CC 39966,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 39967,Cc1nc(=N)[nH]cc1C(N1CCCCC1C1CC1)C(=O)NC1CC1 39968,C1(CNC(C(n2cc(Cl)cn2)C)=O)CCCCN1C(=O)Cc1cccnc1 39969,C1(c2c(C)nn(C)c2)CC(C(=O)N=c2cc(C(C)C)[nH][nH]2)=CC1C(=O)O 39970,c1(C(C)(C)C)nc(C(=O)NCCCC2CCCN2C(=O)CN2CCOC2=O)co1 39971,Cc1nn(C)cc1C1CC1C(=O)NC1CCN(C(=O)CSc2ccccc2Cl)C1 39972,c1(CS(CC2OCCN(c3nccc(OC)c3)C2)=O)cc2c(cc1O)CCCC2 39973,C(=O)(C1CCCn2nccc21)C1=CC=NC(N2CCC3(CCC(O)C3)C2)=NC(CC)=N1 39974,N1(C(C(C2CC2)NC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 39975,C12(C=CCN1C(=O)COC)C(=O)NC2.C(CCN=[N+]=[N-])OC.C12(CCC1)CCS2 39976,C(C(CNC(C1(Cl)CC1)=O)S(C)(=O)=O)NC(C(C(C)C)n1cnnn1)=O 39977,c1(Nn2nc(C(=O)Oc3cc(C)on3)cc2C)ccc2ncsc2c1Br.C1CN[SH]1(C)=O 39978,Nc1ccc(C(=O)NC(CNC(=O)CCc2ncccn2)C2CC2)nc1N 39979,N1(C(c2n[nH]c(CC)c2C)=O)CC(C(N2CCC(C(N)=O)CC2)=O)OC(C)C1 39980,N1(C(=O)N(Cc2c(Cl)ccc(C(C)(C)C)c2)C2CC2)CC23CCC2(COC3)C1 39981,c1(C(=O)NC(C2CN(C(C(=O)NCC)=O)C2)C)ccc2nnc(O)n2c1 39982,c1(C(=O)NC(CCNC(C(C)OCCC#C)=O)C(C)C)cccc(=O)n1C 39983,c1(CN2C(C)CN(C(c3c[nH]c(C(F)(F)F)c3)=O)CC2)cccc([N+](=O)[O-])c1 39984,Cc1ccc(SCC(C2(C)OCCO2)C)cc1C(C)C 39985,O=C(C(O)CC1CCCC1)NC1CN(C(C2CC2(Cl)Cl)=O)C1 39986,Cc1ncsc1C=CC(=O)NC1CCC1CNC(C1CCN(CC(F)F)C1)=O 39987,c1(CCNC(C(C2CCCC2)NC(C2C3CC4C(C3)C24)=O)=O)ncccc1Cl 39988,C1(C(=O)NCC2C(CNC(CC=CC)=O)C2)CCc2ncsc2C1 39989,c1(C(N(CCCCNC(C(=Cc2ccccn2)C)=O)C)=O)cnc2[nH]ccc2n1 39990,Cn1nc(C2CC2)nc1CC(=O)N(C1CCCCC1)C(=O)C(=O)C1CCCC1 39991,C1(NC(=O)CC2(c3cnn[nH]3)OCCO2)CC12CCN(O)C2 39992,c1(C(=O)NC2CC(NC(C3CCCN(C(=O)NC)C3)=O)C2)ccc2n[nH]cc2c1 39993,c1(C(=O)NC2C(NC(CC(C)c3ccco3)=O)C2)cccc(P(C)(C)=O)c1 39994,c1(C(=O)NCCCNC(=O)C=CCO)ccc(OCCCNC(=O)C=CCl)cc1 39995,Cc1nn(C)nc1C(=O)NCc1cn(C)nn1 39996,CCCC(CC(C)C)C(=O)NCC1(NC(c2cc(N)nc(Br)c2)=O)CCC1 39997,NS(=O)(=O)C1CN(C(C2(c3ccc(Cl)c(F)c3)CC2)=O)C2(CCC2)C1 39998,c1(CNC(C(C)(C)C2CCOC2)=O)ccc2c(c1)CC2.c12nc(cs1)CNC2=O 39999,c1(C(=O)NC2C(CNC(C(CCC)OCC)=O)CCC2)cn(C)c(C)cc1=O 40000,CC1(C)C(CC(=O)NCCC2C=CCC2)CCN1C(=O)CCCC1CCC1 40001,Cc1nc(C(C)C)ncc1C(=O)NCCCN(C(=O)CNC(c1ccco1)=O)C 40002,CC(CNC(C1COCC(C)O1)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40003,n1(CC(C)C)c(SCC2NC3CC2C3)nc2sc3c(c2c1=O)CCC3 40004,C=CCC(F)(F)C(=O)NCC1(C)CCC(NC(=O)COCC(C)C)C1 40005,N1(C(CN(C2CCC2)C)=O)CCCN(C(C2CC2F)=O)C(c2ccccc2)C1 40006,CC(C)C(O)C(F)(F)C(=O)NC1CCC(CNC(=O)Cc2ccc(Cl)s2)C1 40007,c1(C(=O)NCC2(CNC(C(COC)O)=O)CC2)c(C)cc(C)oc1=O 40008,C1(C(=O)NCC2(CNC(CCCC(C)C)=O)CC23CCC3)CC2(C1)CC(C)(C)C2 40009,C1(N(CCOC)C)CCN(C(c2cn(C)cn2)C(=O)NCC(C)C)CC1 40010,CCCCCC(C)CC(=O)NCCC(O)CNC(=O)CC1CNC(=O)C1 40011,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40012,C(CCSC)(C(=O)NC(C)(C)CNC(c1cn(Cc2ccccn2)nn1)=O)OC 40013,C1(C(N(CC)CC2CCC2)=O)CCC(O)CN1C(=O)CCCC(C)C 40014,C1(C(N2C(CC(=O)OC)COCC2)=O)CC2OCCC2N(C(=O)CCCCCl)C1 40015,c1(C(N2C(C)CN(C(C3CC4CC4C3)=O)CC2)=O)cc2c(nc1O)CCCCC2 40016,Cc1nn(C2CCC2)cc1C(N1CC(CNC(=O)CCC(=O)C2CC2)C(O)C1)=O 40017,CCCC(CCC)C(=O)N1CC2CC2(C(=O)Nc2cccc(C)c2O)C1 40018,Cc1nc(C(N2CCC3CC3(NC(c3cscc3Cl)=O)CC2)=O)c2ccccn12 40019,Cc1cc2sc(C(=O)N(CCC(C(C)(C)C)NC(c3ccccc3)=O)C)cc2s1 40020,C(=O)(C(C)(C)C(C)(F)F)NCC(C)N(C(C1CC1(C)C(F)F)=O)CC 40021,N1(C(CCS(C)(=O)=O)=O)CCC(C2CCN(C(C3CCSC3)=O)C2)CC1 40022,c1(CC(=O)Nc2ccn(CCOC)n2)nnc2n1CCNC2C 40023,N1(C(CC(CN(C)C)NC(C(=O)NC(C)C)=O)=O)CC2(CNC(=O)O2)C1 40024,C1(NS(CCC)(=O)=O)(NC(=O)Nc2ccccn2)CCCN(C(=O)C(C)SC)C1 40025,c1(C(=O)NCC2CC(NC(c3ccncn3)=O)C(O)C2)cc2c[nH]cnc-2n1 40026,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40027,O=C1CCC2(NC(=O)C(=O)NCCC3=CCCCC3)CCCCC2N1 40028,C1(OC)CN(C(=O)CONC(C2(C)C=CCCC2)=O)CCO1 40029,N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCC2CC(=O)N(C)C2)CC(F)C1 40030,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40031,c1(C(COC(c2nnn(CC(C)C)c2C)=O)OC)c(F)cccc1F 40032,n1(C(C)C)ncc(C(N2CCN(CCNC(=O)CC(C)N(C)C)CC2)=O)c1C(F)F 40033,N1(C(c2sc(C)c(O)n2)=O)CCCC(C2CN(C(c3cccc(F)c3)=O)C2)C1 40034,N1(C(c2c(C)[nH]cc2)=O)CCC2CC2(C(=O)Nc2cc(O)ccc2F)CC1 40035,CC(CCNC(=O)NC1COCCN1Cl)CCN(C)C 40036,c1(C(N2CCC(NC(c3c(C)scc3)=O)C2)=O)cnc2ccccn12 40037,C1(OC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40038,c1(C(N2C3C(CNC(C4C(C)CC4)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40039,N1(C(C=C(CCC)CCC)=O)CCc2nc(CNC(=O)C=C3CCC3)sc2C1 40040,C=C(C)CCCC(=O)N(CCCNC(c1nc(OC)cc(OCC)n1)=O)C 40041,c1(CC(=O)OCC)ccc(C2CC2OC)cc1 40042,CC1=C(C)CC(C(=O)NC(CCN(C(=O)CCCC2CCC2)C)C(C)(C)C)CC1 40043,C(=O)(C(C#N)CC)NC(CC)CNC(=O)CN1CCOCC1 40044,C1(c2nn[nH]n2)(SC)CC2CCC(C1)N2c1cnc(-c2ccc(COC)o2)nc1 40045,c1(OC2CCCN(C(c3ncc[nH]3)C)C2)cc(F)ccc1F 40046,CC(C)(C)CC(C)(C)C(=O)N1CCC1Cn1cc(-c2ccnc(C#N)c2)nn1 40047,C1(O)(CNC(C2C(NC(CN(C)C(N)=O)=O)COCC2)=O)CC(C)(C)C1 40048,c1(C2n3nc(-c4ccncc4)nc32)ccc(Cl)c(Cl)c1.C1(C2(C)CC2)CCCC1 40049,c1(CN2C(C)(C(=O)NCc3cc(C)n(C)n3)CC2)ccc2ccccc2c1 40050,c1(NC(C=C)=O)ccc(C(=O)NC23CC2CN(C(c2cnc[nH]c2=N)=O)C3)cc1 40051,CCC(C)C(O)CC(=O)NCCOCCNC(c1cnc2ccccn12)=O 40052,C1(CC2CCC(C)C2)CCCC(C)(C)C1.N12CCC(CC1)C(=O)NC2=O 40053,c1(C2(C(N3CCC(NC(c4nocc4Cl)=O)C3)=O)CC2)ccc(Cl)c(Cl)c1 40054,N1(C(COCCCCC)=O)CCC(CCC(=O)NCc2scnc2C)C1 40055,c1(C(=O)NC(CNC(CC=CC)=O)CC)csc(-c2nc[nH]n2)n1 40056,Cn1ccc2cccc(C(N3CCC(C)(NC(C4CCCS4(=O)=O)=O)C3)=O)c12 40057,N1(C(C(C)CF)=O)CC2CCC(C1)N2C1CCN(c2ncnc(=N)[nH]2)CC1 40058,c1(C(C(=O)NC2CCCC2)N(CC(C)C)CC#N)cnc2n1CCC2 40059,N1(C(C(C)SC)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40060,c1(C(=O)NC2CCN(C(C(CC)(F)F)=O)C2)cc(F)c(SC)cc1F 40061,c1(CNC(C2N(C(CSCC)=O)CCOC2)=O)ccc2nccn2c1 40062,c1(NC(=O)CC2(NC(=O)Cc3cc(Cl)ccc3O)CCC2)cccc2c[nH]nc12 40063,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40064,c1(OC)nc(C(=O)NCCN(C2CCCC2)C(C2C3CCCCC23)=O)sc1C 40065,C(CC(C)C(=O)N(C1CCCN(C(C2CN(CC(F)(F)F)C2)=O)C1)C)=CCC 40066,CC(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2ccc(CC#N)cc2)=O)C1 40067,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40068,c1(CN2CCC(C(C)NC(CC(CC)C)=O)CC2)ccc(Br)cc1F 40069,CC1(C)COCCC1CCNC(C1C(NC(=O)CCCCCF)C1)=O 40070,C1(NC(N(CCC)CCF)=O)CCC1CNC(=O)OC(C)C 40071,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)Cc2ccsc2)CC(O)C1 40072,C(=O)(C(C)C(O)CCCC)NC1C(NC(CC(=C)C)=O)C1 40073,c1(-n2c3nc(n2)C3C)ccnc2ccccc12.N1(CCSC2CC2)CCOCC1.S.C 40074,N1(C(C(C)Cc2ccc(F)cc2)=O)CCC2(CCN(C(C34COCC3C4)=O)C2)C1 40075,N1(C(C2N(C(CC(C)(C)C(F)F)=O)CCCCC2)=O)CCC2(CCCCO2)C1 40076,Cc1ncc(C(=O)NC(C)CC(=O)N2CCCC2CNC(N)=O)c(C)n1 40077,C1(NC(c2c(C(C)C)onc2)=O)CC(C)N(C(c2cn(C)cn2)=O)C1 40078,N1(C(CN(C2CC2)CC)=O)CCN(C)C(CNC(C2CCCCC(=O)N2)=O)C1 40079,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(C1CCS(=O)(=O)CC1)=O)CC2 40080,C1(NC(=O)CCc2cn[nH]c2)CCN(C(=O)CSC(F)(F)F)CCC1(F)F 40081,Cc1csc(C(F)(F)C(=O)NC(C)C(C)NC(C2(O)CCC2)=O)n1 40082,c1(C(N2CCC=C(CNC(CC3C(C)CCO3)=O)C2)=O)ccc2c(c1)C(=O)NC2=O 40083,c1(C2CC(CC)C2)nc(CCCN2CCC(C)C2)nn1C1CCCOC1 40084,N1(C2CCC(NC(CN(C)CCO)=O)C2)CCN(C(=O)C2=CCC2)CC1 40085,c1(N2CCCC(NC(C3CCCCN3C3CC3)=O)CC2)cc2ncnn2cn1 40086,c1(COCC(N2CCC(CNC(C(C=C)(C)C)=O)CC2)=O)ccc2c(c1)OCC2 40087,Cc1no[nH]c1=NC(=O)C1(C)CCN(C(c2ccccc2)C2CCC2)C1 40088,c1(C(N2CC3C(CNC(CC(C)F)=O)(C3)C2)=O)ccc2c(Br)cnn2c1 40089,N1(C(C(COCC)C)=O)CC(N(C(=O)Cc2cncs2)C)C2(CC2)C1 40090,CN1CCN(CCCCCNC(C2CCCN2Cc2cccc(Cl)c2)=O)CC1 40091,C1(C(=O)NCCN(C(C)C)C(c2ccc(N(C)C)cc2)=O)CCC(N=[N+]=[N-])CC1 40092,c1(OC)ccc(F)c(F)c1.c12nc(co1)C(=O)NC2C.C12CC1NCC(=O)N2 40093,c1(CC(C)C(=O)OCCCn2cc(-c3ccnn3C3CC3)nn2)ccc(F)c(F)c1 40094,CCCCC(C(=O)NC1CCN(C=O)C1)NC(c1c[nH]nc1OC)=O 40095,N1(C(C2(C=C)CC2)=O)CCN(C(c2cn(CC(F)(F)F)nn2)=O)CC(C(=O)OC)C1 40096,CC1CCC=C1C(=O)NC1(O)CN(C(=O)CCNc2ccc(Cl)cc2Cl)C1 40097,c1(OCCC(=O)NCC2N(C(C(C)(C)OC(C)C)=O)CCC2)ccc(Cl)cc1 40098,C1(CCC)CN(C(c2cc(Cl)ccc2F)=O)CCN1C(=O)CC(O)C1CCCC1 40099,Cc1[nH]c2ccccc2c1C(=O)NCC1COCCN(C(c2c[nH]c(Br)c2)=O)C1 40100,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40101,c1(C(=O)NC2CC(C)N(C(C3CCC(=O)N3)=O)C2)cc(F)cnc1Cl 40102,C1(C(=O)NC2CC(NC(C3(c4ccc(O)cc4)CC3)=O)C2)CC2COCC2C1 40103,C(=O)(N=c1nnn(CC)[nH]1)NCC(=C)C(F)(F)F 40104,C(=O)(C(C)(C)C(=O)NC1CCC(NC(c2ncc[nH]c2=O)=O)CC1)OC 40105,C12(COC)COC(C(N3CCCCC3CNC(=O)Cc3ccccc3C)=O)(C1)C2 40106,c1(CC)cc(NCC(C)(C2CCC2)NC(C2CCC(C(F)(F)F)CC2)=O)ncn1 40107,C(C(=O)N1CCCC1(C)C1(C(=O)NC2CCCC(C)(C)C2)CC1)(C(C)(C)C)OCC 40108,c1(C(N(CCCNC(c2ccn(CCN(C)C)n2)=O)C)=O)csc(Cl)c1Cl 40109,c1(CN(C2CCN(C(c3nccn3C)=O)C2)C)ccc(Br)c(CO)c1 40110,C1(CCC(=O)OC)CCCN(C(C2CCCC(CO)C2)C(=O)NC2CC2)C1 40111,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40112,N1(C(CCCC=C)=O)CCC2CCCN(C(c3cc(C4CC4)ccc3F)=O)C2C1 40113,C1(C2CCN(C(C(C)=CC)=O)C2)CCCCN1C(=O)CSc1ccncc1 40114,C(CCCCCCC(=O)NCCCCC1(NC(=O)CC(C)C(C)C)CC1)SC 40115,c1(OC)ncc(C(=O)NC2CN(C(=O)COCC3CCOC3)C2)nc1C 40116,CC(O)(CCNC(N1CCNC(c2ccc(C(F)(F)F)cc2)C1)=O)C(F)(F)F 40117,c1(C2CCN(C(c3n(CC)ncn3)=O)CC2)ccc(C#N)cc1 40118,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40119,N1(NC(CCC)=O)CCN(C(=O)Cc2cnc(C(F)(F)F)s2)CC1C 40120,C1(NC(C(C)Cc2ccccc2F)=O)CC2CCC1N2C(=O)CCC1(CO)CC1 40121,CC1=C(C(=O)NC2CCN(C(=O)C(c3cnccn3)C)CC2O)C(=O)OC1(C)C 40122,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40123,C1(C)(C(=O)NCC2CCN(C(CN(c3ccccc3Cl)C)=O)CC2)CNC(=O)C1 40124,N1(C(C2(OC)CC2)=O)CCC(O)(CNC(=O)CC2CCN(C)C2=O)CC1 40125,N1(C(C2C(CC)CCO2)=O)CCCCC(N(C)C(C2(CC)CCNC2=O)=O)C1 40126,C1(C2CCN(C(C34CC(C3)C4)=O)CC2)(NC(C(CCCC)C(C)C)=O)CCC1 40127,C(c1ccc(C(F)(F)F)cc1C)=CC(N1C(CC(=O)OCC)(C(=O)O)CCC1)=O 40128,C1(C(=O)OC)CC=CCN1C(=O)OCC1CC2CCCC12 40129,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40130,C1(C(C)OC)CCCCN1C(=O)Cn1cc(C2CC2NC(C2CC23CCC3)=O)nn1 40131,n1(CC#C)cccc1C(=O)NCC1CC(CNC(C2(c3ncco3)CC2)=O)CO1 40132,C(C(C)C(=O)NCC(C1CC1)NC(c1ccn(CCF)n1)=O)SC 40133,N1(C(c2c(C(C)(C)C)ccs2)=O)CC(CNC(c2nsnc2O)=O)C1(C)C 40134,C1(C#N)(C(N(CC(=O)N(C2CCCC(O)C2)C)CC)=O)CC2CC2C1 40135,Cc1[nH][nH]c(=N)c1NC(=O)Cn1cc(CC2CCN(C(N3CCCC3=O)=O)C2)nn1 40136,C1(C(N(CCCNC(=O)CC2CCC(C(F)(F)F)O2)CC)=O)CCC(C)(C)O1 40137,CC1CN(C(=O)CSc2nncs2)CCC1NC(=O)C(C)(C)C1(O)CCOC1 40138,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40139,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40140,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2F)=O)CC2(CC2)C1 40141,C(c1cnn(C)c1)=CC(=O)NC(CC=CC(=O)N(C1C(C)CCC1)C)(C)C 40142,C1(NC(CN(C(=O)C(C)OCCCC(=O)SC)CCOC)=O)CC1 40143,C1(CNC(=O)CC2C=CCC2)COCCN(C(=O)CC2CCCS(=O)(=O)C2)C1 40144,C(CCCCC(=O)N1CC1c1cccc(N)c1)n1cc(C2C(OC)OCCC2)nn1 40145,CC1(C)CCC(C(=O)NCC2CN(C(=O)CC3CCSCC3)C2)OC1 40146,C#CC1(C(N2CC(F)(C(=O)NC34CC(C3)C4)C2)=O)CC(=O)C1 40147,CCCC(C(O)C(=O)NCCSC1COCC1O)NC(=O)CNC(=O)OC 40148,c1(NC(C)=O)ccc(F)c(CC2(CC3CC3)CN(NC)C2)c1 40149,C(=O)(CC(c1ccccc1)NC(=O)OC(C)(C)C)NC(CC)CSC 40150,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40151,C1(CN2C(C(=O)NC)CC2C)CN(C(=O)OC(C)(C)C)CC1C 40152,Nc1c(C(N2CC(C3CN(C(=O)CCCCCO)C3)C2)=O)ccc(F)c1Cl 40153,C1(NC(C(CC)NC(C)=O)=O)CC(C)CN(C(C2CCS(=O)(=O)CC2)=O)C1 40154,C(CCCC(=O)NCC(c1cccnc1)O)NC(c1cc(OC)n[nH]1)=O 40155,CN=c1cc(C(=O)NCC2(F)CCC(NC(c3occc3C)=O)C2)cc[nH]1 40156,Cc1nc(C(N2CCC(OC3CC3)C2)=O)ccc1NC(=O)CC1CCCC(C)C1 40157,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCN(CC(F)(F)F)C)C1 40158,C1COC2(COC2)C1.n1(CCC(N2CC(CCC=C)C2)=O)cc(CC)nn1 40159,C1(CCNC(CCC(=O)NCCOCC(=O)OCC)=O)CC(C)NC(C)C1 40160,Cc1ccccc1C(=O)NC(C)CCNC(=O)CCCc1cncs1 40161,C(C(C(=O)N)OC)SCC.c1(C(=O)NC(=O)COCCOC)cc(C(F)F)on1 40162,c1(N2CCN(C(C)C)CC2)nc(NC2CCCOC2C)nc2scnc12 40163,c1(OC)ccc2cc(C(N3CC(CCNC(C4(Cl)CC4)=O)C(C)C3)=O)nnc2c1 40164,C1(NC(CC2C(=O)NC(=N)S2)=O)CCC2CCN(C(=O)C(c3ccccc3)F)C12 40165,c1(C(=O)NC(C)C(F)(F)F)cccnc1C(N1CCC(CC#N)CC1)=O 40166,N1(C(Cc2c(C)con2)=O)CCC(C)(C)C(CNC(=O)Cn2cc(CO)nn2)C1 40167,C1(C2CCOCC2)(NC(C2CC(NC(C(=O)NC(C)C)=O)C2)=O)CC1 40168,c1(C(=O)NC(C)C(c2ccccc2)NC(C2CCNC2=O)=O)cc(Cl)ncc1N 40169,C1(NC(=O)Cc2cccnc2O)C2CC3CN(C(C4CCCSC4)=O)C1C3C2 40170,N1(C(=O)Nc2ccc(C)cc2)CCC2(C(N3CC(COCC)C3)=O)C(F)(F)C2C1 40171,C1(SC)CCN(CC2CC(F)CN2CCCCN2CCCC2)CC1 40172,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40173,C(=O)(C1=CCCSC1)NC1(CNC(C(C)OCc2ccccc2)=O)CCOC1 40174,N1(C(c2cc(CC)no2)=O)CC(NC(C2CC2c2ccccc2)=O)CC(F)(F)C1 40175,C12(C(N3CCN(C(c4ccc(C)c(C)c4)=O)C(C)C3)=O)CCCC1CC(=O)C2 40176,CC1(C)CCC(CNC(=O)C(C2CCCCC2)F)N(C(=O)CN2CCSCC2)C1 40177,c1(C(N2CC(C)C(NC(c3cc[nH]n3)=O)C2)=O)cccc(C(N)=O)c1N 40178,N1(C(C(CC)CCOC)=O)CC2CCN(C(C3CC3(F)F)=O)CC2C1 40179,N1(C(c2nsc(C(F)F)n2)=O)CCC(n2cc(-c3ccc(Cl)nc3)nn2)CC1 40180,C1(OC)(CNC(C2CC(C)(C)C2)=O)CN(C(C2CC2C(C)C)=O)C1 40181,C1(C(=O)NCCOCC(=O)NCC2CCC(C3CC3)CC2)CCCCC1(F)F 40182,c1(CC(N2CCC(CNC(c3snc(C(C)C)n3)=O)C2)=O)cc(C#N)ccc1F 40183,C1(NC(CSCCC)=O)C2CCN(C(c3cnn(C(C)C)c3F)=O)CCC12 40184,CCC(C)(CCC(C)C)C(=O)NC1CC(C(N2CCC(O)C(O)C2)=O)C1 40185,c1(-c2cc(C)[nH]c2C)csc(=Nc2cccc(Cl)n2)n1CCC1CCSC1 40186,C(c1cccc(Cl)c1)=CC(=O)NCCCN(C(CC(=O)OC)=O)CC.CC(F)(F)F 40187,C(CC(C)C(=O)N1CC(CNC(c2cnc(COC)nc2)=O)CC1C)=CCC 40188,C=CCC(C(=O)NCC1CC(OC)CN1C(c1cnc2[nH]ncc2c1)=O)C(C)C 40189,c1(CCNC(C2COC(C3CC3)C2)=O)nc2cc(Cl)cnc2[nH]1 40190,C(=O)(C(C)(C)C(O)C(C)C)NC1CN(C(c2c(C)nn(C)c2F)=O)CC12CC2 40191,N1(C(C=CC(C)=O)=O)CCC(C(C)(C)O)(N(C(C2C3CC4C(C3)C24)=O)CCO)CC1 40192,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40193,c1(N(C2CCSCC2)C)ncc2ccsc2n1.C12CCCN(C1)C2=O 40194,C12(C(N3C(COC)CCCC3)=O)COCC1CN(C(C1CC(C)(C)C1)=O)C2 40195,C(=O)(CC(C)CC(C)C)N1CCC(C(C(=O)N(CCC(CCC)O)CC)C)CC1 40196,c1(CNC(C2CCC(=O)N2)=O)ccc(CNC(C2CCCS2(=O)=O)=O)cc1 40197,c1(CSCC)ccc(F)c(Cn2cccc2C(=O)OC)c1 40198,N1(C(CCCCN(C)C)=O)CC2(CCCC2)C1C(N1CCC2(CCSC2)C1)=O 40199,Cc1cn2cc(CC(=O)NCC(C)CN(C(=O)CC(C)CF)C)nc2s1 40200,c1(NC(N(C(CNC(C(C)O)=O)C)C)=O)nccc(Sc2ccccc2)n1 40201,n1(C(C(=O)NCC(C2CC2)NC(CCSC)=O)C)cc(C(C)O)nn1 40202,C1(NC(c2c(C)noc2)=O)CC=C(C(=O)NCc2ccoc2)C1 40203,c1(C(N(CC(C)NC(c2cnn[nH]2)=O)C)=O)ccc(COc2ccsc2)s1 40204,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)N(C)C)C2)CCO1 40205,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40206,N1(S(C(C)C)(=O)=O)CCC2(COCCN2Cc2ccc(CO)o2)C1 40207,C1(CNC(=O)COCC2CCCO2)C2CCC(C2)N1C(=O)CC1CCCC(CO)C1 40208,c1(CC)sc(C(=O)NC(C)(C)CNC(c2cc(CC(C)C)[nH]n2)=O)cc1C 40209,C(CCCC(=O)NC1CC(NC(c2ccnc(Cl)c2)=O)C1)(OC)OC 40210,CCCCC(CC)C(=O)N1CC(CNC(=O)CN2CCCS2(=O)=O)CC1(C)C 40211,C1(C(=O)NN2CC(CNC(c3cc(Cc4ccccc4)on3)=O)C2)C2CCC(=O)C12 40212,c1(C(=O)NCCC(C)N(C(C(C)c2ccsc2)=O)C)cnc2[nH]nnc2c1 40213,C(=O)(C1CCCn2ccnc21)NC1CCN(C(C(C2CCC2)OC)=O)CC1(C)C 40214,c1(OC(c2ncc(C(N3C(C(=O)OC)CC3)=O)s2)C)ccc(OC)c(C)c1 40215,CC1(NC(c2ccc(F)cn2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 40216,Cc1occc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(O)C2CCOC2)C1 40217,C#Cc1cncc(NC(=O)NCC(=O)NC(c2ccc(Br)cc2)C)c1 40218,c1(C(C)=O)[nH]c(C)c(C(N2CC(CNC(=O)COC3CCOC3)C2)=O)c1C 40219,C(=O)(C(Cc1ccco1)NC(C1CNC(=O)N1)=O)N(CCCC)CCO 40220,c1(C(=O)NC2C(NC(C(c3ccccc3F)OC)=O)CCC2)cnc(O)c(F)c1 40221,C1(C(=O)OCC)OCCNCC1N(c1ncncc1F)C(C1CC(C)C1)=O 40222,CCC(CC(=O)NC1CCC(C)(NC(c2cnn(C)n2)=O)CC1)CC(C)C 40223,c1(C(=O)OCC(=O)NC2CC(NC(Cc3cc(C)[nH]n3)=O)C2)ccc(F)c(Cl)c1 40224,CCCCC(CC)C(=O)NC1CC(C)(C(=O)N(C)Cc2ncc[nH]2)C1 40225,C(=O)(C1=CC2CCC(C1)C2)NCC(CO)NC(CCSC)=O 40226,c1(C(N2CC(CC(=O)OC)C3(C2)CC3)=O)ccc2ncn(C)c(=O)c2c1 40227,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40228,c1(C(=O)NCC(C)CN(C(COC)=O)CC(N)=O)oc2ccccc2c1CS(C)=O 40229,c1(C2CCC(C(=O)NCCCNC(CCC=CCC=C)=O)C2)ccc(F)c(F)c1 40230,C12CCCCC1(C)NC2=O.c1(CNC(CCN(CC)CC)=O)ccc(C)cc1F 40231,N1(C(C(C)NC(N)=O)=O)CCCC1(C)CNC(=O)CCC1CCC(CO)CC1 40232,C1(C(N2CC(CNC(c3cncc(C)n3)=O)OCC2)=O)CCCCC1(C)C 40233,C(C(F)(F)C(N)=O)NC(C1(CCC=C)CN(C(=O)CN2CCC(C)C2)C1)=O 40234,Nc1cc2[nH]c(O)nc2cc1C(N1CC2(CCC2NC(C2CC2F)=O)C1)=O 40235,C(=O)(CCCC(F)(F)CO)N1C(C2(NC(=O)CCC34CCC(CC3)C4)CC2)CCC1 40236,C1(F)(CNC(C(C)OCCC=C)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1 40237,c1(C(=O)NCCc2c[nH]c(=NC)s2)ccc(OC)cc1S(C)(=O)=O 40238,Cc1nc(C=CC(=O)NC2CCC(CCNC(C3CC3F)=O)C2)cs1 40239,c1(C(N2CC(CNC(=O)C(C)(C)N(C)C)C3(CC3)C2)=O)ccc(N)cc1C#N.CO 40240,N1(C(c2ccn(CCC)n2)=O)CCC(C)(C)C1CNC(=O)C(C)(CC)CO 40241,c1(C(=O)NCC2(NC(COC(CC)(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 40242,c1(C(N2C(C)(C(=O)Nc3ccc(O)nc3)CC2)=O)cn2ccc(Cl)cc2n1 40243,c1(OC)cc([N+](=O)[O-])c(C(N2CC3CCCC(C2)N3C(=O)CC#N)=O)cc1SC 40244,C1(O)(C(N2C(CNC(c3cc(CC)nn3C)=O)COCC2)=O)CC2CCC1C2 40245,N1(C(CCC)=O)CCCN(C(c2cc(C)n(C3CCCOC3)c2C)=O)CC1CO 40246,C(=O)(CCCCc1ccc(C)cc1)NCC(CNC(CCc1cc(C)[nH]n1)=O)F 40247,C(CC1CCC1)(C(=O)NOCCO)NC(c1c(CC)csc1)=O 40248,C12CCN(CC1C)C(=O)C(=O)c1cnn(c1)CC(=O)N2CC=C.C(C)(C)(C)O 40249,Cc1cc(N2Cc3nc(C#N)n(C)c3C2)nc(=NCCCc2c(C)noc2C)[nH]1 40250,N1(C(c2c(C)nco2)=O)CCC2(CC(NC(=O)C(F)(F)c3ccnn3C)CO2)C1 40251,c1(C(CC)N(C)C)nnc(CNC2C(OCC)CC2)n1CC 40252,C#CCCCCC(=O)N1CCCC(C)(CNC(=O)C(CCC)OC)C1 40253,C1(C(N2C(C#C)CCC2)=O)CN(C(=O)Cc2cnnn2C)CCC1(C)C 40254,N1(C(c2cc(OC)n(C)n2)=O)CC2CC(NC(=O)C(O)C3CCCC3)CC1C2 40255,c1(-c2ccc(COC(C3(C)CCCN(C)C3)=O)s2)cc(=O)c2ccccc2o1 40256,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC1CN(C(c2c(Cl)cnn2C)=O)C1 40257,C(=O)(CC(O)CC(C)C)N1CCCC(CCNC(CC=C)=O)C1 40258,CC1CN(C(=O)CCNC(=O)C2CC2)CC1NC(C1OCCO1)=O 40259,CC1CC(C(=O)N2CCN2)CC(C)C1.c1(Cc2nc(C3CC3)n[nH]2)ccccc1 40260,N1(C(C(c2cnn(C)c2)C)=O)CCC(C2(NC(=O)Cc3cc(Cl)n(C)n3)CC2)C1 40261,C1(NC(C(C)OC)=O)CCC(NC(=O)Cc2cnn(C)c2C)CC1 40262,c1(C(=O)NC(CC(C)NC(CCN(C)CC)=O)C)cccc(Cl)c1C 40263,N(C)(S(=O)(=O)N(C)C)CC(=O)NCC(=O)NC1CC(n2cc(CC(C)C)nn2)C1 40264,C1(C(=O)NCC2(OC)CN(C(c3cocc3C(N)=O)=O)C2)CCC(C)(C(C)C)C1 40265,C=C(C)CC(C(=O)NC(C)CCNC(=O)COC)OC 40266,C1(C#N)(CSCc2n(C)ccn2)C(C#N)C1(C)C 40267,N1(C(c2n(C)ccc2)=O)CCOC(CNC(c2cn(C)nc2-c2ccoc2)=O)C1 40268,c1(OC(C(=O)NCCNC(C2N(C(C(C)=CC)=O)CSC2)=O)C)ccc(C)cc1 40269,N1(C(c2cc(CC)oc2C)=O)CCCN(C(=O)Cn2ccc(O)nc2=O)C(C)C1 40270,c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)C2)cc(F)c(N)c(F)c1 40271,c1(OC)cc(NC(c2cccc(N3CCNC(=O)C3)c2)=O)ccc1O 40272,N1(C(c2c(SC)cccn2)=O)CCCC12CCN(C(=O)C(C)c1ccco1)C2 40273,c1(CC(=O)NC(C2N(C(C(C(C)C)OC)=O)CCCC2)C)cc(F)ccc1Cl 40274,c1(CC(C(=O)NC(CC)CNC(=O)CCF)(C)C)ccc([N+](=O)[O-])cc1 40275,N1(C(c2c(COC)cc[nH]2)=O)CC(CNC(C2CSC2)=O)CC1(C)C 40276,Cc1nc(C(=O)NC2CCN(C(C3CC(N4CCCC4)C3)=O)CC2C)ccc1C#N 40277,Cc1occ(-c2nn[nH]n2)c1C(F)(F)F.C12(CCCC1)CC(=O)N2 40278,CCCC(C(=O)N(C)C)NC(=O)CCn1cc(CCCC(C)=O)nn1 40279,C1(C(N(C)Cc2c(OC)nsc2)=O)CCOC(c2cccc(F)c2)C1 40280,C(=O)(C=CCN(CC)CC)NCC(=O)NCC 40281,N1(C(CN2CCC(C)C2)=O)CCC2(CCCC2NC(C2C3CNC(=O)C23)=O)CC1 40282,C1(CNC(C2CC(OC)C(OC)C2)=O)CCCN(C(=O)Cc2coc(C)n2)CC1 40283,c1(C(=O)NC(CC)CNC(C2C=CCS2)=O)nnn(-c2cccc(Cl)c2)c1C 40284,C1(C(=O)NC2CCCCN(C(c3cnn(CC)c3C)=O)C2)CNC(=O)CC1(C)C 40285,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NCCc1cncs1 40286,C1(C2CCN(C(=O)CC3C=CCC3)CC2)(NC(=O)CC2CC3COCC(C2)C3)CC1 40287,C(=O)(C(C)(C)CCF)N1CCCC(N2CCN(C(C(C)Cc3cnc[nH]3)=O)CC2)C1 40288,c1(C(=O)NCC(C(C(C)C)C)NC(c2ccc(Cl)s2)=O)noc2c1CCCC2 40289,CC1(C)CCC(C(N2CC=CC2CNC(C2(C(F)F)CC2)=O)=O)C1 40290,N1(C(=O)Cn2ncnn2)CCC(C2CCN(C(C3(F)CCCCC3(F)F)=O)CC2)C1 40291,C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C=C(C)C(C)C)C1C 40292,C1(O)(CN(C(C(C)N2CCC2)=O)C)CCN(C(c2ccc(C#N)cc2)=O)CC1 40293,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40294,Cc1c(Br)cnc(O)c1C(=O)NC(C1(O)CN(C(=O)C=CC2CC2)C1)C 40295,C(C(=O)N1CC(O)C(O)CO1)C1(C)CCN(C(C(CO)OC)=O)CC1 40296,C1(C(=O)NC2C(OC)CN(N3CCC(CC=O)C3)C2)CCC(C)(O)CC1 40297,C1(C(N2CCCC(N(C(=O)COC3(C)CCCC3)C)C2)=O)CC12CC(F)(F)C2 40298,C1(C)(C(=O)NC2CC(OCC(N3CC(C(CC)CC)C3)=O)C2)CCC(=O)CC1 40299,C(=O)(C(C)CC(C)(C)C)N1CCC(N(C(Cn2ncc(CC)c2)=O)C)C1 40300,c1(NC2C(CN(C)C)C2)ncc(S(=O)(=O)NCCC2CC(Cl)(Cl)C2)cc1Cl 40301,CCCCCCC(C)C(=O)N(C)CC1CCCN1C(C1CCCCN1C)=O 40302,N1(CC(=O)NCC(C)N(C(=O)Cc2ccnn2C)C)CCCCCCC1=O 40303,C(=O)(C1=CCOCC1)N1CCC(C(=O)NCC2(O)CCN(C)C2)(CF)C1 40304,Cc1cc(NC(=O)CC2CCN(C(c3ccc(Br)cc3)=O)C2)ncn1 40305,C(c1ccncn1)=CC(=O)NC(CN(C(C1(CC=C)CCC1)=O)C)(C)C 40306,Cc1cccc([N+](=O)[O-])c1C(=O)N(C1CN(C(=O)CC2OCCOC2(C)C)C1)C 40307,c1(-c2nnc(OCc3onc(CC)n3)n2N)c[nH]c2ccccc12 40308,C(=O)(CS(=O)C(F)(F)F)NC1C(CO)CCN(C(CCNC(C)=O)=O)C1 40309,CC1CCc2ncc(C(N3CCC(CNC(=O)C(N)=O)C34CCC4)=O)n2C1 40310,N1(CC(=O)NC(C)C)CCCNS1(=O)=O.C(=O)(C(C)N(C)C)N(CC(C)N)C 40311,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CC3C=CC2C3)=O)CC1 40312,N1(C(CCC)C)CCN(c2ccnc(NC3CCCN3C)n2)CC1 40313,N1(C(c2cc(-c3cccs3)on2)C(=O)NCCSC)CC(CCO)OC(C)C1 40314,N1(C(Cc2c(N)nccc2)=O)CCC=C(CNC(=O)CCN2CCCC2)C1 40315,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40316,c1(C(N2CC(C#N)OCC2)=O)cc(-c2cccc(OC(F)F)c2)c2[nH]ccc2c1 40317,C[S+](C)CCC(O)C(=O)N1CC(O)(CNC(=O)COC2CCOC2)C1 40318,c1(C(=O)NC2C(NC(=O)CN3CCCCC3=O)CC2)cc(SC2CC2)nc(O)c1 40319,c1(C(C(=O)NC)N(C2CCC(F)(F)CC2)C)ccc2c(c1F)CCC2 40320,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40321,c1(C(=O)NC(CCNC(C(C(=C)C)(C)O)=O)C)ccc2c(C)nn(C)c2n1 40322,N1(C(C(c2cn3ccccc3n2)C)=O)CC2CN(CC(=O)NC3CC3)CC2C1 40323,c1(N2CC3OCCN(CCOC)C3C2)cc(C)c(S(=O)(=O)NCCSC(C)C)cn1 40324,C12(NC(=O)Cc3ccccc3Cl)CCN(C(=O)CCN3CCOCC3)CC1C2 40325,Cc1ccc(C(C)N(c2nnc(N3CCOCC3)n2Cc2cccs2)C)cn1 40326,c1(OCC)cncc(C(=O)NC(C2CN(C(c3coc(Cl)c3)=O)CCO2)C)c1 40327,N1(C(Cc2c(C)occ2)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40328,N1(C(COCC#C)=O)CCC(NC(=O)CCc2ccc[nH]2)C1C1CC1 40329,c1(OC)cc(N)ccc1C(=O)NCCN1CCC(NC(=O)C=CCO)CC1 40330,C1(N(C(c2n(C)ncc2Br)C(=O)NC2CC(F)(F)C2)C)CCCC(C)(C)C1 40331,C(N=c1ccc([N+](=O)[O-])c[nH]1)C1C(OCC)CC(=O)N1 40332,c1(C(N(C)CCNC(=O)C(C)(C)COC2CCCC2)=O)cccc2nsnc12 40333,c1(C(N2CC(O)(C3(C4(C#C)COC4)CC3)C2)=O)cc(F)c(C)c(F)c1 40334,c1(C(N2CCC(NC(c3cc(C#N)sc3)=O)CC2)=O)cc(S(N)(=O)=O)ccn1 40335,N#Cc1cc(NC(C2(CNCc3cc([N+](=O)[O-])ccc3Br)CC2)=O)c(Br)cc1F 40336,C1(NC(C2CC(C)(C)OCC2)=O)CCC2CCN(C(=O)CC3CCCCO3)C1C2 40337,c1(C(N2CC(Sc3ccc(C)o3)C2)=O)nccnc1-c1ccccc1 40338,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40339,Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC2CC(C1)N(Cc1ccccc1Cl)C2 40340,C1(CNC(c2scc(C)c2)=O)CC(NC(C2CN(C(N)=O)C2)=O)C12CCC2 40341,C(=O)(C(O)CCNC(C1COCC(C)O1)=O)NC(c1nnc(C)s1)C 40342,C1(CNC(CCCOCC=C)=O)N(C(=O)C(C)SC)CCCC1(C)C 40343,C(=O)(CCCn1cncn1)N(C1CCN(C(=O)C(C)Cc2ccccc2)C1)CC 40344,c1(CC)nc(C)[nH]c1C(=O)NC1CC(C(F)C(=O)NCc2[nH]cnc2C)C1 40345,CC1(NC(=O)COC2CCOC2)CCCN(C(c2c(Cl)nsc2Cl)=O)C1 40346,c1(CC(=O)NCC2(CNC(=O)CC3OCCO3)CC2)ccc(Cl)s1 40347,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1(C#N)CC1)=O)CC2 40348,N1(c2cc(NCCCc3cncnc3)nc(C(C)C)n2)CCCCNC(=O)CC1 40349,CC(C)(C)C(CC(=O)NCCC1CCN(C(=O)CN2C(=O)CNC2=O)C1)C(F)F 40350,c1(C(=O)NCC2CCC(NC(C3(C)CCC3)=O)C2)ccc(CCF)cc1 40351,CN1CCOCC1C(N1CC(C(N2CCC3CCC23)=O)C(F)C1)=O 40352,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40353,c1(C(=O)NC2C=CCC2)cc(S(=O)(=O)N(C)C)cn1C.C12(CC1)CN(C)C2 40354,C(=O)(C1=NOC2(CCN(C(=O)Cc3cccnc3)C2)C1)NCc1cccc(C#N)n1 40355,N1(C(COCCOCC)=O)CCC2(CCCCN(C(c3coc(CC)n3)=O)C2)C1 40356,C12(CNC(CCC=CC)=O)CCCC(CN(C(c3cccc4[nH]ccc34)=O)C1)C2 40357,Cc1cc(N(C2CN(C(c3c[nH]c(C(N)=O)c3)=O)C2)C)no1 40358,c1(N2CC(NC(C3CCC4CC34)=O)(CO)C2)ncncc1Br 40359,N1(C(C2C(C)(C)CC2)=O)CCCCC1C1CCN(C(c2cc(Br)no2)=O)CC1 40360,N1(C(c2cc(OC)n[nH]2)=O)CCCC(C(C)NC(c2sc(N(C)C)nc2C)=O)C1 40361,N1(C(C(C2CCN(C(=O)C(N3CCOCC3)C)C2)C)=O)CCC(O)C(C)C1 40362,C1(C(N2CCC3CN(C(c4cnns4)=O)C3C2)=O)CC12CCS(=O)(=O)CC2 40363,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(N)=O)CO3)C2)=O)c1C#N 40364,C1(C(=O)NCC2(CN(C(c3cnn(C(C)C)n3)=O)C)CC2)CCC(C)(C(N)=O)C1 40365,CC(c1ccccc1)=CC(=O)NCC1CCC1NC(C1CC12CC2)=O 40366,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CSC3CC3)CCCC12 40367,C1(CC(=O)NC2(CF)CCCC2)C2CCC(C2)N1C(C1C=CCCC1)=O 40368,c1(C(CCCOC)NC(=O)C(C2CCC2)OC)c(OC)ccnc1F 40369,N12CCN1CC(O)CCC2.C1(C=O)CSCCN1S(=O)(=O)Cc1ccc(F)cc1 40370,c1(C(N2CC(CNC(C3C(C)CN(C)C3)=O)C2)=O)cnc2ccnn2c1 40371,N1(C(C(C=C)C)=O)CCC2(CNC(c3cccc(C)c3O)=O)CCCC12 40372,Cc1ccsc1C(=O)N(CCC(=O)NC(C)(C)CO)C 40373,C(=O)(CCCS(=O)(=O)N1CCCC1)NCC1CC1NC.C#CCCN1CC(=O)O1 40374,c1(OC)cccc(Cl)c1C(=O)NC1CCN(C(C2(C(C)C)CC2)=O)C(C)C1 40375,c1(NC(COCC(=O)NCC(CNC(=O)OC)(C)C)=O)ccnc(O)c1 40376,N1(C(=O)C2=NOCC2)CC2CCCC1CN(C(c1ccc3nc(O)[nH]c3c1)=O)C2 40377,C(=O)(CCCC(C)(C)C)NCc1occ(C(=O)NC(CC(C)C)C(N)=O)n1 40378,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(c2cc(Cl)c[nH]2)=O)CC1 40379,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)(C)C)nc2C)=O)C1)NC(C)=O 40380,N1(C(C(CO)OC)=O)CCC(C(=O)Nc2cnc(CC3CC3)nc2)=C(F)C1 40381,O=C(C1=CC2CCCC12)NCC1CC(NC(c2ncnc(O)c2Br)=O)C1 40382,CCC(C)C(C(=O)N1CCNC(=O)CC1)N(C(=O)C(C)N1CCCC1)C 40383,CCC(C(=O)OC)C(=O)N1CC(NC(=O)CCNC(N)=O)C2CC2C1 40384,C#CC1(C(=O)NCCN2CCOC(C)C2)CCN(C(=O)C(=O)C2CCCC2)CC1 40385,c1(CC2(C(=O)N(c3nnnn3C(C)C)C)CCC2)ccc(F)c(Cl)c1.CN 40386,c1(C(=O)NC(C2CN(C(c3ccc(CO)cn3)=O)CCO2)C)cnc(F)c(F)c1 40387,Cc1[nH][nH]c(=N)c1C(=O)N(C)CC1(O)CCN(C(=O)CCC2CNC(=O)N2)C1 40388,C1(C(=O)NCCOC(CC)(C)C)CCN(C(=O)COC(C2CCC2)=O)CC1(C)C 40389,c12ncnc3c1ncn3C1CC(C(=O)N=c3cc(C)[nH][nH]3)N2C1.CCOC 40390,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40391,C1(C(=O)NC2(CSC)CCC2)CCCN(C(=O)C(C)SCC(C)C)C1C 40392,N1(C(C)C(=O)N(CCCNC(=O)Cn2nnnc2C2CC2)C2CC2)CCC(O)CC1 40393,N1(C(CS(CCC)=O)=O)CCC2(CCOCC2)C(NC(c2cnn(C)c2F)=O)C1 40394,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40395,c1(C(C)C)cc(C(N2CCOCC2CNC(C2(CO)CC2)=O)=O)ccc1F 40396,c1(CC)cc2oc1=2.C(CC(F)(F)F)SCC(=O)N(C1CC(NC=O)C1)CC 40397,c1(C(=O)NCC(CC)NC(c2cnn(C(C)C)c2C)=O)cccc(F)c1OC 40398,C(=O)(C1=CC2CCC=CCCC12)N1CC(C(C)NC(c2cn(C)c(=O)n2C)=O)C1 40399,C1(NC(=O)C(O)C(F)(F)F)CN(C(=O)CCNC(c2ccncc2)=O)CC2(CC2)C1 40400,C1(NC(C(c2ccc(Cl)cc2)C)=O)(CNC(=O)COCCF)CC2CCC1CC2 40401,C=C(F)C1(CCNC(=O)CCC(=O)NC2CCCN2C(=O)COC)CCOCC1 40402,c1(C(N2CCN(C(CNC(CCC)=O)C)CC2)=O)c2n(c(=O)n1C)CCCC2 40403,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CN(Cc2c(Cl)cc(F)cc2Br)C1 40404,C(=O)(C1=C(C)CCOC1)NC(CC#C)CC(=O)NCC(O)C(C)O 40405,C1(C(N(C)Cc2cncs2)=O)CCCN1NC(=O)c1cn2ccccc2n1 40406,N1(C(c2cc(C)on2)=O)CCN(C(=O)CC(C)(C)O)C2CCCCC2CC1 40407,c1(C(=O)NC2C(CNC(c3n[nH]c(=N)s3)=O)C2)cc2n(n1)CCC2 40408,c1(CC(N2C(CNC(c3cnc(O)s3)=O)CCCC2)=O)cccc(F)c1O 40409,c1(CC(=O)NCC(C)NC(=O)CC2COCC2(C)C)c(F)c(F)cc(F)c1F 40410,Cc1ncc(Br)c(N2CC(CC(C)NC(C3C(c4ccccc4)C3C)=O)C2)n1 40411,CC1CCN(C(=O)C=CC=C(Cl)Cl)CCN1C(C1CC(=O)NC(=O)C1)=O 40412,C1(C)(NC(C2(OC)CCCOC2)=O)CCN(C(=O)C(=Cc2cn(C)nn2)F)CC1 40413,C1(C(N2C(CCNC(=O)Cc3ncc(Cl)s3)COCC2)=O)CC2CCC(C1)C2 40414,C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)Cc2ccc(F)cn2)CC1C(F)(F)F 40415,Cc1cnnc(O)c1C(N1CC(CCNC(C2CC2CN2CCOCC2)=O)C1)=O 40416,C#CC1CC2(CC2)CN1C(C1CCN(C(C2(SC)CC2)=O)CC1)=O 40417,c1(C(=O)NCC(=C)CCNC(c2cnoc2)=O)nn(C)cc1SC 40418,C(=O)(C(Cc1cnc[nH]1)NC(=O)COC1CC=CC1)NC(C(C)SC)C 40419,c1(OC)cccc2c1OCCC2NC(c1nnnn1C)(C1CCOC1)C 40420,N1(C(c2c(C)cncn2)=O)CCC(O)C(N(C(=O)CCOCCN(C)C)C)C1 40421,N1(C(c2nc(OC)oc2)=O)CC2=C(C1)CN(C(=O)CC1COCC3(CCC3)O1)C2 40422,C(=O)(C1CC(C)S(=O)(=O)c2ccccc21)N(CCNC(c1c(CC)con1)=O)C 40423,C1(N(C(=O)CCCc2ccsc2)CC)CCN(C(=O)C=Cc2nnn(C)n2)CC1 40424,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40425,N1(C(Cc2c(C)n[nH]c2)=O)CCCC(N(C(=O)CCc2c(C)n[nH]c2C)CCO)C1 40426,N1(C(CC(CC#C)N(C(=O)C(CC2CC2)OC)CC)=O)CC(C)CCC(C)C1 40427,CN1CCOCC1CC(=O)NC1(CNC(=O)Cn2ccc(=N)[nH]2)CCCCC1 40428,N1(C(C(=O)NCC)=O)C(C(=O)NCCCc2nc[nH]n2)CC2CC12 40429,c1(OCC(=O)Nc2c(C(=O)OCC)cncn2)cc(C)ccc1C(C)C 40430,c1(NC2(CNC(C3(C)CC(C)OCC3)=O)CCCC2)ncc2c(ncn2C)n1 40431,C1(c2c(O)ccc(CC(=O)O)c2)SC(=Nc2ccccc2)NC1=O 40432,N1(C(C(C)N(C(c2ccn(CC)n2)=O)C2CC2)=O)CCC(C)(COC)CC1 40433,CC1(OCC(=O)NC2(N(C(=O)CCOC3COC3)C3CC3)CCC2)CCOCC1 40434,c1(C(N(CCCCCCNC(C(C)=C(C)C)=O)C)=O)cc(=O)n(C)cc1Br 40435,CCC(CC(=O)N(C(C)C(=O)NC1(CC)CCCCC1)CC)OC 40436,C1(C(=O)NC2(c3ccc(CC#N)cc3)CCCC2)CCc2nc(O)nc(O)c2C1 40437,C1(CC(=O)NC(CN(C(COCC#C)=O)C)(C)C)CCC(=O)N1CC 40438,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(CCCC)n2)=O)C1 40439,Cc1ccsc1CN1CCC(C(=O)NCC2SCCS2)C1 40440,C=CCC(C)(C)CCN=c1cccc(S(=O)(=O)N2CC(C)c3cccnc32)[nH]1 40441,C1(CN(CC(C2CCCC23CC3)=O)C)CCCCN1C(c1ccccc1F)=O 40442,N1(C(=O)Cc2ccc(F)c(F)c2)CCC2(CCCN2C(=O)C2=CCCCCC2)C1 40443,c1(NC(c2c(NC(C(CC)CC)=O)cnc(F)c2)=O)cc(F)c(C#N)cc1F 40444,N1(C(=O)NCC)CC2C(C(=O)OCc3ccccc3Cl)C2C1 40445,C1(C(N2C(CCNC(C(C)(Cl)Cl)=O)CCCC2)=O)CCC2CCC1O2 40446,CCC(O)C(F)(F)C(=O)N1CC2C(C1)N2C(C1CCCCC1)=O 40447,C(=O)(CCC(F)(F)C(F)F)N1CCC(OCCNC(C2CCCO2)=O)C1 40448,N1(C(c2c(CC)noc2)=O)CCC(C)(C)C1CNC(c1nccc(OC)c1F)=O 40449,c1(OC)cc(Cl)c(C(N2CCCN(C(C)=O)CC2)C(=O)NC(C)C)cc1OC 40450,c1(C(=O)NC(CCO)C2CC2)ccc(Cl)cc1.n1(CCCSC)nnnc1C1CN1 40451,C1(NC(c2ncn(CCNC(C(C3CC3)OC)=O)c2)=O)CCC(C)(C)C1 40452,C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(C(COC)(F)F)=O)CC1CC2 40453,N1(C(c2cn(C)nn2)=O)CCC2CC2(C(=O)NC2CCCC2F)CC1 40454,c1(NC(C)=O)ccc(CC(=O)N(C2C3CN(C(=O)C(F)=C(C)C)CC23)C)cc1 40455,C1(CNC(Cn2ccc(C)n2)=O)CC12CCN(C(c1cnc(N)c(O)c1)=O)CC2 40456,Cn1nnc(Cn2nnnc2C(C2CC2(Cl)Cl)NCc2nc(C(F)F)n[nH]2)n1 40457,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nccn2C1 40458,n1(CC)c(C(N2CCC(C)(NC(=O)C(F)CC(C)C)C2)=O)nc2ccccc12 40459,c1(C(N2CC(CNC(CC(CC)C)=O)C3(C2)CC3)=O)cnc2c(c1)nnn2C 40460,N1(C(C(C=C)O)=O)CC(NC(C2CC3(C2)CC(F)C3)=O)CC2(CCC2)C1 40461,c1(N2CC(CCOc3c(OC)c(C)cc(C=O)c3)C2)cccc2cn(C)nc12 40462,C1(CC=C)(NC(=O)Cc2c[nH]nc2C)CCN(C(=O)C(C)(C)COC(C)(C)C)C1 40463,S(=O)(=O)(c1ccc(=NCC(C)(COCC(CC)CO)SC)[nH]c1)CN 40464,c1(OC)ccc(NCCCC(=O)NCC2(C(=O)NCc3cc[nH]n3)CCC2)cc1 40465,CC1CCC=C1C(=O)N1CCC(OCCNC(=O)C(C)c2cccs2)CC1 40466,C(C1CCCN1C(=O)CN1CCCCC1C)=CC(=O)NCc1nc(C)oc1 40467,c1(OC)ccc(F)cc1CC(=O)NC1C2CC1N(C(C1CC1C(F)(F)F)=O)C2 40468,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(F)F)c1 40469,C1(C(N2C(COC)CCCC2)=O)CN(C(=O)C(C)c2cc[nH]n2)CC1(C)C 40470,c1(NC(C2CC(NC(Cc3ccc(NC(C)=O)nc3)=O)C2)=O)cc(C)ccc1F 40471,CN1CCN(C(c2ccccn2)=O)C(C(=O)N(C2CCN(C)CC2)C)C1 40472,N1(C(CC(CC)C)=O)CCCCCC(NC(c2c(C)noc2C(F)(F)Cl)=O)C1 40473,c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)CC2C)cc2c(nc1O)CCC2 40474,Cc1cc(F)c(Cl)cc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C 40475,C1(NC(C2C(C)C2)=O)C2CN(C(c3cc(-c4ccccc4)n(C)n3)=O)CC12 40476,C(=O)(CC1=CCCCC1)N(C)CC1CCCN(C(CCCN(C(C)=O)C)=O)C1 40477,c1(C(C(=O)NCCCCNC(c2n(COC)ncc2)=O)C)ccc(Cl)c(Cl)c1 40478,CCC(C(=O)NCC1(O)CN(C(C2(F)CC2)=O)C1)OCC(C)C 40479,C1(NC(C=C(CNC(CC(=O)NCC)=O)C)=O)CCC(COC)CC1 40480,c1(C(=O)NCc2c(C(N3CCC(C(=O)NC)CC3)=O)nco2)ncccc1F 40481,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40482,C(CCNC(C1CCC(O)CN1C)=O)(C(C)(C)C)NC(C1N(CC)CCCC1)=O 40483,c1(C(N(C2CCN(C(c3cnc(C)n3C)=O)CC2)C)=O)cnc(C2CC2)nc1C 40484,CC(C)CC(C)(C)C(=O)NCC(CO)NC(=O)COC1CCC(C)CC1 40485,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40486,C(=O)(C1=CCC(C)CC1)N(CC(C)(C)CNC(C1CC(O)C(F)C1)=O)CC 40487,c1(CNC(CC2(C)CNC2=O)=O)cccc(Cl)c1Cl 40488,C(C)(C)(C(C)NC(=O)C(C)=C1CC1)NC(C1(CC)CCC1)=O 40489,C(=O)(C(C)C(O)C(C)C)N1C(C(=O)NC(CC#C)C)CSC1 40490,C1(C(=O)NC(CNC(CN(CCC)C)=O)(C)C2CCC2)CC=CCC1 40491,C1(C)(COC)CCN(C(=O)C(C2(O)CN(C(c3[nH]nnc3C)=O)C2)F)C1 40492,c1(C(N2CCOCC(NC(C(N)=O)=O)C2)=O)ccc(=O)n2c1COCC2 40493,c1(NC(C2CCCN(C(C)=O)C2)=O)cc2nscc2cc1Br 40494,CCC1CCC(=O)NCCOCCO1.C(=O)(CC)N(C)CC.C(C(F)F)O 40495,C(=O)(C(C)(F)C(C)(C)F)NCC1(NC(CCc2cccc(OC)c2)=O)CC1 40496,C1(C(=O)NC(C)(C)CC2CCC2)CC2CCC1N2C(=O)CCCn1cccn1 40497,c1(CN(CCOCC)C)cc2c(cc1O)CCCC2 40498,C(Cn1cccn1)(C(=O)NC(C(=O)OCC)C1CC1)NC(COCC#C)=O 40499,N1(C(=O)Cc2ccc(C(F)(F)F)s2)CCC(CO)CC1CNC(C1CC12CCC2)=O 40500,C1(NC(c2c(N(C)C)cnnc2)=O)CC(O)CN(C(c2cccc(F)c2Cl)=O)C1 40501,C1(N(C(Cc2cn(C(=O)NC)nn2)=O)CC2CC2)C2CCCC1CC2.C1C(=O)N1 40502,CC1=C(C)CC(C(=O)N(C(C)(C)CC(N2CC(CO)CC(C)C2)=O)C)CC1 40503,c1(C(C)NC(C2OCCC2NC(C2(C)CCCC2C)=O)=O)ccccc1O 40504,C1(C(=O)NCCC=C=C)CCN(C(C2OCCOC2C)=O)CC1(C)C 40505,C=CC(C)(CCOC)C(=O)NCc1ccc(C(=O)NC2CCC(C)(C)CC2)cn1 40506,C1(C(N2CC(C)N(C(c3ccoc3Cl)=O)CC2)=O)COc2cc(Cl)ccc2C1 40507,CC1(NC(=O)COC)CC2(CCC2)C1.c1(OCCN)nc(O)nc(O)n1 40508,C1(C(=O)NCCN(C)C(c2cnns2)=O)C2Cc3c(Cl)cccc3C12 40509,c1(N(C)CC2CCCNCC2)nc2c(F)cc(C(F)(F)F)cc2s1 40510,C1(NC(C(C2CCCOC2)OC)=O)(CNC(C2(CF)CC2)=O)CC2CCC1CC2 40511,c1(C(N2CCCC(N(C(c3ccccc3F)C)C)C2)=O)cccn2nccc12 40512,c1(C(C)(C)C)ccc(NC(=O)CC2COCCN2Cc2ccnc(F)c2)cc1 40513,c1(C(N2CCCN(C(C3(C)CCC(OC)C3)=O)CC2)=O)cccc2c1CCO2 40514,N1(C(C(C2CC=CCC2)NC(c2ccc(F)cc2)=O)=O)CCN2CCC1CC2 40515,C(=O)(C(C)(C)C(C)NC(=O)CC1CC2(CC2)C1)N(CCCCC)CCO 40516,C1(CC2CC2C(N2CC(NC(C(C)Sc3ccccc3)=O)C2)=O)CCS1(=O)=O 40517,C12(CNC(c3ccn(CCOC)n3)=O)CCC(CC1)N2C(C1(F)CCCCC1)=O 40518,C1(C2CCC(=O)NC2)(C(=O)NC(C2CCN(C(=O)C#CC3CCC3)C2)C)CCC1 40519,C1(N(C(C(c2cc(C)sc2)(F)F)=O)C)CN(C(c2n[nH]c(C)c2C)=O)CC1F 40520,C1(CC)(NC(c2cc(C(=O)NC)c[nH]2)=O)CCN(C(c2ccc(F)s2)=O)CC1 40521,c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 40522,Cc1ncc(C(=O)NC(C(=O)N(CCC#N)C)c2nccs2)s1 40523,C1(C(N2C(C)(CNC(C3(CSC)CCC3)=O)CCC2)=O)CCC(F)(F)C1O 40524,c1(CC(=O)NCC(C)OCC(=O)NCC2CCCCO2)ccc(Br)cc1Cl 40525,CC#CCCC(=O)N1CCC(N2CCN(C(c3cnn(C)c3N)=O)CC2)CC1 40526,N1(C(C(C)C2CCOC2)=O)CCC2CCC(C1)N2C(c1cc(Br)cs1)=O 40527,c1(C(=O)NCC2CCC2C(=O)NC2CCCC2(F)F)ccnc2cc[nH]c12 40528,c1(C(F)F)cccc(OC(F)F)c1.c1(CN2CCC2)nnnn1C1CCOCC1 40529,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40530,C(C)(N=c1[nH]c(=N)[nH]c(=NCc2ncn(C(C)C)n2)[nH]1)c1nnc(C)s1 40531,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NCCC2(C)CC2)CC2CCC1C(O)C2 40532,CCCCC(C)CCC(=O)N(CCCN(C)C(c1cccn2c(O)nnc12)=O)C 40533,c1(N(C(C)=O)CCC(C)N(C(CCNC(C)=O)=O)C)c(Br)ccc2n[nH]cc12 40534,C1(=O)CC(C)NC(=O)OCC(C)NC(=O)C2(F)CC2N1.C(C)(C)(C)OC 40535,C1(C(=O)OCC)CC(C(=O)OC)CN(c2ccnc(O)c2)C1 40536,O=C(C1=C2CCCN=C2NN1)Nc1ccc2c(c1)CNC2=O.N12CC3C(C3C1)C2 40537,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(=O)CCc1cnn[nH]1)CC2 40538,C(=O)(CCC(=O)NC1CCC(F)(CNC(c2ccsc2C(F)F)=O)C1)NC 40539,C1(n2cccn2)(C(=O)NCC(C)N(C(=O)Cn2ccnn2)C)CCCC1 40540,c1(NC)snc(C)c1C(N1CC(CNC(c2cn(CC(N)=O)nn2)=O)C(O)C1)=O 40541,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40542,CC1CN(C(=O)CCCC(N)=O)CCCN1C(c1cncc(C(F)(F)F)n1)=O 40543,C1(NC(C2C(CC)CCN2C(=O)C(N2CCCCC2)C)=O)CCCCCC1C 40544,C1(C(=O)NC2C(NC(c3c(CCC)n[nH]c3)=O)CCC2)C(F)(F)C12CC2 40545,C1(CC(=O)OCC(c2c(OC(C)C)occ2C(F)(F)F)=O)CC(C)(C)OC(C)(C)C1 40546,C1(N(C(CCCCOC)=O)C)CCC2CN(C(=O)Cn3nnc(=N)[nH]3)CC12 40547,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40548,C=C(F)C1(CC(=O)NCC2(C(=O)NCC3=NOC(C)C3)CC2)CCC1 40549,CC1(C)COC(CC(=O)NC2(C3CCCCN3C(=O)CCn3cccn3)CC2)C1 40550,C1(CC)(NC(=O)C(C)SC(F)(F)F)CCN(C(=O)C(CO)NC(N)=O)CC1 40551,c1(C(c2n(CC)nnn2)NC2CN(c3nncs3)C2)cc(C)nnc1C 40552,C1(CNC(CCc2ccc(NC(C)=O)cc2)=O)CCCN(C(=O)C(F)C(C)C)CC1 40553,N1(C(CC(CC)C)=O)CC2CC(NC(c3cnc(C(C)C)[nH]3)=O)C1C2 40554,C1(C(=O)NCC(C(C)(C)C)NC(CN2CCN(CC)CC2)=O)CCC2CC2CC1 40555,C(C(C)C(=O)NCC1CCC(NC(c2c[nH]nc2C2CCOCC2)=O)C1)OCC 40556,C#Cc1cn(C)nc1C(=O)N(C1CCN(C(=O)C2=C(C)CCC2)CC1)CCO 40557,c1(C2C(C(C(=O)OC)OC3CCCCCC3)C2)ccc(C)c(C)c1 40558,CC(C)C(CCNC(C1(CO)CCCCC1)=O)NC(=O)CCC1CCOCC1 40559,N1(C(C(CCC)OCC)=O)CC(CNC(c2cn(C)cn2)=O)OC2(CCC2)C1 40560,CC(C)(C)C1=CCN(C(C2CCN(C(c3cc[nH]n3)=O)C2)=O)CC1 40561,c1(CCC(=O)NC2CC(NC(=O)C(F)(F)C3CC3)C(O)C2)n[nH]c2c1CCCC2 40562,N1(C(C(C(C)C)O)=O)CCN(C(=O)CCCCCC#N)CC(CO)C1 40563,C1(NC(C(C2CC(NC(C3(CCC)CC(=O)C3)=O)C2)F)=O)C(O)C2CCOC12 40564,C(=O)(C1=CCC12CCNCC2)NC(CC)(C)CO 40565,c1(OC)ccc(C(N2CCC(CNC(c3cc(F)ccc3N)=O)C2)=O)c(F)c1Cl 40566,c12c(ccn1C)NC2=O.C(C)(C(=O)N(C1CN(C(C)=O)C1)CC1CC1)OC 40567,C1(C(N(CCNC(C(CC)C)=O)CC)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1 40568,c1(C(=O)NCC2(O)CCN(C(C3=NOC(C)C3)=O)C2)ccc2cnsc2c1 40569,N1(C(C2CCN(C(C)=O)C2)=O)CCCC2(NC(C3COCCN3C)=O)CCCC12 40570,c1(C(N(C(CNC(c2ccc(CC)cc2)=O)C)C)=O)cc2oc(Br)cc2[nH]1 40571,C(C)(C)(CN=c1nc(N2CCCN(CC(F)(F)F)CC2)c2c([nH]1)CCC2)N(C)C 40572,CC(COCc1ccccc1)C(=O)NNC(=O)Nc1cn2c(n1)C(C)CCC2 40573,c1(CCCC(=O)N(CC(CC)NC(=O)C(C)=CC(C)(C)C)C)ccc(C#N)cc1 40574,C(=O)(CCCC(C)(C)C#N)NC1C2CC(NC(c3c(OC)ccc(Cl)c3)=O)CC21 40575,N1(C(c2ccc(C#N)o2)=O)C2CCC1CN(C(c1cnc(-c3ccsc3)s1)=O)C2 40576,n1(CC(=O)NCCNC(C(c2ccc(F)cc2)OC)=O)c(=O)oc2ccccc12 40577,N1(C(C2=C(C)OCC2)=O)CC2CN(C(=O)CCc3ncc(C)[nH]3)CC2(C)C1 40578,c1(CC)ncc(C(=O)NCCN(C(c2cc(CC(C)C)[nH]n2)=O)C(C)C)[nH]1 40579,c1(C(N2CC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)ccc(Cl)c2c1OCCO2 40580,c1(C(=O)NCCN(C(C2CN(C)C(=O)N2)=O)C)cccc(C#CCO)c1 40581,N1(C(=O)Cn2cccnc2=O)CCSCC1C(=O)NC(C)C(=O)NC1CC1 40582,CC1CC(NC(C2(CC3CC3)CC3(CCC3)C2)=O)CCN1Cn1ccc(C2CC2)n1 40583,C1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CC2COCC2N1C(=O)CSC1CC1 40584,N1(C(c2csc(Cl)c2)C(=O)NCCC)CCC(C2(C)CC2)CC1 40585,CCCCCCCN(C(c1cc(F)ccn1)c1n(CCC)nnn1)C1CC1.C1CC1 40586,C(CNC(C1(c2ccccc2)CC1F)=O)(CO)(CO)NC(C1C(OC)CCC1)=O 40587,c1(C(N2CCC(N(C(=O)C=C(Cl)Cl)C(C)(C)C)CC2)=O)noc2c1COCC2 40588,C#Cc1cccc(CC(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40589,C1(C)(C(=O)NC(C2CN(C(c3cccs3)=O)C2)C)COC(=O)N1 40590,C1(NC(c2occ(C)c2)=O)CCC(C)N(C(=O)CCc2ccc(F)cc2Cl)C1 40591,C=C(C)C1CCC(C)=CC1CC(=O)NC1CC2C(NC(=O)CCS(C)(=O)=O)C2C1 40592,N1(C(CC(C(=O)OC)C)=O)CCOC2CCN(C(c3ccc(Cl)nc3C)=O)CC12 40593,c1(CC)cc(CC(=O)N(CC(=O)NC2CC(C)(C(N)=O)C2)CC(C)C)no1 40594,n1(CCCN(C(C(C)c2ccco2)=O)C)cc(Cn2ccnc2)nn1 40595,C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCCCN1C(C1COC(=O)N1)=O 40596,C1(NC(c2cnc(C)nc2O)=O)COC2(C1)CN(C(=O)CCC(C)CN(C)C)C2 40597,c1(CCC(=O)NC(C)CNC(=O)Cc2nc[nH]n2)ccncc1Br 40598,C(=O)(C1=COCC1)NCCOCC(=O)N(C)CCOc1ccn(C)n1 40599,c1(C(N(C(C)CN(C)C(c2csc(Cl)c2)=O)C)=O)ccc(F)c(Br)c1 40600,N1(C(CC(C)(C)F)=O)CCC(NC(c2cnn[nH]2)=O)C(CO)C1 40601,C(CNC(C12CC(CCO1)C2)=O)(CC(C)C)NC(C=CC(=O)OCC)=O 40602,N1(C(C2C(C(C)NC(c3cccc(C)n3)=O)C2)=O)C2CCC1CN(C)C2 40603,C1(C(=O)NC2(c3cn(C(CC)C)nn3)CCC2)CCc2ncc(C)n2C1 40604,CN1CCN(C(=O)CN2CCCCC2=O)C(C(N2CCOC(C)(C)C2)=O)C1 40605,C(C1CN=C2C=C(N=CN2)N1)OC.N1(C)CCS(=O)(=O)CC1 40606,C1(NC(CCCOC(C)(C)C)=O)CC2COCC(C1)C2NC(c1cnccn1)=O 40607,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40608,C1(NC(C2CC(CC)C2)=O)CN(C(=O)C(O)C2CCCC2)CC1C 40609,N1(C(C(c2cn(C)nc2)=O)=O)CCCC(CCNC(C2CC(N(C)C)C2)=O)CC1 40610,Cc1cc(C(N2CC(NC(c3nn(C)c(Cl)c3Cl)=O)C(C)C2)=O)cc2nn[nH]c12 40611,c1(C(N2CCCC(N(c3ccno3)C)C2)=O)cc(S(N)(=O)=O)ccc1O 40612,c1(C(=O)NCC2C(NC(CC(C)n3cccc3)=O)CCCC2)n[nH]c2c1CCC2 40613,c1(CC(=O)NC(CN(C(C2C=CC(C(=O)OC)C2)=O)C)C)ccnnc1O 40614,CC1CCOC(C(N2CCC2C(=O)NCc2ncc(CO)o2)=O)C1 40615,CCC(C(=O)NC(C1CCN(Cc2nc(C3CC3)no2)CC1)C)C(C)C 40616,N1(c2cncc(-c3cc(=NC)[nH]cc3)c2)CCCc2cc(C)ccc21 40617,c1(C(CNC(c2cnco2)=O)NC(CCC2CCN(C)C2)=O)cccc(Cl)c1 40618,C1(C(=O)N(CCC(=O)NCCCO)C)(OC)CCC(C)(C)C1 40619,C1(C(=O)NC(CC)CNC(C2(OC)CCCC2)=O)CCCCC1C(C)(C)C 40620,c1(C(=O)NCCCC(C)NC(CCCN(C(C)=O)C)=O)nn(C)nc1C(F)(F)F 40621,C(=O)(C1=NN(C2CC2)C(=O)CC1)NCCC1N(C(CC=C=C)=O)CCCC1 40622,c1(CC2(NC(c3nc(C)c(C)o3)c3n(CCCSC)nnn3)CC2)ccccc1C 40623,C1(OC)CCC12CC(NC(=O)Nc1cn(C3CN(CCCCC(C)CO)C3)nn1)C2 40624,N1(C(CCCC#C)=O)CCCC(O)(CNCC2(CSc3ccccc3)CC2)C1 40625,c1(C(=O)NC2C(NC(=O)C3=NOCC3)CCCCC2)cc2ccc(F)cc2s1 40626,Cc1cc(Oc2cc(NC(=O)C(=O)NC3CC3C)ccc2F)ccc1C(N)=O 40627,N1(C(c2cnn(C)c2C#N)=O)CCC2(CC1)CC(NC(=O)C(F)C1CCCC1)C2 40628,C1(C(=O)NC(C2CCCN(C(=O)CCC3CC3)C2)C)(NC(C)=O)CCCCC1 40629,C(=O)(C1=CCC(C)CC1)N1CCC(C)(CC(NOCCC#C)=O)C1 40630,Cc1ccc2cc(C)nc(N3CCC(C4CCN(C(C)C)C4)C3)c2c1 40631,c1(C(N2CCN(C)CC2CNC(=O)CCCCO)=O)cnc2n1CCOC2 40632,C1(C(=O)N(C)Cc2ncc[nH]2)(COC)CCCN1C(=O)CC(O)CN(C)C 40633,C(C(C(C)(C)C)NC(=O)Cc1ccc(C(F)F)cc1)NC(C(C)OCC)=O 40634,c1(C(=O)NCC2C(NC(c3n(CC)nc(C4CC4)c3)=O)C2)cc2scnc2[nH]1 40635,CN1CCN(C(=O)Cc2cc(O)n(C)n2)C(CNC(C2CCCCC2(F)F)=O)C1 40636,c1(C(=O)NCC=C)oc(CNC(C2(Cl)CC2)=O)nc1C 40637,N1(C(C2CC3(CC(=C)C3)C2)=O)CC2(CCN(C(=O)C=CC3C(C)C3(Cl)Cl)CC2)C1 40638,N1(CCOC)CCN(C(C2(c3cn(C4CCCNC4=O)nn3)CCC2)=O)CC1=O 40639,C#CC1(C(=O)NC(c2nccn2CCC)C)CN(C(c2cc(OC)ncn2)=O)C1 40640,N1(CC(C2(O)CCC2)CC)CCOC(c2n[nH]c(CC3CCC3)n2)C1 40641,c1(CCCNC(c2nnnn2CC(F)F)C(C)C)cccc(F)c1 40642,N1(C(=O)Cc2ncncc2Cl)CCN(C(C2CCCCC2)=O)C2(CCC2)C1 40643,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40644,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40645,N1(C(CC2(NC)COC2)=O)CCC(CNC(=O)CO)C12CC2.c1(C)nc(C)no1 40646,C1(NC(CC2(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2ccc(F)cc2)C1 40647,n1(CC(=O)NC2CN(C(CC3(OC)CCCCC3)=O)CC2C)cc(F)ccc1=O 40648,CC1OC2(C(=O)N(CCCOCCNC(=O)CC(C)C3CC3)C)CCC1CC2 40649,N1(C(c2ccc(CNC(=O)Cn3cncn3)[nH]2)=O)CCN2CCC1C2 40650,CCCC(CCC)CC(=O)N1CCN(C(=O)COCCOC)C(CS(C)(=O)=O)C1 40651,C1(C(=O)NCCNC(C(C(C)C)NC(=O)C(C)(C)C)=O)CCC(C)(C)CO1 40652,C(=O)(C(C)(C#N)CC)NCc1c(CN(C(c2c(CC)nn(C)c2)=O)C)cccc1 40653,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCC(F)F)C2)C1 40654,C(c1cncnc1O)=CC(=O)NCC1(NC(Cc2nn(C)c(Cl)c2)=O)CCOC1 40655,CC(C1CCCCC1)=CC(=O)NC(C)(C)CCNC(c1ccnc(C)c1N)=O 40656,NC(=O)CC(C(=O)N1CCCCC1C1(O)CC1)NC(c1ccc(O)cn1)=O 40657,CCC(C(=O)OC)C(=O)NCC1CCC(C(N2CCC(C(=O)NC)CC2)=O)O1 40658,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C(C)C 40659,N1(C(CC(C)F)=O)CCC(CNC(=O)CNS(C)(=O)=O)C(F)(F)CC1 40660,N1(c2ncc(C(=O)OCC)s2)CCC(C)C(CN(C(c2cnc(C)s2)=O)CC)C1 40661,CC(C)(C)CCCCC(=O)NCc1nc(C(=O)N2CC(O)CCO2)co1 40662,C(C)(C)(C(=O)N(CCCNC(C1(C)CCCC1)=O)CC1CC1F)OC 40663,N1(C(Cc2c(C)cco2)=O)CCCC(C)C1CCNC(C1CCC2(CCC2)C1)=O 40664,CCCC(C)(C)C(=O)N1CC(C(=O)Nc2nnc(CC(C)C)s2)CC(C)C1 40665,O=C(C1CNc2ccccc21)N1CCN(C(=O)Cc2cccc(Cl)c2)C(CO)C1 40666,C=CCC(CC=C)C(=O)NCCNC(N(C(CSCC)=O)CC#CC)CC 40667,CS(=O)(=O)c1coc(C(=O)NCC2CCCN(C(=O)CC3CCCOCC3)C2)c1 40668,Cc1c(CC(=O)NCCOCCN(C(=O)CC2CCC(O)C2)C)ncn1C 40669,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(c2ccc(CO)c(Cl)c2)=O)c1F 40670,CCCCC(CNC(=O)C1=CCCC1)NC(=O)CCc1cnc(C2CCC2)o1 40671,C1(C(N2CC(SCC)C2)=O)C2CC3C(C2NC(=O)C(C)(O)CC)C13 40672,N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)C(C)NC=O)CC1C1CC1 40673,c1(C(N(C(C)CN(C)C(c2n[nH]cc2Br)=O)C)=O)cc2c(cc1O)CCC2 40674,C1(CNC(C2(CNC(CCCN(C)C)=O)CC2)=O)CCOC(C)(C)C1 40675,c1(CC)ccc2occ(CC(=O)NCCNC(c3ccn(CC)c(=O)c3)=O)c2c1 40676,CN1CC(C(N2CC(C3CC3C(=O)NC3(C(O)CO)CC3)C2)=O)CCC1=O 40677,c1(C(N2CC(CC=C)(NC(c3[nH]nnc3C3CC3)=O)C2)=O)c[nH]c(C)c(Cl)c1=O 40678,c1(SC)cc(C(F)(F)F)ccc1F.CCC1C(N)CN1C 40679,c1(C(=O)NCC(CNC(c2nc(C(C)C)oc2)=O)O)cn2c(n1)CCCC2C 40680,c1(CNC(=O)OC(C)(C)C)nnnn1CCSC1CC2CC2C1.CCCO 40681,c1(Cn2cc(CN3CCN(C(CSCCC)=O)CC3)nn2)ccc2ncsc2c1 40682,c1(C(=O)NC(CNC(C=NOC)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 40683,C1(NC(C2(N(C)C)CC2)=O)CCCC(N=c2[nH]c(Cl)nc3ncn(C)c23)C1 40684,C(C1CN(C(c2cnns2)=O)Cc2ccccc21)NC(c1c(C)nccn1)=O 40685,c1(C(C)C)ncc(NC(=O)C(C)NC(=O)CC2CC2C2CC2)cn1 40686,CC(C)(C)C(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(C2CCCC2)=O)C1 40687,N1(C(CSCC(=O)OC)=O)CC(NC(=O)C(C2CCC2)OC)CC2(CCC2)C1 40688,c1(C(N2CCCC(CC(=O)NC3(C)CCCC3)C2)=O)cc(Cl)ncc1N 40689,CC1(C)CCC(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)C1 40690,N1(C(C(CC)CC)=O)CCN(C)C(C(=O)NC(C2CC3(CCC3)C2)C)C1 40691,CCN=C(NCC1CCCC1C(=O)OC)NC(C1CCOC1)COC 40692,C1(CNC(C(CCC)C)=O)COC(C)(C)CN1C(c1ccc(OCCF)cn1)=O 40693,C(=O)(CC1OCCc2ccccc21)NCC1(CNC(C2(C)CCC(O)CC2)=O)CC1 40694,C123CCN(CC1C2)C3=O.c1(C(C)(C)C)nc(CNC(C2(C)COC2)=O)cs1 40695,C12(C(N3C(CNC(c4c(C)onc4O)=O)CCCC3)=O)CCC(CC1)C(C)O2 40696,C1(C(CC)(C)C)CCCN1C(=O)CCN(C(=O)C(C)OC(C)(C)C)C 40697,C=CCC(CC=C)C(=O)NCC(CNC(c1cc(C2CC2)oc1C1CC1)=O)CO 40698,N1(NC(=O)OC)CCCN(CC2CCCO2)CC1.c12ccc(cc1)-c1scc-2c1 40699,C1(F)(CNC(C2(CCC=C)CC2)=O)CC(NC(C2COCC2C(N)=O)=O)C1 40700,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nnnc2c1 40701,N1(C(CCCCOC(C#C)C)C)CCN(CCCc2ccccn2)C(=O)C1 40702,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 40703,c1(C(N2CCC(C)(CNC(CN3C(C)CC3)=O)C2)=O)cnc2[nH]cnc2c1 40704,CC(CNC(=O)CNC(=O)CNC(C1CC2CC2C1)=O)S(C)(=O)=O 40705,c1(C(=O)NCCN(C(CC(COC)(C)C)=O)CCOC)cc(N)c2ncccc2c1 40706,c1(CC(C)(C)C(=O)NC2COCC2CNC(C2CC2F)=O)ccc(F)cc1F 40707,C(C(CC(C)C)NC(=O)C(O)C(F)F)NC(CCCN(C(=O)OC)C)=O 40708,N1(C(C(C)O)=O)CCC2C(C1)NC(=O)N2c1ccccc1Oc1ccccc1 40709,C=CCCC(C)(N=c1ccn(-c2ccc(Cl)cc2C)[nH]1)c1nnnn1CC(F)(F)F 40710,C1(NCC2C(C)C2)CCOCC1C(=O)N(CC(=O)NC)C1CC1 40711,CC(C)CC(O)C(=O)NC(c1cccnc1)C(=O)NC1(CN(C)C)CCCC1 40712,c1(SC)ccc(CCCC(=O)N2CC(CC(C)NC(C3CCCOC3)=O)C2)cc1 40713,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CCC(NC(c2coc(C(N)=O)c2)=O)C1 40714,N1(CCC(N2CCC(N(CCC)C(c3ncoc3C)=O)C2)=O)CCC(C)CC1 40715,CC1CN(C(=O)CN2CCC(=O)CC2)CCC1NC(=O)CCC1CCN(C)CC1 40716,c1(C(=O)NC2C3CCN(C(C(C(C)C)SC)=O)C3C2)ccc2cnsc2c1 40717,CC(C)C(O)C(=O)N1CCC(CCNC(C2(c3ccccc3F)CCC2)=O)CC1 40718,c1(C(=O)OCC2Cc3ccccc3CO2)n[nH]c2c1CCCCC2 40719,CC#CCCC(=O)NCCCCNC(c1sc(Cc2cccc(Cl)c2)nc1C)=O 40720,N1(C(C=CC=CC)=O)CCC(C=C)(CC(=O)NOCc2noc(C)n2)CC1 40721,Cc1cc(C)n(C(C)CCNCc2ccccc2-c2ccc(F)cc2)n1 40722,C(c1cc(Cl)ccc1Cl)=CC(N1C(C)CCC(NC(C2CC(C)(O)C2)=O)C1)=O 40723,C1(C(N2CCC(CNC(c3n(C)cnn3)=O)CC2)=O)CCc2ccccc2C1 40724,N1(C(C2(O)CCN(Cc3n[nH]cc3Cl)C2)=O)CCc2cccc(O)c21 40725,CCCC(CN(C(=O)CCOCCCC(CCC)c1ccco1)C1CCC1)OC 40726,c1(C(=O)NCC(CC(C)C)NC(c2n(CCC)ncc2)=O)cc(C)nc(O)c1 40727,C1(NC(C(C2CC2)OC)=O)CCN(C(C23CC(C)(C2)OC3C)=O)CCC1CO 40728,Cc1c(COC(C2CCCC2N2CCCS2(=O)=O)=O)cccc1S(N)(=O)=O 40729,N(C1CN(C(C2CCC3CC2C3(C)C)=O)Cc2ccccc21)C(C(CC)(F)F)=O 40730,N1(C(CSC(C)C)=O)CC(NC(=O)CC2(C(F)(F)F)CC2)C2CC12 40731,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 40732,N1(C(Cc2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(=O)C2CC2)C1 40733,CC1(C)C=C(C(=O)N2CCN(C3CCCN(C(=O)Cc4ccccc4)C3)C(=O)C2)C1 40734,N1(C(C(CC)Cl)=O)CC2CC(C1)N2C(=O)CN1CCN(c2ccc(Cl)cc2)C1=O 40735,N1(C(C=C(C)C)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CC12 40736,c1(C(N2CC(NCc3cc(C)no3)C(F)C2)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] 40737,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCOC2)=O)CC12CC2 40738,CN1CCC(C(=O)NC2(C)CCN(C(C3CCSCC3)=O)C2)S1(=O)=O 40739,C1(C(=O)NC(c2ccccc2)CNC(c2cnc(CSC)s2)=O)CC2CCC1O2 40740,CC(c1cccnc1)=CC(N1CC(N(C)C(c2cccnn2)=O)C(F)C1)=O 40741,Cc1cc(NC(=O)C(=O)NCC2COCCC2C)cc(-n2c(C)ccc2C)c1 40742,CCC(CC=C)Nc1ccccc1.C12CCN(C1)c1nnc(o1)CO2 40743,Cc1nc(F)ccc1CNC(C1(NC(C2CC(=C3CC3)C2)=O)CCCCC1)=O 40744,c1(CCNC(C=CC(C)NC(c2ccc(F)o2)=O)=O)ccccc1O 40745,c1(C(=O)NCCN(C(=O)C2=CSCCO2)CC)c[nH]c2c(OC)nccc12 40746,C(=O)(CC(C)CC(C)C)N(C(C)CN(C(c1cc(C)c(C)s1)=O)C(C)C)CC 40747,c1(C(=O)NC2CC(NC(C(C3CCCCC3)OC)=O)C2)cccc(C(F)(F)F)n1 40748,CN1CCc2[nH]nc(C(N3CCOC4CC3C4)=O)c2C1 40749,O=C(C1=CSCCO1)N1CCC(CCNC(C2(F)CCCCC2)=O)C1 40750,c1(OC)cc(NC(=O)C(C2CCCN(C(=O)Cn3cccn3)C2)(C)C)ccc1Cl 40751,c1(-c2n(C(C3CCCNC3=O)C)ccn2)cccnc1-c1ccccc1N 40752,CC1CCCC(C)C1NC(C1CCC(CNC(C2(C3(O)CCC3)CC2)=O)C1)=O 40753,c1(C(=O)NCCCCc2cn(C(c3onc(CCC)n3)C)nn2)[nH]cnc1C#N 40754,C(C(CO)CC(C)(C)C)NC(CC(c1cccc(OC)c1)C)=O 40755,C(CC(C)C(=O)NCCOCCNC(=O)CC(O)(c1ccccc1)C1CC1)OC 40756,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 40757,CC1(C(=O)NC2(CO)CC(F)C2)CCCN1C(=O)CSc1ccccn1 40758,N1(C(C2(C#N)CCCCC2)=O)CCC2(CCC2)C(NC(=O)CCOCC2CC2)C1 40759,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 40760,Cc1nc(C(=O)NC2CCCC(NC(c3cc(O)nn3C)=O)C2)c2ccccn12 40761,N1(C(CN(C)CC)=O)CCCC(CCNC(c2cn(C)nc2C(F)F)=O)CC1 40762,N1(C(C2(OC)CCC2)=O)CCC(C2CCCN(C(C3C=C3C)=O)C2)C1 40763,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)nnn1C)=O 40764,C(=O)(CC(CC(C)C)NC(=O)CC(O)CC)NCc1c(CC)nccc1 40765,C(C)(CC(=O)N(C)CCN(C)C(c1cn(C2CCCC2)nn1)=O)=C(C)C 40766,C(=O)(C(CCC1CC1)NC(=O)CNC(=O)CN(C)C)NC(c1nnnn1C)C 40767,c1(C(C(=O)NC2C(NC(CCNS(C)(=O)=O)=O)CC2)O)cccc(N)c1 40768,c1(CC(=O)N(CCCCCNC(C2(C#C)CCC2)=O)C)cccc(F)c1F 40769,C12(C(N3CCC(N(C(c4ccc(Cl)cc4)=O)CC)C3)=O)C3C4C1C1C2C3C41CO 40770,N1(C(C(C)NC(=O)NCC)=O)CC2CC3CC2C1C3NC(c1cn(CC)nn1)=O 40771,Cc1cc(C#N)c[nH]c1=NCC1CN(C(=O)CSS(C)(=O)=O)CC12CCC2 40772,c1(C(=O)NCC2(CNC(CC(CCC)C)=O)CCC2)cc(N)c(Br)c(F)c1 40773,c1(C(=O)NC(C2CCN(C(C3CCC(=O)N3C)=O)C2)C)ccc2nc(O)[nH]c2n1 40774,Cc1[nH]nc2ncnc(N3CCOCC3CN(C(=O)CCc3ccncn3)C)c12 40775,S(=O)(=O)(c1ccc(C(F)F)cc1)NCC(=O)NC1CCC(CC2CC2)CC1 40776,C1(c2onc(CCNC)n2)(C(C)OC(C)(C)C)CCN(C(=O)OC)CC1 40777,C1(C)(CNC(c2scc(C)n2)=O)CN(C2CCN(C(=O)CC=C(Cl)Cl)CC2)C1=O 40778,c1(CC(C(=O)N(CC(C)C)C)NC(C(CC)C)=O)cccc(F)c1 40779,c1(C(N(C2CCN(CC)C2)C(C(=O)NCCC)C)=O)nccnc1CC 40780,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 40781,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 40782,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3(F)COC3)c2)=O)C1 40783,N1(C(c2ccc(C)c(Br)c2O)=O)CCC2CN(C(C3CC3(C)C)=O)CC2CC1 40784,C1(N(C(C(C)CC2CC2)=O)C)CCCN(C(=O)Cc2cncc(Br)c2)C1 40785,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 40786,c1(OC)ccccc1OCCCN(C)C(=O)NCCNC(C)=O 40787,c1(C(=O)NC2(CC(=O)OC)CC2)cc(CNC(c2c[nH]c(=N)o2)=O)on1 40788,C1(NC(c2c(C)n(C3CC3)nc2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)C2)C1 40789,C(C)(C)(C(C)CC(=O)NC(CCO)CC(C)C)NC(c1c(C)snn1)=O 40790,c12ccc(nc1)c(=O)[nH]2.C1(CNC)CCCN1c1ccncn1 40791,C1(NC(COCC(C)C)=O)CC2CC1CN(C(c1coc(-c3ccsc3)c1)=O)C2 40792,N1(C(c2cc(OC)ns2)C(=O)NCCCOC)CC(C2CC2)OC(C)C1 40793,N1(C(c2c(COC)cco2)=O)CCC2C(C1)CN2C(c1cc(C)cc(C)c1)=O 40794,c1(OCC)nccc(C(C)NC(=O)NCCC2(OC)CCC2)n1 40795,N1(C(C=CSC)=O)CCCC1(C)C 40796,c1(CNC(C2C(COC)CC2)=O)nnn(C)c1C(=O)OC1CCN(CCO)C1 40797,Cc1cc(F)c(C(N2CCC(CCNC(=O)CCc3ccc(C)s3)C2)=O)cc1F 40798,C1(C#N)(C(=O)NC(C)CC(C)NC(c2conc2C(F)(F)F)=O)CCN(C)C1 40799,CCC(C)CCCCC(=O)N(C)CC1C2CN(C(=O)C=C(C)C(F)F)CC12 40800,c1(C(=O)NC2C(NC(c3cc(C)c(Cl)s3)=O)CC2)cccc2nn(C)cc12 40801,C1(CC(=O)N(C(CC#C)C)C)CN(C(=O)CC2CCC(=O)C2)CC12CC2 40802,c1(C(C)C)ncc(C(N2CC(CC(C)NC(c3cnccn3)=O)C2)=O)s1 40803,c1(C(=O)NC(C2CCCN(C(c3n(CC)ncc3)=O)C2)C)cc2n(c1)CCSC2 40804,c1(OCCF)ccccc1.C1(=O)C(C)SN1.C(C(C)NC(C)=O)N(C(=O)C)CC 40805,c1(C(=O)N)cnc(O)n1CC.c1(C(N2CC(C(C)CC)C2)=O)[nH]ccc1N 40806,c1(C(N(CC(CNC(C2(SC)CCC2)=O)(C)C)C)=O)ccnnc1C 40807,C=C(CNC(=O)C(CCC1CC1)NC(C1CC(=O)C1)=O)C(F)(F)F 40808,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 40809,C1(CNC(COCCC=C)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 40810,N1(C(C2(F)CN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 40811,c1(C(=O)NCC2C3CN(C(C4(C)CCCS4)=O)CC32)ccc2scnc2c1 40812,N#Cc1ccc(S(=O)(=O)N2CCC(N3CCCC3=O)C2)nc1 40813,c1(C(=O)NCC2(F)CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 40814,Cc1[nH]c(C#N)cc1C(N1CCC(NC(=O)CCc2cc(N(C)C)no2)C1C)=O 40815,C1(C(N(CCNC(CSCCCC)=O)C)=O)C(C)OC(C)C1C 40816,C1CC(CC)(C(=O)NCCCNC(=O)C=CCO)N1CC 40817,c1(CC(N2CCC(NC(CC(C)SC)=O)C(CO)C2)=O)cn(C)c2ccccc12 40818,c1(OCCCC(=O)N2CCCC2CC(c2ccco2)O)cccc2c1OCCC2 40819,c1(Cc2c(C)occ2)cn(C)c(C)n1.C12(CCC1)CC(=O)NCC(C)NC2=O 40820,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 40821,C1(NC(c2cncc(SC)c2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)CC1 40822,C(=O)(N=c1[nH]nc(-c2ccc(C(F)(F)F)cc2)s1)N1C(c2cc(C)on2)CCC1 40823,C1(O)(CNc2c(CNCCOC)ccs2)CCCC1C 40824,O=C(CCCC1CCCC1)NC1OC1C(=O)CCCn1cc(C2CCSC2)nn1 40825,C(CC1=CCCCCC1)NC(C1CCN(C(c2ccc(C)c(F)c2)=O)CC1F)=O 40826,C12CCN(C1=O)C1CN2C1.N(S(=O)(=O)N(C)C)CCNC(c1ncn(CC)c1)=O 40827,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)Cc3cncnc3)CC2)c(C)n1C 40828,C1(O)(CNC(C2CC(C(C)C)C2)=O)CCCN(C(C2CCSC2)=O)CC1 40829,CC1(C(=O)NC2(C(=O)NC3CCOCC3C(N)=O)CC2)CC2C=CC1C2 40830,C#CCC(CC#C)C(=O)N1CC(NC(=O)COCC2CCCOC2)C2(CCC2)C1 40831,C1(NC(=O)C#CCNC(=O)C(C2CCCCC2)F)CCN2CCCCC12 40832,C(CCC(C)NC(=O)Cc1csc(Cl)c1)NC(C1(NC(C)C)CC1)=O 40833,N1(C(CNC(=O)NC)=O)CCC2(CCC2)C(CNC(c2ccc(C(C)O)s2)=O)C1 40834,N1(C(C#CC(OCC)O)=O)CCN(C(c2cc3ccsc3n2C)=O)C(C)CC1C 40835,c1(C(=O)NCC2(SC)CC2)cc(Cl)ccc1.C1(CC=O)CCOC(C(C)C)C1 40836,c1(C(=O)NCCCCC2CN(c3ncnc(Cl)c3Br)C2)c[nH]c2ncccc12 40837,c1(C(=O)NCc2c(C)ncs2)ccc(C(=O)Cc2ccsc2Cl)cn1 40838,C1(NC(c2c(C)oc(C(C)C)c2)=O)CCCN(C(c2[nH]nnc2C)=O)C1C 40839,CC(C)(C)C(CC(=O)NC12CCOC(CNC(=O)CSC3CC3)(C1)C2)C(F)F 40840,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 40841,C(=O)(C1=CCCC1P(C)(C)=O)N1C(C)CN(C(=O)CC(F)(F)Cl)CC1 40842,c1(C(N2CCC(N(C(=O)C(F)OC(F)(F)F)C)CC2)=O)cnc2ncc(Cl)cn12 40843,N1(C(C2CN(CCC)C(=O)C2)=O)CC(NC(=O)CNc2ccccn2)CCC1C 40844,CC(C)(C)C(CO)C(=O)NCC1CC(C(=O)NC2CC3CC(O)C2C3)=NO1 40845,N1(C(c2c(C)ccn2C)=O)CCC2(CC1)CN(C(=O)C1=CCCCC1C)C2 40846,C1(NC(C=CC2C(=O)NCC2)=O)CC2(C1)CC(F)(F)C2 40847,c1(OCC)cc(Cl)ccc1C(=O)NC12C(CN(C(c3cccc(OC)n3)=O)C1)C2 40848,c1(C(N(CC#C)C)=O)cc(CNC(C2CC(F)(F)C2)=O)no1 40849,CCC(C)CC(=O)C(=O)NCC(C(=O)NCC(n1cncn1)C)C(C)C 40850,C(c1cccc(Cl)c1)=C(C)C(N1CCN(CCNC(C2CC=CCC2)=O)CC1)=O 40851,N1(C(CCOc2c(C(C)C)cccc2)=O)CC(NC(C2CC2F)=O)CCC1C 40852,c1(C(=O)NCC2OCC(C(=O)NCC3CC(O)C(O)C3)C2)ccc([N+](=O)[O-])[nH]1 40853,C1(C(=O)NCC#CCNC(c2c(OC(C)C)cccc2)=O)CCCC1S(C)(=O)=O 40854,c1(CN(C)C(c2cnn(CCNC(c3cnccn3)=O)c2)=O)ccccc1Cl 40855,CC1CCN(C(=O)C(C2CCOCC2)F)CC1C(=O)NCCCCO 40856,N1(C(=O)NC(c2ccccc2F)C)CCC(O)(C2CCCC2)CC1 40857,c1(NCCC(N2CC3C(NC(C(C)=C4CCCC4)=O)(C3)C2)=O)oc(C)nc1C#N 40858,C1(C(=O)Nc2ccnn2COCCCF)CCOC(C(=O)Nc2ccccc2)C1 40859,N1(C(c2c(Cl)cn(CCC)n2)=O)CCCC(N=c2nn[nH]n2CCC)C1 40860,c1(C(N2C(C(N(CCO)CC3CCCN(C)C3)=O)COCC2)=O)cc2sccc2[nH]1 40861,c1(CNC(C(CCOCC)NC(c2csc(F)c2)=O)=O)ccc(F)c(F)c1 40862,CC(C(=O)NC(CNC(C1(c2cccc(Cl)n2)CC1)=O)C1CC1)C(C)(F)F 40863,C(=O)(C1CCc2c[nH]nc21)N1C(C)(C)CC(NC(c2cccc(F)n2)=O)C1 40864,c1(CCC(=O)NC(C(=O)N(CC(C)C#N)C)C2(O)CCC2)cn(C)nn1 40865,C1(C(N2CCC(C3OCCO3)C2)C(=O)NCCCSCC)CC2CCC1CC2 40866,N1(C(CC2C=NN(C)C2=O)=O)CC(O)(C2(CNC(c3ccc(CO)o3)=O)CC2)C1 40867,c1(C(=O)NC(CCNC(C2C(C)C2C)=O)C)cc(C(F)(F)F)ccc1N 40868,Cc1ccc2c(c1)CCC2C(=O)NCC(O)CCNC(=O)CCOCC(C)C 40869,C(CC(C)C)(C(=O)NCC(=O)NNC(=O)C1CCN(C)C1)NC(=O)OC 40870,c1(C(=O)NC(C(=O)NCc2ccc(C)c(C)n2)C2CCC2)ccc2nccn2c1 40871,C1(C(=O)NCC2CSCCO2)(COC)CCCN1C(=O)CCCc1ccccc1 40872,c1(C(N(CCNC(C2C3COCC23)=O)CC)=O)nc(C)sc1Br 40873,c1(N(CCC(=O)N(C)CCO)C)cc(C2CC2)nn1C.C1(=O)C=CC(C)N1C1CC1 40874,n1(CCCC)ncc(C(=O)NC2(CO)CCN(C(c3cnc(S)[nH]3)=O)C2)c1C 40875,C=CC1(C(=O)N(C)Cc2cccc(O)c2)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 40876,c1(OC)nc(C)ncc1C(=O)NCC(C)NC(C1CCC2CC2CC1)=O 40877,C1(CNC(c2ccsc2Br)=O)C2CCC1CN(C(C1CCC(F)(F)C1)=O)C2 40878,N1(C(c2nc(C)sc2)=O)CC2CCC1C2NC(C(=O)NC)=O.c1c(C)n[nH]c1C 40879,Cc1cc(F)cc(C(=O)N(C(Cc2cnc[nH]2)C(=O)O)C)c1Br 40880,C1(NC(c2c(SCC)scc2)=O)CN(C(c2ccc(C)cn2)=O)CC1N=[N+]=[N-] 40881,C(=O)(CC(C)CC(C)C)NCC1N(C(c2n(CC)ncc2)=O)CC=C1 40882,C1(NC(CCCc2n(C)cnn2)=O)CCCC12CN(C(=O)Cn1cccn1)C2 40883,c1(C(N2CCC(Nc3c(C)cncn3)C2)=O)ccc(F)c(C#N)c1 40884,CCCC(CC1CCCC1)C(=O)NC(C)(CNC(C1CC(F)(CO)C1)=O)CO 40885,Cc1ocnc1CC(=O)NCC1CC(CNC(=O)CC(F)F)CO1 40886,C1(C(=O)NC(C)C=CC(=O)N(C)CC2CCCOC2)CCSCC1 40887,C12CCN(CC1)C(=O)c1nnc(s1)N(C)C2.c1(C(=O)OC)c(C)ncn1O.CC 40888,c1(CNC(C(=O)NCCOC)=O)ncc(C(C)C)o1.C12CC(C1)N(C)C2=O 40889,C#Cc1cnc(NC(C2(OC)CCN(Cc3ccc(F)c(Br)c3)C2)=O)cn1 40890,C1(C(N2CC(OC3CCN(C(C(C)OC)=O)C3)C2)=O)COC(C)(C)O1 40891,Cn1ncc2nc(Cl)nc(N3CCC4(CCCN4C(C4C5CCC(=O)C45)=O)C3)c12 40892,C1(OCCNC(=O)COc2cccnc2)CCN(C(c2cccnc2CO)=O)CC1 40893,C(CN=c1[nH]c2c(c(=NC3CCCc4ccc(F)cc43)[nH]1)SCC2)NC(=O)NC 40894,C(CC(C)(C)C(=O)NC1CCC(C(=O)NC2CCCC(C)CC2)C1)OC 40895,Cc1[nH]nc(C(=O)NC2CC(CNC(c3nsnc3O)=O)C2)c1C 40896,Cc1ncnc(NC(=O)C(Cc2ccc(F)c(F)c2)NC(=O)N(C)C)c1C 40897,c1(CCC(=O)NC23CN(C(C4CCN(C)C4)=O)C(C2)C3)ccc(Cl)cc1Cl 40898,N1(C(=O)COCC(F)(F)F)CCCC(C2CCCCN2C(c2cccs2)=O)C1 40899,N1(C(CC2CCC(=O)C2)=O)CCCC(F)(C(N2CCC(CCCO)CC2)=O)C1 40900,N1(C(C(C)CF)=O)CCOC2(CCC(N=c3[nH]c4ccc(F)c(F)c4s3)CC2)C1 40901,C1(C(N2CC(NC(c3c(C)nc(CC)s3)=O)C(C)C2)=O)CCCCC12CC2(F)F 40902,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC(C)(C)C)C(CC2CC2)C1 40903,C1(C(=O)NCC2(C)CCN(C(C3N(C)C(=O)CC3)=O)CC2)CC2CC1CC2(F)F 40904,C1(N(C(C2CC(=C)C(=O)CCCCCC(C)N2C)=O)CC)CCc2ccccc2C1 40905,C(CN=c1[nH]c(=NCCN(C)C)[nH]c2ccc(Cl)cc12)(c1ccccc1Cl)SC 40906,CC1CNC(=O)CN1C(C1(NC(C2CCCN2C=O)=O)CCCCC1)=O 40907,C1(CN(C)C(C2CC2(C)C(F)(F)F)=O)CCN(C(=O)CCCc2cncs2)C1 40908,C1(C(=O)NC2(C)CCN(C(C(C)OCOC)=O)C2)CN(C)C(=O)CCO1 40909,C1(SC)CN(C(C2CCC(=O)N2)=O)CC1NC(c1ccnc(Cl)c1)=O 40910,CCC(CC)(CCNC(=O)C(F)C(C)C)NC(c1cc(C(=O)OC)co1)=O 40911,Cc1ccnc(O)c1C(=O)NCC1CN(C(C2CCNC(=O)C2)=O)CCO1 40912,C1(C(N(C)CCn2cc(-c3cn[nH]c3)nn2)=O)CCCN1CC(F)F 40913,c1(CC)ccc(C(=O)C(=O)NC23CC(CNC(c4ncsc4C)=O)(C2)C3)s1 40914,c1(C(c2nnnn2C)NCCCC(=O)NCCOC)coc2ccc(F)cc12 40915,C1(N(C(C2CCC(CC)CC2)=O)C)CCCN(C(c2[nH]c(C)nc2C)=O)CC1 40916,Cn1nccc1CC(N1CSCC1C(=O)NOC1CCOC1)=O 40917,c1(C(=O)NC2C(NC(c3nc(CC)sc3)=O)CCC2)cc(N)c(C)c([N+](=O)[O-])c1 40918,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CCCOC)N(C)C 40919,CN1CCC(C(N2CCN(C(=O)C=Cc3cn(C)nn3)C(CCO)C2)=O)CC1=O 40920,c1(C(N2C3CN(Cc4c(OC)c(F)ccc4F)CC32)=O)cnc2ccc(Br)cc2c1 40921,Cc1c(C(=O)NCC2CC(CC(=O)NCC3CC(C)CO3)CO2)cnn1C 40922,CCCC(C)(C)CC(=O)NCC1CCN(C(C2C3CCC(C3)C2C)=O)CC1O 40923,c1(C(=O)NC2CC(CNC(c3ccc(SC)s3)=O)C2)c(O)nnc(C)c1C 40924,CC1(C)CCC(C(N2CC(CF)(NC(=O)CCOC3CCCCC3)C2)=O)OC1 40925,c1(C(=O)NCCN(C(C(CC)(C)O)=O)C)cc(Br)ccc1C1CC1 40926,C(=O)(CC1=CCCCC1)N1C(C(C)NC(=O)C2=CSCS2)CCC1 40927,c1(NC(N2CC(c3nnc(C)s3)C2)=O)cc(Cl)cc(F)c1F 40928,CC1C(NC(c2csc(Cl)c2Cl)=O)CCN1C(=O)CCSC1CCCC1 40929,c1(CC)ncc(C(N2CCC(CN(C)C(c3ncccn3)=O)CC2)=O)c(C)n1 40930,C1(CNC(c2c(C)ncn2C)=O)CC2(CCN(C(=O)C(C#N)C(C)C)CC2)CO1 40931,C(=O)(C(C(C)C)C1CCC1)NCC(CCNC(C1CC1C(=O)OC)=O)OC 40932,N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC(C)(NC(=O)COC(C)C)C1 40933,c1(OC)ncc(Br)cc1S(=O)(=O)N1CCC(CC(=O)NCC2(C)CC(F)(F)C2)C1 40934,c1(N(CCCSC)C)nnc(-c2ccccc2)n1CC(C)C1CC1 40935,C1(CC)CCN(C(=NCCC(C)(F)F)NCCCCl)CC1(C)C 40936,C(=O)(CCCC(=O)OC(C)(C)C)N1CC(N(C(CC(C)NC(C)C)=O)C2CC2)C1 40937,C(=O)(C1=C(Cl)CC1)NC1(C)CN(C(C(C)CC2CC2)=O)C1 40938,C1(CN(C(c2c(C)cco2)=O)CCO)CC(C(C)C)=NO1 40939,c1(C(N2CC=CCC2C2CC2)C)cnc2[nH]ncc2c1 40940,C1(C(C)C)N(C(=O)CONC(c2ccncc2F)=O)CC12CCC2 40941,c1(C(=O)NC(C(NOCC)=O)C2(O)CCC2)ccc(F)cc1O 40942,CC1CC(=O)NC1C(=O)NCC1CC(F)(CNC(=O)CCCC2CC23CCC3)C1 40943,c1(C(=O)NCC2CCN(C(C3(C)ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 40944,c1(OC)cc(C(=O)OC2CCCC2)cc(C)n1.c12ccnc(c1)C(=O)NC2 40945,C12(C(=O)NCCCCCCN(C(C(CSC)OC)=O)C)CC3CC(CC(C3)C1)C2 40946,C(=O)(C1=C(C)OCC1)NCC1(CC)CN(C(=O)C(C2CCOCC2)O)C1 40947,CC1CCCC(CC(N2CCC(OCCN3CCN(Cc4ccon4)CC3)C2)=O)C1 40948,N1(C(C(C2CCCC2)OC)=O)CC(O)(C(C)NC(C2(CC(F)F)CCC2)=O)C1 40949,c1(OC(c2n(C)nc(CN(C)C)c2Cl)=O)nc(C(F)(F)F)c2ccccc2n1 40950,Cn1ncc([N+](=O)[O-])c1NC(c1nccc(-c2cncc(F)c2)n1)=O 40951,C1(CC(=O)N(CCOC)CCNC(c2ccc(Br)cn2)=O)COCC(C)(C)O1 40952,C1(NC(CCCN(C)C(c2cncc(CO)c2)=O)=O)CCCC(F)C1 40953,N1(C(c2cc(C)c(F)cc2F)=O)CCC2C(CCN2C(C2COCCO2)=O)C1 40954,C1(NC(C(C)SC)=O)CC(C(=O)NOCC(F)F)C1(C)C 40955,C1(CNC(CC(C)NC(C2CCCN2C2CC2)=O)=O)CCNC(=O)C1 40956,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2(O)CCC2)C1 40957,C(=O)(CCCCCS(N)(=O)=O)N1C(NC(C(C)N2CCCC2)=O)CCC1 40958,c1(C(N2CC(CNC(C(CC)NC(N)=O)=O)C2)=O)oc2c(C)ccc(C)c2c1C 40959,C(CC(O)C(=O)Nc1cccc(NC(c2c(Br)noc2C)=O)c1)SC 40960,CCCCC(CNC(=O)CCCNC(N)=O)NC(C1CCNCC1C)=O 40961,C1(C(=O)NC(CNC(CCNS(CC)(=O)=O)=O)C(C)C)CC2(C)CC1CO2 40962,c1(N(C)C)ccc(CCC(=O)NC2CC(C(=O)Nc3ccc(F)cc3)C2)cn1 40963,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CCCC3)=O)CC12 40964,N1(C(C2(CCCC)CCOCC2)=O)CC2CCN(C(C3CCC(=O)C3)=O)CC2C1 40965,CC1C(=O)CCC1CC(=O)NC1(CNC(c2coc(C3CCCCC3)n2)=O)CC1 40966,N1(C(c2cccc(CC)c2)=O)CC=C(CNC(=O)C(C)NC(C)=O)CC1 40967,C1(CNC(CC2(CC(=O)OC)CCCC2)=O)CC(F)CN1C(c1cc[nH]c1)=O 40968,C1(CNCC2N(C(c3cccc(Cl)c3)=O)CCCC2)CC2CCC1CC2 40969,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC=CC2)=O)C(O)C1 40970,c1(CC(N2CC3(CC(NC(C=CC(=O)N(C)C)=O)C3)C2)=O)c[nH]c2ccccc12 40971,Cc1cc(=NC(=O)c2ncsc2Br)[nH]n1-c1cccc(C(=O)OC(C)(C)C)c1 40972,N1(C(C(C)SCCCC)=O)CCN(C(C2OCCCC2(C)C)=O)C(C2CCC2)C1 40973,c1(C(N2C3CN(Cc4ccc(C)cc4Br)CC32)=O)cc(F)c(C)cc1Br 40974,Nc1cc(C(=O)NCC(CO)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 40975,CCC1=C(C(=O)N2CCCCC2C(C)NC(C2(C3CC3)CC2)=O)CCCO1 40976,C1C(C(=O)NCC(O)CF)CC(CC)C(=O)CC(C)C(=O)N1 40977,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 40978,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)CC=C(Cl)Cl)C3)=O)cc12 40979,c1(NC(c2n(CCCSC)nnn2)C(C)(C)C2CCCO2)cnc(Cl)c(Br)c1C 40980,C12CCC3CN(CC3C1)C(=O)c1ccc(o1)C(=O)N2.C1(CO)CCOC1=O 40981,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(C(=O)Cc1ccccn1)CCO2 40982,C1N=C2C=C(N=C(Cl)N2)C(=O)N2CCOC1C2.c1(CC)c[nH]cc1C(=O)OC 40983,CC(=O)CCCCCCC(=O)NC1(CNC(=O)C(C)NS(C)(=O)=O)CCCC1 40984,c1(C(=O)NC2CC(CCNC(CCSc3n(C)nnn3)=O)C2)cccc(CO)c1 40985,CC1(C)C(NC(=O)C2=C(Cl)CCC2)CCN1C(=O)CC1CCOC1=O 40986,N=c1[nH]c2c(s1)CN(C(C1CC1c1ccc(Br)cc1)=O)CC2 40987,N1(C(C(c2n(C)cnn2)(C)C)=O)CC2CCCN(C(=O)Cn3cnnn3)C2C1 40988,C1(COC)CC=C(C(c2nnnn2C)NCc2ccc(F)cn2)CC1 40989,C1(CC(=O)N(CC(C)NC(c2nccc(CC)c2)=O)C)CCCC2(CCC2)CO1 40990,C#Cc1ccccc1CNC(=O)CC1CCCCN1C(c1c[nH]ccc1=O)=O 40991,c1(C(N2CCC(O)(CNC(CCCC(C)O)=O)C2)=O)[nH]nc2cnccc12 40992,C12CCCN(C1)C(=O)N2.c1(NC(c2n(CCC)ccn2)C)cn(C)nc1OC 40993,c1(C(N2CCCC(O)(CNC(C3CC4(CC4)C3)=O)C2)=O)cc2n(n1)CCOC2 40994,CCC(C)CCC(=O)N1CCCC1C(C)NC(=O)C(F)(F)c1ccsc1Cl 40995,n1(CC(C)C)cc(CC(=O)Nc2noc(CCN(C)C)n2)cn1 40996,C(=O)(C(O)CSC1CN(C(C=CCCC)=O)C1)N(CCNC(c1ccoc1)=O)C 40997,c1(C(=O)NCCC2(CNC(=O)CC3CCOC3=O)CC2)cnc2ncnn2c1O 40998,N1(CCC(N2CC(C(C)NC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)CCN(C)CC1 40999,C1(C)(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)CCCO1 41000,N1(C(CCc2cc(C)no2)=O)CCC(c2cn(CC(=O)N(C)C)nn2)C12CC2 41001,C1(OC)CCC2(C(=O)NC(C)(C)C(=O)NC(Cc3ccco3)CO)CC12 41002,N1(C(C2C(C#C)C2)=O)CCN(C(c2ccc3cncn3c2)=O)C(C#C)C1 41003,N1(C(C2(C#C)CCCC2)=O)CC2(CCC(CNC(c3cccc(Cl)c3O)=O)O2)C1 41004,N1(C(Cn2c(C)ncc2)=O)CC2CC(O)C1C2NC(c1cccc2cncn12)=O 41005,c1(-n2nnnc2OC(C(c2ccc(OC)cc2)CC(N)=O)=O)cc(C)ccc1C 41006,c1(C(=O)NCC2CN(C(C(C(C)C)OC)=O)CC2C)cncc2c(O)nccc12 41007,C1(N(C(=O)COCC2CCCCO2)CC)CCCN(C(=O)C(C)(C)O)CC1 41008,N1(C(CS(N)(=O)=O)=O)CCC(C(N2CCCC2C(=O)C2CC2)=O)CC12CC2 41009,C1(O)(C(C)NC(C(CCC)O)=O)CCN(C(c2cc(C)sc2C)=O)CC1 41010,c1(C(=O)O)ccc2nc(NC3CN(C(c4sc(Cl)cc4Br)=O)C3)oc2c1 41011,N(C(=S)N1CC(C)c2ccccc2C1)C(COC)(C)C 41012,c1(C(N(CCCNC(=O)C(C)c2cncs2)CC)=O)cccc2c1NCC2 41013,C1(CC(=O)NCCC(=O)NC(C=CC(=O)OC)C)CCC(C)(C)C1 41014,CC1CCN(C(c2sccc2C2CC2)=O)C(CNC(c2cc(C#N)c[nH]2)=O)C1 41015,C(CCC(=O)NCc1nocc1C(=O)NC1CCCSC1)OC(C)=O 41016,c1(C(=O)NCC2N(C(CCCCOCC)=O)CCCC2)nc2c(s1)COCC2 41017,c1(CC(=O)N(C2(C)CN(C(c3cn(CCC)nn3)=O)C2)C2CC2)cccc2[nH]ncc12 41018,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)CC1CC1 41019,c1(C(=O)OCC)sc(NC(C23CC(C)(CO2)C3)=O)c(C(=O)OC2CC2)c1C 41020,N1(C(C2C3CC(NC(c4cccc(OC)c4)=O)CC32)=O)CCC2(CC2)CC1C 41021,N1(c2ccnc(C)n2)CCN(C(C23CCCCC2C3)=O)CCCC1 41022,c1(C(=O)NC(C)(C)CN2CCCCC2)ncc(F)c(O)n1 41023,N1(C(C2C3(CC(NC(C(CCC)F)=O)C3)C2)=O)CC2CSCC2(C)C1 41024,N12CCOCC1C2=O.C(=O)(C(F)(F)F)NCC(=O)NCCCCCNC(C)=O 41025,C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)C1(C)CN(C(=O)C)C1.c1(C=O)ccnc(Cl)c1 41026,c1(NC(C2(C)CCN(C(c3cccc(F)c3F)=O)C2)=O)cc(Br)cnc1Br 41027,C12(NC(C(CSC)C)=O)CC1CN(C(=O)Cc1ccnn1C)C2 41028,N1(C(C(C)NC=O)=O)CCN(C(c2ccc(N(C)C)cn2)=O)CC1c1cccs1 41029,c1(C(=O)NCCC(C)N(C(=O)CC2CCCC(=O)N2)C)cccc2[nH]nc(O)c12 41030,C(CCC(=O)N1CCCC1NC(C1CCCCS1)=O)NC(=O)NC(C1CCCC1)C 41031,CCC(CCC(=O)NC1CCC(CCOC)C1)NC(c1cncn(C)c1=O)=O 41032,C(c1cc2ccccc2o1)=CC(N1CC(CNC(C(C=C)(C)C)=O)C(O)C1)=O 41033,C(CCCC(CO)NC(c1cc(C2CC2)nn1C)=O)NC(CC(CC)C1CC1)=O 41034,CCCCCC(F)C(=O)NCCC(CC)(CC)NC(C1CCC(CCC)CC1)=O 41035,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41036,C1(C(=O)NC(CNC(CCOCC)=O)(C)C2CC2)CCCSC1 41037,c1(CC)sc(C(=O)NC(C)CCNC(c2nnsc2C)=O)cc1Br 41038,C1(C(N2CCC(NC(C3C(COC)C3)=O)(CO)C2)=O)CN2CCN1CC2C 41039,CC1(C(=O)NCc2cc(Br)cs2)CC(NC(=O)Cc2ccoc2)C1 41040,N1(C(C(C)n2ccnn2)=O)CC2CC(NC(C3(CF)CCC3)=O)CC1C2 41041,C(CSC)(C(=O)NCc1cc(C(=O)NCC(C(C)C)OC)no1)OC 41042,C1(C(=O)NCC(C2(c3cc(C)c(O)nn3)CC2)N(C)C)CCc2ncsc2C1.C=O 41043,C(=O)(CS(=O)CCC(F)(F)F)NCC(=O)NCCC(=O)NC(C(N)=O)CO 41044,Cn1cc(C(C(=O)NC2C3COCC23)N(C(=O)COc2ccsn2)C)cn1 41045,O(NC(=O)CC(CC)NC(=O)CCCN(C)C(C1CC1OC(C)=O)=O)CC 41046,c1(OC)ccc(S(=O)(=O)N2CC3CCC(C2)N3C(c2cc(C)nc(Cl)c2)=O)cc1F 41047,CC1CN(C(=O)CCc2cnco2)CCCN1C(=O)C(c1ccc(F)cc1)O 41048,c1(CC)ncsc1C(=O)NC(C)(CNC(C1CCCC1CC)=O)CO 41049,C1(c2c(C)cc(F)c(C(C)C)c2)NC(=O)N(CCF)C2=C1C(=O)NC(C)C2 41050,C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)CN2C(c1cc(Cl)cnn1)=O 41051,C(N=c1[nH]nc2ccc(Cl)cn12)c1c(-c2ccccc2)c[nH]n1 41052,CC(C)C(C(=O)NC1(C(=O)NCC23CC(F)(C2)C3)CCC1)SC1CCCC1 41053,C1(C(C)C)OCCC1C(=O)N(CCCN(C(=O)C(Cl)=CCl)C)C 41054,C1(NC(c2coc(CO)c2)=O)CCN(C(=O)CSc2ccccn2)C1C1CC1 41055,N1(C(N2CC(NC(=O)OC(C)(C)C)C(C)C2)=O)CC2CCC1C2N(CCC)C 41056,C1(NC(c2n(CC)nnc2)=O)CC2CC1CN(C(c1ccnc3[nH]cnc13)=O)C2 41057,C=CCCC(C(=O)NC(c1cn(C)nc1C)C)NC(c1cnc(OCC)nc1)=O 41058,C1(CNC(C2(C)CCN(C)C2)=O)CN(C(C2CCCC2(C)C)=O)CCC12CCC2 41059,CC1(C)CC(C)(NC(=O)CSCCNC(C2CC2(C)C)=O)C1 41060,C1(C(=O)NC2C(C)N(C(C3CCc4nc[nH]c4C3)=O)CC2)CC2(CCCC2)CO1 41061,C(=O)(C1CCCc2n[nH]cc21)NCC(=O)NCC(C)CNC(=O)C(F)(F)F 41062,N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(C2CC3CCC2O3)=O)CC(C)(C)C1 41063,CC1(C(=O)NC2CC(NC(=O)C=C(Cl)Cl)C2)CCC(=O)N1 41064,CC1(OC(F)F)CCN(C(=O)CC2(NC(C3(C)CCCOC3)=O)CC2)CC1 41065,c1(C(N2CCCC(n3cc(CN(C)C)nn3)C2)=O)cc(O)nc(Cl)c1 41066,C=CCC(CNC(C1(C)CC1)=O)NC(=O)CC1CCCCC1 41067,C1(CCNC(CN2CCC(C)C2)=O)CN(C(=O)Cc2ccnc(C(N)=O)c2)CC1C 41068,C(=O)(N1CC(n2cc(CCCCC3CCCC3)nn2)CO1)c1c(C)nccc1 41069,c1(C(=O)NCC2C(NC(c3ccc(OC)cc3)=O)C2)cccc(C2CC2)c1C 41070,N1(c2snc(CCC)n2)CCC(C)(C)C(CNC(=O)CCCN(C)C(C)=O)C1 41071,CC1(C)Cc2cccc(S(=O)(=O)NCCn3ccc(O)nc3=O)c2O1 41072,C1(O)(C(C)NC(=O)CCOC2CC2)CCN(C(C2CC2c2nccn2C)=O)C1 41073,CN(CCCC(=O)NCCOCCNC(C1(CC2CCC2)CCCC1)=O)N=O 41074,c1(C(C(=O)NC(C)C(CO)NC(C2(CCF)CC2)=O)(C)F)ccccc1F 41075,N1(Cc2c(OCC)c(Cl)ncc2)CCC(N=c2[nH]cnc3cc(I)sc23)CC1 41076,c1(CN(C(=O)C=CC(=O)NC2CCCC2)CCC)ccccn1 41077,C(=O)(C1=CC2(CCOC2)C1)N1CC(CNC(CC=C)=O)OCC1 41078,c1(C(c2n(CC(=C)C)nnn2)NCC(c2ccccc2)CO)nnc2sccn12 41079,C12C(CCN1C(C1(F)CCCCC1)=O)C(=O)N2.c1(OCC)ccc(OC)nc1 41080,c1(CC)cc(Cl)ccc1C(=O)NCC1(CNC(=O)C(C(C)C)NC)CCCC1 41081,C(c1ccc(OCC(C(=O)NCC(COC)OC)OC)cc1OC)=CC(=O)OC 41082,C(=O)(C(CC(C)C)N(C)C(c1cc(CO)on1)=O)N1CCC(C(CC)C)CC1 41083,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41084,N1(C(C(C)OCC)=O)CC2CC(O)C1C2NC(c1cc(C)sn1)=O 41085,C1(C(=O)OC)CCC(C2(C(=O)NCC3(COC)CC3)CNC2)C1.C1CC1 41086,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41087,N1(C(c2ccc(OC)c(O)c2)=O)CC2OCCN(C(=O)COCC3CC3)C2C1 41088,c1(C(=O)NCC2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)ccc2c(c1)CCO2 41089,c1(CC)ccc(C(N2CC(C)(NC(c3n[nH]cc3F)=O)C2)=O)cc1[N+](=O)[O-] 41090,C1(C)(NC(C2CCC(CNC(CCCOC)=O)O2)=O)C=CCCC1 41091,N1(C(CC(=O)NCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41092,N1(C(c2c(C)n[nH]c2)=O)CC2CCCCN2CC1CNC(c1cc(O)ncn1)=O 41093,C1(C(=O)NCc2nc(C(N3CC(n4ccnc4)C3)=O)co2)COCCOC1 41094,C1(CC(=O)NC2CCN(CCC)C2)CCC(C)(C)CN1C(C1CCOC(C)C1)=O 41095,C(C)(C(=O)NC1COCCN(C(c2cc(F)ccc2Cl)=O)C1)(C(C)C)OC 41096,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)C(C2CCCCC2)F)C(C(C)(C)C)C1 41097,c1(C(N2CC(C(N3CCC(COC(C)=O)C3)=O)C3C2C3)=O)ncc2ccccn12 41098,c1(C2C(=O)N(C)CC2)c(F)cccc1F.C=CCC(C)C(=O)OC 41099,c1(C(N(CC(=O)O)CCC2C(C)C2)=O)ccc(CO)s1 41100,N1(C(C(C)C(C)NC(=O)C(=O)NC2CC2)=O)CC2(C1)CC(C)(C)C2 41101,CC(O)(C(=O)NC1C=CC(C(=O)Nc2cc(C(F)(F)F)cc(I)c2)C1)C(F)(F)F 41102,N1(CC2CC(C(=O)OC)(C(F)F)C2)CC(CO)CC(c2ccccc2)C1 41103,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC1CCN(C(c2cn(CCC)nc2)=O)C1 41104,c1(CN2C3CC(C3)C2=O)ccc(F)c(C#N)c1.C1(OC(C)C)CCOCC1 41105,C1(Cl)(C(=O)NCCN(C(c2ccc(C(C)=O)cn2)=O)CC)CC12CCC2 41106,CC(C(C)C(=O)N1CC(CNC(C23CCCCN2CCC3)=O)C1)S(C)(=O)=O 41107,O=C1Nc2ccc(C(N3CCCC3(C)CNC(=O)CC3CC(F)C3)=O)cc2C1=O 41108,C(CCN=c1ccnc(N2CCOC3(CCOCC3)C2)[nH]1)OC=C 41109,CN1CCN2CC1NC(=O)CC1CCN(CC1)C(=O)C1C(C1)C2=O.C1(C)CC1.C 41110,c1(C(N2CCCCC(NC(c3n(OC)cnc3C)=O)C2)=O)cnc(O)n(C)c1=O 41111,c1(C(=O)NCCC(CNC(c2nn(C)c(C3CC3)c2)=O)O)cc(F)c(F)cc1N 41112,C1(n2cc(CN(C(CCc3cnc(C)o3)=O)C3CC3)nn2)CCCNC1=O 41113,c1(C(N2CC3C(CNC(c4cn(CCCC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41114,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(c1cnccc1C(C)(C)C)=O)C2 41115,C1(NC(c2c(C)nc(C)n2O)=O)CCN(C(c2cc3n(n2)CCC3)=O)C12CCC2 41116,C12CC(C(C)(C)C)CN(C1)C(=O)C(=O)N1CCN(CC1)CCNC2=O.C1(CC)CC1 41117,C1(NC(COCCC)=O)CC2CCCC(C1)N2C(C1CC12CC2)=O 41118,N1(C(Cc2c(C)cc(OC)c(OC)c2)=O)CCN(C(=O)C(N)=O)CC(CO)C1 41119,Cc1cc(C(=O)NC(C)(C)CN(C)C(C2CCCC(=O)O2)=O)nn1C(C)C 41120,c1(OC)cc(F)ccc1CC(=O)N(C)CCN(C)C(c1nccnc1C(N)=O)=O 41121,c1(C(N2CCC(NC(C(C=CC)O)=O)C2(C)C)=O)c(N)cc(F)cc1Cl 41122,C1(CC(=O)N(C)CC)CCCCC1F.n1(CCOCC)cc(COC)nn1 41123,c1(C(N2CC(CCC)C(NC(C)=O)C2)=O)ccc2cnn(C(C)C)c2c1 41124,C(=O)(C1CC(=O)Nc2ncccc21)N1CCCC(CNC(=O)CC2(O)CCC2)C1 41125,N1(C(CSC)=O)CCOC(C(N2CC(O)CC2CO)=O)CC1 41126,N1(C(c2ccon2)=O)CCN(C(C2CSCCS2)=O)C2(CC2)C1 41127,c1(OC)cccc(Br)c1C(N1CC(O)(CCNC(C23CCC(CC2)O3)=O)C1)=O 41128,CC1C(=O)CCC(C(=O)NCC2CCN(C(=O)COc3ccccn3)C2)C1(C)C 41129,C=C1CC(CC(=O)NCCC2(CNC(=O)C=C(C)C(F)F)CC2)C1 41130,CC1=CCC(C(N2CCC(OCC(=O)N(CC(F)F)CC3(F)CC3)CC2)=O)CC1 41131,C#CCCC(C(=O)NCC#CCC)NC(=O)CC1(O)CCCCC1 41132,c1(C(N(C(CSCC)C)C)=O)ccc2c(c1)C(=O)CCN2C.C12(CC1)C(=O)N2 41133,c1(C(N2CCC(OC(CC)(C)C)C2C)C(=O)NC2CC(F)(F)C2)ccccc1I 41134,CCC(C)C(O)C(=O)N1CCCC1C1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 41135,c1(CCC(=O)NCCC(C)NC(c2cccnc2)=O)ccccc1OC1CCC1 41136,c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41137,CC(C)CC(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)C)cc1)C(N)=O 41138,CCCC(C(=O)NCC1(NC(=O)C(=O)NCCC(N)=O)CCCC1)OCC 41139,Cc1c(Cl)ccc(N(C)C(C(C)CC(C)C)=O)c1Cl.NC 41140,N1(C(c2cccc(OC)n2)=O)CCC2CCN(C(=O)Cc3sccc3Cl)C2C1 41141,CCCC(CNC(=O)Cn1cc(CNCC2(OC)CC2)nn1)OC 41142,C(=O)(CC(F)(F)C(F)F)NC(CN(C(CCCCC#C)=O)C)(C)C 41143,C12(C(c3ccno3)CC)CC(NC(=O)C(C)=C3CN(C(C4(O)CCOC4)=O)C3)(C1)C2 41144,C1(NC(C(C)SCC)=O)CC2CC1CN(C(c1cc(C#N)cc(C)n1)=O)C2 41145,C1(COC(Cc2c(C)c[nH]c2-c2ccccc2)=O)CC2(CCC2)C(=O)O1 41146,c1(C(=O)NC2CN(C(C3(O)C(C)(C)C3)=O)CC(F)C2)cc(F)c(F)cc1F 41147,C1(CNC(=O)C(O)C2CC2)CC2CCC1N2C(c1cccc(C2CC(F)(F)C2)c1)=O 41148,C12(C(=O)NCC3N(C(=O)CCOC4CCC4)CCCC3)CC3CC(CC1C3)C2 41149,CC(C)CC(C(=O)NCCN=[N+]=[N-])NC(C1CCCC1F)=O 41150,C(=O)(CC(O)CNC(=O)C(CC)OCC)N1CC(N(CC=C)C)C1 41151,CC1CC(C(N2CCC(C(C)(C)CNC(=O)CSC(F)(F)F)CC2)=O)CCO1 41152,C1(C(N(CCNC(C(CC=C)C)=O)Cc2ccccc2)=O)CCC(C)=C(C)C1 41153,C12(C(C)C)CCC(NC(=O)NC(C)CCc3ccc(C(F)(F)F)cc3)C1C2 41154,N1(C(C(C)=CC)=O)CCN(C(C2CC3CCC2O3)=O)C(c2ccc(F)c(F)c2)C1 41155,C=Cc1cnn(C)c1C(=O)Nc1ncc(C(c2ccc(F)cc2)O)s1 41156,C1(NCC=CCNS(C)(=O)=O)CCC(NC(c2cnc(-c3ccoc3)s2)=O)C1 41157,c1(CN(C(C)C(=O)NC2(CCNC(C3CSC3)=O)CC2)C)ccccc1 41158,S(=O)(=O)(c1cccnc1NCCCCS(C)=O)NCC(C1CCCO1)C 41159,C(=O)(C1=NOC2(CCCN(C(=O)C(O)Cc3cccc(Cl)c3)C2)C1)NCCSC 41160,Cc1cccc(NC(C2OCCC2NC(c2cnsc2C)=O)=O)c1C 41161,C(=O)(C1CCc2c[nH]nc21)N(C1CCCN(C(CC(=C=C)C)=O)C1)C 41162,c1(CC(N2CC3C(NC(CC4C(C)C4)=O)C3C2)=O)cccc2c1OC(C)(C)C2 41163,c1(OC)ncccc1C(=O)NCCN(C1CCCCC1)C(c1cc(F)n(C)n1)=O 41164,CCCCC(CNC(c1c(C(C)C)noc1C)=O)NC(=O)C(C(=O)OCC)OC 41165,Cc1cc(=NCCCOC(C)C)[nH]c(N2CCC3(CCC(C)C3)C2)n1 41166,c1(OC)cc(N)ccc1C(N1C(C2(NC(C3CCCCC3O)=O)CC2)CCC1)=O 41167,CCC(CC(=O)NC1CC(CCC(=O)NCCOC2CCCC2)C1)C1CCC1 41168,C#Cc1ccc(F)c(C(N2CCC(C3CCCCN3C(c3csnn3)=O)C2)=O)c1 41169,CCC(CCOC)C(=O)NC1C=CCN(C(=O)CCF)C1 41170,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41171,c1(COCCN2C(NC(C(=O)NCC)=O)CC2)ccccc1.C1(=O)C(OC)CN1 41172,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(c1cocn1)=O 41173,N1(C(C(C)S(N)(=O)=O)=O)CCC2CCC(NC(=O)Cc3ccon3)C1C2 41174,CC1(C)CCN(C(C2CSCC(=O)N2)=O)CC1CNC(c1cc(Br)no1)=O 41175,c1(C(N(CC(C)O)CC#C)=O)c(CNC(=O)COCC(F)F)nnn1C 41176,c1(C(=O)NCC(CC)(C)NC(=O)COCC2CCOC2=O)ccc(CO)c(Cl)c1 41177,N1(C(C)=O)CCC2(CCC(CNC(=O)CNC(N)=O)O2)CC1 41178,Cc1ccc(F)c(C(N2CCCC2CN(C)C(C2CCS(=O)(=O)N2)=O)=O)c1F 41179,C(=O)(C1OCCc2c(O)cccc21)N1C2CC(CN(C(CC(=O)NC)=O)C2)C1 41180,C1(CNC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(=O)CNC(N)=O)CC1 41181,C#CC1(NC2CCn3nccc3C2)CC2(CCCC2)C1 41182,c1(NC(CCOCCCC)=O)cccc(NC(c2cc(Br)sn2)=O)c1 41183,Cc1ncc2n1CCN(C(C1CCCC1CNC(C1(C3CC3)CC(=O)C1)=O)=O)C2 41184,C(=O)(CC(C)(C)CCOC)N1CCC(O)(CNC(C(CC=C)NC(C)=O)=O)C1 41185,C1(C(N2CC(C(C)(C)O)(CNC(C=NOC)=O)C2)=O)CCN(C)S1(=O)=O 41186,N1(C(C2(CC)CCC2)=O)CCCC(C2CC2NC(c2ccccc2O)=O)C1 41187,CN1CC=C(CC(=O)N2CCCOC(CNC3Cc4ccncc4C3)C2)CC1 41188,C12(C(=O)NC3C(NC(C(C)C4CCOC4)=O)CCC3)CCC(C(C)=O)(CC1)CC2 41189,N1(C(c2cc(C)sn2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1C 41190,C(CCCCC(C)C)NC(CN(CCOC)C(C1CCCC(F)C1)=O)=O 41191,Cc1cc(C)c(C(=O)NC(C)CN2CCN(C(=O)C(F)(F)CC3CC3)CC2)o1 41192,C1(N(C(=O)CC2(O)CCOCC2)C)CC2CCC(C1)N2C(=O)C1=C(Cl)CC1 41193,C1(NC(c2cc(CNC(CC3C(C)(C)C3)=O)on2)=O)CCC(C#N)CC1 41194,Cc1ccc(F)c(CC(N2CC(CC(=O)NCc3nncn3C)C3(CC3)C2)=O)c1 41195,N1(C(c2cn(CCNC(c3cn(CC=C)nc3)=O)nc2)=O)CCC(C)(CO)C1 41196,C1(NCc2c(C(C)C)ccc(C(=O)OC)c2)CC2(CCOCC2)CCO1 41197,CC(N=[N+]=[N-])C(=O)NC(C(=O)NCC1COCCOC1)C1CCOC1 41198,CCCCCCC(CC)C(=O)N1CC(OC)C(NC(=O)C(C)(C)F)C1 41199,C1(C(=O)NC2(CCC(=O)NC3(CCCCO)CC3)CCC2)COCOC1 41200,CCC(CNC(c1cn(C)nc1OCC(F)F)=O)(CC)NC(=O)C(F)=C(C)C 41201,N1(C(C2C(c3n(C)cnn3)CC2)=O)CCCC2(CC=CCC2)C1 41202,Cc1ncc(C(=O)NCCC(C)(C)NC(C2COCCN2C)=O)cn1 41203,C12(CNC(CNC(C)=O)=O)CC1CN(C(=O)CCc1ccc[nH]1)C2 41204,c1(C(N(C(C)CC(N2CCC(C)(C)C2C)=O)C)=O)cccc2cc[nH]c12 41205,C1(CNC(CC2(C=C)CC2)=O)CC(OC)CN1C(C1CCC(=O)N1)=O 41206,c12cccc(c1)NC(=O)CCCO2.C(C(=O)NC1(CO)CC1)SCC=C 41207,N1(C(C(CC#C)O)=O)CC2CCC(CNC(c3nc(C4CC4)sc3C)=O)(C2)C1 41208,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COc2cncc(Cl)n2)CC12CCC2 41209,CC1C(C(=O)NCC2CC2NC(=O)CCc2csnn2)=NOC1C 41210,C1(C(=O)NC(CCCNC(C(CC)c2ccccc2)=O)C)CC12CCCCCC2 41211,CCC(CC)C(=O)NC(C1(NC(=O)COc2ccccc2COC)CC1)C 41212,c1(CN(C(C)C)CCO)cccc(NC(=O)C(=O)NS(C)(=O)=O)c1 41213,c1(C(C)C)cc(CC(=O)N(CCC(C)NC(=O)C(=O)Nc2ncc[nH]2)CCO)on1 41214,C1(=O)CC(CCCC(C)C)N1.C1(N(C(=O)OC)C)CC1(C)C.C(C)(C)(C)O 41215,CC1(NC(C2(CO)CC(O)C2)=O)CCCOC1.C1(=O)C(F)CC2CN1C2 41216,N1(C(C=CC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(c2ccccc2)CC1 41217,c1(C(=O)NC(CNC(C(C)NC(=O)NC)=O)C2CC2)cn2ccc(F)cc2n1 41218,CCCCC(C)C(=O)N1CCC(CN(c2cccc(Cl)c2Cl)C)C1 41219,N1(C(C)C)CCN(C(C23CC(CN2C(=O)C(C2CCC(=O)N2)C)C3)=O)C(C)C1 41220,N1(C(C=CCC)=O)CC(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC1C 41221,C1(C(=O)OCC)CN(C(C2COCCN2CCCO)=O)C2(CCC2)CO1 41222,N1(C(C=C)=O)CCC2C(CCN2C(c2ccn3c(O)nnc3c2)=O)C1 41223,N1(C(C(C)=CC(=O)O)=O)CCCC1c1cn(CCN(C)C(N)=O)nn1 41224,C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(=O)CSCCN(C)C)CCC1 41225,N1(C(c2ccc(C(C)=O)s2)=O)CC2CC(NC(c3oncc3C)=O)CC1C2 41226,c1(CCC)ccc(C(=O)OC)cc1NC(=O)NC1CCN(C)CC1 41227,C(=O)(C(C)(O)Cn1ccccc1=O)NCCCNC(c1ccc(OC)s1)=O 41228,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(C2(c3noc(C)n3)CC2)=O)C1 41229,C1(O)(CNC(=O)Cc2cc(CO)ccc2Cl)CCN(C(c2cc(F)c[nH]2)=O)CC1 41230,C1(NC(c2c(Cl)ccc(OC)n2)=O)CN(Cc2nc(Cl)cs2)CC(F)(F)C1 41231,C(=O)(C(C)NC=O)NCCCN(C(=O)CC1CC(OC)C1)CCC 41232,C=CCC(C(=O)N1CCN(C(=O)CCC(=C)Cl)CC12CC2)C(C)C 41233,Cn1cc(NC2CS(=O)(=O)CC2NC(=O)CC(O)c2ccccc2)c(C#N)nc1=O 41234,c1(C(=O)NCC2COCCN2C(=O)C(O)C2CC2)nc[nH]c2nccc1-2 41235,C1(NC(Cc2c(C)nccc2)=O)COCCN(C(c2c(Cl)nn(C)c2C)=O)C1 41236,C1(CNC2CC(CC(=O)O)OCC2)CC2CC(=O)C1C2 41237,C1(C(=O)NC(CC#C)C)CSCCN1C(=O)CCCC1CC1C 41238,CC1CC(NC(=O)CC2(Oc3ccccc3)CC2)CN1C(c1cc(F)c[nH]1)=O 41239,c1(C(=O)NCC(CN(C(c2cnc(C)n2C)=O)C)(C)C)cnc2ccc(F)cn12 41240,c1(OC)cc(Cl)cc(Cl)c1-c1ccc(CNC(c2cnc(O)cc2OC)=O)nc1 41241,C(=O)(CCCCC1CC1)N(CCCCNC(CCOCC#C)=O)CC 41242,CC1(C)CC(C(=O)NCC2CCC3CC23)CN(C(c2cnc[nH]c2=N)=O)C1 41243,c1(C(=O)NC(C2CN(C(CCCC)=O)C2)C)c(Br)cncc1OC 41244,c1(CNC(C2C(OC(C)=O)C2)=O)ccnc(C(=O)NCCC2CCOC(C)C2)c1 41245,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41246,Cn1ccc(=NC(=O)C2CC(O)CN2C(c2ccn(C(C)(C)C)n2)=O)[nH]1 41247,C1(CNCC(C(=O)OCC)Cc2ccc(F)cc2)C2CCC(C2)C1C 41248,c1(OC)ccc(F)c(F)c1CC(N1CCN(Cc2cc(CO)nn2C)CC1C)=O 41249,C(=O)(CCCCC(N)=O)N1CCC(N(CCOC)CC)CC1.c1(N)cnc(OC)nc1 41250,Cn1cc(C(=O)NCC2(NC(C3CCC(F)C3)=O)CCCC2)c(=O)[nH]1 41251,c1(CC)nnc2n1CCCC2C(=O)N1CCC(NC(=O)CNS(N)(=O)=O)C(O)C1 41252,CCCCC(O)CCC(=O)OCC1CN(C)CC(C)O1 41253,C1(C)(C(=O)Nc2nccn2C)CC2CCC(C1)S2.C(C1CN1)OC 41254,CCCCCCCCNC(C1C(C(N2CCC(N(C)C)C2C)=O)C1(C)C)=O 41255,C(=O)(CC1=CCN(C)CC1)NC(CCC)CC(=O)N1CCC(C)(NC(=O)OC)C1 41256,C1(C#N)(CC(=O)NCCOCCCNC(c2ccc(CC)cn2)=O)CCCCC1 41257,C1(NC(=O)C=CC=C(Cl)Cl)CC2C(NC(c3ccc(Br)s3)=O)C2C1 41258,N(C1CCCn2cnnc21)C(c1cc(CNC(C(c2cnn(C)c2)C)=O)no1)=O 41259,C1(CC(=O)N(CCCNC(Cc2cncc(C)c2)=O)CCO)COCC(C)(C)O1 41260,CCCC(CCC)C(=O)NCC(C)NC(C1CC=C(C(C)C)CC1)=O 41261,N1(C(C2(C)CCC2)=O)CC2CS(=O)(=O)CC2(CNC(=O)Cc2cc(Cl)cs2)C1 41262,C1(NC(COCCC#C)=O)CCCN(C(=O)CC(CC#N)c2ccccc2)CC1 41263,CCC(CCCO)NC(C1CCCCC1NC(C1(CF)CCOCC1)=O)=O 41264,C1(CNC(C2C(NC(C3CSC3)=O)CCCC2)=O)CCCCC1(F)F 41265,c12ccc(cc1)C1(CCC1)N2.CC1(CN)CC(C(=O)O)C1 41266,c1(CNC(C=CCC)=O)ccsc1C(=O)NC(C)COC(F)(F)F 41267,c1(CC(=O)NC2(CN(C(=O)C(CC3CCCC3)C3CC3)C)CC2)cccc(F)c1F 41268,C=CC1CCCCN1C(C12CCC(OC)C1C2)=O.C1(=O)CC(C)(C)CN1 41269,c1(CNC(C2(C(=O)OC)CC2)=O)ccc(CNC(C2CC3(CSC3)C2)=O)nc1 41270,c1(NC(C(N2CCC(c3cn(C)nc3)C(C)(C)C2)=O)=O)cccc2c1CC(=O)N2 41271,C12(CNC(C3CC(C)C3)=O)CCCCC1N(C(=O)C=C1CCN(C)C1)CCC2 41272,c1(C(N(C2CN(C(Cc3c(C)cco3)=O)C2)C)=O)cnn(CC(C)C)c1C 41273,n1(CCOC)cc(C(=O)NCC(C)(C2CCC2)NC(=O)COCC(C)(C)C)nn1 41274,S(=O)(=O)(c1c(Cl)ccc(C)c1F)NCC(COCC)O 41275,CC1(F)CCN(C(C2CN(C(=O)Cc3ccccc3F)CC2F)=O)C1 41276,C1(C(=O)NC(C(=O)NC(c2ccccn2)CCC)C2CC2)CC(=O)CCO1 41277,CCC(CC(=O)NCC(CC)(CC)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41278,CC1CC(C(=O)NCC2(CNC(=O)C(Cl)=CCl)CC(F)(F)C2)CCO1 41279,C#CCC(C)C(=O)NCC(C)(C)CN(C(=O)C(c1ccccc1)SC)C 41280,C1(C(N2CC(O)(CNC(C3(C)CC=CC3)=O)C2)=O)CCC(OCCF)CC1 41281,CC(CCCc1ccccc1)C(=O)N1CC(NC(=O)CCn2cnnn2)C1 41282,c1(C(C)NC(=O)COC2CCN(C(=O)C=C3CCN(C)C3)C2)cccnc1 41283,CCC(C(=O)NC1CCN(C(c2oc(C)nc2C)=O)CC1O)C(F)(F)F 41284,CC1(C)CCN(CCNC(=O)C(c2ccoc2)NC(=O)CSC2CC2)C1 41285,c1(NC(N2C(CC)CC(C(=O)OC)CC2)=O)cc2c(s1)CCC(C)(C)C2 41286,c1(C(=O)NC2CC(NC(C3(C)ON=C(C)C3)=O)C2)ccc(N)c(C)c1Br 41287,Cc1ccc(F)cc1C(N1CC(CNC(c2nc(C3CC3)cs2)=O)C(O)C1)=O 41288,N1(C(c2c(C)nc(CCC(=O)ON)s2)=O)CC(CN)C(C2CC2)C1 41289,c1(CNC(COCC)=O)nnc2n1CCN(C(c1cscc1OC)=O)C2 41290,C(=O)(C(C)(C)C(C)O)NCC1(OC)CN(C(c2c(Cl)c(CC)nn2C)=O)C1 41291,c1(NC2CN(C(C(C(C)C)SC)=O)CC2(C)C)ncnc(N(C)C)c1[N+](=O)[O-] 41292,C1(CC)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(CC)n2ccnc2)C1 41293,N1(C(C2C(OCC)C2)=O)Cc2ccccc2OC2(CCC2)C1 41294,C(=O)(CCCCC1CC1)NCC(C=C)O.C12(CC1)C(=O)N2C 41295,c1(C(N2CC3CN(C(c4ccon4)=O)CC32)=O)cn2cccc(Br)c2n1 41296,C12(CNC(c3ccc(N)cc3)=O)CCC(NC(c3ncsc3C3CC3)=O)(CO1)C2 41297,n1(CCC)cc(C(=O)NC2CC(O)CN(C(c3cc(C)[nH]c3C)=O)C2)ccc1=O 41298,N1(C(=O)OC(C)(C)C)CCN(C(c2cncc3[nH]ccc23)=O)CC1(C)C 41299,c1(NCC)ccc(C)cc1C(=O)NCc1cccc(CNC(=O)C(C)N(C)C)c1 41300,CCC(C)C(O)C(=O)NC1(C(=O)N(C(C)CC(F)(F)F)C)CCCCC1 41301,N1(C(C2(C)C=CCC2)=O)CCCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 41302,N1(C(C(C)CBr)=O)CCC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 41303,c12c(cccc1F)S2.c1(N(CC)CC)ccc(=O)n(C)c1.c12csc(n1)NC2 41304,CC12CC(C(=O)NC(CCCNC(=O)C(F)n3ccnc3)c3cccs3)(C1)C2 41305,N1(C(C(=O)NC(c2ccc(Cl)cc2)C(F)(F)F)=O)CC2CCC1CO2 41306,c1(C(=O)NC2(C3N(C(C(CC)O)=O)CCC3)CC2)cc(F)c(Cl)c([N+](=O)[O-])c1 41307,c1(-c2cc(C(=O)NCC(C)N(C(C(C)=C(CC)C)=O)CC)no2)ccc(Cl)cc1 41308,CC1(CNC(=O)COC2CCOC2)CCCN(C(=O)CSC2CCCC2)C1 41309,c1(CN2C(C(N3CCCOCC3)=O)CC(=C)C2)cccc(Cl)c1F 41310,CC1(CNC(c2ncn3c2CCC3)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 41311,C1CCCC(N=c2[nH]c(=NCC3CCCSCC3)c3ccc(C)cc3[nH]2)CC1 41312,c1(CC)ccc(C(=O)NCCC2(NC(=O)CSC)CCCCCC2)c(F)c1 41313,c1(C(C(=O)NCCOC)N(CC(C2CCC2)OC)C)csc(Cl)c1 41314,N1(C(C)CNC(=O)CCn2cccc2)CCN(C(=O)CCc2ncc[nH]2)CC1 41315,C(c1ccc(C(N)=O)cc1)=CC(=O)NCC(C)N(C(C(C)OCC)=O)C 41316,C1(C(N(C)Cc2ccsc2)=O)CCN(C(=O)CCOC2CCC2)O1 41317,Cc1[nH]c(C)c(C(=O)NC2CC(C)(NC(c3ccn(C(F)(F)F)n3)=O)C2)c1C 41318,CN1CC(CNC(=O)C(N2CCCC2C(F)F)=O)C(O)C1 41319,C12(C(N3CC(C)C(NC(C4(F)CCCCC4C)=O)CC3)=O)C3CC(CC13)C2(F)F 41320,N(C(=NCCOc1ccc(Cl)cn1)NCC1CCC(=O)N1)CC1N(CC)CC1 41321,N1(C(C23N(C(CS(CC)=O)=O)CC(C2)C3)=O)CC2C(C1)C2(F)F 41322,c1(C(=O)NCC2CCC(C(=O)OC)CC2)nc(C)ccc1C.C12CC1CNC2=O 41323,C1(NC(=O)COc2cccnc2)CN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1F 41324,C1(OC)(CNC(c2cncc(C3CC3)c2)=O)CCN(C(C2CC(SC)C2)=O)C1 41325,C1(C#N)(C(=O)NCCc2c(C(=O)NCC3(O)CCN(C)C3)c[nH]n2)CCOCC1 41326,c1(C(=O)NCCCN(C(=O)C(c2ccccc2)C2CC2)CCO)cc(Cl)ccn1 41327,c1(C(N)=O)cc(CC(=O)NCCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41328,c1(CC)c(C(=O)NC2CCCC2NC(c2conc2C(F)(F)F)=O)cccc1C 41329,CCCC(C)CC(=O)NCC1CCCN(C(c2cc(CC)ccc2C)=O)C1 41330,CCCC(C)CN=c1cccc(S(=O)(=O)NCCn2ccnc2C(C)C)[nH]1 41331,c1(OC)ccc(C)c(OC)c1C(=O)N(CC(C)CNC(=O)CCOC)C 41332,C12(C(=O)OCC)CCN(N3C(CCC(=O)O)C[SH](c4ccccc4)C3)CC1C2 41333,C1(C(N(C(C=C)C)C)=O)C(CNC(=O)CC2CC=CCC2)C1(C)C 41334,c1(CC)[nH]nc(C(=O)N(CCCNC(=O)C(O)C(C)SC)C2CC2)c1Cl 41335,C=CCC(C)C(=O)N1CCC(N(C(=O)CC(c2ccccc2Cl)C)C)CC1 41336,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41337,c1(C(N2C(CNC(c3ccc(Br)nc3Br)=O)COCC2)=O)cc2cccnn2n1 41338,C(=O)(C(CC(C)C)NC1(C(C)(C)O)CC1)N(CC(COC)O)C 41339,C1(C)(CC)CC(NC(=O)CCc2csnn2)CN1C(=O)CN(C1CCCC1)C 41340,N1(C(COCC#C)=O)CC2CCC1CN2C(C1CCS(=O)(=O)CC1)=O 41341,c1(C(=O)NCC23CC(NC(CCCOCC)=O)(C2)C3)ccc(C(F)(F)F)c(N)c1 41342,N1(C(C(CC)=CC)=O)CCCC12CCN(C(C1CCN(C3CC3)C1=O)=O)C2 41343,CN1N=C(CC(=O)N2C3CCCC2CC(NC(=O)C(C)(C)CF)C3)CC1=O 41344,N1(C(C2CC(C(C)(C)C)C2)=O)CCC(CO)(NC(=O)CC2CCC(=O)N2)C1 41345,N1(CN(c2nccc(OC)c2)C)CCN(C(=O)C(c2cccnc2)O)CC1=O 41346,CCCCCCC(F)C(=O)NC1(C)CCN(CCOc2c(C)cccc2C)C1=O 41347,C(CN=C(NCC1CCCCO1)N(C)Cc1ccc(Cl)s1)c1n(C(C)C)nnn1 41348,c1(CC)c(-c2nc(C3CCCN(C(=O)NCC(C)C)C3)no2)c(C)nn1C 41349,c1(NC(CCCNCC(CC)OCCC)=O)c([N+](=O)[O-])c(C)nn1C(C)C 41350,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41351,CC1CC(C(=O)NCCC2(NC(C3(C)CCCCCC3)=O)CC2)CC(C)C1 41352,C(CO)(CCCCNC(c1ccnc(Cl)c1O)=O)NC(C1CC(C)C1)=O 41353,CC1CN(C(c2cnn(CC(F)(F)F)c2)=O)CC1CCNC(c1c[nH]c(=N)o1)=O 41354,c1(C(C)SCCOC)nc(-c2ccc(OC)cn2)nn1CCCO 41355,Cn1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cc(Cl)c1Cl 41356,N1(C(C(C)CC2CCC2)=O)CCOCC(C(=O)NC2CN(C)CC2(F)F)C1 41357,c1(OCC)ccc(C(C)NC(=O)Nc2ccccn2)c(OCCOC)c1 41358,CC(C)CC(O)C(C)C(=O)N1CCC1C(N1CCN(CC(F)(F)F)C(=O)C1)=O 41359,C1(C(N2CCN(CCCNC(=O)CCOCC(F)F)CC2)=O)C2CCCCCC12 41360,N1(C(c2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(O)CC3CCOCC3)CC12 41361,Cn1ncnc1C(=O)NCC(N1CC(NC(=O)CCc2ccccc2)C1)=O 41362,CC#CCC(C(=O)NCC#Cc1ccco1)NC(C1CN2CCN1CC2)=O 41363,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41364,c1(SCc2n(CC(=O)OC)ncc2)nc(N(C)C)nc(N)n1 41365,c1(CN(c2conc2CC2CCCCC2)C(C)=O)cc(C)oc1C.c1(CN)cccs1 41366,N1(C(c2cc(COC(C)(C)C)on2)=O)CC(NC(c2ccc(=O)oc2)=O)C(O)C1 41367,C1(O)(CNC(C(C)C2CCC2)=O)CCCN(C(c2nc(Cl)cs2)=O)C1 41368,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cc(Br)sn1)=O 41369,C1(NC(CCSC)=O)CCN(CCCNC(C2SCCS2)=O)C1C 41370,C(CN=c1nc(-c2cc(Cl)cc(Cl)c2)[nH]s1)C1(NC(c2ncc(C(F)F)s2)=O)CC1 41371,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41372,c1(C(=O)OCC)cccc(C(N2CC(N3CCOCC3)C2)C)n1 41373,N1(C(C(C)=C(CC)C)=O)CCC2CN(C(C3(C)CCCS3)=O)CC12 41374,CCC(C)(CNC(=O)Cn1cc(CN(C(C)CO)C)nn1)C(N)=O 41375,c1(C(=O)NCC(CNC(=O)CNC(c2ccncc2)=O)O)cncc([N+](=O)[O-])c1 41376,C1(C(=O)NC2C=CC(CNC(=O)CCCC3CCCO3)C2)CC2C=CC1O2 41377,C(=O)(C(C(=O)NCC1CCN1C(c1cc(O)n(CC)n1)=O)C(C)C)OCC 41378,C(=O)(CC(C)CNC(=O)Cc1cccnc1)N(C1CCOC1)CC 41379,Cn1c(C(N2C3CN(C(=O)CCc4ccc(F)nc4)CC23)=O)cc2ccccc12 41380,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41381,c1(C(=O)NCc2nc(CNC(c3ccc(C)s3)=O)sc2)ccn2nncc2c1 41382,c1(CNCC(CNC(C(C)SC)=O)C)cncc(C)c1 41383,c1(C(N2CC(CC(C)NC(C3CCCCC3C)=O)C2)=O)cn(C)c2ccccc12 41384,C1(F)(NC(C=CC)=O)CCN(C(=O)CCNC(=O)Nc2ccccc2)C1 41385,CC(=O)CCCC(=O)NC1C2CN(C(c3cc(C)c(C)s3)=O)CC12 41386,C(=O)(C(F)(F)CCC=C)N1CCC(N(C(=O)C(CC(C)C)C2CCC2)CC)C(O)C1 41387,CC(C(=O)NCCc1ccc(Cn2cc(COC)nn2)c(Cl)c1)P(C)(C)=O 41388,Cc1ccccc1CCC(=O)NCCN(C(C1(Br)C(C)C1C)=O)C1CC1 41389,CC(C)(C)CC(O)C(=O)NC(Cc1cc[nH]n1)C(N1CCCCCC1)=O 41390,c1(C(=O)NCC(CC)NC(=O)C(C(C)C)SC)cn(-c2cccc(Cl)c2)nc1C 41391,CCC1CC(=O)N(C)CCC(C)N1.C1(C(C)C)(NC(=O)COC)COC1 41392,c1(CCC(=O)NCC2N(C(C3(CCC)CC3)=O)CCCC2)n[nH]c2ccccc12 41393,C1(C)(C(N(CC(C(=O)OC)(C)C)C2CC2)=O)CCC(=O)NC1.C1CC=CC1 41394,N1(C(C2N(CC)CC2)=O)CC(CO)C2(C1)CN(C(c1ccc(C(F)(F)F)o1)=O)C2 41395,C1(C(=O)NC(C)C2CCC2)(CO)CCN(C(=O)C=CC2CCCN2C)C1 41396,C(=O)(CC(C)(F)F)N(CCNC(C1C(C)C1C)=O)C(C)C 41397,Cn1cc(C2=CCN(S(=O)(=O)C(F)(F)F)CC2)cn1 41398,N1(C(C2(N=[N+]=[N-])CC2)=O)CCC2(NC(c3ncccc3CO)=O)CCCC12 41399,c1(C(=O)NC(Cn2cc(C=CC)nn2)C)cc(C)ccc1C(F)(F)F 41400,c1(C(=O)NCC2(NC(C#CC3(CC)CC3)=O)CCCC2)cccc2ccnn12 41401,CCC(C)CCN(C)C(C1CCN1C(=O)COCC(=O)NC)=O 41402,N1(C(C(C(CC)C)N)=O)CC(NC(c2cc(C#N)c[nH]2)=O)C2(COC2)C1 41403,n1(CC(=O)NC2CCCC(C(=O)NCc3cncs3)C2)cc2ccccc2n1 41404,C(=O)(C(CC)CC(C)C)NCC1CC(OC)CN1Cc1ccc(C(C)=O)cc1F 41405,C1(C(=O)NCC(CNC(CN(C(C)=O)C)=O)C)CCCN(Cc2ccccc2)C1 41406,N1(C(CC(CC)NC(N)=O)=O)C2CCC1CN(C(=O)CC1CCN(C)CC1)CC2 41407,Cc1nn(C)c(Cl)c1CC(N1CCN(CC(C)NC(c2csnn2)=O)CC1)=O 41408,CCC(C(=O)N1CCC(NC(C2CCCN2CC)=O)C1C)C(C)(C)CC 41409,c1(CC(=O)N(C)CC2N(C(C(C)=C(CC)C)=O)CCC2)cc(Cl)sc1Cl 41410,c1(C(=O)NC(CNC(C(CC)(CC)OC)=O)COC)nccc2nn[nH]c12 41411,c1(C(C)NC(C(F)OC)=O)nc(C(=O)N(C)CC2CCN(C(C)C)C2)co1 41412,CCN=C(NCc1ccc(Cc2ccoc2)cc1)NC.C1(C(=O)OC)CCCC(F)C1 41413,CC(O)(C(=O)N1CC(O)(CCNC(=O)C(C2CCCC2)N(C)C)C1)c1ccccc1 41414,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41415,c1(C(=O)NCC(C)N(C(=O)CO)C)cc[nH]c1C1CCCC1 41416,CCCCC(COC)N=c1[nH]c(=NCC(N)CCO)[nH]c2cc(C)ccc12 41417,CC(C)CC(CNC(=O)CCC1COC(C)(C)O1)NC(=O)CCN1CCCCC1 41418,C12(CCNC(C=CCN(C)C)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41419,CS(=O)(=O)C1CCCN(S(=O)(=O)Cc2nc(O)nc(O)n2)C1 41420,N1(C(COCCCC#C)=O)CCCC(O)(CCNC(c2c(Cl)csc2Cl)=O)C1 41421,Cc1c[nH]c(C(=O)NC(C)(CNC(=O)CCc2cc[nH]n2)Cn2cccn2)c1 41422,c1(C(N2CCSC(CO)C2)=O)ncc(Sc2ccccc2)cn1 41423,C(=O)(C(C)(C)C(N)=O)NC(C1CCN(C(=O)CCS(C)(=O)=O)CC1)C(C)C 41424,N1(C(C(CC)CN(C)C)=O)CCC(C(=O)N(C)CC2(C)CCC2)C12CC2 41425,c1(CN2CC3C(C(Nc4c(C)cccc4F)=O)(C3)C2)ccc(O)c(C#N)c1 41426,c1(C(=O)NC2COC3(C2)CN(C(=O)COCCF)C3)cc2cc(F)ccc2s1 41427,CC1(CNC(=O)Cc2ccsc2)CCCN1C(=O)C(O)c1ccsc1 41428,CC1CCCC=C1C(=O)N(C(C)CN(C)C(c1cc2ncccc2[nH]1)=O)C 41429,C(=O)(CCCC(C)(F)F)NCCC1OCCN(C(c2c(C)csc2)=O)C1 41430,C1(NC(C(CC)=CC)=O)CCC2CN(C(=O)CC(C)C(=O)OC)CC2C1 41431,N1(C(CSCCC)=O)CCOC2CN(C(c3ccsc3-n3cnnn3)=O)CC12 41432,C1(CC(=O)NCc2cc(C)[nH]c2)COCCN1C(C1(C(N)=O)CC1)=O 41433,Cc1ncc(Cl)c(C(N2CCC(O)(C(C)NC(C3CCCC34CC4)=O)CC2)=O)n1 41434,N1(C(C=C(CC)CC)=O)CCCCC1CNC(c1cnc(C)cn1)=O 41435,N1(C(CCc2onc(C)n2)=O)CCC2(CO)CN(C(=O)C3=CC(C)(C)C3)CC2C1 41436,N1(C(C2(N(C(CSCC)=O)C)CC2)=O)CC(O)(CC(C)C)C1 41437,N1(C(CCc2cn(C)nn2)=O)CCCC(C2(C(N3CCCCCC3)=O)N=N2)C1 41438,N1(C(C(CC)CN(C)C)=O)C2CCC1CN(C(c1ccc(C(O)CF)cc1)=O)C2 41439,CC(C)CCC(C)NC(C1CCCCN1C(C1(NC(N)=O)CC1)=O)=O 41440,C1(CNC(C2(C(C)C)CC2)=O)CN(C(C23CC(C2)C(C)O3)=O)CCC1C(F)(F)F 41441,C1(CNC(C(C=C)O)=O)CCN(C(CCNC(=O)CC2CCCCO2)=O)C12CC2 41442,C(=O)(C(C)(CC(C)C)NC(=O)C(C(C)(C)O)c1ccccc1)OC 41443,N1(CCC(=O)NC2(C)CC(NC(C(CC)F)=O)C2)CCN(CC)CC1 41444,c1(CNC(C2COCCN2C(=O)CCCCC2CC2)=O)ccc(F)cc1 41445,c1(CN2CC3C(CNC(c4cnc(CC(C)C)s4)=O)C3C2)cc2nc[nH]c2cn1 41446,C12OC(CC1C)OC2OC.C1(OC)CCC(NC(=O)NCCC)N1C1CC1.C1CC1 41447,C1(CC)CN(C(C2COCCOC2)=O)CCN1C(C12CCCC1(C(N)=O)C2)=O 41448,c1(C(=O)NCC(CNC(C(CCCC)N(C)C)=O)F)oc2ccccc2c1CO 41449,c1(C(=O)NCCC(=C)CNC(=O)C(O)C(C)CC)ccc(Cl)c(OC)c1 41450,C1(C(=O)NCC2(C)CCC(NC(c3ccc(C)nc3)=O)C2)CCCCNC1=O 41451,c1(C(=O)NCCN(C(C(CC)Cc2ccccc2)=O)CC)cc2cccnn2n1 41452,N1(C(CCNC(=O)OCC)=O)CCN(C(=O)CSc2ccc(Cl)c(F)c2)CC1C 41453,N1(C(CC(C)F)=O)CC2CCOC2(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41454,C1(NC(c2cc3oc(Br)cc3[nH]2)=O)CC2CN(C(c3cccs3)=O)CC2C1 41455,c1(-c2c(C(N3CCCC(C(=O)O)C3)=O)c[nH]c2)ccc(-c2ccncn2)cc1 41456,CN1CCC(F)(C(=O)NCCC(O)CNC(c2ccccn2)=O)CC1 41457,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41458,C(=O)(C(C)C(CC)CC)N1CCCC(CNC(CN(CCC)C)=O)C1C1CC1 41459,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41460,C(=O)(C1=CC(O)C(NC(=O)C=C(C2CC2)C2CC2)C1)Nc1cc(C)sc1 41461,C(=O)(CC(F)(F)CS(C)(=O)=O)NCC1N(C(c2c(C)nccn2)=O)CCC1 41462,C(CCC(=O)NC1CC1CNC(=O)CSc1n[nH]c(C)n1)OCC=C 41463,c1(OC)ccnc(C(C(=O)NCCCC2CC2)N(C2CCCCC2C)C)c1C 41464,N1(C(C2N(CC)CCC2)=O)CCC(C(=O)NC(CC2CC2)COC)C1(C)C 41465,c1(OC)cc(SC)ccc1C(N1CC(O)(C(C)NC(c2nccnc2C)=O)C1)=O 41466,C1(CC(=O)N(C2CCCN(C(c3sc(C)nc3C)=O)C2)CC)CC2(CCC2)CO1 41467,Cc1cccc(CN(C(=O)C(C)c2ccco2)C(=O)NC2CCSC2)c1 41468,c1(C(N2CC(C(C)NC(C(C)NS(C)(=O)=O)=O)C2)=O)ccn(CO)c(=O)c1 41469,c1(C(N2CC(C(C(=O)C(O)CCl)=O)C2)=O)nc2ccc(F)cn2n1.O 41470,C1(C(=O)NC(C2CCN(C(c3cnc4sccn34)=O)C2)(C)C)CCS(=O)(=O)CC1 41471,C1(C(=O)NCCCOC)CCN1C(=O)C=CC(C)C 41472,C1(C(=O)Oc2nc(CCOCC)sc2)CCCC(CC)C1.C(CN(C)C=O)OC 41473,C(=O)(CCCC(=O)NCCOC1CC1(F)F)OCCN1CCC(C(C)C)C1 41474,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41475,Cc1nc2cc(C(=O)NC3CCCN(C(=O)CCCc4cncs4)C3)ccc2o1 41476,c1(C(N(C2CCN(C(CCC(C)SC)=O)CC2)C)=O)ccc(F)c(F)c1F 41477,C1(CC)CCC(C(=O)NC23CC(C(=O)NCC(F)(F)CO)(C2)C3)CC1 41478,C1(C(=O)NCCCOC=C)CN(Cc2cc(Br)c(Br)s2)CCS1 41479,c1(C2(C)CC2)ccc([N+](=O)[O-])c(NC(CC2CCC2)CO)n1 41480,c1(C(N2CC(NC(CS(CCC)(=O)=O)=O)(COC)C2)=O)ccc(C=NOC)cc1 41481,C1(N(C(C(C(C)C)NC(Cc2cn(CC)nc2)=O)=O)C)CCOC(C)(C)C1 41482,C1(C(N2CC3C(CNC(c4c(CC)[nH]cc4)=O)(C3)C2)=O)CC(C2CC2)=NO1 41483,C(C(=O)NC12CC(NC(c3csc(Cl)c3)=O)(C1)C2)(C(C)(C)C)NC(C)=O 41484,c1(C(=O)NCC2C(C)CCN2C(=O)C(F)=CCCF)cnn2c1OCC2 41485,CCC(CC)CC(=O)NCCC1CN(C(=O)CCc2ccc(C#N)cc2)C1 41486,N1(C(CN(CCO)C(C2OCC(=O)C2)=O)=O)CCCC(OCCO)C1 41487,N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(=O)CS(=O)CC)CC2(CC2)C1 41488,C=CCCCCCC(=O)N(C(C)C(=O)NC1CCCC(CC)C1)C 41489,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41490,N1(C(CC2(C)CCC2)=O)CC2C(NC(c3occc3F)=O)C2C1 41491,CCCCCC(F)C(=O)NCC(O)CC(N1c2ccccc2CC1C)=O 41492,CCC(CN=c1[nH]c(N2CCN(C)C(=O)C2)nc2ccccc12)ON(C)C1CC1 41493,c1(NCC)cccc(C(=O)NC2CCCCC2CNC(C2CCCCN2C)=O)c1 41494,CC1(C)Cc2occc2CN1C(c1ccc(Cl)cc1I)C(=O)NC1CCOC1 41495,c1(CC(=O)NCC2C(NC(C3C(C(C)=O)C3(C)C)=O)C2)ccc(S(N)(=O)=O)cc1 41496,C1(C(=O)NC(C(C(C)C)NC(CN(C2CC2)CC)=O)C)CC2(C1)CC21CCC1 41497,c1(CNC(c2ccc(C(N3CCC(O)(CO)C(O)C3)=O)o2)=O)c(F)ccc(Cl)c1F 41498,C1(NC(=O)OCC(C)(C)C)CCCC(C(=O)OC)CC1.c12cn(nn1)C2 41499,C(CC(=O)NNC(=O)C(N)CC1COCCO1)OCCCCC 41500,C(=O)(C(C)N(OC)C(=O)C=CCNC(=O)C(C)NC1CC1)N(C)CC 41501,N1(C(c2nccc(C)c2)=O)CC(C)(C)CC1CNC(=O)Cn1cc(Cl)cn1 41502,N1(C(CC=C)=O)CCC(O)(CN(C)C(C2CN(C3CCOC3)C2)=O)C1 41503,c1(CNC(CC)C2(C(C)C)N=N2)cc(-c2ccccc2)n[nH]1 41504,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCC(CCNC(CC=CC)=O)C1 41505,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41506,C1(c2cccs2)(C(N2C(CNC(c3c(CC)nns3)=O)C=CC2)=O)CCOCC1 41507,Cc1ncncc1C(N1CCC(F)(CNC(c2ccccc2)=O)C1)=O 41508,C1(N(C)C(c2ccnc(OC(F)F)c2)=O)CCCN(C(=O)C(O)C(F)F)C1 41509,C#Cc1ccc(OC)c(C(=O)NCC2(C)CC2C)c1 41510,C(=O)(C(CCNC(=O)CCC1CCOC1)OC)NCC1(CCC=C)CC1 41511,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41512,N1(C(c2ccc(Nc3c(CC#C)cccc3)cc2)=O)CC(C)C2CCCCC12 41513,CC1(CCNC(=O)Cn2cnnn2)CCN(C(c2ncncc2F)=O)CC1 41514,CC1CC(CO)CN(C(=O)C(Cc2ccoc2)NC(c2ncccc2Cl)=O)C1 41515,C(=O)(C(C)CC(N)=O)N1CCC(CN(C(CCCCC)=O)C)CC1 41516,CCN=c1ccc(C(=O)OC(CC)C(=O)Nc2ccc(Cl)cc2)c[nH]1 41517,c1(NC(CC(C)N(C)C(C2CCCN2C)=O)=O)ccc2cnccc2c1 41518,CC1CN(C)CCN1C(=O)C(O)CNC(c1ccc(Cl)cn1)=O 41519,c1(C(=O)NCC(=O)NCCO)coc(CCCNC(=O)C(O)Cn2cncn2)c1 41520,C1(C(N(CCN(C(C2CC(F)C2)=O)CC)CC)=O)CCCN(C)C1 41521,c1(C(N(CCCCN(C(C(CC)O)=O)C)C)=O)c(C)sc(C)c1C#N 41522,c1(C(=O)NCC2CCC(CNC(c3c(C)scc3)=O)CC2)cnn2ccccc12 41523,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41524,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41525,Cc1cncc(CC(=O)NCCC2CCCN2C(C2COCCO2)=O)c1 41526,N1(C(CC(CC)C)=O)CC2CN(C(c3cccc(C)c3Br)=O)CCC12 41527,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41528,C(=O)(CCC(C)NC(=O)C(O)C(C)C)NCc1occ(C)n1 41529,CCC(C)C(C)CNC(=O)CC1CCC(NC(c2cnn(C(F)F)c2)=O)CC1 41530,C(=O)(C#CC1CC1)NC(CN(C(c1nc(CC)oc1)=O)C)(C)C 41531,C1(NC(=O)Cc2cnsc2)CC12CC(NC(c1csc(-c3cnccn3)n1)=O)C2 41532,N1(C(Cn2c(C)ncc2)=O)CCCC(C)C1CCNC(c1cncc(C(N)=O)c1)=O 41533,C1(NC(CSCC(=O)OC)=O)CN(C(=O)C(F)(F)C2(O)CCC2)CC1O 41534,C1(NC(C(COC)N(C)C)=O)CC(OC)CN(C(=O)CSS(C)(=O)=O)C1 41535,c1(OC)cccc2c(C(=O)NCC(O)CCNC(=O)C=Cc3cscn3)c[nH]c12 41536,c1cc(OC)cc(NC(N2C(CC)COCC2)=O)c1.C1(N(C)C)(CO)CCNCC1 41537,C1(NC(c2cccc(F)c2F)=O)CN(C(c2csnc2Cl)=O)CCC1CO 41538,N1(C(c2nnn(C(C)C)n2)=O)CC2(CCC2NC(=O)C(C)(C)COC(C)(C)C)C1 41539,C(=O)(C(F)(F)C(F)F)N1C(C(C)NC(C(c2ccc(C)cc2)(F)F)=O)CCCC1 41540,c1(C(C(C)NC(=O)CC2CC2C(F)(F)F)NC(c2cc[nH]n2)=O)ccccc1 41541,c1(C(=O)NCC2C(NC(C(C)C(C)(F)F)=O)C2)cc2sc(Br)cc2[nH]1 41542,N1(C(CCNC(C)=O)=O)CCC2(CC1)CCN(CC(O)C1CC1)CC2 41543,C1(C(F)(F)F)(NC(=O)NCC2OCCC(NC(=O)CO)C2)CC2C=CC1CC2 41544,CC1OC2(CNC(C3CC3F)=O)CC1(NC(c1nccc(F)c1Cl)=O)C2 41545,N1CC2CN(c3ccccc3)CC2C1.CC1CC(c2ccccc2)CCN1CCSC 41546,N1(C(C2CC(C)(F)C2)=O)CC(CNC(c2nnc(O)nc2O)=O)C2CCCCC12 41547,C1(NC(CC=CC=C)=O)CCC2CN(C(=O)CCn3c(C)csc3=O)CC2C1 41548,CC1=NOC(CC(=O)NC2(C(=O)NCc3csc(C)n3)CC(O)C2)C1 41549,Cc1csc(C)c1C(=O)NC(C)C=CC(=O)NCCc1ncccc1F 41550,c1(C(N2CC3CC2CS3)C(=O)NCCOC)noc2c(Cl)cccc12 41551,C(CN=c1[nH]c(=NCc2cccc(Cl)c2Br)[nH]c2c1COCC2)N(C)C 41552,C(=O)(C(C#N)(CC)CC)NCCC1(OC)CN(C(C2CC(C(C)C)=NO2)=O)C1 41553,C1(OC)CC(NC(C2CC(F)(F)C2)=O)CN(C(C2CCN(C3CC3)C2=O)=O)C1 41554,CC1CCCC(C)N(C(C2CC3CCC(C2)N3C(c2ccncc2Cl)=O)=O)C1 41555,C(=O)(C#CC1CCOC1)NCCC(C(=O)NC1(C(=O)OCC)CC1C)C 41556,C1(C(N(CCC(C)NC(C(CC)=CC)=O)C)=O)CCCCC1C(F)(F)F 41557,Cc1ccc2occ(C(=O)NC3CC(C)(NC(=O)C4=CC5CCCC45)C3)c2c1 41558,Cc1nc(C)c(C(=O)N(C2CCN(C(c3cc(-c4ccco4)cs3)=O)C2)C)s1 41559,C(=O)(C(C(C)(C)C)C1CCC1)N(CCCCCC)CCNC(=O)C(C)S(C)(=O)=O 41560,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CN(C(=O)CC(F)(F)Cl)C)C1 41561,O=C(N=c1[nH]oc2cc(Cl)ccc12)C1CCN(C(=O)Cc2cccc(Br)c2)CC1 41562,C1(NC(C(C2CCOCC2)OCC)=O)CC2C(NC(=O)Cn3cncn3)C2C1 41563,N1(C(CNC(C=C)=O)=O)CCCC(CC(=O)NCCc2ccnc(O)c2)C1 41564,C1(N(CCCCC)CCC(=O)NC)CCN(C(=O)C(F)C(C)C)CC1 41565,Cc1cccnc1C(=O)NC1CCCCC1CNC(C1(CC2CC2)CCC1)=O 41566,C1(N)CS(=O)(=O)C2CN(C(=O)CC3CC3)CC12.c12cccc(c1)CC(=O)N2.NC=O 41567,c1(CCNC(N(C(C)CO)C)=O)cc2ncc(Br)cn2n1 41568,CCC(C)C(O)C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(CC)(CC)CO 41569,C(=O)(CCCCC(=O)c1ccc(C)cc1)NC1(C)CCCN(C(C(C)OC)=O)C1 41570,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)NCCC)CC1CCC)=O 41571,c1(CN(C)CCN(C(=O)C(=O)NC2CCCC2)C)ccnn1C1CC1 41572,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(CC)nn1 41573,CCCCC(C)CCC(=O)N1C(C(=O)NCCOC2CCC2)CCC1C(C)C 41574,c1(CC)cnn(CC(=O)NCC(C)N(C)NC(C2CC2C(=O)OC)=O)c1 41575,N1(C(=O)C=CCn2cncn2)CC2CC(C(N3CCSCC3CO)=O)CC2C1 41576,C1(C(=O)NC(Cn2cc(COC(C)C)nn2)C)CCC2(CC1)NC(=O)N(C)C2=O 41577,c1(SCC=C)ccc(C(=O)N(C(C)CNC(C2CC2CCC)=O)C)cc1 41578,c1(C(N2CCCC(C(C)NC(=O)C(F)F)C2)=O)ccc(F)c(F)c1 41579,C(c1ccc(Cl)s1)=CC(N1CCC(CC2CCN(C(CSCC)=O)CC2)CC1)=O 41580,N1(C(c2ccnn2CC(F)F)C(=O)NC(C)C)CC2CC(O)C(O)CC2C1 41581,N1(C(C=CC(C)(C)C)=O)CCC(C)(NC(=O)Cc2cc[nH]n2)CC1 41582,CC(F)(F)C(C)(C)C(=O)N1CC(NC(c2cc(Br)ccn2)=O)C(O)C1 41583,c1(SC)ccc(C(=O)NC2CC(CCNC(C3CC(C)(C)C3)=O)C2)cc1 41584,N1(C(C(C)Cc2ccc(O)cc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)C2 41585,C(=O)(C(C)COC)NC(CC)(C)C.C1=CC(=O)NC1(C)C 41586,N1(C(CSc2cc(C)c(Br)cc2C)=O)CCN(S(N)(=O)=O)CC12CCCCC2 41587,N1(C(CC2(N(C(Cn3nnc(C)n3)=O)C)CC2)=O)CCOC(C)C1 41588,C1(CN(C(C)C)C(c2cocn2)=O)CCCN1C(=O)CCCc1ncco1 41589,c1(C(=O)NC(CCN(C(c2c(C)ncs2)=O)C)C(C)C)ncnc(O)c1Cl 41590,C#CCC(C)(C)C(=O)NCc1cc(C(=O)N(C2CCC2)C2CC2)co1 41591,C1(C(=O)OC)CCC(CNC(CC2(C)CCOC2)C(=O)NCc2ccccc2)O1 41592,N1(C(CSSC)=O)CC(CNC(=O)COCC(C)C)OC2(CCC2)C1 41593,c1(-c2n(C(C3(C)CC3)C)nc(-c3ccnn3C)n2)nsc2cc(Br)ccc12 41594,C12(CC(=O)N(C)CC3CCNC(=O)C3)CCC1CN(C(=O)Cc1cn[nH]c1)C2 41595,Cc1cccc(CC(=O)NCC(C)(C)NC(c2cnn(C3CC3)c2C)=O)c1 41596,c1(C(=O)NC2CCCN(C(C(CCSC)O)=O)C2)ccnc(C)c1O 41597,N1(C(COCCC#C)=O)CC2CC(NC(c3nc(C(F)(F)F)oc3C)=O)C1C2 41598,c1(C(=O)NC2C(NC(c3cc4scnc4[nH]3)=O)C2)cccc2ccnc(O)c12 41599,CC1CN(C(c2ccc(CO)s2)=O)CC1(C)C(=O)NC1CCN(C)C1=O 41600,Cc1scc(C(=O)NCC(C)N(C)C(c2csc(CC(F)F)n2)=O)c1C 41601,C1(C(N(CCC(N2CCC(OCC#C)C2)=O)C)=O)CC12CCC(C)(C)CC2 41602,CC1(CO)CCN(C(C23CCC(CC2)C3)C(=O)NCCc2cccs2)CCO1 41603,N1(C(C(COCC)C)=O)CCC(CNC(=O)CCc2n[nH]c(=N)s2)(COC)CC1 41604,C(=O)(CCCCC(N)=O)NC1CCC(C)(CNCC2(CO)CC(F)(F)C2)CC1 41605,CCCC(CC)C(C(=O)NCCCOC)N(C1CCN(C2CCNC2=O)CC1)C 41606,N1(C(C(CC)=CCCC)=O)CCC2(C=C(C(=O)NC(C)C(=O)N3CCCC3)C2)C1 41607,C#CC1(C(=O)NCC2(C)CCCN(C(C3(C)CCC(=O)NC3)=O)C2)CCOCC1 41608,N1(C(CNC(=O)C(=O)Nc2cc(F)c(F)c(F)c2)=O)CC2C3C=CC(C3)C2C1 41609,C1(C(=O)OCC)(C(=O)NCCNC(=O)CNC(=O)CC2CC2F)CC(O)C1 41610,N1(C(C(CC)=CC)=O)CC2CN(C(=O)CCC(=O)Nc3ccccn3)CC2C1 41611,Cc1cc(C(N2CCCC(NC(=O)C(C)(C)OC(C)C)CC2)=O)c(F)cc1F 41612,CCC(C)CC(=O)C(=O)NC(CC(=O)NCC1OCCC1(C)C)C(C)C 41613,N1(C(C=C(C)C(C)(C)C)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41614,C(CCCC(C)(C)C(=O)NNC(=O)C1CC1)NC(CCCCC#C)=O 41615,Cc1cnnc(O)c1C(=O)NCc1nc(C(=O)NCCCc2nncs2)co1 41616,Nc1cc(-c2cn(CC3CCCN(C(=O)CCN4CCOCC4)C3)nn2)ccn1 41617,C1(N(C(C(C)Cc2ccccc2)=O)C)CCN(C(c2cncn2C)=O)CC1C 41618,c1(C(C(N2CCC(CCNC(c3c(SC)snn3)=O)C2)=O)C)ccc(O)cc1 41619,Cc1cc(-n2nc(-c3ccco3)nc2CCc2nc(O)n[nH]2)cc(Br)c1 41620,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41621,c1(C(N2C(C(=O)Nc3nnc(Br)s3)CC(C)C2)=O)cc(F)c(Cl)c(F)c1 41622,CC(C)CC(O)CNC(C1(C)CCCN1C(=O)C1CC1)=O 41623,C1(CNC(c2cnn(C3CCC3)c2)=O)CCCN(C(=O)CC2CC3CC3C2)CC1 41624,C1(C(=O)NC(C)(CO)C2CCC2)CCN(C(C2CCCCS2)=O)C1 41625,N1(C(CSCC)=O)CCC2CN(C=O)CC2C1.c1(C(=O)OC(C)(C)C)ccc(C)nn1 41626,C(=O)(C(F)C1=CCCCC1)NC(CC)(CNC(=O)C=CC=C(Cl)Cl)CC 41627,C12(COC)CCC(C(=O)NC3COCC3NC(c3cnsc3C)=O)(CC1)CO2 41628,c1(C(=O)OC(COCC)COC)c[nH]c(=NC2CC2)cn1 41629,c1(C(C(=O)OCC)NC(=O)CC2CC=CCN2C)ccc(Br)cc1 41630,N1(C(C23CC(C)C2C3)=O)CCCN(C(=O)Cc2ccc(O)c(F)c2)CC1 41631,C(C(C(=O)N(CC(O)CN(C(=O)CC1CSC(C)O1)C)C)N(C)C)OC(C)C 41632,N1(C(C2C(C)C2C)=O)CC2CCCC(NC(c3ccc(CO)c(Cl)c3)=O)C2C1 41633,CC(C)C#CC(=O)NCCN(CC(C)O)C(=O)Cn1cccnc1=O 41634,C1(C(=O)NC2COCC(C(=O)NCCC3CCCCC3O)C2)CCCC12CCC2 41635,C1(NC(C2N(CC)CC2)=O)CCC(O)CN(C(c2cn(C)nc2OC)=O)C1 41636,N1(C(c2ccc(N)cc2O)=O)CCCC2CCN(C(C3(F)CCCCC3)=O)CC12 41637,C1(C)(C(=O)NCCCN(C(=O)C(O)CC(C)C)CC)CCCC(F)(F)C1 41638,N1(C(C2C3CN(C)CC32)=O)CCC(C(=O)NC2(C)CCC2)C12CC2 41639,C1(C(=O)NC(C(=O)OCC)CO)CC(C)CCN1C(C1CC2(CCC2O)C1)=O 41640,N1(C(c2cn(C)nn2)=O)CC2C(C(=O)N(C3CCCC3)Cc3ccccc3)C2C1 41641,c1(C(=O)NCCN(C(CC2(OC)CCC2)=O)CC(C)O)cc2scc(C)c2[nH]1 41642,C(=O)(C1CCc2cccnc21)NCC1(C)CCN(C(=O)COC2CCOCC2)C1 41643,CC(C)CC(F)C(=O)N(C)CC1COCCN1C(=O)Cc1cncnc1 41644,N1(C(CC(C)Oc2ccccc2C2CCC2)=O)CC(NC(N)=O)CC2(CC2)C1 41645,CC(C)CCCC(=O)N1CCN(C(=O)C(CO)N(C)C)CC1CCO 41646,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(C3CCCC3)n2)=O)C1 41647,c1(OC)ccc(N(C2CC23CCNCC3)C(=O)NCC(C)(C)F)c2ccccc12 41648,N1(C(C(COC)C)=O)CC2(CCN(C(=O)C=Cc3cocn3)CC2)C1C(C)C 41649,C1(C(=O)NCC(Cc2ccccc2)NC(c2cc[nH]n2)=O)CCC=CCC1 41650,C1(CNC(c2cc(OCC)n[nH]2)=O)CC2(CC2)CN1C(=O)CC1CC(C)C1 41651,N1(C(c2cnc(OC)s2)=O)CCC(NC(=O)CCn2ccnn2)C(O)C1 41652,C(C(=O)NC(C(=O)NC(c1nc[nH]n1)(C)C)C1CCC1)(C(C)C)OCC 41653,c1(C(N(C2CCN(C(=O)CC3CCCO3)C2)C)=O)ccc2cnnc(O)c2c1 41654,c1(-c2nc(C(CC)C)nn2-c2c3c(nn2C)CCC3)cc2c(O)cccc2o1 41655,C#CC(C)(C)C(=O)N1CC(=O)CC1CN1CCC(CC)C1 41656,c1(C(=O)NC2CC(C)(NC(CC(C)(C)OC)=O)C2)ccc(S(=O)(=O)N(C)C)o1 41657,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41658,c1(C(=O)N(C2(c3ccc(C4C(C)=C4)cc3)CC2)C2CC2)cn2c(n1)CCC(C)C2 41659,c1(CNC(CCC=C(C)C)=O)cccc(NC(=O)C(F)(F)c2ccnn2C)c1 41660,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)c3cccnc3)C1C2 41661,N1(C(c2cnc(C)s2)=O)CC(NC(C2(C)COC2)=O)CC(O)C1 41662,c1(C(=O)NC(CNC(CCc2n(C)ccc2)=O)C2CCC2)coc2ccccc12 41663,N1(C(C2CCCC(C)C2)=O)CC2(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCC1CC2 41664,C12(C(N3C(CNC(C4C(OCC)C4C)=O)CC3)=O)CC(C)(C1)OC2C 41665,c1(OC)ccc(OCCC(=O)N2CC(C(C)NC(=O)CC=CC(C)(C)C)C2)cc1 41666,N1(C(C(C2CN(C(c3cc(N)ccn3)=O)C2)OC)=O)CCC(N2CCC2)CC1 41667,c1(C(N2CC(F)CC(NC(=O)CC3CC(C4CC4)C3)C2)=O)cc2ncccc2o1 41668,C(=O)(C(CC(C)C)NC(=O)Cc1sc(O)nc1O)NCCNC(=O)NCC 41669,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41670,N1(C(C(CCC)C)=O)CCC2(C1)CN(C(C1CCCN1c1cnccn1)=O)C2 41671,C1(C(=O)NC(c2cccnc2O)C)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41672,C1(CC(=O)N(C2CC(C(=O)N)C2)C)(CC2C(C)CCO2)CCCCC1.N(C)C 41673,c1(CC)nccnc1C(N1CCN(CCNC(=O)C(O)Cc2ccccn2)CC1)=O 41674,C1(CC)CN(C(C2(O)CC2(C)C)=O)CCC1NC(c1ccc(SC)s1)=O 41675,c1(C(=O)NCC2(NCc3ccncc3)COC2)cccc2nc[nH]c12 41676,C(=O)(CC(C)CC(=O)N1CCCN(C(c2ncc(Cl)cc2F)=O)CC1C)OC 41677,c1(CC(=O)NCC2CCCC2NC(=O)CNC(c2cccs2)=O)cncc(F)c1 41678,c1(OC)cccc(-c2cc(-c3n(C)nc(-c4ccsc4)n3)n[nH]2)c1.SC 41679,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41680,C12CCCCN(C1)C(=O)C1CN(C1)CC(=O)N2C.c1(CC)ccc(Cl)c(F)c1 41681,C1(NC(CC(C)c2ccco2)=O)CN(C(C2CC3(C2)CC32CC2)=O)CCC1(C)C 41682,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41683,C1(NC(=O)Nc2cc(C)c(-n3cccn3)cc2)C2Cc3ccc(Br)cc3C12 41684,c1(NC(CCC(=C)C)C)ncc(CO)cc1Cl 41685,c1(NC(COC(C)(C)CNC(=O)CC2CCCS2(=O)=O)=O)coc2c1COC2 41686,N1(C(c2sccc2F)=O)CCC(NC(C2(CO)CC(F)C2)=O)C(CO)C1 41687,c1(NCCC(=O)N(CCN(C(=O)CO)C)C)ccc(Br)c(OC)c1[N+](=O)[O-] 41688,C1(CC)CN(C(C2(CC(C)C)CCC2)=O)CCC1NC(=O)NC(=O)COC 41689,N(C1CN(C(C2CC3(CC3)CO2)=O)CCc2ccccc21)C(C(C)(C)C#N)=O 41690,Cc1nc(=NCC2CCCCN2C(c2ccnc(C3CC3)c2)=O)[nH]cc1[N+](=O)[O-] 41691,CC(CC(=O)NCc1ccnc(C(N2CCCC2(C)CO)=O)c1)CC(C)(C)C 41692,CCCC(CC)CCC(=O)NCc1cn(CCNC(=O)C(F)=CC2CC2)nn1 41693,N1(C(CCc2cc(C)on2)=O)CC(NC(=O)CCc2cccnc2F)C(F)C1 41694,c1(C(=O)NCC(C)(C)CNC(=O)C=Cc2cnc[nH]2)ccc2nc(O)sc2c1 41695,NS(=O)(=O)N1CC(C(=O)NC2CCOCC2F)C1 41696,CC(C)CC(C)CN=c1[nH]c(N2CCC(c3ncc[nH]3)C2)nc2c1CSC2 41697,C(=O)(CCC(F)(F)C(F)F)N(C)CCN(C)C(c1ncn(C)n1)=O 41698,CC1COC(C(=O)NCC(c2ccccc2)C)C1 41699,N1(C(=O)OC(C)(C)C)CCN(Cc2cn(C3C=CCCC3)nn2)C(C(N)=O)C1 41700,N1(C(c2cnc(N(C)C)s2)=O)CCN(C)C(C(=O)NC2CCNC(=O)C2)C1 41701,C1(NC(c2n(CC)ccn2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 41702,Cc1ccc2c(c1)CC(C(=O)N(C)CC1(NC(=O)CCC3CC3(C)C)CC1)O2 41703,N(C1COc2ccccc21)CC.N12CCC(c3nnnn3C(C)C)(C1)NC2=O 41704,C1(C(N(C(C=C)C)C)=O)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 41705,N1(C(CCNC(C2C(C)C2)=O)=O)C2CCC1CC(C(=O)NCC1CC13CC3)C2 41706,N1(C(CC(C)(C)SC)=O)CC2(CCN(C(=O)CC3CCCN3C)CC2)CC1C 41707,c1(NC(=O)OCc2onc(C(=O)OCC)n2)cccc(Oc2ccccc2)c1 41708,C1(NC(c2cnc(OCC)s2)=O)CCCCCC1NC(c1c[nH]nc1F)=O 41709,N1(C(CNC(=O)NC)=O)CCC(C2CC2)(CNC(c2ccc(C)n2C)=O)C1 41710,c1(CC(=O)NCC2CCC(CN(C(CC=C)=O)C)CC2)cnc2c(=O)[nH]ccn12 41711,C(CC)(C(=O)N1CC(N(C(=O)CCc2scnc2C)C)C1)=CC 41712,Cc1ccc(C(N2CC(O)CC2C(=O)N(C2CC3(CCC3)C2)C)=O)c(O)c1 41713,c12ccc(cc1)[nH]c(=O)c2=O.C1(CNC=O)CCC(NC(C(C)O)=O)C1 41714,c1(C(N(c2cc3ccccc3[nH]2)C)=O)ccc2nccn2c1 41715,N1(C(c2sc(C)c(Br)c2)=O)CCN(C(c2cn(C(C)C)nn2)=O)C(C(=O)O)C1 41716,N1(C(CNC(C2(COCC)CCC2)=O)(C)C)CCN(C(C2OCCC2C)=O)CC1 41717,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCCCCC1)=O 41718,N1(C(C(C)CN(C)C)=O)CCN(C(C2(Cn3cncn3)CC2)=O)CC1CO 41719,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 41720,Cc1cn2c(=O)c(C(=O)NCC(C3CCC3)NC(C3C(C)C3C)=O)cnc2s1 41721,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(C1CSCCS1)=O 41722,N1(C(C(=O)NC(CN(C(C(OCC)O)=O)C)(C)C)=O)CC(F)(F)C1.C(C)(=O)N 41723,c1(OC)ncc(C(=O)NCCC(C)(C)NC(c2cnn(C3CC3)c2Cl)=O)c(C)n1 41724,CC(C)CC(C)CC(=O)N1CCC=C(CNC(c2cn(C(C)C)cn2)=O)C1 41725,N1(C(C(c2c(C)noc2C)=O)=O)CC2(C1)CN(C(=O)C(C)(Cl)Cl)CCO2 41726,N1(C(CC2CCCC(C)C2)=O)CC2(CC(NC(=O)CC=CC(C)(C)C)C2)C1 41727,c1(OC)cc(N2CCC3(NC(=O)C=CBr)CCCCC23)ccc1[N+](=O)[O-] 41728,C(=O)(C1=CCC(C)CC1)N(CC(C)NC(c1c[nH]c(=NC)o1)=O)CC 41729,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCn2c(cnc2C(F)F)C1 41730,c1(NC(CC)=O)ncc(C)cc1C.C12CC1COC2=O 41731,c1(C(N(c2nccc(N(C)CCN3CCCC3)n2)C)C2CC2)cccc(Cl)c1 41732,C=CC(C)(CC)C(=O)N1CCC(CCCNC(=O)C(C)(C)OCC)C1 41733,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)n2cnnn2)CC1 41734,C1(C#N)(C(N(CCOCCN(C)C(C2(C3CC3)CCC2)=O)C)=O)CC1C(F)(F)F 41735,C1(=O)C2=C(C)NC(=O)NC2N1.N1(C(=O)OCC)CCCCC1c1cccc(Cl)c1 41736,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 41737,CC1(C)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CN(C(=O)CCC2CC2(F)F)C1 41738,c1(N2C3CC(CC(NC(C=CS(CC)(=O)=O)=O)C3)C2)nc(Cl)nc2c1cnn2C 41739,N1(C(COC(c2ccns2)C)=O)CCC(CN(C(=O)Cc2nccn2C)C)CC1 41740,C1(C(=O)NC(C(=O)OCCC)C)CC2CCC1N2C(c1cc(C(C)=O)[nH]n1)=O 41741,c1(C(CC(C)NC(=O)C(=O)NCCOc2ccccc2N)C)ccc(Cl)cc1 41742,CC(C)(CCCNC(=O)C(O)CC(N)=O)C(=O)N1CSC(CC2C(O)CC2O)C1 41743,c1(C(=O)NCC2C(C(N3C(C)(CCC)CC3)=O)CCC2)cc(C#N)[nH]c1C 41744,c1(N2CCCC(NC(N)=O)C2)nc2c(c(=NCc3ccc(Br)s3)[nH]1)COC2 41745,C1(O)(CNC(C#CCNC(C(n2cc(CO)nn2)C)=O)=O)CCCOC1 41746,c1(CCC(=O)NCC(F)F)c(C)nn(C)c1C.C1(=O)C(=O)NCC(C)N1CC 41747,N1(C(=O)NC(C(CC)OC(F)(F)F)=O)CCCC2CN(CCNC(C)(C)C)CCC12 41748,c1(COC)cccc(NC(=O)CNC(=O)NCc2csc(CO)n2)c1 41749,c1(NC(C2CCC3(CCCN3)CC2)=O)ccnc2c(Br)cc(F)cc12 41750,c1(C(=O)OCC2C(C(=O)OCCC)C2)ccc(S(C)(=O)=O)s1 41751,CC1(C)CC(NC(c2cc3ccsc3s2)=O)CN(C(=O)C=Cc2ccc(F)cc2)C1 41752,C(=O)(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccccn2)=O)C1)NC 41753,c1(C2(CSCC)OCCCN2)nnnn1CCSCCCF.OC 41754,C#CCC(CC#C)C(=O)N1CC(NC(=O)C(c2ccc(C)c(C)c2)=O)CC1C 41755,C1(NC(C(CCCC)C)=O)CC2CCC1CN2C(C1CC1c1ccoc1)=O 41756,n1(CC(=O)NC2C(CNC(C=C(CC)CC)=O)C2)cccc([N+](=O)[O-])c1=O 41757,CC1(C)CN(C(=O)CC(O)C2CCCC2)C1C1CCN(C(=O)C(O)C2CC2)CC1 41758,N1(C(C2CCCN(C(CC)=O)C2)=O)C2CCC1CC(CCN(C(=O)CSC)C)C2 41759,c1(OC)ncc(Cl)cc1C(N1CC(CCNC(C2CCC(C)(O)CC2)=O)C1)=O 41760,O=C(O)CCCCCCBr.C1(N2CCN(C=O)CC2)Cc2cccnc2C1 41761,c1(-c2c(C)csc2)cc(C(=O)Nc2c(C(C)C)cccc2C)c2[nH]ccc2c1 41762,CC1CN(C(=O)C#CC2CCC2)CCC1NC(c1c[nH]nc1C(C)(C)C)=O 41763,c1(N(CC(CN(C)OC(c2ccccc2)C2(F)CCC2)O)C)nnc(C(C)(C)C)s1 41764,c1(CC(N2CCOCC(NC(C(C(C)C)O)=O)C2)=O)ccc(C#N)cc1F 41765,c1(C(=O)NC(C(C)NC(=O)CC2CCCOCC2)CO)cnc2sccn12 41766,C1(OCc2cn(CCNC(c3c(OC)cccn3)=O)nn2)CCC(=O)NC1=O 41767,CCC(C)(CNC(=O)CCc1cccs1)NC(C1CC=CCC1)=O 41768,c1(C(=O)NC(C(=O)N(CCCC)CC)CO)cnncc1OC 41769,c1(C(=O)NC(CC)CN(C)C(c2ccc(N)cc2Cl)=O)cc(P(C)(C)=O)ccn1 41770,Nc1ccc(C(=O)NCCCOC2CCN(C(C3(F)CCOC3)=O)CC2)cc1F 41771,Cc1n[nH]cc1CCNC(=O)C(O)C1CN(C(C2CC(F)(F)C2)=O)C1 41772,CC(C)(CN=c1nc(N2CCCC(C(C)(C)C)C2)c2c([nH]1)CCC2)C(N)=O 41773,C1(CC(=O)NCCOC(C)(C)CSC(=O)CSC2CC2)CS(=O)(=O)C1 41774,C1(OC)CCn2cc(C(=O)NC3CCCC(CNC(C4(O)COC4)=O)C3)nc2C1 41775,C1(C(=O)NCCSCC(=O)NC2(CSC)CC2)CCOCC1C 41776,C(=O)(CC(C(F)F)NC(c1ccccc1Br)=O)N(CC(C(=O)OC)C)C 41777,CCCS(=O)(=O)CC(=O)NCC1CN(C(c2sc(C)c(C)c2C)=O)CC1O 41778,Cc1cccc(C)c1C(=O)NCC(=O)NCC1COCCN1C(=O)COC(F)F 41779,C1(CNC(=O)CC2CCOC2)CN(C(=O)Cc2ccc(O)c(Cl)c2)CCCO1 41780,c1(NC(C2(C)CN(C(=O)C(F)(F)C(C)(C)O)C2)=O)ccc2c(c1)CNC2=O 41781,c1(CC(=O)NCCCNC(c2scc(C(=O)OCC)c2)=O)cnn2ccccc12 41782,CC(N=c1ccnc(N(CCCn2ccnc2)CCO)[nH]1)c1cccnc1 41783,N1(C(C2(c3ccc(C)cc3)CC2)=O)CCC(NC(=O)CCCCF)C(F)C1 41784,c1(C(N2CC(NC(c3cccc(C#C)c3)=O)C(C)(C)C2)=O)ccc2occc2n1 41785,C1(NC(=O)CCCC2CCCC2)CCC12CN(C(=O)COCC1CCOC1)C2 41786,C1(CC(=O)N(CC(C)(C)CNC(c2cocc2C(N)=O)=O)C)CCCC12CC2 41787,c1(SCC(C)(C)CCNC(C2CCCC(=O)O2)=O)nnc2n1CCCCC2 41788,CC1C(CNC(=O)C#CC2CCCC2)C(C)CCN1C(=O)CSc1cccs1 41789,N1(CC(N2CCC(NCc3ccc(OC)s3)C2)=O)CCC(F)CC1 41790,C1(O)(CCNC(c2c(C)cns2)=O)CCN(C(C2CCCC(O)C2)=O)C1 41791,C12CCCCN1C(=O)C1(n3cc2nn3)CC1.C1(OC(C)C)CCCC1(C)C 41792,C1(C(N2CCC(O)(CN(C(C(C)=CC)=O)C)C2)=O)Cc2cncn2C(=O)N1 41793,C(=O)(C#CC1(CC)COC1)NCC(CC)NC(=O)C=Cc1ccccc1C 41794,C(C)(CN(C)OC(c1ccnn1Cc1ccccc1)=O)(CO)OC 41795,C1(NC(CCOC)=O)CCN(C(c2cnc(S)nc2)=O)CCC1(F)F 41796,c1(C(=O)NC(CC)CNC(=O)C=Cc2ncco2)cnc(O)n1CC 41797,C1(C)(C(=O)NCC(C)N(C(c2c(C)cccc2C)=O)C)CC(C(C)C)=NO1 41798,CC1(C)CCC(C)(C)N(c2cc(NC3CCC(CC#N)C3)ncn2)CC1 41799,N1(C(COCCOC)=O)CCC(c2nnc(C(=O)OC(=O)C3CC3)s2)CC1 41800,C1(C(N(C2CN(C(=O)CC3(C)CC3(F)F)C2)C)=O)C2CCC1(c1ccccn1)C2 41801,C1(CNC(CCC2N(C)CCC2)=O)CCCC(NC(=O)C=C(Cl)Cl)C1 41802,CCC(CC(=O)NCCc1cnc(C)cn1)N(C(=O)C(O)CSC)C 41803,C(C)(C(C)N=c1c(C#N)c[nH]c2ccccc12)NC(C1(C(=O)NC)CC1)=O 41804,c1(C(=O)OC)ccc(F)c(NC(C2CCN2Cc2c[nH]c(Br)c2)=O)c1 41805,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(=O)C(F)(F)n2ccnn2)C1 41806,c1(C(=O)NCC2(OC)CN(C(c3cc(C#N)c[nH]3)=O)C2)ccc2ccccc2n1 41807,C(C(F)(C(=O)N1CCC(N2CCC2)C1)C(C)C)NC(c1c(C)snc1)=O 41808,C1(C(=O)N(C(C)CCNC(C)(C)C)C)(NC(C)C(=O)NS(C)(=O)=O)CCCCC1 41809,c1(OCC)cncc(CC(=O)NC2CCN(C(=O)CNC(c3ccco3)=O)C2)c1 41810,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 41811,c1(C(=O)NC2(CC=C)CN(C(=O)C(O)C(C)SC)C2)c(C(C)C)cnn1C 41812,C12(CNC(=O)C=Cc3ncc[nH]3)CC(CN1C(C1CCCN1C1CC1)=O)C2 41813,CC1(C)CCC(C(N2CC(CNC(c3sccc3Cl)=O)C(C(F)(F)F)C2)=O)C1 41814,C1(CCNC(C=C(C)Cl)=O)C(C)CCCN1C(c1ccc(N)c(Cl)c1)=O 41815,C=C(C)C1OCCC1C(=O)NC1CC(CC(=O)NC2CCC3(CC3)C2)C1 41816,N1(C(C(C)OCC2CC2)=O)CCC(CNC(c2c[nH]cc(Cl)c2=O)=O)C1(C)C 41817,C1(F)(C(N(C2CCN(C(c3cnc(C(N)=O)s3)=O)CC2)CCC)=O)CCOCC1 41818,C1(CC=C)(C(=O)NC2(c3ncco3)CC2)CCN(C(=O)CCn2cnnn2)C1 41819,c1(CC2CN(NC(C3CCC(C(=O)OC)C3)=O)C2)nn(C)cc1C 41820,C(c1cc(F)cc(F)c1)=CC(N1C(CN(C(=O)C2=CCCSC2)C)CCCC1)=O 41821,Cn1cncc1CC(=O)NC1CCCC1NC(=O)C(N1CCOCC1)C1CC1 41822,C1(C(=O)NCc2scc(C)c2)C=CCCN1C(C1CC1[N+](=O)[O-])=O 41823,c1(CNC(c2c(C(C)NC(C(CSC)OC)=O)noc2)=O)ccnc(F)c1F 41824,c1(CNC(C(CSC)C)=O)cc(C(=O)NCCc2noc(=O)n2C)ccn1 41825,N1(C(C(C)NC=O)=O)CCC(F)(F)C(CNC(=O)C2=CCS(=O)(=O)C2)C1 41826,N1(C(C(CO)NC(C23CCCC2C3)=O)=O)CCCCC1C(=O)NCC 41827,c1(C(=O)NCC(CNC(C2(C#N)CC2)=O)O)nn2c(c1Br)OCCC2 41828,CCC(C)(C(=O)Nc1cccc(NC(=O)C(N2CCCCC2=O)C)c1)OC 41829,C1(CCCC2N(C(C(=O)NC)=O)CCC2)CCCCN1C(=O)C=Cc1cocn1 41830,C(=O)(C(C)(C)CF)NC(CCN(C)C(C12CSCC1C2)=O)(C)C 41831,Cn1ncnc1C(C(=O)NC1(CCO)CCCC1)NC(=O)CCC1CC1(F)F 41832,C(=O)(CC(C)C(F)(F)F)N1CCCCC(NC(c2ccc(CC)cc2)=O)C1 41833,Cc1ccoc1C(=O)N(CC(=O)NC1CCC(CO)C1)CC(C)C 41834,c1(CC(=O)NCC(CC=C)NC(=O)CCCn2ccnc2CC)cnn(C)c1C 41835,CC1(C)CN(CC(C2CCOC2)=O)CCS1=O 41836,c1(N(CCOC2CC3CCC2C3)C)nc2cc(C(=O)O)ccc2n1CCO 41837,CC(C)C(C(C)NC(c1ccsc1CO)=O)CCNC(=O)Cc1cc[nH]n1 41838,C1(C(C)NC(C2CCN(C(Cc3nc(C)[nH]n3)=O)C2)=O)CC2CCC1C2 41839,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(=O)C(C2CCCCC2)=O)C1 41840,c1(C(=O)NCC(C2CC2)NC(C2(CC=C)CC=CC2)=O)ccc(CSC)cc1 41841,C1(CNC(=O)C=Cc2ccsc2)CC(COCCO)CN1C(c1ccn(C)c1)=O 41842,C1(NC(CN(C)CCO)=O)CN(C(C2(n3ccnc3)CCCC2)=O)C2(CCC2)C1 41843,O=S(=O)(c1cccc(N2CCn3cnnc3C2)n1)NCc1nc(O)n[nH]1 41844,c1(CC(=O)NCC(C2CCCC2)NC(CCC)=O)coc2cc(Cl)ccc12 41845,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 41846,C12(CNC(c3cccc[n+]3[O-])=O)CCCC(CN1C(C1CCCCC1)=O)C2 41847,C(C(CC(C)C)C(=O)N1CCCC(CC2CCC2)C1)NC(COCCCC)=O 41848,N1(C(CSCC#C)=O)CC(C2CC2C(N2CC(N3CC(O)C3)C2)=O)C1 41849,c1(C(=O)NCC2CCN(C(C(CCC)N(C)C)=O)C2)c[nH]c2ncccc12 41850,c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)C)cc([N+](=O)[O-])oc1C 41851,C1(NC(c2snnc2C)=O)CCN(C(C2(Cl)C(C(=O)OC)C2)=O)CC1 41852,c1(C(=O)NCC(C2(O)CCN(C(CC3(OC)CC3)=O)C2)C)cncc(OC)c1C 41853,C1(NC(C(C)NS(CCC)(=O)=O)=O)CC(CNC(=O)CCC2CC(OC)C2)CC1O 41854,C1(NC(CCSCCC)=O)(CO)CCCN(C(c2cc(Cl)cnc2O)=O)C1 41855,c1(C(N2CCCC(CCNC(=O)COCC(F)(F)F)C2)=O)ccc2nsnc2c1 41856,N1(C(CC(=O)NCC)=O)CCC(OCCNC(C2CC(OCC)C2)=O)C1C1CC1 41857,C(=O)(C#CC1CC1)N1CCC(C(C)Cc2ccccc2)C1.N(S(N)(=O)=O)CC(=O)N 41858,C1(C(=O)NCCCN(C(C#CC(C)(C)O)=O)C2CC2)CC2(CCOCC2)CO1 41859,N1(C(c2c(NC)snc2C)=O)CC(NC(=O)Cn2cnccc2=O)C2(CC2)C1 41860,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 41861,c1(C(=O)NCC2C(NC(c3c(CC)ocn3)=O)CC2)c(C)nn2cccnc12 41862,Cc1ccc(Cl)c(C(C)NC(=O)OCCC(O)CF)c1 41863,c1cnnn1C.C1(COC)(CN)CC1C(=O)OC.C12CC1C(=O)N2 41864,c1(CC)ccccc1C(=O)NC(CCF)C(=O)N(CCC1CC1)CC 41865,C1(CC(=O)NC2C(NC(=O)CNC(=O)Cn3cncn3)C2)CN2CCN1CC2 41866,C1(CNC(C=CCN(CC#C)C)=O)CCCCCN1C(=O)CC(C)(C)COC 41867,C(=O)(CCCCCCC)NC(CSCC)C(=O)N(CC(O)CO)CCO 41868,C=CC1(C(=O)NC(c2ccccc2F)(C)CNC(C2CC(C)C2)=O)CCCCC1 41869,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 41870,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsc2CO)=O)C1 41871,c1(C(=O)NCC2(OC)CN(c3nnc(C)s3)C2)ccc2cccnc2n1 41872,N1(c2nc(OCC)c(Cl)cn2)CCC2(NC(c3nsnc3O)=O)CCCCCC12 41873,Cc1ccc(C(=O)NCCCCCC(=O)NCC2CCC=CCC2)nc1C 41874,N1(C(C=C(CC)C)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC12CC2 41875,O=C1NCc2ccc(NS(=O)(=O)c3ccccc3N3CC(F)(F)C3)cc21 41876,c1(C(N(C2CC(NC(c3cc(C)c(C)s3)=O)C2)C)=O)coc2c(F)c(Cl)ccc12 41877,N1(C(c2cn(CC)nc2)=O)CCC2CCCC12C(=O)NC(C)Cc1nncn1C 41878,C(=O)(C1=CCCCC1C)NC1C(CNC(c2c(C)nc(C3C(COCC)C3)s2)=O)C1 41879,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 41880,C(=O)(C(C#N)(CC)CC)NCCC(C)NC(C1(CCC)CC1)=O 41881,c1(CN(C(C(=O)NCC)=O)CCc2nn[nH]n2)ccccc1 41882,C1(C(N2CC(C(=O)Nc3cnc(O)c(Br)c3)C2)=O)CCC2(CC1)OCCO2 41883,c1(CC(=O)N(C2CCN(C(c3cocc3C(N)=O)=O)CC2)C)ccccc1Cl 41884,CC1CCCCC1C(=O)NC(C1CN(C(C2(C)CC(F)C2)=O)C1)C 41885,Cc1nc(CNC(=O)C(c2cn(C)nn2)NC(=O)CC2(O)CCC2)cc(O)n1 41886,c1(C(C)C)ncccc1C(=O)NC1CC(CNC(=O)COCC2CCOC2)C1(C)C 41887,N1(CC(=O)NC)CCC(F)(F)C2(CCOC2)C1.c12ccccc1NC2=O 41888,c1(C(N(C2CCC(NC(=O)CCc3ccco3)C2)C)=O)ccnnc1O 41889,c1(Cn2c(N(CCCC)C)nnc2C(O)COCC)ccc2cc(C)sc2c1 41890,c1(C(F)(F)F)ccc2occ(-c3nc(C(F)F)nn3CCCN3CCOCC3)c2c1 41891,N1(C(c2c(C)csc2)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CCC(O)C1 41892,CC1(C(=O)NCc2cccc(NC(=O)Cc3ccccc3O)c2)CC(C2CC2)=NO1 41893,Cc1c(C(N2CCC(NC(c3ccc(N)cc3)=O)C2)=O)c(=O)oc2ccccc12 41894,C1(OC)CN(C(=O)CC(O)CNC(C2CC23CCCCC3)=O)CC12CC2 41895,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 41896,N1(C(C2OCC(C)(C)C2)=O)CC2(CC2)CC1CNC(c1cc2n(n1)CCC2)=O 41897,C1(NC(C(C(=O)NC)(C)C)=O)CCN(C(C2CC3C=CC2C32CC2)=O)CC(O)C1 41898,c1(C(N2C(CNC(C(C(C)(C)C)O)=O)C3CCC2C3)=O)sc2ncccc2c1N 41899,CC1(C)CNc2ccc(C(=O)NCC(F)CO)cc21 41900,C1(OC)CCCC(CC(=O)OC2CNCC2c2ccccc2Cl)C1 41901,C1(NC(CCc2cc(C)on2)=O)CCOC(C(=O)NCc2ccc(Cl)cn2)C1 41902,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)C1CCC1 41903,C1(OC)CS(=O)(=O)CC1NC(=O)NC(c1ccc(Cl)nc1)C 41904,c1(CC(N2CC(CNC(C3C4CS(=O)(=O)CC34)=O)C2)=O)cnc2cccnn12 41905,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(=O)Nc2c(OC)cnnc2OC)C(C)C1 41906,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccnc(O)c1)=O 41907,C(CC)(CCC(=O)NCC1(C)CSC(C)=N1)NC(CCC#C)=O 41908,C1(NC(C2(CF)CCN(C(COCC(C)C)=O)C2)=O)CCCCC1C#N 41909,C(N=c1[nH]c(=NCC(C)C#N)[nH]c2c1SCC2)c1cccc(C)c1C 41910,c1(OC)c(NC(=O)C=C2CCN(Cc3c(Cl)ccnc3Br)CC2)cccc1C#N 41911,C1(C)(C(N(CCC(C)NC(C2(C(C)(C)O)CCC2)=O)C)=O)CC(C(C)(C)C)=NO1 41912,C(c1ccccc1F)=CCC(=O)N(C1CN(C(C2(CC#C)CC2)=O)CC1F)C 41913,CCC(C)(C)C(=O)C(=O)N1CC(O)CCC1C(N1CC2C=CC2C1)=O 41914,c1(C(=O)NC2C(NC(Cc3c(OC)ccnc3)=O)C2)cnc2onc(CC)c2c1 41915,c1(C(=O)NC2CC(O)CN(C(C3CCOC3)=O)C2)ccc2c(c1)CCCS2(=O)=O 41916,C1(OC)CC(NC(=O)C2=C(Cl)CC2)C12CCN(C(=O)CC1(O)CCCCC1)CC2 41917,N1(C(C2(C(=O)OC)CCCC2)=O)CC(C2(NC(C3(F)CC3)=O)CC2)C1 41918,CON1CCC(C(N2CC(c3cn(-c4ccc(Cl)cn4)nn3)C2)=O)CC1 41919,C1(CC(=O)NCCCCN(C)C(C2CNC(=O)C2)=O)(CN(C)C)CCOCC1 41920,C1(NC(c2cc(CC)oc2C)=O)CCN(C(=O)CCOC(C)C)CC1F 41921,Cc1c(C(=O)NCCC2CC(NC(=O)C(C)c3cccs3)C2)cnn1CC(F)F 41922,N1(C(C(N2C(CCOC)CCCC2)=O)=O)CCCc2ccc(F)cc21 41923,C1(CC)CC(C)N1C(=O)CCc1cncn1C 41924,N1(C(c2nc(COC)sc2)=O)CCC(C2CCCN(C(=O)CC3(C)CC3)C2)CC1 41925,C(=O)(C(C)C(C)(C)C)NC(C)CNC(c1cn(C)nc1C(C)(F)F)=O 41926,N1(C2(NC(=O)NCc3cnn(CC(F)F)n3)CC2)CCCCC1=O 41927,Cc1cn2c(CN3CCN(c4cccc(C)c4F)CC3)c(C)nc2s1.C(=O)(N)NC 41928,c1(C(=O)NC2(C)CCN(c3nc(SC)nc(Cl)c3)C2)cc2cc(C)ccc2cn1 41929,c1(NC(C(C2CN(C(=O)CCC3(C#N)CCC3)C2)OC)=O)cnc2ncnn2c1 41930,C1(NC(=O)C(c2ccccc2)=O)CC(NC(c2ccccc2Br)=O)C12CCC2 41931,N1(CN(C(c2ccc(N3CCCC(CC)C3)nc2)=O)O)CCCc2ccccc21 41932,Cc1cc(C(=O)N(C2CC(NC(=O)CNC(=O)CNC(N)=O)C2)C)ncn1 41933,C1(C(=O)N(CCC(=O)NC(C)CC(F)(F)F)C)(CC)CNC(=O)C1 41934,c1(OC)ccc(C(C)NCC2CC(F)(F)C2(C)C)c(OC)c1 41935,C(c1cc(C)ccc1OC)=CC(=O)NCC(CC)NC(c1occc1C)=O 41936,c1(C(=O)NC(c2cccc(Cl)c2)CNC(CN(C2CC2)CC)=O)nc(C)nn1C 41937,N1(C(c2cccc(CC(C)C)c2)=O)CCC(F)C(NC(C2CCC2CF)=O)C1 41938,CCCC(O)CC(=O)NC(CNC(C1CCCS1)=O)(CC)CC 41939,c1(C(N2CC(NC(=O)C(F)(F)C3CCCC3)C3CC23)=O)ccc(OC(F)F)cc1 41940,CC(C)CCCCC(=O)NC1(CNC(=O)C(C)C2CC2)CCCC1 41941,Nc1c(Cl)cc(C(=O)NCC2(F)CC(NC(C3CC3[N+](=O)[O-])=O)C2)cc1[N+](=O)[O-] 41942,N1(C(CCc2c(C)scc2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1C 41943,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(=O)CC23CCC(CC2)C3(C)C)[nH]1 41944,c12csc(n1)CNC2=O.n1(C(C)C(=O)O)cc(CC2CC2)nn1 41945,C1(NC(C2(SC)CC2)=O)CC(NC(=O)C(C)(C)Cc2ccc(O)cc2)C12CCC2 41946,N1(C(c2ccn(COC)c2C)=O)CC2CC1CN(C(C1CCCCO1)=O)C2 41947,CN1CCOC(C(N2CCC(OCCNC(=O)C(C)(C)CC3CC3)CC2)=O)C1=O 41948,N1(C(COCCC=C)=O)CC2CCC(NC(c3c(Cl)ccnc3F)=O)CC2C1 41949,c1(C(C(=O)N(CC(O)CN(C(=O)COCc2nc[nH]n2)C)C)OC)cnn(C)c1 41950,N1(C(CC(=O)OCC)=O)CCC(O)(C(C)CNC(c2cc(O)n(C)n2)=O)C1 41951,C(=O)(C(C1CCC1)NC(=O)C=CC(F)F)NCCCOC 41952,n1(CCC)cc(Cl)c(C(=O)NCCN(C(=O)CC(c2ccccc2F)C)CC)n1 41953,C1(O)(C(C)C)CCN(C(=O)CCCCCN(C(=O)CCCC#N)C)CC1 41954,C(CCCCCCCO)=CC(=O)NCC1C(NC(CCCCOC)=O)CCC1 41955,CC1C(NC(c2ccc(F)c(Cl)n2)=O)CC2CCC1N2C(C1(O)CCOC1)=O 41956,c1(C(=O)NCC(CCC)NC(C2CCCC2F)=O)cc(C)c(C)o1 41957,c1(OC)cc(F)c(F)cc1S(=O)(=O)N1CC(C)(C)CC1C 41958,C(CC(C)C)(C(=O)N(CCO)CCOC)NC(C(C)=CC1CC1)=O.N(C)C 41959,N1(C(c2c(CNC(CC(C=C)CCC)=O)c[nH]n2)=O)CCc2cc(C)ccc21 41960,c1(C(=O)NC2CCC(CC(=O)N(C)CCN(C)C)CC2)cccc(OCC2CC2)n1 41961,C1(NC(c2c(C)nsc2N)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 41962,N1(C(C2C3CN(C(C(CC)(C)COC)=O)C2C3)=O)CC(C)N(C)C(C)C1 41963,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 41964,C1(C(N(C(C=C)C2CC2)C)=O)CCCC(NC(c2cccc(C)c2O)=O)CC1 41965,N1(C(C(C2CC2)SC)=O)CC2CC(NC(c3coc4ccccc34)=O)CC1C2 41966,c1(NC(CC(CC#C)N)=O)cc2c(cc1Cl)NC(=O)C2 41967,N1(C(C(=O)NC(C)C)=O)CC2CCCC2(CNC(c2cc(Cl)cn2C)=O)C1 41968,CCC(O)C(F)(F)C(=O)N1CC(CNC(=O)C(CC)C2CCOCC2)(OC)C1 41969,c1(C(N(CC(C)NC(=O)CCCn2cncn2)CC)=O)c(C)cccc1C 41970,C1(O)(CNC(C(CC)(C)F)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 41971,N1(C(C=CC2(C)CCOCC2)=O)C2CCC(C2)C1C(=O)NCC1CCC(=O)N1 41972,C(CNC(=O)CCCC1CC1C)(CC(=O)NCc1cnn(C)c1O)OC 41973,C1(COC)(NC(C23CC(C)(C2)C3)=O)CCN(C(C2CC(C)(C)CO2)=O)CC1 41974,CCCC(C(=O)NCC1(C(F)F)CCN(C(c2cc(C)co2)=O)C1)C(C)C 41975,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 41976,CC1C(C)N(C(=O)Cc2ccn3nnnc3c2)CCN1C(=O)CC12COC(C)(C1)C2 41977,N1(C(c2c(CC)noc2)=O)CC(NC(=O)Cc2ccc(C)cc2)C(C)C1 41978,C1(CC(=O)NC(C(C)NC(CC2C(CC)C2)=O)CO)(CO)CCCCC1 41979,Nc1ccc(C(=O)NC(CNC(=O)C(O)C2CC2)CC(F)(F)F)c(Br)c1 41980,c1(OC)ccc(Br)c(C(N2CCC(F)(CNC(c3cccnc3O)=O)C2)=O)c1 41981,CCC(CC)C(=O)NC(COC)C(N1CCCC(O)C1)=O 41982,C12(CCNC(c3cncc(C)c3)=O)CCC1CN(C(C1CCCN1C(N)=O)=O)C2 41983,C12(C(N3CC(CC(=O)OC)C3)=O)CC1CCN2C(c1ccc(C(N)=O)o1)=O 41984,c1(-c2cnc(Sc3ccccc3C(=O)NC3CC(C)(O)C3)s2)ccc2cc[nH]c2c1 41985,C(c1sc(Cl)nc1Cl)=CC(=O)NC1CCC(NC(COC(C)C)=O)CC1 41986,N1(C(C2C(C#C)C2)=O)CCC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)(C)C1 41987,c1(C(=O)NC(CN(C(c2n(CC)ccc2)=O)CC)C)ccc2c(c1)COC2(C)C 41988,CC(C)C(CCN(C(=O)CCc1cncc(O)c1)C)NC(C1CC2CCC1O2)=O 41989,Cc1cc(C(=O)NCC2CCN2C(c2ccc(CC3CC3)cc2)=O)nc(O)n1 41990,C1(C(c2n(CC=C)nnn2)NCc2ncc(COC)[nH]2)(OC)CCCCCC1 41991,c1(NC(C2C(C(=O)NCCc3ccccc3O)C2)=O)cc2ccccc2cc1O 41992,c1(CC2CCC(CN(C(C(F)=CC)=O)Cc3cnc[nH]3)C2)nnc2ccccc2n1 41993,C1(NC(c2n(CC)ccc2)=O)CCCN(C(=O)CCc2n[nH]c(=N)s2)CC1 41994,CC(CC(=O)N(C1CC(NC(c2sc(Br)cc2F)=O)C1)C)C(F)F 41995,C1(C(C(=O)NCC(C2CC2)NC(=O)CC2(N(C)C)CC2)OC)CCOCC1 41996,C(C(=O)C(C)(O)Cc1ccccc1)N1CCCC(N(C)Cc2cccc(N)c2)C1 41997,N1(C(c2c(CC#C)con2)=O)CCC2CN(C(C3(C(=O)OCC)CC3)=O)CC2CC1 41998,C(C(N=c1ccn2nccc2[nH]1)C1CCCC1)NC(C(CCC)C(C)C)=O 41999,c1(C(=O)NC(CN(C(CCNC(=O)OC)=O)C)C)cnc(N(C)C)c(Cl)c1 42000,c1(OC)cnnc(C(=O)NC(CNC(C2(C)CC3CC3C2)=O)C(C)(C)C)c1 42001,N1(C(Cc2cnn(C)n2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C1CC1 42002,c1(C(=O)NCCCNC(C2(OC)CC(CF)C2)=O)cc(Br)c(Cl)cc1N 42003,Cc1ccnc(C)c1NC(=O)NCc1cnn(CCNC2CC2)c1 42004,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42005,c1(C(C(=O)NCCCNC)NC(=O)COCC(=O)OC)cnc(O)nc1O 42006,C(=O)(NNC(=O)C(N)C1CCCCC1)NC(c1ccnc(C)n1)C 42007,N1(C(C(=O)N(C)CCc2cn(CCF)nn2)=O)CCCC(CC2CC2)CC1 42008,c1(CCN(CC)CC)cn(C2CCC(C(=O)NS(=O)(=O)CC3(C)CCC3)C2)nn1 42009,C(=O)(C(C)S(C)(=O)=O)NCC(C)(C1CCC1)NC(Cc1cc(C)n(C)n1)=O 42010,C1(C(N2C(C3(C(=O)NCC(N(C)O)=O)CC3)CCC2)=O)CC2(CCCO2)C1 42011,c1(C(=O)NCC2(C)CCN(C(c3nc(C)oc3)=O)C2)n[nH]c2ccccc12 42012,CCS(=O)(=O)CC(C)N(CC(O)COc1cccc(C)c1C)C=O 42013,C1(NC(c2cc(CC)on2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42014,CCC(C)C(C(=O)NC1CC1)NC(C1CC1C1CCCO1)=O.c1(C)cnsc1 42015,Cn1cc(C(=O)C(N2CC(O)(C3CCCN3C(c3cnn[nH]3)=O)C2)=O)cn1 42016,CS(=O)(=O)C1CN(C(=O)C=Cc2cnccn2)CC1NC(=O)C(=O)NC1CC1 42017,c1(CSC)ccc(C(N2CCCC(NC(=O)C=C(C)C)C2)=O)cc1 42018,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42019,c1(C(=O)NCCC(CNC(C2CC3(CCC3)CO2)=O)OC)cc2cnccc2[nH]1 42020,c1(C(=O)NCC2N(C(c3c(OC)ccs3)=O)CCC2)cc(C(F)(F)F)cc(O)c1 42021,C(C1CN(C(=O)N(C)Cc2ccc(-c3ccccn3)s2)CCO1)=CC(=O)OC 42022,c1(CC(N2C(C)CC(NC(C3CN(C)C3)=O)CC2)=O)coc2cc(F)ccc12 42023,CCCCCCCC(C)NC(=O)NCCC1CCN(C(=O)OC(C)(C)C)C(C)C1 42024,N1(C(C2(NC(c3c(C)cns3)=O)CC(O)C2)=O)CC(C)C1(C)C 42025,C1(=CC(=O)N(C2CCN(C(C3CCC(C)(O)CC3)=O)C2)C)CC2CCC(C1)N2C 42026,N1(C(C)=O)CCCC1(C)C(=O)NC1(C)CC(NC(=O)C#CC2CC2)C1 42027,C1(C2CCC2)(C(=O)NCCN(C2CCCC2)C(C2CCC(C)C2)=O)CC1 42028,N1(CC(C)(C)NC(COCC(C)C)=O)CCC(NC(=O)CC2CCCO2)CC1 42029,C1(CNC(c2ccc(C)nc2)=O)CC2CCCC2C1.C12(CCC1)C(=O)N2 42030,c1(CC(=O)N(C(C(N2C(C=C)CC2)=O)c2ccco2)CC)cnn(C)c1C 42031,C1(OCC(=O)NC(C2CCCN2C(=O)C(=Cc2c[nH]cn2)F)C)CC(F)(F)C1 42032,N1(C(Cc2cc(C)sc2C)=O)CC2CCC(C1)N(C(=O)CCC(C)(C)N(C)C)C2 42033,c1(CC(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccccc1CC#N 42034,Cc1c(-c2cn(CCCC(=O)N(CC(N)=O)C)nn2)c(=O)oc2ccc(O)cc12 42035,C(=O)(CCCCCCN=[N+]=[N-])N1CCC(NC(C2CC(CC)C2)=O)(CF)C1 42036,N1(C(C2CCCC(C(=O)NOC3CCOC3)CC2)=O)CCC2(CCCC2)C1 42037,c1(CCNC(C(=O)N(C(c2c(C)cccc2)C)C)=O)ccc2c(c1)CC(C)O2 42038,c1(COC(c2scc(CC3CC(=O)NCC3)n2)=O)ncnc2[nH]cnc12 42039,N(C1CCc2ccc(Br)cc21)C(C1CCCN1S(=O)(=O)c1ccc(Cl)c(Cl)c1)=O 42040,C#CC1(NC(c2occc2CNC(C2CCCCC2F)=O)=O)CCOC1 42041,N1(C(=O)CCOc2cccc([N+](=O)[O-])c2)CCNC2(CCNCC2)C1 42042,C12CCCN(C1)C(=O)c1csc(n1)NC2=O.C(C)(C)(C)N(C(=O)CNC=O)C 42043,C1(C)(C(=O)NCC(CN(C(=O)C(C)COC)CC)(C)C)CCC(=O)NC1 42044,c1(C(N2CCCN(C(C(C(C)C)F)=O)CC2)=O)coc2cc(F)ccc12 42045,C(=O)(C1=CC2(CN(C(C3CC4(CCC4)CO3)=O)C2)OC1)NCCN=S(C)(C)=O 42046,CCC(O)C(=O)N1CC(OCCNC(=O)CC2CC(c3ccccc3)C2)C1 42047,Cc1ccc(F)cc1C(N1CC2(CNC(c3cc(Cl)c(Cl)n3C)=O)CCC1C2)=O 42048,C1(NC(C2N(C(C3(CC)CC(C)(C)C3)=O)CCCC2)=O)CCCOC12CCC2 42049,C1(NC(C2CCc3nncn3C2)=O)CC1C1CCCN(C(=O)C=CCF)C1 42050,c1(NC(CC)=O)nccc(=NCCCNCc2nnc3ncccn23)[nH]1 42051,C1(C(N2CCC(N(C(CCCC)=O)CCO)CC2)=O)CN(C)CC(C)O1 42052,CN1CC(O)CC1(C)C(=O)NCC1CCCCN1C(C1CCCCC1)=O 42053,C1(C2(O)CCOCC2)(NC(N(C2CCC(OC)CC2)C)=O)CC1 42054,C1(c2nnc(O)o2)CCCCN1CC#CC(F)(F)F 42055,C1(NC(c2cnco2)=O)Cc2ccccc2N(C(c2cocn2)=O)C1 42056,c1(CNC(c2c(OC)cncc2)=O)cc(O)ccc1Cl 42057,N1(C(C(C)OCOC)=O)CCC(C(=O)NCCc2cnnn2C)C(C)(C)C1 42058,N1(C(c2cc(-c3cc(F)cc(OC)c3)[nH]n2)=O)CCc2cccc(Br)c2C1 42059,C1(NC(CC2CC(=O)NC2)=O)CCCCN(C(=O)C=CC=C(Cl)Cl)C1 42060,C1(OC)CCCN(C(C2CCCC(Nc3ccnc(C)n3)C2)=O)C1 42061,c1(CNC(=O)NCC2C(c3n(C)ncc3)OCC2)n[nH]c2ccc(Br)cc12 42062,c1(N(C)C)ccc(Br)c(Cl)c1.n12cc(nn1)CCC(=O)NC(C1CC1)CC2 42063,c1(CC)nn(C)cc1C(=O)NCC(C)(C1CCC1)NC(=O)C(F)F 42064,CCC(C)(CCC(C)C)C(=O)N1CCC(CCNC(=O)CC2CCNC(=O)C2)C1 42065,c1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)cc(C)cc2c[nH]nc12 42066,C1(NC(C(c2ccc(F)cc2)(C)C)=O)C2CCC1CN(C(c1cc(O)n[nH]1)=O)C2 42067,c1(C(N2CC(CC(C)NC(=O)CC3=CCCC3)C2)=O)ccc2c(c1)C(=O)NC2=O 42068,Cc1cc(C(N2CCCC2CCNC(=O)CS(=O)(=O)N(C)C)=O)nc(O)n1 42069,CC(CC(=O)NC1CCCC1NC(C1(C(F)F)CC1)=O)n1cccn1 42070,O=C(CC1CC2CC1C2)NNc1ccc(Br)c(F)c1F 42071,Cc1ccc(C(=O)NCC23CC(CN2C(=O)Cn2ccc(C4CC4)n2)C3)c(C)c1 42072,c1(N2CC(NC(C3CC4C=CC3C4)=O)CC3(C2)CC3)nc2cc(F)ccc2o1 42073,c1(CS(=O)(=O)NCCCCCC)ccc(NC(=O)NC2(O)CCCSC2)cc1 42074,CCCC(CC)C(=O)NC1CCN(C(=O)NC2CCC2C(=O)OCC)CC1 42075,C(=O)(C(F)C(F)(F)F)NC(CC)CNC(=O)COCc1ccncc1 42076,CC1(C)CC(NC(=O)C(C)(O)C(F)(F)F)CCN(CC2CCCC2)C1 42077,Cc1nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnc(C)s3)C2)c2ccnc-2[nH]1 42078,c1(N2CCN(c3c(C)nc(-c4cccc(F)c4)s3)C3C2C3)ncnc2sccc12 42079,C1(NC(C)=O)CN(C(c2ccccc2N(C)C)=O)CCC1O.C1CO1 42080,C12(C)CCC(CC1)OC2.C1(S)C(C(=O)N(C2CC3CC2CN3)CC)CCN1C 42081,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42082,c1(C(=O)NCCCC2N(C(C(C)(CO)OC)=O)CCC2)cc2c(cn1)COCC2 42083,c1(OC)cc(OC)c(C(N2CC3CC(C2)O3)C(=O)NC2CCOC2)c(OC)c1 42084,C1(C(=O)NCCC(=C)CNC(=O)CCc2cn(C)nc2C)CCOC(=O)CC1 42085,CC(C(=O)NCC1CN(C(C2CCC(F)C2)=O)C1)S(=O)(=O)C1CCOCC1 42086,c1(C(N2CC(COC)(NC(=O)CC(C)SC)C2)=O)cccc2c1COC2 42087,N1(C(CC2(C)CN(C(CCOC)=O)C2)=O)C2C=CCC1CCC2 42088,c1(C(N2CC(OC)C(NC(C3CCCN3C)=O)C2)=O)nnc2ccccn12 42089,C1(C(=O)NCC2C(C)CN(C(=O)C=Cc3ccsc3)C2)CCCCC(C)(C)C1 42090,CCCCC(O)CC(=O)NC1CCCC(NC(=O)COc2c(F)cccc2F)C1 42091,C1(CCNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42092,Cn1oc(C(=O)NCC2CCN(C(=O)COCC3CCOC3)C2)cc1=O 42093,N1(C(Cn2c(C)cc(C)n2)=O)CC(C)N(C(c2nnn3c2CSCC3)=O)CC1C 42094,C(=O)(C#CC1CCCCC1)NC1(C)CC(C(=O)NC(CC=C)CC(F)F)C1 42095,C1(C(=O)NCC2CCCO2)(CC)CCCC1O.c12ncoc1CNC2=O 42096,n1(CCC)ccc(C(=O)NCC2COCC2NC(C2CC=CCO2)=O)n1 42097,Cc1ccc(CO)c(O)n1.C12(CN(C(=O)C(C)C3CCCO3)C1)CC(=O)N2C 42098,C1(C(=O)NC(CC=C)CC)CCN(C(=O)CC2CCSCC2)C12CC2 42099,NC1CN(Cc2nc(-c3nccs3)no2)C2(CCCOC2)C1 42100,CC1CC2CN(C(c3cnc4[nH]cncc3-4)=O)CC2N1C(=O)Cc1cn[nH]c1 42101,C1(C)(C(=O)NC(C#C)C2CCC2)CCN(C(=O)CC2CCC=CCC2)C1 42102,c1(N(C)CC2CC2C2CC2)cccc(-c2cnn(C)c2)c1 42103,c1(CNC(C(C2CCN(c3ccc(CC)cc3)CC2)C)=O)c(F)cc(Br)cc1F 42104,c1(C(N2C(C3(NC(=O)C=Cc4cc[nH]c4)CC3)CCC2)=O)ccc2nnnn2c1 42105,C(CC(=O)NCCC1(C)CCN(C(C2(CO)COC2)=O)C1)(C(F)(F)F)OC 42106,c1(OC)cccc(OC)c1S(=O)(=O)NC1C2CN(C(=O)Cc3nc(C)cs3)CC12 42107,C1(N(C(=O)C(c2ccnn2C)N(CC)CC)CC#C)CCN(C(=O)CSC)CC1 42108,C(=O)(CCCC(F)(F)CO)NCC(c1ccccc1)NC(C1C(C)OC(=O)N1)=O 42109,CCC(CNC(c1sccc1C)=O)(CC)NC(C1CC(OC(F)F)C1)=O 42110,c1(SC)cc(C(=O)NC2CC23CCN(C(=O)CSC2CCCCO2)C3)ccc1F 42111,C(C1c2ccsc2CCN1C(C1CCSCC1)=O)NC(C1C(OCC)C1)=O 42112,c1(OC)ccc(CN2CCN(C(=O)CC3CCCC(C)O3)C(C)C2)nc1Cl 42113,c1(C(=O)NC2CC(C)N(C(C3(C)CCCS3)=O)C2)cccc2cc(O)ccc12 42114,C1(CC(=O)NC2(C)CCOC2=O)N(C(c2csc(F)c2)=O)CCC1(C)C 42115,N1(C(c2c(CC)cc(F)cc2)C(=O)NCc2ccccc2)Cc2cccc(C)c2C1 42116,Cc1c(NCCC(N2CCC(C(F)F)C2)=O)occc1=O 42117,C(=O)(C(c1cccs1)NC(=O)C(C)N1CC(C)C1)NCC(=O)OCC 42118,N1(C(C(C)NC(=O)OC)=O)CCCC(NC(c2cccc(C(F)F)n2)=O)C1 42119,C1(NC(C2C(C)CCN2C(C2C3CCCC23)=O)=O)CC2(C1)CC(C)(C)C2 42120,C(C(F)(F)CCC(=O)NCC1CCN(C(C)(C)C)CC1)n1c(C)nc(C)n1 42121,c1(C(=O)NCC(C)NC(c2c(CC)ncs2)=O)cc[n+]([O-])cc1 42122,N1(C(c2cnn(CC)c2Br)=O)CCC(NC(=O)Cn2cnnc2O)CC1C 42123,C12(CNC(C3(SCC)CC3)=O)COCC1CN(C(=O)C(C1CC1)OC)C2 42124,C(CCCCCNC(C(C)SCC)=O)N(C(=O)C(O)C1CCC1)CCCC 42125,c1(C(=O)OC)sccc1S(=O)(=O)NC1CN(C(=O)Cn2nc(C)cc2C)CC1O 42126,C(=O)(C(C)(C)C(C)C)N(CCOC)CCNC(c1sc(CO)nc1C)=O 42127,c1(C(=O)NCC2(F)CCN(C(c3c(C)con3)=O)C2)cnn2c(N)ccnc12 42128,C1(C(=O)OCC)CC1C1CCN(C(=O)CN(CC)Cc2ncc[nH]2)CC1 42129,C(=O)(C(O)CCCNC(c1cnn(C)c1)=O)N(CC(C)C#N)CC 42130,N12CC(C)C(C(C)C1)CNC(=O)CCNC2=O.c1(NC(COCC)=O)cccs1 42131,N1(C(c2n(C)nc(C3CCC3)c2)=O)CCCC(CNC(c2c[nH]c(=N)s2)=O)CC1 42132,c1(-c2nnc(N(C(C=C)C)C)n2CCCC(=O)OCC)cc(Cl)ccc1OC 42133,Cc1cc(NC(C2CSCCN2C(c2ccc([N+](=O)[O-])cc2)=O)=O)c(C)cc1Cl 42134,N1(C(CCC#C)=O)CCCN(C(=O)C(O)Cc2ccccc2)CC1CO 42135,C(=O)(C1=CC2(CCOC2)C1)NC(C1(O)CN(C(c2c(C)nc(O)[nH]2)=O)C1)C 42136,C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(NC(=O)Cc2cnn(C)c2C)C1 42137,c1(OC)cc(C)sc1C(=O)NCCCN(C(=O)C(C)n1cccn1)C 42138,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42139,C1(CC)CN(C(c2cc(Cl)cnc2C)=O)CCN1C(c1ccc(C)o1)=O 42140,Cn1nc(C(F)F)cc1C(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42141,CC1CC2CC(C2)NC1=O.C1(CCNC(=O)OCCC(C)(C)C)OCCC1C 42142,N1(C(C(C)(N(C(=O)CCCC2CCCO2)C)C2CC2)=O)CCC12CCCC2 42143,N1(C(c2n(C)nc(C(F)(F)F)c2)=O)CCC2(CCC2CNC(C2(F)CC2)=O)CC1 42144,C1(C(N(C2C(C)CCNCC2)C2CCOCC2)=O)Cc2ccccc2C1C 42145,Cc1cc(C)c2cc(C(N3CC(NC(=O)Cc4nncs4)CC3(C)C)=O)sc2n1 42146,C=CC(C)(CCOC)C(=O)NC(CNC(=O)C(C)C(=O)OC)CO 42147,c1(C(N2C(C(=O)Nc3ccno3)COCC2)=O)cc(F)c(F)cc1Br 42148,C1(C)(C(N2CCCC(C(C)NC(=O)CN(C)C3CC3)C2)=O)CCC(C)C1(C)C 42149,c1(C(=O)NCC(CCC)NC(=O)C(F)CC2CCOC2)nccc(C)c1N 42150,c1(C(N(C2CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)CCCC)=O)n[nH]c(C)c1Cl 42151,O=C1CC2CC(C(N3CC4C(C(=O)NOC5CCOCC5)C4C3)=O)C1C2 42152,Cc1nc(O)nc(O)c1CCC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42153,c1(CC)cc(C)c(C(=O)NCC(Cn2cc(C3CCCC3O)nn2)OC)o1 42154,Cc1nocc1CC(=O)NCC1(C2CCCN2C(=O)COCC2CCC2)CC1 42155,C1(CNC(CCSCCC)=O)CC2CCC1N2C(=O)CC1CCCCC1(C)C 42156,C(=O)(C(C(C)(C)C)C1CCCC1)N(C(CNC(COCC(=C)C)=O)C1CC1)CC(C)=O 42157,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42158,S(=O)(=O)(c1cccnc1NC1(CO)CCSC1)N(CCCS(N)(=O)=O)C 42159,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)CC3CCCC3)CCCO2)c1F 42160,C=CC1(C(=O)NCC(=O)NC2CC2)CCN(C(c2ccc(F)s2)=O)C1 42161,C(CC1=CCN(C(C23CCC(O)(CC2)CC3)=O)CC1)NC(C1(C)CC1(F)Cl)=O 42162,C1(C(=O)NCC2(F)CC(CNC(COCC=C)=O)C2)Cc2ccc(F)cc2O1 42163,C1(C)(NC(=O)NCC2(OCC)CN(C(=O)Cc3ccccc3C)C2)CCC(=O)N1 42164,N1(C(=O)NC(C(=O)OC)COC)CCCC(c2nnc(S)n2C(C)C)C1 42165,C1(C(=O)NCCN(C(C2CC(OCC)C2)=O)C2CC2)C2CCC1(C)C2(C)C 42166,c1(C(N2CC(SC)C(NC(=O)C(F)n3ccnc3)C2)=O)cc(C)cc(C)c1 42167,N1(C(CN(C2CCC2)C)=O)CC2CC(NC(C3(CC#N)COC3)=O)C(C2)C1 42168,N1(C(C(COCC)OC)=O)CCOCC1CCNC(c1c(C)ncn1C(C)C)=O 42169,CCC(C)(C)C(=O)NCCOC1CCN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 42170,c1(C(=O)OC)c(C)[nH]c(NC(c2cnc(Br)s2)c2nnnn2C2(C)CC2)c1C 42171,C1(CNC(C(C=C)(F)F)=O)CC2CC1CN(C(=O)CCc1cnn(C)c1)C2 42172,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CCC(F)(F)F)=O 42173,CCCC(CNC(=O)CCCCNC(N)=O)C(=O)N(C)C(c1ccccn1)C 42174,C1(CNC(c2c(OC)cnnc2)=O)CC(C)CN(C(c2ccnnc2O)=O)C1 42175,N1(CC(=O)NC(C(=O)NCCC(=O)OC)(C)C)CCC(F)CC1 42176,CCC(C)(C)CCNC(=O)CCC1CCCN1C(=O)C(C)NC(=O)NC 42177,CN1CCCC(C(=O)N(CCCNC(C2CSCCS2)=O)CCO)C1 42178,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42179,N1(C(C2(C=C)CCC2)=O)CCC2(CC1)CC(C)N(C(c1cn3c(n1)SCC3)=O)C2 42180,c1(COCC(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)cccc(C(F)F)c1 42181,N1(C(C(C=C)(C)C)=O)CC2CCC(C(=O)NCCSCC(=O)OC)(C2)C1 42182,c1(NC(=O)Nc2ncn(C)n2)cc(F)ccc1C(N1CCC(CO)C1)=O 42183,CC1(C)C(CNC(c2ccc(C3(C#N)CC3)cc2)=O)CCN1C(=O)CCCCF 42184,c1(C(C(=O)NC2C(NC(C(CO)N(C)C)=O)CCC2)(C)C)ccccc1F 42185,C1(C2(O)CN(C(=O)CCc3cnc(O)[nH]3)C2)(CNC(C(C)NC(CC)=O)=O)CC1 42186,C#Cc1cccc(CC(=O)NC2CN(C(C3COCC3C(N)=O)=O)CC2OC)c1 42187,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42188,C1(C(=O)Nc2ccc(C(C)(C)C)o2)CC2CC2N1C(c1cc(O)ncn1)=O 42189,N12CC(CC1(C)COC)NC(=O)CN(CP(C)(C)=O)CCCC2=O.CCOCC 42190,CC#CCCC(=O)N1CCCCC1C(C)(C)CNC(=O)COCc1ccncc1 42191,C(=O)(C(C)C(O)CCCC)N(CCNC(c1cccc(C#C)c1C)=O)CC 42192,n1(C(CCC)CCO)cnc2c(N3CCCC(N4CCOC4=O)CC3)ncnc12 42193,Cc1ccc(OC(C)C(=O)NC2(N3CCOCC3=O)CC2)cc1.C12CN(C1)C2=O 42194,C1(C(=O)N(C2CCN(C(C34CC5CC3C4C5)=O)CC2)CCO)CC2(CCCO2)C1 42195,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(CNC(c1cc[nH]n1)=O)CO)C2 42196,c1(C(N(CCC)CCNC(c2n[nH]c(C)c2Cl)=O)=O)ccc2nnnn2c1 42197,c1(-n2c(-c3csc(Cl)n3)nc(COC)n2)c(C)cc(C)cc1C 42198,C1(N(CC#C)C)CCCN(C(=O)C(=O)Cc2cscc2OC)C1 42199,c1(CCC(=O)NCC(CNC(C(C)=C(CC)C)=O)F)cccc([N+](=O)[O-])c1 42200,C(=O)(C(CC)C(=O)NCC1C(NC(c2ccnn2C2CC2)=O)CC1)OCC.C1CC1 42201,c1(C(=O)NCC2(C)CCN(C(C=C(C)C)=O)C2)nn(C)c(C)c1N 42202,C1(C(=O)NCC(O)CO)CCC2(CC2)N1C(C1CC=CCO1)=O 42203,N1(C(=O)COC2CC2)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42204,n1(CC)c(C(=O)N(C2CN(CC)C2)C)cnc1O.N12CC(C)C1C2=O 42205,C1(C(=O)NCC2CCN2C(c2csc(Cl)n2)=O)CC1C1CCC1 42206,c1(CN2CCC=C(C)C2)cc(=NC2CCCN(S(=O)(=O)N(C)C)C2)[nH]c(CO)n1 42207,N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(=O)CC2CCCC(F)(F)C2)C1 42208,n1(CCSS(C)(=O)=O)nnc(C(=O)NCC(C)NC(=O)CCCOC)c1C.CC 42209,C(=O)(C#CC1CCCO1)N1CC(CNC(c2[nH]c(=N)sc2)=O)C(C(F)(F)F)C1 42210,Cc1ncn(C)c(=O)c1C(=O)NC1CN(C(=O)C(C)C(O)C(C)C)C1 42211,C(=O)(C(CC(C)(C)C)OC)N1C(C(=O)NC2CC(=C)C2)CCC(O)C1 42212,N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42213,Cc1nn(C)cc1OCC(=O)OC(c1cccc(C(F)(F)F)n1)C 42214,c12ccc-1cc2.C1(NC(CNC(CC)=O)=O)CCN(C(=O)C(C)CC)C1C1CC1 42215,c1(CNC(C(CNC(=O)CCC2CCCN2C)OC)=O)cnccc1Cl 42216,CCC(C)C(C)C(=O)NC1CN(C(=O)CN2CCCC(C(F)(F)F)C2=O)C1 42217,C1(=O)C(CC2CC(F)(F)C2)N1C1CC1.C1(CCN(C)C)CCCN1C(=O)NC(C)(C)C 42218,C1(C(N2CC(NC(CCn3ccc(C)n3)=O)C(C)C2)=O)CC(C)(C)OC(C)(C)C1 42219,Cc1cnccc1C(=O)NCC(C)(O)CNC(=O)C(c1cccnc1)C 42220,CCN=C(NCC(C1CC1)C1CC1)N1CCCC(OC)(OC)C1 42221,C1(NC(COc2cn(C)nc2)=O)CCN(C(=O)C(C)(C)C2CCC2)CC1F 42222,C(=O)(C(CCNC(=O)CC1OCCC1C)N(C1(C2CC2)CC1)C)OC 42223,c1(C2C(C(=O)OC)C2)cccc2c(C(N3C(CC)COCC3)=O)cccc12 42224,N1(C(CSS(C)(=O)=O)=O)CCC2CN(C(=O)COCc3nc[nH]n3)CC2C1 42225,c1(-c2ccc(N3CCN(C(CNS(CC)(=O)=O)=O)CC3)cc2)nc(=N)[nH]c(=N)[nH]1 42226,C#Cc1c[nH]nc1C(=O)NC(C1CN(C(c2cnc(C3CCC3)s2)=O)C1)C 42227,C=C(Br)CN=C(NCc1ccc(SC)cc1)NC(C)C 42228,c12cccc(c1)OCc1cnc([nH]1)NC(=O)C(=O)N2.c1(C(C)NC)nccn1C 42229,C1(CC)(CNC(=O)C(C2CCC2)NC(c2csnc2C)=O)CCOCC1 42230,c1(C(=O)NCC2C(CNC(COCc3cn(C)nn3)=O)C2)nc[nH]c2ncnc1-2 42231,CCCCC(C)CCC(=O)N1CC=C(CCNC(C2CC2C2CC2C)=O)CC1 42232,CC12CCCN1S(=O)(=O)C(C(=O)NCC(c1ccco1)COCc1ccccc1)C2 42233,N1(CC)C(=O)CCC1C(=O)NCC(C)(C1CC1)NC(=O)CC1CCCCO1 42234,C1(CC)CN(C(=O)C(C2CCC2)NC(c2cc(C)ccc2O)=O)CCN1C 42235,C1(NC(CCC=CC)=O)CC2C1CCN2C(=O)CC(c1ccccc1)C1CC1 42236,N1(C(CCCSC)=O)CC2(CCN(C(c3csc(C)c3C)=O)CC2)C2COCC12 42237,C1(C)(C(=O)NC(c2cnn(C)c2)C(=O)NCc2nnc(CC)s2)CCC(O)CC1 42238,C1(NC(CCc2nc(C)sc2)=O)CN(C(=O)C(C)OCC2CC2)CC1(C)C 42239,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCCC2CC(N)=O)=O)nn1C 42240,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42241,CN1CC(CNC(=O)C(C2CC2)NC(c2ccc(CO)o2)=O)CC1=O 42242,C1(C)(CC)C=C(C(=O)NCCC2CCCN(C(C3CC3(C)C)=O)C2)C1 42243,c1(C(N(CCNC(C(C2CC2)SCC)=O)C2CC2)=O)cc2ccnn2cn1 42244,c1(OC)cc(CN(C(C(=O)NC2(C)CC2)C2CCOC2)C2CC2)cc(F)c1OC 42245,N1(C(C(F)=CCC)=O)CCCCC1C1(NC(=O)CCCCNC(=O)OC)CC1 42246,N1(C(c2n(CC)nnc2)=O)CCC2(CCC2NC(c2cccc(F)c2C)=O)CC1 42247,C1(C(C(N2CCC(OC)(CNC(=O)CNC(C)=O)C2)=O)O)CCS(=O)(=O)CC1 42248,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42249,N1(CC(=O)N(CC(CC)NC(=O)Cn2nnc(C)n2)CC)CCC(C)C1 42250,c1(-c2nc(C(C)NC(C3OCC3(C)C)C)on2)cccc(Cl)c1 42251,c1(-c2ncc(CN=C(NC(C)CF)NC(C3CC3)C3CC3)s2)c(F)cccc1F 42252,C1(CC)CCCCC1OCC(=O)NC(C1CCN(C(=O)C(=O)NC)C1)C 42253,C12(CCn3cc(-c4n(C)ccn4)nn3)CCC1CN(C(=O)C(C)(Cl)Cl)C2 42254,c1(C(=O)NCC=CCNC(C2OCC(C)C2)=O)cc(F)cnc1Cl 42255,C1(NC(CN(CCC)C(C2COCOC2)=O)=O)Cc2nccn2C1 42256,n1(CC(=O)Nc2c(C)cc(C(F)F)cc2)nc(CN)c2c1CCC2 42257,c1(C(N2C3C(NC(C4C(C)(C)C4)=O)(CCC3)CC2)=O)nc(Br)c2ccccn12 42258,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42259,c1(C(=O)NC(C(C)NC(c2nc(OC)nc(O)c2)=O)CO)c(F)cc(N)cc1F 42260,N1(C(C2(NC(C(COC)C)=O)CCC2)=O)CC(O)(C2CCC2)C1 42261,N1(C(c2c(OC)scc2)=O)CCC(C(=O)Nc2ccc(C)nc2)C1(C)C 42262,C=C1CN2C(=O)CCC2(C(=O)NCCN(C(c2sccc2C)=O)CC)C1 42263,Cc1cccc2c(CC(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)c[nH]c12 42264,N1(C(c2c(C)cnn2C)=O)CC2(CC(C(N3CCCC(O)C3)=O)C2)C1 42265,c1(C(NOCC(=O)NC(CC#C)C(=O)OC)=O)cc(C)ccc1F 42266,c1(C(N2C(CNC(C(CC)(C)CO)=O)CCCCC2)=O)onc2ccccc12 42267,N1(C(CCc2nc(C)sc2)=O)CCC(C(C)(C)CNC(c2cn(C)nn2)=O)CC1 42268,C1(C(=O)NC(CO)(C2CC2)C2CC2)CCCC(C(=O)Nc2ccc(CO)o2)CC1 42269,CCCC(CC1CCCC1)C(=O)N1CCC(O)(CNC(c2[nH]ncc2C#N)=O)CC1 42270,CC12CCN(CC1)CC2NC(c1coc(CNC(c2cscn2)=O)c1)=O 42271,C1(S(C)(=O)=O)(C(=O)NC(C(C)NC(c2c(C)ccc(C)c2)=O)C)CC(O)C1 42272,N1(CC(=O)N(CCN(C(c2cncc(OC)c2)=O)CC)CC)CCCCS1(=O)=O 42273,N1(C(C=CCC)=O)CCC2CC2(CNC(=O)CCN2CCC(CO)CC2)CC1 42274,c1(NC(N(C)C)=O)cccc(CN2CCCC(N(C)C)C2)c1 42275,N1(C(C2N(CC)CC2)=O)CCC(C)(CCNC(c2ccc(NC(C)C)cc2)=O)C1 42276,C1(CC(=O)NC2CC2)CCCN(C(C2CCNC2=O)=O)CC1.c12cccc(c1)OC2 42277,C(=O)(CC(C(F)F)c1ccccc1F)NC(CC)CN(C(C1(O)CCC1)=O)CC 42278,c1(COC)nc(N2CCCC(NC(c3ccc(O)nc3)=O)CC2)cc(Cl)n1 42279,N1(C(C(F)=CCC)=O)CC(C)CCC1CNC(C1CC(OC(F)F)C1)=O 42280,c1(CC(=O)N(C(C)CNC(=O)Cc2c(Cl)cncc2Cl)C)cccc2nonc12 42281,c1(C(N(CC)CCSC)=O)ccc(C)c2cccnc12.C12(CCSC1)C(=O)N2 42282,c1(CNCC2C(C(=O)Nc3cccc(OC)n3)C2)cccc(F)c1Cl 42283,c1(C(=O)NCC(C)(C)NC(C(C(=O)OCC)F)=O)ccc2c(c1)COCCN2 42284,C=CC1(C(N2CC(CNC(C3(CO)CC3)=O)C2)=O)CCCCC1 42285,COn1cnc(C)c1C(=O)NCCCN(C)C(c1sc(Br)cc1C)=O 42286,C1(CC(=O)N(CC(=O)NC(C)CC(C)C)C)(NC(C)=O)CC1 42287,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42288,Cc1nc(C(C)C)sc1C(=O)N(CCNC(=O)COc1ccsc1)C(C)C 42289,c1(C(N(C(CN(C(=O)C(O)CCC#N)C2CC2)C2CC2)C)=O)csc(C2CC2)n1 42290,N1(C(C2CC(OCOC)C2)C(=O)NC2CCCC2)C2CCC1CC(CO)C2 42291,C1(C(=O)NC(CC)CN(C(=O)CNS(=O)(=O)NC)CC)CCOC1C(F)(F)F 42292,Cc1ncc(NC(C2CN(C(c3nn(C)cc3Br)=O)CCN2)=O)cc1O 42293,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42294,c1(C(N2C(CNC(C(C3CC3)OCC)=O)C=CC2)=O)cc(F)c(C)cc1N 42295,C12(C)CCCC1CN(C(=O)COC)C2.N1(CC)CCOCC1C(=O)NCCOC1CC1 42296,n1(CC(=O)NCC2N(C(CCCC=C)=O)CC(F)C2)nc2n(c1=O)CCCCC2 42297,C(C(=O)NCC(C)NC(=O)C(c1ccc(F)cc1)(C)C)(C(C)C)NC(CCC)=O 42298,C(=O)(C(C)(C)CC(C)C)NCCCCN(CCCNC(CC(CC)C1CC1)=O)C 42299,N1(C(C=COCC)=O)CCC(CNC(=O)Cn2cnnn2)(OCC)CC1 42300,CC1(NC(C2CCC(N=[N+]=[N-])C2)=O)CCCc2ccccc21 42301,c1(C(=O)NCC2CN(C(C3C(C#C)C3)=O)C2)ccc(CNC(C)=O)cc1 42302,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC(NC(=O)CCC2CCC(=O)N2)C1 42303,C(CC(=O)NCC1CCOC1=O)(CC(C)C)NC(CSCC#C)=O 42304,CCC(CC(=O)NCCCC(C)(C)NC(=O)C(CO)C(C)(C)C)C(C)(C)C 42305,C1(OC)(OC)CC(C)(C(C(=O)Nc2ccccc2C)N(c2cscc2Br)C)C1 42306,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(C)C3CCCCC3)CC12 42307,c1(C)cccc2oc(C)nc12.C=CC(C)(C)C1c2nnnn2CCCN1 42308,Cc1ccccc1C(C)NC(C1C(CNC(=O)CN(C)C)C1(C)C)=O 42309,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42310,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42311,Cc1c(C(N2Cc3c[nH]nc3C2)C(=O)NCCCOC2CC2)cccc1F 42312,c1(SC)cc(N2CCC(C)(CNC(=O)Cc3sc(O)nc3O)CC2)nc(SC)n1 42313,N1(C(C2(C)CCOCC2)=O)CCCC(NC(=O)CCC2(O)CCC2)CC1 42314,C(=O)(C(C(C)C)SSC)N(C(CN(CC)CC)C)CC.CCC(C=O)OC 42315,c1(CC(N2CC3C(NC(=O)COc4ccsc4)C3C2)=O)ccc2ncnn2c1 42316,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42317,c1(C(N(CCCCCNC(C(CSC)C)=O)C)=O)ccn2cccc2c1 42318,N(C1CN(C(=O)C=C2CCC2)CCc2ccccc21)C(c1ccc(Cl)nc1O)=O 42319,C1(NC(C2CC(CCC)C2)=O)CCCC(C(N2CCSCC2)=O)CC1 42320,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CC2CNC(c1cc(CSC)on1)=O 42321,C1(NC(=O)CSC(F)(F)F)CCN(C(c2ccc(CO)cc2F)=O)CCC1(F)F 42322,N(C1CN(C(C2(C)CC(F)C2)=O)Cc2ccccc21)C(c1cc(C)[nH]n1)=O 42323,C1(CC(=O)NCCC2CN(C(c3ccn(CCF)n3)=O)C2)CC2CCC1O2 42324,c1(C(=O)NC(C(C)NC(CCC(=O)NCCC)=O)C)cc(C)c(C)nc1C 42325,c1(CC2(NC(C(C)OCCOCCOCCOC)=O)CCC2)c(OC)cccc1F 42326,C1(C(=O)NCC2CC2CO)CCCN(C(c2ccncc2-n2cccn2)=O)C1 42327,CC1CC(C(=O)Nc2cccc(CO)n2)N(C(c2ccc(C(F)(F)F)nc2)=O)C1 42328,CC(C)(C(=O)NC12CC1CN(C(=O)CCOc1cc(Cl)cc(Cl)c1)C2)C(F)F 42329,c1(C(=O)NCC2CCC(C(=O)NCc3nc(C)sc3)C2)ccnnc1O 42330,c1(OC)ccc(C(N2CCC(CNC(=O)CC(C)OC)(OC)C2)=O)cc1F 42331,c1(NCN(CCCC)CCCC)cccc(-c2scnc2C)c1 42332,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42333,C1(CNC(C=CC(C)(C)C)=O)CC(NC(c2coc(C3CCOCC3)n2)=O)C1(C)C 42334,C(=O)(C(C)CC(N)=O)Nc1nc(C2N(c3nc(C)c(C4CC4)s3)CCCC2)on1 42335,N1(C(COCC=C)=O)CC2CC1CC2NC(=O)C(C)(C)c1ccn(C)n1 42336,c1(C(=O)NC(c2ccc(C)nc2)CNC(=O)CC2CC23CC3)cc(F)cnc1O 42337,N1(C(CC2C(C)=NNC2=O)=O)CC2CCOC2(CNC(=O)CCC2OCCO2)C1 42338,c1(OC)cc(C)nc(N(C)CC2CCN(C(=O)CC(C)SC)CC2)n1 42339,C1(C(C)C)C(C(=O)NCc2nc(CO)n[nH]2)CCN1C(=O)CCc1cncnc1 42340,C1(c2n(CCC)nnn2)(NCCCC2CCOC2)CCC2(CCOCC2)C1 42341,Cc1ccc(C(=O)NC2CCOCC2C(=O)NCCC(C)C)c(O)c1 42342,c1(C(N2CCC(SC)C2)=O)n[nH]c2c1CCN(C(=O)Nc1ccnc(Cl)c1F)C2 42343,c12ccccc1C(=O)N1CCC(C)(C1)C(=O)N2C1CC1.N1(CC)CCCCCC1 42344,CC(=O)CCCC(=O)NC1(C2CCCCN2C(=O)CCc2cccnc2)CC1 42345,c1(N2CC(C)(N(C(CC)=O)CCO)C2)nc(C(F)(F)F)ccc1C(=O)OC 42346,CCC(C)C(C)CN=c1[nH]c(C)cc(=NCc2ccc3nn[nH]c3c2)[nH]1 42347,C1(C(CNC(c2n(C)cnc2)=O)(C)O)CCCN(C(=O)C=CC(=O)N(C)C)C1 42348,S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N(C(C(c1c(C)cccc1C)O)=O)CCO 42349,N1(C(CC2(C(=C)F)CCC2)=O)CC2CCC(C1)N2C(=O)Cc1cnn2ccccc12 42350,C1(C)(CNC(C(c2ccnn2C)C)=O)CCN(C(=O)Cc2cccs2)C1 42351,c1(C(N2CCCC(C)(NC(CN(C)C)=O)C2)=O)ccc2c(Br)nn(C)c2c1 42352,C#CC1(C(N2CCC2CC)=O)CCN(C(c2cccc(C)c2F)=O)CC1 42353,C1(C(=O)NC(CCSC)C(=O)OC)N(C(c2ccco2)=O)CC12CCCC2 42354,C(C(=O)N1CCCO1)NC(=O)NCc1ccncc1C1CC1 42355,C(C)(C)(CC(=O)NCC1(F)CCC(NC(c2cc(OC)cnn2)=O)C1)OC 42356,c1(C(N2C(CNC(C(CC)(C)COC)=O)CC2)=O)n[nH]c2cc(Br)ccc12 42357,CCC1=C(C(=O)N(CCCOC)C)CCCO1.c12cccc(OCC)c1NC2=O 42358,c1(C(=O)NCC(CC)NC(=O)C(C)C)ccc(NC(c2cc(C)[nH]n2)=O)cc1 42359,N1(C(C=CC(CC)C)=O)CCC2(C=C(C(=O)NCc3ccc(C)cn3)C2)C1 42360,C(C(=O)NO)(c1cn(C)nn1)OC.N1(CC(=O)N2C(C3CC3)C2=O)CCCC1C 42361,C=CCC(C)(C(=O)N(C)Cc1ccc(CNC(=O)C2=CCCC2)cc1)N(C)C 42362,C#Cc1cn(C)nc1C(=O)NC(C(=O)N(c1cccc(Cl)c1)C)C(C)C 42363,N1(C(C)=O)CCN(CCCNC(=O)C(F)CN(C)C)CC1.C1CO1 42364,N1(C(Cc2nc(CC)sc2)=O)CCCC(C(C)NC(=O)C=Cc2ccsc2)C1 42365,c1(CNC(C)CCC2CCCCC2)cc2ccc(Cl)cc2o1 42366,c1(NC(c2n(CC(=C)C)nnn2)CCCSC)ccc2c(c1)C(C)(C)CO2 42367,Cc1ccc2oc(C(=O)N(CCCNC(C3(F)CCCCC3)=O)C3CC3)cc2n1 42368,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(CC3CC3)C1)=O)CC2 42369,C1(NC(=O)Cc2ccon2)CCCC(NC(c2csc(C(F)(F)F)c2)=O)C1 42370,CC(CO)CCCN=c1[nH]c(=NCc2cccc3c2OCCO3)c2sccc2[nH]1 42371,C(=O)(CC(C)CCC=C(C)C)NC1C(CNC(c2nncc(OC)c2)=O)C1 42372,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(c1cn(C)nc1O)=O 42373,N1(C(c2ncccc2O)=O)CC(C2CCCCN(C(=O)C(F)OC(F)(F)F)C2)C1 42374,c1(NC(=O)CC2(O)CN(C(c3ccno3)=O)C2)ccc(Cl)c(Br)c1 42375,Cc1cccnc1CC(=O)NCCC1COCCN1C(=O)CO 42376,c1(C(=O)NC(CCCCNC(C(COCC)N=[N+]=[N-])=O)C)cccc2nccn12 42377,C1(NC(c2c(C)cccc2Cl)=O)COC2C(NC(C3CC(F)(CO)C3)=O)COC12 42378,c1(C(C)NC(C2(CNC(C3COCCN3C)=O)CC2)=O)ccc(F)cc1 42379,C(=O)(CC(C)CCCCC)N(C1(C#C)CC1)C1CC1.N12CCC(C1)C2=O 42380,CN1CCC(C(N2CC3CC2(CNC(c2ccc(O)nn2)=O)C3)=O)CC1 42381,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42382,C1(NC(c2cn[nH]c2)=O)CC1C1CCN(C(=O)C(=CC2CCCCC2)F)CC1 42383,CCC(CC(=O)N1CCC2C(C(N3CCOC(C4(O)CC4)C3)=O)C2C1)C(C)C 42384,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42385,c1(C(=O)NC(C2CCN(C(CC(=O)OC)=O)C2)C)c(C(F)(F)F)ccc(F)c1F 42386,N1(C(=O)Cc2ccsc2)CC2=C(C1)CN(CC1CC1c1ccccc1OC(F)F)C2 42387,Cc1ccc2[nH]cc(C#N)c(=NCc3coc(C4CCN(C)CC4)n3)c2c1 42388,Cc1c(F)cc(C(N2CC3CN(Cc4ccc(O)c(I)c4)C3C2)=O)cc1Br 42389,c1(N2CCC(COc3c(C)cccc3C)C2)ncnc2sc(I)cc12 42390,Cc1n[nH]c(C)c1CC(=O)NC(C)CC(C)NC(=O)CCC(F)F 42391,S(=O)(=O)(CCC(=O)NC(C#N)C(C)(C)C)N(C)C 42392,C(c1cccc(CO)c1)=CC(=O)N(C(C)CNC(c1nc(O)[nH]c(=O)n1)=O)C 42393,C12(CNC(=O)CN3CCCC3c3ccccc3)CC(CO1)N(c1nccc(OC)n1)C2 42394,CC(CN(C)C)CCC(=O)N(CC(C)(C)NC(=O)Cc1csnn1)C 42395,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCC1CC1 42396,C1(C)(C(=O)NC(C)CNC(=O)CCOCC(F)F)COc2ccccc2O1 42397,CCCCC#CC(C)(C)NC(c1csc(CNC(=O)CCCC(C)=O)c1)=O 42398,c1(CC(=O)NC2CCC(CCNC(CC=C(C)C)=O)C2)ccc2nn[nH]c2c1 42399,C1(C(N(CCCCNC(C2(C)CCN(C)C2)=O)C)=O)CCc2ccccc2C1 42400,N1(C(C2(NC(c3c(C)ccs3)=O)CCSC2)=O)CCC(=C(F)F)CC1 42401,Cc1cccc2[nH]c(-c3ccnc(NC(c4ccccc4[N+](=O)[O-])=O)c3)cc12 42402,C(=O)(C(C)(F)C(F)(F)F)N1CCC(CCCNC(C2(C)CN(C)C(=O)C2)=O)CC1 42403,N1(C(COC)=O)CCCC(N(C(=O)CCc2nnc(C3CCCC3)o2)C)CC1 42404,C(c1nc2ccccc2s1)=Cc1ccc(OCC)o1 42405,CC1(F)CC(C(=O)NC(C(=O)NCc2nn[nH]c2C2CC2)c2ccoc2)C1 42406,N1(C(C(C)OCc2cccc(Cl)c2)=O)CC=C(CNC(C2(C)CCCS2)=O)CC1 42407,c1(NC2CC(=O)CC(=O)C2)[nH]c(=O)n(C)c(=O)c1C#N.CC1CC2CN1C(=O)N2 42408,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCN(C(=O)COCCF)CC1C1CC1 42409,C(=O)(C(C(C)C)C(C)C)NC1CC2C(NC(CC3CN(C(=O)NC)C3)=O)C2C1 42410,C1(CN(C(C(C)OCC=C)=O)CC)CCN(C(c2ccn(CC)n2)=O)CC1 42411,c1(OC)ccc(C(=O)NC2CCN(c3ccnc(N(C)C)n3)CC2O)c(F)c1F 42412,C(CC1=CCCCCC1)n1cc(C(C)NC(=O)C(O)C(C)(C)c2ccccc2)nn1 42413,O(NC(=O)CCC1(NC(=O)C2=COCC2)CCC1)C(CC)C 42414,c1(C(=O)NC(CC=C)CNC(=O)CC2CC(C)C2)ccn2cnc(C)c2c1 42415,C(=O)(CCCCCn1cc(-c2cnn(C(F)F)c2)nn1)N(C)CCN(C)C 42416,C(=O)(C1=CCN(C(c2csc(C(C)=O)n2)=O)CC1)NC1(CC)CCCC1 42417,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(C2CC2)n1)=O 42418,c1(C(=O)NC2(CCCNC(C(COC)COC)=O)CC2)cncc(S(C)(=O)=O)c1 42419,N1(C(c2n(C)nc(C(F)F)c2)=O)CCC2(CCCN2C(=O)CC2C=CS(=O)(=O)C2)C1 42420,c1(C(=O)NC(CNC(CN(C)CC)=O)CC(C)C)cnc2n1CCS2 42421,c1(CN(C)CCNC(=O)C=CC(=O)NC(C2(O)CCCC2)=O)ccccc1 42422,C1(C(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)C)CC2CCC1CC2 42423,C12(C(N3CC(CNC(CC=CCC)=O)C4C3C4)=O)CCN(CC1)S(=O)(=O)C2 42424,CC(C)(CC1CCOCC1)C(=O)NC1CN(C(=O)CCn2cncn2)C1 42425,n1(C(C)C)cnnc1C(=O)NCC1(C(=O)NCCSC2CC2)CCCO1 42426,c1(-n2c(CC(CCC)C)nc(CN(C)C(C)C)n2)ccc2c(c1)OCCO2 42427,N1(C(CCC#C)=O)CCC=C(C(=O)N2CCC2CC(C)C)C1 42428,c1(CN2CCC(c3nnnn3CCCF)(OCC)CC2)cccc2c1nnn2C 42429,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(=O)NC2CCOC3(CCC3)C2)C1 42430,c1(N2CC(C)(C)NCC2)nc(N)c2ccsc2n1.C1(N)CCC2C(CC1)C2(F)F 42431,C1(C(=O)NC(CC(C)NC(C2CCC3CC2C3(C)C)=O)C)CCC2CCCCC2C1 42432,c1(OC)ccc(C(N2CCN(C(=O)C=CC3CCC3)CC2CO)=O)c(OC)c1 42433,S(=O)(=O)(CCC(=O)N(C1CN(C(c2ccc(C(=O)N(C)C)cc2F)=O)C1)C)NC 42434,C1(C(=O)NC(C)(C)CN(C)C)CC2(CCC2)CN1C(=O)CC1(C=C)CCC1 42435,C(=O)(CC(C)(C)C(=O)NC(C)CCCNC(=O)C(F)(F)c1cnccn1)OC 42436,C1(SCCC(=O)NCCSCCCNC(C2CC2F)=O)CCCCO1 42437,C1(OC)CC2CC1CC2NC(=O)NC1CC1C1CCC1 42438,CC(C)C1C(=O)N1.N1(C(CCOC(=O)C2CC2)C)CCOCC1 42439,N1(C(=O)CC2CC2)CCC(S(=O)(=O)N2CCCC2c2ccc(Cl)c(Cl)c2)C1.N1CCCC1 42440,N1(C(C(C)N(C(CC2(CC)CC2)=O)C)=O)CC(C(=O)NC)C2(CCC2)C1 42441,c1(C(=O)NCCN(CCC)C(c2cnc(C(C)C)o2)=O)c(C)coc1C1CC1 42442,c1(C(C(=O)NC(CCC)CNC(=O)C(C)Cc2ccnn2C)O)cccc(C)c1 42443,c1(NC(=O)CCOC2CN(C(C3CC3C3CC3)=O)C2)ccc(Cl)cc1O 42444,c1(CC(N2C(C(=O)OC)CCS2(=O)=O)=O)ccc2cc(O)ccc2c1 42445,C1(CC=C)(NC(=O)CC2CCC(=O)N2)CCCN(C(=O)CC(C)c2ccco2)C1 42446,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)NCC(O)C2CCC2)c1C 42447,N1(C(C(C)NC(=O)NC)=O)CCN(C(c2c[nH]nc2F)=O)C(CCO)C1 42448,C1(CN(C)C(c2cn(CCF)nn2)=O)COCCN1C(C1CC1c1cccs1)=O 42449,c1(C(=O)NCC(n2cc(CCC3CCC3)nn2)C)ccc(Br)c(Cl)c1 42450,C1(C(=O)NCC(C)N(C(=O)CC2(C#N)CCCCC2)C)CCc2n[nH]cc2C1 42451,C12CCN(CC1)C2.C1(C(C2CCCCS2)=O)CCC(CN2CCCC2)O1 42452,c1(C(=O)NCC2CC2NC(C2(F)CCOC2)=O)cnn2ccccc12 42453,CCCCCCCC(=O)N(C)CC1CN(C(=O)CC2CC(CC)C2)CCO1 42454,Cc1cocc1CNC(C1(NC(=O)COC2CCOC2)CCSC1)=O 42455,C(=O)(CCCC1CCCO1)N(C)CCOCCC(=O)NCCCCCO 42456,N1(C(CCC(=C)C)C(=O)OC)CC2CCCC2(C(=O)OC(C)(C)C)C1 42457,C1(C2(NC(=O)Cc3cnoc3)CC2)CCCN1C(=O)C(O)C1CCC1 42458,c1(OC)ccc2c(NC(=O)NC3CC3)cnn2c1.c12cc(nn1C)CNC2=O 42459,C(C(C)CNC(=O)CCNC(=O)C=CCl)NC(C1(C(=O)NC)CC1)=O 42460,C1(NC(=O)COc2ncccn2)CCCCC1Oc1cnc[nH]1 42461,C(=O)(C(CCC)NC(=O)OC(C)(C)C)NC(CNC(CCC=C)=O)(C)CO 42462,c1(C(=O)NC(CNC(C(CC=C)(C)CC)=O)CO)cc(S(N)(=O)=O)sc1C 42463,C1(C(=O)Nc2ccc(COC)cc2)CCC(C)(C)N1C(=O)C(F)Br 42464,C(=O)(C(C(C)(C)NC(C)=O)N1CCC(OCCO)C1)NC(C)C.c1(CC)ccccc1 42465,c1(COC(=O)C(=O)NC(CC(=O)OC)c2ccccc2)ccc(F)cc1F 42466,CCCC(C)CN=c1cc[nH]cc1S(=O)(=O)NC(c1c(C)noc1C)C 42467,c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C(CO)C2)cccc2nn[nH]c12 42468,N1(C(C2(NC(=O)CCC3OCCO3)CCCC2)=O)CCC2C(C1)C2(F)F 42469,c1(C(=O)OCC)cc(NCC(C)NC(C2(C)CC2(C)C)=O)n2nccc2n1 42470,c1(NC)cccc(C(=O)NCCC(C(C)C)NC(c2nocc2C(C)(C)C)=O)n1 42471,c1(C(CC)(C)O)cn(CCC2CN(C(c3coc(C(C)(C)C)n3)=O)C2)nn1 42472,CC1(C)CC(O)CN(C(=O)Cc2ccc(SCCC#N)cc2)C1 42473,CCC(C)(C)C(O)C(=O)N1CCCCC(CNC(C2CN3CCN2CC3)=O)C1 42474,c1(NC(C2CCN(C(C3(O)CCSC3)=O)CC2)C)ncc([N+](=O)[O-])cc1CO 42475,c1(C(=O)NCC(C)NC(=O)C(C)(C)CS(N)(=O)=O)cc2c(cc1Cl)NC(=O)C2 42476,c1(C(N(C2CCN(C(=O)CCCC(C)(C)C)CC2)CC)=O)ccnc2ncnn12 42477,c1(C(=O)NCC)ccc(CN2CCCCC2CN2CCCS2(=O)=O)cc1 42478,Cc1n[nH]c(C)c1CC(N1CC2C(CNC(=O)C(C)(C)C)C2C1)=O 42479,C1(C(N(CC(CC)NC(c2c(CC)non2)=O)CC)=O)CC(F)(F)C12CCC2 42480,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2CN(C(=O)Cn3cccn3)CCC12 42481,CC1CCC(CNC(c2cc(CO)[nH]n2)=O)CN1C(=O)COC1(C)CCOCC1 42482,c1(C(C(=O)O)NC(=O)NC(c2nc(C(F)(F)F)cs2)C)cccc(Cl)c1 42483,c1(SC)ncc(Cl)cc1C(=O)NCC#CCN(C1CC1)C1CC1 42484,C1(NC(C2(OC)CCC2)=O)CCN(C(C2CC(CSC)C2)=O)CC(C)(C)C1 42485,CCCC(CCC)C(=O)NC1CC1NC(=O)CCC1(C)CC1 42486,Cc1nnc2c(C(=O)NC(C)C(C)NC(c3ccncc3N)=O)cccn12 42487,c1(Cc2nnnn2C2CC2)cccc(C(F)(F)F)c1.C(COCCO)SC 42488,c1(C(=O)NC2CC(C)N(C(=O)Cc3ccnn3C)CC2)cncc2[nH]ccc12 42489,C1(C(CC)=O)COCCN1C(=O)CN(C(C1CC(F)CN1C)=O)C(C)C 42490,C(=O)(C1=CC2CC(C1)CC2O)NC(CNC(Cn1nc(C)oc1=O)=O)C(C)(C)C 42491,S(=O)(=O)(c1ccc(F)c(C(N2CCN(C)C(C(C)C)C2)=O)c1)NC(C)C 42492,C1(C2CC2)(CNC(=O)CCN2CCCCC2=O)CCN(C(=O)C(O)C2CCCC2)C1 42493,N1(C(c2c(CNC(C(CC)C#N)=O)nnn2C)=O)CC2(CO)CC2(CO)C1 42494,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)C=C2CCSCC2)CC1O 42495,c1(C(=O)Nc2ccc(C3CCCCCC3)nc2)cnc(Br)nc1 42496,CCCC(C)(CCC)C(=O)N1CCC(CO)(NC(=O)CN(C)C(C)=O)C1 42497,c1(NCCCCC#CC)cc(=NCC(C(C)C)C2CCCCO2)[nH]c(C(C)C)n1 42498,C1(CCC(=O)NC(C2(CNC(=O)C(=O)Nc3cccnc3)CC2)C)CCN(C)CC1 42499,c1(C(=O)NC2CCN(C(CC(C)c3ccco3)=O)C2(C)C)ccc2[nH]ccc2c1 42500,CCC(Cc1ccccc1)C(=O)NCC(C)(Cn1cccn1)NC(=O)CCF 42501,Cc1nc(CCCC(=O)NCCC2CC(NC(c3cscc3C(N)=O)=O)C2)cs1 42502,C1(CC)C(C(N(C)CP(C)(C)=O)=O)CCCN1C(c1ccccc1F)=O 42503,N1(C(COCCCOC)=O)CCC2(CCCN2C(=O)CCn2cccc2)CC1 42504,C1(NC(COCC(=O)NC)=O)CC2CC(CNC(=O)CCC3CCOC3)CC12 42505,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42506,c1(C(N2CCC(NC(CCOCC)=O)(CO)C2)=O)cc2occc2n1C 42507,C1(CC(=O)NC(C(=O)NC(C#C)C(C)OC)C2(C)CC2)CCCCN1C 42508,CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CC(CCNC(C2(C(N)=O)CCC2)=O)O1 42509,c1(C(=O)NCC(CC(=O)N(CC(=C)C)C)OC)cnn2c1OCC2 42510,C1(c2nnnn2C)(NC(c2cnn(C)n2)c2nnnn2C)CSCCSC1 42511,N1(C(C(C2CCCC2)OC)=O)CC(NC(c2cc(CC3CC3)on2)=O)C(F)C1 42512,c1(COCC)nc(NC(=O)CCc2cncc(Cl)c2)sc1-c1ccc(OC)cc1 42513,C1(C(=O)OC)CN(C(=O)C(=O)N(C)C)c2ccccc2O1.c12cc(n[nH]1)NC2 42514,c1(C(N2CCC3(C(NC(COCC)=O)C3)C2)=O)scc2c1OCCO2 42515,C(=O)(CC(C(C)C)C(C)C)NC(CCNC(C1C(=C)CC1)=O)(C)C 42516,Cc1cnn(C)c1CNC(C1C2CN(C(=O)Cc3ccsc3C)CC12)=O 42517,C1(C(C)C)C(NC(=O)C(C)NC(=O)CC(C)(C)C)CCN1C(=O)CC1CCSCC1 42518,C1(CNC(c2nc(CC)oc2)=O)CC(C)(C)CN1C(c1cnccc1Cl)=O 42519,c1(OC)c[nH]c(C(N2CC(C)(C)CC2CNC(C2CC(C)(C)CO2)=O)=O)cc1=O 42520,CCC(C)C(C(=O)N1CCC(CCO)CC1)NC(=O)C(C)C 42521,N1(C(C(C)Cc2ccc(F)cc2)=O)CC(CO)CC(C)C1 42522,CC12CC1CN(C(=O)C(N1CCN(c3ccccc3F)CC1)=O)C2 42523,c1(OCCC)ccc(C(=O)NC2CCCN(C(=O)C(O)CC3CC3)CC2)cc1N 42524,N1(C(C(CC)OCC)=O)CCC(C(=O)NCC(C)F)C1(C)C 42525,C1(O)(CNC(=NCC=C)NCc2nc(C)cc(C)n2)CCC2(CC1)OCCO2 42526,O=C(C1COc2ccccc21)NCC12CCC1CCN2C(=O)CCOC1CC1 42527,C=C=CCCC(=O)N(c1ccccc1)CCCOCCNC(=O)CCC1CC1(C)C 42528,C(C(C(=O)N1CCCC1CN(C)C1CC1)C(C)C)NC(Cc1c(C)n(C)cn1)=O 42529,c1(CC(=O)NCCC(CNC(=O)Cc2cnoc2)O)nnc(S)nc1O 42530,S(=O)(=O)(CCC(=O)NC1CN(C(c2ccoc2C2CC2)=O)CCC1F)NC 42531,C(C(O)CS(C)(=O)=O)NC(=O)NCc1sc(C)c(-c2ccccc2)n1 42532,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1O 42533,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1C(C)C(NC(=O)CCNS(C)(=O)=O)CCC1 42534,C1(C(=O)NCCCN(C(c2cc(O)nn2C)=O)CC)OCCOC12CCC2 42535,N1(C(C23CC(OC)C2C3)=O)CCC(CCNC(c2ncccc2Br)=O)CC1 42536,C1(C(=O)NC(CC)CNC(C2CC(F)(CC)C2)=O)COCCN1CC 42537,C=CC(C)CC(=O)N(C1(C(=O)NC2CC(CO)C2)CC1)C 42538,O=C(C1=CCN(C(=O)C(F)F)CC1)NCC1CC1[N+](=O)[O-] 42539,C(=O)(C(F)(F)C1=CCOCC1)N(CC(C)NC(=O)C1CCc2ccccc21)CC 42540,c1(CCN(C)C)ccc(C(=O)NC23CC(NC(C4CC45CCC5)=O)(C2)C3)cc1 42541,C1(C(=O)NC2C(C)CCN(C(c3n(CC)nnc3)=O)C2)CCc2nc(O)[nH]c2C1 42542,c1(C(=O)NCC(CNC(C2CC=CCC2C)=O)OC)ncc(F)cc1F 42543,C1(NC(C(=O)NCc2ccccc2)=O)CCCCC1Cc1cc(Cl)ncn1 42544,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CCN(C(C)=O)C(c2nccn2C)C1 42545,C1(CSC)CCN(NC(C(=O)NC(c2nc[nH]n2)=O)C2CC2)C1 42546,c1(C(=O)NCC2C3CN(c4c(C#N)nccn4)CC32)cc2cc(Cl)cnc2[nH]1 42547,C(CCCC(=O)NCC(O)C(=O)Nc1cccc(F)c1O)(OC)OC 42548,N1(C(C(C)NS(C)(=O)=O)=O)CC2CC3CC2C1C3NC(c1cc(Cl)ccn1)=O 42549,c1(CN2C(CC(=O)Nc3c(C(=O)OC)csc3C)CCC2)c(O)ccc(Cl)c1Cl 42550,N1(C(C(C)Sc2ccc(F)cc2)=O)CCN(C(=O)CNC=O)C(c2nccn2C)C1 42551,c1(CC(C(C(CC)O)c2ccccc2)=O)cc(-c2nn[nH]n2)n(C(C)CC)n1 42552,Cc1cc(C(N2CCN(C3CCN(C(C4COC4)=O)C3)CC2)=O)cnc1C 42553,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3ccsc3C)C2)cc1CO 42554,C(C(C(=O)N1CCC(NC(=O)OC(C)(C)C)C(O)C1)C(C)(C)C)OCC(C)C 42555,c1(C(=O)NCCCNC(c2ncc(C#C)cc2C)=O)ccc2c(c1)NC(=O)CC2 42556,C1(C)(CC(N2C(C(=O)NC3CCCN(C)C3)CCCC2)=O)CCS(=O)(=O)N1 42557,C(=O)(C(C)(C)C(=O)OC(C)(C)C)NC1CN(C(C2CC(C)OCC2)=O)C(CO)C1 42558,Cn1ncc2cc(C(N3C4CCC3CC(NC(c3c[nH]nc3F)=O)C4)=O)cnc12 42559,CCCC(CCC)CCCC(=O)N(C)CCNC(c1cc2c(cn1)CCCC2)=O 42560,CC(C1CC1)=C(F)C(=O)NC(C)C(C)NC(C1(CN(C)C)CC1)=O 42561,c1(C(=O)Nc2c(CC)cccc2)cc2c(-c3ccc(F)nc3C)cncc2s1 42562,CCS(=O)(=O)c1ccc(S(=O)(=O)Nc2csc3c2C(C)CCC3)cc1 42563,C1(CC(=O)NCCn2ncc(C)c2)CCCN(C(c2ccc(F)nc2)=O)C1 42564,Cn1cc(Br)c(C(=O)NCC2C=CC(NC(=O)C(c3ccccc3)O)C2)n1 42565,c1(C(N(C(CNC(C(c2ccc(C)o2)C)=O)C)C)=O)nc2ccccc2[nH]1 42566,N1(C(c2cccc(C#C)c2)=O)CCCC(NC(=O)COCC2(F)CC2)C(F)C1 42567,C1(C(=O)NC2C(NC(CC(CN(C)C)O)=O)CCCC2)Cc2cncn2C(=O)N1 42568,C#Cc1c[nH]nc1C(=O)NC1CN(C(c2csnc2C2CC2)=O)CC1O 42569,c1(C(=O)NCC2(F)CC(NC(c3c(CCC)n(C)nc3)=O)C2)cc2ccsc2s1 42570,N1(C(CN2CCC(C)(O)C2)=O)CC2CC(NC(=O)CN3CCNC(=O)C3)C(C2)C1 42571,C=CC(CC)CC(=O)NC(C)CCCNC(=O)Cc1cc(F)cc(F)c1 42572,C(=O)(CC(=O)NC1COCC1C(=O)NCC(C)(C)CSC)NCC#C 42573,C(=O)(C(CCCOC)NC(=O)C(=CC1CCCC1)C)NC(C#C)CCCC 42574,c1(C(C)NC(c2csc(Br)c2)=O)ccnc2ccc(O)cc12 42575,C1(C(=O)NCC2(COC)CCC2)CCN(C(c2cc(C)[nH]n2)=O)C1C 42576,C1(CNC(CC(C)(C)C2CC2)=O)CC(F)(F)CN1C(=O)CC1(CO)CCCCC1 42577,c1(C(=O)NC2C(NC(C(CC#C)(C)CC)=O)CC2)ccc2ccccc2c1 42578,c1(OC)cc(C(=O)NC2CCC2NC(C2CC(C)(O)C2)=O)ccc1O 42579,C#CCCC(C(=O)NC1CCCC(O)C1O)NC(C1COCC(C)O1)=O 42580,C(C(=O)N1CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1)(C(C)C)OCC 42581,CCC(C(=O)N(C)CC1(O)CN(C(=O)CN2CCCC2)C1)n1cncn1 42582,C(C(C)C(F)C(=O)N(C1CC(C(N)=O)C1)C)NC(C(C)C1CC1)=O 42583,N1(C(CC2ON=C(CC)C2)=O)CC2(CCCC2)C1C(=O)NCCCc1nccs1 42584,C1(CC=C)(NC(c2ccnn2C)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 42585,N1(C(CC2CCC(C)C(C)C2)=O)CC2=C(C1)CN(C(=O)COc1cnn(C)c1)C2 42586,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42587,c1(CC(=O)NCC(CNC(=O)C(O)CC2CC2)OC)c[nH]c2cccc(Cl)c12 42588,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NCC(C#C)OC)C12CC2 42589,c1(C(C)NC(C2N(C(COCC#C)=O)CC=C2)=O)nc(C)oc1C 42590,C1(O)(N(C(C)=O)C)CCN(C(=O)NCc2ccccc2C)C1 42591,N1(C(C=Cc2c(C)n[nH]c2)=O)CC2CN(C(=O)CC3CCCN(C)C3)CCC12 42592,c1(CN(CCCN(C)C(=O)NC(C)C(C)(C2CC2)OC)C)ccn(C(C)(C)C)c1 42593,N1(C(c2cn(C(C)C)nc2)=O)CC(n2cc(C(O)C3CC3)nn2)C(C)C1 42594,N1(C(C=C(CC)CC)=O)CCN(C(c2ccn3c(O)nnc3c2)=O)C2CCC12 42595,CC(C)S(=O)(=O)c1cccc(C(N2CCC2CNC(c2ccsn2)=O)=O)c1 42596,N1(C(c2c(C)nsc2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC(CO)C1 42597,CC(C)C(C)CC(=O)N1CC(N(C(=O)CCc2cc(Br)ccc2F)C)C1 42598,N1(C(CC2C(C)(C)CCO2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 42599,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42600,c1(OC2CCN(C)CC2)ccc(NC(N2CCC(NC(C)=O)CC2)=O)cc1Cl 42601,c1(C(N2C(CNC(c3cccc(CC=C)c3)=O)CC2)=O)nn(C)c(C)c1N 42602,N(C(=NCCC(C)C)NCC1(C)CCC(NC(C)=O)CC1)C1CN(C(=O)OC)C1 42603,C1(C(=O)NC(CC(C)C)CNC(C2CN(C)C(=O)N2)=O)CC(C2CCCC2)C1 42604,C1(C)(C(=O)NCCNC(C(C)N(C)C)=O)CC(F)(F)C1.c12cn(nn1)C2 42605,C1(CNC(CN(C(=O)C(O)C2CCCC2)C)=O)CCCCC1C(N1CCOCC1)=O 42606,C1(C(N2CCN(S(=O)(=O)c3cccs3)CC2CC#N)=O)CCc2ccccc2O1 42607,N1(C(C(c2scc(C)n2)C)=O)CCC(C)(C)C(CNC(=O)C(F)(F)C2CC2)C1 42608,N1(C(C(COCC)NC(=O)CC(=O)NC)=O)CCC(C)C(C2CC2)C1 42609,c1(C(N(C(C=C)(C)C)CCOC)=O)cn(CCCNC(c2cc(C)cs2)=O)nn1 42610,CCCCCCC(CC)(CC)C(=O)N(CCCNC(=O)CNS(N)(=O)=O)CC 42611,C1(CCNC(=O)NC2CC(CC(=O)OC)C2(C)C)CCC(F)(F)CC1 42612,C(C)(C(C)S(C)(=O)=O)NC(C(=O)NC1CN(C(C)C)C(=O)C1)=O 42613,N1(C(=O)OC(C)(C)C)CCCC1C(C)(C)CO.c12cnc(o1)oc2=O 42614,c1(C(=O)NCc2c(C)nn[nH]2)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)C2 42615,c1(NC(C2(C)CCN2C(c2cccc(Cl)c2F)=O)=O)ccc2ncccc2c1 42616,C1(C(=O)N(C(CCCC)C)CC)N(C(C)=O)CCC1(C)C 42617,c1(CCC(=O)N(C2CC(C)(OC(F)F)C2)C(N)=O)cncc(F)c1 42618,c1(C(=O)NC2CC(F)(CNC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42619,c1(N(CC=C(C)C)C)cc(C)[nH]c(=NCC2CCN(C(C3CCCCC3)C)C2)n1 42620,N1(C(C23CC(OC)C2C3)=O)CCCC(O)(CN(C(=O)Cc2ccc(N)cc2)C)C1 42621,c1(C(=O)NCC(=O)NC(c2ccc(C)s2)C)cnc(C)c(C)c1 42622,c1(C(=O)NC2(CNC(c3cccc4ncnn34)=O)CCC2)ccc(O)c(F)c1F 42623,c1(CC)ccc(C(=O)N(C)CC2CCN(C(C3CC(=O)NC3(C)C)=O)C2)c(C)n1 42624,N1(c2nc(C)nc(=N)[nH]2)CCC2CS(=O)(=O)CC2C1 42625,c1(OC(C)C)ccc(C(=O)NCC(CNC(=O)COCC2CCCO2)CO)cc1 42626,C(C(C)C(=O)N(CCCO)C(c1cccnc1)C)OCCNC(C)=O 42627,C1(C(C(=O)NCCN(C)C(C2(C)CCCN2C)=O)(C)C)CCC(O)CC1 42628,c1(C(CC)C(=O)N(CC(O)CNC(=O)C(C)=CCOC)C)ccc(F)cc1 42629,C12(CC(=O)NCCCSC)CCC1CN(C(=O)CCCNC(C)=O)C2 42630,N1(CCN(C)C(c2cccc(F)c2)=O)CCN(C(=O)Cc2ccncc2Cl)CC1 42631,c1(-c2cc(C(N3CCC(=CCC)C3)=O)n[nH]2)cncc(N2CCOCC2)c1 42632,c1(C(CCO)NC(CC(CC)(C)C)=O)ccc2c(c1)OCCO2 42633,c1(C(=O)NC2CCCC(NC(c3nsnc3O)=O)C2)ccc2nc(Cl)nn2c1 42634,N1(C(CC2(OC)CCC2)=O)CC2=C(C1)CN(c1ncc(Br)c(C(=O)OC)n1)C2 42635,Nc1c(CNC(=O)NC2CCCC2c2cccc(Br)c2)cccc1F 42636,c1(C(N(C(C)CNC(=O)Cn2cccn2)C)=O)ccccc1C1(C#N)CC1.C1CC1 42637,c1(C(=O)NC(CCNC(c2c(C)[nH]nc2C(C)C)=O)C)cnc2nccnc2c1 42638,c1(OCC)ccc(C)cc1.N12CC(C)(C1)CCOCCC(=O)NCCC2=O 42639,C1(N(C)C)CCOC(C(N2CC(O)(c3cn(CC4COCCO4)nn3)C2)=O)C1 42640,C(C(=O)NC1CCC1CNC(C12CCC(CC1)CC2)=O)(C(C)(C)C)SC 42641,c1(OC)nc(NC(C2C3CC2N(C(c2c(O)cc(O)cc2O)=O)C3)=O)c(Cl)cc1Cl 42642,c1(CSC)cc(C(=O)NCC2C(C)CCCN2C(=O)CC(=O)N(C)C)ccc1F 42643,CC(C)(CNC(=O)NC1CCCC1)CC1CCN(C(=O)CCOC(C)(C)C)C1 42644,CCC(C(=O)N1CCOCC(CNC(c2sc(CC3CC3)nc2C)=O)C1)C(C)(F)F 42645,C(CCC(F)(F)F)N(C(C1N(C(Cc2c(C)con2)=O)CC1)=O)C 42646,c1(C(N(CCCCCC)CCNC(=O)C(C)C#N)=O)ccc2nonc2c1 42647,CC(C)CC(C)(CNC(=O)C(C)(C)n1cnnn1)NC(c1ccnn1C(F)F)=O 42648,c1(C(N2C(CNC(CCC=C(C)C)=O)C=CC2)=O)cnc2ccc(C#N)cn12 42649,Cc1ccc2[nH]c(C(=O)NCCC(C)(C)CNC(C3(CO)CCC3)=O)cc2c1 42650,CC(CCN=c1nc2c3cc(ccc3[nH]1)OCCN(CCN(C)C)C2)=C1CC1 42651,c1(C(CNC(C23CC(C)C2C3)=O)NC(C2(CC(F)F)CCC2)C)ccccc1F 42652,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42653,Cc1cc(Cl)cc(C(=O)NCCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42654,CCC(CC)NC(=O)CO.C1(=O)CC=CCN1.C1(=O)CN1 42655,c1(OCC)cccnc1C(N1CC(O)(CCNC(c2cccc(F)c2)=O)C1)=O 42656,N1(C(COCCCCC)=O)CCCC(C2CN(C(c3cnn(C(C)C)c3)=O)C2)C1 42657,c1(C(=O)NC2(CN(C(C=CC(C)C)=O)C)CC2)cccc(C(C)C)n1 42658,Cn1ncc(C(F)(F)F)c1C(=O)NC1(CNC(=O)C2=CCCC2)CCOCC1 42659,C(=O)(C(C)CC(F)(F)F)NC(c1occ(C(N(CC(C)C#N)CC)=O)n1)C 42660,C(=O)(CCn1ccnc1)N(C1(CC(=O)N(CC(C)O)C)CC1)C1CC1 42661,c1(-c2cn(C3CCC(C(=O)NC(C4CCOC4)(C)C)C3)nn2)ccc(CO)cc1 42662,c1(NC2(C(=O)OC)CC3CCC(C3)C2)sc2cccc(F)c2c1C 42663,c1(C(N2CC(NC(=O)C(F)(F)CO)CC(C)C2)=O)nc2cccnc2s1 42664,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42665,N1(C(C2C(CC)C2)=O)CCC(n2ccc(C)n2)CC1.n12cc(nn1)CC2 42666,c1(CC(=O)NC(C2CCN(C(C3CC=CC3)=O)C2)C)ccc(C(F)(F)F)nc1 42667,N1(C(C)=O)CCCC(NC(=O)CCOCCNC(=O)Cn2cccc2)CC1 42668,C(=O)(CC(COC)COC)NC(CC=C)CNC(C1CCNC(=O)C1)=O 42669,N1(C(CN(C2CCCCCC2)C)=O)CC2CCN(C(=O)C#CC3(C)CC3)CC12 42670,c1(OCC(N)=O)ccc(C(=O)NCCNC(=O)C=CSc2ccccc2)cc1 42671,c1(CC(=O)N(C2CCN(C(c3ncccc3Br)=O)C2)C)ccc(O)cn1 42672,C1(NC(c2c(CC)c[nH]n2)=O)CCN(C(=O)CSc2cccc(F)c2)CC1(C)C 42673,C(=O)(C1COc2ccccc21)N1C(C)(C)C(NC(C2(F)C(C)(C)C2(C)C)=O)CC1 42674,c1(N(CCOC)CCNC(C2CCC(=O)N2)=O)nc(C)cc(C)n1 42675,N1Cc2ccc(Cl)cc2C1.c1(O)ccccc1NCCN1CC1CCN(CC)CC 42676,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42677,N1(C(CCC#C)=O)CCN(C(c2cc(CCCC)n(C)c2C)=O)C(C)C1C 42678,c1(C(=O)NCC(C)(C)CNC(CC(CCCC)O)=O)ccc(S(N)(=O)=O)cc1Cl 42679,c1(CC(=O)NC(CC=C)CO)cn2cc(-c3cc(C)cs3)ccc2n1 42680,N1(C(C(C)(C)F)=O)CC2(CCC(C(=O)Nc3ccc(Cl)c(C#N)n3)O2)C1 42681,c1(C(=O)OC)nc(Br)cnc1NC(C1CCC(C)N1Cc1ncc(Cl)cc1C)=O 42682,C(=O)(CS(=O)(=O)C1CC1)N1CCN(C(C(C)(C)C2(O)CCC2)=O)CC1C1CCCC1 42683,C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2ccccc2)CC2CCC1C2 42684,C1(C(=O)NCC2C(CNC(C(CCC)=CCC)=O)C2)COC2COCC2O1 42685,c1(C(N2CCCC(C(N(CC(=C)C)CC)=O)CC2)=O)ccc2[nH]nc(Cl)c2c1 42686,CCCN=C(NCc1ccc(SC)s1)NC1CCOc2ccccc21 42687,c1(CC)cc(C(=O)NC(C2CN(C(=O)CC3CC(CC)CO3)C2)C)on1 42688,C(=O)(CS(=O)(=O)C1CC1)N1CCC(C2N(C(CSCC=C)=O)CCC2)C1 42689,C(=O)(C1=C(Cl)CCCC1)N1CC(NC(C(=Cc2ccncc2)C)=O)C(CO)CC1 42690,N1(C(c2cc(C)sc2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42691,c12ccc(Br)cc1NC(=O)CCc1ccccc1-2.N1(CC)CCC(O)CC1CC 42692,C(C)(C(=O)NC1CC(NC(=O)CCc2nc[nH]n2)C1)=CC 42693,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 42694,C1(NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1CNC(=O)C=CBr 42695,c1(OC)cc(C=CC(=O)NCc2ccc(CNC(C3CCNC3=O)=O)cc2)sn1 42696,Cc1ccncc1C(c1nnnn1CC1CCOC1)NCCc1cn(C)nc1C 42697,c1(C(NCP(=O)(O)O)C(N2CC3CCN(C(CC)=O)C3C2)=O)ccc(C)cc1[N+](=O)[O-] 42698,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OCC 42699,N1(C(C(CC=C)C)=O)CCCCC(NC(c2cc(-c3ccc(F)cc3)sn2)=O)C1 42700,C(=O)(C(C)(C)C(C)O)N(CCCCC(=O)N(C)CC)C.N12CCC(C1)CCC2 42701,c1(SC)cccc(NC(C2(CCCF)CN(C(C)CC(N)=O)C2)=O)c1 42702,c1(C(N2C(C(C)(C)NC(C(C)C3CCC3)=O)CCC2)=O)cnn2c1CCC(C)C2 42703,c1(N2C(Cc3c(C)n(-c4cc5sccc5s4)nn3)CCC2)cc(C)ncc1C 42704,c1(CC(=O)NC(C2CCN(C(C3(OC)CC3)=O)CC2)C)ccc2cccnc2c1 42705,CC1CC(CNC(c2cccnc2)=O)CN1C(=O)CCCC1CCCC1 42706,CC1Cn2nc(C(=O)NC3CCN(C(c4cc5c(s4)CCC5=O)=O)C3)cc2CN1 42707,C#CC1CN(C(=O)C(C(C)OC)NC(=O)C(O)Cn2cncn2)CCO1 42708,N1(C(C(C)Cc2ccncc2)=O)CC(NC(c2cncc(F)c2)=O)CC12CCC2 42709,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 42710,N1(C(CC(C)OC)=O)CCCC(C)(NC(c2ccc(O)cc2C(F)(F)F)=O)C1 42711,N1(C(=O)CCCCn2cc(CC3CCCC3)nn2)CCc2oncc2C1 42712,Cc1ccc(O)c(CNC(=O)CC=CCNC(c2cn(C)cn2)=O)n1 42713,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)CCCC1CCOCC1 42714,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 42715,CC1(C(=O)NCCC2CCCN(C(c3ccc(O)c(N)c3)=O)C2)CCC12CCC2 42716,Cc1ccc(CC(=O)NC2CC(NC(=O)CC3COC4CC3C4)C(O)C2)c(Cl)n1 42717,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)N(C1CC1(C)C)C 42718,Cc1cnc(C(N2CC(C(O)C(=O)NCCN3CCC(C)C3)C2)=O)cn1 42719,c1(C(=O)OC)c(C)cc(CCNCCC(F)(F)CO)cc1I 42720,c1(C(=O)NC(C)CN(C(=O)CO)C)ncccc1Br 42721,C1(C(N2C(C)C(NC(c3ccc(CC#N)cc3)=O)CC2)=O)CCCC(F)(F)C1 42722,c1(C(C(=O)N(C2CN(C(C3CCCN3C)=O)C2)C)OC)ccc(F)cc1 42723,C=CC1(C(N2CCC(C(=O)NC(C#C)CC(C)C)C2)=O)CCCCC1 42724,CCCCC(O)C(=O)N1CC(NC(=O)CCCCCC)C(c2cnn(C)c2)C1 42725,C1(OC)CC(NC(C2(C)CCC2)=O)CN(C(=O)C(C2CCC2)C2CCC2)C1 42726,C1(OC)CN2CCCC2(C(=O)NC2CC(CN=c3nc(-c4ccoc4)[nH]s3)C2)C1 42727,c1(C(=O)NC(C)CN(C)C(C23CCCC2C3)=O)cnc(N(C)C)c([N+](=O)[O-])c1 42728,C1(C(N)=O)CC(F)CN(C(=O)CC2CCN(C(=O)Cc3ccc(O)cn3)C2)C1 42729,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 42730,c1(C(N2CC(C)(CC(=O)Nc3cc(C4CC4)[nH]n3)C2)=O)cccc(C(N)=O)c1 42731,C(C(=O)N=S(C)(=O)N(C)C)c1nc(NC(C(CC)CC)=O)sc1.c12cc(ccn1)CS2 42732,c1(OC)cc(NC(C)=O)ccc1N1CCOCC1.S1(=O)(=O)CCOCC(=O)N1 42733,C1(CCNC(C2(F)CCCCC2)=O)CCN(C(C2CCCCO2)=O)CC1 42734,N1(C(CC2(OCC)CCC2)=O)CC(C)C(C)(C(=O)N(C(CC(C)C)C(N)=O)C)C1 42735,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1CCOC1)=O 42736,N1(C(C2CCN(C(C(=O)NC(C)C)=O)C(C)C2)=O)CC(C#N)C2(CCC2)C1 42737,N1(C(=O)CC2CCS(=O)(=O)C2)CCCN(C(C2CCS(=O)(=O)N2)=O)CCC1 42738,c1(OC)ccc(F)c(C(=O)NCCCNC(=O)C=CCNC(=O)OC)c1 42739,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 42740,C1(COC)(NC(C2CN(S(N)(=O)=O)C2)=O)CCCN(C(=O)Cc2cccnc2)C1 42741,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 42742,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 42743,c1(CN=C(NC(c2c(OC)cccc2)COC)NCCF)c(C)nn(C)c1C 42744,c1(NC(C2CC3CC3N2C(c2n[nH]c3c2CCCC3)=O)=O)nc(Br)c(Br)cc1Br 42745,C1(NC(C(CCC)N(C)C)=O)CN(C(=O)CNC(C)=O)Cc2nccn2C1 42746,C(=O)(CC(C=C)CC)NCC(C(=O)N(CC#C)C)CC1CCCC1 42747,c1(CC(N2CCC(O)(C(C)NC(C(C)n3cncn3)=O)C2)=O)c(O)ncnc1O 42748,C1(OC)CC2CC(C(=O)NCCCC(C)NC(=O)CC3CC(=O)C3)CC12 42749,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 42750,c1(CNC(c2cc(-c3ccc(F)cc3)no2)=O)cnc2[nH]ccc2c1 42751,C1(CC(N2CC(O)(CNC(C(CN(C)C)N(C)C)=O)C2)=O)COCC2(CCC2)O1 42752,CCCCC(O)C(=O)NC1CC1NC(=O)CCNC(=O)Nc1ccoc1 42753,N1(C(C(C2CC2)OC)=O)CC(O)(CCNC(C2(c3ccccc3)CC(C)C2)=O)C1 42754,c1(C(=O)NCC2C(NC(C(CC)COC)=O)C2)cc(Br)cc(Cl)c1C 42755,C(=O)(C1=CCCCCC1)NC1(CCO)CN(C(c2nc(C)n(C(F)F)c2)=O)C1 42756,C(=O)(CCCC(=O)N1CCC(O)C1)NCC(N1CCC(O)(C(F)(F)F)C1)C 42757,C1(NC(c2cc(Cl)ccn2)=O)COC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 42758,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(F)c(N)c(F)c1 42759,N(C1CS(=O)(=O)Cc2ccccc21)NC(NC(CC#C)C)=NCCCF 42760,C1(C(=O)NCC2OCC3(CN(C(C=CC=CC)=O)C3)C2)CCC(C2CCCO2)O1 42761,C1(OC)CCC(CC(N2CCCC2CNC(=O)CC2CCCC(CN)C2)=O)CC1 42762,C1(NC(C(C(C)C)NC(=O)OCC)=O)CC2(CCN(C(C3CC(C)C3)=O)CC2)C1 42763,C(C)(CN=c1nc2scnc2c(N2CCN(C)CC2)[nH]1)c1cc(OC)ns1 42764,C(C(O)CO)N(C(=O)CC=CCNC(=O)C(C)OCOC)C 42765,C1(OCC(=O)OC)CCN(C(C2C(C)OC(C)C2C)=O)C1(C)C 42766,CC(C)CC(C(=O)N1CCCC(NC(=O)CN(C)C(N)=O)C1)Nc1ccccc1 42767,C1(NC(COC2(C)CCC2)=O)CC2CC(C1)N(C(C1CC3CCC1O3)=O)C2 42768,C1(C(C)NC(=O)CN(C)CCO)CCCN(C(=O)CCCn2cccn2)C1 42769,C1(c2ccccc2)(C(=O)NCC(CO)NC(COC(C)C)=O)CC=CCC1 42770,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 42771,c1(SC)cn(C)nc1C(N1CCC(C(C)(C)NC(=O)CS(C)(=O)=O)C1)=O 42772,c1ccc(C2CC(NCC3(C4CCCO4)CNC3)C2)cc1 42773,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 42774,c1(N(C(C=C)C)C2CC2)ncc(S(=O)(=O)N2CCCC(c3ccco3)C2)cc1Cl 42775,Cc1ccc(SCCC(=O)NCC2(F)CCC(CNC(C3CC3(C)C)=O)C2)cc1 42776,c1(N)ccccc1Cl.C12(F)CC(C1)CNC(=O)C(=O)NC2.CCC(=O)C(CN)=O 42777,C1(NC(c2n(C)cc(Br)n2)c2nnnn2C2CCCC2)CC2(CCCC2)C1 42778,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(-c3ncc[nH]3)c1)=O)C2)OC 42779,CC1=C(C)CC(C(=O)NC(C)C=CC(N2CCCC2C2(C)CC2)=O)CC1 42780,C1(CCC)(NC(=O)Cc2c[nH]nc2O)CCN(C(C23CCOC(C)(C2)C3)=O)CC1 42781,C(C(CC(C)C)NC(c1ccc(F)cn1)=O)NC(CC1(CSC)CC1)=O 42782,C(C)(CC(C)NC(=O)Cc1sccc1C)NC(C1(OCC)CCC1)=O 42783,N1(C(C2(C)CC(F)(F)C2)=O)CCN(C(c2ccc(F)s2)=O)CC1CF 42784,CC1CCN(C(=O)CCc2nc(CNC(c3cnoc3)=O)no2)C(C(N)=O)C1 42785,C1(NC(CNC(N)=O)=O)CCC12CCN(C(C13CCCCC1C3(F)F)=O)CC2 42786,c1(C(N(CC(C)N(C(=O)C=CS(C)(=O)=O)C)C)=O)cc2cc(F)ccc2o1 42787,c1(C(=O)NC(C2CCN(C(c3nnc(C)s3)=O)C2)C)cc2cccnc2s1 42788,C(=O)(C(=O)C(C)(C)CC)NC(CC(N1CC(C)(OC)C1)=O)C1CC1 42789,C#Cc1cc(C(=O)NCC(C)CN(C)C(C2(C)CCCS2(=O)=O)=O)ccc1C 42790,c1(C(=O)NCC23C(CN(C(C(C)=O)=O)C2)C3)cc(Cl)cc(Cl)c1O 42791,CCCC(CC)CC(=O)NC1CC(NC(c2c(N)cc(F)cc2F)=O)C1 42792,C1(NC(Cc2c(C)n[nH]c2)=O)COC2C(NC(=O)CCCC(F)F)COC12 42793,c1(C(=O)NC2(CS(=O)(=O)NC)CCCCC2)cc(C)nc2c1c(C)nn2C 42794,c1(SCC(N2CCC(c3ccccc3)C2)=O)nc(Cl)cc(Cl)n1 42795,Cc1cc(C#N)nc(NCC(C2CC2)NC(c2ccc(Cl)cc2C(F)(F)F)=O)n1 42796,N1(C(CN(C(C)=O)C)=O)CCC(CO)(NC(=O)C(N2CCCCCC2)C)CC1C 42797,Cc1nc(C(N2CC3(NC(c4ncoc4C)=O)CC2C3)=O)n(C)n1 42798,N1(C(=O)NC2CCC(NC(CC)C)C2)CCN(c2ccnc(OC)n2)CC1 42799,C12(NC(c3ccc(=NCC)[nH]c3)=O)CCOCC1CN(C(=O)C(C)CN(C)C)C2 42800,C1(c2cn(C3CC(C)SCC3)nn2)CCc2n[nH]cc2C1 42801,c1(CC(=O)NC2CN(C(c3cccn3C3CC3)=O)CC2O)ccc(Cl)c(F)c1 42802,O=c1cccnn1CC1CCC(c2ccccc2)CC1 42803,Cc1ccc2cc(NC(C3CN(C(=O)C(C)n4cccn4)CCN3)=O)ccc2n1 42804,C(=O)(C1=CCCOCC1)N(CCNC(=O)C(C(C)(C)C)C1CCC1)CC 42805,c1(CCC(=O)NCC(C)CN(C)C(C2CC3C=CC2O3)=O)ccc(C#N)cc1F 42806,c1(C(C(=O)O)N(C(=O)C(=O)NC(C)(C)C)CCCC(F)(F)F)ccccc1 42807,c1(C(C)OC2CC(C)(O)C2)cn(CC2CCOCC2)nn1 42808,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 42809,N1(C(CCCCC#C)=O)C(C(=O)NCC2CCN2C(C)=O)CC2CCCC12 42810,CCCCC(CNC(=O)C(C)NC(=O)NC)NC(c1cocc1C)=O 42811,CCCC(C(C(=O)N(CC(F)Br)C)NC(=O)C(C)C(O)C(C)C)OC 42812,c1(C(N2C(CNC(CCP(C)C)=O)CC2)=O)ccc(N)c(Cl)c1O 42813,CC(N=c1[nH]c(=NC2CCOC2)[nH]c2cc(F)cc(F)c12)C1(c2ncccn2)CC1 42814,c1(C2OCCN(C(c3nc(C(F)(F)F)no3)C)C2)ccc(Cl)cc1Cl 42815,Cc1nc(SC(F)F)nc(O)c1CC(N1CCCC(n2cccn2)C1)=O 42816,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(=O)CC2SC(=N)NC2=O)C1 42817,Cc1cc(N)c(C(=O)NCC2CC(NC(C3CCCC3)=O)C2(C)C)cc1F 42818,C1(NC(c2ccc(CSC)cc2)=O)CCC(C)(C)CC1.CC1C(=O)N1C1CC1 42819,CC(C)CC(C(=O)NC(C)CNC(c1ccncc1Cl)=O)N1CCCCC1=O 42820,c1(C(=O)NC2CC(OCC(=O)NC3C(C)CN(C)C3)C2)cccc(F)c1O 42821,c1(C(CNC(=O)NC2CC(OCC)C2)N(c2ncn(C)n2)C)ccc(F)cc1 42822,C1(N(C(=O)CCn2cccc2)CC#C)CCCN(C(C2CN(C)C2)=O)CC1 42823,c1(C(C)=O)cccc(F)c1C(N1CC(O)(C(C)(C)CNC(C2(O)CC2)=O)C1)=O 42824,Cc1ccc(C(N2CCN(C3CCC(NC(c4cc[nH]c4)=O)C3)CC2)=O)cn1 42825,CC(C)C(CC(=O)N1CCN(C(C2(CF)CCCOC2)=O)CC1)c1ccc(N)cc1 42826,C(=O)(C1=NN(C)C(=O)CC1)NCC1C(CC(NOC)=O)C1 42827,CCC(CNC(=O)Cc1ccc(C(C)C)cc1)(CC)NC(=O)C=Cc1scnc1C 42828,c1(C(=O)NC2C(CNC(c3cc(OC)ncc3)=O)CC2)noc2c1COCC2 42829,N1(C(c2cc(CC)ncc2)=O)CCC(C)N(C(=O)CCCC2CCCCC2)CC1 42830,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2(NC(c3c(F)cccc3Br)=O)CC2C1 42831,C12CCC3(CN(C3)C1=O)O2.Cc1cc(C(=O)NCCNC(c2cccnc2)=O)c[nH]1 42832,C1(C(=O)NC2CC(F)(F)CC2NC(C2SC3C=CC2CC3)=O)CN2CCC1CC2 42833,N1(C(c2c(C)cccc2Br)=O)CC2(CCN(C(C3CC3(C)C(C)C)=O)C2)C1 42834,c1(CC(C(=O)NCC2CNC(=O)O2)NC(C=C(C)C2CC2)=O)cnn(C)c1O 42835,c1(C(N2CCC(NC(c3cncc(C#C)c3)=O)C2C)=O)cnn2c1CC(F)(F)C2 42836,Cc1cccc(CN(C)CC2CCN(C(c3ccc(C(F)F)o3)=O)CC2)c1 42837,N1(C(C(C)(C)OC)=O)CCN(C2CCCN(C(c3cnsn3)=O)C2)C(=O)C1 42838,N1(C(CCCCCOCC)=O)CCC(CNC(=O)C(O)C2CC2)C(F)(F)CC1 42839,CC1=CCC(C(=O)NCCCOCCCNC(=O)CC(C)OC(C)=O)CC1 42840,CCCC(O)C(CO)NC(=O)C(C(C)C)NC(C1CCC2(CC2)C1)=O 42841,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 42842,C1(C(=O)NC(c2cccs2)C)(CNC(C2CCCCC2)=O)CC(C)(C)C1 42843,N1(C(COC)=O)CCC(CNC(C2CC3CCCC23)=O)C(F)(F)CC1 42844,C(=O)(CC(O)CCCC)N1CC(CNC(CC=C)=O)C(c2cnn(C)c2)C1 42845,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 42846,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 42847,CC1CN(C(=O)Nc2cc(C3CC3)c(Cl)cn2)CCN1C1CCC1 42848,C(CC(C)CC)(C(=O)N1C2CSCC1C2)NC(CC=C=C)=O 42849,n1(CC(N2CCC(CNC(C(C(C)C)OC)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 42850,N(C1CC2(CN(C(C3CC34CC4)=O)C2)n2ccnc21)C(c1[nH]n(C)c(=O)n1)=O 42851,N1(C(c2ncn(-c3c(N)nc(Br)cc3)n2)=O)CCC2(C1)CN(CC(F)(F)F)C2 42852,CC(C)N=C(NCC1(CNc2ccccn2)CC1)N1CCC(C2CC2)C1 42853,N1(C(C2(CCOC)CCCC2)=O)CCC(C)(C)C(NC(=O)NC)C1 42854,c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(C1(C)CCOC1)=O)C2 42855,C1(NC(C2(CC#C)CCC2)=O)CN(C(C2COC2)=O)C2(CCOC2)C1 42856,C1(C(=O)NCc2c(C(=O)NC(C)CCCCO)cccc2)CC2(CCC2)CO1 42857,CCC(C)(C)CCCC(=O)N(CCN(c1nc(C)ncc1Br)C)C(C)C 42858,CC(C)(CC(=O)NC(C1CCCC1)CNC(=O)CCCC(F)(F)CO)CC(F)(F)F 42859,c1(C(=O)NCC(CO)NC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 42860,C(=O)(C1=CCN(C(=O)C(CO)NC(N)=O)CC1)NC1C(C)(C)OC(=O)C1 42861,c1(C(N2CC(C)OC(C3CCNCC3)C2)=O)cc(Br)cc(F)c1N 42862,N1(C(=O)NC2N(Cc3c(C#N)cccc3)CCC2)CCc2ccccc2CC1 42863,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 42864,C1(CC)(NC(C2CCSCC2)=O)CCCN(C(=O)CCN(CCC(C)(C)C)C)C1 42865,c1(C(C(=O)N(CC(C)C)Cc2c(C)nc[nH]2)=O)cnn2ccccc12 42866,C1(C(=O)NC(CCNC(c2[nH]cc(C)c2)=O)C)COCCN1CC(F)(F)F 42867,N1(C(c2cc(C)c(O)cc2)=O)CCC(F)(F)C(NC(c2ccc(Cl)nc2F)=O)C1 42868,N1(C(c2c(C)cnn2C)=O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C(C)C1 42869,C(CCC(C(=O)NCC(CO)C(C)(C)C)NC(C1CN(C(N)=O)C1)=O)OC 42870,N1(C(C2C(CC)OCCC2)=O)CCC(C)(NC(=O)Cn2cc(CO)nn2)CC1 42871,C1(NC(C2CN(C(C)=O)C2)=O)CCC2(CC1)CC2NC(c1cncc(N)c1C)=O 42872,CC1CCN(C(=O)Cn2ncnn2)CC1NC(c1cnc(N)c(Br)c1)=O 42873,N1(C(C2C(NC(c3[nH]cc(C#N)c3)=O)COC2)=O)CCC(CO)C12CCC2 42874,C(=O)(C(CCNC(c1nnsc1N)=O)OC)N1CCC(CSC)C1 42875,c1(C(=O)NC(c2ccccc2)CNC(C2CC(=C)C2)=O)ccn(O)c(=O)c1 42876,CC1CN(C(=O)CC2CC3CCC2CC3)CCC1CNC(C1(O)CCCCCC1)=O 42877,c1(C(=O)NCC(C)(O)CNC(c2ccc(C(F)F)s2)=O)ccn2c1CCCC2 42878,c1(C(N2CC3(CN(C(C4(CC)COC4)=O)C3)C2)=O)cnc2sc(C)cn2c1=O 42879,c1(C(C(=O)NC2CN(C(c3cnc(Cl)nc3)=O)CC2F)=O)cc(F)c(F)cc1F 42880,C1(NC(c2ccnc(Br)c2F)c2n(CCC3(C)CC3)nnn2)CC2OC(=O)CC12 42881,C1(N(C)C(C2(CO)CCC2)=O)CCC(NC(=O)Cc2c[nH]nc2O)C1 42882,c1(C(N2CCC(C)(F)C2)C(=O)NC(CC)(C)C)c2ccccc2nn1C 42883,C1(C(=O)NC2CN(C(C(C(C)(C)C)N(C)C)=O)CC2F)Cc2ccncc2N1 42884,c1(CC)cc(F)ccc1C(=O)NCC(C)(C)CNC(c1ccc(N(C)C)nc1)=O 42885,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 42886,N1(C(c2c(C)ncc(C)c2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 42887,N12CCCN(CC1)C(C)C2=O.CCC(CC(=O)N(C)CCC1CCCO1)C1CCC1 42888,C1(N(C(=O)NC(c2nnc(C)s2)C)Cc2cccc(Cl)c2)CN(C)CCO1 42889,N1(C(=O)Cc2cncs2)CC(CNC(c2cc(-c3ccccc3)on2)=O)C2CC12 42890,N1(C(C2(C(=O)NCc3[nH]nc(OC)c3Cl)CCC2)=O)CCCCC(CC2CC2)C1 42891,c1(C(=O)NC2(CNC(C3C(C(N)=O)C3)=O)CC2)nnn2c1CSCC2 42892,C(CCCCC(=O)NC(C)CCC(=O)NCCCc1ccncc1)=CC 42893,C(C)(CCCN=c1nc(NC2COCC2N(C)C)c2ncccc2[nH]1)OC 42894,C=CC(C)C(C)C(=O)NCC1CN(C(C2(N(C)C)CCCC2)=O)C1 42895,c1(CN(c2ccc(C#N)c(NC3(C)CC(N)C3)c2)C)cc(Br)cc2c1cnn2C 42896,CC1CN(C(c2cnn(C)c2Br)=O)CC1NC(c1ccnn1CC#N)=O 42897,c1(C(=O)NC23CC(NC(=O)Cc4cnc[nH]4)C(OC2)C3)nnc2n1CCCCC2 42898,C#Cc1ccc(C(N2CC(NC(=O)C(C)SC)C(c3nccn3C)C2)=O)c(F)c1 42899,c1(C(=O)NCCN(C(=O)C(C)NC(=O)CC)CCC)cn2cccc(F)c2n1 42900,C(N=c1[nH]c(N2CCC(C)(C)C2)nc2cc[nH]c12)c1n(CCCC)ncc1 42901,c1(OCC)cnc(N2CCC(CCNC(c3csc(C)c3OC)=O)CC2)nc1 42902,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C)c2cc[nH]n2)CCC1C 42903,C(c1c(Br)ccc(Cl)c1Cl)=CCNC(=O)NC1CC(C)OC1 42904,c1(C(=O)NCC(CN(C)C(c2ccc(N)c(F)c2F)=O)O)nn(C)c2c1CCC2 42905,Cc1oc(C(C)C)nc1C(=O)NCC(C)NC(=O)CC1CC(CF)C1 42906,CC(C)C(C)COCCC(=O)N1CC(CCNC(=O)C=CCO)C1 42907,c1(N2CC(C)S(=O)CC2)ccc(S(=O)(=O)NC(c2cn(C)nn2)C)cc1Cl 42908,CC(C)CC(F)(F)C(=O)NC12CC(CNC(C3C(C)(C)C3(C)C)=O)(C1)C2 42909,N1(C(C2C(CC)OCC2)=O)CCC(CN(C(C2(C3CC3)CC2)=O)CC)CC1 42910,c1(CC)cccnc1C(=O)NCCC1(O)CCN(C(=O)C(C)OCCC(C)C)C1 42911,c1(C(N2CCN(C(c3c(C)ccnc3O)=O)CC2C)=O)cccc(C#N)c1Br 42912,O=C1CCCCC(c2nnc(Cn3cc(C(F)C(F)(F)F)nn3)o2)N1 42913,c1(CCC(=O)OC)nnc(O)nc1O.C12CCCN1C(c1ccccc1)C2 42914,c1(OC)cc(C(=O)NCCSCC(N2CCC2C)=O)sn1 42915,C(CNC(=O)C(C)CN(C)C)(CC(F)(F)F)NC(C=Cc1nnc(C(C)C)o1)=O 42916,c1(CNC23CC(C(=O)NC4CCCN(C(C)C)C4)(C2)C3)c(F)cc(Br)cc1F 42917,CCC(C)C(C(=O)NC1CCOC1C(N)=O)N(C(=O)Cn1cc(C(C)=O)nn1)C 42918,c1(C(=O)NC2(COC)CCN(C(C3=C(C)CCC3)=O)C2)c(C)nn2c1CCCC2 42919,c1(NC(C(CC2CCN(C(=O)C(C)(Cl)Cl)C2)NC(C)=O)=O)cncc(Cl)c1 42920,CCCN(OC)C(=O)C(F)C1CCN(C(c2cc(C(C)=O)c(C)o2)=O)C1 42921,C1(OC)CNCC1NC(=O)CC1(c2cccs2)CC1.c12ccc(cc1)[nH]c2=O 42922,N1(C(CSc2c(OC)cccc2)=O)CCc2cc(C(=O)OC(C)C)ccc2C1 42923,C1(Nc2nccc(CC#N)n2)CCCCCN(C(c2cc(CCCO)on2)=O)C1 42924,c1(C(=O)NCC(CNC(C=CC(=O)NC2CC2)=O)F)ncoc1C1CCCO1 42925,C1(C(=O)NC(c2cn[nH]c2)C)CCC(n2cc(C3CCCO3)nn2)C1 42926,CCCC(C)CC(=O)NCCOCCCNC(=O)CC=C(Cl)Cl 42927,CC1CC(NC(=O)C=CCC(=O)C=Cc2ccoc2)c2nccn21 42928,N1(C(C(CC2CC2)NC(CC2COCC(C)O2)=O)=O)CCC2CCCC2CC1 42929,CC(C)C(C(C)NC(C12CCN(CC1)C2)=O)NC(c1cc(C(F)(F)F)n[nH]1)=O 42930,C12(C(=O)NC(CC=C)CNC(=O)CC3CC(n4cnnc4)C3)CC(C)(CCO1)C2 42931,C(=O)(C(F)C(C)C(F)(F)F)NC1C(SC)CN(C(=O)C=Cc2cn(C)nn2)C1 42932,Cc1cncc(C(=O)NCCN(CC(C)O)C(c2cn(C3CCOC3)cn2)=O)c1 42933,c1(C(N2C(CC)C(NC(C3(C)CC3(C)C)=O)CC2)=O)n[nH]c2c(OC)cccc12 42934,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 42935,C1(CNC(C2CC3(C2)CS(=O)(=O)C3)=O)CCCC2(CN(C(=O)C3=NOCC3)C2)O1 42936,Cc1ncc(C(=O)NCCCCC(C)NC(=O)CC2COCCO2)c(C2CC2)n1 42937,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 42938,C(C(C)(C)CN(C(=O)CC1CC1C(F)(F)F)C1CC1=O)NC(C1C(OCC)C1)=O.COC 42939,C1(C(=O)NCC#Cc2cccs2)(CC)CCN(C(=O)CCCC2CCOCC2)CC1 42940,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)Cc2cccc(F)c2)C2CCCC12 42941,C1(c2n(CCSC)nnn2)(NCC2CC2(C)C)CCOCCC1C 42942,N=c1[nH]c(=NCc2ncc(Br)cc2F)[nH]c(=NCc2ccc(F)c(F)c2)[nH]1 42943,c1(C(N(C(CNC(=O)C(Cl)=CCl)C2CC2)C)=O)cc(N)c(Cl)cn1 42944,C1(C(=O)NC2CCN(CC)CC2)CCCN(C(=O)CC2CCCO2)C1C 42945,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 42946,C1(C(=O)NCCCCCNC(c2cn(CCC(C)C)nn2)=O)CN2CCC1CC2 42947,c1(C(C)=O)cc(NC(C2CCN2Cc2sccc2Br)=O)ccc1O 42948,C12CCCCN1N1CCC(C1)n1nc(C3CSC3)nc12.c1(C(C)C)ccccc1 42949,N1(C(C(CN(C(C=C(C)C(F)F)=O)C)C)=O)CCC12CC(CO)C2 42950,c1(C(=O)Nc2cnc(C#N)nc2Cl)ccc2cccc(-c3cnoc3)c2n1 42951,C1(C(=O)NC(CC(C)C)=O)(N(C(CCC)=O)C(C)CO)CCN(C)C1 42952,Nc1ccc(-n2cccn2)cc1C(=O)NCCC1(CNC(=O)C(F)(F)F)CCC1 42953,c1(C(N2CCC(C(=O)NCC(C)CN3CCCC3)CC2C)=O)cccn2nccc12 42954,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(C(C)C)C)=O 42955,C1(C(=O)NCc2cc[nH]n2)COCCC12CN(C(c1cc(C(F)(F)F)on1)=O)C2 42956,N1(C(CCOCC)=O)CCC(C(CO)NC(C23CCC2C3)=O)CC1 42957,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCCC1)OC 42958,C1(C(=O)NC(C)(CNC(=O)CN(C)C(N)=O)C2CC2)(OCC)CCOC1 42959,N1(C(CC(C)c2ccccc2)=O)CCN(C(C2(CNC(N)=O)CC2)=O)C2CCC12 42960,c1(NC(c2n(CC)nnn2)c2ccsc2)cc2n(c1)CCCC2 42961,c1(CN2C3(c4onc(C)n4)CCC3CC2)nc2ccc(C)cc2s1 42962,C1(C(=O)NCC(CNC(=O)Cc2ccccc2F)OC)NC(=O)OC1C 42963,N1(C(C2C(O)CCN(C(=O)Cc3ccc(F)cc3F)C2)=O)CCC2(CC1)COC2 42964,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 42965,c1(NCC(=O)CNCC2N(C(C3C(OC)C3C)=O)CC=C2)ccc(F)c(F)c1 42966,Cc1cc(C)c(C(=O)N(CCCNC(=O)C=C2CCSCC2)C)c(=O)o1 42967,c1(CN(C(C2N(CC)CC2)=O)C)cnn2c1CN(C(=O)COC1CCOC1)CC2 42968,c1(CC(C(=O)N2C(CNC(=O)Cc3ccnn3C3CC3)CC2)O)cccc(Cl)c1 42969,N1(C(C=COCC)=O)CC12CCN(C(=O)C(c1ccc(OC)cc1)(C)C)CC2 42970,c1(C(N2CC(NC(=O)Cc3cc[nH]n3)C(F)C2)=O)cccc([N+](=O)[O-])c1Cl 42971,N1(C(c2cc(Cl)ccn2)=O)CCc2cnccc21.C1(CCN(C)C)COCCN1 42972,c1(C(N2CC(F)CC(C(=O)NCc3ccsc3Br)C2)=O)c(F)ccc(Cl)c1Cl 42973,C(CS(=O)(=O)CC(=O)NC1CCC(CNC(c2csc(Cl)n2)=O)C1)OC 42974,c1(N(C)CCC2CCCN(C(C3CCS(=O)(=O)CC3)=O)C2)ccc2ocnc2c1 42975,N1(C(c2c(C)csn2)=O)Cc2[nH]nc(C(=O)NOCC(C)(C)C)c2C1 42976,N1(C(COC(CC)CC)=O)CCCCC1CC(=O)NCCCS(C)=O 42977,Cc1c(C(C)(C)NC(c2ccc(C#N)cn2)=O)cc(F)cc1[N+](=O)[O-] 42978,N1(C(CCCCC=C)=O)CCC2(CCN(C(=O)CC(CC)CC)C2)C1 42979,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(c2cnn(CC(F)F)n2)=O)CC1 42980,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(N)c(C)c1 42981,c1(C(=O)NCC2CN(C(=O)C(C3CC3)C3CC3)CC23CC3)ccc2ocnc2n1 42982,c1(OC)cnn(C2CCN(C(=O)COC(C)(C)C)CC2)c1C 42983,C1(N(C(C(C2CN(C(Cc3ccc(C)o3)=O)C2)O)=O)C2CC2)CNC(=O)C12CC2 42984,c1(NC(CC(C)N(C(C(CCOC)C)=O)C)=O)ccc2nccn2c1 42985,C1(CC)CN(C(=O)C(c2cccnc2)O)CCN1C(C1OCC1(C)C)=O 42986,C1(N(C2CC3CNC2C3)C(c2cccnc2)=O)CCOC2(CCCCC2)C1 42987,C(CCC(C(=O)NCC(C)(O)C1CCC1)NC(=O)CS(C)(=O)=O)OC 42988,C=CCC(C)(CC=C)NC(C1C(C)CCN1C(=O)CCC1OCCO1)=O 42989,c1(C(N2C(CN(C(=O)CC#N)C)CCC2)=O)cnn2c1CCC2 42990,N1(C(C(N2CC3CC3C2)C)=O)CCCC2CN(c3ncc(C)c(O)n3)CC12 42991,C1(OC)CN(C(=O)C(O)CNC(=O)C(C)(C)CC#N)CC1(C)C 42992,C#CCC(CC(=O)NC(CC)C1CCC1)NC(=O)CCCNC(N)=O 42993,c1(OC)cncc(C=CC(=O)NCCCCNC(c2c(C3CC3)cnn2C)=O)c1 42994,C(C(C)C(C)C(=O)NCc1ccnc(NCCN(C2CC2)CC2CCC2)c1)OC 42995,c1(C(=O)NCC(C)CNC(c2ccc(C#N)s2)=O)n[nH]c2ccccc12 42996,N1(C(C)=O)CCCC1(C)n1cc(-c2cc(C(N3CC(CO)C(O)C3)=O)sc2)nn1 42997,C(=O)(NN1CCCC1C(=O)NC1CN(C)CC1OC)c1cc(CC)nn1C 42998,Cc1sc(Cl)nc1C(N1CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1)=O 42999,C1(CC(=O)NCC(=O)OCC#C)N(C(=O)C(C)SCC)CCC1(C)C 43000,Cc1ncnc(C)c1C(=O)NCC1CC(F)CN1C(C1CC1(C)C(F)F)=O 43001,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)CC(=O)Nn2cncn2)C2(CCC2)C1 43002,N1(C(C2C(C)C2)=O)CCC(O)(CNC(c2csc(Cl)n2)=O)CC1 43003,c1(C(=O)NC(C2(O)CN(C(C3(O)COC3)=O)C2)C)ccc(F)cn1 43004,c1(C(C(=O)NCC(=C)C)N(C)C)ccc(OC(F)(F)F)cc1 43005,C(=O)(CC(C)(C1CC1)NC(=O)Cc1ccsc1Cl)OC 43006,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)c(F)ccc(F)c1F 43007,c1(C2C(NC(=O)Nc3cncc(NCC)c3)C2)cc(Cl)ccc1Cl 43008,c1(C(=O)NC(CN(C(C2(CC)COC2)=O)C)C)cc(C(C)=O)cs1 43009,C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CCc2cnn[nH]2)CCN1C 43010,c1(C(=O)NC2CCN(C(C3COCO3)=O)CC2O)cnc2c(c1)C(=O)CCC2 43011,C1(O)(CCNC(CC(=O)NCCOC)=O)CCN(C(=O)CCS(C)=O)C1 43012,N1(C(C(C(C)C)SCC)=O)CCN(C(=O)Cc2c(C)cnn2C)CC(C)(C)C1 43013,C(=O)(CCC(C)(F)F)NCC(C)C(=O)NCCN1CC(C)(O)C1 43014,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)sc3CC)=O)C2)C1 43015,c1(N2C3C(C(N4CCNCC4)=O)(CCC3)C2)ncnc2[nH]ccc12 43016,N1(CCn2ncc(C)c2)CCCCC1c1cn(CCn2cc(C(N)=O)nn2)nn1 43017,C(CC)(CCCC(=O)Nc1cc(C#N)cs1)NC(=O)Nc1n(CC)ccc1 43018,C(CCC(N)=O)(C(=O)NCCCCCNC(C1(CF)CC1)=O)N(C)C 43019,CCCCC(CC)C(=O)NC(C)CCCNC(=O)Cc1ccc(OC)cc1 43020,C1(C)(CNC(C=CCN(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)=O)CCCCC1O 43021,C=CCC(F)(F)CNC(c1c[nH]nc1CCNC(=O)CCCCC)=O 43022,C(=O)(C1CCCn2ncnc21)NCCC1CC(NC(C2=C(C)OCCS2)=O)C1 43023,c1(C(=O)NS(c2cc(C(=O)OC)nn2C)(=O)=O)cnc2ccc(C)cn12 43024,c1(CC(=O)Nc2c(C(C)(C)C)c(-c3ccccc3)cs2)csc2ccc(Cl)cc12 43025,Cc1nc(N2CC3C(NC(c4coc(Cn5cccn5)c4)=O)C3C2)[nH]c(=N)n1 43026,c1(NC(C2N(C(C(CC)OCC)=O)CCC2)=O)cccc(Cn2cncn2)c1 43027,C(=O)(C(C)(C)C1CCCN1C(c1ncsc1C)=O)NCCN(CCCC)C 43028,c1(C(N2CCC(C)C(NC(C3(C)CC(C#N)C3)=O)C2)=O)ccc(Cl)c2occc12 43029,C(=O)(C1=C(C#N)CCC1)NCCC1OCCN(C(C=COCC)=O)C1 43030,c1(C(N(C(CNC(CCN(C(C)C)C)=O)C)C)=O)ccc(F)cc1 43031,C1(C(C(=O)N(CCC)CCC)C)CCN(C(=O)Cc2cc(O)n(CC)n2)CC1 43032,c1(OCC)cccc(NC(=O)Cc2ccc(OCC3CC3)nc2F)c1C(=O)OC 43033,N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)CCC2OCCO2)CC)C1 43034,C(=O)(C(C)C(C)C(C)(C)C)NCC1(F)CC(NC(c2c(C)cc(CC)o2)=O)C1 43035,N1(C(CCC(N)=O)=O)CC2(CC(NC(=O)C=Cc3cnc[nH]3)CO2)C1 43036,N1(C(c2c(CC)oc(C)c2)=O)CC(C(N2CCC3C(OC)CC23)=O)C(F)(F)C1 43037,C(C(C)(C)C(=O)NCC1CCC(NC(=O)C#CC2CC2)C1)OC 43038,c1(NC(N2CCN(C3COCC3O)CC2)=O)ccc(C2CCC(=O)N2)cc1 43039,C1(C(=O)NCCC(C2CC2)OC)CCC(C)CN1C(=O)COCC1CC1 43040,C(=O)(C1CCCCc2ccccc21)NCC(=C)CCNC(=O)CC(O)CCSC 43041,c1(OC)ccc(N2CCC(OCC(C)C(=O)Oc3ccccc3)C2)cc1 43042,C=Cc1ccc(C(N2CCC(c3cn(CC4CCCO4)nn3)C2C(=O)O)=O)cc1 43043,c1(C(N2CC(CCNC(c3ccnn3C3CC3)=O)(OC)C2)=O)cc(C#N)oc1C 43044,C1(C(N(C(C)CN(C(=O)CNC(c2cccs2)=O)C)C)=O)CCCC1S(C)(=O)=O 43045,C1(C(=O)OCC)CC(F)(F)CN1C(c1ccnc(OC2CCOC2)c1)=O.C1(C)CN1 43046,N1(C(CCOC2CN(C(CC3CCC(C)CC3)=O)C2)=O)CCCNC(=O)C1C 43047,C1(C(N2CC3CC3(C(=O)NCCOc3ccccc3F)C2)=O)CCn2cnnc2C1 43048,C=CCC(C(=O)N1CCC(O)(CNC(C2(C3CCCCO3)CC2)=O)CC1)C(C)C 43049,c1(COCC(=O)NCC2CCCN(C(c3cccc(F)c3)=O)C2)ccnc(O)c1 43050,N1(C(c2n[nH]c(C)c2N)=O)CC(C2CCCN(C(=O)C(C)CS(C)=O)C2)C1 43051,C1(C)(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(c2cncnc2)=O)CCO1 43052,Cc1nc(C(=O)NC2CCN(C(c3c[nH]cc3Br)=O)C2C)cn(C)c1=O 43053,c1(C(N2CCCC(CC)(N(C(=O)CC3CC3)C3CCC3)C2)=O)ccc2nncn2c1 43054,C1(F)(C(=O)NCC(C(=O)NC(C)CCC2CCCC2)N(C)C)CCCCC1 43055,C12(CNC(C(CC)c3ccccc3)=O)CC(NC(c3cc(C)[nH]n3)=O)(CCO1)C2 43056,c1(C(C)C)ccc(C(=O)N(C2CCC(NC(C3(Br)CC3)=O)C2)C)nc1 43057,C1(CNC(C(C)(C)c2ccno2)=O)CN(C(C2CCCC2O)=O)C2CCCC2O1 43058,c1(C(c2ccccc2)C(N2CC(NC(CC3(N(C)C)CC3)=O)C2)=O)cncn1C 43059,c1(C(N2C(C(=O)NC(C(=O)NC)(C)C)CSC2)=O)cc(F)cnc1O 43060,c1(N(C)Cc2cc(Br)cs2)nc(N2CCOC(c3cn[nH]c3)C2)nc2cccnc12 43061,C1(NC(c2c(C)cc(C)s2)=O)CN(C(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 43062,c1(N(c2ccccc2)CC2CCN(CC)C2)nc(C)cc(O)n1 43063,C1(CNC(=O)CC2CS(=O)(=O)C2)C2CN(C(c3cnccc3Cl)=O)CC12 43064,c1(C(N(CCCNC(C2(CCC)CC2)=O)CC)=O)cc(CSC)cc([N+](=O)[O-])c1 43065,c1(C(=O)NCCC(C)NC(C2COCCO2)=O)cc2cc(F)cc(F)c2[nH]1 43066,c1(C(=O)NC2CCC(NC(C3C(CCC)C3)=O)C2)ccc2c(c1)NC(=O)CS2 43067,n1(CC(N2C(CCCNC(CC=CC)=O)CCC2)=O)nc(C)cc1C(F)F 43068,C1(CNC(C(CC)(F)F)=O)CC2CCC1N(C(=O)C(CO)CNC(N)=O)C2 43069,CC(C)(CNC(=O)CC(O)CNC(=O)CS(C)(=O)=O)C(N)=O 43070,C(=O)(C1=C(C)CCCC1)NC1C(SC)CN(C(=O)C(=Cc2ccc(F)cc2)C)C1 43071,N1(C(C(CCCC)C)=O)CC2(CCC(CNC(=O)C(C)C3CCCO3)O2)C1 43072,c1(OC)c(C(=O)NC(C)CNC(C2CNC(=O)C(C)(C)C2)=O)oc2ccccc12 43073,c1(CC)cc(C(=O)NC(Cc2cn(C)nn2)C(=O)NC(C)COC)n[nH]1 43074,c1(C(N(CC(C)NC(=O)C2=C(Cl)CC2)C)=O)ccc(CSc2nncn2C)cc1 43075,n1(CC)nc(C(=O)NC(C)(CSC)C(=O)NCC(O)COC(C)=O)c(C)n1 43076,c1(OC)ccccc1C(=O)NC1CCCN(CCC2CCCCO2)C1 43077,c1(OCC)ccc(F)c(CNC(C23CC2CN(C(c2ccc(Cl)s2)=O)C3)=O)c1 43078,N1(C(C(C)Sc2nncn2C)=O)CCN(C(c2nncs2)=O)CC1CCO 43079,N(C(=NCCCF)NCC(c1ccc(OCF)cc1)O)C(c1ccncc1)C 43080,CCC(O)(C(=O)NC(C1CN(C(C2CNC(=O)N2)=O)C1)C)c1ccccc1 43081,C1(C(=O)NCC2CC(NC(c3c(Cl)nc(OC)s3)=O)C2)CCCC2(CCC2)C1 43082,C1(CCOCCC(C)C)CCC(NC(=O)CNC(=O)CCN2CCC2)C1 43083,CC(C)(CO)C(=O)NCCC1CCN(C(=O)CCN2CCCC(C(N)=O)C2)CC1 43084,c1(NC(c2ccc(N(C)C)nc2)=O)c(C(=O)NCC2(CC)CCC2)cccc1Br 43085,C1(CS(=O)(=O)NCCOC)(OC)CCOCC1.c12ccc(cn1)CN2 43086,N1(C(c2ccn(CC)c2C)=O)CCCC2CN(C(C34CC(C)(C3)C4)=O)CC12 43087,c1(NCC(=C)Cl)cccc2c(C(=O)OC)ncc(Br)c12 43088,Cc1cccnc1NC(C1CCN1C(=O)CC1CC1)C1(c2ccon2)CC1 43089,C1(CCC=O)CCCN(C(=O)C2CC2)CC1.CC1CC(CSC)N1 43090,N1(CCC)CC(CNC(=O)NCC(C2(O)CCCCC2)C2CC2)CC1=O 43091,Cc1cc(C(F)(F)F)nn1CC(N1CC2CC2(CNC(C2C3COCC23)=O)C1)=O 43092,C1(C(N2CCC(NC(=O)Cn3cnnn3)C2C)=O)(OC)CCCOC1 43093,c1(C(N2C3CCC(NC(c4cc5n(n4)CCC5)=O)(C3)C2)=O)nnn2c1CCCC2 43094,Cc1cc(NC(=O)C(c2ccnn2C)NC(C2CC=CCC2)=O)cnc1C#N 43095,Cc1c(C(=O)NCC2CCCN2C(=O)CC2COCCN2C)cccc1Cl 43096,Cc1cccc(OCC(=O)NC(C)(CNC(C2OCCN(C)C2=O)=O)CO)c1F 43097,Cc1c(NCC2CC23CCC3)ncnc1N1CCOC(C(C)(C)C)CC1 43098,c1(N)cnc2sccn12.N1(c2cc(N(CC)CC)ncn2)CCOCC(CO)C1 43099,N1(C(C(=O)N(C)CCn2ccc([N+](=O)[O-])n2)=O)CCCC2(CNC2)C1 43100,c1(OC(CC)C)ccccc1C(=O)NC1CCN(C(=O)C(C)c2cccs2)CC1 43101,CC(N=c1[nH]nc(-c2ccccc2)s1)c1ccc(NCC(N)=O)cc1 43102,C1(C(=O)NCCOC2CN(C(C3(C#C)CCCC3)=O)C2)CN2CCCC2CO1 43103,CC(N=c1[nH]c(=NCCF)[nH]c2c1COC2)c1snnc1C1CC1 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43172,N1(C(Cc2n(C)ccn2)=O)CC2ON=C(CNC(C3CC(S(C)(=O)=O)C3)=O)C2C1 43173,N(C(=NCC)NCC(CC)OC)CC1CCC(CCCC)O1 43174,Cn1ncc2c(C(=O)NC3CCC34CN(C(=O)CC3CC=CCC3)C4)ccnc12 43175,CC1(C)CC(C(N2CCCCC2CNC(=O)CC2COC(=O)C2)=O)CO1 43176,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43177,N1(C(c2n(CCC)ccc2)=O)CCOCCC1C(N1CC(CC2CC2)C1)=O 43178,C1(NC(=NCC)NCCC2CCCN(CC)C2)CCn2nnnc2C1 43179,C12(NC(CCCSC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 43180,Cc1cccc(NCCC(N2CC(CNC(c3cccnc3S)=O)C(C)C2)=O)c1 43181,C(C(N=c1ccnc(NCCN2CCS(=O)(=O)CC2)[nH]1)c1ccccc1)OCC 43182,C1(C)(C(=O)NCC2C(C)CN(C(c3ccc(F)cn3)=O)CC2)CCC(C)(C)CC1 43183,CCC(C)CC(C)C(=O)N1CCC(=CCNC(c2cc(=O)c(OC)co2)=O)CC1 43184,N1(C(C(C)=C(C)C)=O)CCCC1COC(=O)NC(C1CCC1)=O 43185,N1CCCC(C2CCN(CC(=O)OC)C2)C1.c1(OC)ncccc1NCCCCCC 43186,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43187,C1(C(=O)Nc2[nH]c(CC)c(Cl)n2)CCN(Cc2ccc(N(C)C)cc2)CC1C 43188,Cc1ccccc1NC(=O)CN1CCCC1CCCNC(=O)CNC(N)=O 43189,N1(CC)CCN(C)C(CO)C1.c1(SC)nn(C)cc1C(=O)NCC1CC1C(=O)N 43190,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2CCCNC2=O)CC1C 43191,N1(C(C)C(=O)NCC23CC(C2)C3)CCC(NC(=O)OC(C)(C)C)C(F)(F)CC1 43192,c1(C(N2C(CNC(C3C(C)C3)=O)CC(F)C2)=O)ccc(N=NC(N)=O)cc1 43193,C(=O)(CCC(=O)C1CC1)NCC(C)(C)CNC(=O)C(C)(C)c1cscc1Cl 43194,CC1(CO)CCCN1C(=O)Cn1cc(I)nn1 43195,c1(C(N2CC(COC)N(C(C3CC(OC)C3)=O)CC2)=O)cc(F)c(C)cc1F 43196,C(C(CC(C)C)C(=O)N(C)Cc1ccoc1)N(CC(=O)NCCC)C.C1C(=O)N1 43197,c1(C(N2CCCCC(NC(c3n[nH]c(C)c3O)=O)C2)=O)c(C)cc(O)nc1C 43198,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43199,C1(C)(CNC(c2n(C)ncc2)=O)CN(C(C2(CF)CC(F)(F)C2)=O)CCO1 43200,C1(NC(CC2C(=O)NCC2)=O)CCOC(C(N2CCOC(CCN(C)C)C2)=O)C1 43201,C1(CNC(C2C(CC)CCN2C(=O)CCOC)=O)CCCC2(CC2)C1 43202,C12(NC(c3c(C)oc(-c4cccs4)n3)=O)CC(CNC(=O)C(C)NC=O)(C1)OC2C 43203,CCCCCC(C(=O)N1CCC(C)(NC(c2onc(C)c2C)=O)CC1)C(C)C 43204,C(=O)(C(CCC(N)=O)n1ccnn1)NCc1nnc(C)o1.N1(NC)CCCC1=O 43205,c1(C(=O)NCCCC(C)NC(c2cn(C)cn2)=O)nc(Cl)sc1Cl 43206,CC1(C)CCCC(CNC(C2CCC(CNC(=O)OC(C)(C)C)O2)=O)O1 43207,CC(C(=O)N1CC(CNC(=O)CC2CC(=O)N2)C1)OCC.C(C(F)(F)F)O 43208,C12(NC(C(CC=CC)CC)=O)CCC(CN(C(c3ccc(OCC)nc3)=O)C1)C2 43209,CN1CCN(C(C2CCOC2CNC(=O)C(F)C(C)(F)F)=O)CC1CO 43210,C1(NC(C2(CC)COC2)=O)CC(NC(=O)C(C)OCC(C)C)CC1O 43211,C1(NC(C(C)NC(C)(C)C)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1 43212,Cc1nc(C)c(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)nc1C 43213,CC1CC(C(=O)N(C)C)CCN1C(C1CCCN1Cc1ccccc1)=O 43214,C=C(CNC(=O)COC1CCC1)CCNC(=O)COC(F)(F)F.C1CC(=O)N1 43215,c1(CN2CCC(CNC(Cc3c(C)n[nH]c3)=O)CC2C)cn(C)c2ccccc12 43216,C1(NC(C=C(CCC)C)=O)C(C)CCN(C(c2ncc(C(F)F)s2)=O)C1C 43217,C1(C)(C(=O)NC(C2CCOC2)(C)C)CCCN(C(c2cccc[n+]2[O-])=O)C1 43218,C(Cn1cccn1)(C(=O)NC1(C2CCCO2)CCC1)NC(=O)CCC1CC1 43219,c1(C(=O)NC2C(C)CCN(C(c3cc(Cl)cnn3)=O)C2)ccc2nc(O)oc2c1 43220,C1(NC(C(CC)SC(F)(F)F)=O)(NC(=O)CN(C)C)CCCC1C 43221,C1(C(N2CCCC(F)(C(=O)NCn3nc(C)c(Br)n3)C2)=O)CC(=O)CC12CCC2 43222,N1(C(C)=O)CC(O)CC1C(=O)NCC1(CNC(c2ccon2)=O)CC12CCC2 43223,c1(OCCOC)ncccc1C(=O)NCCC(C)(C)NC(=O)CC1CCC(C)(C)C1 43224,N1(C(C2C(C(N)=O)C2)=O)CC2CC1C2CNC(=O)C(C1CC1)SC 43225,c1(C(=O)NCCC(C)NC(C(C=C)O)=O)cc(C)cc(C)c1N 43226,C(=O)(CC(C)(C)C1CC1)NC(C1N(C(C(c2ccc(Cl)s2)OC)=O)CCC1)C 43227,C1(CNC(c2ccc(-c3nc[nH]n3)cc2)=O)CN(C(c2cnc(S)[nH]2)=O)CC1(F)F 43228,C12CCCN1C2=O.C(CC(=O)N(C)CC1(NC=O)CC1)N(C)CCO 43229,c1(C(=O)NC2C(C(N3CCC(C=C)(O)C3)=O)CC=CC2)cc2ncccc2[nH]1 43230,C1(C(C)NC(=O)Cc2csc(S)n2)CCCCN1C(c1ccncc1C(F)F)=O 43231,C(=O)(C(CO)C(F)(F)F)N(C)CC1CC(F)CN1C(c1cnn(CCF)c1)=O 43232,N#Cc1ccc(N)c(C(=O)NCC(CC2CC2)C(N2CC(O)CC2CO)=O)c1 43233,c1(N(CC=C)CCC)nc(=NCC2(C)CC2(F)F)[nH]c2c1CCCCC2 43234,C1(C(N2CCN(CC3CN(C(C(C)(C)O)=O)C3)CC2)=O)CC2(C1)CC(C#N)C2 43235,N1(COC)CCN(C(c2ccccc2I)C(=O)NCC2CCOCC2)CC1=O 43236,C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(c2ccc(C#N)s2)=O)C1 43237,O=C(N=c1ccn(C(F)F)[nH]1)C1=C(F)CN(CCF)CC1 43238,C1(C(C)C)CN(C(c2c[nH]nc2C(F)(F)F)=O)CCC1NC(=O)C1=CCCO1 43239,C1(CNC(c2ccc(F)s2)=O)CN(C(c2ccc(C3CC3)s2)=O)CC12CCC2 43240,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CCC3CCOC3)CC2)nn1 43241,C12(C(=O)NCc3cc(C)sc3)CC(C)(CN1C(=O)CC1CC3CCC1O3)C2 43242,C(C(CCC)C(=O)NC1CCCN(O)C1=O)NC(CCC#C)=O 43243,c1(C(N2C(C(N3CCC4CCCC4CC3)=O)CCC2)=O)cn2cccnc2n1 43244,C12(CN(C(C#C)C3CCC3)C)CCCCC1CNC2 43245,Cc1cccnc1C(=O)NCc1cn(CCCCCCNC2CCC(F)CC2)nn1 43246,C1(C(N(CCCN(C(=O)CCc2cccc(O)n2)C)C)=O)CCC2CCCCN12 43247,C(=O)(C(C)(C)CNc1ccccc1)NCCCC1(NC(C(COCC)F)=O)CC1 43248,N1(C(CN(C)C)=O)CCC2CN(C(c3cc(C4CCOCC4)[nH]n3)=O)CCC12 43249,N1(C(C2(C(C)C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43250,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(OCC(N1CC3(CCC3O)C1)=O)C2 43251,CCC(CCCC(=O)NCC1(CCF)CCC1)NC(c1cc(OC)n(C)n1)=O 43252,c1(CC(=O)N(C2CN(C(CC3(OC)CC3)=O)CC2O)C)nn(C)c2ccccc12 43253,C1(NC(c2ccc(O)nn2)=O)CCN(C(=O)CCC2CCC2)C2CC12 43254,N1(C(C(CC)N(C)C)=O)CCC(NC(C2C3CCC2CC3)=O)C12CCCC2 43255,N1(C(C(C)OCCC=C)=O)CCC2CN(C(c3ccc(F)c(Cl)c3F)=O)C2C1 43256,O=C1CCC(CCN(C(=O)C)C)N1.C1(OC(=O)C2CC2)CCOCC1 43257,C1(NC(c2cccc(-c3cccs3)c2F)=O)CN(Cc2ccsc2)CC1(F)F 43258,N1(C(C2(CCOCC)CCC2)=O)CC(C)(CNC(C2CCCC2)=O)CC1(C)C 43259,c1(CCNC(C2N(C(C(C3CC3)OC)=O)CCC2)=O)ccnc(C)n1 43260,C1(C)(CNC(CN(CCC#C)C)=O)CCC(NC(C2CCN(C(C)C)CC2)=O)C1 43261,C1(CNC(C2CCCOC2)=O)CC12CCN(C(=O)CC1CC3CC(=O)C1C3)CC2 43262,N1(C(c2c(C)cncc2)=O)CC(C)CN(C(c2nc[nH]c3nccc2-3)=O)C(C)C1 43263,c1(NC(C2CCN(CCC)CC2)=O)c([N+](=O)[O-])cc(CO)c(C)c1[N+](=O)[O-] 43264,n1(-c2nc(C34CC(OC(C)(C)C)(C3)C4)on2)cc(C(C)(C)C)cn1 43265,C(CCCC(C(=O)Nc1ccccc1CO)N1CCS(=O)CC(C)C1)OC 43266,C1(C(=O)OC)(NC(=O)CCc2c(N)cccc2F)CCS(=O)(=O)CC1 43267,CCCC(O)C(=O)NC1(C)CN(C(=O)C(=O)NCC2CC2)C1 43268,C(CN=c1[nH]c2ccc(Br)cc2s1)N(C(=O)CCCCC1CC1)CCO 43269,CC(C)C(CCNC(c1ncoc1C(C)C)=O)NC(=O)CC1CCCC12CC2 43270,C1(NC(CN(C)C(N)=O)=O)CN(C(c2cn3cccnc3n2)=O)CCC12CCC2 43271,C(CCC(=O)N1CCCC(N(C)C)C1)(C(C)C)NC(c1c(C)coc1)=O 43272,C12(C(N(C)CC3CN(C(=O)Cc4ccc(F)cc4)C3)=O)CCC(C1)C2(C)C 43273,C(=O)(CC(C)(C)C(=O)NCC1CC1NC(C1(O)CCCC(C)(C)C1)=O)OC 43274,Cc1ccccc1NC(=O)CN1CCC(C(=O)NCC2COC(C)(C)N2)C1 43275,N1(C(COCCC=C)=O)CC(CNC(c2cc(C(N)=O)co2)=O)OC2CCCC12 43276,C1(C)(CNC(C2C=CC(NC(C(C)=CCC)=O)C2)=O)NC(=O)NC1=O 43277,c1(C(=O)NC(CN(C(C(C(C)C)n2cncn2)=O)C)C)ccnc2c1CC(=O)N2 43278,N1(C(C(CC2CCC2)NC(C(C)OCC)=O)=O)CCCSCC1C 43279,CC(C)C(C(=O)NC(C)CC1CN(C(=O)CCc2cccnc2)C1)NC=O 43280,C1(C(=O)NCC(c2cnc[nH]2)O)(NC(=O)Cc2ccsc2)CCCCC1 43281,CC(C(=O)NC1CN(C(c2ncccc2N)=O)CCC1c1ccccc1)C(C)(C)C 43282,C(=O)(C(F)C(F)(F)F)N(CCC)CCNC(C1CCC1C(C)(C)C)=O 43283,C(=O)(C1CCc2cccnc21)N1C2CCC(NC(C34CC(CC)(C3)C4)=O)(CC2)C1 43284,N1(C(c2c(COC)ccs2)=O)CC(CNC(c2cc(OC)ncn2)=O)CC1C 43285,c1(OCC(=O)N(CC(CNC(C(C)O)=O)O)C)cccc(Cl)c1 43286,c1(NS(=O)(=O)Cc2cccc(C(=O)NCC(N)=O)c2)cc(Br)cnc1Br 43287,C1(C(=O)NCC2C(NC(c3c(C(C)C)c[nH]n3)=O)CC2)CCCN(C)C1 43288,Cn1c(C(N2CCC(C)(CNC(=O)C(O)C(C)(C)C)CC2)=O)c(Cl)c2ccccc12 43289,CCC(CC)C(=O)N1C(CNC(c2cccc(CC(C)C)c2)=O)CC2CC12 43290,c1(C(=O)NCC2CC(NC(CCC=C=C)=O)C2)cc(C)ccc1OCC 43291,Nc1ccc(F)c(C(=O)NC2(C3CCCO3)CC2)c1.C12CN(CC13CC3)C2=O 43292,C1(NC(C2=C(C)CCC2)=O)C2CC(CN(C(=O)C=CCF)C2)C1c1ccccc1 43293,C1(CC(=O)N(C2CCN(C(=O)CCCF)C2)CCC)CCN(Cc2ccccc2)C1 43294,C(=O)(C1=NNC(=O)C1)NCC(C)(C)NC(C1CN(C2CCOC2)C1)=O 43295,C1(C(=O)NCC(CNC(CCCOCC)=O)C)CCCC12OCCO2 43296,N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCCN2C=O)=O)CC1c1cccnc1 43297,c1(CNC2C(C(N(CCC(F)(F)F)CC)=O)CCC2)ccc(F)c(F)c1Br 43298,C1(C(=O)NCc2ncccc2Cl)C(C2CC2)CCN1C(=O)Cc1cccs1 43299,Cc1nc(C)c(C(N2CCC(OCCNC(=O)C(c3cccc(F)n3)F)C2)=O)[nH]1 43300,C1(NC(C(CC=CC)CC)=O)CCCCCN(C(c2ncsc2CC)=O)C1 43301,Cc1nn(CCN(CCN(C)C)Cc2cn(C3CCC(N)C3)nn2)c(=O)n1C 43302,c1(CN(C(=O)C(F)C2CC(NC(C3(C)CCC3)=O)C2)C)ncnn1C 43303,C1(OC)(CNC(=O)COC2CC2)CN(C(C2(c3ccnn3C)CC2)=O)C1 43304,c1(NC(c2n(C(C)C)cnn2)C)[nH]c(=NCCn2cc(Br)cn2)nc2scnc12 43305,Cc1c(-c2nccn2CC(N2C(Cn3ccnn3)CCC2C)=O)nc2sccn12 43306,c1cc(NCC2CCC2C2CC2)cc(-n2cnnn2)c1 43307,c1(N(C)Cc2ccn(CC)n2)cc2nc(n1)CCN2.N1(CC)CC(C)(C)C1 43308,Cc1oc(C(C)C)cc1C(N1CCOCC1CNC(=O)Cc1cnoc1)=O 43309,c1(COCC(=O)NCC(CNC(C(C)c2cncs2)=O)CO)ccnn1C 43310,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43311,c1(CN2CC3C(NC(CCc4cc(C)cc(C)c4)=O)(C3)C2)cccc(C=O)c1Br 43312,C(=O)(C(CNC(C1CCCOC1)=O)N(C)C)N(CC(=C)C)C 43313,C1(NC(c2c(CC)nc[nH]2)=O)CN(C(=O)COc2cc(C)on2)CCC1C 43314,c1(C(=O)NC2CC(CNC(c3sc(C)c(O)n3)=O)C2)ccc(=NCC2CC2)[nH]c1 43315,C12CN(C3CCN1C3)CC(=O)N2.CC1(C)COC1 43316,N1(CCC)CCN(C(C2CCCN(C(=O)NC3CCCO3)CC2)=O)CC1=O 43317,c1(C(=O)NC2CC(C)N(c3ncc(Cl)cn3)C2)cc(O)nc(O)n1 43318,Cc1ccnc(CNC(=O)CCC2CCCN2C(=O)CCc2ncc(F)cn2)n1 43319,c12ncc(cc1O)c1ccsc1[nH]c(=O)[nH]2.c1(NC=O)ccccn1 43320,CC(C(=O)N1CCC(OCC(=O)NC2(O)CC2)C1)C(F)F 43321,N1(C(CC(C)C)=O)CC(NC(c2ccn(C)c2-c2ccccc2)=O)CC(O)C1 43322,C1(C)(C(N2C(CNC(c3n(CC)nc(C)c3)=O)CCCC2)=O)CCC12CCC2 43323,N1(C(c2cc(CCC)on2)=O)CCC(C(F)CNC(C2CC2C#C)=O)CC1 43324,c1(OC)cnc(C(N2CC(C(F)(F)F)C(CNC(c3n[nH]cc3Br)=O)C2)=O)cn1 43325,Cn1cnc2cccc(C(N3CCCC3CN(C(=O)C=CC(N)=O)C3CC3)=O)c12 43326,C=CC(C)(C)CCCNC(C1(NC(C2CC(=O)OC2(C)C)=O)CSC1)=O 43327,C(C)(CCCCNC(=O)COCc1ccc(OC)cc1)NC(C(C)OC)=O 43328,c1(C(C)C)cc(CN(C)Cc2csc(NS(C)(=O)=O)n2)no1 43329,CC1(C(=O)NCCC2CCCO2)CCN(C(c2ccnc(O)c2)=O)C1 43330,Cc1ccccc1C1(C(=O)NC2C3CC2N(C(=O)COCCCN(C)C)C3)CC1 43331,c1(C(N2CC(OC)(CNC(=O)CCCn3ccnn3)C2)=O)cc(C)c(F)cc1Cl 43332,N1(C(c2c(C(C)C)nco2)=O)CCC2CCCC12CNC(C1CCCOC1C)=O 43333,C1(C(N(CC(CNC(c2c(C)nc(O)cc2)=O)(C)C)C)=O)CC2CCCCC2O1 43334,C1(CC)C(=O)NCCCN1C(C1C2CCC(C2)N1C(C1(CC)CNC(=O)C1)=O)=O 43335,n1(CCC)cc(C(=O)NCC(C)(C)NC(c2n[nH]cc2Br)=O)nn1 43336,N1(C(=O)NCC(C(C)C)C)CCCC(C(N)=O)C1 43337,c1(C(=O)NC(C)C(C)(C)NC(C2(C3CCCO3)CC2)=O)cc2sc(Cl)cc2s1 43338,N1(CC)CC(C(=O)NC2CC23CC(NC(=O)CC2(C(F)F)CC2)C3)CC1=O 43339,N1(CC(C)(C)NC(C(C)=CC)=O)CCN(C(=O)Cc2nccc(OC)n2)CC1 43340,C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(=O)c2cccnn2)O1 43341,c1(CCCC)cc(=NC(=O)Cc2cccc(Cl)c2Cl)[nH][nH]1.C12(CC1)C(=O)NC2=O 43342,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=COCC2)C(O)C1)=O 43343,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43344,c1(CCNC(CC2(NC(Cc3cc(C)[nH]n3)=O)CCCC2)=O)c(C)noc1C 43345,N1(C(CC=C)=O)CC(NC(C2(COCC)CCCO2)=O)C(c2cnn(C)c2)C1 43346,C1(NS(=O)(=O)C2CC3(CC3)C2)CCOC2(CCC(F)(F)CC2)C1 43347,N1(C(C(C)C2CCC2)=O)Cc2ccccc2C(NC(c2cccc(CO)n2)=O)C1 43348,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43349,C1(CC)CC(F)(F)CN1C(C1CCCC1c1ccccc1)=O.C1(C(=O)O)(CCF)CC1 43350,c1(C(=O)NC2CC2NC(=O)C(O)Cc2cnc[nH]2)cccc2[nH]nc(O)c12 43351,N1(C(C(C)c2ccsc2)=O)CCOC2(CCN(C(c3ccc(F)nn3)=O)CC2)C1 43352,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(c2cccs2)=O)C1 43353,c1(OC)cccc(C(=O)NCC(C)(C)CNC(C2CC3CCC2O3)=O)n1 43354,Cc1nc(CC(=O)N(C)CCN(C(=O)C2=CCCC2)C)c(Cl)s1 43355,c1(OC)ccc(Cl)c(F)c1C(=O)NC1CC1NC(c1occc1C)=O 43356,c1(OC)cc(C(N2CC(C(C)NC(c3occc3C)=O)C2)=O)cc(N)c1O 43357,c1(OC(N(C2(CO)CC(CO)C2)C)=O)nc(C(=O)N(C(C)(C)C)C)cs1 43358,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1 43359,C(CCCCC(=O)NCc1n[nH]cc1C(=O)NC1CN(C)CC1(F)F)OC 43360,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CC#C)CO 43361,N1(C(C2(Cl)C(C)(C)C2)=O)CCC2(CCC2NC(=O)CCP(C)(C)=O)CC1 43362,C1(C(=O)Nc2cncc(C)c2)CCC(C)N(C(=O)C(CO)N(C)C)C1 43363,C1(CNC(=O)C=CC2CC2)CCCCC1C(=O)N(CCO)CCO 43364,N1(C(C2CC(=C)C2)=O)CCC(C(N2CCC(N3CCC3)C2)=O)C1(C)C 43365,C(C(=O)NC(c1ncccc1C)C)(C(C)C)NC(=O)OC.C12CN(C1)C2=O 43366,Cc1cc2sc(C(N3CC(F)(CNC(=O)CCn4ccnc4)C3)=O)cc2s1 43367,N1(C(C2(C#C)CN(C(c3ccc(CO)o3)=O)C2)=O)CCC(C2CCC2)C1 43368,c1(C(N(CC(C)NC(c2cnc(Cl)c(N)c2)=O)C)=O)cnc2ncc(Cl)cn12 43369,c1(C(=O)NC(CC=C)CNC(=O)C(CC2CC2)OC)cccc(N(C)C)c1 43370,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1F 43371,c1(CNC(C(=O)OC)C2CN(C(C3CCCC3CF)=O)C2)cccc(=O)n1C 43372,CS(=O)(=O)CCCCCCC(=O)N1CCC(CO)C(NC(=O)Cc2cccnc2)C1 43373,C1(NC(C(CSC)O)=O)C2CC1CN(C(c1cn3ccsc3n1)=O)C2 43374,C(=O)(CC(C(C)(C)C)NC(=O)C(C)n1ccnn1)N(CC)Cc1ccnn1C 43375,Cc1cncc(C(=O)NC(C2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)(C)C)c1 43376,C1(C(=O)OC)CCc2cc(OC)ccc2N1C(=O)CCc1ccc(C)cn1 43377,c1(N2CCCC(NC(C3CC(OC)C3)=O)CC2)c(F)cccc1[N+](=O)[O-] 43378,N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCN(C(=O)CC23CCCC2C3)C(CF)C1 43379,C(=O)(C(CNC(=O)CC(=O)OC)CC(C)C)Nc1cc(CC)c(C)nc1 43380,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)Nc1c(OC)nsc1 43381,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43382,N1(C(CC2CCCC(NC(CCCCC=CC)=O)C2)=O)CC(C)CCCC1C 43383,C1(NC(CCc2onc(C)n2)=O)CCN(C(=O)CCc2scnc2C)CC1(C)C 43384,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCC2)=O)=O)C1 43385,c1(C(N(CC(C)NC(C(C)=CC2CC2)=O)C)=O)ccc(-c2nc[nH]n2)cc1 43386,N1(c2cc(N(C)CC)nc(C)n2)C2CCC1CC(NCC1CCN(CC)CC1)C2 43387,CC1CC2(CCN(C(=O)CCN3CCCC3=O)CC2)CN1C(C1CCC1(C)C)=O 43388,c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2nnn(C)c2C)=O)CCOC1 43389,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43390,C1(CCC)CN(C(=O)CSSC)CC1NC(c1nccn1C1CC1)=O 43391,C1(CNC(C(CC)CCOC)=O)CCC(C)(C)CN1C(=O)Cc1cc(C2CC2)on1 43392,CC(C)C(F)C(=O)NC1CCCN(C(c2cc(C3CCC3)[nH]n2)=O)C1 43393,C1(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CC(F)(F)C2)CCc2nc[nH]c2C1 43394,C=C(C)C(C)(N)C(=O)NCCc1ccn(-c2ccccc2)c1C 43395,c1(CN(C)C(C2(CO)CCC2)=O)cnc2cc[nH]c2c1.N12CC3C(C3C1)C2 43396,C12OCCC1NC2=O.c1(CN)ncc(I)s1 43397,c1(C(=O)NCC2CCN(C(C(C)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43398,c1(C(=O)NC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)C)cnc2sccn12 43399,c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1ccc(C)c(Cl)c1)=O)c1ccccc1 43400,C1(CCNC(C(CC)N(C)C)=O)CCCN(C(C2(c3ncco3)CCC2)=O)CC1 43401,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2ccc3[nH]ccc3n2)=O)CC(O)C1 43402,CC1C(C(=O)N(C(C)(C)CC(N2CC3C=CC2CC3)=O)C)=NOC1C 43403,c1(CNCc2ncc(F)cn2)cnn2ccccc12 43404,C#CCCCCC(=O)NCCCC(C)NC(C1CC(CC)(CC)C1)=O 43405,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43406,N1(C(c2cc(C)[nH]n2)=O)CC(F)(F)CC1C(=O)NC1CC(C)CCC1O 43407,C1(C(=O)NC2(CNC(C3(CC#C)CCCC3)=O)CCCC2)CCOC(C)C1 43408,c1(CN(C(c2occc2F)=O)CCO)cccc(F)n1 43409,C(=O)(C(O)CC(C)C)C1C(N2C(C(C(=O)OC)(C)C)CC2)C(O)C1 43410,CCCC(CC)C(=O)N1CCN(C(=O)Nc2ccc(F)c(F)c2)C(C)C1 43411,C(N=c1[nH]c2c(c(=NC3CCc4cccc(Cl)c43)[nH]1)SCC2)c1ccc(O)nc1 43412,C=CCC(CC=C)NC(=O)C(CC1CC1)NC(=O)C(C)=C(C)CC 43413,Cc1ncc(C(N2CC(C)(NC(=O)CCC3CC(C)C3)C2)=O)cc1C#N 43414,c1(C(=O)NCC2N(C(c3cnc(C)s3)=O)CCN(C)C2)ccc2c(c1)COCC2 43415,c1(CC)csc(C(F)(F)CNC(=O)C(=O)N(CC)Cc2cc(C3CCCC3)on2)n1 43416,c1(C(N2C(CNC(CC(C=C)(C)O)=O)CN(C)CC2)=O)cc(Cl)c(F)cc1C 43417,c1(C(=O)Nc2ccc(C=CC)cc2)ccc(COC(C)C)nc1C(F)(F)F 43418,C1(NC(c2cc(OC)ns2)=O)CCN(C(C)C(=O)N(C)C)CC1C 43419,C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)C(C)(C)OC(C)C)CC(C)(C)O1)OC 43420,C1(CC(=O)NCC(C)(C)CNC(C2(CCCF)CC2)=O)CC(C)(C)CO1 43421,N1(C(CCC(=O)NC)=O)CCC2(CC1)CC2(C)C(=O)NCCc1csc(C)n1 43422,Cc1cc(C(N2CCC(C)(CNC(C3(C)CC3F)=O)CC2)=O)cc(N)c1Cl 43423,C1(NC(=O)CCCCC2CC2)CC12CCN(C(=O)C=Cc1cncs1)C2 43424,C1(CC)CCN(C(=O)Cn2c(O)nnc2O)C(NC(C2COC(C)(C)C2)=O)C1 43425,N1(C(c2cccc(C)c2C)=O)CC(C2CN(C(=O)CC3CC4C=CC3C4)C2)C1 43426,c1(CC)c(C(=O)Nc2cccc(Cn3cnnc3)c2)cnn1C 43427,CC1CCN(C(=O)CCCC2CC2)CC1NC(c1ccc(Cl)c(N)c1)=O 43428,C1(C(N(C2CN(C(C3CCCCCC3)=O)C2)C)=O)CN(S(N)(=O)=O)C1 43429,C1(CC(=O)OCCN(C2C3(C(C=O)C3)C2)CCN(CCO)CC)CCCCC1(C)C 43430,c1(CC2(C(=O)NC(c3c[nH]nc3C(=O)O)=O)CC2(F)F)ccccc1 43431,N1(C(CCCCN(C(CCCOCC)=O)C)=O)CC(C)CCC1CC 43432,C1(OC2(C#C)CC2)CCCC1CN(C(c1sccc1OC(N)=O)=O)C1CC1 43433,c1(CNC(C(C)N(C)Cc2cccnc2)=O)cccc(NC(=O)N(C)C)n1 43434,N1(C(CNC(C(C)(C)C)=O)=O)CCCN(C(=O)CCc2ncco2)CC1C(C)C 43435,C1(C)(C(N(C)CC2CCCN2C(C2CCCN2C)=O)=O)CCOCC1 43436,C1(CNC(CCC(=C)C)=O)CC2COCC2N1C(c1ocnc1C(F)F)=O 43437,c1(C(=O)NCC(CNC(c2c[nH]c(=NC)o2)=O)F)ccc2nccnc2c1 43438,c12ccc(c(Cl)c1C)OCC(=O)NC2C.C(C(O)COC)N(CCC)C 43439,C1(CC)CN(C(c2cc(C)[nH]n2)=O)CC1C(=O)NCCCn1cnnn1 43440,C(=O)(C(C)C1=CCCC1)NCCCNC(C(=Cc1cccnc1)C)=O 43441,C#Cc1ccc(CCC(=O)NCC(C)N(C(=O)CN2CCOCC2)C)cc1 43442,N1(C(CC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43443,c1(C(C)C(=O)NC2CC(Cn3cc(C(C)(C)C)nn3)C2)ccc(C(N)=O)cc1 43444,C1(C2CN(C(=O)C=Cc3nccs3)C2)(NC(c2c(C)occ2)=O)CC1 43445,C1(C(=O)NC2(CC(N)=O)CCC2)CCCN1C(=O)CC1CCC1 43446,N1(C(C(CCC)C)=O)CC2(CCNC(=O)CCSc3ccco3)CCC1C2 43447,Cc1ccnc(C)c1C(N1CCC1(C)CC(=O)NCc1nn(C)c(=O)n1C)=O 43448,c1(C(C(=O)NCC2N(C(c3c(CC)cco3)=O)CCSC2)C)c(C)nn(C)c1C 43449,O=C1CCC(C(N2CCC(CNC(=O)C(O)CCc3ccccc3)C2)=O)CCO1 43450,c1(CC)cc[nH]c1C(=O)NC(CNC(=O)C(C)N(C)C(C)=O)CCOC 43451,c1(C(=O)NC2(CNC(C3CCCCO3)=O)CC2)cc(F)cc([N+](=O)[O-])c1 43452,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43453,c1(C(N2CCC(NC(C(C(CC)C)OC)=O)CC2C)=O)ccc(C#N)cc1F 43454,c1(C(=O)NCC23C(CN(C(c4scc(C)c4)=O)C2)C3)cnc2cnn(C)c2c1 43455,C(c1ccncc1C)=CC(=O)N(C(CNC(C(CCOC)OC)=O)C)C 43456,c1(CSCc2onc(-n3cc(C)nc3)n2)cc2nc[nH]c2cn1 43457,Cc1ccc(C(=O)NCC(C2CCC2)NC(C23CSCC2C3)=O)nc1 43458,c1(CN(C2CC3CC2CN3)C(c2ccc(C)s2)=O)cc(Cl)c(N(C)C)c(Cl)c1 43459,N1(C(C2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(=O)CCc1ncco1 43460,c1(C(N(CC(CNC(C2=C(C)OCC2)=O)(C)C)C)=O)cc(=O)c2ccccc2o1 43461,C1(C(=O)NC2(C(N(CC#C)CC3CCCO3)=O)CC2)CC1C1(C)COC1 43462,c1(CC)cnccc1C(N1CCCC1CC(=O)OC)C(=O)NC(C)CC 43463,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(c2cccc(CC)n2)=O)C1 43464,c1(CC(=O)N(CC(O)CN(C)C(C2CC2F)=O)C)ccnn1C 43465,C(=O)(CCN=c1[nH]cncc1Br)NC(C)C(=O)NCCO 43466,c1(C(N(CC(C)(C)NC(C2CCCC2O)=O)C)=O)nccc2ccncc12 43467,N1(C(c2c(OC)nsc2)=O)CCN2CCN(C(C3CCCC(=O)N3C)=O)CC2C1 43468,C=CCC(C)(C(=O)N1CCC(N(CCO)C(c2cc(C)ncc2C)=O)C1)N(C)C 43469,C(=O)(C(CC)NC(c1ocnc1C)=O)NC1CN(C(CC)=O)C1 43470,C(CC(C)(C)C(=O)NCC1COCCN1C(=O)C=CCOC(C)(C)C)OC 43471,C1(NC(C(C)(c2cn(C3CCOC3)nn2)N2CCCC2)=O)CC2CCC(C1)C2 43472,C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(c2cccs2)=O)C1 43473,C1(CCNC(C(C)n2cnnn2)=O)CCCN(C(c2cnoc2)=O)CC1 43474,c1(C(=O)NC2C(NC(CCN(C(C)C)C)=O)CC2)cnc(Cl)c(N)c1 43475,C1(NC(C2CC3(CC(=C)C3)C2)=O)CN(C(=O)CCCC(C)O)CC2(CC2)C1 43476,C1(C(=O)NC2(CCC(N3C(C)CCC3)=O)CCC2)CC=CC(O)C1 43477,C(CNC(=O)CN(C1CC1)CC)(CC(F)(F)F)NC(CCC(C)OCC)=O 43478,C(CCC(O)C(=O)NC)NC(c1c(CC)c[nH]n1)=O.N12CC3CC3(C1)C2 43479,c1(C(=O)NC2C(CNC(C(c3cccs3)SC)=O)C2)cc2ccc(F)c(F)c2o1 43480,c1(CC)nc(CC(=O)NCCCCN(C)C(C2CCC(C)O2)=O)cs1 43481,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(N1CC(OC(=O)N(C)C)C1)=O 43482,c1(-n2cc(C(=O)NCCCCNC(C3(CC)CCOC3)=O)nn2)ccccc1F 43483,c1(OC)ccc(CN2CCCCC2(C)C(=O)O)c(O)c1OC 43484,CON(CSC)C(=O)C(F)(CNC(CCCCC(=O)OC)=O)C(C)C 43485,N1(C(C)=O)CCCCC1C(=O)NC(C)CCN(C(=O)CSc1cccnc1)C 43486,Cc1cc2nc(C(=O)NC3CC(C)N(C(=O)C#CC4CC4)C3)cn2cc1C 43487,O=C(C(F)C(F)(F)F)NCC1CCCCC1C(=O)NCC1CC2CCC1O2 43488,C1(NC(c2ccc(CNC(C3C(C)C3C)=O)cc2)=O)CCC(=O)NC1C 43489,c1(CC(=O)Nc2ccc(C(=O)NCc3c(CC)occ3)cc2)c(C)cccc1C 43490,N1(C(C(C)(C)c2cccs2)=O)CC2CCCN(C(C34COCC3C4(F)F)=O)C2C1 43491,C#CCCCC(C)C(=O)N1CCC1CC(=O)Nc1ncc(CC#C)s1 43492,C1(NC(Cc2n(C(C)(C)C)ncc2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43493,S(=O)(=O)(c1cc(C)c(Br)cc1F)NCCc1ccc(C(=O)NC)cc1Cl 43494,C1(NC(CCC2CCC(NC(CC(C)(F)F)=O)C2)=O)CCCCCC1O 43495,N1(C(C(=O)NC)C2CC(OCOC)C2)CCC(N2CCC(C)(O)C2)CC1 43496,c1(C(=O)NC23CC(CNC(C(C)SC)=O)(OCC2)C3)ccn2cnnc2c1 43497,N(C1=NCCC(=O)ON1)CC1(COC)CCC1.C1(C(N)=O)CCCCO1 43498,C(=O)(CCCCCN(C1COCCC1c1ccccc1)C)OCC 43499,C(c1ccc2ncccc2c1)=CC(=O)NC(CNC(C(C)=CC)=O)C1CC1 43500,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43501,c1(C(=O)NCCCCCNC(C2(CCC)CC2)=O)ccc(F)c(OC(F)F)c1F 43502,c1(C(=O)NC(C)CCCNC(c2cnn(C(F)F)c2)=O)ccc(C(F)(F)F)nn1 43503,N1(C(c2c(C)n(C)cn2)=O)CCC(NC(C23CC(C2)C3)=O)C(C)C1 43504,C(=O)(CCC(F)(F)CN)OCC.c12ccc([nH]1)c(=O)[nH]2 43505,c1(C(N2CC(C)C(NC(=O)CS(C)(=O)=O)CC2)=O)ccc2c(O)nc(=N)[nH]c2c1 43506,c1(NC(C(C2CCN(C(C3(C)CC(=C)C3)=O)C2)C)=O)ccc(F)cc1C 43507,c1(C(=O)NCc2cccc(P(C)(C)=O)c2)ccc2cc(Cl)ccc2c1 43508,C1(CNC(Cc2c(C)con2)=O)(NC(c2ncsc2C)=O)CCCCC1C 43509,N1(C(C(C)NC(=O)NC)=O)CC(NC(c2cnn(C)c2SC)=O)C2(CC2)C1 43510,N1(C(C(CNC(C(C(C)C)OC)=O)(C)C)=O)CC(=O)N2CCCC2C1 43511,C(=O)(CC(CNC(=O)CC1(C)OCCO1)C1CCC1)N(CC(C)C)C 43512,C=CCC(CNC(=O)CNC(=O)CC(C)CC)CC(C)C 43513,Cc1ccc(O)cc1NC(=O)CCCCCNC(=O)C(F)C1CCCC1 43514,CC1(C)CCN(C(=O)COCC(=O)NC2CCC2)CC1C(=O)N(CCO)C1CC1 43515,C=CCCCCCCCC(=O)NCc1cn(CCC(N2C(C(N)=O)CC2)=O)nn1 43516,C1(NCC(=O)NCC)CN(C(C2CCCN(C)C2)=O)CC1C.C1(=O)CN1 43517,c1(C(N2CC(CNC(=O)C=Cc3ccco3)C3C2C3)=O)cccc2nc(Cl)cn12 43518,S(=O)(=O)(c1cccnc1NCc1cc(Cl)n(C)n1)NCc1ccc(OCC)nc1 43519,N1(C(c2cnc(CC)o2)=O)C(CC(=O)NC2C=CCCC2)C2CCCC12 43520,c12ccccc1C(=O)N2.C1(CC(=O)NCc2csnn2)(COC)CCC1 43521,c1(CC(=O)NCCN(C(c2c(OC)noc2C)=O)C)ccc2c(c1)ncn2C 43522,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)F)cccc(Br)c1F 43523,c1(OC)nc(C(=O)Nc2cccc(OCc3cccnc3)c2)ncc1F 43524,C1(O)(CN(C(C)=O)C)CCN(C(=O)CC2(C)CCOCC2)C1 43525,C1(O)(C(=O)NC2CN(C(c3c(C(C)(C)C)[nH]cn3)=O)C2)CC(F)(F)C1 43526,N1(C(c2n(C(C)C)ncc2)=O)CCCCCC(NC(=O)C(C)n2ccnc2)C1 43527,N#Cc1ccc(F)c(C(N2CCC3CCC23CNC(c2cnncc2O)=O)=O)c1 43528,CC1CCN(C2CCCC2)CC1.[nH]1c(-c2ccc(C)o2)nnc1C 43529,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43530,c1(C(=O)NCC2(CCNC(C3C(C)OC(=O)N3)=O)CC2)nc2ncccn2n1 43531,C1(CC(=O)N(CC(CC)OC)CCO)CCCC1NC(=O)C=Cc1cncs1 43532,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43533,c1(OC)nccc(C)c1C(N1CC(CNC(=O)Cn2cncn2)C(O)C1)=O 43534,c1(C(c2n(CC(=C)C)nnn2)NCC(C)(C)C2CCC2)cccc(C)c1C(=O)OC 43535,C(CC(C)C(=O)NCC(CC)NC(C1(C)CCCC1)=O)=CCC 43536,C1(C(=O)NC2CCN(C(C3CCOC3)=O)C23CC3)CCC2(CC1)OCCO2 43537,c1(C(=O)NCC2(COC)CN(C(C3COC(=O)N3)=O)C2)ccc(C)cc1C 43538,C(=O)(CC(C)C(F)F)NC1CCCC(CNC(C=Cc2cnc(C)s2)=O)C1 43539,c1(CC)cc(C(=O)NC2CN(C(c3ccc(-n4ccnc4)o3)=O)C3CC23)n(C)n1 43540,c1(C(=O)NC2(C)CCN(C(c3ccc(Cl)c(O)c3)=O)C2)ccc2nn[nH]c2c1 43541,Cc1c(C(=O)N(C)CC2(Cl)CCC2)sc2nc(-c3ccco3)ccc12 43542,N1(C(CC=C(C)C)=O)CC2CC2(CNC(=O)CCN(C)C)C1 43543,c1(N2CC(CC(C)NC(C(CC)SC)=O)C2)nc(C(=O)OC)nc2ccccc12 43544,c1(CC(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)CC2F)c(F)cc(Br)cc1F 43545,C(CCO)(C(=O)O)c1cn(C(c2ccc(Cl)cc2)C(=O)N(C)Cc2cccnc2O)nn1 43546,n1(CC)cnc2nc(NCC3CCCN(CCF)C3)nc(CC3CCN(C)C3)c12 43547,C#CCCCC(C)C(=O)NC1CCC(NC(c2c(C)cnn2C)=O)C1.Cc1occc1 43548,Cc1cc(C(N2CCC(CCNC(C3CCN(C)C3)=O)C2)=O)cnc1C(F)(F)F 43549,C12(CC)COC(C(=O)NCCCC(C)(C)NC(=O)COC3CCCC(C)C3)(C1)C2 43550,Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(=O)CNS(C)(=O)=O)s1 43551,CC(N=c1ccnc(C2CCC2)[nH]1)C1CC(NC(c2cccc3nc[nH]c23)=O)C1 43552,CC1=NOC(C)(C(N2CCC(CNC(c3c(OCF)noc3C)=O)C2)=O)C1 43553,c1(C(N(C2CCNCC2)CCCC)=O)cc(C)ccn1.C1(=O)CO1 43554,c1(CN(C(=O)CCCNC(=O)C(O)CN2CCCC2)C)nccc(O)n1 43555,c1(C(N2CCC(C(C)NC(C3C(C)COCC3)=O)C2)=O)ccc(N(C)C)c(F)c1 43556,C1(C(N2CCOC(C3CN(C(=O)C=C4CCSCC4)C3)C2)=O)(CC)CC(C)(C)C1 43557,N1(C(c2ncc(C)cc2F)=O)CC2CCC(N(C)C(C3CCCC3O)=O)C2C1 43558,c1(C(N2C3(C(=O)NC4C(C)(C)C4)CC3CC2)=O)ccc2ccoc2c1 43559,C(=O)(CCS(C)=O)NCCN(C(C(C)N(C(C)=O)C)=O)Cc1ccccc1 43560,C1(NC(N(c2nc(C)c(C3CCCCC3)s2)C)=O)CNC(=O)C12CC2 43561,C(CCCCC(=O)N(CCOCCO)CCNC(C1CCC(C2CC2)C1)=O)SC 43562,c1(OC)ccc(C)c(C(=O)OCC(=O)NC(=O)Nc2cc(Cl)ccc2OC)n1 43563,C(=O)(CC(C(F)F)c1cccc(F)c1)N(CC(C)N(C(C=C(C)Cl)=O)C)C 43564,CC1(C)C(NC(C2CCN2C(C)(C)C)=O)CC1O.c12nn[nH]c1CNC2=O 43565,c1(CCNC(C(N(CCSC)C(C)(C)CO)=O)=O)cccc2ccccc12 43566,N1(C(C(C(C)C)SC)=O)CC2CCC1C(C(=O)NCCCc1n[nH]c(C)n1)C2 43567,N1(C(c2c(CC)occ2C)=O)CCC2(CC(C(=O)NCC#CCOC)C2)C1 43568,C1(N(C(c2cc(F)c[nH]2)=O)C2CC2)CCCCCC1.C12CCN(C1)C(=O)CC2(C)C 43569,C1(NC(Cn2nnc(=N)[nH]2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43570,c1(OC)c(C(=O)NCCNC(=O)C(CSC)OC)cc(Cl)cc1C.C1CC1 43571,N1(C(c2c(OC)ccc(Br)c2)C(=O)NCC(F)F)C2CCC1CC(F)C2 43572,c1(C(=O)NC(c2cn(CCO)nn2)C)cc(F)cc(Br)c1 43573,CC1CN2CCN12.C(=O)C(CC(F)F)N(C)C(c1ccnn1C1CCC1)=O 43574,Cn1nc(C2CC2)cc1CC(=O)NC1CN(C(c2cncc(F)c2)=O)CC1F 43575,c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2)ccnc2c1cnn2C 43576,N1(C(C2(C)N(C(CC)=O)CCC2)=O)CC2CC(NC(=O)COCCO)C2C1 43577,N1(C(C(C)Oc2cc(F)cc(Cl)c2)=O)CCC2OCCN(C(=O)C(N)=O)C2C1 43578,C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CC2CCC(C1)N2C(=O)COC1CCC1 43579,C1(C(N(C)CCC2OCCO2)=O)CCN(C(c2cc(Cl)cnc2Cl)=O)CC1O 43580,c1(C(N(CC(CNC(C=C(C)C2CC2)=O)(C)C)C)=O)cc(C2CC2)nn1C 43581,C1(C(N2C(CN(C(C3CCN(C(C)=O)C3)=O)CC)CCCC2)=O)OCCOC1(C)C 43582,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CCCC1 43583,N1(C(c2c(OC)ccc(F)c2)=O)C2CCC1CN(C(=O)C=CC1CC1)C2 43584,CC1CN(C)C(=O)CN1C(=O)CCN(C)C(c1ccc(Cl)cc1)=O 43585,C(=O)(C(CCC)OCC)N1CCC(C(N2CC(CCCC)C2)=O)C1 43586,C#CCC(C(=O)NCCCNC(N)=O)NC(C1CC=CCC1)=O 43587,C1(CC(=O)NC2C(NC(CSCC=C)=O)C2)OCCCC1(C)C 43588,C(=O)(C(O)C(F)(F)F)N1CC2(C(C(=O)NCc3ccc(OC4COC4)cc3)C2)C1 43589,N1(C(CSCCC)=O)CC2CC1CN2c1cc(Cl)nc(SC)n1 43590,C1(C(=O)NC(CNC(c2cc(C)n(C)c2)=O)C2CC2)CC(c2cccc(F)c2)=NO1 43591,c1(C(N2CCC(CN(C)C(C3CC3CF)=O)C2)=O)cccc2nccn12 43592,c1(-c2cn(C3CN(C(COCCCCC)=O)C3)nn2)ccc(OC(C)C)cc1Cl 43593,c1(CCCCNC(c2ccccc2)CCC)ccc(N2CCC(N)CC2)cc1 43594,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCC(C(C)C#N)CC1 43595,n1(CC(=O)NCCn2cc(C(=O)NC3CN(c4nncs4)C3)nn2)cnnc1O 43596,c1(C(N2CCC(O)(C(Cl)(Cl)Cl)C2)=O)ccc(C(=O)OC)nc1 43597,N1(CC(=O)NC(CC)(C)C)CCC2(CC1)CC2(C)C(=O)NCC1CC2CCCC12 43598,C1(C(N(CC#C)C)=O)CC12CCN(C(=O)CN1CC(C)(C)C1)C2 43599,C(c1cocn1)=CC(=O)NCCCN(C(C1CCC1c1ccccc1)=O)C1CC1 43600,C1(NC(c2ccc[nH]2)=O)CN(C(C23CCC(CC2(F)F)C3)=O)Cc2nccn2C1 43601,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43602,N1(C(C(C)C)=O)CC(C(=O)O)CO1.n12cc(nn1)CNC(=O)C2C(=O)OC(C)(C)C 43603,c1(C(N2CCC3(NC(c4cc(Cl)sc4Cl)=O)C(C2)C3)=O)ccc2[nH]nc(O)c2c1 43604,C1(F)(C(N(C2CC(C#N)C2)CC#C)=O)CCN(C(=O)CCCOC)C1 43605,CC(C)(C(=O)N1CC(=O)N1)c1ccno1.C1(CO)(SC2CC2)CC1 43606,Cc1nn(CC(N2CCC(C(C)CNC(c3cc(C#N)c[nH]3)=O)CC2)=O)cc1Cl 43607,N1(C(C2C(=C)C2)=O)CCC2(CC1)CN(C(=O)C(C)n1cccc1)CC2CO 43608,c1(C(N2CCC(CCNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43609,C1(CNC(c2c(CC)nccc2)=O)CN(C(C2OC3CCC2CC3)=O)CCN1C 43610,C(=O)(C#CC1CC1)NC(CC)C(=O)NC1CCCC1N 43611,C(=O)(C1OC1)OCC.C(=O)(C(F)C1CCCC1)N(CC=O)C1CC1.C1CC1 43612,CC1COC2(CCC2)CN1C(=O)C(=O)Nc1ccc(C2CCN3CCC2C3)cc1 43613,N1(C(C(C)(O)C(F)(F)F)=O)CCC2(C1)CN(C(=O)COc1cn[nH]c1)CCO2 43614,C(=O)(C(CC(C)C)N(C)C)N1C2(CC2)C1.C1(C(F)(F)C(=O)OC)(OC)CCOCC1 43615,C1(C(=O)NC(C(=O)NCc2cc(C)n(C)n2)Cn2ccnn2)CN2CCN1CC2 43616,c1(C(N(C2CCN(C(CCC(=C)C)=O)C2)C)=O)ccc(Br)cc1OC(F)(F)F 43617,CCCC(C(=O)NC(C)(C)CNC(c1cccc(COC)c1)=O)S(N)(=O)=O 43618,c1(CC)nnc2cc(N3CC(CNC(=O)C(C)C(F)F)(OC)C3)ncn12 43619,C1(O)(CNC(C(C2CCN(C(CCSC)=O)C2)C)=O)CC2C=CC1C2 43620,c1(C(C(=O)NC2CC2)N(C2CCC(F)(F)C2)C)cccc(C(F)F)c1 43621,C(=O)(C1=CCCCCC1)NC(C)CCNC(=O)Cn1cc(Br)cn1 43622,c1(CNCC(O)C(F)(F)F)c(O)ccc(F)c1F 43623,CCC(=O)CCC(=O)NC(C)CCNC(c1ccc(C2CC2(Cl)Cl)cc1)=O 43624,C1(N)CCN(C)C(=O)C1.CC(C)CC(O)c1cn(C2CCC(C(=O)NNC=O)C2)nn1 43625,N1(c2cc(NCC(CC)N(C)C)ncn2)CCc2c(F)ccc(F)c2C1 43626,C1(C)(NC(CCCNC(C(C)C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43627,C(=O)(C1CC(=O)c2ccccc21)N1CC2C(CN(C(=O)C3=CCOC3)C)C2C1 43628,CN1CCCCC1C(=O)N(CCC(N1CC(N(C)C)C(CO)C1)=O)CCO 43629,CCC(C)C(C(=O)N(C1CCN(C)CC1C)C)N(C(=O)CC)C.c1nc(=O)o[nH]1 43630,Cc1ccc(C)c2[nH]c(C(=O)NCC3CCC3NC(C3CCS(=O)CC3)=O)cc12 43631,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43632,C1(C(=O)NCC(CC=C)OC(=O)NC2(C)CC2)CCCN(C(=O)OC(C)(C)C)C1 43633,c1(C(=O)NC2(CC)CN(C(=O)C=CCF)C2)cc2c(s1)COCC2 43634,C1(C(=O)NC2CCCC(C)C2)CC2(CCC2)CN1C(=O)Nc1ccc(=N)[nH]c1Cl 43635,c1(C(N2CC(N(C)C(C3(c4cccs4)CCC3)=O)C2)=O)cnn(C)c1N 43636,C(CCCCCNC(c1cc(Cl)c[nH]1)=O)N(C(C(c1cccc(Cl)c1)C)=O)C 43637,C1(CNC(=O)Nc2occ(C(C)(C)C)n2)CCN(c2ccc(Cl)cc2)C1=O 43638,C1(C)(CC)CC(OCC(c2cccnc2)c2cnc(C)o2)CCO1 43639,CCCCCC(F)C(=O)OCC.C12CCCC(C1)CC(=O)C(OC)OC2 43640,c1(C(N2CC(CN(C)Cc3ccccc3)C2)=O)ccc2nc(O)oc2c1 43641,C1(CC(=O)NCCN(CC(C)O)C(c2cscc2F)=O)CCC(C)(C)CO1 43642,c1(C(N(C)CC2CN(C(=O)C(F)OC(F)(F)F)CCO2)=O)cccc2nccn12 43643,c1(C(=O)NCCC2(C(N3CC(n4cnnc4)C3)=O)CCC2)ccnnc1 43644,c1(C(N(C(C)C)CCNC(C2(C)CC=CCO2)=O)=O)cc2ccc(O)cc2n1C 43645,C(=O)(C(F)(F)C(O)C(C)C)NCC1=CCN(C(c2ccc(C(C)C)cc2)=O)CC1 43646,c1(C(=O)OCC)cnc(N2CCS(=O)C(C)(C)C2)cc1C 43647,C1(NC(C=CC(C)C)=O)CC(NC(=O)Cc2ccccc2)CC1O 43648,N1(C(CNC(CCC(C)C)=O)=O)CCC2(CNC(=O)CC(F)(F)F)CC2C1 43649,C1(OC)CC(CNC(c2nnc(C)s2)=O)N(C(C2CCC(C)S2)=O)C1 43650,C1(CC(n2cc(CSC)nn2)C)CCCN1N1CC=CC1c1ccccc1 43651,N1(CC(=O)N(C(CCNC(Cc2nnc(C)o2)=O)C)C)CCC(CO)CC1 43652,c1(CCC(=O)Nc2ccc(Cl)cc2)cnc(Br)cn1 43653,CC(C(=O)N1CCCC1C1(O)CN(C(C2C3CCCCCC23)=O)C1)S(N)(=O)=O 43654,c1(C(N2CC3C(NC(=O)CO)CC(C3)C2)=O)n[nH]c2ccc(Cl)cc12 43655,Cc1cnc2cccc(C(=O)NC(C)C(C)NC(c3sccc3C(C)C)=O)n12 43656,C1(CNC(C(c2ccc(F)cc2)OC)=O)COCCN1C(C1CC(=O)N(C)C1)=O 43657,C(=O)(C(C)(CO)CO)N1CCCC(C(=O)Nc2c(C(C)(C)C)cccn2)C1 43658,c1(C(=O)NC2CCN(C(C3OC4CCC3C4)=O)CC2)ccc2nccnc2n1 43659,C(CCC(N)=O)(C(=O)N1CC(CCNC(=O)CC2CCCC(C)(C)O2)C1)N(C)C 43660,Cc1cccn(CC(=O)NC(C2CN(C(C3CC3c3cc[nH]n3)=O)C2)(C)C)c1=O 43661,C1(NC(N(C)CC2CC(=O)N(c3ccc(Cl)cc3)C2=O)=O)CCS(=O)(=O)C(C)(C)C1 43662,N1(C(CN(CCC#C)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)CCC1C 43663,N1(CC(=O)NCC(C2CCC2)OC)CCC(O)(CN2C(=O)CN(C)C2=O)CC1 43664,c1(C(N2CCC(F)(CNC(CC3C(CC)C3)=O)C2)=O)cc2c(cn1)CCCC2 43665,O=S(=O)(c1cnccc1N1C2CCCC1COC2)NCc1nc(C(F)F)ccc1Br 43666,C1(F)(CNC(C(CC2CC2)OC)=O)CCN(C(=O)CC2CC(=O)C2)C1 43667,C1(CC(C)C)COCCN1C(=O)CCc1c(CC(F)(F)F)cccc1F 43668,c1(CCC(=O)N(CCCN2CCC(COC)C2)CCC)cc(C)no1 43669,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)C2CC2)C(C)C1 43670,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43671,N1(C(c2cc(C(C)C)[nH]n2)=O)CCCCCCC1C(N1CCCC(N=[N+]=[N-])C1)=O 43672,c1(C(=O)NC2CC(C)N(C(c3cc4cccnn4c3)=O)C2)ccc2nonc2c1 43673,c1(C(=O)OCC2(CN3CCN(C)CC3)CC(F)(F)C2)ccc(NC(C)=O)cc1Cl 43674,CC1(C)C(CC(=O)NC2CCC(NC(c3coc(Cl)c3)=O)CC2)CC1O 43675,Cn1cc(S(=O)(=O)CCNC(c2ccn(O)c(=O)c2)=O)cn1 43676,C(C(C)(C)C#CC(=O)NCCNC(=O)C1CC1)NC(CN1C(C)CCCC1)=O 43677,C=C(C)C1OCCC1CNC(C1CCCN(S(=O)(=O)C(CCC)CC)C1)=O 43678,C1(C#CC(=O)N2CCC(CCN(C(=O)CCCC(=O)N(C)C)CC)C2)(CC)CC1 43679,C1(C(=O)OCCCOCCS(C)(=O)=O)OCC2COCCC12 43680,Cn1cncc(C(=O)NC2CCC(CC(=O)Nc3ccccc3O)C2)c1=O 43681,C(=O)(C(F)CC1CCOC1)N(CCN(C(=O)CC1(C)CC1)C)C1CC1 43682,N(C(=NCCOCC)N1CCC2(CCCCCC2)C1)C(C#C)CC 43683,C1(NC(C2N(C(c3cnc(C)nc3)=O)CC2)=O)CCCC(O)CC1 43684,c1(CNC(C2C(NC(C3N(C(C)=O)CCC3)=O)CC2)=O)n[nH]c(C)c1[N+](=O)[O-] 43685,c1(CC(=O)NC(CNC(CSC)=O)C2CCC2)cnns1 43686,C1C(OC(c2csc(O)n2)=O)C(=O)NC2CC(F)(C2)CN1.C1(OC)CCCC1 43687,C1(O)(C2CCN(c3n(C)nnn3)C2)CCN(C(=O)Nc2c(Br)ncn2C)C1 43688,Cc1cc(C(=O)NCC#CC(=O)N(C)CC2CC2(F)F)ccn1 43689,C(=O)(C1CCCc2c1ncn2C)N1CC(NC(c2c(C)occ2)=O)C(O)C1 43690,C1(C(N(CCN(C)C)CC)=O)C=CCN(C(=O)C(CSC)OC)C1 43691,C1(NC(CCCCNC(c2c(CC)cccc2)=O)=O)CCCOC12CCC2 43692,N1(C(C2(C(C)(C)OC)CCCC2)=O)CC(C)CN(C(=O)CCN(C)C)C(C)C1 43693,c1(CCC(=O)NCCN(C(CC=CC)=O)C)ccccc1 43694,Cn1c(C(=O)NC2CC(F)C2)ccc1C1COCCN1C(=O)Cc1cnc[nH]1 43695,c1(C(N2CCN(C(c3ccn(COC)n3)=O)C3C2C3)=O)cn2c(C)cccc2n1 43696,C1(C(=O)NC2CC(CCNC(CSC)=O)C2)CSc2ccccc2O1 43697,c1(C(=O)NC2(CNC(C(CC)(C)F)=O)CCOC2)ccc(Cl)cc1Cl 43698,c1(N2CCC(CCOC)(NC(c3c(C)cnn3C)=O)C2)nc(Cl)nc(C)c1C 43699,N1(C(C2(C(C)C)CCN(C(c3n[nH]cc3Cl)=O)C2)=O)CC2(CCCO2)C1 43700,C1(C(N2CCC(C(C)(C)NC(C3CC4(CSC4)C3)=O)C2)=O)CC2CCC1C2 43701,Cc1cccc(C(=O)NCC2CCC2C(=O)N(CCCO)CCOC)c1 43702,C1(N(C(C=CC(=O)NC(C)CN(C)C2CC2)=O)C)CCCC1C 43703,CCC(CCC(=O)N1CCCCC1CCO)NC(c1cc(C)ncn1)=O 43704,C1(CNC(CC2(C)CC2(F)Cl)=O)C2CN(C(c3ccn(C4CCC4)n3)=O)CC12 43705,C=CCCCC(=O)Nc1cccc(OCC(F)(F)F)n1.C12CC1CNC2=O 43706,CC1(C)C2CC(C(=O)NC3CN(C(C4CCS(=O)(=O)CC4)=O)C3)CC12 43707,CCC(C)C(C(=O)NCCN1CCN(C(C2CC2OC)=O)CC1)NC(=O)OC 43708,c1(C(=O)NC(C(C)C)CNC(=O)CN2CCCCC2)cc(N)c(O)c(F)c1 43709,CC(CNC(=O)CCN1CCOCC1)C(F)C(=O)NC(C1(O)CCC1)(C)C 43710,c1(C(=O)NCC(CC)NC(=O)Cn2ncccc2=O)ccnc(S)c1 43711,C1(CCNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 43712,c1(NC(C2N(C(COCC)=O)CCC2)=O)cc(I)cnc1Cl 43713,C(C(N=c1[nH]c(=N)[nH]c(=NCC(C)OC)[nH]1)c1ccco1)OC 43714,N1(C(C=C(C)C(F)F)=O)CCC(C2CC2)C1C(=O)NCC(CC1CC1)CO 43715,C(C(CC(C)C)C(=O)NCCOC1(C(N2CC(OC(C)C)C2)=O)CCOC1)OC 43716,CS(=O)C1(CNC(=O)C(CC2CCC2)NC(c2csnc2Cl)=O)CCC1 43717,c1(C(N2CC(CNC(C3=NOC(C)C3)=O)C(C)C2)=O)cncc2c1CCCC2 43718,C1(CC(=O)OCC(F)(F)F)CCCC(OCc2ccc(Cl)nc2)C1 43719,c1(C(N(C)CC2N(C(c3nnn(CC)c3C)=O)CCOC2)=O)ncc(F)cc1F 43720,C1(OC)(CNC(=O)Cn2cc(-c3cnc(C)cn3)nn2)CCSCC1 43721,c1(OC)c(F)ccc(C(=O)NCCN(CC(C)O)C(C2CCS(=O)(=O)C2)=O)c1F 43722,c1(CC(=O)NC2CCN(C(COCCC)=O)C2)ccccc1CS(N)(=O)=O 43723,Cc1cc(C(N2CCC(NC(C3CC34CCCC4)=O)C(CO)C2)=O)ncc1CO 43724,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC2C=CC1O2)=O 43725,c1(C(=O)NC2C(NC(c3c(C)cc(C(F)F)o3)=O)CC2)n[nH]c2c1COC2 43726,Cc1nc2ccccc2n1CC(=O)NC1CC(NC(c2[nH]nnc2C)=O)C12CCC2 43727,C1(CCC(C)(C)F)NC(=O)N(Cc2nn(C)cc2Br)C1=O 43728,C1(CC=C)(C(N2CCC(C#N)C2)=O)CCN(C(=O)COC(C)=O)C1 43729,c1(C(C(=O)NCC(F)F)N(C(C23CC(C2)C3)C)C)cncc(Cl)c1 43730,CC1C(NC(=O)C(C)(Cl)Cl)CCCN1C(c1cnn(C(F)F)c1)=O 43731,C1(C(N2CCC(C(N)=O)C2)=O)(CC)CCCN1Cc1cc(Br)c[nH]1 43732,N1(C(=O)NCC(c2ccsc2)C)CCn2c(C3CCOC3)nnc2C1 43733,c1(NC2CCCN(C)C2)nc(N2CCC3CCCC3C2)nc2c1ncn2C 43734,N1(C(C(CC=C)CNC(=O)CN2CCN(C)CC2)=O)CC(C2CC2(F)F)C1 43735,C(CC1CCCC1)(C(=O)NCC(CO)NC(=O)Cn1cnnc1O)NC(C)=O 43736,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 43737,Fc1cc2nc(Cl)nc(NCC3CCCN3S(=O)(=O)c3ccc(Br)s3)c2cc1Br 43738,C12(C(N3CCC(COC)C3)=O)COCC1CN(C(c1ccon1)=O)C2 43739,C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1ncccc1CSC)=O 43740,C1(CC)CCCN(C(C2(NC(=O)C(C)NC(C)=O)CC2)=O)CC1 43741,Cn1nc(C(=O)NCCNC(=O)Cc2ccc(F)c(C(F)(F)F)c2)ccc1=O 43742,c1(C(N2CCCC(NC(C(CCSC)(C)C)=O)C2)=O)cc([N+](=O)[O-])cc(C)n1 43743,C(CC1=CCN(C(c2coc(C(N)=O)c2)=O)CC1)NC(CN1CCN(C)CC1)=O 43744,C1(NC(CCC#C)=O)CS(=O)(=O)CC1NC(c1cc(SC)c(C)o1)=O 43745,c1(C(N(CCCCN(C(c2nn(CC)c(O)c2)=O)C)C)=O)c(C)cnnc1O 43746,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 43747,Cc1cc(C#N)ccc1COCC(=O)NCCCc1nnc(C(C)(C)C)s1 43748,c1(CC(N2CCC(NC(CNS(NC)(=O)=O)=O)(CF)C2)=O)cc(F)cc(Cl)c1 43749,CCC(C)CC(C)NC(=O)CC1CCC(NC(c2cnn[nH]2)=O)CC1 43750,C12(CNC(=O)CC3CC=CC3)CCCC1N(C(=O)C=Cc1cccnc1)CCC2 43751,C1(NC(CCc2cc(C)on2)=O)CC1C1CCCN(C(=O)CN2CCN(C)CC2)C1 43752,n1(C)c(=O)c2cccnc2s1.c12ccc(cc1)C(=O)CCC(=O)OC2 43753,N1(C(CCOCCNC(C2(C)CC2(Cl)Cl)=O)=O)CC2(CCCC(CO)O2)C1 43754,S(=O)(=O)(c1ccc(NCc2ccc3c(c2)CN(C)C3)c(F)c1)NC1C(CC)C1 43755,C1(CS(=O)(=O)N(CCOC)Cc2cccnc2)CCCCCC1.C1CC(=O)O1 43756,c1(C(=O)OC)ccc2c(c1)CCO2.c1ccc(C)c(C(=O)NC(=O)OC)c1 43757,C1(CCN(C)C(C2(N(C)C)CC2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)CC1 43758,N1(C(C(=O)NCC(C)C)=O)CCCN(C(CC2(C)CC2)C(=O)N(C)C)CC1 43759,C1(NC(C=NOC)=O)CC(NC(c2cscc2Cl)=O)C12CCOCC2 43760,C1(CN(C(COCCCCC)=O)C)CCCCN1C(=O)Cc1csc(S)n1 43761,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 43762,C(=O)(C1COc2ccccc21)NCCCC(CCC)NC(=O)C=Cc1cnc[nH]1 43763,c1(COC(C)C)cccc(OC)c1.n12nnnc1C2NCc1cc(I)cs1.CC 43764,CC(C)(C)C(CNC(C1CCC(C)(C)C1)=O)NC(=O)CN1CCC1 43765,C(=O)(CCC(=O)N(CC(C)NC(C1CSCN1C(C)=O)=O)C)NNC(C)=O 43766,c1(C(=O)NCC2CCC(C)CN2C(=O)C(F)F)cnc2sccn2c1=O 43767,C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(c2c(C)cn(C)n2)=O)C(O)C1 43768,C(C(=O)N1OC2C=CC1CC2)(C1CCOC1)NC(C1C=CCS1)=O 43769,c1(N(C)C)ccc(C(=O)NC2CCOC(C(=O)NCC3CC3Cl)C2)nc1 43770,NC1C2CCC1N(C(c1ccnc(OCC(F)(F)F)c1)=O)C2 43771,c1(C(C)C(C)N(C(C)C)CC23COC(CO)(C2)C3)ccc(S(C)(=O)=O)cc1 43772,c1(N(C(COCC)C)C)nnc(-c2cc[nH]n2)n1CC1CC(OC)(OC)C1 43773,c1(C(N(C2CN(C(c3ccc(CO)o3)=O)C2)C)=O)n[nH]c2c1CC1CC21 43774,C(=O)(C(CCc1ccc(Cl)cc1)C(C)(C)C)NC1CC1C(=O)N(C1CC1)CC 43775,c1(S)ccccc1.c1(CNC(C(C)SC)C)cn(C2CCOC2)nn1 43776,c1(C(N2CC(CC(=O)NCCC(=O)NCC)OCC2)=O)ccc2ccoc2c1 43777,c1(C(N2CCC(CC=C)(NC(=O)C(C)Cc3cccnc3)C2)=O)cc(F)ccc1N 43778,CC1=C(C)CC(C(=O)NCC2CC(F)CN2C(c2cscc2F)=O)CC1 43779,O=C(C1=CCCCC1)NCC(c1ccoc1)NC(=O)Cc1cccnc1 43780,S(=O)(=O)(c1ccc(N2CCn3nnc(CO)c3C2)c(C#N)c1)NC(CCC=C)C 43781,C1(C)(NC(CCNC(=O)NC)=O)CCC(NC(c2ccc(F)c(Cl)n2)=O)CC1 43782,C=CC(C)CC(=O)NC1CC(CNC(c2ccsc2-n2cnnn2)=O)C1 43783,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 43784,n1(CC(=O)NC2CC(CNC(c3cnc(C(C)=O)s3)=O)C2)nc(C)n(CC)c1=O 43785,C1(NC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1CO 43786,c1(CN2CCC(c3[nH]nc(C(C)(C)C)n3)CC2)cnn2c1CCC2 43787,C1(C(=O)NC(CCSC)C(=O)N(C2(C)CC2)C)CN(C)CC(C)O1.N(C)C 43788,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCOC(C)C)C2)C(=O)C1 43789,C1(C(=O)NC(C(CC)C)CO)CCC2(CC2)N1C(c1cncc(NC)c1)=O 43790,c1(OC)nn(C)cc1C(=O)NC1CCC(CNC(=O)C(C)n2ccnc2)CC1 43791,C(=O)(C(C)C(C)NC(c1c[nH]nc1CNC(=O)CCOC(C)=O)=O)NC 43792,N1(C(C(CC=C)OC)=O)CCC2(CCC(NC(=O)Cc3ccccc3C)CC2)C1 43793,c1(NC(C2(CC)CN(C(C(CC)CC)=O)C2)=O)ccc(F)cc1SC 43794,c1(OC)cccc(C(c2cn(C)nc2C(F)(F)F)N(C=O)CC2(F)CCCC2)c1 43795,c1(C(=O)NC(C)CCNC(=O)C(O)c2cnc[nH]2)ccc(Cl)o1 43796,c1(C(=O)NCCCNC(c2ccn(C(CC)CC)n2)=O)cc(C)nn1CC 43797,N1(C(C(CCC#C)O)=O)Cc2ccccc2C(NC(=O)Cc2ccc(C)o2)C1 43798,c1(CC(N2CCC(O)(CCNC(CSCCOC)=O)C2)=O)cccc(C#N)c1 43799,c1(NC(c2n(CCCOC)nnn2)(COC)C2CC2)ccc2nncn2c1 43800,c1(C(N(CCN(C(CCC(C)c2ccccc2)=O)C)C)=O)cnc2[nH]cnc2c1 43801,C(=O)(C1=C(Cl)CCOC1)N1C(CN(C(c2c(OC)cc(F)cc2)=O)C)CCC1 43802,C1(C(N2CC(CNC(c3cn(CC=C)nc3)=O)C(O)C2)=O)CC=C(C(C)C)CC1 43803,N1(C(C(CCC)(C)C)=O)CCC2(CCN(C(=O)CC3CCC(=O)NC3=O)C2)C1 43804,N1(C(CC=C)=O)CCC(C(=O)N2CC3(C)CCC3(C)C2)=C(F)C1 43805,C(=O)(CC(C)CC(C)(C)C)OS(c1cc(N(C2CCS(=O)(=O)C2)CC)ncc1)(=O)=O 43806,C1(c2cn(CCC(=O)N(CC)Cc3ccncn3)nn2)C2CCCCC12 43807,Cc1nc(C(C)C)ccc1C(=O)NCC(O)CCNC(c1cc(F)ccc1N)=O 43808,CC1CCN(C(=O)C2=CCCCC2)CC1CNC(=O)C=Cc1ccoc1 43809,Cc1cc(N(CCCN=[N+]=[N-])C)ccc1S(=O)(=O)N(C)C 43810,C#CCC(C)(C)C(=O)N(C)CC=CC(=O)NCCCc1ncnn1C 43811,N1(C(c2c(C)occ2)=O)CCCC(CNC(=O)C(c2ccc(N(C)C)cc2)C)C1 43812,c1(NCC(CNC(=O)CON2CCCC2)OC)nnnn1C(C)(C)C 43813,c1(C(c2nnnn2CCCF)(C)NCC=Cc2ccco2)nnc2n1CCCC2 43814,c1(C(N2C(CNC(C)=O)CCCCC2)=O)cc2ccc(C)n2c(C)n1 43815,n1(CC)c2ccccc2c2cc(C(N3CC(C)C3(C)C)=O)ccc12 43816,Cn1ncc2nc(Cl)nc(N3CC(C)CCC3NC(=O)CC(C)(C)C(F)F)c12 43817,C1(O)(NC(COC2CN(C(c3c(C)c(N)ccc3)=O)C2)=O)CCCC(C)(C)C1 43818,C1(N=c2cc(-c3n(C(C)C)nnn3)n(C)[nH]2)(Sc2cccc(Cl)c2)CCOC1 43819,c1(C(=O)NCCSC)cc2cc(-c3cn(C)nc3C)ccc2oc1=O 43820,C1(NC(CCc2cccc(NC(C)=O)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C1 43821,C(=O)(C(C)C(=O)N1CCN(CCNC(=O)C(C)(C)C2CCCO2)CC1)OC 43822,c1(C(=O)NCCC2N(C(c3c(C)con3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 43823,C1(C)(C(=O)NCCCN2CCN(C(C(C)SC)=O)CC2)C(C)(C)C1(C)C 43824,C1(C(N(C(C)C)CCc2ccco2)=O)CCN(C2CCOC2C)CC1 43825,c1(C(=O)NC(C2(O)CCN(C(c3nc(C)oc3)=O)C2)C)[nH]nc2ncnc(O)c12 43826,c1(C(=O)NC(CCOC)C(=O)NCC2CCC(O)CC2)cccc2[nH]ccc12 43827,CC1(C)CC(=O)NCC1C(=O)NCCNC(=O)CCCc1cccnc1 43828,c1(CC(=O)NC(CC=C)CNC(=O)CCCNC(N)=O)ccc(Cl)c(OC)c1 43829,C1(NC(C2CC(O)(CC#C)C2)=O)CCCN(C(c2cccnc2CC)=O)C1C 43830,c1(C(=O)NC(C2CCN(C(=O)CCNC(=O)C3CC3)CC2)C)ncc(F)cc1C 43831,c1(C(=O)NCC(CC)NC(C2CNC(=O)C2)=O)cc(C2CC2)cs1 43832,C(=O)(CC1=CCOCC1)NC1CCCC(C(=O)NOC2CCCCCCC2O)CC1 43833,N1(C(c2ncc[nH]2)=O)CCC(C2CCCN(c3nccn4nnnc34)C2)CC1 43834,C#CC1CC(CONC(=O)C2CC2(F)F)C1 43835,C#CC1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(c2cc(OC)ccn2)=O)C1 43836,c1(COC)ccncc1NC(C1COC(CNC(=O)Cn2cccn2)C1)=O 43837,N1(C(CC2(C)CC2)=O)CCC2C1CCCN2C(=O)C=CCCCc1ccco1 43838,c1(CCn2cc(-c3cccc(SC)c3)nn2)cccc2c1CN(CC(F)(F)F)C2 43839,c1(C(C(=O)NC)N(C)CC2CC2(F)F)ccc(C2CCOCC2)cc1 43840,CCN=c1ccc(C(=O)NC(C)CC2CN(C(c3nnsc3C)=O)C2)c[nH]1 43841,C1(C)(N(C)CC)CCN(c2ncc(OC(C)C)cn2)C1.C(=O)(CC=C(Cl)Cl)N 43842,C1(C(N2CCCC(C(C)(O)CNC(=O)CC3CC3)C2)=O)CCOC2(CCC2)C1 43843,C(=O)(C1CCc2nccn21)N(CCC1CCN(C(C2CC(C)(CC)C2)=O)CC1)C 43844,C1(NC(C(CC)C(C)O)=O)CN(C(=O)CC(c2ccc(F)cc2)C)CCC12CCC2 43845,N1(CC#CC(=O)NCC2CCC3(CC3)C2)CCOC2C(O)CC12 43846,C(c1cccc(CO)c1)=CC(N1CCC(C)(NC(=O)CCCc2ncco2)C1)=O 43847,N1(C(c2c(CC)oc(C)c2)=O)CCC2(C1)CN(C(=O)CC1CC=CCC1)CCO2 43848,c1(C)noc(CNC(C2CC2C(=O)OC(C2(O)CN(OC)C2)C)=O)n1 43849,c1(C(N(CCNC(=O)CCC2CCC(=O)N2)CC)=O)cc(C(F)(F)F)nn1C 43850,C1(C(N(CC#CC)C)=O)CN(C(=O)Cc2scnc2C)CCO1 43851,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 43852,C(=O)(CCCn1ccnc1)NCC1(C(=O)NCC(=O)NCc2cnn[nH]2)CCC1 43853,CC1CC(C)N(C(c2oc(S(N)(=O)=O)cc2C)=O)CCN1C(=O)CCF 43854,C1(=O)CCCCCCN1.C1(N(C)C)CCCN(CCN2CCCC2=O)C1 43855,n1(C2CN(C(C(N(C(C=CC(=O)OCC)=O)C)SC3CC3)=O)C2)cc(C)cn1 43856,Cc1cc2ncnc(N3CCC4(CCN(C(c5conc5C)=O)C4)C3)c2[nH]1 43857,C12(C(=O)NC3(CO)CN(c4cc(N)ncn4)C3)CCCCC(=O)N1CCC2 43858,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 43859,c1(C(=O)NC2C(CNC(=O)C3=CCCCC3)CC2)ccc2oc(=O)oc2c1 43860,C1(n2cc(CN(C)C(c3cccc(F)c3)=O)nn2)CCCC(F)(F)C1 43861,c1(C(N2C(C)(C(=O)OCC)CCC2)=O)ncnc(CC2CCCCC2)c1C 43862,n1(C(C)C)cc2ncc(C(N3CCC(NC(=O)C(C)CF)CC3C)=O)cc2n1.C(=O)O 43863,N1(C(C(C)C2CC2)=O)CCC2CCC(C1)N2C(c1cc2c(o1)CCCNC2=O)=O 43864,C=Cc1ccc(C(=O)NC(CCNC(c2cnc(OC)nc2)=O)C(C)(C)C)cc1 43865,c1(C(N2C(CNC(C(CC)C#N)=O)CCCC2)=O)sc2ccc(F)cc2c1C 43866,N1(C(C(C)C)=O)CCCC1CCCNC(=O)COC1CCN(C(=O)C2CC2)C1 43867,C1(C(=O)NC(CC=C)C(=O)NC(CCO)C2CCC2)CC2(CCO1)CC2 43868,CC1CCn2c(C(=O)NCC3CC(F)CN3C(=O)CN3CC(C)(C)C3)cnc2C1 43869,N1(C(C(C(C)C)C)C(=O)NCc2ccccc2Br)CCn2ncc(CN(C)C)c2C1 43870,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 43871,C1(OCC)(CNC(C2CCCN(C(C3CCS(=O)CC3)=O)C2)=O)CCCCC1 43872,N1(C(C2(N(CC(F)(F)F)C)CCS(=O)(=O)C2)=O)CCCC2CN(CCF)CCC12 43873,CCC(C)(CNC(=O)CSC(F)(F)F)NC(C1(O)CCOC1)=O 43874,C(CC(C)C(=O)N1CCCC(N(C(=O)CC2(OC)CCC2)C)C1)=CC 43875,C12(NC(CCSC)=O)CCOCC1CN(C(=O)Cc1cc(C(C)(C)C)c[nH]1)C2 43876,c1(C(=O)NCCCN(C(=O)CCOCC(F)F)C)ccc(-c2nc[nH]n2)nc1 43877,C(=O)(C(O)C(C)(C)C)N(CC(C)O)CCNC(C1CC(O)(CC#C)C1)=O 43878,N1(C(C2CN(C(CCS(C)(=O)=O)=O)CC2(F)F)=O)CCC(O)CC(O)C1 43879,c1(C(N2CCC(C)(C(=O)NC(CC)C3CC3)C2)=O)c(C)nn(C)c1C 43880,c12ccc3c(c1)C(NC2)CCO3.C1(NC(=O)OC(C)(C)C)CC(CO)CO1 43881,c1(C(=O)NCC2COCCN2C(=O)COC2CC2)ccc2c(n1)CCOC2 43882,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 43883,N1(C(c2scc(C)c2)=O)CCC(F)(OCC(N2CC(CC(F)(F)F)C2)=O)C1 43884,C1(CNC(C2(OC)CCCC2)=O)CC(NC(c2cncn2C)=O)CC1O 43885,C1(NC(c2n(C(C)C)ncn2)=O)CCCC(NC(c2cn(C)[nH]c2=N)=O)C1 43886,N1(C(C(=O)NC)C(C)CC2CCC2)CCc2sc(C)nc2C1 43887,C(=O)(C(C(C)(C)C)NC(C1(C)CC(=O)N(C)C1)=O)N(CCOCC#C)C 43888,C(=O)(C(C(C)(C)C)C1CCCCC1)N1CCC(NC(c2cn(C)cn2)C)C1 43889,c1(CNC(C(C)N(C)C)=O)ccoc1C(N1CC(c2nncn2C)C1)=O 43890,C(=O)(C(O)CC(C)C)NCC1C(C(N2CC(CC)(Cn3ccnc3)C2)=O)OCC1 43891,N1(CC(=O)NC2C(NC(C(C)NC(COC)=O)=O)C2)C(=O)C2CCCCC2C1=O 43892,C1(NC(C(C)=C2CC2)=O)CCCC12CN(C(C1CC3COC(C)CON13)=O)C2 43893,O(NC(=O)CCCCCNC(=O)C(C)CCCOC)CC(=C)Cl 43894,CCC(C)(O)C(=O)NC1CC(n2ccc(C3CC3)n2)C1.N12CCN(CC1)C(=O)C2 43895,c1(NC(C2N(Cc3c(OC)ccc(CO)c3)C3C(C2)C3)=O)nc2ccccc2[nH]1 43896,C1(O)(CNC(C(C)OCCC#C)=O)CCCN(C(=O)C(Cl)=CCl)CC1 43897,c1(C(=O)OCC)cc(F)c(C(=O)NC(C(C)NC(=O)C=C(C)C)C(C)C)cc1F 43898,C1(NC(c2n(C)cc(Cl)c2)=O)CC2CN(C(c3ccc(S(N)(=O)=O)o3)=O)CC2C1 43899,C1(C(=O)NC2C(NC(Cn3ccc(C)n3)=O)COC2)CCC(O)CN1C 43900,c1(C(=O)NCC2N(C(C(C)OCCC=C)=O)CCCC2C)ccc2occc2c1 43901,C1(NC(CC(C)(C)O)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 43902,C12(NC(C(C)=C3CCC3)=O)CCCC(CN(C(c3ccc4ccoc4c3)=O)C1)C2 43903,c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cc(C)c(Br)o1 43904,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 43905,CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CCOC2C)CC1)C1CC1 43906,N1(C(c2c(C)con2)=O)CC(CNC(=O)CCC2CCCN2C=O)CC1C 43907,C(=O)(CCCC(=O)NC1CCC(F)(CNC(=O)CCCCCOC)C1)NC 43908,c1(C(N(CCCNC(C2N(C(CCC)=O)CCCC2)=O)C)=O)c(C)cn(C)c1C 43909,C(=O)(C1=CCC(C)CC1)NCC1N(C(C2(COC)C=CCC2)=O)CCC1 43910,C(=O)(CCCCC(F)(F)F)NCC1CCN(C(C(CC)C(C)C)=O)C1(C)C 43911,N1(C(c2nccs2)=O)CC2CN(C(=O)C3CC3)CC2C1.c1ccccc1I 43912,CC12CCC(CC(=O)NCC3(C)CCC(NC(=O)C=Cc4ccsc4)C3)(CO1)C2 43913,N1(C(C2=C(C)CC2)=O)CC2(CC(NC(=O)C(c3ccnn3C)O)CO2)C1 43914,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)CN(C)C)C 43915,C(C)(CCC(=O)OC)N(CC(F)(F)F)C.C1C(=O)N1CCNC(=O)C=C(C)Cl.CS 43916,CN1CCOCC1CC(=O)NCCn1cc(C(=O)N(C2CCC2)C2CC2)cn1 43917,C1(NC(C(CCC)c2ccccc2)=O)CN(C(c2ccc(F)cc2)C)CCC1C 43918,c1(C(=O)NCCCCN(C)C(C2CCCO2)=O)cn2ccnc2s1 43919,N1(C(CCCCCSC)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 43920,N1(C(c2cc(Cl)ccn2)C(=O)NCC=C)CCOC2(CCSC2)C1 43921,C1(NC(C2(COC)CC=CC2)=O)CCN(C(=O)C(C)C2CCOC2)CC1C 43922,C(=O)(C#CC(C)(C)O)N1C(CNC(C2CCCN(C(C)C)C2)=O)CC(COC)C1 43923,c1(C=O)ccn2cncc2c1.CC(CN1CCC1)NC(=O)C=CCC1CC1 43924,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 43925,c1(OCC)ncc(C(=O)NC2CCC(NC(C3CC3C#N)=O)CC2)cn1 43926,C(=O)(C(F)CC(C)(C)SC(C)(C)C)NCCN(c1cnn(C)c1CCCO)C.C1CO1 43927,c1(C(=O)NCc2ccccn2)cc([N+](=O)[O-])n[nH]1.C12CCC(O1)CNC2=O 43928,c1(OC)cc(O)c(C(N2CCC(F)(C(=O)Nc3cn[nH]c3)CC2)=O)c(Br)c1 43929,N12CCCC(C1)C(=O)OC(=O)N1CC(C1)C2=O.C1(COCC)(C)CC12CCC2.OC 43930,C1(C(N2CCOC(C)(CNC(=O)CNC(N)=O)C2)=O)(CC)CCCNS1(=O)=O 43931,N1(C(C=NOC)=O)CCCC2(CC(NC(=O)CC3CN4CCC3CC4)C2)C1 43932,c1(SC)ccc(NC(C2CC2CNC(C2(C)CCOC2)=O)=O)cc1 43933,N1(C(C2C(OC)C2)=O)CCC(NC(C2CN(CC(C)C)C2)=O)C1(C)C 43934,N1(C(c2c(Cl)cnc(CC)n2)=O)CC2CCCC2(NC(=O)Cc2c[nH]nc2C)C1 43935,C1(NC(CCNC(=O)CO)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 43936,CC(C)C(C)C(C)CC(=O)NCC1(C)CCCN1C(c1nccc(Cl)c1F)=O 43937,N1(C(C(CC)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc(N(C)C)nc1)=O)C3 43938,C(=O)(C(CC)N(C)C)N1CC(C)(CCC(=O)NC(c2cscn2)C)C1 43939,N1(C(c2ccc(CCC=C)cc2)=O)CC2CC(NC(c3snc(C)c3N)=O)C1C2 43940,Cc1nc2ccc(C(=O)NC3CC(NC(c4cc([N+](=O)[O-])cn4C)=O)C3)cn2n1 43941,c1(NC(c2nnnn2CCSc2ccccc2)C2(C(N)=O)CC2)ccc(Cl)cc1F 43942,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 43943,C(=O)(CC(O)CCCCC)NCC(CC=C)NC(=O)CN1CCN(C)C1=O 43944,c1(OC)cc(N)c(Cl)cc1C(N1CC(C)(NC(C23CSC(C2)C3)=O)C1)=O 43945,c1(C(=O)NC(CNC(C2(CCC)CCC2)=O)C)cc(C)c(Br)c(C)c1 43946,N1(C(C(CC)NC(C)=O)=O)CC(CNC(C2CCC(=O)N(C)C2)=O)CC(C)C1 43947,N1(C(CN2CCN(C(C(CCC)F)=O)CC2)=O)CCC(O)C(F)C1 43948,c1(C(N2CCCC(N(C(C(CC=CC)C)=O)C)CC2)=O)cc2nc(C)sc2[nH]1 43949,C(C(O)C(=O)O)NC1CCN(C2C(C(C)(C)C)C2)C1.C1CC1 43950,c1(C(=O)NCCOCCNC(c2cncc(N)c2)=O)cc2cc(Cl)cnc2o1 43951,N1(C(c2n(C)cc(NC(=O)COC3CCOCC3)n2)=O)CCC(CO)C(C)(C)C1 43952,c1(C(N(CCCNC(c2c(C)snn2)=O)C2CC2)=O)cncc(N)c1 43953,Cc1cccc(Br)c1-n1cc(C(C)N(C(=O)C(=O)OC(=N)O)C)nn1 43954,c1(CC(=O)NCCC2CCN(C(C(C)C3CC3)=O)CC2)cn(C)c2ccccc12 43955,c1(NC(C2C(NC(CN3CCC(C)C3)=O)C2(C)C)=O)cncc(CO)c1 43956,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 43957,CC(C)C(C(=O)NC1CCCC1NC(C1CCCN(C)C1)=O)n1cncn1 43958,C(C)(CCC(=O)N(CC(O)CNC(=O)CSc1nncs1)C)NC(C)=O 43959,c1(C(N2C(c3c(OC)cc(Cl)cc3)CCC2)C(=O)NC)cn2cc(F)ccc2n1 43960,C1(NC(c2cnc(OCC)s2)=O)C2CCN(C(=O)CSc3nncn3C)CCC12 43961,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 43962,N1(C(C(C)NC(C)=O)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 43963,c1(NC(C(N2CC(NC(=O)CC3(CO)COC3)(CO)C2)=O)=O)ccc(O)cc1 43964,c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(C)C2CCC2)C)ccc(CC)cn1 43965,N1(C(c2c(CNC(CNC(C(N)=O)=O)=O)occ2)=O)CCC(O)(CO)C1 43966,C1(CC)CCC(C)N(C(=O)CCOCCN(C)C(c2nnc(S)n2C)=O)C1 43967,N1CCN(C(=O)Cc2cncc(Br)c2)C(C2CC2)C1.c1(COC)cc(OC)ncn1 43968,C1(C(=O)NCCC#C)CCN(C(=O)c2cccc(Cl)c2)O1 43969,CC1COCCCN1N1CCN(Cc2ccc(Cl)cc2)CC1 43970,C1(C)(C(=O)NC(CCC)CO)CN(C(=O)CC2(C)CCC2)CC1C 43971,c1(SC)cc(C)c(C)nc1C1CCN(c2nnc3n2C3)CC1.C1(CO)CCCCO1 43972,Cc1nc2[nH]c(C(N3CCC4(NC(c5cnc(S)[nH]5)=O)CC4C3)=O)cc2s1 43973,C1(C(=O)NCC(C(C)O)O)CC2CCC1N2C(C1(C)CC=CCC1)=O 43974,CC1(CC(=O)NCC2CCN(C(=O)C(O)COCc3ccccc3)C2)CCOC1 43975,CC(C)(CO)CCCNC(C1CCC(C)N1C(C1COC(=O)N1)=O)=O 43976,C12(C(=O)NCC(C)N(C(C3(c4cccc(C)c4)CCC3)=O)C)CCC(F)(CC1)C2 43977,C1(Cc2cn(CCC)nn2)CN(C(C2CCCC2c2ccccc2)=O)CCO1 43978,c1(NC(=O)NC(c2ccccc2F)C=C)cccc2cncc(C)c12 43979,CCCCCC(CC)C(=O)NCC1(CNC(=O)C(n2nccc2C)C)CCCC1 43980,Cc1cc(CC(=O)N(CCCCN(C(=O)C(C)(C)OC(C)=O)C)C)n(C)n1 43981,c1(C(=O)NC(CN(C(=O)C(C)(O)CC)CC)C)ccccc1S(=O)(=O)C(F)F 43982,C(C(=O)NC12CC(CNC(=O)CSC(F)F)(C1)C2)(c1ccccc1)=C(C)C 43983,Nc1cccc(F)c1C(=O)NCC1CCN1C(C1CC1c1ccncc1)=O 43984,C(=O)(CCCC(C)(C)C)N1CC(CC)C(NC(c2cccc(NC(C)=O)c2)=O)C1 43985,CC(C(C(=O)NC1CC1)N1CCN(c2ccncc2Cl)CC1)C(C)(C)C 43986,c1(OC)cc(Cl)ccc1CNC1CC1C(N1CCC2(CCO2)C1)=O 43987,C1(CNC(=O)CNC(=O)C2CC2)CCCC1CNC(C1CSCCS1)=O 43988,N1(C(C(C(C)(C)C)N(C)C)=O)CCC2(CC1)CC2CNC(c1cc(N)ccn1)=O 43989,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 43990,C(=O)(C1COc2ccccc21)N(C1CCCN(C(=O)CSC2CC2)CC1)C 43991,N1(C(c2c(CCC)cccc2)=O)CCC2(CC(NC(=O)CCC(C)(F)F)C2)C1 43992,C1(CC)CN(C(c2ncc(Br)cn2)=O)CCC1NC(C1CCC(=O)N1)=O 43993,c1(C(=O)NC(CC)CNC(=O)CCS(N)(=O)=O)cnc(COC(C)(C)C)nc1O 43994,n1(CC#C)c(C(=O)OCC(=O)Nc2nccc(Br)c2Cl)cc2ccccc12 43995,N1(C(c2cnc(CC(C)C)s2)=O)CCCC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1 43996,c1(OC)cncc(C(=O)NCCC2CN(C(=O)CSCc3cccs3)CC2O)n1 43997,c1(C(=O)NCCCC(C)NC(C2(C)CC(C)C2)=O)cccc2c1COCCN2 43998,C(C(C)C)(C(O)C(=O)OCc1c(C)nsc1Br)OC 43999,N1(C(C2CCCN(S(CC)(=O)=O)C2)=O)CCCC2CN(C(=O)C(O)C3CC3)CC12 44000,c1(C(N2CC(CNC(C3(CC=C)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44001,O(N(C)C(=O)C(C1(O)CCCCC1)NCC)CC.C(C(C)CC)=CC(=O)C(=O)C=C 44002,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44003,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44004,C1(C)(C(=O)NCC2(CNC(C(C(C)C)C3CCC3)=O)CCCC2)CCCCCC1 44005,N#Cc1ccc(NC(=O)C(F)CC2CN(C(c3cnc4n3CCC4)=O)C2)cc1 44006,c1(C(N2CCC(n3cnnn3)C2)C(=O)NCCCOC)cccc2c1OCO2 44007,c1(N(C(CC(n2c(C(C)C)ncc2)C)=O)CC2CC2)ccc(F)cc1 44008,C(C)(C)(CCC(=O)N(C(C(=O)NCC1C=CCOC1)C1CC1)C)OC 44009,C1(CC(N2CCC(CN(C(CC3CN(C(C)=O)C3)=O)C3CC3)C2)=O)CCN(C)C1=O 44010,N1(C(C(=O)NCC(C)C)C2CC2(C)C)CCn2ncc(-c3cc[nH]n3)c2C1 44011,C(=O)(C(C)(O)Cn1ccccc1=O)N1CCC(C(c2ncc(O)cn2)C)CC1.N 44012,N1(C(CS(=O)(=O)NC)=O)CC2CC1CCC2NC(c1ccc(C2CCCCO2)o1)=O 44013,c1(CN(CC)CC2CC2C(=O)O)ccc(O)cc1 44014,CN1CCOCC1C(=O)NCCCNC(c1ocnc1C(F)(F)F)=O 44015,C12(CC)COC(C(=O)NC3CC(NC(c4c(C)coc4C4CC4)=O)CC3O)(C1)C2 44016,C1(CC(=O)N(CCONC(C2CCC(O)C2O)=O)C2CC2)CCS(=O)(=O)CC1 44017,C1(CC(=O)NCCc2cc(C(=O)NCc3ccc(C)o3)no2)CCCCC1C 44018,N1(C(C(F)OC)=O)CC(CNC(=O)Cc2cc(C)on2)CC(C)C1 44019,C#CCC(C)(C)CNC(C(=O)OC(C)(C)C)C1CCC1.C1(=O)C2=CC(C2)N1 44020,c1(N(C)CCn2cc(C3COCCOC3)nn2)ccc(F)cc1.C12CCCN1C2 44021,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(c3cccc(N)c3)=O)C2C1 44022,C1(C(=O)NCCC2CC(NC(CC(=O)OCC)=O)C2)CS(=O)(=O)CC12CC2 44023,C(=O)(CC(C)CF)N(CCCNC(CCN(CCOCCOC)C)=O)C1CC1 44024,C(=O)(N=c1c(Br)c[nH]cc1I)C1CCC(C(C)NC(c2ccc(F)cc2)=O)CC1 44025,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44026,c1(CC(=O)NCC2(O)CN(C(c3c[nH]nc3C3CCCO3)=O)C2)ccccc1 44027,N1(C(CC2CC(=O)C2)=O)CCC2CCC(C1)N2C(=O)CC1CCC2CC12 44028,O=C1CCc2ccc(OC(=O)COc3cccc(Br)c3)cc21 44029,c1(C(=O)NC(c2cn(-c3ccc(C)o3)nn2)CCC)ccnn1C(C)C 44030,C1(CCNC(Cc2ccn(CC)n2)=O)CCCCN1C(C1CCCN1C)=O 44031,C1(CN(CCn2nccc2C(=O)OC)CC)CCN(C(=O)Cn2cccn2)CC1 44032,C1(CNC(C(C(C)(C)C)O)=O)CN(C(C2CN3CCC2C3)=O)CC12CCOCC2 44033,C(=O)(C(CCC1CCC1)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)COC 44034,C1(NC(c2ccn3nccc3c2)=O)CN(C(=O)CC2CC2(Cl)Cl)CC2(CC2)C1 44035,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)C(NC(C2CC23CCC3)=O)C1 44036,c1(C(C)C)cc(C(N2CCC(F)(C(=O)Nc3cc(C(C)(C)C)n[nH]3)C2)=O)n(C)n1 44037,c1(OC)cc(C)c(C(N2CC=CC(NC(c3c(Cl)noc3C)=O)C2)=O)cc1Cl 44038,N1(C(=O)NC2C(SCC)C2(F)F)CCN(c2cc(C(N)=O)ccn2)CC1 44039,N1(C(c2c(C)cccc2)=O)CC2CCCC(C1)N2C(=O)COC1CCCCC1 44040,c1(C(=O)NC(C(=O)N(CC(C(=O)NC)C)C)CCF)cc(OC)cc(C)c1 44041,N1(CCC2C(C)(C)C2)CC(O)(CNC(c2cc(CO)on2)=O)C1 44042,N1(C(c2c(CC)ocn2)=O)CCCC(NC(=O)CCc2cnn(C)n2)C(F)C1 44043,C(CO)(C(=O)N(C)CCNC(C1(c2ccncc2)CCCC1)=O)NC(C(C)C)=O 44044,c1(C(=O)NCC2(F)CC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44045,N#CC1CCCC(CC(=O)NCC2(NC(=O)Cn3cnc(C(F)(F)F)n3)CC2)C1 44046,C12(NC(C3C4CCN(C(C(N5CCCCC5=O)C)=O)CC43)=O)CCC(O)(CC1)CC2 44047,c1(SCn2cc(C(c3cccc(C)c3)CCC)nn2)c(F)cc(C#N)cc1[N+](=O)[O-] 44048,C1(C(N(C2(C(F)(F)F)CC2)C(C)C)=O)CC(C)CN1Cc1ccco1 44049,C1(CNC(c2cc(OC)no2)=O)CCC2(CO1)CC(NC(=O)C(C)CSC)C2 44050,Cc1ccc(NC(C2CC2NC(c2ccc(F)cc2F)=O)=O)cc1Br 44051,CN1CCN(C(=O)CC2(O)CCCCC2)CC1C(=O)NCc1cncnc1 44052,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cc2cncs2)C2(CCC2)C1)=O 44053,c1(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)cc(Cc2ccccc2)c[nH]1 44054,C(C(=O)NC(CCC1CCC1)C(=O)NCC1C=CCCC1)(C(C)C)OCC 44055,c1(Oc2c(-c3nc(C(CC)CSC)n(OC(C)C)n3)nccn2)ccc(F)c(Cl)c1 44056,C=CCN=C(NCCC1CSC1)N1CCC(C)(c2cccc(Cl)c2)C1.OC 44057,C=C1CCCN(C(=O)CCC(C)NC(=O)CC2(O)CCOCC2)C1 44058,c1(C(N(C(CNC(C(C2CCOC2)OC)=O)C)C)=O)cnc(C(C)(C)C)[nH]1 44059,c1(NCC(N)=O)[nH]c(=NCC2CC=CCC2)nc2scnc12 44060,Cc1ccc(CN2CCC(NC(C3(C4CC4)CC3)=O)C2)nc1Br 44061,C#CCC(O)C(=O)N1CCCC1C(C)NC(C1(COC)CC1)=O 44062,CCC(C)(COC)C(=O)NCCC(C)N(C(=O)C1=COCCC1)C 44063,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44064,N1(C(C2C(C(C)NC(c3c(NC)cncc3)=O)C2)=O)CCC(O)C(C)(O)C1 44065,c1(Cn2cc(C3N(C(CC(CN(C)C)O)=O)CCC3C)nn2)cccc(C)c1Br 44066,O(NC(=O)C(C(CC)CC)NC(=O)CC(=O)NCC1CCCC1)CCCC 44067,N1(C(C2CCN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CCc2n[nH]cc2C1 44068,CC1CN2CC1CNC(=O)OCC2=O.c1(CC(=O)OC(C)(C)C)csc(S)n1 44069,C1(CC)CN(C(CCc2ccco2)C(=O)NCC2CCOC2)CC1O 44070,C(C(=O)NCC(O)CCNC(=O)CCc1cccs1)(C(C)O)NC(C)=O 44071,c1(C(=O)NC2CCCC(NC(CN3CC(C)C3)=O)C2)cnn(C)c1C#N 44072,C(=O)(CC(C)(C)CN(C)C)NC(C(=O)N(C(CCC(C)C)C)C)C1(C)CC1 44073,CC1(C)C(C(=O)NCCCCCO)CCN1C(=O)C(O)CN1CCCC1 44074,Cc1nc(N)n(CCC(=O)NC(C)CN2CCN(C(=O)Cc3ccon3)CC2)n1 44075,CCC1C(=O)ON1C.C1(NC(=O)N(CCCCO)C)CCCCO1 44076,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(CC(CC)SC)=O)C(CC2CC2)CC1 44077,C1(C(=O)NCCNC(CC2CC(COC)C2)=O)CC(=O)N(Cc2ccccc2)C1 44078,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(c2cc(F)cs2)=O)CC1 44079,C1(C(N2CCC(N(C(c3ccn(CC)n3)=O)CC)C2)=O)CC12CC(C)(C)C2 44080,C1(NC(C(C=C)C)=O)CN(C(c2cnn3c2OCC3)=O)C2CCCC12 44081,C(=O)(CCCCC(N)=O)NCC1(CNC(C2CC3(CC(=C)C3)C2)=O)CC12CCC2 44082,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(C3(C)CCN(C)CC3)=O)CC2C1 44083,C1(NC(C2CC(N(C)C)C2)=O)COCCC1NC(c1nc(Cl)sc1Cl)=O 44084,C(C1c2ccsc2CCN1C(=O)Cc1nnc(S)n1C)NC(C(C)(CO)OC)=O 44085,N1(C(C(C(=O)OCC)OC)=O)CCN(C(=O)CC(CC)C(C)C)CC2(CC2)C1 44086,CC(C)C(CN(CCCO)CCO)C(=O)NC1CCC(F)CC1 44087,C1(C(N(C(C)C)N(C2CN(C(=O)CSC3CC3)C2)C)=O)CCOC(=O)CC1 44088,c1(C(N2CCC(CSc3ccccc3)C2)C(=O)NC(C)C)ccn2nccc2c1 44089,c1(C(CC)C(=O)NN2CCCC(N3CCCC3=O)C2)ccc(Cl)c(F)c1 44090,C#CC1CCC(c2nnnn2CC(F)F)(Nc2cccc(O)c2)CC1 44091,O=C(C1=CCCN(Cc2nc(C)ccc2C(F)(F)F)C1)Nc1ccc(Cl)nc1Cl 44092,CC1CC(NC(C2CC(O)C2)=O)CN(C(=O)C(C)(O)c2ccccn2)C1 44093,c1(C(N(CC(=O)NC(C(C)C)c2nc[nH]n2)C)=O)ns[nH]c1=O 44094,c1(OC)ccc(C(=O)NCC(CO)NC(c2c[nH]ccc2=N)=O)c(C)c1 44095,N1(Cc2cccc(N(C)C)c2F)CC(N=c2ccn3ncc(I)c3[nH]2)C1 44096,C(=O)CN=c1cc[nH]cc1.C12CN(CC(C)(C)O1)C(=O)C2=O.CO 44097,C1(CNC(C(CC)F)=O)CC2(CCN(C(c3c[nH]cc3CC)=O)CC2)C1 44098,c1(C(=O)NCC23CCOCC2C3)cc2cccc(Br)c2[nH]1 44099,N1(C(C(C)OC)=O)CCN(CCNC(C2CCN(C(c3cnn(C)n3)=O)C2)=O)CC1 44100,C1(NC(c2c(C)[nH]nc2C(F)F)=O)CN(C(=O)CN2CCCC2)CCC1CO 44101,Cc1nc2cccc(Cl)c2s1.O=C1CN(CCC2CCCC2(F)F)C(=O)N1CC 44102,c1(OC)ccccc1C(C1CC1)NC(=O)C(=O)NC1CCCCC1 44103,c1(C(N2CC(C)(CCC(N3CCC(O)(C(C)C)C3)=O)C2)=O)nc(O)nc(O)c1N 44104,c1(C(N2CC(CNC(c3n(CC)ccc3)=O)(OC)C2)=O)ccc2cnccc2n1 44105,CC1=NNC(=O)C1CC(N1CCOC(CCNC(=O)C(C2CC2)C2CC2)C1)=O 44106,C1(CC(=O)NC2CC23CC(NC(C2(CO)CCC2)=O)C3)Cc2cccc(Cl)c2O1 44107,C1(CNC(CCSCCCOCC)=O)CN(C(=O)Cc2nc[nH]n2)C2CCN1C2 44108,CCCC(O)C(CO)NC(=O)C(C1CC=CCC1)NC(c1ncncc1N)=O 44109,c1(CC)ccc(OC)cc1C(N1CCCC1CCCNC(C1CC(C)(C)C1)=O)=O 44110,C1(C(N2CC(C(=O)OCC)C2)C(=O)NC)CCC(CNC2CCC3(CC3)C2)CC1 44111,C12(CC(=O)NC3(CCCC)CCCC3)CCC(CC1)N(C(=O)C(C)C(=O)OC)C2 44112,C(CC1=CCN(C(=O)CC2CSCCO2)CC1)CC.c1(C2(C)CC2)cc(C(=O)N)[nH]n1 44113,C12(C(N3C(C)(C(=O)NCc4ccc(OCC#C)cc4)CC3)=O)CCC(C)(C1)OC2 44114,c1(NCc2c(C)noc2)[nH]c(=NCCn2ccnc2C)nc2ncn(C)c12 44115,N1(C(c2c(SCC)nccn2)=O)CCCC(n2cc(C3CC34CC4)nn2)CC1 44116,C=C(C)c1ccccc1NC(=O)CCC1CCN(C(=O)C=CCCOC)CC1 44117,C1(NC(C=CC(C)(C)NC(C(C(C)(C)C)OC)=O)=O)CCn2cncc2C1 44118,C1(C(N(C)C)=O)CCCN(C(=O)C(=O)NC2COCC2OC2CC2)C1 44119,c1(C(=O)NCC2CC(CNC(C3C(CCC)C3)=O)C2)cc2cccnc2s1 44120,CC1(CNC(=O)CCN2CCOCC2)CCCN1C(=O)CC1(CO)CC1 44121,C1(CN(C(C=CC=CC)=O)C)CN(C(c2ocnc2C2CCCO2)=O)CC12CC2 44122,c1(C(=O)NC2C(C)(C)CN(C(c3ccccc3Cl)=O)C2)cncc(N=[N+]=[N-])c1 44123,c1(C(C(=O)NC(CNC(C=CC(CC)C)=O)C)O)ccc(Cl)c(F)c1 44124,c1(C(=O)O)c(NC(c2cn(-c3ccc(C(F)(F)F)nc3)nn2)=O)ccc(Cl)c1Cl 44125,c1(C(N(C2CC3CC2CN3)Cc2c(OC)c(Br)ccc2)=O)coc2cccnc12 44126,C=CCC(C)(C)CC(=O)N1CCN(C(=O)Cc2cc(OC)no2)CC1CF 44127,C12(NC(C(C)OC)=O)CC(C)(C1)OC21CN(c2nncs2)C1 44128,c1(NC(C(C)C)CNC(C2CCCO2)=O)ncncc1I 44129,c1(CN2C(C(=O)Nc3c(C(=O)OCC)csc3C)CC2)cccc2c1OC(F)(F)O2 44130,N1(C(C(C)(C)n2cnnn2)=O)CC(OC)CC(C)C1.c1(CC(=O)OC)cc(C2CC2)no1 44131,C1(CCNC(c2nc(C)sc2)=O)CN(C(C2OCCC2(C)C)=O)CCS1(=O)=O 44132,C1(C)(CNC(C2(CCCC)CC2)=O)CCN1C(=O)OC(C)(C)C 44133,Cc1ccc2c(c1)CN(C(=O)C(=O)NCCC1CC3COCC13)CC(C)(C)C2 44134,C(C(O)C(=O)N(C)Cc1cn(CCc2ncccn2)nn1)OC 44135,Cc1cc(C)c(C(=O)NC(c2cn(-c3ccc(C4CC4)nc3)nn2)C)c(S)n1 44136,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3ccco3)[nH]2)=O)C1 44137,O(NC(=O)C(CC(F)(F)F)c1ccc(Cl)c(F)c1)CCCOCC(=O)OCC 44138,N1(C(C#CC2(CC)CC2)=O)CC(C)(CNC(=O)Cc2ccc(O)nc2)CC1(C)C 44139,c1(NC(C2C(C(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44140,N1(C(CCCNC(C)=O)=O)CCN(C(=O)Cc2ccc(Br)cc2)C(C)C1 44141,n1(CC(=C)C)nnnc1C(c1ccc(C2CC2)o1)NCCCc1nncs1 44142,CCCCCC(C)CC(=O)N1CCC(N(C(=O)C(O)C2CCCC2)CCC)CC1 44143,C=CCC(CNC(C1C2CCC(C2)C1C)=O)C(=O)NCCC(O)COC 44144,C1(c2cn(CC(C)NC(=O)CSS(C)(=O)=O)nn2)COC(C)(C)O1 44145,C1(CC)(NC(c2ccc(O)nn2)=O)CCCN(C(=O)Cc2ccc(O)cn2)C1 44146,Cn1cc([N+](=O)[O-])c(C(=O)NCC2(F)CCN(C(=O)CN3CSCC3=O)C2)n1 44147,c1(CC)oc(C(N2CC(CC(=O)N(CC(C)C(=O)OC)C)C(C)C2)=O)cc1C 44148,n1(CC(=O)NCC2CN(C(c3oc(C)c(CO)c3)=O)C(C)C2)ccc(O)nc1=O 44149,C1(NC(=O)Cc2cncs2)CCCCN(c2nc(C3CCOCC3)ns2)C1 44150,C1(NC(C2C(C=C)C2)=O)CC2(C1)CC(CNC(=O)Cc1cccc(C)c1Cl)C2 44151,C(=O)(C1=CCCC1C)NCC1CC(COC)CN1C(C1OCCC1C)=O 44152,C1(C(C)C)(C(=O)NC(C2CN(C(=O)C(O)C(F)F)C2)C)CNC(=O)C1 44153,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44154,C(CCN(C)C)(C(=O)N1CCOCC1C(F)F)NC(c1scc(C)c1)=O 44155,c1(CC(=O)NC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C2CCC2)nc(O)n[nH]1 44156,c1(C(=O)NC(C2CCN(C(=O)C(CO)c3ccccc3)C2)C)cnnn1C 44157,N1(C(C(C=C)O)=O)CCC2(CCN(C(c3nccnc3CC)=O)C2)C1 44158,C(C(=O)N1CCC(O)(CNC(N)=O)C1)(C(F)(F)F)NC(Cn1c(C)ncc1)=O 44159,C1(NC(NC(c2c(C)cccn2)C(C)C)=NCc2ccccc2)CC12CC=CCC2 44160,S(=O)(=O)(c1ccc(F)c(C(=O)NC2C3CC2N(C(=O)C(C)N(C)C)C3)c1)NC(C)=O 44161,C1(CNCc2ccc(OCCC)cc2)CC2(CCC2O)C1 44162,c1(C(=O)OC)csc(S(=O)(=O)N(C)CC2CCO2)c1 44163,N1(C(C(c2c(C)cncc2)C)=O)CC2(C1)SCCC2NC(=O)CSc1cn[nH]c1 44164,N1(C(CSCC#C)=O)CCC(C=CC(=O)NCC2CC(C)C2)CC1 44165,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC2(CC1)CCN(CC1CCC1)CC2 44166,c1(C(N2C(CCNC(C3CC34CCC4)=O)CCC2)=O)nccc2nn[nH]c12 44167,C(=O)(CC(C)P(C)(C)=O)NCC(CCCC)NC(=O)CN(C)C(c1ccoc1)=O 44168,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnn(C)c3F)=O)C2)cc1C 44169,n1(C(C(N2C3CC(CNC(COC)=O)CC2CC3)=O)C)cnc2cc(C)ccc12 44170,C(=O)(C1=CCCCC1C)N1C(CC(=O)NCc2c(CC)con2)COCC1 44171,c1(C(N(C)CC2CCCN2C(=O)C(=O)NC2CC2)=O)ccc2c(c1)CCCCN2 44172,n1(CC(=O)NC(C)(CNC(=O)C(C#N)C2CC2)C2CC2)nnc(-c2ccsc2)n1 44173,CCCC(CC)C(=O)NC1(c2ccccc2)CC(NC(C2CCS2(=O)=O)=O)C1 44174,c1(NCC(=O)NC2CC(N(C(CCNS(CC)(=O)=O)=O)C)C2)cc(C)ccc1F 44175,CCC(CC(=O)N(C(C)CCNC(C1(C(=O)NC)CC1)=O)C)CC(C)C 44176,CC1(NC(=O)C(C2CCN(C(=O)Cc3csnn3)C2)F)CC2(CCC2)C1 44177,C12(CCNC(c3c(C)nn[nH]3)=O)CCC(CC1)N(C(c1ccc(F)c(F)c1)=O)C2 44178,c1(COC)ccccc1C(=O)NCCCCC1CN(C(c2nn(C)nc2C)=O)C1 44179,Cc1nc(Cl)c(NC(C2CC2C(=O)NCc2cc(F)cc(I)c2)=O)cc1Br 44180,Cc1c(C(=O)NCc2cc(C(=O)NC3CCCCC3O)co2)cnn1C 44181,c1(OC)cnc(C(=O)OC(CN(C(COC)=O)C(C)C)(C)C)cn1 44182,c1(C(N2CCC(O)(CCNC(C(COC)C)=O)C2)=O)cc(F)c(C)cc1Cl 44183,CC1CCN(C(=O)CN2CC3CCC2C3)C(C)C1NC(=O)CCc1cscn1 44184,c1(CC(=O)NCC2N(C(C(C)CC3CCCC3)=O)CCOC2)nnc(S)nc1O 44185,C1(CO)CC2(CCOCC2)CN1Cc1cc(N)ccc1F 44186,c1(C(=O)NC2(CN(C)C(C3CCCC3n3cccc3)=O)CC2)cc(C(F)F)on1 44187,c1(N2CC3CN(S(CCCC)(=O)=O)CC(C2)O3)ncnc2ccc(OC)cc12 44188,C12(CC)CN(C1)C(=O)C1N(CSC1)C2=O.C1(NC(=O)C2CC2)CN(C(N)=O)C1 44189,C1(OCCNC(N2CCCC(OCCC)C2)=O)CCC2OCCC2C1 44190,N1(C(=O)C(N2CCOCC2=O)C2CC2)CCc2[nH]nc(-c3ccncc3)c2C1 44191,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44192,N1(C(CCN(CC)CC)=O)CC(NC(C23CC(CN2C)C3)=O)CC(O)C1 44193,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44194,C12(NC(c3cc(C)n(C4CC4)n3)=O)CCC1CN(C(=O)CC1CCS(=O)(=O)C1)C2 44195,N1(C(C(C)N(C(=O)COC)CCC)=O)CCC2(CNC(=O)N2)C1 44196,c1(C(N2CCC(O)C2C(N2CCC2CO)=O)=O)cccc(Cl)c1F 44197,CC1CCCC(N(C(=O)CC2CCCCO2)C)C1C.C12CC3(CC(C3)NC1=O)C2 44198,C(c1cc(C)c(C)cc1C)=CC(=O)NCC(c1cccc(C)c1)NC(=O)CO 44199,C1(OC)CN(C(=NCCF)NCC2(C)CCCC2(F)F)CC1O 44200,C1(C(=O)NCCCNC(C(C)C)=O)CC(C)N1C(=O)C=Cc1cc[nH]c1 44201,O=S(=O)(c1cccc2ccccc12)NCc1ccnc2c(Br)cccc12 44202,c1(CC(=O)NC(CNC(c2ccc(C3CC3)o2)=O)C2CCC2)ccc(F)cc1Cl 44203,N1(C(CCc2c(C)ccs2)=O)CC2C(C(=O)NC(c3nn[nH]n3)C3CC3)C2C1 44204,C1(C#N)(OC)CC(C(=O)NC(C)CNC(=O)CSc2nncn2C)C1 44205,c1(CN(C2CCN2)C(=O)Nc2c(C(F)(F)F)ccc(C)c2)ccc(O)cc1[N+](=O)[O-] 44206,c1(NC(CNC(c2ccc(COC)s2)=O)C)ncc(Br)cc1C#N 44207,c1(CCCC(=O)NC(CC)CNC(=O)Cc2noc(C(N)=O)n2)c(C)n[nH]c1C 44208,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)CO)CCCC2(CCCCC2)C1 44209,c1(NCC2N(C(c3c(C)cc(Br)cc3F)=O)CCC2)c(C#N)oc2ccccc12 44210,N1(C(c2cc(C)n(C)c2C)=O)CCC(NC(c2cnc(CO)nc2)=O)CC(O)C1 44211,C1(CC=C)(C(=O)N(CC(C)(C)C)C)CCCN1C(=O)CCCc1ncco1 44212,N1(C(CCC(=O)N(CC)CC)=O)CC2CCCN(C(=O)C=CC=C(Cl)Cl)C2C1 44213,C1(C(N(CC(=O)O)CCc2cn(C3CCS(=O)(=O)C3)nn2)=O)CCCC1(F)F 44214,Cc1cnc2ccc(C(N3C4CCC3CN(C(=O)CCCF)C4)=O)cn12 44215,S(=O)(=O)(c1cnn(-c2ccccc2)c1)NC(C1CC2CC2N1C1CC1)=O 44216,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCCC3)=O)CC2)C1)=O 44217,c1(C(N2CC(CNC(c3scc(C)c3)=O)OCC2)=O)cccc2ncc(C)n12 44218,N1(C(CC2CCC(=O)C2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44219,c1(C(=O)NCCCC(C)NC(c2ncc(OCC)nc2)=O)c[nH]c2nccc-2c1 44220,C1(CC)CC2CCC1N(C(c1nc(Cc3ccccc3)sc1C)=O)C2 44221,c1(C(N2C(C)CC(CNC(CCCC(=O)OC)=O)C2)=O)cc2n(c(=O)c1)CCS2 44222,C12(CCC)CC(C(=O)N(C)CCN(C(C3CC=CCO3)=O)C(C)C)(C1)C2 44223,c1(NC2(CCC)CCN(C(=O)C(C)CC3CCCCC3)C2)ncnc(OC)c1F 44224,CC(C(=O)NCC=Cc1cscn1)C(C)NC(=O)C(N)=O 44225,N1(C(c2scc(CC)n2)=O)C2CC1CN(Cc1ccc(F)cc1I)C2 44226,C1(C)(CC)CCN(C(C2CC2C2CN(C(c3n[nH]cc3Cl)=O)C2)=O)CC1 44227,N1(C(C2COCCOC2)=O)C2CC=C(C(=O)NC3(C)CCCC3)C1CC2 44228,CC(C)C(C(=O)NCc1ccccn1)C(C)NC(C1CC(=O)N(C)C1)=O 44229,Cc1cnn(CC(N2CCC3C(NC(=O)C(CCO)NC(N)=O)C23)=O)c(=O)c1 44230,c1(C(N2CCN(C(COCC=C)=O)C(CO)C2)=O)cnn2cccc(Cl)c12 44231,c1(C(=O)NCC2(CNC(=O)CC(F)F)CCCC2)ccc(O)cc1F 44232,C(C)(C(=O)NC(C)CC1CCC1)CCNC(C1(CCOC)CC1)=O 44233,c1(CC)cc(C(N2CCC(CCNC(=O)CC3(C)CC3(F)F)CC2)=O)cc(O)n1 44234,C1(NC(C2CC(O)(CNC(C(n3ccc(C(F)F)n3)C)=O)C2)=O)CCC(C)(C)C1 44235,N1(C(CCC#C)=O)CCCCC(NC(c2ccc(NCc3ncc[nH]3)nc2)=O)C1 44236,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCN1C(=O)CCCn1ccnc1 44237,C1(CNC(C2CCC2)=O)CN(C(C2CCCN2C(C2(CCO)CC2)=O)=O)CC1O 44238,c1(C(N2C(C(C)(C)CNC(=O)CC3CC3C(F)(F)F)CCC2)=O)cnc(=N)[nH]c1 44239,CCC(C)C(CO)NC(c1conc1C)=O.C(=O)(C(F)=C(C)CN1CCCC1)N 44240,C1(CC#C)(OCC(C(=O)NC)NC(=O)CC(=O)NC)CCCC1.C1CC1 44241,C12(CC)CC(CNC(C)CC(C)(C)c3ccccc3)(CO1)C2 44242,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44243,N1(C(=O)NC2CNC(C3CC3)C2)CCc2c(-c3ccccc3)cccc21 44244,c1(C(=O)NCC2(F)CC(CNC(c3cccnc3O)=O)C2)cc(C2CC2)ccn1 44245,Cc1cncc(C(=O)NCCOCCCN(C)C(C2CCC(N(C)C)CC2)=O)c1 44246,C(CN=c1cc(NC(C)C)nc(C(C)C)[nH]1)(c1ccccc1)OC(C)C 44247,c1(CNC(C2(CC#C)CCC2)=O)ccnc(C(N2CCC(O)(CN(C)C)C2)=O)c1 44248,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44249,c1(-c2n(C3CCN(C)CC3)ccn2)cn(C)ccc1=O.c1(CC)ncno1 44250,N1(C(C(COC)(F)F)=O)CCC(C2(O)CN(C(C3CCCS(=O)(=O)C3)=O)C2)CC1 44251,CC1CN(C)CC1CNC(=O)OC(C)(C)C.c12nc(cn1C)NC2 44252,c1(C(=O)NC2C3(CC(NC(C(C)(C)N4CCCC4)=O)C3)C2)ccc2nonc2c1 44253,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44254,N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CC2NC(=O)Cc1cc(C)cc(F)c1 44255,c1(COC)ccc(Cl)cc1C(=O)NCCCN(CCO)C(C1(O)CCCC1)=O 44256,C(=O)(CCS(=O)(=O)CC(C)C)N1CCCC(O)(CNC(C(CCC)OCC)=O)C1 44257,C1(CC(=O)NC2CCOC2=O)CC2(C1)CN(C(=O)Cn1cc(CC3CC3)nn1)C2 44258,c1(C(=O)NC2CC(NCCCCS(C)=O)C2(C)C)cccc2c1OCCO2 44259,C1(C(N(CCC(=O)NCCCOC(=N)O)C2CCCC2)=O)CC(O)C(F)C1 44260,c1(C(N(CC(CC)C)CC(N)=O)=O)conc1C(C)NC(c1csc(O)n1)=O 44261,C1(c2cn(CCN(C(c3cnc(C)nc3)=O)CC)nn2)CCC(F)(F)CC1 44262,N1(C(C)=O)CCc2ccc(CN(C)C)cc2CC1.c12ccc(s1)NC(=O)CC2 44263,CCC(CC)CCCC(=O)NCC1=CCN(C(c2nc(F)c(F)cc2F)=O)CC1 44264,c1(CCNC2(c3n(C(C)C)nnn3)CC(Cc3ccccc3)C2)cc(F)cc(F)c1 44265,C(=O)(C(CCOCCO)NC(=O)CC1CCOC1=O)NCCOCC 44266,c1(C(N(C2C3CN(C(CSCCCC)=O)CC32)C)=O)ncc([N+](=O)[O-])cc1C 44267,N1(C(c2c(C)cccn2)=O)CCC(NC(=O)CSC(F)(F)F)C2(CCC2)C1 44268,CC1COCC(CC(N2CCC(C(O)CNC(c3cccc(O)n3)=O)CC2)=O)O1 44269,c1(C(=O)Nc2cncc(C(N3CCC(CC(=O)OC)C3)=O)c2)cc(Cl)ncc1I 44270,c1(C(=O)NCC2CCCCN(C(C3(C(F)F)CCC3)=O)C2)ccc2nccn2c1 44271,c1(SCC)nc(C)c(CC(=O)NC2CCN(C(=O)C=CBr)C2)c(O)n1 44272,c1(C(=O)NCC2CC(CNc3nc(SC)nc(Cl)c3)OC2)cc2ncccc2o1 44273,C(=O)(CCS(=O)(=O)NC)NC1C(NC(C2N(OCC)CCCC2)=O)CCC1 44274,C(=O)(C(C)(F)C(=O)NCCC(O)CNC(=O)CCc1c(C)n[nH]c1C)OC 44275,C1(CC(=O)NCC(CN(C(=O)COC(F)F)C)O)CCN(Cc2nnnn2C)CC1 44276,N1(C(C2CC(C)(CC)C2)=O)CC2(CCCC2)C1C(=O)NOCC1(O)CCC1 44277,C1(C(=O)NC2CCC(CCC(=O)NCc3nc(O)n[nH]3)C2)CC2(CSC2)C1 44278,C(=O)(C(C)(C)C(F)F)N1CC(O)(CCNC(CC(C)NC(=O)OC(C)(C)C)=O)C1 44279,CCC(C)(CNC(=O)CC(C)F)C(=O)NCC1CC(O)C(F)C1 44280,C1(NC(C=C(C)C2CCCCC2)=O)C(CNC(c2csnn2)=O)CCC12CCC2 44281,C1(C(=O)NC(CCC)CCCNC(c2ccc(CC)s2)=O)CC(C(C)(C)C)=NO1 44282,C1(CC(=O)N(CC(CNC(C(C)C2CCC2)=O)O)C)COC(C)(C)C1 44283,N1(C(c2n(CC)ccc2)=O)CCN(C(=O)Cc2ccc(C)cn2)CC1C(C)(C)C 44284,C12(C(=O)NC3CC(N(C(C4C(C=C)C4)=O)C)C3)C3CC(CC13)C2(F)F 44285,Cc1nccc(Cl)c1C(=O)N(C1CN(C(C23CCC(CO)(CC2)C3)=O)C1)C 44286,c1(C(N2CCCC(NC(C3C(C)CCS3)=O)CC2)=O)ccc(F)c(Cl)c1F 44287,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1CC(=O)N(C)C1)=O 44288,CC1(C)OCC(Nc2cccc(NC(N3CCCCC3c3cnccn3)=O)c2)O1 44289,N1(C(CCC(=O)NCC)=O)CCC(NC(=O)C(c2cn(C)nc2C)O)C(C)(C)C1 44290,N1(C(c2cnc(CC)o2)=O)CCC=CC1C(=O)NCC(C#N)CC 44291,C(=O)(C1=CCC2CCC1N2C(c1ccc(C)c(C)c1)=O)NCc1n(CC)cnc1 44292,N1(C(C(CC#C)C)=O)CC(C)OC2(CCN(C(c3cc(OCC)cs3)=O)CC2)C1 44293,C(=O)(CC(C)C(=O)N1CC(C(C(=O)NCCC(C(C)C)OC)OC)C1)OC 44294,Cc1cc(Br)c(F)cc1N(C)C(c1cncc(C(F)(F)CF)c1)=O 44295,C1(C(N(CCCC=C)CC)=O)CCCN(C(C2(CC)CCCCC2)=O)CC1 44296,C#CCCCCC(=O)NC(C)(C)CNc1nc(OC)cc(COC)n1 44297,C(C#CC(=O)N(CCCCO)CC)NC(C1CC(=C)C1)=O 44298,CC12CC(C(N3CC(C(n4cc(COC5CCOCC5)nn4)C)C3)=O)(C1)C2 44299,C(=O)(C(O)C(C)CC)N(C)CC1(NC(C=CC(=O)OCCCC)=O)CC1 44300,C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1(NC(c2cc(C(C)(C)C)on2)=O)COC1 44301,C1(C(=O)NCC2(OC)CN(C(c3ncccc3N)=O)C2)CN2CCC1CC2 44302,C(N=c1ccnc(Cl)[nH]1)C1(O)CN(C(C(C)O)=O)C1 44303,c12ccc(cc1)oc2=O.C1(C(=O)OC)CCC(C(=O)OC(C)(C)C)C1 44304,C1(NC(=O)Nc2c(OC)nccn2)CCC(C)N(C(C2CCS(=O)(=O)CC2)=O)C1 44305,C(=O)(C#CC(C)(C)C)N1CCC(N(C(c2c(OC)nsc2)=O)C)CC1 44306,c12cc(Cl)c(OC)cc1[nH]c(=O)[nH]2.C(=O)(C(C)CCC)OCC(F)(F)F 44307,c1(CC(N2CCC(CCNC(COC(CC)C)=O)C2)=O)ccccc1F 44308,N1(C(C2C(COC)(COC)C2)=O)CCC2CN(C(=O)C3=CS(=O)CCC3)CC2C1 44309,C1N=C2C=C(N=CN2)N1.C12(CNC(C3CN(C)CCO3)C)CCC(CC1)C2(C)C 44310,c1(C(N2CC(NC(CC(C)OC)=O)C(C)(C)C2)=O)cccc2oc(C)nc12 44311,N1(C(c2nc(COC)sc2)=O)CCN(C(=O)CC(C)C)C(CC(=O)N(C)C)C1 44312,Cc1cc(Cl)ncc1NC(C1CCCCN1C(=O)Cn1cccn1)=O 44313,CCCCCC(=O)N1CC(O)CC1NC(=O)N(C1CCOC1)CC 44314,CCC(C)(C)CCCC(=O)N(C)CCOCCNC(C1CCC2CC1C2(C)C)=O 44315,c1(C(=O)NCCC2CC(OC)CN2C(=O)CC(C)(C)C)cc2nn[nH]c2cc1F 44316,Cc1ccc(N2CCC(NC(=O)NCCC3CC3)C2=O)cc1 44317,N#Cc1cc(C2C(C(=O)NC3CCC3NC(=O)CCSc3ccccc3Cl)C2)no1 44318,C1(CC(=O)NC)CN(C(=O)CC=Cc2cccnc2)CCN1Cc1cc[nH]c1CC 44319,C1(C(N(c2ccsc2Br)C)=O)CCN(C(=O)C=CC2CC2)CC1(C)C 44320,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)COCCCF)C)cc1C 44321,C1(OC)C(C(=O)OCC)C(C)C(N(C)C)CC1N1CC(=O)NCC1c1ccccc1 44322,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44323,c1(C(N2CCN(C(C3C(=C)C3)=O)C(C)C2)=O)cccc2nc(O)[nH]c12 44324,c1(C(=O)NC(c2ccccc2)CNC(C=CCCC)=O)nccnc1C(=O)NC 44325,C(=O)(C(F)C(F)(F)F)N(CCCN1CC(C)(C)C1C(F)(F)F)C 44326,N(C1CC2(CN(C(C3(F)CC3)=O)C2)n2ccnc21)C(N1CC(C)C1)=O 44327,c12ccnc(c1)C(=O)C2=O.c1(C(N2CC(N)C2)=O)ccnc(Br)c1.CO 44328,c1(C(N2CC(CCNC(COC)=O)OCC2)=O)cncc(N=[N+]=[N-])c1 44329,c1(CC)cc(C(=O)NCC(C)(O)CNC(=O)CC2CC(C)=NO2)cc(O)n1 44330,C1(CNC(=O)CC23CC(C2)C3)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)CC1 44331,C(=O)(C1Cc2ccccc21)N1CCC(C)(NC(c2n[nH]c(CC)c2C)=O)CC1 44332,c1(SC)ccc(C(=O)NC(C)CC2CN(C(C3CCCC3O)=O)C2)cc1 44333,C1(NC(CC2C(NC(C=CC(=O)N(C)C)=O)CCC2)=O)CCCN(C)C1=O 44334,c1(C(N(C)CC2N(C(CSCC#C)=O)CCC2)=O)ccc(NC(=O)CO)cc1 44335,CC1(C)OCC(CCC(=O)NC2CC2c2cnn(-c3ccccc3)c2)O1 44336,C1(COC)CCCCN1C(=O)NCC12CC(C3CC3)(CO1)C2 44337,C1(C)(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(c2nnsc2C)=O)C1 44338,C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(C2CCC=CO2)=O)CC1 44339,n1(CC)ncc(Cl)c1C(=O)NC1CCC(C)(C(C)(C)C)C1 44340,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44341,Cc1nc(C)c(C(N2CCC(C)(CNC(c3scnc3C)=O)C2)=O)[nH]1 44342,N1(C(C(C(C)C)OCC)=O)CCN(C(C2CC(C)(F)C2)=O)CC1CC(F)(F)F 44343,Cc1cc(C(=O)OCC(N2CC=CC(NC(C3CCCC3)=O)C2)=O)c2c(c1)CCC2 44344,N1(C(CCC(=O)N(CC)CC)=O)CCC(CNC(=O)Cc2ccsn2)C1(C)C 44345,c1(C(=O)NCCCCC(CO)NC(C2CCCO2)=O)cnc2cccnn12 44346,C(=O)(C1=CC(O)C(NC(=O)C2=CCCC2C)C1)NCCC1CC(C(=O)OC)C1 44347,C1(C(=O)NCCC(CNC(C#CC(C)(C)C)=O)O)Cc2ccccc2C(=O)O1 44348,N1(C(C(C2CCCC2)NC(C)=O)=O)CC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C1 44349,C1(NC(c2cc(OC)no2)=O)CCCCN(c2nnc(-c3ccon3)s2)C1 44350,C1(CNC(CCNS(CC)(=O)=O)=O)CC(F)(F)CN1C(=O)CC1CCOC1 44351,S(=O)(=O)(CC(C)C)NC1CN(CC(=Cc2ccco2)C)C1 44352,N1(C(C(C)OC)=O)Cc2ccccc2C(NC(c2cc(C)ccc2Br)=O)C1 44353,CN1CC(O)CC1(C)C(N1CCC(C(=O)NCC2COCCN(S(C)(=O)=O)C2)CC1)=O 44354,N1(C(C2C(C)C2(F)F)=O)CCN(C(=O)CCNC(C2CCC2)=O)C(C(C)C)C1 44355,c1(C(C(=O)NC(C)C)NC(c2c(C)n(C3CC3)nc2)=O)ccc2c(c1)C=CCC2 44356,N1(C(c2csc(C(F)F)c2)=O)CC2(CCN(C(c3sccc3F)=O)C2)C1 44357,C1(CC)CCN(C(=O)CC2(O)CCC2)C(C(N2CCNC(=O)C2C)=O)C1 44358,CC(C)(C)C(CO)C(=O)NC1(C(=O)NCC2CC2Cl)CC(F)C1 44359,C(C(CN(C)C(c1ccccn1)=O)S(C)(=O)=O)NC(C(C=C)C)=O 44360,C1(NC(CCC=CCC=C)=O)CCN(C(c2ccc(F)cc2O)=O)C12CCC2 44361,C#Cc1ccccc1NC(=O)C(CCC=C)NC(=O)CCCC 44362,C(CCCCC(=O)N(C)CC1OCCC1(C)C)NC(c1cc(C)ns1)=O 44363,Cc1cc(C(N2CC(NC(C3(C)CCC(F)(F)C3)=O)C(C)(C)C2)=O)ncc1CO 44364,N1(C(c2c(OC)nccc2)=O)CC(C(=O)NCCc2cnc[nH]2)CC12CCC2 44365,C1(O)(CNC(NC2C(C)C2)=NCC2CCC(F)CC2)CN2CCCC1C2 44366,C1(CNC(c2cnnn2C2CC2)=O)CCN(C(c2cn3c(n2)SCC3)=O)CC1O 44367,N1(C(C=Cc2cn(C)nc2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1Cl)C2 44368,C(=O)(CC(C)(C)CNC(C1CCCC1O)=O)NCC(C)(C)C(F)F 44369,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C(C)N(C(C)=O)C)=O 44370,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(C2CCCN2C(C)C)=O)C(C)C1)=O 44371,CC1CC(C)(C)CCC1NC(=O)C(=O)Nc1cccc(CN2CCOCC2)c1 44372,C(=O)(C(C)(O)C1CCC1)NCC(C)CNC(C1(Br)CC1)=O 44373,N1(C(COCCC=C)=O)CCC(C)CC1CNC(c1ccc(OC(C)=O)c(F)c1)=O 44374,C1(C(=O)NC2CC(OC(F)F)C2)CCC2(CCCC2)C1 44375,CC1(C(=O)NCCCCC(=O)NCC2(CO)CCOC2)CCC(=O)C1 44376,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44377,C1(NC(=O)CCCc2ccc3ncccc3c2)CCCOC12CCS(=O)(=O)CC2 44378,c1(C(N(CCCNC(COCCCCC)=O)C)=O)cnnc(-c2ccccc2)c1 44379,C1(=O)C(C(C)(C)C)n2cc(nn2)C(C)N1.C1(OCC)C(C(=O)O)CCC12CC2 44380,c1(CNC(c2cnn(CC)n2)(C)C)c(F)cccc1Cl 44381,C1(CN(C(=O)Cc2cncs2)CC)CCCCN1C(C1CC(OC(F)(F)F)C1)=O 44382,c1(C(=O)NC(CCNC(C(C)OCCOCC)=O)C(C)C)cc(S(N)(=O)=O)c[nH]1 44383,C1(C(=O)NCC2CCC(NC(C3CCCC(F)C3)=O)C2)CC2(CSC2)C1 44384,N1(C(C(CC)SC)=O)CCc2ccccc2C1CNC(C1CC2(C1)CC(C)(C)C2)=O 44385,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44386,C=C(C)CCCN=c1nc2ncn(CC)c2c(NC(CCNC(C)C)=O)[nH]1 44387,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(=O)C=Cc3ncco3)CCC2F)c1Cl 44388,C(=O)(C1=CCCSC1)NC1(COC)CCN(C(=O)CC2CC23CC3)C1 44389,c1(C(=O)NCC2C(NC(c3c(C)n[nH]c3)=O)C2)coc(C#N)c1 44390,C(=O)(C#CC(C)(C)O)NC(C1(CNC(C2COC(C)(C)C2)=O)CC1)C 44391,c1(C(N2CC3(CCC3)C2)=O)ccc(NC(C2CCC(=O)N(C)C2)=O)nc1C.CO 44392,C(=O)(C(C)(C=C)CC)N1C(CC(=O)NC(C#C)CCC)CC1 44393,c1(C(=O)NC(C2CCN(C(c3cc(C(=O)O)n(C)n3)=O)C2)C)ncc(Cl)cc1F 44394,C=C1COc2c(C(=O)NCCC(C)NC(C3(Br)CC3)=O)cnn2C1 44395,C1(C(=O)NCC(CNC(COCC(C)C)=O)O)CCCCCN1C 44396,CC1COc2cc(C(N3CCCCC(c4ccccc4)C3)=O)ccc21 44397,C1(CC(N2CCC(CCC)C2)=O)CCCN(C(=O)CC2CC(C)=NO2)CC1 44398,C1(COC)(NC(C2C=CC=CC=C2)=O)CCN(C(=O)CCc2cn(C)nc2C)C1 44399,c1(CN2CCC(C(N(C3(C)CCCC3)C)=O)C2)ccc(Br)c2cccnc12 44400,C1(CC#C)(C(N2CC(F)(CNC(c3ccc(C(C)C)nc3)=O)C2)=O)CCCCO1 44401,Cc1cc(N)c(C)nc1C(=O)NCCCOCCN(C)C(C1C=CCCCC1)=O 44402,c1(CC(=O)NCCC(CNC(C=C(C)C(F)F)=O)O)csc2c(F)cccc12 44403,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44404,N1(C(C(CC(=O)OC)(C)C)=O)CCCC12CCCN(C(=O)C(O)C(C)C)CC2 44405,c1(OC)cc(CN2CCOCC(Nc3cn(C)nn3)C2)ccc1OCC(=O)O 44406,C(=O)(C1OCCc2ccccc21)N1CC(SC)C(NC(=O)C(O)CCN(C)C)C1 44407,Cc1c(CC(=O)NCC(CO)NC(=O)C=Cc2cn(C)nn2)ccc(Cl)c1Cl 44408,C#Cc1cncc(C(=O)N(C(C)CCNC(C2CC(F)C2)=O)C)c1 44409,Cn1cc(C(=O)NOCC(C2CCCO2)=O)nn1.C(C)(CO)(C1CCC1)N 44410,C1(CC(=O)OC)(c2nnnn2CCF)CN1.C(=O)(CCCNC(C)C)OCC 44411,C1(C(=O)NCC2(NC(=O)CNC(c3ccccc3)=O)CCC2)CC2CC1C2 44412,N1(C(C2CC(N3CCCC3)C2)=O)CCCN(C(c2snnc2SC)=O)CC1 44413,c1(OC)cc(CCC(N2CC(NC(=O)C(N)=O)C(O)C2)=O)ccc1Cl 44414,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44415,Cc1cc(C)nc(SCC(=O)NCC(C)CN(C)C(C2(F)CCCC2)=O)n1 44416,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44417,C1(C(CNC(C(C)C#N)=O)O)CCN(C(=O)CSCC2CCCOC2)CC1 44418,n1(CC)cc([N+](=O)[O-])c(C(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)n1 44419,C1(NC(COCc2cc(C)no2)=O)CN(C(c2cnn(CCO)c2C)=O)CCC1F 44420,C#CCC(C)(C(=O)NCc1nn(C)cc1C)NC(=O)CCN1CCCC1=O 44421,c1(C(=O)OCc2cccc(C(F)(F)F)c2F)nnn2c1COCC2 44422,Cc1ccc(C(=O)C=CC(=O)N(C2CCN(C(=O)C(=O)NC(C)C)CC2)C)cc1C 44423,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44424,N1(C(C(C2CC(NC(C(CC)=CC)=O)C2)F)=O)CCN(CCO)C(C)C1 44425,C1(C)(CNC(C2CCC(C)O2)=O)CCN(C(c2cnccc2Cl)=O)CC1 44426,c1(OC)c(Br)ccc(F)c1CN1CC2CC2(C(=O)Nc2cncnc2C)C1 44427,C(N=c1cc(C)nc(NCc2ncccc2Cl)[nH]1)c1ccc(C)cc1Br 44428,C1(N(C(=O)Cc2csc(Cl)c2)CC)CCC(CNC(=O)CC2OCCC2C)CC1 44429,C(CCS(=O)(=O)C(C)(C)C)N(C(=O)NC(c1cccs1)CC)C 44430,c1(NC(CN(C(C(C)CC2CC2)=O)CC2CC2)=O)cc2ccccc2o1 44431,CCC1=C(C(=O)N2CCN(C(c3c(CC)cccc3F)=O)CC(O)C2)CCCO1 44432,C1(C(=O)NCC(C)(C)CCNC(=O)C(O)C(F)(F)F)CCCC2(CCC2)O1 44433,C#CCCCC(C)C(=O)N1CCS(=O)(=O)C(CCNC(=O)CCCC(=O)N(C)C)C1 44434,C(CCCC(=O)NC(C)(C)CC(=O)NC1C=CCC1)N(C)C 44435,C(=O)(CC(Cc1ccccc1)OC(c1ccccc1)=O)N1C(CN=[N+]=[N-])CSCC1 44436,c1(OC)cc(CCNC(=O)C(c2ccc(Cl)c(F)c2)O)cc(Br)c1 44437,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44438,S(=O)(=O)(c1ccc(C#N)c(N2CCCC(C)(F)C2)c1)NCC(N(C)C)C1CC1 44439,Cc1cc(CC(=O)NC(CNC(=O)C(C(C)C)c2ccn(C)n2)C2CC2)n(C)n1 44440,N1(C(=O)OC(C)(C)C)CC2CCCC1C2c1noc(-c2cc3n(n2)CCC3)n1 44441,Cc1ccc(F)c(N)c1C(=O)OC(CC(C)C)C(N)=O.C12CCN(CC1)C2=O 44442,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CC(=O)OC)C1)(C(C)C)OCC 44443,N1(C(c2cc(OC)nn2C)=O)Cc2ccnn2CC(NC(=O)CCC2(C)CC2)C1 44444,N1(C(c2nn(C(F)F)cc2Cl)=O)CCN(C(C2(F)CCOCC2)=O)CC1C1CC1 44445,N12CC3(CCC3)CC1NC(=O)C2.CC(COc1ncccn1)(CO)c1ccccc1 44446,C(C(CO)C(F)(F)F)NC(c1sccc1CNC(C1CCCCS1)=O)=O 44447,N1(C(CN(c2ccccc2)C)=O)CCOCC1CCNC(C1CC1C1CC1)=O 44448,CCC(C)C(CO)NC(C1(F)CN(C(=O)COC(C)(C)C)C1)=O 44449,N1(C(C=CCC)=O)CCCC(C)C1CCNC(=O)CCc1ccnc(C)n1 44450,N1(C(C(C=C)c2ccccc2)=O)CCC(CC)C1CNC(c1cnc(S)n1C)=O 44451,c1(NC(C(C)N(C(=O)CCc2scnc2C)CCC)=O)cccc2ccncc12 44452,N1(C(CCOC)=O)CCC(C)(C(=O)NC(c2ncc(C)o2)C)C1 44453,c1(C(=O)NC(CN(C(=O)C(C)CC2CCCC2)CC)C)cccnc1C 44454,C(=O)(C1CCCc2c[nH]nc21)NC1C(CNC(CSCC(C)C)=O)COC1 44455,C1(NC(C2C(OCC)C2C)=O)C=CCN(C(c2cc(OC)n(C)n2)=O)C1 44456,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC2(CCC2)C1 44457,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCSC(F)(F)F)CCC1F 44458,Cc1nnc2n1CCC(N=c1[nH]c(=NC3CCCOC3)[nH]c3ccsc13)C2 44459,Cc1ccc(NC(C2(n3cnnn3)CCOCC2)=O)cc1N1CCCC1=O 44460,C1(CNC(C2(C)CC(C)C2)=O)CN(C)CCN1C(C1CCN(CC(F)F)CC1)=O 44461,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC(C)C)CC1O 44462,CC1CN(C(=O)C(=O)NC2CCC2)CC(C)N(C(c2cccnc2C(F)F)=O)C1 44463,N1(C(C=CCN(CC)CC)=O)CCC=C(C(=O)N(C2CCSCC2)C)C1 44464,N1(C(CC2C(C(C)(C)C)C2)=O)CC2CC(CNC(=O)CCC3CCOCC3)C1C2 44465,N1(C(CC=C=C)=O)CCC2(CC1)CC2C(=O)NCCc1nncn1C(C)C 44466,c1(N2CC(NC(C3C(C)(Br)C3)=O)C2)ncc(O)cn1 44467,C(C(=O)N1CC(NC(C2CN(CC(C)C)C2)=O)C(C)C1)(C(C)C)SC 44468,C=CCC(F)(F)C(=O)N1CC2CC(NC(=O)CN3CCC(C)CC3)C1C2 44469,Cc1cc(C(C)NC(N2CCCC2C2CCCOC2)=O)cc(C)c1 44470,C(=O)(C(CC(C)C)C(C)C)NC(CN(C(c1cn(C2CC2)nn1)=O)CC)C 44471,C1(NC(CC2(C(C)C)CCCC2)=O)CCN(C(C2(COC)CC2)=O)CC1C1CC1 44472,c1(NC(C2(C)N(Cc3cn(CCC)nc3)CC2)=O)ccc(C#N)cc1C 44473,O=C(C1=CC2CC=CCC12)NCCCC1CCCN1c1ncc(F)cn1 44474,C1(F)(CC)CCC(NC(=O)C(=O)Nc2ccccc2OCC)C1c1ccccc1 44475,C1(CNC(CC2C(NC(=O)Cc3ccc(O)cc3)CC2O)=O)CCC(F)(F)CC1 44476,c1(C(CC)NC=O)cc2cc[nH]c2cc1C(=O)Cn1cc(Cl)cnc1=O 44477,CC1CCN(C(C2CCCN2C)=O)CC1CC(=O)NC1C(C)C1(C)C 44478,N1(C(C(C)=CC)=O)CCCCC2(CCN(C(c3ccn(CCO)c3C)=O)C2)C1 44479,C1(C(=O)NC2(NC(CCCCNC(=O)NC)=O)CCC2)CC2CC1CC2O 44480,N1(c2nc(=N)nc(N3CCC(CC(C)C)CC3)[nH]2)C2CCC1c1ccccc12 44481,c1(C(=O)NCC(C)NC(C(C2CCCCC2)OC)=O)c(C)cc(Br)cc1C 44482,N1(C(C2CCC(C)O2)=O)C2CCC(C2)C1C(=O)N(C)CC1(O)CCC1 44483,N(C(=NCCc1nccs1)NCC1CCS(=O)(=O)CC1)C(c1ccoc1)C 44484,C1(NC(COc2cc(C)on2)=O)CN(C(C2CCOC2)=O)CC1C(F)F 44485,CC1(C(=O)NC(CNC(=O)C=C2CCC2)C2CC2)CCC(=O)N1 44486,CC(N=[N+]=[N-])C(=O)N1CCCC1CNC(C1C2CCC(F)C12)=O 44487,CC#CCC(C(=O)NCc1cc(C)sc1C)NC(c1ccn(CC)n1)=O 44488,C1(NC(C2(CC=C)COC2)=O)CCC(C)N(C(c2cnn(C)c2C(F)(F)F)=O)C1 44489,C1(OC)CCC(CCN(C(=O)C=CSc2nc[nH]n2)C(=O)Cc2ccccc2)C1 44490,C12CCN(C1C)C(=O)N2.C1(C)(CC(=O)NC)CSCCO1 44491,C1(O)(CCNC(c2cc(C(F)(F)F)cc(O)c2)=O)CCCN(C(=O)C=CBr)C1 44492,c1(OC)c(C(=O)NC2CN(C(=O)C(C)C#N)C2)csc1C 44493,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(NC(C(CSC)OC)=O)C2)C1 44494,c1(N2CCC(N(C(c3cn(CCC)nn3)=O)CC)C2)ncc2cccnc2n1 44495,N1(CC2(C)CC2)CCC(NC(=NCC2CCO2)NC2CCCCC2)CC1 44496,N#CC1(Cn2cc(C3CCN(C(=O)COC(F)F)C3)nn2)CCC1 44497,c1(OC)ccc(S(=O)(=O)N(CC(N2CCS(=O)CC2)=O)CC(C)C)cn1 44498,n1(CC)cc(Br)c(CC(=O)NC2CC2NC(=O)Cc2cncs2)n1 44499,CC(CCc1ccccc1)CC(=O)NCC1CCCC1c1ccccc1 44500,c1(NC(N2CCOCC2c2ccoc2)=O)ccc(C(F)(F)F)nc1 44501,C1(N(C(=O)Cc2cccnc2)CC)CCCN(C(c2ccc(Cl)cn2)=O)C1 44502,Cc1ccc(S(C)(=O)=O)cc1C(=O)NCCCCC(C)NC(c1ccc(F)cc1)=O 44503,c1(Nc2c(C(=O)Nc3cccc(SC(C)C)c3)scc2)nccc(Cl)c1Cl 44504,O=C(CCS(=O)(=O)Cc1ccc(C(F)(F)F)cn1)NCCOC1CCOC(C2CC2)C1 44505,N1(C(C)C)CCCC1C(=O)N(CCC(=O)Nc1cc(C2CC2)co1)C1CC1 44506,c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)csc(=NC2CC2)[nH]1 44507,c1(C(N2CCC(C)(C(=O)OCC)C2)=O)cc(C(C)=O)ccc1OC 44508,C1(C(=O)NCC#CCC)CN(C(C2CCCN2C=O)=O)CCN1C 44509,N1(C(Cc2ccc(OCCC)cc2)=O)CCC(NC(c2cc(C)ns2)=O)C(F)C1 44510,S(=O)(=O)(CCC(C(F)(F)F)OC)N1CC(CC(=O)OCC)OCC1 44511,c1(C(=O)NCC2C(NC(CC(C)c3cccnc3)=O)CC2)ccc(O)cc1F 44512,n12c(nc3ccccc13)N(OC(c1ccoc1C)=O)C(=O)CC2.N1(CC)CC(O)C1 44513,N1(CC(=O)N(c2cccc(F)c2)CC)CC2CN(C(C3COCCO3)=O)CC2C1 44514,c1(C(=O)Nc2cc(C)[nH]n2)ccccc1F.CC(CCC1CC1)N 44515,C1(CNC(c2nnc(CC)s2)=O)CCCC(NC(=O)Cc2ccc(Cl)s2)C1 44516,c1(C(=O)OC)cc(OC)ccc1NC(=O)NNC(=S)Nc1ccccc1C(N)=O 44517,C#CCC(CC(=O)NCC=CCNC(=O)C(C)=CC(C)(C)C)c1ccccc1 44518,c1(C(=O)OC)cccc(CC(F)(F)F)c1.CCC1CNC(=O)N1 44519,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)COc1cccc(F)c1C)C2 44520,c1(C(=O)NC2CCC(C(=O)Nc3cn(CCOC)nc3)C2)ccc(C)cc1C 44521,c1(C(N2CCCC(C(C)NC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44522,c1(C(N2CCCC(CNC(c3cc(C)n(CCO)n3)=O)C2)=O)cccc(N)c1C 44523,N1(C(C=C(C)C(C)(C)C)=O)CCC(C(=O)NCC2CN3CCC2CC3)CC1(C)C 44524,C1(C(=O)NCC(C)(C)NC(C2(F)CCOC2)=O)CC2CC1C1C2C1(F)F 44525,CCC(C)CC(=O)N1CC(OC)C(CNC(=O)COCCOC)C1 44526,N1(C(c2ncnc(C)c2C)=O)CCCC2(NC(C34CCCC3C4(F)F)=O)CC2C1 44527,N1(C(C2C(CC)C2)=O)CCc2cc(CNC(C3CCCN3C(N)=O)=O)ccc2C1 44528,C1(CNC(c2n(C)ncc2)=O)CN(C(c2ccc(C(F)F)nn2)=O)C2CCN1C2 44529,C(=O)(CCCC(CC)NC(=O)CCc1ccoc1)NC(C#C)(C)C1CC1 44530,C(=O)(CC(C)(C)CNC(=O)Cc1occc1CNC(=O)C(C)c1cc[nH]n1)OC 44531,N1(C(C(C)N(C)C)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44532,c1(CC2CCC(C(N(CCCC)CC)=O)CC2)cccc(S(N)(=O)=O)c1 44533,N1(C(C)C)CCCN(CCCCNC(C2CCOC(=O)CC2)=O)CC1 44534,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44535,C1(CNC(c2ccc(C(C)C)s2)=O)N(C(c2ccc(F)c(Cl)n2)=O)CCC1(C)C 44536,Cc1nc2nccc(C(N3CC(NC(C4(CCN(C)C)CC4)=O)C(F)C3)=O)n2n1 44537,N1(c2nnc(CC)s2)CCCCC(NC(c2nn(C)cc2C)=O)C1 44538,N1(C(Cc2ccn(C)n2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44539,S1(=O)(=O)c2ccc(c(C#N)c2)NCC2CCN1C2.C(CC(C)CC(C)(C)C)SC 44540,c1(C(N(C2CCCC2)CCCNC(C(C)=C2CC2)=O)=O)cccc(C(C)(C)C)c1 44541,Cc1ccc(C(=O)NCc2nc(C(=O)NC(C)(C)CN3CCCC3)c(C)o2)cn1 44542,c1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCCC2)cnn2cccnc12 44543,CCC(CC)C(C(=O)NCC(C(C)(C)C)NC(c1cc(O)nn1C)=O)OC 44544,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)N(C)C 44545,N1(C(C2CC(=C)C2)=O)CCC2(NC(=O)COc3ccccc3OCC)CC2C1 44546,CCC(CNC(=O)C=CC(=O)N(C)C)(CC)NC(=O)C(C)Cc1ccccn1 44547,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44548,O=C(O)CC(C(=O)Nc1ncccc1OCc1ccc(Cl)cc1O)c1ccccc1 44549,c1(C(=O)NC2(C)CCCN(C(C(F)=CCC)=O)C2)ccc(CCC)c([N+](=O)[O-])c1 44550,Cn1nnc(C(=O)NCCCC(C)(C)NC(=O)CC2CC3(CC3)CO2)c1C(F)F 44551,C(=O)(C1=CCCSC1)NCCn1cc(C(=O)NC(CCCC)CC)nn1 44552,O(C=CC(=O)N1CC(O)C(O)CO1)Cc1c(C#N)ccnc1 44553,Cc1cn2c(n1)CC(C(=O)NC(C)CC1CN(C(=O)CNC=O)C1)CC2 44554,n1(CCC(=O)NC(C(C)NC(=O)C=Cc2ccsc2)CO)ccc(O)nc1=O 44555,c1(-n2cc(CCN(C(=O)NCc3nccn3C)CC)nn2)cnccc1C(C)C 44556,C(=O)(CCCS(N)(=O)=O)NCC1OCCN(C(c2ccc(C(C)C)cc2O)=O)C1 44557,c1(C(=O)NCC(C(C)(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44558,Cn1nc(Br)cc1CC(=O)NC1CC1NC(C1CCC(OCCN(C)C)CC1)=O 44559,C1(C(C(=O)N(CCNC(c2ccc(C(C)O)cc2)=O)C2CC2)O)CCC(C)(C)CC1 44560,CC1CN(C(C2CCC(=O)N2C)=O)CCC1NC(c1cnc2sccn12)=O 44561,C(C)(CCC(=O)NCCOCCOCCN(C)C(=O)Nc1ncccc1Cl)OC 44562,C1(F)(CNC(c2n(C)ncc2)=O)CCCN(C(C2CC(=O)N(CC3CC3)C2)=O)C1 44563,N1(C(c2ncn(C)c2)=O)CCC2(CC1)CN(C(c1cc(F)nn1C)=O)C2 44564,N1(C(C(C)OCCCC)=O)CCCC(CCNC(C2(O)COC2)=O)C1 44565,C1(CN(C(CC2(OC)CCC2)=O)C)CN(C(=O)CC2(OC)CCC2)CC12CC2 44566,N1(C(c2ccc(O)nn2)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)C2CC12 44567,N1(C(C(Cc2cnc[nH]2)OCC)=O)CCN(C)C(=O)C1.C1(C)C(=O)O1 44568,C(=O)(CCCC(F)(F)F)N(C)CCNC(=O)C(C1CCCCCC1)F 44569,c1(SCC(N2C(CNC(CC=C=C)=O)CCC2)=O)nc(O)c2c(C)c(C)sc2n1 44570,C1(Cn2cc(C3OCC(CNC(C(C)(C)C)=O)C3)nn2)CC2COCC(C1)C2 44571,C12(NC(=O)NCc3c(F)ncc(C)c3)CCC(C(N)=O)(CC1)CO2 44572,N1(C(C2(NC(CCCNC(N)=O)=O)CCSC2)=O)CC(CO)C(C2CC2)C1 44573,C1(CC)(NC(=O)C(C)(F)F)CCCN(C(C2CC(C)(C)CN2C)=O)C1 44574,C1(C(N(C(CC#C)C)C)=O)CCCN1C(=O)CC1(C)CCC1 44575,C12(NC(=O)Cc3ccco3)CCCC1N(C(=O)Cc1ccccc1)CCC2 44576,C(=O)(CCCCC(=O)N1CC(C)(C)CC1CNC(=O)C(=O)N(C)C)OC 44577,N1(C(C(C)OC)=O)CCN2CCN(C(=O)C(C)Cn3cccn3)CC2C1 44578,c1(OC(C)C)ccc(C(=O)Oc2ccc(C(C)(C)C)cc2)cc1.C1(=O)CCO1 44579,N1(C(C(COC)(F)F)=O)CCCCC(NC(c2cnn(C)c2C)=O)C1 44580,N1(C(CN2CCN(C)CC2)=O)Cc2nccn2CC(NC(C2CCSCC2)=O)C1 44581,c1(CC(=O)NCC(c2ccccc2)NC(CC2CC(OC)C2)=O)ccc(Cl)nc1 44582,C1(NC(c2nccc(CNC(C(C(=O)OC)OC)=O)c2)=O)CCC2(CC1)CC2 44583,N1(C(CC2CC(OCC)C2)=O)CCC(CC(N2CCCC2CF)=O)C1(C)C 44584,N1(C(=O)NCC2CC(OC)C2)CCCC(Cc2nn[nH]n2)C1 44585,C(CCCCCC)(C(=O)OC)N1CCC(C(=O)NOCCCCF)(CC#C)C1 44586,N1(C(c2ccc(CSC)cc2)=O)CC(NC(=O)COC(C)C)C2(CC2)C1 44587,C12(C(=O)NC(C)C(C)NC(c3ccc(O)nn3)=O)CCCN(CCC1)C2 44588,C(CC(C(=O)NCc1ccc(CO)o1)NC(=O)CC(O)c1ccccc1)OC 44589,CCC(C)(CNC(=O)CCC1OCCO1)C(=O)NCCCC1CCCCO1 44590,O=C(C1=CCOC1)NCC1CN(C(=O)COc2ccc(F)cc2)C2CC12 44591,C(=O)(CCCC(=O)C1CC1)NCCCNC(Cc1cc(C)sc1Cl)=O 44592,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44593,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccnc(C)n2)=O)CC1 44594,N1(C(C2N(Cc3cc(SC)ncn3)CC2)=O)CCCCCCC1C 44595,C(CNC(=O)C(=O)C(C)C)(CC(=O)N(C(CO)C1CC1)C)OC 44596,CCC(C)C(C(=O)NC)NC(C)=O.C12CC(=NO1)C(=O)NC(C)CNC2=O 44597,c1(C(=O)NCC23CC2CN(C(=O)Cc2nc[nH]n2)C3)cc2ccc(F)cc2[nH]1 44598,CC(CC(F)(F)F)C(=O)NCC(C)(C)CN(C(=O)C(C)CC(C)(C)C)C 44599,c1(C2C(C(c3c(C)nsc3Br)Nc3n(CC)nnn3)C2)ccccc1OC(F)F 44600,C1(C(=O)NC(c2ncccn2)CCC)CCN(C(=O)CS(=O)CC)CC1C 44601,c1(C(N2C(C)CC(NC(C(CC)(C)O)=O)C2)=O)cc(C)cc(Br)c1 44602,CCC(O)C(C)(C)C(=O)NC1CC(C(=O)NCC2(CO)CCN(C)C2)CC1O 44603,C(=O)(CS(=O)CC)N1CC(C(N)=O)(CNC(c2ccc(SC)o2)=O)C1 44604,c1(C(=O)NC2C3CC2N(C(=O)C(F)OC(F)(F)F)C3)cc(F)ccc1F 44605,N1(C(C2N(C(CCN(CCC)C)=O)CC2)=O)CCCC1CC(N)=O 44606,CC1CC(NC(=O)CCc2ccccc2O)CN1C(=O)C(N)=O 44607,N1(C(C2N(C(c3[nH]cc(C)c3)=O)CC(C)C2)=O)CCC(O)C(C)C1 44608,CC1(CNC(=O)C(C2CCOC2)NC(c2ccccn2)=O)CCCOC1 44609,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44610,C1(C(=O)O)C(CNCCC(O)c2cccs2)C1(F)F 44611,C1(CN(C(C(c2ccccc2)N(C(C)C)C)=O)C)CCCN1C(C1CN(C)C1)=O 44612,N1(C(c2cc(C)oc2C)=O)CC(C)(C)CC1C(=O)NCC1CC(C2CC2)=NO1 44613,N1(C(COC2(C)CN(C(C(C3CC3)OC)=O)C2)=O)CCCNC(=O)CC1 44614,O=C(C1=NOC(CNC2C(C(=O)N(CCO)CCO)C2)C1)NC1CCOCC1 44615,N1(C(=O)CC2CCC3CC23)CC23CCCC2(C1)CN(C(c1ccnnc1)=O)C3 44616,N1(C(c2c(I)ccnc2Cl)=O)CCN(CC(N2CCCCC2)=O)C2CC12 44617,C(CS(=O)(=O)CC(=O)NC(C)(C)CC=CC(=O)NCCCN(C)C(C)=O)OC 44618,CC(CC(C)(F)F)C(=O)NCC=CCNC(=O)CCCc1nncn1C 44619,c12ccc(cc1)NS(=O)(=O)NC2.N1(CCC)CCC1 44620,C(=O)(C(C)CC1CC1)NCCCN(C(c1ncoc1C1CCC1)=O)CC 44621,C=CC(C)(C)CCCN=c1cc(C)nc(N2CCN(c3cnn(C)c3)CC2)[nH]1 44622,C1(NC(c2cccc(C3CCC3)c2)=O)COC2(CNC(C3CS(=O)(=O)C3)=O)CC1C2 44623,C1(N(C(c2cc(C3CCC3)no2)=O)CC)CCCN(C(=O)C(F)CC2CCOC2)C1 44624,Cc1ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(=N)[nH]c2)c1 44625,N1(C(Cc2c(C)cccn2)=O)CCCC(C2CC2NC(c2cc(C(N)=O)cs2)=O)C1 44626,N1(C(CC2N(CC)CCOC2)=O)CC(CNC(=O)CNC(C)=O)OC2(CCC2)C1 44627,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(F)(F)F)s1 44628,C1(C(=O)NC2CCCOC2)(CC)CCCN(C(c2ccc(C(N)=O)cc2)=O)C1 44629,C=C1CC2(C1)CC(C(=O)NN1CC(C)NCC1=O)C2.c1(OC)cccc(OC)c1 44630,C#Cc1cc(C(N2CC(C)N(C(C3(OC)CCCC3)=O)CC2C)=O)cc(F)c1 44631,N1(C(c2cncc(C)n2)=O)CCC(NC(c2ccc(Cl)cc2)=O)C1(C)C 44632,C12(NC(=O)Cc3nc(F)c(F)cc3F)CCCN(C(c3cnsc3)=O)CC1C2 44633,C1(NC(C(COC)COC)=O)CN(C(c2cnc(O)cc2OC)=O)CCC1C 44634,N1(C(COCCC=C)=O)CCC(CC)(OCCCCC)CC1 44635,C(N(C1CC1)N1CCCCC(F)(F)C1)c1ccc(CC(F)(F)F)cc1 44636,CCS(=O)(=O)c1cccc(NC(=O)NCC2CCCC2n2cccn2)c1 44637,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44638,CC(CC(=O)N1CCC(=C(F)F)CC1)C(C)(C)C.N12CC3CCC(C1)N3CC2=O 44639,c1(SC(C(=O)NC(C)CNC(=O)C(O)CC2CCCC2)C)ccc(F)cc1 44640,N1(C(CCCCN(C)C)=O)CC2CCCC(CNC(=O)Cc3nnc(O)s3)C2C1 44641,c1(CC)cc(C(N2CCC(NC(c3cc(Cl)n[nH]3)=O)C(F)C2)=O)ccc1OC 44642,C(c1ccccc1F)=CCC(=O)NCC1(O)CN(C(c2ccc(C#N)o2)=O)C1 44643,C(=O)(C1OCCc2c(Br)cccc21)NCC(CN(C(C(CC)(F)F)=O)C)C 44644,C(=O)(C#CC1CCCCC1)NCCN(C(C)C)C(C1CCC(C)S1)=O 44645,c1(CC)cc(C)nc(N2CCC(CCNC(c3ccc(C(C)=O)[nH]3)=O)CC2)n1 44646,CCCCCCC(=O)NCC1CCC(F)(CNC(=O)C(O)C(C)C)C1 44647,CC(N=[N+]=[N-])C(=O)NC(c1ccnn1C)C(=O)NCCC1CCCC1 44648,CCCCC(O)C(=O)N1CCC(CO)C(NC(=O)CCC2CCC2)C1 44649,C1(Cc2c[nH]nc2C)CN(C(C2CC3CCC2CC3)=O)CCN1OCC 44650,c1(CC)cc(S(=O)(=O)NC2CCCC2CCCC(=O)O)n(C)n1 44651,c1(C(=O)NCC(C)N(C(C(CCOC)C)=O)C)cc(OC(C)C)ccc1Cl 44652,c1(OC)cc(C)ccc1OCCC(=O)NC(C)CCCNC(c1c[nH]c(=N)s1)=O 44653,c1(C(=O)NC2CN(C(CC(C=C)(C)C)=O)CC(C)C2)c(F)ccc2n[nH]cc12 44654,O=S(=O)(c1c[nH]ccc1=NCC1COCO1)NCC1COc2cscc2O1 44655,Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1(CCNC(C2CCC(=O)O2)=O)CC1 44656,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44657,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44658,c1(C(=O)NC2C(CNC(C(C)n3cnnn3)=O)C2)c(O)nnc2c1COCC2 44659,C12(NC(c3c(C)nc(CO)nc3)=O)CCN(C(c3cccc(Br)n3)=O)CC1C2 44660,N1(C(C2=C(C#N)CCC2)=O)CCN(C)CC(CO)C1.c1(C(C)=O)ncsc1CN 44661,C=CC(F)(F)C(=O)N1CCC1CNC(c1ccc(C(C)(C)C=C)cc1)=O 44662,N#CC1CC12CCN(C(C1(F)CCN(C(C3CCNC3=O)=O)C1)=O)CC2 44663,C12(CNC(CCC(=O)NC)=O)CCC(CNC(C3CC3(C)C(C)C)=O)(CC1)OC2 44664,c1(CC(=O)NC)ccc(C(=O)NCCC(O)CNC(c2cccn2C2CC2)=O)cc1 44665,c1(C(C)=O)cncc(C(=O)NC(CNC(=O)CCc2c(C)noc2Cl)CO)c1 44666,N1(C(c2ccn(CC)c2C)=O)C2CCC1C(NC(c1ccnc(Cl)c1N)=O)C2 44667,CC(C)(C)CCCC(=O)N1CCN(C(=O)CC2CC2(C)C)CC1CC(F)F 44668,c1(CN(c2c(Br)cnn2C)C(=O)Nc2n(CC)ccc2)ccc(F)cc1 44669,c1(OC(C)C)nccc(C(=O)NCC2CCCC2NC(C2CNC(=O)C2)=O)c1F 44670,CC(C)C(O)C(F)(F)C(=O)NCCC1CN(C(=O)C(C)O)C1 44671,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44672,C1(CC)C(=O)O1.C(C(F)(F)F)=CC(=O)OC 44673,Cc1cc(=NC(C)c2ccc(C)o2)[nH]c(=NCCC(=O)NCP(C)(C)=O)[nH]1 44674,C(C1=CCC2CC1C2(C)C)(CCCC=C)c1nnnn1Cc1cccc(OC)c1 44675,N1(C(CCc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44676,C1(CC)(NC(C2CCCCC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 44677,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2C)=O)cnc2n1CCCC2C 44678,N1(C(c2c(OC)ccnc2)=O)CC(C(=O)NOCCCC(F)(F)F)C(F)(F)C1 44679,c1(CNC(C(CC)N(C)C)=O)ccccc1CNC(=O)CC1CC2CC2C1 44680,c1(C(C)=O)c(C)[nH]c(C(N2CCC(O)C(NS(=O)(=O)CCCl)C2)=O)c1C 44681,c12ccccc1C(=O)NCC2OCC.C(=O)(CCC(=O)OC)NC(C)C 44682,c1(N(C2CN(C3CCCCC3CO)C2)C(c2ccco2)=O)ncc2cccnc2n1 44683,C1(Cn2cc(C3N(C(Cc4nc(C)c(C)s4)=O)CCC3)nn2)CCCCC1(C)C 44684,n1(CCCC)ncc(C(N2CC3C(NC(c4n[nH]c(C5CC5)n4)=O)C3C2)=O)c1C 44685,c1(CCC(=O)N(C(C)C)CC2CCCN(C)C2)cccc(-c2cccc(F)c2)c1 44686,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(c1conc1C)=O 44687,c1(OC(C(C)C)C(=O)NCCC2CCCN2C(=O)C2CC2)ccc(F)cc1F 44688,c1(CC(=O)NC2C(NC(C3(COCC)CCC3)=O)CCC2)ccc(Br)nc1 44689,c1(C(=O)NCC(CCNC(CCCOCCC)=O)O)c(F)cc(O)cc1F 44690,CC(C)(C(=O)N1CC2CCC(NC(c3ncsc3Br)=O)(C2)C1)S(C)(=O)=O 44691,c1(C(N2CCC(CCNC(c3occc3Br)=O)C2)=O)ccc2c(c1)OCCC2 44692,C1(CNC(c2cc(C)n(C(C)C)n2)=O)CN(C(=O)Cn2cccc2)CC12CC2 44693,CCC(F)(CNC(=O)CC1CCCCN1C(=O)CCCOC(C)=O)CC 44694,N1(C(CCc2ccc(C)s2)=O)CCC(C)C1CNC(C1CCCN1S(C)(=O)=O)=O 44695,Cn1cnc(C=CC(=O)NCC(c2ccccc2)NC(C2(C(N)=O)CCC2)=O)c1 44696,C1(CNC(C2(C)CC2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1O 44697,n1(CC)nccc1C=CC(N1CC(NC(=O)Cc2cn[nH]c2)C(C)C1)=O 44698,C(=O)(C1=COCCO1)NCC1CCN(C(C(CC)=CC)=O)CC1 44699,C1(CNC(c2cc(-c3ccoc3)[nH]n2)=O)CN(C(C2C3CCC2CC3)=O)CCO1 44700,c1(CC)c(C(N2CC(N(C(=O)C(C)(C)COCC(F)F)C)C(F)C2)=O)csc1C 44701,Cc1nc(Cl)ccc1C(=O)NCC(O)CNC(C1CCC(O)CC1)=O 44702,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCC(=O)C4)=O)CC3O)cc12 44703,C1(C)(C(=O)NCCN(C(c2nccc(N)c2Cl)=O)CC)CCC(F)(F)C1 44704,c1(C(=O)NC2C(NC(C3N(C=O)CCC3)=O)CCC2)c(F)c(F)c(F)c(F)c1F 44705,c1(C(CNC(C(C)(C)N(C)C)=O)NC(C2CCCC2O)=O)ccccc1F 44706,c1(C(N2CCC(O)(CN(C(=O)CSCC(N)=O)C)C2)=O)oc2ccccc2c1Cl 44707,C1(CNC(=NC)NCCOCCS(N)(=O)=O)Cc2ccccc2C1 44708,c1(C(=O)NC(C(C)NC(=O)Cc2cnoc2)CO)cccc(N)c1N 44709,N1(C(C(C)CC(N)=O)=O)CCOC2CCCC12.n1(CCCO)cc(C(C)O)nn1 44710,Cn1nnc2cc(C(=O)NCC34CCCC3CCN4C(c3cnc[nH]3)=O)ccc12 44711,N1(C(CSCCNC(C2C3CC(=O)CC32)=O)=O)CCN2C(=O)NCC2C1 44712,c1(C(=O)NCCCC2(NC(C(C(C)C)CO)=O)CC2)cccc2ncnn12 44713,CC1C(C(=O)O)CCCN1Cc1cc(Br)no1.C(=O)CCCCCn1ccnn1 44714,c12ccc(c(F)c1Br)[nH]c2=O.n1(SCC)cc(CNC2CC(CC)C2)nn1 44715,n1(CC)ncc2c1CCCC2N.c1(N)nccc(N2CCC(N(C)C(C)C)CC2)n1 44716,C1(CN(C(=O)CSc2ccccn2)C)CC(NC(C2CC(C#N)C2)=O)C1(C)C 44717,N1(C(C(CCSC)OC)=O)CCC(C)(C)C(CNC(=O)C(C)(C)C2CCCC2)C1 44718,c1(C(N(C2C(C)CCN(C(=O)C=Cc3cccs3)C2)C)=O)cc2scc(Cl)c2[nH]1 44719,CC1OC2(C(N3CC=C(CNC(c4ccnn4C4CC4)=O)CC3)=O)CCC1CC2 44720,c1(C(=O)NC2(CO)CCN(C(c3cc(C(C)=O)on3)=O)C2)noc2ccccc12 44721,C1(C2CCN(C(=O)C3=C(C)CCC3)C2)(NC(C=CCC)=O)CC1 44722,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CCF)CC 44723,C(CC(F)(F)F)NC(c1cn(CCO)nn1)=O.C12(CC1)C(C)N(C1CC1)C2=O 44724,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(=O)Cc2cc(C)ns2)CC(C)(C)C1 44725,CC(CC1CCCO1)C(=O)NCC1CCCN1C(c1cc(C(F)F)cs1)=O 44726,C1(SC)COC2(CCN(Cc3ccc(C)nc3Cl)CC2)C1.c12cc-1cc(F)c2 44727,c1(C(=O)NC(C2CCOC2)C)coc2c1CN(C(c1[nH]ccc1C1CC1)=O)C2 44728,C(C(CCOC1CCCO1)OC)NC(C(C1CCCC1)OC)=O 44729,C1(C(=O)OC2CCCCC2)CC(O)CN1C(=O)C1CC1 44730,N=c1[nH]c2ncc(C(=O)NC3(C4CCCN4C(C4CCCS4)=O)CC3)cc2s1 44731,Cc1occc1CC(=O)NC(c1ccccc1)C(=O)NC(C)Cn1ccnc1 44732,C(=O)(C(CCSC)NC(c1ccco1)=O)N(CCNC(C)=O)C 44733,O=C1CCC(CCC(N2CCCC2CNC(=O)CC2CSC2)=O)N1 44734,C1(c2cn(CC3N(C)CCCC3)nn2)CCOCCN1Cc1cc(F)ccc1N 44735,C1(CC=C)(C(=O)NC2CC(CO)N(C)C2)CCCN1C(C)=O 44736,N1(C(Cn2ncc(CC)c2)=O)CC(C)CC1CNC(C1CC1F)=O 44737,c1(C(=O)NC2CC(NC(c3c(C)cc(C(F)F)o3)=O)C2)ccc2ncc(=O)[nH]c2c1 44738,c12ccc(cc1)OCC(=O)N(C)CC(CC)NC2=O.C1(C(=O)NC)CC2CC2C1 44739,N1(C(C2(CC)COC2)=O)CC2COCC(C1)C2NC(C1C2COCC12)=O 44740,CCCCC(C(=O)NCCCC(C)(C)NC(c1cccc(CF)c1)=O)NC(N)=O 44741,C(CC(F)(F)Cn1cc(Cn2cccn2)nn1)NC(Cc1n(C)cnc1)=O 44742,c1(N(C=O)Cc2n(C(C)C)ncc2)ccc2c(c1)ncn2C 44743,C1(NC(CCOC)=O)CCOCC1NC(=O)CC1CC(C)(C)C1 44744,N1(C(C(CC)=CC)=O)CCC(NC(c2sc(F)cc2C)=O)C(CC)C1 44745,C(CC(C)(C)C)(C(=O)N(CC1CC1)CC1CC1)NC(C1C(CC(C)(C)C)C1)=O 44746,Cc1nc(CC(N2CCC(N(C(=O)CCOC3COC3)C)C2)=O)n[nH]1 44747,C1(C(N2CC(NC(C3(C=C)CC3)=O)(COC)C2)=O)CC2CCC1CC2 44748,C1(O)(C(=O)Nc2cnn(CCC3CCCC3)c2)CCN(Cc2ccccc2I)CC1 44749,C1(C(=O)NC(C(=O)N(C2CC3CC3C2)C)C2(O)CCC2)(CO)CCCO1 44750,C(C)(CCCC(=O)N(CC1CCC1)CC1CC1)NC(c1c(CC)cc[nH]1)=O 44751,Cc1ccc(CC(=O)NC2CCN(c3cccc(C(F)(F)F)n3)C2)c(C)c1 44752,c1(C(=O)NCCC(C)N(C(C(C)OCCC=C)=O)C)ccc(C(C)C)s1 44753,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 44754,C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCC2CN(C(C3(F)CCCCC3)=O)CC12 44755,CN1CCC(F)(F)C(CC23C(NC(=O)OC(C)(C)C)C4CC2C3C4)C1 44756,C1(C(=O)NCC(C(N2CC3C(COC)C3C2)=O)(C)C)CCC(C)=C(C)C1 44757,CC(CCNC(=O)CCCCN(C(=O)CC1CC1)C)CCO 44758,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 44759,C1(C(=O)NC(c2c(F)cccc2F)C)CC(c2cccc(F)c2)=NO1 44760,N1(C(c2oc(C)c(CO)c2)=O)CCC(C2CC2)(CNC(c2ccc(CO)s2)=O)C1 44761,c1(NC(C2CN(C(c3ncc[nH]3)=O)CCN2)=O)nc2c(s1)COCC2 44762,CC1CN(C(c2c(F)cncc2Br)=O)CC2(CCN(C(=O)CO)C2)O1 44763,Cc1ccc(Nc2nnc(NC(=O)NC3(Cc4ccc(Cl)cc4)CC3)s2)cn1 44764,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)N(CC(F)(F)F)C)=O)C(O)C1 44765,Cc1cc(CC(=O)NCC2(CN(C(=O)C(C)C3CCOC3)C)CC2)cc(F)c1 44766,CC(C)CC(C)(CNC(=O)CC1CC1(C)C)NC(C1(C(F)(F)F)CCC1)=O 44767,N1(C(CN2CCC(OC)C2=O)=O)CCN(Cc2cccc(CC)c2)CC(O)C1 44768,C(=O)(CCCCC(C)C)N1C2(C(=O)NCC3(COC)CCC3)CC2CC1 44769,N1(C(C2C(CC)OCC2)=O)CCCC(C2CC2NC(=O)Cc2cc(OC)no2)C1 44770,c1(C(N(CCNC(c2c(SC(C)C)nccc2)=O)C2CC2)=O)cc(=N)[nH]c(Cl)n1 44771,c1(C(=O)NC2(CNC(CCOCC)=O)CC2)cccc2nn[nH]c12 44772,c1(OC)ccc(C(C2CCC2)Nc2cccc(-c3cnn(C)c3)c2)c(Cl)c1OC 44773,c1(C(=O)NCCCC(C)NC(C(C)Oc2cccc(C)c2)=O)cc(F)c(N)cc1F 44774,c1(-c2cncc(C)c2)cc(C(=O)NCc2ccc3c[nH]nc3c2)cc2[nH]ccc12 44775,C1(NC(c2cc(SC)oc2)=O)CC2CCC1CC2NC(c1cc(C)nc(C)c1)=O 44776,c1(OC)ccc2onc(CC(N3CCN(C(c4cn[nH]c4)=O)CCC3C)=O)c2c1 44777,C=C(C)C1OCCC1CNC(C1CN(C(c2cnc(C)cn2)=O)CC1CC)=O 44778,c1(CNC(=O)NCC2C(c3n(C)cnn3)CCC2)cc(Cl)cc([N+](=O)[O-])c1 44779,C(C(C)(C(=O)N1CC(NCCCC(=O)OC)C(O)C1)OC)OC 44780,c1(OC)ncnc(OC)c1CN1CC2CC1C2C(=O)Nc1ncc(Cl)s1 44781,C1(NC(C=Cc2c(C)cccc2)=O)CC1C1CCN(C(C2(C)COC2)=O)CC1 44782,CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CC(CNC(=O)CC2(C)CCS(=O)(=O)N2)C1 44783,C1(C(C)C)N(C(=O)CCCn2cc(C(C)N(C)C)nn2)CC12CCC2 44784,C(c1cccnc1)=C(C)C(=O)NCCN(C1CCCC1)C(=O)CC1CCN(C)C1 44785,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(C2CC(F)(F)C2)=O)CC1 44786,N1(CCC#N)CCC(CCNc2nc(-c3ccco3)no2)CC1 44787,C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCCNC(C)=O)=O)C(C)C1.CC=O 44788,C1(N=c2cncc(Cl)[nH]2)(CNC(=O)CN2CCCCC2=O)CCOC1 44789,OCC(F)CN=c1[nH]c(N2CCN(C(=O)C3CC3)CC2)nc2c1COC2 44790,n1(CCOCC(CNC(=O)CCC2CCCO2)O)cc(C2CC2)nn1 44791,CCCCC(O)C(=O)NC(CNC(C1CC1C(C)(F)F)=O)C1CC1 44792,C1(CNC(C(C2CN(C(C(C(=O)OCC)F)=O)C2)O)=O)OC(=O)NC1(C)C 44793,CC(C)CCC=CC(=O)NC(C)C(=O)NCC(C1CC1)N(C)C 44794,N1(C(C(C)OCC(F)(F)F)=O)CCC(N(CCO)C(c2cncc(N)c2)=O)CC1 44795,N1(C(CC(CC#C)c2ccccc2)=O)C2CCC1CN(C(=O)CC(O)CC(C)C)C2 44796,N1(C(CC)C)CCN(C(=O)C(CNC(C2(C)CC(C)(C)C2)=O)CC2CC2)CC1 44797,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(c2cc(Cl)c[nH]2)=O)CC12CC2 44798,n1(CCC(=O)NCc2ccnn2-c2ccccc2)cc(CCc2cc(Cl)cs2)nn1 44799,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 44800,N1(C(C2CC(CC)C2)=O)CCCCC1CNC(=O)C(O)Cc1ccccn1 44801,NS(=O)(=O)CCN=c1[nH]c(NCc2ccc(S(C)=O)cc2)nc2c1CCC2 44802,c1(C(N2CC(F)(C(=O)Nc3c(C(=O)OC)nccc3)C2)=O)cc(Cl)c(O)cc1F 44803,N1(C(C=CC)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1C1CC1 44804,CC1(C(=O)NCC2CCCCN2C(=O)CC2CCC2)CCC(F)(F)CC1 44805,CC1CCN(C(=O)CC2C=CCCC2)C1C(=O)N(C)CCC1CCCC1 44806,C1(CN2CC(c3cn(C(C)COc4ccccc4)nc3)OCC2)CCC(C)(C)CC1 44807,N1(CC#N)CCCC1C1CCCCN1C(c1cccc2nc(O)[nH]c12)=O 44808,C(CC1CC1)(C(=O)NCCC1CCC(NC(C2(CC(F)F)CC2)=O)C1)OC 44809,c12ncnc(Cl)c1CC1(NC(c3cc(C4(C)CC4)n[nH]3)=O)CCN2C1.CC=O 44810,C1(C(=O)NC(C2C(C(=O)OC)C2)C)CC2(CCN(C(C3(C)CCC(=O)N3)=O)C2)C1 44811,N1(C(C(C)N)=O)CC(CCO)C2(CCNCC2)C1.C1CN1.C1CO1 44812,c12cc(OC)cc(OC)c1SCC(=O)N(C)CC(C)N(C)C(=O)C2.C=CCSC 44813,C1(NC(C=CC=CC)=O)CC2CC(NC(c3ccnc(-c4ccccn4)n3)=O)C1C2 44814,N1(C(c2c(C)cc(F)s2)=O)C2CCC1C(C(=O)Nc1nnc(O)cc1O)C2 44815,c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)C(CO)C2)ccc2nncn2c1 44816,C(=O)(C1=CS(=O)CCC1)N1CCCC(CC=C)(NC(=O)CCC(=O)NC)C1 44817,Cc1nn(C)c(-n2cccn2)c1C(=O)NC1CCCN(C(=O)C(Cl)=CCl)C1 44818,N1(C(C2CCC(C)(C)O2)=O)CC2(CCCN(C(C3CCCC4(CCC4)O3)=O)C2)C1 44819,c1(C(N2CCCCCC(NC(CC=CC=C)=O)C2)=O)cc2cc(Br)cn2cn1 44820,c1(CCC(N2CCN(C(CS(C)(=O)=O)=O)CC2CF)=O)ccc(S(C)(=O)=O)cc1 44821,N1(C(C2C(C(=O)OC)C=C2)=O)CCC2(CCCN2C(C23CCCC2C3(F)F)=O)C1 44822,c1(N2CC(c3ccccc3)(NC(C3(C)C=CCC3)=O)C2)cc(C)c([N+](=O)[O-])cc1F 44823,c1(NC(C(CCC)NC(c2sccc2CO)=O)=O)c(C)cccc1F 44824,c1(C2(C(N3C(c4onc(C)n4)C(C)(C)C3)=O)CC2)c(Cl)cccc1Br 44825,CCCC(C)CCCC(=O)NC1CCC(C)N(C(=O)C=Cc2ncc[nH]2)C1 44826,C(=O)(C#CC1CCCOC1)N1C(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCC1 44827,C1(c2ccc(C(=O)Nc3nccc4c(Br)c[nH]c34)cc2)CC2(CO1)CC1(C2)OCCO1 44828,N1(CCC)CC2(CCC(C(N(C(C(=O)Nc3ccccc3C)C)C)=O)C2)C1 44829,S(=O)(=O)(c1cccc(N2CCOC(C3CC3(F)F)C2)n1)N(C)CCn1ccnn1 44830,C1(N(C(c2c(COC)cc[nH]2)=O)C)CCC(NC(C2CC3(CC3)CO2)=O)CC1 44831,N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CCCN2C(=O)C(F)C(F)(F)F)C1 44832,CC1CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)Cc1n[nH]c(=N)s1 44833,c1(C(N2C(C)CC(NC(c3ncn(CC)c3)=O)C2)=O)ccc2sccc2c1 44834,c1(CC)nc(C(=O)NCCCCN(C(=O)CN2CCSCC2)C)cs1 44835,C1(NC(CC2N(C(CCC(C)=O)=O)CCCC2)=O)CC2(COCCO2)C1 44836,S(=O)(=O)(CCC(F)(F)F)N1CCCC(N(c2ncc(C#N)cc2Br)C)C1 44837,N1(C(c2ncn(C)n2)=O)CCN(C(c2ccccc2F)=O)CC1CO 44838,C1(NC(c2cc(C)c(C)nc2)=O)C2CC3CN(C(=O)CC(C)(C)C(F)F)C1C3C2 44839,N1(C(c2[nH]cc(C#N)c2)=O)CC2(CCC2)CC1CN1CCCC1.C12(CCC1)C(=O)N2 44840,N1(C(c2c(C)n[nH]c2C)=O)CC2(CCC2)CC1CNC(C1(F)CC=CC1)=O 44841,N1(c2c(OC)nc3ccccc3n2)C2CCCC1CN(C(C1CCOC1)=O)CC2 44842,C(C(=O)N(CCCCN(C(=O)CC1C(=O)NN=C1C)C)C)(C(C)C)OCC 44843,C(C(CC)(CC)C(=O)NC(c1ccccc1)CF)NC(C(CC=CC)C)=O 44844,c1(N2CC(C(C)NC(C3(C)CC(O)CN3C)=O)C2)ccc([N+](=O)[O-])cn1 44845,N1(C(Cc2cnc(C)[nH]2)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CCC12 44846,C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 44847,C(=O)(CCC(C)(C)NC(=O)CC1CCC(=O)C1)N(CC#C)C 44848,c1(CC(=O)NC)ncc(F)cc1F.C1(N)CCN(C(C2CCCN2C(N)=O)=O)C1 44849,C(CC(C)C(=O)N(C1CC(NC(C2CCOC2c2cccnc2)=O)C1)C)=CCC 44850,C1(CC)(NC(=O)C(Cn2cncn2)NC(=O)Cc2cnn(CC)c2)CCCC1 44851,c1(OCCOC)ncc(C(=O)NCC(O)CNC(C2CCCCNC2=O)=O)cc1Cl 44852,C#CCC(CC(=O)N1CCCCC1C1CCC1)NC(C)=O.C1(=O)C(=C)N1 44853,c1(N(C)CC2CC2Cl)nc(=NCCc2nnc3n2CCC3)[nH]c2c1CSC2 44854,CC1(C)CC(CCNC(C2(C)C=CCN2C(=O)Cc2ccnc(O)c2)=O)CO1 44855,CCCC(CCCNC(c1c(OC)noc1C1CC1)=O)NC(=O)C(CC)C(C)C 44856,CCP1(=O)CCN(C(=O)CC2CCCCC2C)CC1 44857,c1(C(C)CNC(=O)Cn2cnc(-c3cccs3)n2)cccc(Cl)c1 44858,N1(C(c2nc(SC)sc2)=O)CC2CN(C(=O)CCC(=O)N(C)C(C)C)CC2(C)C1 44859,C1(CNC(CCC=C=C)=O)CC(C)CN(C(=O)C(C)CCC)C1 44860,C1(NC(C(CC=C)CNC(C2CCN2CC)=O)=O)CC12CCCCCC2 44861,C1(NC(=O)Nc2c(Cl)ccc(C)c2)CCC(F)(CNC(=O)Nc2ccccc2)CC1 44862,c1(OC)ccnc(C(=O)NCCCN(C(C2CCOC(C)C2)=O)C(C)C)c1O 44863,C(=O)(C(C1=CCC(C2CCOCC2)O1)OC)NC(COCC=C)COC(C)C 44864,N1(C(C(CCNC(C2OCCO2)=O)OC)=O)CCOC(C)(C)C1C 44865,C1(NC(c2nc(C)oc2)=O)CCCCN(C(=O)COCC2CCCC2)CC1 44866,Cc1cc(F)cnc1C(=O)NCC1CN(C(=O)CCn2ccnc2)CC1O 44867,N1(C(COCCC)=O)CCOC(C)(CNC(=O)CNc2ccnc(C(N)=O)c2)C1 44868,C(C)(C(O)C(=O)NCCCC1(NC(c2ccncc2)=O)CC1)OC 44869,CCCCCC(C)(C)CNC(=O)C=CC=CCOC.C1(=O)C(C(C)CC)N1 44870,C1(C(N2C(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 44871,N1(C(C(CC)=CCCC)=O)CC(=O)CC1C(=O)NCc1cc(O)ncn1 44872,c1(C(C)NC(=O)C(=O)NC2NCCCC2C(F)(F)F)ccc(F)c(Cl)c1 44873,CC1(NC(c2ccnc(OCCO)c2)=O)CCCN(C(C2C=CC=CC=C2)=O)C1 44874,c1(C(CNC(C2(CCO)CC2)=O)NC(C2(CC)C=CCC2)=O)ccccc1SC 44875,C(=O)(C(C)(C)CN1CCCCC1)N(CC(=O)N(C1CSC1)C)CC 44876,c1(C(N2C(CNC(C(C)OCCCCCC)=O)CC2)=O)nn(C)c2c1CCC2 44877,c1(C(=O)NC(c2nc[nH]n2)CC)ccoc1CNC(C1CC1(C)C(F)F)=O 44878,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2COC2)nn1)=O 44879,CC(C(=O)NCC(C)CN(C(=O)COc1ccc(OC)cc1)C)S(N)(=O)=O 44880,c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCC2)cnc2scc(C)n2c1=O 44881,C(CN=c1[nH]c(C)ncc1F)(CC(C)C)NC(COCc1ccc(C)s1)=O 44882,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 44883,C(CC(=O)CCO)N(C(C=CC)=O)CCN(CCO)CCN(C)C 44884,c1(NCCCC)ccc(C(=O)NC2(C)CC(NC(=O)CC3CC3)C2)cc1[N+](=O)[O-] 44885,c1(C(=O)NCC2(NC(C3C(C)(CC)C3)=O)CC2)ccc(Br)c(F)c1 44886,N1(C(C2C(OCC)C2)=O)CC2(CNC(=O)C=Cc3ccnn3C)CC(F)(C1)C2 44887,CC1(C)CCCCC1(N(C=O)Cc1cccc(Cl)c1F)CN 44888,CC(C(=O)NC(CNC(c1c(F)cncc1Cl)=O)C1CCC1)C(F)(F)C(F)F 44889,N1(C(C2(O)CC(C)(C)C2)=O)CCC(NC(c2[nH]nc3ncccc23)=O)C(F)C1 44890,CCCCCCCCCC(C(=O)NCC(=C)C)N(C1CCCC(OC)(OC)C1)C 44891,C(C1CCCc2cccnc21)NC(NCC)=NCCOCCNS(C)(=O)=O 44892,C1(NC(c2cc(OC)ncc2Cl)=O)CN(C(C2CC=CCC2C)=O)CC(F)(F)C1 44893,c1(C(=O)NC2(C)CCN(C(C(CCC)OC)=O)C2)ccc(N)c(C)c1Cl 44894,CCCCC(O)CNC(=O)COC(C1CCCC1)C1CC1 44895,c1(N(C(C2CCCN(C(=O)CN3CC(=O)NC3=O)C2)=O)C2CC2)cnccn1 44896,C1(C(N2CC(CC)OCC2)=O)C2CCN(C(C34CCC(C3)C4)=O)CC12 44897,CN1CCN(C(=O)CC2(NC(=O)CC3CC4CC4C3)CC2)CC(O)C1 44898,c1(C(=O)NCCOCC=C)cc(-c2cc(OC)c(C)cc2C)c2cn[nH]c2c1 44899,c1(C(N(C2CCN(C(C(C)(C)OC)=O)CC2)CCO)=O)ccc(C(C)C)cc1O 44900,c1(C(C(=O)NCC(=C)CCNC(=O)C(C)CO)(C)C)ccc(Br)cn1 44901,Cn1cc(C(F)(F)F)cc1C(=O)NC1(CCNC(=O)CC2C(=O)NN=C2C)CC1 44902,C(C(F)C(=O)N1CCCC1C1(OC)CC1)N(C(COCC(=O)NC)=O)C 44903,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cncn2)CC1C1CC1 44904,N1(C(CN(C(c2cccc(C#N)c2)=O)CC)=O)CC2(CC(F)C2)C1 44905,C(=O)(CCCNS(C)(=O)=O)N1C(CN(C)C(C2(c3ccccc3)CCC2)=O)CC1 44906,N1(C(C2CCC(CC)CC2)=O)CCC(F)(F)C(Nc2ccc3ncsc3c2)C1 44907,c1(OC)cc(C(N2CC(CNC(c3cn(C)nc3OC)=O)C(C)C2)=O)ccc1F 44908,C1(O)(CNC(=O)CCCc2ncco2)CCCN(C(C2CC2CC(F)(F)F)=O)C1 44909,C#CCCC(O)C(=O)NCCC1CCCCN1C(C12CC(CCO1)C2)=O 44910,N1(C(C2C(CN(C)C)C2)=O)CCC(CNC(C2CN(N3CCOCC3)C2)=O)CC1 44911,C(=O)(C(CC1CC1)NC(=O)CCc1ccoc1)NCC1(C(C)C)CCC1 44912,CC1(C)CC(CNC(c2cccnc2)=O)N(C(=O)Cc2cncnc2)C1 44913,c1(CC(=O)NC2C(NC(C3C(C#N)CC3)=O)CC2)ccc(C2CCCCC2)cc1 44914,c1(CC(=O)OC(C)C)ccc(NCCCCNC(c2nc(=O)n(C)[nH]2)=O)nc1 44915,C(=O)(C(C(C)NC(=O)CCCn1cccc1)C(C)C)NC(C1CCC1)CC 44916,Cc1c(C(=O)NCCCN2CCC(=O)NC2=O)c(=O)oc2cc(N)ccc12 44917,Cc1cc(C(N2CC3(CCC3NC(C3CCSCC3)=O)C2)=O)n2nc(C)cc2n1 44918,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(c1csc(F)c1)=O 44919,CCC(CC(=O)NC1CC(CC(=O)N(CC(O)(CC)CC)C)C1(C)C)C(F)F 44920,c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)ccc(Br)c(Cl)c1 44921,C1(C(=O)NCC(CC(=O)NCC(C)(C)OC(C)C)C)CC2COCC2C1 44922,N1(C(C(=O)NCC2CC2)C2=CCCCC2)Cc2nccc(Cl)c2C1 44923,c1(CC(C(=O)NC(CCCNC(c2occ(C)c2)=O)C)C)c(C)n[nH]c1C 44924,c1(C(=O)NCC(C)NC(CCn2ncc(C)c2)=O)ccc(Cl)cn1 44925,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 44926,N1(Cc2cnc(C)n2C)CC2(CCC(C(=O)NCCC(=O)NC(C)(C)C)O2)C1 44927,C1(N(C)C(c2cccn2C)=O)CCN(C(C2(C)CCNC2=O)=O)CC1 44928,Cc1cc(-c2nn(-c3ccc(Cl)cc3)cc2C(=O)NCCC(C)C)ccc1F 44929,c1(C(=O)NC2CC2CC(C)(C)C)ccc(C)n1C.C12CCC(C1)N(CC)C(=O)C2 44930,CC#CCC(C(=O)NCC1C=CCCC1)NC(=O)CC1CCCCC1O 44931,c1(C(=O)NC2CC(CNC(C(C)CC(N)=O)=O)OCC2)ccc2c(c1)CCC2 44932,C1(C)(CNC(c2cccc(CCC)c2)=O)COCCN(C(=O)C2=CCCCO2)C1 44933,C1(CNC(C2CC23CC(O)C3)=O)CC12CCN(C(=O)CS(=O)(=O)CCO)CC2 44934,c1(CC)cc(Br)ccc1C(N1C2CCC(C2)C1C(=O)Nc1cnncc1Cl)=O 44935,CC(O)C(C)C(=O)NCC(F)CNC(C1CCCN1Cc1ccccc1)=O 44936,c1(C(=O)NC(c2cccc(C)c2)CNC(C=COC)=O)nn2c(c1C)CCCC2 44937,Cc1cc(C(N2CCC(O)(CNC(C3COCC3O)=O)C2)=O)n(C)n1 44938,C(C1CN(N2CCSCCC2C)CC1C=O)=CC 44939,c1(C(C)NCCNC(=O)NC2CC2C(=O)Nc2cnn[nH]2)ccccc1F 44940,C=CC1(C(N2CC3CC2(C(=O)N(C2CCCC2C#N)C)C3)=O)CCCC1 44941,C(=O)(C(F)C(C)(C)O)NC1CC(NC(c2c(OC)c[nH]n2)=O)C1 44942,c1(NC(=O)NC2CC2c2ccc(Cl)cc2Cl)cc(O)c(Cl)cc1Br 44943,N1(CC(=O)NCC(CNC(c2cc(CC)n[nH]2)=O)OC)CCS(=O)(=O)CC1 44944,c1(SC)ccc(C(=O)NCC(C2CC2)NC(=O)COC(C)C)cc1 44945,c1(-c2nc(CCC(C)C)nn2C(c2ccc(Cl)cc2)C)cnc2c(c1)ncn2C 44946,N1(C(C2N=C(C)SC2)=O)CCCOC(CNC(c2cc(C)n(C)c2C)=O)C1 44947,c1(C(=O)NCc2c(CN(C(CCCC)=O)C)cccc2)cc(C#N)c(N)cc1O 44948,C(=O)(C(C)CC(C)C(C)=O)NCCC1CC(C(=O)NCC)C1.C(C)(C)(C)O 44949,c1(C(=O)NCC(O)CC(=O)N2CC(NC(=O)C3CC3)C2)cc(F)cc(F)c1 44950,c1(CC)nn[nH]c1C(N1CCC(CCNC(=O)COCC2CCCOC2)C1)=O 44951,C#Cc1ccc(F)cc1C(=O)NCCOCCNC(c1cc2c(ccn2C)[nH]1)=O 44952,c1(CN(CC(=O)NC2C(CNC(CSC)=O)C2)C)cccc(C(N)=O)c1 44953,CC1CCC(C)C(C)C1NC(=O)C(=O)NCc1ccn(C(C)(C)C)n1 44954,C1(C(=O)NC(CC)CN(C)C(c2ccsc2)=O)CCCCN1N1CCOCC1.C=O 44955,C(CC(C(C)C)NC(=O)CCN(C(=O)C(C1(O)CCCC1)F)C(C)C)OC 44956,c1(NC(COC2CCN(C(CCC(C)NC(N)=O)=O)C2)=O)ccc2sncc2c1 44957,C12(C(N3CCC(CCCC)C3)=O)CCCC1CCN2C(=O)Cc1cncn1C 44958,c1(C(C(=O)NCCC)N(C)C(C2CC3CCC2C3)C)ccc2c(c1)NC(=O)CO2 44959,c1(CC(=O)NCc2nccc(CC)n2)c(F)c(F)cc(F)c1F 44960,Cc1cc(C#N)ccc1S(=O)(=O)N1Cc2[nH]nc(-c3ccc(C(C)=O)cc3)c2C1 44961,CC(C)(C(F)(F)F)SCCOC1(CCNC(COC(C2(F)CC=CCC2)=O)=O)CC1 44962,c1(C(N2CCC(OCC)(Cc3ccc(OC)cc3)CC2)=O)ccc(C)c(C)c1O 44963,N1(c2snc(CC)n2)CC(CNC(C2CC23CCOC3)=O)OC2(CCC2)C1 44964,C12C3CN(CC13)C(c1ccc(C)s1)C(=O)C(=O)CC(=O)NC2.CO 44965,c1(C(C(=O)NCCC(C)NC(C2(C(F)F)CC2)=O)=O)cc(F)cc(Cl)c1 44966,C1(Nc2nc(C)ns2)CCCC1CNC(c1sccc1F)=O.CS(=O)(=O)NCC=O 44967,Cc1noc(-c2ccccc2)c1C(=O)NCC(C)(O)CNC(C1CCOC1=O)=O 44968,c1(CNc2ncn(C)n2)ccc(CN(C)C(c2ccc(C(C)C)cc2)=O)cc1 44969,c1(N2CC(CN(C)C)OCC2)cc(Br)ccc1S(=O)(=O)NCC(F)C1CCC1 44970,C(=O)(C1COc2ccccc21)N1CC(CCNC(c2cc(C)n(C)c2)=O)OCC1 44971,Cc1cc(C(=O)N(CCCCNC(=O)CCC(=O)c2ccncc2)C)c(C)s1 44972,N1(C(C=CSC)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 44973,C1(C(=O)NC(C#C)CCC)CC(=O)CN1C(C1(C(=O)C2CC2)CC1)=O 44974,N1(C(C2C(NCC)CC2)=O)CCC(N(C(C)OCc2onc(CC)n2)C)CC1 44975,n1(C(CC)C)ccc(=NC(=O)C2CN(C(c3nocc3C)=O)CCC2(C)C)[nH]1 44976,N1(C(C2C(OC)CCCC2)=O)CCN(C(C2OCCCC2(C)C)=O)CC1CO 44977,C1(CC(=O)NCC2C=CCN2C(=O)C=CI)CC2(CCC2)C1 44978,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 44979,N1(C(Cc2nc(C)sc2Cl)=O)CCCC(NC(C2C(C)OC(C)C2C)=O)CC1 44980,C1(C(N(CC(C)C(=O)NC2C=CC(C)(C)CC2)C)=O)CCC(C)(O)CC1 44981,c1(CC(=O)NCCCCNC(=O)C(c2ccccc2)F)ccc(NC2CC2)cc1 44982,CC(CS(C)=O)C(=O)NC(=O)CC=CCNC(=O)CCCCNC(N)=O 44983,C(C(CO)(c1ccccc1)NC(=O)Cc1csc(Cl)c1)OC 44984,C(=O)(CC(C(F)F)NC(C1(C)CCCC1)=O)NC(C(=O)OC)C 44985,C(=O)(CS(=O)(=O)c1cc(Cl)ccc1Cl)NCc1cn(CCCOC)nn1 44986,c1(C(N2C(C(N(C3CCOCC3)CC)=O)CC2)=O)cnc(Cl)o1 44987,c1(NC(C2(CNC(c3c(OC)nsc3)=O)CC3(CC3)C2)=O)cc(Cl)ccc1C 44988,C#CC(CNC(C1C=CCN1C(c1cnc(O)o1)=O)=O)CC1CC1 44989,N1(C(c2cc(CCC)[nH]n2)=O)CC2CC(C(=O)NCCCOC(=N)O)CC2C1 44990,c1(CC(=O)NC2C(CNC(COc3ccn(C)n3)=O)C2)c(Cl)cncc1Br 44991,n1(CCCC)ncc(C(=O)NCC(O)CN(C)C(c2nnn(C)c2C)=O)c1CC 44992,N1(C(C(C2CC2)OCC)=O)CCCC1CC(=O)NCC1(C(C)C)CCC1 44993,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2cncn2)CC1 44994,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)N(C(C)C(=O)NC)C 44995,C1(C(N2C(CN(C(CCCOCC=C)=O)C)CC(F)C2)=O)CCS(=O)(=O)CC1 44996,Cc1cnc2[nH]cc(CN3CC4C(C(=O)NC(=O)C(Cl)(Cl)Cl)(C4)C3)c2c1 44997,c1(OC)ccnc(-c2cn(C3CCN(C(C4(C)C=CCCC4)=O)C3)nn2)c1 44998,c1(C(=O)NCC(CNC(Cn2nc(C)c(C)c2C)=O)O)cnc2cnccc2c1 44999,c1(Cn2cc(C3C(C)CCN3C(=O)CCF)nn2)cccc2nccn12 45000,N1(C(n2cc(-c3c[nH]nc3F)nn2)=O)CCC(C2CC2)C1Cc1nccc(O)n1 45001,N1(C(CCCOC(C)C)=O)CCCOC(CNC(C2CC=CCC2)=O)C1 45002,CC1(C(=O)NC2CC(CNC(C3(C(F)F)CCCC3)=O)C2)CCCNC1=O 45003,c1(CC(N2CCC(C(CO)NC(C3=C(C)CC3)=O)CC2)=O)c(C)nn(C)c1C 45004,C1(NC(c2nc(Cl)c(Cl)s2)=O)CC2CCC(C1F)N2C(C1CCCSC1)=O 45005,C12(CC(C)CC(C)C1)C(=O)N1CCN(CC1)C2.c1(S)ccccn1.CO 45006,CC1CCC=C1C(=O)NCC1(CNC(=O)CC(O)c2ccccc2)CCCC1 45007,N#CC1CC(C(=O)NC2(C(=O)N(CC(O)CF)C(N)=O)CC2)C1 45008,C12(C(N(C(CC#C)C)C)=O)CC(CN(C(C3CC=CCC3C)=O)C1)C2 45009,CCCC(C)CC(=O)N1CCOC(CN(C(=O)CN(C)C2CC2)C)C1 45010,N(C(=NCCC)NCC1CCCC(CC)O1)CC1CC(CC)C1 45011,N1(C(c2ccc(C)nn2)=O)CC(C(N2CCOCC(N(C)C)C2)=O)C(F)(F)C1 45012,N(C1CN(c2cc(Cl)ncn2)CCc2ccccc21)C(=O)CCc1cnc[nH]1 45013,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45014,C(=O)(CC(O)C(C)C)NCCC(c1ccc(C)cc1)NC(=O)Cc1cc(Cl)no1 45015,C12(CNC(=O)C=CC=C3CCCC3)CCCC(CN1C(=O)Cc1ccccc1)C2 45016,c1(C(=O)NC2CCN(Cc3c(C#C)cccc3)CC2O)ccc(O)c(O)c1Cl 45017,c1(COC2CCN(C(c3cc(SC(CC)C)no3)=O)CC2)ccc2nccn2c1 45018,c1(CN=[N+]=[N-])nc(CSc2cnn(CC3CCCNC3)c2)cs1 45019,c1(C(N(CCCNC(C2C(=C)C2)=O)C2CC2)=O)ccc(NC)c(S(N)(=O)=O)c1 45020,N1(C(C(C)C)=O)CCC(C)(C)C(NC(=O)COc2ccccc2C(N)=O)C1 45021,c1(OC)ccccc1C(F)(F)C(N1CC(NC(=O)C(C)N(C)C)C(O)C1)=O 45022,Cc1[nH]c2c(C(N3CCC(C(C)(C)NC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45023,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3cc(-c4ccoc4)[nH]n3)=O)CC2)C1 45024,c1(OCC(N2CC(CCCSCC(=O)NC3CC3)OCC2)=O)cc(F)ccc1F 45025,N1(c2c(OC)c(Cl)ncn2)CCCC(C2CC2NC(c2nccc(Cl)c2F)=O)C1 45026,c1(CN2C(C)CC(OCC(N3CCC(OC)CC3)=O)C2)cc(C)cc(C)c1 45027,C1(O)(CCNC(C2CC(NS(CC)(=O)=O)C2)=O)CCN(C(=O)C=C(C)Cl)CC1 45028,N1(C(c2c(C)nc(-c3cnn[nH]3)s2)=O)CCN(C(=O)CO)C(c2ccncc2)C1 45029,Cc1cc(N2CC(c3nc(-c4ccco4)no3)CC2=O)nc(C)c1 45030,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45031,C(=O)(C1=CCCN(C(=O)C=CCF)C1)NC(CC)C(C)CN(C)C 45032,c1(C(=O)NC(C(C)NC(C2(CCC=C)CC2)=O)(C)C)cc(Cl)cc(F)c1N 45033,c1(C(N(CC(=O)N(C)CC2CCCS2)C2CC2)=O)occ2c1CCC2 45034,C1(NC(C)C(c2ccccc2Cl)O)CC2CCC(C1)C2N 45035,c1(C(N2CC(NC(c3n(CC)c(O)nc3)=O)(COC)C2)=O)cncc([N+](=O)[O-])c1 45036,C#CC1(NC(=O)C(C2CCC2)NC(=O)C(F)C(C)(C)O)CCCCC1 45037,c1(C(C(CN2CCCC(CC(N3CCCC3)=O)C2)O)OCF)ccnc(Cl)c1F 45038,C1(CC=C)(NC(=O)Cc2cccc(C3CC3)c2)CCN(C(c2ccccc2)=O)C1 45039,CC(C)CCC(C)N(C(=O)C(C)N(C(C1CCC2CC12)=O)C1CC1)C 45040,c1(C(=O)NC2CC3CN(C(C(CC)CC)=O)CC3C2)ccc2cnnc(O)c2c1 45041,C(C1CCOCC1)=CC(=O)N(CC(=O)NCC1(CC)CCCO1)C1CC1 45042,c1(C(N2C(CNC(C=C(COC)C)=O)CC(F)C2)=O)cccc(OC(F)F)c1C 45043,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45044,N1(C(CN(C)C)=O)CC(C)(C)CCC1CNC(=O)CCn1ccnn1 45045,N1(C(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2ncccc2O)=O)CC(F)C1 45046,c1(CNC(CC=CCC)=O)nn(C)c2c1CN(C(=O)CC1CC3CCC1C3)CC2 45047,C1(F)(CNC(C(C2CCC2)OCC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45048,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45049,N1(C(=O)Cn2cc(-c3ccsc3)nn2)CCCC1Cc1ncco1 45050,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45051,Cc1ccc(F)c(CC(=O)N(CCCCCCO)CC(=O)O)c1 45052,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45053,c1(C(N(CC(CC)NC(C=CCN(CC)CC)=O)C)=O)ccnn1C1CC1(F)F 45054,CC1CC(NC(=O)CCCN(C)C(N)=O)CCN1C(=O)CN(C)C 45055,c1(OC)ccc(F)cc1CC(N1CCN(C(c2ccc(CO)nc2)=O)CC1)=O 45056,N1(C(C2C(C)CCC2)=O)CC(F)(F)CC1C(=O)NCc1cc(Cl)ccc1Cl 45057,CC1CCN(C(=O)CCNCCS(C)(=N)=O)CC1CC(=O)NC1CCCCCC1 45058,C(=O)(CC(O)C(C)CC)NC1(C)CC(F)(F)C1.C1(C(=O)OC)CN2C1(C)C2=O 45059,N1(C(CC(C)(C)O)=O)CC2(C1)SCCC2NC(c1ccc(SC2CC2)cc1)=O 45060,C(=O)(C1=CC2(CCOC2)C1)N(C1CCCCCN(C(=O)COc2ccsn2)C1)C 45061,C(=O)(C(C)CC=CCC=C)N1CCC(CNC(c2ccc(CC#C)s2)=O)C1 45062,C1(NC(CC=CC(C)(C)C)=O)CC12CCN(C(C1CCCOC1)=O)C2 45063,Cc1nn(CC(=O)NCCC2CCN(C(c3nccnc3Cl)=O)C2)c(=O)n1C 45064,N1(C(C(C)=C2CC2)=O)C2CCC1CC(CNC(c1ccc(=N)[nH]c1Cl)=O)C2 45065,N1(C(c2cc(C3(C)COC3)no2)=O)CC(NC(=O)C(C)(Cl)Cl)C(O)C1 45066,c1(C(CNC(c2[nH]ccc2NC(c2cnc(C)o2)=O)=O)OC)c(F)cccc1F 45067,N1(C(c2cc3cccc(F)c3s2)=O)CCCC(C2CN(C(C3(F)CC3)=O)C2)C1 45068,c1(CC(=O)NC2C(CNC(CCC3N(C)CCCC3)=O)C2)cnn2c1OCCC2 45069,C1(NC(CCSC)=O)CCC(CCNC(=O)Cc2ccn(CC(C)C)n2)C1 45070,C(=O)(C(C)(C)CCC#N)N1CCC(CC(=O)NCc2ccc(C#C)cc2)C1 45071,C#CC(C(C)OC)NC(=O)CC1CC(NC(=O)CC(C)C2CCCCC2)C1 45072,C1(CS(=O)(=O)NCC2CC(C)(C)OC2)CCCC2(CCOC2)O1 45073,Cc1nc(C(=O)NC2(CCNC(=O)C(F)CC3CCOC3)CC2)n[nH]1 45074,C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(c2c(COC)noc2)=O)CCC1 45075,C1(C)(COCC(=O)NCC(C)CNC(=O)CC2CCCC2)CCC(=O)N1 45076,C1(C(=O)NCCC2CN(C(C(C)(C)OC(C)=O)=O)C2)CC1C1CCCC1 45077,c1(CC(=O)N(CC(C)NC(C2(Cl)CC2(F)F)=O)C)cccc(C2CC2)c1 45078,C1(CNC(CCc2c(OC)cccc2)=O)CN(C(C23CC(CO2)C3)=O)CCC1C 45079,CCC(C)C(O)C(=O)N1CCCC1C(N1CC(=O)N(CC)C1)=O 45080,C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCCNC(Cn1c(C)c(Cl)cn1)=O 45081,c1(CC)[nH]nc(C(N2CC(OCCNC(c3cccnc3C(F)F)=O)C2)=O)c1Cl 45082,N1(C(c2ccccc2F)=O)CC2CCN(C(=O)CCCCc3ccccc3)C2C1 45083,C(=O)(C(O)CC(F)F)NC1(CNC(c2c(OC)n[nH]c2)=O)CCCC1 45084,CC1(C)CN(C(=O)CC(F)(F)Br)C(CNC(C2CCC2)=O)CO1 45085,CC1CC(NC(c2ccn(C3CCCC3)n2)=O)CN1C(=O)CN1CC2CC2C1 45086,c1(C(=O)OC)cc(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)CO)no1 45087,C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C(CC=CC)C)=O)C1 45088,C1(C(N2CC(C(=O)NCCC(CNC(C3(C)CCC3)=O)O)C2)=O)CCCN1C=O 45089,C1(NC(c2cc(C)c(F)cc2)=O)CCCC12CN(C(=O)C(C1CCC(=O)N1)C)C2 45090,CC1CCC(NC(=O)C(=O)C=Cc2ccc(F)cc2)CN1C(C1(CF)CC1)=O 45091,c1(OC(C(=O)NC(CNC(C(=CC2CCCC2)C)=O)CO)C)ccc(F)cc1 45092,N12CCCCC(C1)CCC2=O.N1(C(Cc2n(C)ccn2)=O)CCOC(CN=[N+]=[N-])C1 45093,N1(C(=O)NC(c2cncc(C)n2)C)CC(=O)OC2(CCC2)C1 45094,C1(NC(C2(C=C)CCOCC2)=O)C2CCN(C(=O)CC3(C#N)CCC3)CCC12 45095,CC(C)(C)C(C(=O)NCCOC1CN(C(=O)C(c2ccccc2)O)C1)N(C)C 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45148,N1(CC(N2CCC(O)(COC)CC2)=O)C(=O)C(=O)N(C)C1=O 45149,Cn1nc2c3c1CCN(C3)C2.C1(NC(C2CCC2)=O)CCC(C)(C)CO1 45150,c1(OC(C(=O)NC2C(NC(Cc3c(C)con3)=O)C2)C)ccc(F)c(F)c1 45151,CS(=O)(=O)c1ccsc1C(=O)NC1CCC(CNC(C2CC(C(=O)OC)C2)=O)C1 45152,N1(C(Cn2c(C)ccn2)=O)CC2(C1)CN(C(c1cccnc1CO)=O)CC2CO 45153,C1C(CC=C)C(=O)N2CCCC2C(=O)O1.C#Cc1cnn(CC(=O)NCC)c1 45154,Cc1ccc(CCNC(=O)CC2CCCN(C(C3OC4CCC3C4)=O)C2)cc1 45155,CC1(C)CCOC1CC(=O)NC1CCN(C2CCOC2)CC1.C12CCCN1C2 45156,C1(NC(c2cnc(S)nc2)=O)(CNC(C2C3(CC3)C23CC3)=O)CCCCC1 45157,c1(OC(C)(C)C)ccc(F)c(F)c1.C12(CCCC1)CNC(=O)N2C1CCCC1 45158,N1(C(c2noc3c2CCCC3)=O)CCC2CCC(C1)N2C(=O)C=CC1CCCC1 45159,N1(Cc2ccc(OC)cc2)C(=O)C(CCCO)N(Cc2cccs2)C1=O 45160,c1(CNC(C(N2C(C(C3CCOC3)=O)CC2)=O)=O)nncn1CC1CC1 45161,C1(C(=O)OC)CCN(C(=O)C(CC2CC2)NC(C2CC(C(C)C)C2)=O)O1 45162,N1(C(=O)NC(c2cc(Cl)ccc2Cl)CC)CCC(F)(F)C(C(=O)OC(C)(C)C)C1 45163,c1(C(=O)NC2CCN(C(C=CC)=O)CCC2C(C)C)cnc2c(cnn2C)c1O 45164,C(=O)(N=c1ccn(C)[nH]1)c1ccc(S)o1.N1(C(=O)C=CC(=O)NC(C)=O)CC=CC1 45165,CCC(CC)CCCC(=O)N1CCCC(O)(CNC(=O)C(C(C)C)OC)CC1 45166,C(=O)(CS(=O)(=O)CCO)NCCCN(C)C(c1cn(CC2(C)CC2)nn1)=O 45167,C1(NC(CN(CC#C)C(c2ccoc2CNC(N)=O)=O)=O)C2CCCC12 45168,N1(C(C2C(C=C)C2)=O)CCC(C2CC2)(CNC(=O)CC(C)P(C)(C)=O)C1 45169,C(CCCCC(=O)N1CCN(C(C2CCN(C)C2=O)=O)C(c2ncc[nH]2)C1)OC 45170,c1(C(N2CC(OC)CC(NC(COCCC)=O)C2)=O)csc2c1CCC(C)C2 45171,C1(N(C(c2ccc(CCC)s2)=O)CC)CCCN(C(C2(SC)CCC2)=O)C1 45172,Cc1cc(C(C)C)ccc1C(=O)NC1C=CC(CNC(c2sc(C)cc2Cl)=O)C1 45173,c1(C(N2CCN(C3CCN(C(c4c[nH]c(=N)o4)=O)C3)CC2)C)ccc(F)c(F)c1 45174,c1(NCc2cn(CCF)nc2)nc(N2C3CCC2COC3)nc2ncn(C)c12 45175,C1(C(=O)NCC(C)(C)NC(C(C)C(C)N2CCCC2=O)=O)CCC(O)CN1C 45176,c1(C(N2C(C(N(C)CC3(O)CCCC3)=O)CCC(O)C2)=O)ccc2[nH]ccc2c1 45177,C(=O)(C1CCCc2nncn21)N(CCNC(C1CCC(CF)C1)=O)C1CC1 45178,CCCC(C(=O)N1CC2CC2(NC(=O)C(CC)OCC)C1)C(C)C 45179,c1(C(N2CCC(N(C(c3cc(C)nn3C)=O)C)C2)=O)nc2ccccc2s1 45180,c1(C(=O)NC2CC(NC(c3coc(C4CC4)n3)=O)C2)csc2ccc(F)cc12 45181,C1(NC(=O)COC2CC2)C2CC1N(C(c1conc1-c1ccccc1)=O)C2 45182,C1(CC(=O)NCCN(C(Cc2n(C(C)C)cnn2)=O)C)CCCCN1C 45183,N1(C(=O)OC(C)(C)C)CC2CCC(O)C(O)C12.c1(C2C(=O)O2)cccnc1 45184,N1(C(C)C(=O)Nc2ccc(Cl)cc2)CCCN(C(c2cccc(F)c2)CO)CC1 45185,C1(F)(C(=O)NCCC2CCC(NC(=O)C=Cc3ccccc3)C2)CC2(CCC2)C1 45186,c1(CC)ccc(C(=O)NC2C3CCN(C(=O)C(N4CCC(C)C4)=O)C23)cc1 45187,c1(C2C(=O)NCCCN2CC)cccc(N=[N+]=[N-])c1.C#CC1(OC)CCC1 45188,c1(C(=O)OC)c[nH]c(=NC2CCCCC2N2CCOCC2)nc1C(F)F 45189,C1(CC2N(C(CNC(=O)OC)=O)CCC2)CN(C(=O)Cc2cn[nH]c2)CCC1C 45190,C(CO)(CCCCNC(=O)CC1CCCO1)NC(C1(OCC)CCOCC1)=O 45191,N1(C(C2C(C)OCC2)=O)C2CCC1CN(c1ccnc(-c3ccccn3)n1)CC2 45192,c1(CNC(C(N(C(=O)CCc2cscn2)C)C2CC2)=O)ccc(CO)cc1 45193,N1(C(=O)C#CC2CCCO2)CCC2(CCN(C(c3ccc(F)s3)=O)C2)C1 45194,C1(CNC(c2cnc[nH]2)=O)CC12CCN(C(C1CC3CCCCCCC13)=O)CC2 45195,Cc1[nH]c(=NC2CC(NC(=O)C3CC3)C2)ccc1C#N 45196,N1(C(Cc2c(C(C)C)con2)=O)CC(NC(C2C3CC(F)(F)CC23)=O)C2(CC2)C1 45197,c1(C(N2CCC(N(C(c3sccc3C)=O)CC)C2)=O)cnc(C)nc1C 45198,N1(CC2(C(F)F)C(NC(=O)NCC3(C)CCOCC3)CCC2)OC(C)(C)CC1=O 45199,N1(C(C2(C)CCC2)=O)CCC2(CC1)CC2CNC(c1[nH]nnc1C1CC1)=O 45200,CCCCCCCC(=O)NC1CCc2nnnn2C1 45201,c1(CC)ccc(F)c(C(N2CCCC(C)(CNC(c3nnccc3C)=O)C2)=O)c1 45202,C1(NC(C2(CC)CC2(F)F)=O)CCN(C(=O)CCOC(C)C)CC(C)(C)C1 45203,c1(C(=O)NC2C(C(N3CC(C(=O)NC)C3)=O)CC2)ccc(C)cn1 45204,CC1C(NC(=O)C(C)(C)n2cc(Br)cn2)CCCN1C(=O)C(=O)NCC(F)F 45205,C1(c2n(C)ccn2)CC(C)(C)CN1C(=O)CCn1cc(-c2cccnc2)nn1 45206,C1(CNC(C(c2cccc(C)c2)F)=O)N(C(C2CCNC2=O)=O)CCCC1(C)C 45207,N1(CCNC(C(COC(C)C)N(C)C)=O)CCC(NC(=O)C=CCF)CC1 45208,N1(C(C=C(C)C)=O)CCCC(C2CC2NC(c2cn3ncccc3n2)=O)C1 45209,C(=O)(C1=CCCCC1P(C)(C)=O)NCCC1N(C(CC=C)=O)CCC1 45210,c1(C(C2CC2)NC(C(C)(C)c2ccccn2)=O)cccc(F)c1 45211,C1(N(C(CC(=O)NCC)=O)C)CN(C(=O)CCCC2CCCO2)CC12CC2 45212,C1(NC(C2(C=C)CCC2)=O)CC(C)N(C(=O)Cc2ccc(O)cc2)C1 45213,C1(CCNC(=O)CC2CCCC2)CCCN1C(C1(Sc2ccccc2)CCC1)=O 45214,Cc1cc(C(=O)N(CC(C)NC(=O)Cc2cc[nH]c(=N)c2)C)c(C)cn1 45215,C1(C)(CNC(c2c(C)con2)=O)CN(Cc2ccc(F)cc2Cl)CCO1 45216,CC(CN(C)C(C1(C)COC1)=O)C(=O)NCCCCNC(N)=O 45217,N(C1CN(C(c2ccc3nc[nH]c3c2)=O)Cc2ccccc21)C(=O)CSC(F)F 45218,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1CNC(=O)CSC 45219,CC1C(NC(=O)CC2OCCO2)CCN1C(=O)C(=Cc1cn(C)nn1)F 45220,Cc1ccc(NC(C2C3CC2N(Cc2cnccc2Cl)C3)=O)c(F)c1F 45221,c1(NCCC(C)OC)nc(N2CCC(C(C)CO)CC2)nc2c1ncn2C(C)C 45222,C1(NC(=O)CCC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45223,C=Cc1cncc(C(=O)NCC2CN(C(=O)CCC3CCCN(C)C3)CCO2)c1 45224,C(=O)(C(C(=O)OCC)OC)N1C(C(C(=O)NC(CCC)C2CC2)(C)C)CCC1 45225,C12CCCN(CC1)C(=O)C(C)(C1CC1)N2CC.C(C)(C(=O)O)=CCC 45226,c1(C(=O)N)cc(C(=O)NCC2C=CC(CC3CN(C(=O)OC)C3)C2)no1.OCC 45227,C=C(C)C1CN(C(=O)CC2CCCN(C(=O)Cc3cnns3)CC2)CCO1 45228,c1(NC(C2CCCN(C(C(CC=C)NC(C)=O)=O)C2)=O)cc(Br)ncc1[N+](=O)[O-] 45229,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45230,CCC(O)(CC(=O)NC1(CCNC(=O)C(C)SC)CCC1)c1ccccc1 45231,C1(CC(=O)NCC(C)N(C(Cc2c(C)nc(C)s2)=O)C)COc2ccccc2O1 45232,c1(NC(C(C(C)NC(CC(CC)SC)=O)(C)C)=O)cnn2c1CCCC2 45233,C#CCC(C)(C)C(=O)N1CCN(CC(C)NC(=O)C(C2CCOCC2)O)CC1 45234,C(CC(C)C)(C(=O)NCCC1(NC(C)=O)CN(C(=O)C(=O)NC(C)C)C1)OC 45235,c1(C(=O)NC2CC(CNC(CCNC(C)=O)=O)C2)ccn2nnnc2c1 45236,CN1CCC2C1CCCN2C(C1(CNC(c2n[nH]c3c2CCC3)=O)CCC1)=O 45237,C1(C(=O)NCC2(C)CC(NC(C3(C)C(C)(C)C3(C)C)=O)C2)CC2CCC(C1)C2O 45238,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(F)(F)Cl 45239,c1(CNCC23C(CN(C(C4CC(F)C4)=O)C2)C3)cccc(F)c1Cl 45240,O=C(C1=C(Cl)CCC1)NC1CC(NC(c2n[nH]c3c2COC3)=O)C1 45241,N1(C(c2nc(C)nn2C)=O)CCN(C(C2(N3CCCC3)CCC2)=O)C(C)C1C 45242,C(=O)(C1=CCC(F)(F)CC1)N1CC(CNC(C2C(C)C2)=O)OC(C)(C)C1 45243,CP(C)(=O)CCC(=O)NCC#CCNC(C1CN(C(N)=O)C1)=O 45244,C1(CC(=O)N(CC(C)C)CCCN(C)C)C2CN(C(=O)C(F)=CC3CC3)CC12 45245,C1(OC)CN(C(=O)CC2CC2)CC1NC(c1coc(C(c2ccccc2)C)n1)=O 45246,c1(C(=O)NC(CC)CNC(=O)C(F)n2cccn2)cncnc1 45247,N#CC1(CC(N2CC(C(O)C(=O)NCc3csc(C(N)=O)c3)C2)=O)CCCC1 45248,C1(F)(CNC(=O)CCCN2CCCCC2)CCN(C(C2CCCSC2)=O)CC1 45249,C#CCC(C)(CC)C(=O)N(CC(=O)Nc1nccn1C(C)C)CC(C)C 45250,C1(CCNC(C(F)=CCC)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45251,c1(Cc2n(-c3cc(C)on3)ncn2)ccc(Cl)c(COC)c1 45252,N1(CC(=O)NC2CCCN(C(C(C)(C)F)=O)C2)CCCC(C(F)(F)F)C1=O 45253,N1(C(CCC#C)=O)CCN(C(c2cn(C)nn2)=O)CC1CC1CC1 45254,C(C)(CCC(=O)N1CCCC(C(C(C)C)NC(=O)CNC(=O)N(C)C)C1)SC 45255,c1(C(=O)NCCCC(C)NC(=O)CN(C)C)cnccc1C(F)(F)F 45256,c1(C(N2C(CN(C(CSC(C)C)=O)C)COCC2)=O)n[nH]c2c1COC2 45257,N1(C(c2c(C)snn2)=O)CCC2(CCCN(C(c3cc(CO)n(C)n3)=O)C2)C1 45258,c1(C(=O)NCC2(OC)CN(C(C3CC34CCOC4)=O)C2)ccc2c(c1)NCC2 45259,Cc1ccc2oc(C(=O)NC3CN(C(c4cn(C)c(C(F)F)n4)=O)C3)cc2n1 45260,C1(NC(c2c(CC)nccn2)=O)(COC)CCN(C(c2cccn2CC)=O)CC1 45261,CCC(C)C(C(=O)NCCn1ccc(C(=O)NCC2CCSCC2)c1)N(C)C 45262,CC(CCNC(C1(CNC(=O)CC2CCC(C)C2)CCCC1)=O)C(C)(C)C 45263,Cc1cccc(Cl)c1NC(C1CN(C(=O)C(C(C)C)Sc2ccccc2)C1)=O 45264,C1(C(CC(CC)NC(C2(C(CC)=O)CC2)=O)=O)COC2COCC12 45265,C1(C(N2CC(C(N)=O)(CNC(C3C(=C)CC3)=O)C2)=O)CCc2nnc(O)n2C1 45266,C1(C(N(C2CC(NC(C(CCC)NC(N)=O)=O)C2)C)=O)CC2CCCC(C1)C2 45267,n1(C(COC)C)nc(C2CCCCC2)nc1COC(C)CC(C)C 45268,N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(=O)C(C)(C)N(C)C)C2CC12 45269,C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(=O)CC1CC=CCC1 45270,C1(n2c(OCC)nc(CCc3ccccc3)n2)CCC(F)(F)CC1 45271,N1(C(c2c(N)non2)=O)CC(NC(=O)Cc2csc(-c3ccsc3)n2)CC(O)C1 45272,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45273,c1(C(N2CC(C(C)(C)C)C2)=O)n[nH]c2c1CN(C(C1C3COCC13)=O)C2 45274,CCC(C(=O)NC1CC(NC(=O)C=C(C)C2CCC2)C(O)C1)C(C)(F)F 45275,C12(C(=O)NCC(CC)(CC)NC(c3ccc(OC)nc3OC)=O)CCC(F)(CC1)C2 45276,CCCCCC(O)C(=O)N1CC(CN(C(=O)CN2C(=O)CNC2=O)C)C1 45277,CS(=O)(=O)c1ccsc1C(=O)NCC(C1CCC1)NC(C1(C#N)CC2CC2C1)=O 45278,C(=O)(C(O)C(C)(C)C)NCCn1cc(C(N(CC#C)C)=O)nn1 45279,C1(CN(C(=O)CN2CCOCC2=O)C)CCCN(C(C2CCCS2(=O)=O)=O)C1 45280,c1(C(=O)N(C2CCCC2)CCNC(C23CC(O)C2C3)=O)cc(Cl)ccc1Cl 45281,C(=O)(C1=COCCO1)N1CCC(N(CCCCCNC(=O)C2CC2)C)CC1 45282,c1(C(N2C(CNC(C(C)(Cl)Cl)=O)CC2)=O)cc(C2CC2)oc1C1CC1 45283,Cc1cccnc1C1(F)CC1.C12CCCN(C1)C(=O)c1ccnn12 45284,C1(CC)CCCCC1C(N1CC(NC(=O)CCCOCc2cccnc2)C(O)C1)=O 45285,C1(C(N2CCC3(CC2)CC3C(N2CCC(F)C2)=O)=O)CCc2cc(F)ccc2O1 45286,CCCC(C(=O)N1CCCC1(C)c1cn(Cc2cnc[nH]2)nn1)OC 45287,N1(C(c2c(C)ocn2)C(=O)NCc2cccc(Cl)c2)CCCCC1Cc1cccs1 45288,CC(C)(C)C(C)(C)C(=O)NC1CCC(NC(=O)Cc2ccn(CCF)n2)C1 45289,C1(NC(c2cccnc2OC(F)F)=O)CC2CN(C(=O)C3CC3)CCN2C1=O 45290,c1(N(C(c2ccccc2SC)=O)CC)nccc(OC)c1F.C12CC1CNC2=O 45291,c1(C(C)C)cncc(C(=O)NC2(C)CC(NC(=O)C(F)C3CCOC3)C2)c1 45292,C1(C(N2CC3(C(NC(c4c(C)nsc4)=O)CCC3)C2)=O)Cc2ccccc2CO1 45293,Cc1ccc(C=CC(N2CC=CC(C(=O)NC(C3CCOC3C)(C)C)C2)=O)cc1 45294,C(C1COC(C)(C)O1)=CC(=O)NC1CC(C)(NC(C(C=C=C)C)=O)C1 45295,c1(C(=O)OC)cnc(NC(C2CCCN(C(c3ncsc3Br)=O)C2)=O)nc1C 45296,CCCC(CCC)C(=O)N1CC=CC(NC(c2cc(C(F)F)ccc2Cl)=O)C1 45297,c1(C(=O)NCC2(C(C)(C)C)CCN(C(C3CCN(C)C3)=O)C2)c[nH]nc1[N+](=O)[O-] 45298,N1(C(C(C)(C)SC)=O)CCC(NC(c2ccc(-n3ccc(C)n3)cc2)=O)C(C)C1 45299,c1(CC(C(N2CC(n3cc(CCOC)nn3)(C(=O)OC)C2)=O)C)ccc(O)c(F)c1 45300,Cc1ccc2nc(C(=O)NC3(CNC(c4nc(C)oc4C)=O)CC3)c(N)n2c1 45301,c1(NC(C)=O)ccccc1CCC(=O)N(CCCNC(=O)C(F)C1CCOC1)C 45302,C=C(C)CC(C(=O)N(CC(O)CC)C)NC(C1CC2CC(=O)C1O2)=O 45303,C(N=c1[nH]c(=NCCc2csc(=N)[nH]2)[nH]c2cc[nH]c12)c1nccc(N(C)C)c1 45304,CCCC1C(=O)NCC(=O)N2CC(OCC2)CC(=O)N1.C(C)(C)[SH3]=O.COC 45305,C(C(C(=O)N(C1CC1)CC1CC1)NC(=O)C(C)OC1CCOC1)SC 45306,c1(CC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)ccc2c(c1)CC(C)O2 45307,C1(C(=O)NC(CN(C)C(c2cc(Cl)nn2C)=O)(C)C)CCC2CC2CC1 45308,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(Cl)cc2)O)c[nH]c2nccc-2c1 45309,c1(OCCOC)cnc(C(=O)N(C(C)CNC(=O)Cc2scnc2C)C)cn1 45310,C(=O)(C1=CCN(C(=O)C(c2cnn(C)c2)=O)CC1)NC(CC(CC)C)C 45311,CCCC(CC(=O)NC1CCC(OC)C1)NC(c1cc(C#N)oc1C)=O 45312,c1(OC(C)C)cnn(C)c1.c1(CCC(=O)N2CCCNC(=O)C2)ccncc1 45313,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45314,CN1CCC(NC(=O)CC(C)(C)C#N)C12CCCN(C(c1cscc1Cl)=O)C2 45315,Cc1c(C(=O)NCCC2(O)CN(C(=O)CCC3CCOC3)C2)cc(N)cc1O 45316,c1(OCC)ccc(C(=O)NC2CCC2CNC(=O)C(c2cccnc2)OC)cn1 45317,Cc1ccnc2ccc(C(=O)NCC3(NC(=O)CN4CC(C)C4)CC3)cc12 45318,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CC(C)CN(C(=O)C(C)(CC)OC)C1 45319,N1(C(c2ccc(CC=C)cc2)=O)CCN(Cc2nc(=N)[nH][nH]2)CC1C 45320,C1(C(=O)OCC)CC2(CCN2C(=O)C(c2ccc(Br)cc2)(C)C)C1 45321,C1(NC(CCC(C)SC)=O)CCN(C(c2cc(F)c(F)cc2Cl)=O)CC1(C)C 45322,N1(C(C(C)(C)C(F)F)=O)CC2CCC(NC(=O)CCc3cscn3)C2C1 45323,CC(C)C(=O)NNC(=O)C1CCN(C(=O)OC(C)(C)C)C1CCc1ccccc1 45324,CCC(C(=O)NC(CNC(c1cccc2c1CCO2)=O)CO)C(C)(F)F 45325,c1(CC(=O)NCC2OCCN(CC3CN(C)C(=O)C3)C2)ccnc(Cl)c1F 45326,C1(C(N2CCC(N(C(c3csc4nccn34)=O)CC)C2)=O)CCCCC12CCC2 45327,CCCCCCC(C)NC(c1cc(C(C)C)n(CC(=O)OCC)n1)=O 45328,N1(C(=O)NCCc2coc(Cl)n2)CCC(CCn2cc(C(N)=O)nn2)C(F)(F)C1 45329,Cc1c(C(=O)NCc2csc(CNC(=O)C(C)C3CC3)n2)sc2cccc(F)c12 45330,C=CCCCCC(=O)NCC(C)NC(=O)CCCSCc1ccccc1 45331,N1(C(CC2CC(NC(CCCSC)=O)C2)=O)CCc2nc(O)[nH]c2C1 45332,N1(C2CCN(C(C(C)(C)OC)=O)C2)CCN(C(=O)CC2(C(F)(F)F)SCCS2)CC1 45333,c1(C(C(=O)NC(CC)CNC(C2CSCC(=O)N2)=O)(F)F)cccc(Cl)c1F 45334,C1(COC)CCCCN1C(c1n[nH]c(C2CC2)n1)C(=O)NCCCN(C)C 45335,C1(CC(=O)NCC2CCN(c3ncc(Br)cc3Br)C2)CCc2n[nH]cc2C1 45336,c1(SC)ccc(NC(c2c[nH]nc2CNC(c2cnc(C)nc2C)=O)=O)c(F)c1 45337,Cc1nccnc1C(=O)N(C)CCNC(=O)CC(C)Cc1cccc(F)c1 45338,N1(C(C(C)NC=O)=O)C2CC1CN(C(c1cc(-c3cccc(Cl)c3)ns1)=O)C2 45339,C12(C(N3C(CN(C(=O)Cc4cc[nH]n4)C)CCCC3)=O)CCC(CC1)OC2 45340,Cc1c(C(=O)Nc2ccc(N3CCCCC3)nc2)cc(I)cc1Cl 45341,C(Cn1cncn1)N=c1[nH]c(N2CCN3CCCCC3C2)nc2ccsc12 45342,CC1(C)COC(C(=O)NCC2CCCC(CNC(c3cc(F)c[nH]3)=O)C2)C1 45343,C(=O)(CC(C)(O)C1CC1)NCC(C)CN(C(=O)Cc1n[nH]cc1Br)C 45344,N1(C(Cc2ccc(C)cc2)C)C(=O)CN(CC2(C(F)F)CCCO2)C1=O 45345,C1(F)(CNC(CCc2nc(C)c(C)[nH]2)=O)CCCN(C(=O)CCC(C)(F)F)CC1 45346,n1(CC)ncc(Cl)c1C(=O)NCC1CCC(CNC(c2cc(C(=O)OC)c[nH]2)=O)C1 45347,N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2C(C(=O)NCC3(C)CC3(F)F)C2C1 45348,C1(CCC)CN(C(C2CC(CO)C3CC23)=O)CCN1C(c1cn[nH]c1)=O 45349,c1(C(=O)NCC(C2CCC2)NC(CSCC)=O)cc(Br)ccc1Cl 45350,c1(C(N(CCCOCCNC(c2ccc(SC)cc2)=O)C)=O)nc(C)ccc1F 45351,C(CC(=O)NNC(=O)c1cnn(C2CC2)c1C)SC 45352,C1(c2cn(Cc3c(OC)cccc3)nn2)(NC(=O)CC(F)F)CC2(C1)OCCO2 45353,c1(NC(C2(CN(C(CS(CC)=O)=O)C)CC2)=O)cccc(F)c1O 45354,c1(C(N2CCCC(C(=O)OC)C2)C(=O)NCC(CC)C)ccc(F)c(F)c1 45355,n12cnc3c(nc(=NC)[nH]c13)N1C3CCC1CC2C3.C(=O)(COC)NCCSC.CC 45356,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45357,c1(OCC(NC(NCC(COC)C)=NC)C)ncc(-c2ccccc2F)n1C 45358,C1(CNC(CN(C(C)=O)C)=O)CCCC1NC(c1cnn(-c2ccncc2)c1)=O 45359,CN=c1[nH]cc(C(=O)NCc2ccccc2CNC(c2cc(C)sn2)=O)o1 45360,c1(C(=O)NC(C(C)C)CCNC(=O)C(c2ccccc2)O)cc2cnccc2[nH]1 45361,c1(CN(C2CCCOC2)C(C23CC2CN(C(=O)CC2CC2)C3)=O)cc(F)ccc1F 45362,Cn1ccc(C(=O)NCC2CCN(C(C3CC4CCC3O4)=O)C23CC3)cc1=O 45363,C1(C(N(CC(C)NC(C2SCCS2)=O)C)=O)CS(=O)(=O)CCO1 45364,c1(C(NOC(CC)CC)=O)cc(CSC)ccn1.C12(CCC1)C(=O)NC2 45365,Cc1ccc(C2(NC(=O)Nc3cccc(C(=O)N(C)C)c3)CCC2)c(F)c1 45366,N1(C(c2ccc(C)nc2C)=O)CCCC(F)(CNC(=O)C(O)C(C)(C)C)CC1 45367,c1(OCC)c(C)n[nH]c1C.C12(OCC)CN(C1)C(=O)C1C(C1(F)F)C(=O)NC2 45368,N1(C(C(C2(C)CC2)NC(Cn2ccc(C)n2)=O)=O)CCC12CN(C)C2 45369,c1(C(=O)OCC)ccnc(C(=O)NC(CNC(C2CC2(F)F)=O)CC(C)C)c1 45370,C1(CC(N)=O)(CNC(C2(C)CC(=C)C2)=O)CCN(C(=O)C(O)CC(=O)OC)CC1 45371,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45372,CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)C(O)CCSC)C1 45373,C12CCCCCN1C2=O.c1(C(=O)NCC2CN(C3CCOC3)C2)cccc(N)n1 45374,c1(OCC)ccc(C(=O)NC2CCCCC2CNC(c2ccnnc2O)=O)nn1 45375,Cc1cc(C(N2CC3C(CNC(=O)C(O)CN4CCCC4)C3C2)=O)c(O)c(C)c1 45376,c1(C(=O)Nc2ccc(OC)c(C(C)C)c2)ccc2cncn2c1 45377,C(C)(CC(=O)NCCN(C1CCCCC1)C(c1nocc1Cl)=O)SC 45378,Cn1ncc(Cl)c1C(=O)NCC1CCCN(C(c2cccc(OC(F)F)c2)=O)C1 45379,CC12CC(CC1C(=O)NCCCN(C(C1(O)CCOCC1)=O)CC1CCCC1)C2 45380,n1(CC(=O)N(CCCNC(C(C)OCC=C)=O)C)c(C)cc(O)cc1=O 45381,N1(CC2CC(=O)N2)CCC2(CCN(C(c3ccn4ccnc4c3)=O)CC2)CC1 45382,c1(C(N2CC(NC(Cc3c(C)noc3C)=O)C(F)C2)=O)ccc2nsnc2c1 45383,Cc1cnc(C(C2CC2)NC(C2CS(=O)(=O)C2)=O)s1 45384,n1(CCOC)ccc(C(=O)N(CC(C)(C)NC(c2ncoc2C(C)C)=O)C)n1 45385,C1(C(N(CCNC(c2cncc(C3CC3)c2)=O)CC)=O)CCN(C)C(C)C1 45386,C(C(C)CC(F)(F)F)O.C1(C(=O)OC)CCCN(C(C2(C)CCCCC2CO)=O)CC1 45387,Cc1ccc(F)cc1S(=O)(=O)N1CCC(O)CC12CC2.c12nnc(o1)s2 45388,C#CCC(CC)NC(C1(CNC(=O)C(O)C=C)CCCC1)=O 45389,C1(NC(CN2C(=O)OCC2)=O)CCN(C(C2CC3C=CC2C3)=O)C12CCC2 45390,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CCCC2)CC12CC2 45391,c1(C(N2CC3CCN(C(CC(=O)OC)=O)C3CC2)=O)cnc2c(C)cccc2c1 45392,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccccc1Cl)C 45393,N1(C(c2c(CC(C)C)onc2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C2(CC2)C1 45394,N1(C(CC=C(C)C)=O)CC(F)(F)CC1CCNC(c1coc(Br)n1)=O 45395,C1(NC(c2cn(C)nn2)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)C12CC2 45396,C1(OCCC)CN(N2CC(OCC)C2)C1.N(C)C 45397,CN1N=CC(CC(=O)N(CC(N2CC(C(N)=O)C(CO)C2)=O)CCO)C1=O 45398,CCCCCCCCOC(=O)N(C1CCC1)C(c1ccc(C#N)cc1)C 45399,c1(SC)cncc(C(=O)N(C)CC2CN(C(=O)C(C3(O)CCCC3)F)CCO2)c1 45400,C#Cc1cc(SCCCCO)nc(C)c1 45401,C1(NC(CCCOC(C)C)=O)CCC(CNC(c2csc(S)n2)=O)CC1 45402,c1(C(=O)C(N2CCC(NC(C34CC(F)C3C4)=O)C2)=O)ccccc1Cl 45403,C1(C)(NC(CN(C)C(c2ccsc2)=O)=O)CN(C(=O)CCC2CCCN2C)C1 45404,N1(C(Cc2c(C)noc2)=O)CCC(NC(=O)CCc2ccccn2)C1C(C)C 45405,C1(OC)CN(C2=NCCNCCN2)CCC1O.S(=O)(=O)(C1CC1)CN1CCCCC1 45406,C1(NC(C(C)C)=O)CCCCN(C(c2ccc(N)c(OCc3cccs3)c2)=O)C1 45407,Cc1ccccc1C1(C(=O)NC2COCC2NC(C23CCC2C3)=O)CCOCC1 45408,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(c2c(C)oc(C(C)C)c2)=O)CC(F)C1 45409,c1(NC(c2ccc(Cc3cncc(C)c3)cc2)=O)nn(C)c(Cl)c1C(F)(F)F 45410,N1(C(S(CCCOC)(=O)=O)=O)CC2CC1CC2CNC(c1ccc(SC)cc1)=O 45411,C(C)(C)(C(F)(F)F)OCC(=O)NC(C)CN(C)C(n1cc(C2CCC2)cn1)=O 45412,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(=O)CC(=O)NC3CC3)C2)C1 45413,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45414,C=C1CCN(C(c2ccn(CCNC(=O)Cc3nocc3C)c2)=O)C1 45415,C1(CC(=O)NC(CC)CN(C)C(C2CCC(F)CC2)=O)SC2=NCCN2C1=O 45416,C1(NC(C2(C=C)CCC2)=O)CCN(C(c2c(C(F)(F)F)cnn2C)=O)CC1F 45417,Cc1c(CNC(=O)NC2CCCSCC2)nnn1C 45418,Cc1nn(C)cc1CCNC(=O)C(C1(O)CN(C(C2CC2C(N)=O)=O)C1)F 45419,N1(C(c2c(C)nsc2)=O)CCC(C2CCN(C(C3CC3CC(C)(C)C)=O)CC2)CC1 45420,C(=O)(C1=CCCCCC1)N1C(C)CC(CNC(=O)C(O)C2CCCC2)C1 45421,C1(NC(CCC(C)OCC)=O)CCN(C(=O)CSC(C)(C)C)CC12CCC2 45422,C(=O)(C1=C(C)OCCS1)N1CC(C(N2CCC(O)(CCC)CC2)=O)N(C)CC1 45423,N1(CC(=O)N(C2CCN(C(C3CC(C(C)C)C3)=O)C2)CCOC2CC2)CCOCC1 45424,C1(OC)CC(NC(=O)CCCCCF)CN(C(c2[nH]c(C)c(C)c2C)=O)C1 45425,N1(C(C=CC(=O)NCC=CCOCC)=O)CCC2(CC1)C(C)(C)C2 45426,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45427,N1(C(C(CC(C)C)O)=O)CCc2sc(C(N3Cc4ccc(F)cc4C3)=O)nc2C1 45428,c1(OC)cc(N(C2CNC2)Cc2ccc(C(C)C)cc2)nc(C(F)(F)F)n1 45429,C12(OC)CCC(C(=O)NCCC3CN(C(=O)CCF)C3)(CC1)CC2 45430,CON(CCO)C(=O)CC1CCN1C(C1C2CC(=O)CC12)=O 45431,N#Cc1ccc(NC(C2C=CCN2C(C2(N(C)C)CCOC2)=O)=O)cc1 45432,C1(C(N2CCC(CC)C2CNC(c2ccncc2Cl)=O)=O)CC2CCC(C1)C2O 45433,c1(C(N2C(C(N3CC(C(C)C)OCCC3)=O)CCCC2)=O)cccc2ccnn12 45434,c1(C(=O)NCC2CCN(C(c3ccc(N)c(F)n3)=O)C2)cnc2c(c1)CCCC2 45435,c1(C(N2C(C(N3CCC=C(F)C3)=O)CC3CC32)=O)cccc(C(F)F)c1F 45436,CC(C(=O)N1CC(CNC(=O)CCc2cncnc2O)C(C)(C)C1)S(N)(=O)=O 45437,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)C(F)=C1CCCC1)C2 45438,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45439,Cc1cc(Cl)oc1C(=O)NCCC(C)N(C)C(c1cc(CO)ccn1)=O 45440,Cc1cn2c(CC(=O)NC(c3ccc(F)cc3)CNC(c3ccsn3)=O)csc2n1 45441,C(CC1=CCN(C(c2n[nH]c(C)c2N)=O)CC1)NC(C1(CC)CCOCC1)=O 45442,C1(NC(CC2CC(=C)C2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1F 45443,C#Cc1cc(C(=O)NCC(C)NC(=O)C(C)C2CCC2)cc(F)c1 45444,N1(C(CCC=C(C)C)=O)CC(NC(C2(O)CCC2)=O)CC12CCOC2 45445,C(=O)(CC(C)C(C)(C)NC(c1cccnc1S)=O)N1CCC(C#C)C1 45446,N1(C(c2cn(C)nc2-c2ccncc2)=O)CC2CCCC1(CO)C2 45447,C1(OCC(=O)NCc2cccs2)CCOCC1.CCC(CNC(=O)CSC)N 45448,c1(CC(C)NC(CC(C)(C)CNC(=O)CC23CCCC2C3)=O)ccccc1Br 45449,c1(OC)ccnc(N(C)Cc2ccccc2-n2cc(C(C)N(C)C)nn2)c1 45450,C1(CNC(c2c(CC)c[nH]n2)=O)CN(C(c2cc(C)oc2C)=O)CC1C(F)(F)F 45451,Cc1nc(CNC(=O)CC2CCN(C(c3cnn(C4CCCCC4)c3)=O)C2)c(C)[nH]1 45452,C(=O)(CCCC(C)(C)C)NC(CC#C)CC(=O)NC(CO)CCC1CC1 45453,C1(CNC(c2cn(CC(C)C)nc2)=O)CC2CN(C(C3CC4CCC3O4)=O)CC12 45454,CC(CNC(=O)C(=O)NCCC(F)F)(C1CC1)NC(=O)CC1CCCO1 45455,C1(C(=O)NCCC2N(C(C3C(C)C3)=O)CCC2)(CC2CCCCC2)CCCCC1 45456,O=C1CC2(CCN(C(C3CC(NC(=O)CCc4nc(O)n[nH]4)C3)=O)CC2)CN1 45457,C12(CNC(c3c(OCC)nccc3)=O)CCCC1N(C(=O)CSC1CC1)CCC2 45458,N1(C(C2CC=CCC2)=O)CCN(C(C2CCc3nccn3C2)=O)C2COCC12 45459,C1(NC(C2(NC(CN(C)CC)=O)CCC2)=O)CC(C)N(C(c2ccccc2)=O)C1 45460,c1(C(=O)NCCC2(NC(c3cc[nH]c3C3CC3)=O)CCC2)ccn(C(F)F)n1 45461,C12(N(C)C)CC(C1)N(C(=O)OC(C)(C)C)C2.N12CCCCC1CNCCC2 45462,c1(C(N(CC(C)(C)CNC(=O)CC2(COC)CC2)CC)=O)cn2cc(C)sc2n1 45463,Cc1ccc(CN2CCN(C3CCCC3(C)C)CC2)c([N+](=O)[O-])c1 45464,c1(C(=O)NC2(CO)CN(C(c3ccnc(C)n3)=O)C2)cccc2nccn12 45465,C1(CNC(c2cnc(CC)[nH]2)=O)CC(OC)CN1C(=O)CCc1nc[nH]n1 45466,N1(C(C2C(C)C2C)=O)CCC2C(CCCN2C(c2ccc3cccnn23)=O)C1 45467,c1(C(=O)NCC2C3CN(C(C(C)OC)=O)C2C3)ccc(-n2cnnn2)cc1O 45468,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45469,Cc1nn2ncccc2c1C(=O)NCCC1(CNC(=O)CCCCC(N)=O)CC1 45470,CCC(CNC(c1c[nH]c(=S)cn1)=O)(CC)C(=O)NC1CCCCC1C#N 45471,Nc1nc(C(N2CCC(CNC(C3CC(O)(c4ccco4)C3)=O)C2)=O)ccc1O 45472,c1(CCC(=O)NC2CC(F)(CNC(c3nc(COC)oc3)=O)C2)ccc(Cl)nc1 45473,C1(NC(N(C2CC2(C)C)CC)=O)(CF)CCN(C(=O)C(C)C2CCCC2)C1 45474,Cc1c(C(N2CCOCC2CNC(=O)CCc2ccccc2)=O)ncn1C 45475,C(CO)(C(=O)NC1(CCO)CN(C(C2CC2F)=O)C1)OC 45476,Cc1ccc(C(=O)Nc2ccc(C(N)=O)nc2)c(Cl)c1Cl.C12CCCC1C(=O)N2 45477,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 45478,C1(NC(C(=O)NCC(CC)C(=O)OCC)=O)CC2CCC(C1)S2 45479,C(=O)(C(=O)C(C)CC)N(CC(CC)NC(=O)Cc1ncn(C)c1C)CC 45480,c1(CC)ccoc1C(=O)NC(C)(CNC(c1cnoc1C1CCOCC1)=O)CC 45481,C1(O)(CN(C(=O)Cc2cccc(Cl)c2)C)CCN(C(=O)C(O)C2CCCC2)CC1 45482,C1(=O)CCC(=O)N2CCC(C2C)N(c2cnn(C)c2)CCN1C.CCCO 45483,N1(C(Cc2ccc(C)s2)=O)CC(NC(c2cc(C(N)=O)n(C)n2)=O)CC(O)C1 45484,CC1CN(C(=O)COCC2CCCO2)CC1CCNC(c1ccsc1C#N)=O 45485,CC1CC(C(N2CCC(NC(c3nnc(C(C)(C)C)s3)=O)C(C)C2)=O)CC(C)O1 45486,S(=O)(=O)(CCC(=O)NC1CC(NC(=O)C(O)C(C)(C)C)C(O)C1)NC 45487,N1(C(COC(CC)C)=O)CCC1C(=O)NC1(CC(N)=O)CC1 45488,c1(O)ccc(O)c(CO)c1.c12nc(c(C)o1)C(=O)NC(CCOC)CNC2=O.CC 45489,N1(C(c2c(C(C)C)cccc2)=O)CC2CCN(C(=O)C(F)n3ccnc3)CC2C1 45490,Cc1ccc2c(N3CCCC4(CC3)CC4(F)F)nc(=NCC3CN(C4CC4)C3)[nH]c2c1 45491,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45492,CC1CCc2ncc(C(N3CCC(C(O)C(F)(F)F)CC3)=O)n2C1 45493,N1(C(c2nc(C(C)=O)sc2)=O)CCCC1(C)CNC(=O)CCS(C)=O 45494,C1(CNC(C(CC)C)=O)CCN(C(=O)Cc2cccc(NS(C)(=O)=O)c2)C1(C)C 45495,C12(C(N(C(C)CN(C(=O)C3=COCCC3)C)C)=O)CC(C)(C1)OC2(C)C 45496,C1(C(N2CC3C(NC(C(=O)NCCOC)=O)C3C2)=O)CC(C)(C)CCO1 45497,C1(CC)CCCC1C(=O)NC12CC(C(N3CCC3(C)C(=O)N(C)C)=O)(C1)C2 45498,Cc1ccc(CCC(N2CC3(C2)CN(C(=O)C(C)Cc2ccco2)C3)=O)c(C)c1 45499,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C(F)(F)F)n1)=O 45500,Cc1ccc(C(=O)N(C)CC2(O)CN(C(=O)C(C)N3CCCC3)C2)o1 45501,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45502,C1(NC(CSCC#C)=O)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45503,c1(C(=O)NC(C2(O)CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C)cc(F)cnc1O 45504,c1(-c2cn(CC(=O)NCCCN3CCCCCC3)nn2)ncc(Cl)cc1F 45505,N1(C(CC2CCN(C(CC(COC)(C)O)=O)C2)=O)CC2(COCC(=O)N2)C1 45506,c1(CCNC(=O)NC(c2c(Br)cn(CC)n2)C)cccc2cnccc12 45507,c1(OC)cc2cc(N(C3CCNCCC3C)C(c3cocn3)=O)sc2cc1OC 45508,n1(CCOCCOC2CC2C(=O)OC)cc(Br)nn1 45509,c1(CNC(N2CC(C)(CC(c3ccccc3)O)C2)=O)ccc(Cl)cc1F 45510,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45511,c1(SC)cc(C)ccc1C(N1CCN(C(=O)C(C)N(C)C)C(COC(F)F)C1)=O 45512,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1C 45513,n1(CCCNC(C2CC(N(C)CC)C2)=O)cc(-c2ncc(C(=O)O)o2)nn1 45514,C1(NC(c2cc(=O)cc[nH]2)=O)CN(C(c2ccnc(S)c2)=O)C2(CCCOC2)C1 45515,CN1N=C(C(=O)NC2CCN(C(c3cc(F)cs3)=O)CC2(C)C)CCC1=O 45516,C1(NC(c2c(C)nn(C)c2C)=O)CC12CCC(NC(C1(F)CCOC1)=O)CC2 45517,C1(F)(C(N2CC(NC(C3C(c4cccc(OC)c4)C3)=O)C2)=O)CC2(CCC2)C1 45518,C=C=C(C)CC(=O)NCC1(F)CCN(C(c2cc(-c3ccccn3)ns2)=O)C1 45519,N1(C(=O)CCc2cc(Cl)sc2Cl)CCC2(CCCN2C(=O)CC2CC(F)C2)C1 45520,N1(C(c2ccc(OC)c(Br)n2)=O)CCc2ccccc2C1CCNC1(C)CC1 45521,N1(C(=O)Cc2nc3ncccn3n2)CCC2C(CCN2C(C2SCCCS2)=O)C1 45522,CCCCC(O)C(=O)NC1(C2CCCN2C(c2cscc2C2CC2)=O)CC1 45523,Oc1ccc2[nH]cc(CN3CC(O)(CNc4cnccc4Br)C3)c2c1 45524,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45525,C(=O)(C(C)C(F)(F)C(F)F)NCCN(C)C(=O)OC(C)(C)C.C12CC(C1)NC2=O 45526,C#CCCN=C(NCCc1ccc(C)cc1F)NCC(O)(COC)CO 45527,C1(NC(C#CCNC(c2n(CC)ncc2)=O)=O)CCCCC1(C)C 45528,CC1CCc2[nH]nc(C(=O)NCCCCCNC(c3cn(CCO)nn3)=O)c2C1 45529,C1(OC)(CNC(=O)C(C)(C)OC)CCN(C(C2COCCC2C)=O)C1 45530,N1(C(CC)=O)CCCC(C(=O)N(C(C)Cc2cncs2)C2CC2)C1 45531,Cc1ccnc(C(=O)NC2CC2CNC(c2ccc(Cn3cccc3)cc2)=O)c1 45532,N1(C(CC(=O)NCC)=O)CCN(C(C2(C)CC(C)=NO2)=O)CC1CF 45533,C1(NC(CCCCCC#C)=O)CCN(C(=O)CN2CCCS2(=O)=O)C12CCCC2 45534,c1(CC)ccc(CC(N2CC=CC(NC(=O)Cc3cnc[nH]3)C2)=O)cc1 45535,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45536,c1(C(=O)NC(CNC(CCNC(=O)OC)=O)(C)C2CCC2)nn(C)nc1C 45537,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)CC1O 45538,c1(N2C(CNC(C3N4C(C)CN(CC4)C3)=O)CC(F)C2)nc(Cl)nc2c1COCC2 45539,N1(C(c2c(NC)nccc2)=O)CCCC(CO)(NC(=O)COCC(F)F)C1 45540,N1(C(c2cnc(CC)s2)=O)CCSCC1N.c1(-c2c[nH]nn2)nccc(C)n1 45541,N1(C(c2n(CCC)ncn2)C(=O)NCc2ccco2)CCCC(O)(C(N)=O)C1 45542,S(=O)(=O)(c1ccc(Br)cc1NCC(c1ccccc1)O)NCc1ccc(C)nc1 45543,CCC(CC)(CO)NC(=O)CCn1cc(CC2N(CC3CCC3)CCC2)nn1 45544,C1(C(=O)OC)CCc2cn(CC3CN(C(=O)OC(C)(C)C)C(C)CO3)nc2C1 45545,c1(-c2cccc(OCC)c2)cccc2cc(C(N3CCn4cnnc4C3)=O)sc12 45546,C1(C(=O)NCC(C2CC2)NC(c2cc(C)sc2)=O)CC2CC1CC2O 45547,C(=O)(C(CNC(=O)CCNC(=O)NCC)N(C)C)N1CCC(CC#C)C1 45548,C1(NC(C2C(C)C2)=O)CN(C(=O)C(c2ccc(Cl)c(F)c2)O)C(C)(C)C1 45549,c1(C(N(CC(C)O)CCNC(c2c(C#C)cn(C)n2)=O)=O)cn2cc(C)sc2n1 45550,c1(CC(=O)NC(CNC(C2CN(C(CC)CC)C(=O)C2)=O)C)cccc(F)c1O 45551,c1(N(C)C)cc(C(=O)NC2CCN(C(c3nccn3C)=O)CC2CO)cc(Cl)n1 45552,c1(N2C(CNC(c3ccc(C(F)(F)F)nc3)=O)CCC2)nc(Cl)nc2sccc12 45553,C1(Nc2n(C)cc(NC(c3cnc(OC)nc3)=O)n2)CCC(C2CC2)C1 45554,c1(C(=O)NC2(CNC(=O)COC(F)(F)F)CCOCC2)ccc2n[nH]cc2c1 45555,c1(CC(=O)NC(C)CCc2cn(CSc3ccccc3)nn2)ccn(C)c(=O)c1 45556,C(=O)(CCNC(C1CN(C(C2CC2(F)Cl)=O)C1)=O)OC 45557,N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1C(=O)NCCCCCN(C)C 45558,N1(C(CCNC(=O)OC)=O)CC(O)(C2CCCN2C(=O)C(O)C2CCCC2)C1 45559,C1(CCN(C)C(C2CCCO2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 45560,C1(Cc2n(C)cnc2)CN(C(C2CCCN(C(=O)C(F)(F)Cl)C2)=O)CCC1F 45561,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCOC2(C)C)=O)CC1(C)C)=O 45562,C(=O)(CC(C)CC(F)(F)F)OC.n1(C(C)C)ccc(CN(C2CCCCC2)C)n1 45563,Cc1ccc(OC(F)F)c(NC(N2CCN(C(=O)CP(C)(C)=O)C3CC23)=O)c1 45564,c1(CC(=O)NC2CC(NCc3cccc(F)c3F)C2)ccc2c(c1)CCO2 45565,c1(C(N2C(CCNC(c3cc(Br)c[nH]3)=O)COCC2)=O)c[nH]c2c(F)cccc12 45566,N1(C(C(C(C)C)O)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45567,CC1(C)C2CCC1(C(=O)NCC1CC(F)(CNC(C3CC34CC4)=O)C1)CC2 45568,CC(C(=O)N(C)CCOCCCN(C)C(C1(C#N)CC1(C)C)=O)C(F)F 45569,Cc1ccc2[nH]cc(C(=O)NCCN(CC(=O)NCCN3CCC(O)C3)C)c2c1 45570,C1(CC)CN(C(C)=O)CCC1(F)NS(=O)(=O)CC1CC12CCOCC2 45571,c1(C(N2CCC(C(N(CC)Cc3nccs3)=O)C2)c2ccccc2)ccccc1 45572,c1(C(=O)NCC2C(NC(CC3ON=C(C)C3)=O)CC2)cc(F)cnc1Cl 45573,C1(N(C(CC(C)F)=O)C)CCCCC1N(C)C(c1cc(-c2ccccc2)cs1)=O 45574,c1(CN(CCCC=C)C)cc(Cl)cc2ccccc12 45575,c1(OC(C(=O)NC(CSC)C(=O)NC(C)CN(C)C)C)ccc(F)c(F)c1 45576,c1(CC)cc(C(=O)NCC(F)CNC(c2cn(C)cc2C(N)=O)=O)oc1CC 45577,Cc1ncsc1CN(C(=O)Cc1cocn1)C 45578,c1(C(=O)NCC2CC(NC(CC3(C)CCOC3)=O)C2)ccnc(-c2ccco2)c1 45579,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)CN(C)C1CC1)OCC=C 45580,C(=O)(CCCCN(C)C)NCC(C)CNC(c1ccc(=O)oc1)=O 45581,C(=O)(C#CC1CCCO1)NC1CC(OC)CN(C(=O)Cc2cccc(O)c2F)C1 45582,C1(O)(CCNC(COCC(C)C)=O)CCCN(C(=O)CC2CCS(=O)(=O)CC2)C1 45583,c1(C(C2C(C(=O)NC(C3CCCCC3)CNC(=O)CS)C2)=O)ccncc1 45584,C1(n2cc(CSc3cccc(Cl)c3)nn2)OCCCC1Cn1c(C(=O)OC)ccc1 45585,N1(C(CCOCC)=O)C2CCC1(Cn1cc(C3CC3C(=O)O)nn1)CC2 45586,C1(NC(Cc2cc(C)nn2C)=O)CCN(C(=O)CNc2ccccn2)CC1O 45587,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45588,c1(CNC(C2(SC)CN(C(=O)CC3(C)OCCO3)C2)=O)cc(F)ccc1O 45589,N1(C(c2cccc(C(C)C)n2)=O)CC(C2CN(C(C3(O)CC3(C)C)=O)C2)C1 45590,C1(C2CC2)(CNC(C(C)OCCOC)=O)CCN(C(=O)CN=S(C)(C)=O)C1 45591,C1(NC(=O)C=Cc2nccs2)CC(=O)N(C2CN(C(=O)C=CCF)C2)C1 45592,C1(C2CCCOC2)(NC(=O)C(CC(F)F)NC(C2C3CCCCCC23)=O)CC1 45593,C(=O)(CC(O)CNC(c1cc(OC(F)(F)F)c[nH]1)=O)NCC1(SC)CCCC1 45594,N1(C(C(CNC(=O)C(c2ccc(F)cc2)(F)F)N(C)C)=O)CC2OCCOC2C1 45595,N1(C(CNC(=O)OCC)=O)CCC(C(N2CCOC(COC)C2)=O)C(C)C1 45596,C(C(C)(C)CN(C(=O)CCC1(C)CC1(F)F)C)CNC(CCNC(COC)=O)=O 45597,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C2=CCC2)C1 45598,c1(C(=O)NCC2CCN(C(CNC(C)=O)=O)C2)nc(Cl)cc(N)c1Cl 45599,C=CCC(CNC(=O)C(C)=CCC)C(=O)NCCS(C)(=O)=O 45600,Cc1nc(CCNC(=O)C(N)Cc2cccc(F)c2)c(C)o1 45601,C=CCC(CNC(C1CCC(C)(C)CC1)=O)C(=O)NCC1CC=CCN1C 45602,N1(C(c2ccc(C)c(C)n2)=O)CCC(C(N2CC(CF)C2)=O)CC1(C)C 45603,C1(N(C(c2c(CC)ncs2)=O)C2CC2)CCN(C(=O)Cc2nc(CC)cs2)CC1 45604,CCC(CNC(c1cccc(CO)n1)=O)(CC)C(=O)N1OC2CCC1CC2 45605,C=C(Cl)CC(C(=O)NCc1cc(C)ccc1OC)NC(=O)CCCOC 45606,c12cccc(O)c1CNC2.C1(C(=O)OC)CCC(C(=O)N(CCO)CCO)O1 45607,c1(C(C)C)nc(N2CC(NC(=O)CC(C)C(C)C)C(C)(C)C2)cc(Cl)n1 45608,Cc1ccc(C)c(CC(N2CCC(CNC(=O)C=C3CCC3)C(C)C2)=O)c1 45609,C1(NC(CCOCC)=O)CCC2(CC1)CC(NC(=O)C(c1ccccc1F)O)C2 45610,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C2CC2)=O)cccc(C)c1F 45611,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2c1)=O)NC(CC#CC)CO 45612,CC(CC(F)(F)F)C(=O)N1CCC(OCCNC(=O)C(F)C(C)(F)F)C1 45613,CC1CC(NC(=O)COc2ccsc2)CN1C(=O)CC1(C)CC1(Cl)Cl 45614,c1(CNC(C(CC)NC(c2occc2C(C)C)=O)=O)cnc(C)n1CC 45615,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45616,N1(C(C2CCOC(C)C2)C(=O)OCC)CCCNC(=O)C1SCCOC 45617,C12CCN(C(=NCCCCl)NCC1c1cncn1C)C2.C1(CCOC)CCCC1 45618,c1(SC)ccc(NC(N2CCN(CCc3cccnc3OC3CC3)CC2)=O)cc1 45619,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC(O)c1ccccc1)C2 45620,Nc1ccc(C(=O)NCCC2CCCN2C(=O)CN2CCS(=O)(=O)CC2)cc1Cl 45621,C=CC1(C(N2CCC(O)(C(C)CNC(c3scc(C)c3C)=O)C2)=O)CCCC1 45622,c1(C(=O)NC(c2n(CC#C)ccn2)CC(C)C)cc(C)cc(O)c1 45623,N1(C(C(C)NC(C)=O)=O)CCOC(C(C)NC(=O)CC2CC(C)C2)C1 45624,Cc1oc(C2CC2)nc1NS(=O)(=O)CC1CC1(F)F 45625,C(CNC(C1CCC(F)C1)=O)(C(=O)NCCC1CCCCO1)N(C)C 45626,c1(C(=O)NC(C2(O)CCN(C(C3C(=C)C3)=O)CC2)C)cc2sccc2n1CCC 45627,C#Cc1ccc(CNc2cccnc2C(=O)NC(c2ccccc2OC)C#N)s1 45628,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(c3cnnn3C)=O)CC2)CC1 45629,c1(C(=O)NC2CC(C)N(C(=O)C=C3CCC3)CC2)cncc2ccc(F)cc12 45630,C1(C(F)F)CCC(C(c2nnnn2C2CCCCC2)NCC2CC(=O)NCC2)CC1 45631,c1(CCNC(C(C2CC2)NC(COCCC)=O)=O)cnc(C)cn1 45632,N1(C(=O)NCC(CCC)CCC)CC2CN(CC)CC2C1 45633,c1(C(=O)NCC(CC)NC(c2ccc(C3CC3)cc2)=O)cc2c(nn1)CCCC2 45634,c1(C(=O)NCC2CC=C(C)CC2)cc(C)ccc1F 45635,c1(NC(=O)C(F)CC2CNC2)cnccc1CO 45636,C1(C(C)NC(C(C)OCC#C)=O)CCCN1C(c1c[nH]nc1-c1cccnc1)=O 45637,N1CCC(C=O)CC1.c1(NC(C2CC(C(N)=O)C2)=O)cnc(C2CC2)o1 45638,c1(C(=O)NCC2N(C(C=C(CC)C)=O)CC(C(F)(F)F)C2)ncn2c1CCCC2 45639,N(C(=NCc1ccccn1)N1CCC(Cc2ccsc2)C1)C(=O)Nc1ncccn1 45640,c1(C(N(C2CCCN(C(=O)C3=COCCC3)CC2)CC)=O)ccc(C)c(O)n1 45641,C(=O)(C(C(C)(C)C)N1CCOC1=O)N(CCCCNC(C(C(C)O)N(C)C)=O)C 45642,C1(CN2CCC(C3N(C(C4(O)CCC4)C)CCCC3)CC2)CCN(C)CC1 45643,C#CCC(C)(C(=O)N(CCCCN(C)C)C)NC(=O)CC1CCOC1=O 45644,C1(CC=C)(NC(c2coc(Cl)c2)=O)CCN(C(c2ccc(C3CC3)cc2)=O)C1 45645,N1(C(C2OCCN(C(C3(CC(C)C)CCC3)=O)CC2)=O)C2CCC1CN(C)CC2 45646,c1(C(=O)NC(COC)(C)C)cn2c(n1)CCN(c1scc3c1OCCO3)CC2 45647,C(=O)(C#CC1CCOCC1)NCCCOCCNC(C(CC(=O)OC)C)=O 45648,c1(C(=O)NCC2CC2NC(C2CC3COCC3C2)=O)cc2ncccc2[nH]1 45649,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45650,CCCCC(CC)CC(=O)NC(C(C)N=c1[nH]ncs1)c1ccccc1 45651,C1(F)(CNC(C(C)=C(C)C)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 45652,c1(C(N2C(CNC(=O)C=CC3CCCCC3)CC3CC32)=O)cc(=O)cc(Cl)[nH]1 45653,c1(CNC(c2n(CCOC)nnn2)c2n[nH]cc2Br)c(O)cccc1F 45654,C(C(C)(C(=O)N(C)CCNC(=O)CNS(=O)(=O)NC)OC)OC.C1[NH+]([O-])CN1 45655,C(c1ccc2cccnc2c1)=NC(COCCNC(C#CC(C)C)=O)=O 45656,N1(OS(N2C(CO)CNCC2)(=O)=O)Cc2c(ccc(F)c2Br)C1=O 45657,C(=O)(CCC(C(C)C)NC(=O)C1=C(Cl)CC1)N1CCCC(OC)C1CC 45658,N1(C(C)C)CC(CNC(=O)NCCCc2ccccc2C(F)(F)F)CC1=O 45659,Cn1ncc(C(=O)NC2(C)CC(NC(=O)C(=O)NCC(F)(F)F)C2)c1S(N)(=O)=O 45660,C=CCC(F)(F)C(=O)NCC1COC(C)(CNC(=O)Cn2nnc(=O)[nH]2)C1 45661,c1(-c2ccc(NCN3CCC(c4ncc(C)cn4)CC3)nn2)ccc(Cl)c(F)c1 45662,Cc1cccn2nc(C(=O)N(C3CN(C(C4(C#N)CCCCC4)=O)C3)C)cc12 45663,CC1(C)CC(NCc2nc(Cl)ccc2Br)CN1C(=O)OC(C)(C)C 45664,C1(C(N)=O)CCCC(CNC(=O)C(=O)NC(c2ccccc2Cl)C2CC2)C1 45665,N1(C(=O)CCOC2CCCC2)CCC(C(C)(C)C)(CNC(C23CC(F)C2C3)=O)C1 45666,CC1CC(NC(=O)C(N2CCCC2)C2CCCC2)CN1c1nnc(CO)s1 45667,N1(C(C2CCC(C(=O)OC)CC2)=O)CCSCC(C)C1.N12CCC1C2=O 45668,C1(C)(C(N(CCC(C)(C)C)C)=O)CCCN1C(=O)CCc1ncnn1C 45669,C1(C(=O)NC23CC(CNC(C(COC)O)=O)(C2)OC3C)CCCCC12CCC2 45670,c1(OCC(N2CCC(N(C(C(CSC)(C)C)=O)CC)C2)=O)c(C)ccc(C)c1C 45671,N1(C(c2cn(CC)nn2)=O)CCN(C(=O)CC2OCCC2C)C(CO)C1 45672,N12CCN(CC1)CC(C)NC(=O)N2.C(C)(C)(C)N(CC)CC.C1CN1 45673,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 45674,C1(C(=O)NC2(C)CC(NC(c3ccc(O)c(C(N)=O)c3)=O)C2)CCc2cnnn2C1 45675,c1(OC)ccc(NC(c2nn(C(C)C)c(N)c2C#N)=O)cc1[N+](=O)[O-].C(COC)S 45676,CCCCC(C)CCC(=O)N1CCC=C(C(=O)NCc2cnccc2Cl)C1 45677,C1(CCNC(C(C=CC)O)=O)CC(C)CCN1C(=O)CN(S(=O)(=O)CC)C 45678,c1(C(CC(=O)OC)NC(=O)Cc2c[nH]nc2O)cccc2ccccc12 45679,C1(N(c2n(C)ncc2O)C(=O)CC2NC(=O)NC2=O)CCC2(CC1)CNC2 45680,N1(C(C(C)Cc2cccnc2)=O)CC2C(CNC(=O)C=Cc3cnc[nH]3)C2C1 45681,c1(CC(C(=O)C(O)Cc2ccccc2)=O)ccnc(O)c1.C1(N)CC(N)C1 45682,C1(C(=O)NCC2CCN(S(=O)(=O)Cc3ccccc3)C2)CCC12CCC2 45683,C1(N(C(Cc2nc(OC)sc2)=O)C)CCC(NC(=O)CCc2ncc(C)[nH]2)CC1 45684,N1(C(CNC(=O)NC)=O)CCN(C(=NCCF)NCCc2ccccc2)CC1 45685,c1(CC(=O)NCC=CC(N2CCC(CF)CC2)=O)ccc2c(c1)CC2 45686,N1(C(CC2(OC)CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C2(CCC2)C1 45687,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 45688,C(=O)(C(C(C)C)NC(=O)C(C)CC1CCCC1)NC(CC#C)(C)C 45689,Cc1cc(C(=O)NCC(CNC(=O)CCN2CCCC2=O)CO)on1 45690,C1(CC(C)NC(c2cc(F)n[nH]2)=O)CCN(C(C2(C)CC=CC2)=O)CC1 45691,N1(C(CC(=O)OC)=O)CCC2(CC1)CC(NC(=O)C(CC1CCCC1)C(C)C)C2 45692,Cc1ccc(F)c(CC(=O)NC2CCC(NC(=O)C(F)C3CCC3)C2)c1 45693,C1(CCOC)(C(=O)NCC(O)CNC2CCC(c3ccccc3)C2)CCCC1 45694,N1(C(C=CCNC(C2CCC(C3CC3)C2)=O)=O)CCC2(CCOCC2)C1 45695,c12ccccc1CCNC2=O.C(=O)(COCC(F)F)NCCCCNC=O 45696,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 45697,CCCC(C)CCCC(=O)N1CC2(NC(C3CC3CCOC)=O)CCC1CC2 45698,c1(C(=O)NCC(CN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C)O)ccnc(Cl)c1N 45699,CC1CCC(C(=O)NC2CCCC(CN3CCCC3)C2)CC1.C12(CCC1)C(=O)N2 45700,C1(NC(C2CCCN(C)C2)=O)COC2(C1)CN(C(c1ncnc(O)c1F)=O)C2 45701,c1(C(N2CCC3CN(C(C4C(C=C)OCC4)=O)CC32)=O)cnc2ccccc2n1 45702,c1(OC)cc([N+](=O)[O-])ccc1-c1ccc(C(F)(F)F)cc1C(F)(F)F 45703,C1(=O)C2=CCC(C2)N1.c1(CN(C)C(C2CC2C(C)(F)F)=O)nnc(O)o1 45704,CCC(Cc1ccccc1C)C(=O)OCCOc1cnc(C)s1 45705,N1(C(C2(C)CC2(F)Cl)=O)C(CNC(C2CCCO2)=O)CC2COCC12 45706,c1(C(=O)OC)ccc2ccc(NC(C3CC(F)CN3C(C)=O)=O)nc2c1 45707,CC#CCC(C(=O)NCc1ncccn1)NC(=O)CN1CCCCCC1 45708,CC(CN=c1[nH]c(=NC(C)c2nccs2)[nH]c2ccc(Cl)cc12)N1CCCC1 45709,N1(C(C2C(=O)OCC2)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 45710,C(=O)(C(C)CC(F)(F)F)N1CC(O)(CN(C(C(C)C)=O)C)C1 45711,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(CC)=CC)=O)C(C2CC2)CC1 45712,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 45713,C1(NC(c2c(OCC)con2)=O)COCCC1NC(=O)OC(C)C 45714,C1(C(F)(F)F)(C(=O)NC(C)(C)CCNC(=O)CC2C=CCCC2)CCCCO1 45715,c1(C(=O)OCC(c2ccc(C3CCOC3)s2)=O)cccc2[nH]ncc12 45716,c1(C(=O)NCCC2(NC(c3c(C)coc3)=O)CC2)cccc(N(C)C)n1 45717,N1(C(=O)CC2CC(C3CC3)C2)CC2(CCCC2)C1C(N1CC2(CO)CCC1CC2)=O 45718,c1(N2Cc3c(C)cccc3C2)[nH]c(=NCc2ccc(Br)o2)nc2scnc12 45719,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(=O)C=Cc3ccc(C)o3)C12 45720,c1(NC(C2(C)CN(C(=O)C(O)CCl)C2)=O)ccc(S(=O)(=O)c2ccccc2)nc1 45721,N(C(=NCCC(C)(C)S(C)(=O)=O)NCC1CC(SC)C1)CCOCC 45722,N1(C(C2(OC)CCSC2)=O)CC(CNC(=O)CCc2nc[nH]n2)C2(CCC2)C1 45723,c1(OC(C)C(=O)N(CC(C)NC(C2CCCCC2)=O)C)cccc(Br)c1 45724,CC1CCN(C(=O)CN2CCC(C)(O)C2)CC1CNC(C1CCC(C2CC2)O1)=O 45725,c1(CCCC(=O)NC(CNC(C2CC3(CC3)CO2)=O)C2CC2)ccc(Cl)c(Cl)c1 45726,c1(C(=O)NCC(C)CN(c2ccnn2CC(F)F)C)cnc2ccccc2n1 45727,N1(C(CSCC)=O)CCSC(C(=O)NCCc2nc[nH]n2)C1 45728,C1(CC(N2CC(CC(C)NC(=O)C=Cc3nccs3)C2(C)CO)=O)CCN(C)C1=O 45729,C1(NC(c2ncn(CC)c2)=O)CCN(C(c2ncsc2C(F)(F)F)=O)CC1(C)C 45730,c1(C(N2CC(O)(c3cn(CC4CCCCC4)nn3)C2)=O)cc2ncccn2n1 45731,C1(C(=O)NC(C2CN(C(=O)CCc3ccc(Cl)nc3)C2)C)CCOC(=O)CC1 45732,C1(c2n(CCOC)nnn2)(NC2CC(n3cncn3)C2)CCCC1CN(C)C 45733,Cn1cnc2cc(C(=O)NCC3CCCN(C(c4cc(C(N)=O)co4)=O)C3)sc12 45734,C1(CNC(C(C)(C)CC(F)F)=O)CN(C(=O)C(O)C2CCCC2)C2(CCOCC2)C1 45735,c1(OC)ccc2c(c1)C(NS(=O)(=O)CCCN1CCN(C)CC1)CCC2 45736,CN1CC(O)CCC1C(N1CCC2(CC2C(=O)NC2CC3CCC(C2)O3)C1)=O 45737,C1(CNC2CCC(O)(c3ccccc3)C2)CNC2(CCOCC2)C1 45738,N1(C(=O)CCN2CCOCC2)CC2CCN(Cc3ccc(O)c(O)c3Cl)C2C1 45739,C1(CNC(c2ccc(C)o2)=O)CC2(CCN(c3ncncc3Cl)C2)CO1 45740,Cn1cnc2sc(C(=O)NCC3(O)CN(C(C4(O)CC(C)(C)C4)=O)C3)cc12 45741,c1(C(N2CCC(NC(C(C)(C)F)=O)C2)=O)cc2ccc(Cl)cc2c(=O)o1 45742,N1(C(C(CC)(CC)OC)=O)CCOC2(CCN(C(=O)C(C(C)C)OC)C2)C1 45743,C1(NCCNC(=O)Nc2ccccc2)CCCC(N)C1 45744,C1(CC=C)(NC(c2ncoc2C2CCCO2)=O)CN(C(C2(F)CC=CC2)=O)C1 45745,C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(C1CC(C)(c2ccccc2)C1)=O 45746,CC1CCN(C(=O)CCCNC(c2ccc[n+]([O-])c2)=O)CC1C(F)(F)F 45747,N1(C(c2c(C)csc2)=O)CC2CC(NC(=O)Cc3cc4ccccc4o3)C(C2)C1 45748,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 45749,C=CCC(C(=O)N1CCC(F)(CNC(c2cccc(C)n2)=O)C1)C(C)(C)C 45750,CC1(C)CCN(C(c2ccc3sncc3c2)=O)CC1NC(=O)CCc1cncnc1 45751,c1(CC(=O)NCCCCN(C)C(C2CC2C(C)(C)C)=O)ccc(S(C)(=O)=O)cc1 45752,CCC(=O)CCC(=O)N1CC(C)(CCC(N2CCC(CO)(CO)C2)=O)C1 45753,CC(C)CC(O)CC(=O)NCC1(O)CC2CCC(C1)N2C(=O)CC(C)O 45754,O=C1CCN(C(c2cccc(C3CC3)c2)C(=O)NCC2CC2)CCN1 45755,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCOc1cccc(Cl)c1)OCC 45756,c1(C(=O)NC2(C(C)C)CCN(C(C3CC3F)=O)C2)cc(Cl)cc(C(F)(F)F)n1 45757,c1(CC(N2CCC(NC(C(CC)(C)COC)=O)C2)=O)cc(F)c(F)cc1Br 45758,CC1(c2ccc(NC(C3CN(c4ncncc4I)C3)=O)cc2)NC(=O)NC1=O 45759,c1(C(=O)OC)ccccc1CCC(=O)NCC1(F)CN(C(=O)CC2OCCO2)C1 45760,c1(C(=O)NC2CC(NC(C(C(C)c3ccccc3F)O)=O)C2)cc(C#N)ccc1F 45761,C(CC(C(C)(C)C)NC(=O)Cn1ncnn1)N(C(C(CC#C)C)=O)C 45762,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 45763,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCCCCN(C)C)C2(CCC2)C1 45764,C=CCC(C)C(=O)NC1CC(CO)N(C(c2cc(Cl)c(Br)s2)=O)C1 45765,N1(C(C2(C(N(C)C)=O)CC2)=O)CCC2(CCCN(C(c3ccn(C)n3)=O)C2)C1 45766,c1(C(N(CCNC(C2CC2c2cccc(C)c2)=O)CC)=O)ccc2nn[nH]c2c1 45767,c1(C(N2CC(O)(CCNC(C3(C(C)C)CC3)=O)C2)=O)ccnc(Cl)c1Cl 45768,C1(C(=O)NCCCN(C(c2cnc(S)nc2)=O)CC)CCCC2(CC2)C1 45769,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(F)CNC(C)=O)C2 45770,C1(NC(c2cc3sccc3[nH]2)=O)CC2(NC(C3CC4CC4C3)=O)COC1C2 45771,C12(C(N(CC(CC)O)C3CC3)=O)CC(C)(CN1C(c1cc(C(N)=O)c[nH]1)=O)C2 45772,C(=O)(C1CCc2nccn21)N1CCN(C)CC1C(=O)NC1CCCCCC1 45773,C#Cc1cncc(C(=O)NC(C2CCCCN2C(=O)C(C=C)CC)C)c1 45774,C1(C(=O)N(C)Cc2ccn(C)n2)(NC(C2CC(=C)C2)=O)CCN(C)C1 45775,c1(OC)ccc(C(C)N(C2C3CCC(C3)C2N)C2CC2)c(OC(C)C)c1 45776,N1(C(CCN(C(c2c(C)nccc2)=O)CC2CC2)=O)CC2(CCC2)CCC1CO 45777,CC(C(=O)NNC(=O)CCCn1cc(CN(C)C)nn1)NC(C1CCCCO1)=O 45778,N1(C(C2CCC(CN(C)C)O2)=O)C2CCC1CN(C(C1CCC3(CCC3)O1)=O)C2 45779,C1(CNC(CCC(C)SC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 45780,C1(C(=O)OC)C=CCCN1C(=O)CCC1(C)CN(C(=O)CCOC(C)C)C1 45781,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 45782,N1(C(C(CC=C)(C)N(C)C)=O)CCOC2(C1)CN(C(C1CC1C(C)C)=O)C2 45783,CC(=O)CCC(=O)NC1CCCCC1N(C)C(c1cscc1Cl)=O 45784,c1(CNC(CCC2N(C(COCCSC)=O)CCC2)=O)cccc(O)n1 45785,C1(C(=O)NC(C(=O)NCCN(CCOC)C)CO)CC2(C1)CC2(F)F 45786,c1(CC)cccc2sc(NC(C3CC4(CCOC4)C3)=O)nc12.CCC 45787,C(CCCCC(=O)NC(C)CC1(O)CCN(C(c2cc(CO)n(C)n2)=O)C1)OCC 45788,C(=O)(C(C)(C)C(O)C(C)C)N(C1C2CCN(CC=Cc3ccccc3)CC12)CC 45789,C1(NC(CC2C(C)(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 45790,C1(C(=O)OCC(=O)Nc2ccc(C)cc2)CC2OC(C)CC12 45791,O=C1CC(C(=O)NC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C2CCC2)=NN1 45792,C1(N(C(C(C)O)=O)C)CCCN(C(c2cccc(Br)c2)C2CC2)C1 45793,Cc1cc(CNCC2CCCCN2C(C2(O)CCSC2)=O)n(C)n1 45794,N1(C(C(C)C2CC2)=O)CCC(C2CC2)(CNC(c2ccc3nc[nH]c3n2)=O)C1 45795,C(=O)(C(F)CC(CC)CC)N1C(CC)(CNC(C23CCN(CC2)CC3)=O)CCC1 45796,N1(C(c2n(CC)ncc2)=O)CCC2CC2(C(=O)NCc2n[nH]c3c2CCC3)CC1 45797,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 45798,NC(=O)CCC(C(=O)NC1CCCC1)n1cc(C(n2cccn2)C2CC2)nn1 45799,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 45800,c1(C2(C(=O)NC(C3CCCC3)CO)CNC2)ccccc1Cl 45801,C1(NC(C2CC(=C)C2)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2F)=O)C1C 45802,C(=O)(C1=CCC(C)(C)CC1)NC12C(CN(C(C(CC=CC)CC)=O)C1)C2 45803,c1(C(=O)NCc2ccc(CN(C(CSCC)=O)C)cc2)coc2c1COC2 45804,C(=O)(CCCC(F)(F)CO)NC1(C)CCN(C(c2cc(NC(C)=O)ncc2)=O)C1 45805,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 45806,c1(CC)ccc(CCC(=O)NC2CC(CNC(C3CCN(C)CC3)=O)C2)cc1 45807,c1(CCOC)nc(=NC2CCCC(NC(C3(O)CCSCC3)=O)C2)s[nH]1 45808,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(c3c[nH]c(=N)s3)=O)C2C1)=O 45809,C(C(CNC(=O)C(C1CCC(=O)N1)C)S(C)(=O)=O)NC(C1(CC)CNC(=O)C1)=O 45810,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)N(CC2CC2)CC2CC2)CCC1C 45811,O=C(C1CCCc2cncn21)NCCC1(O)CN(C(=O)CC2CC2)C1 45812,c1(NCC(CC=C)(C)CO)nc(-c2ccco2)nc2cc(OC(C)C)ccc12 45813,C1(NC(C2N(C(C(CC)C)=O)CSC2)=O)CN(C(=O)COC)C2(CCCCC2)C1 45814,c1(C(=O)NCC#CCNC(CC2CCCC(C)C2)=O)c(F)cccc1Cl 45815,Cc1ncc(C(=O)NCC2(CO)CC2)cc1CCNC(C1(O)CC1)=O 45816,Cc1c(NCC2CCN(CC(C)C)C2)ncnc1N(C)CCOCCO 45817,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 45818,C1(C(=O)NC2C(OC)CN(C(COCC=C)=O)C2)CCCC(C)(C)O1 45819,c1(OC)ccc(C(N2CCCC2CC(C)O)C(=O)NCC2CCCO2)cc1Cl 45820,C(=O)(CC(C)(O)C(F)(F)F)NCC1CCN(C(c2ccc(CC)cc2C)=O)C1 45821,c1(N2CC3(C(CNC(C4=C(C)OCCS4)=O)CC3)C2)c(C)cc([N+](=O)[O-])cc1F 45822,c1(C(=O)NC2CC(CCC(=O)NCc3nccc(C)c3)C2)ccc2nc[nH]c2c1 45823,c1(C(=O)NCC2CC(O)(CNC(C(OC)OC)=O)C2)nc(C)ccc1F 45824,C(=O)(C1CCCn2nccc21)N(CC(C)(C)CNC(=O)COC1CCOC1)C 45825,c1(OCC)cnccc1C(F)(F)F.c12ccc(s1)c(=O)[nH]c2=O 45826,c1(C(=O)NC2CC(C)(CNC(=O)Cn3cnccc3=O)C2)ccc(F)cc1N 45827,n1(CC)nnc2cc(C(=O)NCC3(CNC(=O)C(C)CC(C)(C)C)CC3)ccc12 45828,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 45829,CC1CC(NC(=O)Cc2cc(F)ccc2O)CCN1C(c1nc(Cl)cs1)=O 45830,c1(C(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)ccc2nc[nH]c2c1F 45831,c1(CC(C)C(=O)N2CCCC2CN(C)C(c2cccs2)=O)ccc(F)cc1F 45832,C1(=O)CCC(C)O1.N1(CC(=O)O)CCCC(C)C1.C(COCC)OCC 45833,C1(NC(CCC(=O)NCC)=O)CCCN(C(C2CC2c2ccccc2)=O)CC1F 45834,c1(C(CC)C(=O)N(C(C)CN(C(=O)COCC(=O)NC)C)C)c(C)noc1C 45835,C123CC4CC(CC(C4)(C1)C(=O)N2)C3.CC(O)C(C)O.C1(C(=O)N)(C(=O)N(C)C(C)C)CC1 45836,C1(NC(c2c(CC)noc2)=O)C=CCN(C(c2ccccc2OCC(N)=O)=O)C1 45837,c1(C(=O)NC2CN(C(c3cc(C#N)ncc3)=O)C2)ccc2ccnc(O)c2n1 45838,C1(CNC(CC(=O)NCC)=O)CN(C(C2CCC(O)C2)=O)C(C)(C)C1 45839,N1(C(c2ccc(C)o2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C1C(C)C 45840,c1(C(N(C2CCN(C(=O)C(N3CCCC3)C3CC3)C2)C)=O)ccc2[nH]nc(Cl)c2c1 45841,c1(C(=O)OC2(COC)CCOC2)cc2c(OC)c(OC)ccc2[nH]1 45842,O=C1COc2ccc(CN(Cc3ccccc3)Cc3cncs3)cc2N1 45843,C1(CNC(C=CC=CC)=O)(CO)CC12CCN(C(C1CCC(=O)N1)=O)CC2 45844,CCCC(C(=O)N1CCN(C(C23CCCN(CC2)C3)=O)CC1CO)C(C)C 45845,N1(C(C2CC2C(F)(F)F)=O)CC(C)CCC1=CCNC(C)=O.C(=O)(C(=O)N)NC 45846,c1(NC(C(=O)NC(C2CCOCC2)CC)=O)ccc(-c2ccc(F)cc2F)cc1C 45847,CC1(C)CN(C(c2cc(Cl)ccc2O)=O)CCCN1C(c1csc(=N)[nH]1)=O 45848,C(=O)(CS(=O)(=O)Cc1ccc(Cl)s1)NCCN1CCN(C(CS(CC)=O)=O)CC1 45849,N1(C(c2c(SCC)nccc2)=O)CC2(C1)OC1(CO)CC2(NC(=O)CCCF)C1 45850,CC(CCCNC(c1csc(F)c1)=O)NC(=O)CCc1ccc(Br)s1 45851,NC(Cc1cnc[nH]1)C(=O)N1CCCC1CNSc1ccccn1 45852,C1(CC)CCCN(C(C2CN(C(C)C)C2)=O)C1C(=O)NC1CN(C)CCC1O 45853,C1(CC)CCCCN(C(C23CC(CO2)N(C(=O)CCc2cn(C)cn2)C3)=O)C1 45854,Cc1cccc(NC(C2CC2C(=O)Nc2cnc(Br)nc2)=O)c1C 45855,C=CCCC(C(=O)NC1(CO)CC(OC)C1)NC(=O)CCCCC=CC 45856,c1(C(N2CCC(O)(CCNC(CN(C)CCO)=O)C2)=O)cc(=O)n2nccc2[nH]1 45857,C1(NC(CN(CCC)C(C2CN3CCN2CC3)=O)=O)CCCCC1C#N 45858,C1(C(=O)NC(c2cscn2)C)CCN(C(=O)C(C)NS(C)(=O)=O)C1 45859,N1(C(c2ccc(C(C)C)cn2)=O)CCC(C)C(N(C(=O)CCN2CCCC2)C)C1 45860,CC1CCC(CNC(c2cnn(CCn3cc(CCC#N)nn3)c2)=O)CC1 45861,C(CC(C(=O)N(C1CCCN(C(c2csc(C(F)F)c2)=O)C1)C)OC)OC 45862,CC1(C)OC(=O)NC1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC(N)=O 45863,c1(OC)c(C(=O)NCC2(NC(=O)CC3(CSC)CC3)CCC2)sc(Cl)c1Cl 45864,C=C(C)CC1C(=O)NC2CC3(C(C3)C(=O)N1)C2.C1(=O)C(C)N1.OC 45865,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCC2(CC2NC(=O)C2=C(Cl)CCC2)C1 45866,N1(C(N(C)CCN(C)C(C2(C(N)=O)CCC2)=O)=O)CCSC(C)(C)C1 45867,C1(C(=O)NCC(C)(C)Nc2nc(C3CCCC3)ns2)CCc2c[nH]nc2C1 45868,C(=O)(C(CC(F)F)Nc1nc(C)cs1)NCC1C(NC(C(OC)OC)=O)CC1 45869,C1(C)(C(=O)NCCc2cn(C)nc2)CCCN1C(=O)C(N)=O 45870,C=C(Cl)CC(C(=O)N1CC(c2ccon2)C1)NC(=O)C(CCC)CO 45871,C1(C(N(C)CCNC(c2cnn(-c3ccccc3)c2)=O)=O)CCCC(C2CC2)O1 45872,C1(CC(=O)NCC(c2ccc(F)cc2)NC(CC=C)=O)CCS(=O)(=O)CC1 45873,C1(C(=O)NCC2(CN(C)C(c3ccco3)=O)CC2)CCC(CO)CC1 45874,C1(C(=O)NC2CC(NC(c3cn(C)nc3Cl)=O)C2)COC2(CCC2)CO1 45875,c1(-c2ccc(COC)cc2)ccc2c(Cl)c(C(=O)Nc3nc(C)co3)cnc2c1 45876,CN1CCCC(C(N2CCC(CO)(NC(=O)COCc3ccccc3)C2)=O)C1 45877,c1(C(=O)Nc2cc(C(=O)NC(c3nccs3)C)n(C)c2)cc(F)c(F)c(F)c1C 45878,c1(C2(C(=O)NCCNC(C3C=CCN3)=O)CC2)cccnc1 45879,N1(C(CC#C)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1Cl)=O 45880,c1(C(=O)NCC(C)N(C(c2ncsc2Br)=O)CC)c[nH]c2cc(C)ccc12 45881,C(=O)(C(CC(C)C)N(C)C)NC1CC(N(C)C(c2sccc2C(=O)OCC)=O)C1 45882,c1(C(C(=O)NCC(=C)C)N(C2CC2)C(C)C)ccc2nsnc2c1 45883,C1(CC=C)(NC(=O)Cc2ccnn2C2CCCC2)CN(C(c2cc(Br)c[nH]2)=O)C1 45884,N1(C(c2cccc(CC)c2)=O)CC(C)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CC1C 45885,CCCCCCCCC(C)CC(=O)N1CC(CO)(NC(=O)C=CCO)C1 45886,C1(CNC(C2(OCC)CCC2)=O)CC2CCC1N2C(=O)Cc1ccccc1OC 45887,N1(C(C2C(C)C2)=O)CC(NC(c2cncc(Cl)c2)=O)C2(CCS(=O)(=O)CC2)C1 45888,N1(C(C2(COC)CC=CC2)=O)CC(CCNC(c2nn[nH]c2Cl)=O)OC(C)C1 45889,Cc1c(C(=O)NCCN(C(c2cn(CCC(C)C)nn2)=O)C2CC2)cccc1Br 45890,C=CCC(C)(CC)C(=O)Nc1cc(-c2ccc(CC)[nH]2)c(C)cc1F 45891,C1(C(=O)OC)(NC(C2CCCN2Cc2ncc(C(F)(F)F)[nH]2)=O)CCOC1 45892,C1(CC(=O)N(CC(N2CC(O)(CC=C)C2)=O)CC2CC2)CCC(=O)NC1 45893,c1(NC(C2(C)CN(Cc3cncnc3)C2)=O)ccc(F)c(F)c1Br 45894,C1(NC(c2c(CC)cccc2)=O)CCN(C(c2nn(C)cc2C)=O)CC1CO 45895,C1(NC(c2cc(CC)sn2)=O)CCCCC1CC(=O)NCCC(O)C1CC1 45896,C1(SCC)CCCCN1C(C=Cc1ccccc1)C(=O)NCCC1CC1 45897,c1(C(=O)NCC2C(NC(C3CC(CC)C3)=O)CCC2)cc(CS(C)(=O)=O)c(C)s1 45898,N1(C(=O)CCCF)CCN(C(=O)C(c2cc(F)cc(Cl)c2)C2CC2)CC(O)C1 45899,c12nc(ncc1OC)N1C(=O)NC(C1=O)CN2C.c1(CC)cc(C(C)=O)ccn1 45900,N1(C(C2(F)CCN(C(C(C(C)C)OCC)=O)CC2)=O)CCC2CCCC2CC1 45901,c1(NCC2(N(C(C)C)Cc3cccc(Br)c3)CCOC2)c2c(nn1C)CCSC2 45902,C1(C(=O)NCC(C(N2C(CO)CC(OC)C2)=O)CC2CC2)CCC2(CC1)CC2 45903,CCCCC(C)(F)C(=O)NC1CC(CCC(=O)NCCC(C)(O)C2CC2)C1 45904,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 45905,c1(N2CCC(CNCc3cc(C)sc3)C2)ncnc2cnn(C)c12 45906,CC(C)CC(C)CC(=O)N1CC(C)(OC(F)F)C1.c12cc(ccn1)OCC(=O)N2 45907,c1(OCOC)ccccc1S(=O)(=O)NC1CN(c2cc(C)nc(C)n2)C1 45908,N1(c2nnc(C)o2)CCc2c(CNC(C3CCCNS3(=O)=O)=O)cccc2C1 45909,C1(C)(CNC(CNS(NC)(=O)=O)=O)CN(C(c2nc(O)nc(O)c2F)=O)C(C)(C)C1 45910,CC(C)(C(=O)N(C1CCC2(CCC2)O1)C1CCN(C(=O)CCP(C)(C)=O)C1)S(C)(=O)=O 45911,CCCCCC(F)C(=O)NCC1CCN(C(C2CCC2)=O)C(C)C1 45912,c1(C(N2CCC(C)(C)C2CC(=O)NC2CC2)=O)cc[nH]c2nccc1-2 45913,Cc1ccc(-c2ccc(-c3nc(-c4ccc(N)cc4)nn3CC(F)F)o2)cc1 45914,N1(C(CN2C(C)CC2)=O)CCC(O)(CNC(c2cnc(C3OCCO3)s2)=O)CC1 45915,C(=O)(CS(=O)C(F)(F)F)N1CC(C)C(NC(C23CCC(F)(CC2)C3)=O)C1 45916,c1(C(N2CCCCC(NC(c3ccsc3Cl)=O)C2)=O)cccc2c(Br)cccc12 45917,CCCC(C)C(=O)N1CC(CC2CCCC2)(CC)C1.c12conc1C(=O)NC2 45918,N(C1COCc2ccccc21)C(=O)CCSc1ccc(-c2ccc(Cl)cc2)o1 45919,C1(CC(=O)NCCC(C)(C)NC(C2C(C(=O)OC)CCO2)=O)CCCCC1(F)F 45920,c1(OC)cc(C(=O)NCC2CCC2NC(c2cscn2)=O)cc2c1OCC2 45921,N1(CC(=O)NCC(C)(CC(F)F)NC(=O)Cn2ccc(Br)n2)CCC(O)CC1 45922,CC1(CNC(=O)C(F)n2cccn2)CCC(NC(=O)CC2CC(F)(F)C2)CC1 45923,c1(CC)cc(=NCC2CC(OC(C)(C)C)C2)[nH]c(CC2(Sc3ccccc3)CC2)n1 45924,CC1CC(C2CN(C(=O)C(CC(F)F)NC(c3c[nH]c(=N)o3)=O)C2)=NO1 45925,N(C(=NCCc1ncccn1)N1CC(C)N(C2CCCC2)C(C)C1)C(C=C)C 45926,CC1(C)C(CNC(=O)Cc2ccnc(F)c2F)CCN1C(C1CSC1)=O 45927,Cc1cc(=O)c(C(=O)NC(CNC(c2nnc(C)cc2O)=O)C(C)C)c[nH]1 45928,Cn1nc(C(=O)NC2CCC(NC(=O)CC3CC(F)C3)CC2)cc1C(F)(F)F 45929,c1(C(=O)NCCOCC(C2CCCC2)O)csc2c(Cl)cccc12 45930,N1(C(CN2C(C)CC2)=O)CCN(C(=O)C(C)(Cl)Cl)CC(CN(c2ccccn2)C)C1 45931,c1(CNCc2cccc(-c3c(OCC)nccc3)n2)ccc2c[nH]nc2c1 45932,C1(NC(CC2(CC(=O)OC)CCC2)=O)CN(C(=O)CC2(O)CC2)CC12CC2 45933,N1(C(CC(=C=C)C)=O)CC2(CNC(=O)CC3CCSC3)CCC1C2 45934,C(CCC1CCC1)(C(=O)NCc1cccs1)NC(C(C)n1ccnc1)=O 45935,Cc1nc(C(N2CCCC2C2CCOC2)C(=O)NC2CCC2)oc1C 45936,Cc1nc[nH]c1CCNC(=O)CC(C)NC(=O)Cc1cn[nH]c1 45937,Cn1cc(C(C)(C)C(=O)NC2CCC2NC(=O)CC2(c3ccon3)CC2)cn1 45938,c1(C(=O)NC(C2C(C(N(C(CC)CC)CCO)=O)C2)C)cnc(C)cn1 45939,C(=O)(NOC)N(CCC(=O)NC(C)COC(=O)NC)CC=C 45940,N1(C(C2C(C)C2)=O)CC23CCCCC2(C1)CN(C(=O)CC1(C#N)CCOCC1)C3 45941,C1(C(N(CCNC(C2C(NC)COC2)=O)C)=O)CC2COCC(C1)C2 45942,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 45943,N1(C(CN2C(=O)COCC2)=O)CC2(C1)CN(C(=O)C(F)(F)C13CC(C1)C3)CCO2 45944,N1(C(CSC(C)C)=O)CCCOC(CNC(C2CC(O)CN2C)=O)C1 45945,N1(C(C=C(C)C)=O)CC=CC1(C)C(=O)NCC(N1CCOCC1)=O 45946,C(CCN=C(NCc1ccc2c[nH]nc2c1)NCC1CC=CCC1C(F)F)SC 45947,c1(C)cnn2ccccc12.C1(CC)(NC(=O)Cc2cncn2C)CCN(C=O)CC1 45948,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3sccc23)=O)C1 45949,c1(C(=O)NCCN2CCN(C(C3C(OCC)CCC3)=O)CC2)c(C)cccc1Cl 45950,N1(CC(c2ccccc2)OCC)CC2CCCN(C(=O)CC3CC=CC3)C2C1 45951,C1(N(C)C(c2c(O)cccc2O)=O)CN(C(c2cc3n(n2)CCO3)=O)CC1(C)C 45952,n1(CC)nnc(C)c1CNC(=O)NCc1n[nH]c(C)c1C 45953,Cc1ccc(C(=O)NC23CC2CN(C(C2(C)CC=CCC2)=O)C3)c(Cl)c1 45954,c1(CN=[N+]=[N-])ccc(C#N)cc1.n12cnc(c1)SCCNCC2 45955,C12COC3(CCN(C3)C(=O)C3(CCC3)N1)C2.c1(N(C)C)ccc(C#N)cc1CO 45956,c1(NC(C2=CCCN(C(C=CC)=O)C2)=O)ccnc2ccc(Cl)cc12 45957,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 45958,C1(C(=O)NN(C)CC2CCN(C(c3cnc(C4CC4)s3)=O)C2)CC12CCCCC2 45959,c1(C(=O)NCC(C)NC(c2cc(CC)on2)=O)c(C)nn(CSC2CC2)c1C 45960,c1(C(=O)NC2CCN(C(c3cc(SCC)no3)=O)CC2C)n[nH]c2c1CCSC2 45961,C1(C(=O)NCC(C)CC2CCCC2)(NC(C(C)SC)=O)CCCCC1C 45962,C(=O)(CS(=O)C(F)(F)F)NCC(CCNC(C(C)CF)=O)(C)C 45963,c1(CC)ccc(C(=O)NC(C)CNC(c2ccc(CSC)o2)=O)c(C)c1 45964,C1(NC(C(C)N(CCC)C(c2cc(CC)[nH]n2)=O)=O)CC2(CCOC2)C1 45965,Cc1noc2ncnc(N3CCC(C)C3CNC(=O)COCCN(C)C)c12 45966,Cn1cc(CC(O)C(=O)NC2(CNC(=O)CCC3(C#N)CCC3)CCC2)cn1 45967,N1(C(C(C)C2CCCC2)=O)CC(O)(CN(C(=O)CCCN(C)C)C)C1 45968,N1(C(CSCC#C)=O)CC2CCN(C(=O)Cc3ccc(OC)nc3)CC2C1 45969,N1(CC)CCC=C(c2cnc(NC(c3cc(F)c(Cl)cc3F)=O)c(O)c2)C1 45970,c1(C(N(CCNC(C2CC2C(F)F)=O)CC)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 45971,CC1CCCN(C(c2cc(CNC(=O)CN3CC(C)(C)C3)no2)=O)C1C(N)=O 45972,c1(NC(CC2N(C(=O)OC)C(=O)CC2)=O)ccc2[nH]cc(C(F)(F)F)c2c1 45973,c1(C(=O)NCC(C)(CO)NC(C(C)CC(C)(C)C)=O)cccc2c1C(=O)NC2 45974,C(=O)(CCCC(C)C)NCC(CCCC)NC(c1sc(OC)nc1Cl)=O 45975,c1(C(=O)NCC2C(NC(CCC(C)(C)N(C)C)=O)CCC2)cccc2ccnn12 45976,C1(NC(CNC(C)=O)=O)CC2CN(C(c3ccccc3)c3cccs3)CC12 45977,CC1=C(C)CC(C)(C(=O)NC(C2(CNC(C3CC(=O)N(C)C3)=O)CC2)C)CC1 45978,CC1CCc2cc(C(=O)NCCN(C(=O)CC3(O)CCCCCC3)C)ccc2N1 45979,O=C(C1=CCCSC1)NCCC1CN(C(C23COCC(C2)C3)=O)C1 45980,c1(OC)cc(NC(C)=O)ccc1NC(CNC(C1CC1CN)=O)=O 45981,N1(C(CNC(CN(C)C)=O)=O)CCN(C(C2CC(C)(C)C2)=O)CC1C1CC1 45982,c1(N2CCC(N3C(CN(C)C)CCC3)C2)nc(C#N)c(Cl)s1 45983,c1(C(=O)NC2CCN(C(COCCCC)=O)C2)ccc(C(C)C(F)(F)F)cc1 45984,c1(C(=O)NCC2CCC(NC(C3(NC(C)=O)CCC3)=O)C2)cnc2c(C)cccn12 45985,CC1CCSCCN1C(=O)NC12COCC(CO)(C1)C2 45986,C1(CNC(C(C)NC(C)=O)=O)C2CC1N(C(c1csc(-c3cnccn3)n1)=O)C2 45987,C(C(C)(O)CC(=O)N(CC(C)NC(=O)Cc1ccc(C(F)(F)F)nc1)C)OC 45988,N1(C(c2nncc(OC)c2)=O)CC(NC(c2n[nH]c3c2COC3)=O)CCC1C 45989,Cn1cc(C(=O)NC2CCN(C(c3ccc(C(N)=O)nc3)=O)C2)c2ccccc12 45990,C(=O)(C(CC(C)(C)C)OC)NC(C1OCCN(C(CCNC(COC)=O)=O)C1)C 45991,c1(C(=O)Nc2c(C3CN(C(CN(CC)CC)=O)C3)ocn2)cccc(OC)c1F 45992,C1(NC(c2[nH]cc(SCC)c2)=O)CCN(C(c2nc(C)c(C)s2)=O)CC1C(N)=O 45993,Cc1cc(C(N2CCC(N(C(=O)CN(C)C)C3CC3)C2)=O)nn1-c1ccccc1 45994,c1(C(=O)NC2C(C)CCN(C(C(COC)C)=O)C2)cc2cccc(Cl)c2nc1C 45995,C1(C(=O)NC(CCCNC(C2(CC#C)CC2)=O)(C)C)Cc2cc(Br)cnc2C1 45996,C1(C(=O)NC(C2(NC(c3n(CC)ccn3)=O)CCCC2)C)CC(O)CN1C 45997,C1(CNC(=O)C=CBr)CCC(F)(CNC(=O)CCc2ncccn2)CC1 45998,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CNC(c2ccccc2)=O)CC1 45999,C1(C(=O)Nc2cccc(Oc3ncc(Br)cn3)c2)Cc2ccc(O)cc2N1 46000,c1nc(C)c(C)nc1C.C1(NC=O)CS(=O)(=O)CC1NC(CC1(OCC)CC1)=O 46001,c1(C(N2CC(NC(C(CCCC)=O)=O)C(C)CC2)=O)cnn2ccccc12 46002,CCCCC1CN=C2NN=C(O2)N1.C1(C(=O)NC(C)(C)C2CC2)CC(O)C1 46003,c1(C(=O)NC2CN(C(C3CCC(CN(C)C)O3)=O)CC2C)cccc(Cl)c1O 46004,c1(CC(=O)N(CCOC)CCNC(=O)C(F)C2CCOC2)ncoc1C 46005,C(=O)(C1CCc2nccn21)N(CC(C)NC(C(n1c(C)ncc1)(C)C)=O)C 46006,C=C(C)CC(C(=O)NC1CCC2CC1CO2)NC(=O)C(C)CSC 46007,Cc1cccc(F)c1C(=O)NC1CCN(C(C23CC(F)C2C3)=O)C12CC2 46008,C(C(C(=O)NC(CN1CCCC1)CO)NC(C(C1CCCC1)OC)=O)OC 46009,Cc1cnc(C(=O)NC(C)(C)CNC(=O)Cc2cnc(C)nc2O)c(Br)c1 46010,N1(C(c2c(CC)csc2)=O)CCCC(n2cc(C(O)C3CC3)nn2)C1 46011,C1(NC(C(C2CCC2)OCC)=O)CN(C(c2ccc(Cl)cc2C)=O)CCC1CO 46012,N1(C(C=CCOC)=O)CCC(N(C(=O)CN2CC3CC3C2)CCO)C1 46013,C1(C(=O)NC(C2CCN(C(c3sncc3Br)=O)C2)C)(CO)CCOCC1 46014,C1(CNC(c2ccn(CC)n2)=O)CN(C(C23CCC(CC2O)C3)=O)CCN1C 46015,C(=O)(CC(CC(N)=O)c1ccc(Cl)cc1Cl)N(CC(C)CNC(=O)CNC=O)C 46016,C(=O)(CCCS(C)(=O)=O)N1CCCC(C)(N(C(C2(C(O)C(F)(F)F)CC2)=O)CC)C1 46017,n1(CC)nc(C(C)C)cc1C(=O)C(c1cc(C(=O)NCCNOC)nn1C)=O.C(N)(=O)N 46018,C1(CN)CCCCN1C(C1CNCC(Sc2ccccc2)C1)=O 46019,c1(C(=O)NCC(CO)NC(c2cnn(C(C)C)n2)=O)cn(C)nc1Br 46020,N1(C(C(C)CSC(F)(F)F)=O)CCC2(C1)CN(C(c1nccnc1N)=O)CCO2 46021,c1(C(NOCC#C)=O)coc2c1CN(C(C1COCCN1C(C)=O)=O)C2 46022,C(C(CC(C)C)NC(N1C(C(=O)OC(C)(C)C)C(C)CC1)=O)NC(C=CC=CC)=O 46023,CC(C(CO)NC(c1cc(Cl)ns1)=O)NC(C1CCCS1)=O 46024,c1(OCC)cc(C(=O)N(CC(CC)NC(=O)C(C)CC)C)ccc1C(F)F 46025,CCC(CC(=O)N(C(C)CNC(=O)COCCCF)C1CC1)OC 46026,C1(C(N2CC(CC=C)(NC(=O)CC34COCC(C3)C4)C2)=O)C2CCCCCC12 46027,C1(C(C)NC(=O)CNC(=O)C2CC2)CCCCN1C(C1CC2CC1C2)=O 46028,c1(C(=O)NCC(C)N(C)C(c2ccn(CCO)c(=O)c2)=O)cc(O)cc(O)n1 46029,C(C)(c1ccco1)=CC(=O)NC1C(NC(C2(C(CC)(F)F)CC2)=O)CCC1 46030,CCCCC(F)(F)C(=O)N1CCC(=CCNC(c2ncoc2CC)=O)CC1 46031,C(=O)(CC1COCc2ccccc21)NC(C1CN(Cc2cnn(C)c2)CCO1)C 46032,C(=O)(CCCC(C)(C)C)NCC1(C(=O)NC2CC(C#C)C2)CC(=C)C1 46033,N1(C(CCC=CC)=O)CCCCC1CNC(=O)Cn1cccc1 46034,C(C)(C(=O)N(C(C)C(=O)N(C)CCn1cnnc1)C)N(C(C)=O)C 46035,C1(C(C)NC(c2cnoc2C2CCC2)=O)CCCCN1C(=O)CS.n1(C)cncn1 46036,C(C(C(C)(C)C)NC(c1cc(Cl)c(Cl)[nH]1)=O)NC(C=C1CCC(C)C1)=O 46037,N1(Cc2cccc(OC)n2)CCOCC(C)C1.C12CC(C1)C(=O)N2CC(C)C 46038,C(=O)(C(F)CCC(C)(C)C)NC1CC(C(C(N2CC3(CC(OC)C3)C2)=O)F)C1 46039,C1(CNC(C2N(CC)CCOC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CC1(F)F 46040,S(=O)(=O)(c1ccccn1)N1CC(C(N2CCN(S(C)(=O)=O)CC2CC#N)=O)C1 46041,N1(C(CCC=C)=O)CC(CCNC(c2cnc(C)cn2)=O)OC(C)C1 46042,c1(CC)ncncc1C(=O)NCCN(C(C1CCN1CC)=O)CC 46043,C#Cc1ccccc1CN=C(NCC(=O)NC(C)(C)C)NCc1cnn(C)c1 46044,N1(C(=O)CC23CCCC2C3)CC=CC(C(=O)NC2CC(N3CC(O)C3)C2)C1 46045,C1(C(=O)NC(C2CN(C(c3cc(C(F)F)n(C)n3)=O)C2)C)CC2(CC2)CO1 46046,CC(C)(O)C(F)(F)C(=O)N1CCC12CN(C(=O)C(C1CCCCCC1)O)C2 46047,c1(NC(=O)Nc2ccc(Cl)c(F)c2)c(F)cccc1[N+](=O)[O-].S1(=O)(=O)CCN1 46048,C(=O)(CCCS(C)(=O)=O)N1CC(CC)C(NC(c2cc(C(N)=O)n(C)n2)=O)CC1 46049,N1(C(C2(OCC)CCC2)=O)CC2CCC(CNC(C3(OC(C)C)CC3)=O)(C2)C1 46050,N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(C)Cn2ccnc2)C2(CCCC2)C1 46051,NS(=O)(=O)c1ccc(CCNCc2ccccc2CCCCCCl)cc1 46052,C1(C#N)(C(=O)NC(C)CNC(c2cn(C)cc(Br)c2=O)=O)CC12CCCC2 46053,C1(COC)CC(C)CN1C(=O)CC(=O)NC(C)C.C12(CC=CC1)C(=O)NC2 46054,N1(C(=O)OC(C)(C)C)CC2CCN(C(N3CCOCC3)=O)C2C1.C1CN1 46055,CCC(CC(=O)NCCCN(C)C(c1cc(C2CC2)ccn1)=O)C(C)C 46056,C(N=c1[nH]nc(C(F)F)s1)C1N(CC2(C(=O)OC)CC=CC2)CC1 46057,c1(CNC(CCCC(=C)C)=O)nc2c(s1)CCN(C(=O)C(=O)NCC)C2 46058,c1(CNC(C2CCCN(C(C(C(=O)OCC)F)=O)C2)C)ccnc2nc(C)nn12 46059,CCCC(C)C(=O)N1CCC(O)(CNC(=O)C(c2ccccc2F)(C)C)C1 46060,CCCCCCC(=O)N1CCC(=CCNC(c2cc(O)nc(C3CC3)n2)=O)CC1 46061,C1(NC(c2ccc(C(C)=O)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2)C1 46062,c1(CC)ncc(C(=O)NCC2(CN(C(=O)CN3CCCCC3)C)CC2)c(O)n1 46063,C1(C(=O)NC2CCCN(C(C(C)OCCOC)=O)CC2)Cc2ccccc2S1 46064,c1(C(N(C2(C(=O)NC(CC(=O)OCC)(C)C)CC2)C)=O)cccc(F)c1C 46065,c1(CCOC)nc(=NCCOC2CC2)s[nH]1.N12CCCCCC(C1)NC(=O)C2 46066,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46067,c1(C(=O)NCC(C)NC(CNC(C2(OC)CCOCC2)=O)=O)ccc(F)c(Cl)c1N 46068,O=C(N=c1[nH]ccnc1SCCO)C1CCCN(C(c2cccn2C2CC2)=O)C1 46069,CC(CNCC(F)(F)F)C(=O)NNC(=O)Cc1ccccc1 46070,C#Cc1cnc(NC(C2CCC(NC(C3(c4cccs4)CC3)=O)CC2)=O)cn1 46071,C#CC1(C(N2CCC(CNC(c3cncs3)=O)C2)=O)CCCC1 46072,N1(C(C2C(=C)CN2C(=O)C=Cc2ccco2)=O)CCOC(CN(C)C)C1 46073,c1(C(=O)NC(C(C)NC(c2cc(O)nc(Cl)c2)=O)C)n[nH]c2cccnc12 46074,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CCC(NC(C2(CC=C)COC2)=O)CC1 46075,c1(N2CCCC(C)(CNC(c3n(CCC)ccc3)=O)C2)ncnn2cccc12 46076,C1(CC(=O)NC2CC(CNC(C34C(C(=O)OC)(CCC3)C4)=O)C2)CCC(C)(C)CO1 46077,C(c1ccc(Cl)cc1F)=CC(N1CCC2C(NC(CSCC)=O)C2CC1)=O 46078,Cc1nn(C)nc1C(=O)NCC1CC(C)N(C(=O)COC2CCCCC2)C1 46079,CCCS(=O)(=O)N1CCCC1C(N1CCCC1C(C)(C)CNC(=O)C(C)(F)F)=O 46080,C1(CNC(CCSC)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C 46081,c1(C(N)=O)ccc(F)c(NC(=O)CNC(=O)CCc2ccccc2Br)c1 46082,N1(Cc2onc(C(C)OC)n2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46083,N12CCOC(C1)C2=O.C1(N(CC=O)C)(CCO)CCC1.C1(CNC(=O)NC)CCC1 46084,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(C)C)=O)C1 46085,c1(C(N2CCC(C(=O)NC(C)C)CC2)=O)ccc2cc[nH]c2c1 46086,N1(C(c2c(Cl)cc(C#N)s2)=O)CCC2(NC(=O)Cc3cnco3)CCCCC12 46087,N1(C(=O)OC(C)(C)C)CCC(C)(C(N2CC(CCO)(NC(=O)C(C)(F)F)C2)=O)CC1 46088,N12C(=O)CCN(C1=O)NCC(OCC)C2.C1(CN2CCOCC2)CCCS1(=O)=O 46089,C1(NC(=O)CCCC2CCOCC2)C2CC1N(C(C1CC(CC3CC3)C1)=O)C2 46090,C1(COC)(CNC(c2cc(O)nn2C)=O)CCN(C(C2CC(O)CN2C)=O)C1 46091,c1(C(=O)NCC2C(C)(C)C(=O)NC2)coc2c1CN(C(=O)CC13CCCC1C3)C2 46092,C1(C(N(CCOCCCNC(c2c(C(=O)OC)occ2)=O)C)=O)CC12CCOC2 46093,C(=O)(C(C(C)(C)C)N(C)C)NC(CNC(c1c(OC)cccn1)=O)C(C)C 46094,C1(N(C)C(c2cc(-c3cccc(Cl)c3)no2)=O)CCCCN1Cc1nccn1C 46095,C1(N(C)C)CN(C(C2CC3CC3N2C(=O)CCCN2CCOCC2)=O)CCO1 46096,N#Cc1ccc(C(C(=O)NC2CCOCC2)N(C2CCOC2)C)cn1 46097,Cn1ccnc1CN1CCC(Cn2cc(CNS(C)(=O)=O)nn2)C1 46098,N1(C(CCc2ccc(C)o2)=O)CC(CNC(c2scc(C)c2Cl)=O)CC1C 46099,C1(NC(C2C3(CC(OCC)C3)C2)=O)CCN(C(c2ccn(CC)c2C)=O)C(C)C1 46100,C1(C(C2(C(CC(=O)NCCOCCON(CC(C)C)C)=O)CC2)=O)CCC=CCC1 46101,c1(C(N2CC=CC23CCC3)C(=O)Nc2cccc(OC)c2)cccc(C#N)c1 46102,c1(C(=O)NC(C)C(C)NC(c2cc[nH]c2C2CC2)=O)cc(F)c(F)c(F)c1F 46103,c1(C(N(C2CN(C(C3CN(C(N)=O)C3)=O)CC23CC3)C)=O)n[nH]c2ccc(F)cc12 46104,C(N=c1cccc(OCC(O)CO[Si](C)(C)C(C)(C)C)[nH]1)C1(C)CC(F)(F)C1 46105,CCC(C)(C)CCCC(=O)NCCC1CN(C(=O)CCC(C)N(C)C)CC1C 46106,CC1CCC(Cl)=C(C(=O)NCCCCNC(c2ccc3nccnc3n2)=O)C1 46107,C(c1ccc(OC(C)C)c(OC)c1)=CC(N1CC(CNC(C=CC)=O)OCC1)=O 46108,C1(OCC)(CNC(=O)C(O)c2ccsc2)CCN(C(=O)CSCC(F)(F)F)CC1 46109,C12(C(=O)NCC3(F)CC(NC(C4C(C(=O)OC)C4)=O)C3)CCC(C(F)F)(CC1)C2 46110,N1(C(C(CSC)(C)NC(=O)COCC(F)(F)F)=O)CC2CCN(C)C2C1 46111,c1(C(=O)NCCc2ccccc2)ccc(Cn2cc(C3CCOCC3)nn2)cc1 46112,C(C)(CO)(C(=O)NCc1cccc(Cl)c1)NC(c1c(CC)c[nH]n1)=O 46113,c1(C(N2CC(C)N(C(=O)CC3CCCC(C)(C)O3)CC2)=O)ccc2nsnc2c1 46114,N1(C(C(CC=C)OC)=O)CCC(CNC(c2cnc(COC)nc2O)=O)C(C)C1 46115,c1(CC(=O)NC2C(C)(C)CN(C(=O)C=CBr)CC2)ccc(O)c([N+](=O)[O-])c1 46116,C1(O)(C(=O)NCCCN(C(c2cc3ccncc3o2)=O)CC)CCCC(C)CC1 46117,N1(C(c2cnn(C)c2C(F)(F)F)=O)CC2(CCN(C(=O)CO)C2)C1 46118,c1(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)cccc(Cl)c1Cl 46119,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46120,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46121,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46122,c1(CC)nn(C)c(CC)c1C(c1nnnn1C1CCCC1)NCc1ccc(F)cc1 46123,N(C1CCNc2ccccc21)C(=O)Cc1ncnc(O)c1Br 46124,C1(n2ncc(CNC(C3C4CNC(=O)C34)=O)c2)CCN(CC2CCC(F)CC2)CC1 46125,Cc1cc(=NCC2CCOC2c2cnn(CCO)c2)[nH]cc1S(N)(=O)=O 46126,c1(NC(C(C)=CC2CC2)=O)ccc(SCc2ccccc2OCC(F)(F)F)cc1 46127,c1(CCNC(C(CC2CN(C(COC)=O)C2)F)=O)ncc(C)cn1 46128,C(CCCC(=O)N1CC(C(=O)NCc2cccc(C#N)c2)CCC1C)(OC)OC 46129,Cc1cc(N(c2nnnn2-c2ccccc2Cl)C(C2CCC2)C)c(O)c(I)c1 46130,C1(C(=O)NCC(C2CCC2)NC(=O)CC2CCCC2)CCN(C)S1(=O)=O 46131,C(=O)(CCC1=CCCCC1)NCc1c(C(=O)NC2CN(C)CC2(F)F)[nH]cc1 46132,C1(n2c(-c3c(-c4cc(C)c(F)nc4)csc3)ncc2)CCc2ccccc2C1 46133,C(=O)(C1OCCn2ccnc21)NCCCC(CCC)NC(C1CCN(C)CC1)=O 46134,CC(C)(CNC(=O)CC1CCCC(C2CC2)O1)CCNC(=O)Cc1ccno1 46135,N1(C(c2ccc(C(F)(F)F)cn2)C(=O)NC2CC2)CCC2CCCNC2C1 46136,N(C(=NCCn1ccc(COC)n1)NCC12CCCC1CC2)CC(=C)C 46137,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nnc(C)cc1O)=O 46138,C1(C2N(C(C3N(N=O)CCC3)=O)CC2)CCN(C(C23CCCC2C3(F)F)=O)CC1O 46139,c1(C(=O)NCC2C(C)(C)N(C(=O)CC3CCCO3)CC2)cnn2cccnc12 46140,Cc1cccc2c(CC3CCN(c4nc5ccccc5s4)CC3)cnn12 46141,CC#CCCC(=O)NCC(C)NC(=O)C(C)CC1CCCCC1 46142,c1(NC(C2C3CCC2CN(c2ncc4cn[nH]c4n2)C3)=O)cc(Br)cc2cn[nH]c12 46143,C12(NC(C(N(C(=O)C#CC3CCC3)C)C3CC3)=O)CCC(CC1)C2(C)C 46144,C1(NC(=O)NCC(c2ccccc2)N(C)C(C2CCCCC2)=O)CCOC(=O)N1 46145,C1(N2C(=O)C2)CC(C#N)C1.CN(C(C1CC1)=O)OCCNC.C1(C)CC1 46146,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46147,C(=O)(CC1CCCc2ccccc21)N1CCN(C(c2c(C)scc2)=O)CC1CF 46148,N1(C(C)C)N=C(C(=O)N2CCCC2CNC(=O)C(O)CC2CCCC2)CCC1=O 46149,C(=O)(C(CC1CCOCC1)NC(C1CCC1)=O)NCC(C)F 46150,Cc1cc(NC(C2CCC(NC(c3ccccc3CO)=O)CO2)=O)c(Cl)cc1Cl 46151,c1(C(=O)NC2C(N(C(CNC(=O)OCC=C)=O)C)CCC2)cnn(C)c1C(C)C 46152,CCCCC(C(=O)N1CC=CC(C(=O)NCCc2ncnn2C)C1)NC(N)=O 46153,c1(CNC(C=CC(CC)C)=O)cccc2c1CN(C(=O)CN(C1CC1)CC)C2 46154,CCC1CN(C(C2(N(C(=O)CCCC3CCCC3)C)CC2)=O)CC(=O)N1C 46155,CCC(COC)C(=O)N(CCCNC(c1sc(C)nc1C)=O)CCO 46156,N1(c2nccc(Br)c2Br)CCC2CCCCC2C1 46157,CCC(C)CC(C(=O)Nc1cnc(Cl)c(C)c1)NC(c1cnn(C)n1)=O 46158,c1(C(=O)NCCNC(c2cnn[nH]2)=O)ccc(-c2ccccc2)cn1 46159,CC1CCCC(C(=O)Nc2cccc(NC(=O)Cc3cnn(C)n3)c2)CC1 46160,C1(C(=O)NCC2(C3CC3)CCCO2)CC(CNC(c2c[nH]c(=O)cn2)=O)CC1O 46161,c1(OCCC)ccc(C(=O)NCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C)cc1 46162,CC1CCOC(C(=O)NC(CC(F)(F)F)c2ccccc2)C1 46163,Cc1cc(C#N)cc(C)c1C(=O)NC1CCN(C(C2CCCC2)=O)CC1O 46164,c1(-c2cn(CCc3c(C)cccc3)nn2)ccc(F)cc1O 46165,c1(OC)ccc(C(=O)NCC2CCC2NC(=O)CC2CCCO2)c(C)c1 46166,Cc1ccc(Br)c(NC(c2cc(-c3cccc(N4CCOCC4)c3)cs2)=O)c1 46167,N1(C(C2CC(NCc3c[nH]nc3-c3ccncc3)C2)=O)CCN2CCCCC2C1 46168,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCN(C(=O)C(F)=C3CC3)C2)C1 46169,c1(C(N2CCCC(NC(C(C)C#N)=O)C2)=O)cc2c(s1)CN(C)CC2 46170,O=S(=O)(c1[nH]c(=NCC2CC(N3CCCC3)C2)ccc1Br)NC1CCCCC1F 46171,Cc1cc(C(=O)N(CCN(C)C(c2scnc2C2CCCC2)=O)C(C)C)no1 46172,C1(CN(C(=O)C(C2(C)CC2)NC(=O)CN(C2CCCC2)C)C)CC1(C)C 46173,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46174,c1(C(=O)NCC2C(C)CCN2C(C2CC2c2ccccc2)=O)ccc(F)cc1Cl 46175,c1(C(=O)NCC=CCNC(C2CCN(c3ccncc3)C2)=O)cc(Cl)nnc1O 46176,O=C(NNc1cc(-c2nn[nH]n2)ccn1)C1CCC2CCC(=O)N12 46177,C1(C(=O)NCC2C(OC)CC2)(NC(c2cnn(C)c2C)=O)CCN(C)C1 46178,N1(C(C(CSC)C)=O)C2CCC1CN(C(c1ncnc3ccsc13)=O)CC2 46179,C1(C(=O)NC(C(=O)N2CC(N3CCOCC3)C2)C2(C)CC2)CCC2CC1CO2 46180,CC(C)(C(O)C(F)F)NC(C1CCCC1CNC(C1(n2cccc2)CC1)=O)=O 46181,Cc1cc(=O)oc(C)c1C(=O)NC1C=CC(CNC(C2COCCN2C)=O)C1 46182,CCCC(CCC)C(=O)NC1CN(C(c2cc(C)c(OC)c(C)c2)=O)CC1C 46183,C#Cc1ccc(C(=O)NCC2CCCN(C(c3ccn(C(F)F)n3)=O)CC2)cc1 46184,c1(CC(=O)NC(c2cccc(F)c2)CC)ccc(S(C)=O)cc1 46185,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46186,N1(CC(=O)NC(C(=O)NCCN(CCC)CC)C2CCCO2)CCC(=O)CC1 46187,Cc1nc(C)n(Cc2cn(CCCCNC(=O)C(C)N3CCC3)nn2)n1 46188,N1(C(c2ccn(C(CC)CC)n2)=O)CC(OC)CC1CNC(C1(C)CC1(Cl)Cl)=O 46189,N1(C(c2nccc(C)n2)=O)CCCCC(NC(=O)C=CC(C)C)CC1 46190,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(CCOCC(C)C)=O)CC1 46191,N1(C(C(C)Cc2cnc[nH]2)=O)CC2CC1C2NC(=O)CS(C)(=O)=O 46192,CCC(CC(=O)N1CCC(CN=c2nc(C3CC3)[nH]s2)(C)C1)C(F)F 46193,C1(C(=O)C(C)C2(O)CCC2)CCN(C(=O)CCc2cn(C3CC3)nn2)CC1.CO 46194,Cc1c(-c2cc(CN3CCOC(c4ccccc4F)C3)[nH]n2)oc2ccccc12 46195,c1(C(C)SCCNC(=O)C(C)C2CCC2)ccc(-c2cnn(C)c2)o1 46196,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46197,C(=O)(CC(O)C(C)C)NC1CCC(CC(=O)NCc2cc(C)ncn2)CC1 46198,c1(C2(C(N3CC(C(C)NC(C4OCCC4C)=O)C3)=O)CC2)ccc([N+](=O)[O-])cc1 46199,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46200,CCCCC(C(=O)NOCC1CC1)NC(c1nonc1N)=O 46201,c1(C(CC)(C)C)n[nH]c(=NC(CCNC(C2CCCN(C(N)=O)C2)=O)C(C)C)o1 46202,N1(C(c2c(C)csc2)=O)C(C(N)=O)CCC1C 46203,C(=O)(C1CCCc2scnc21)N1C(C)CN(C(C2CCCN2C2CC2)=O)CCC1 46204,c12nccc(c1C#N)NC2=O.C1(C(CNC(=O)NC(C)(C)C)OC)CCCCC1 46205,c1(SCC(N2CC(C=C)C(NC(=O)NC)C2)=O)cc(S(N)(=O)=O)c(C)s1 46206,c1(C(N2CCC(F)(CNC(c3sccc3Cl)=O)C2)=O)cc(O)nc(C2CC2)n1 46207,N1(C(C=Cc2c(C)noc2)=O)CC=C(CO)CC1 46208,CCC(C)CCCCC(=O)NCC(CSC)C(=O)N1CC(C)C(C)C1 46209,C(CC(C)C(C)C)NC(C(CN(C)C)NC(Cc1scc(C)c1)=O)=O 46210,c1(C(N2CC(NC(c3cscn3)=O)C(CC3CC3)C2)=O)cc2nc[nH]c2cn1 46211,N1(C(CC=CC)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46212,C1(CNC(c2c(C)con2)=O)CCN(C(C2CCOC2)=O)CC1C1CC1 46213,N12CCCN(CC1C)CC2=O.c1(N(S(CC)(=O)=O)C)cc(C(F)(F)F)ns1 46214,c1(CN2CC3(CCC(C(=O)Nc4ccnnc4Br)O3)C2)ccc2nc(O)[nH]c2c1 46215,CCP(=O)(CC)c1ccccc1CNC(CC(N)=O)C(=O)C1CC1 46216,C1(NC(C2(CC=C)CCCC2)=O)C2CCN(C(=O)CCCCCCC)CCC12 46217,Cc1ncnc(C(=O)NCC2CCC(NC(c3c(C)nn(C)c3Cl)=O)C2)c1C 46218,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46219,n1(CC(C)NC(C2(n3cccn3)CCC2)=O)cc(CCC2CCCCO2)nn1 46220,c1(OC)cc(NC(=O)NCC2(O)CCOCC2)ccc1F 46221,C(C)(CC(C)N=c1c(C#N)c[nH]c2c(F)ccc(F)c12)NC(c1cc(C)no1)=O 46222,n1(CCC2CN(C(c3csc(Br)c3)=O)C2)cc(CC2CCCCO2)nn1 46223,c1(SC)nc(N2CCCOC(CNC(=O)CC(C)(C)C)C2)cc(Cl)n1 46224,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46225,C1(NC(CCOCC#C)=O)CC2CC(C1)N(Cc1ccc(C)c(Cl)c1)C2 46226,C1(NC(CCc2c(C)noc2C)=O)CN(C(c2coc(O)n2)=O)C2(CCOC2)C1 46227,CC(C)CCCC(C)C(=O)NCC1CCC(C)N(CC=CC(C)(C)C)C1 46228,N1(C(C(=O)NCc2c[nH]c(=O)cn2)=O)CC2CC2(NC(C2CC2)=O)C1 46229,C1(C(=O)NC2CCCCC2)(COC)CCCN1C(=O)CCC1CC1 46230,CCC(C)C(C)CN(CCCCCC)C(C12CC(N)C1C2)=O 46231,c1(C(N2CC(O)(CNC(=O)Cc3ccc(Cl)s3)C2)=O)cc(O)cc(Cl)c1 46232,c1(C(=O)NC2C(CNC(CN(C(C(C)C)=O)C)=O)COC2)cnn2cccc(Cl)c12 46233,c1(C(=O)NC2C(C)N(C(=O)CCCCCN(C)C)CC2)cccc2c1C(=O)OC2 46234,C(=O)(CC1=CCCCC1)NC(C1CN(C(CN(C(C(C)C)=O)C)=O)C1)C 46235,N1(C(C=CC=CC)=O)CCC2CCC12CNC(c1cn(CC)nc1C(F)F)=O 46236,c1(NC(C2(NC(=O)COC(F)(F)F)CC2)=O)cccnc1SCCO 46237,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46238,CC1(CNC(c2ccnc(OC(F)(F)F)c2)=O)COCCN(C(C2CCCO2)=O)C1 46239,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC1C2C3O 46240,c1(CCNC(=O)Nc2cc(Br)cc([N+](=O)[O-])c2)ccc([N+](=O)[O-])c(O)c1 46241,C1(C(=O)NC(C)CN(C)C(c2csnc2Cl)=O)C2CC3C(C2=O)C13 46242,c1(C(=O)NC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)N2)=O)cc1 46243,C1(NC(COC(CC)C)=O)CC(CNC(c2ccn(CC)c2C)=O)CC1O 46244,C(N=c1[nH]cncc1I)C1CC(NC(c2cn(-c3nccs3)nn2)=O)C1 46245,C(C(CCC(F)F)COC(C)(C)C)OC(C1(C(=O)OC(C)(C)C)CCOC1)=O 46246,C(=O)(CC(C)(C)C(=O)N1CCCC1CNC(c1cn(CC)c2c1CCC2)=O)OC 46247,c1(C(=O)Nc2c(C)ccc([N+](=O)[O-])c2)ccc(C2=CCC(O)CC2)s1 46248,C1(C(=O)NCCOC)(CO)CCN(C(C2CC(OC3CCCO3)C2)=O)CC1 46249,CC(C)C(O)C(=O)N1CC(NC(C2(O)CC(CF)C2)=O)C(O)C1 46250,c1(N2CCC(NCC3(CC)CCCC3)CC2)cc(Cl)ccc1Cl 46251,c1(C(=O)NC(C)C)cc(SC)oc1C.c12nc(n[nH]1)CNC(=O)C2.CCOC 46252,c1(OC)ccc(F)c2c1CN(C(C)C(=O)OC(c1ccsc1)OC)CC2 46253,c1(Cn2cc(CCCSCCN3CCC(OC)CC3)nn2)ccc(F)cc1F 46254,C1(CC)(CC)CCCN(C(=O)CC2CCN2C(c2ccc(O)cn2)=O)C1 46255,CCCC(C(=O)N1CCN(CC(=O)NC(C(N)=O)C2CC2)CC1)C(C)C 46256,c1(C(N2CCCC(C(CNC(CCC=CC)=O)(C)O)C2)=O)cc(N)c(C)cc1C 46257,c1(C(=O)NCCC2CCCN(C(C(C)OC(C)(C)C)=O)C2)ncc(Br)cc1F 46258,CCC(CC)C(F)C(=O)N(C)CC1COCCN1C(=O)CCc1csnn1 46259,c1(OC)ncc(C(=O)N(C2CCC(NC(c3cnc(CC(C)(C)C)o3)=O)C2)C)s1 46260,c1(C(=O)NC2CC(O)(CNC(C(C)OCCCC#C)=O)C2)cc(F)c(F)c(F)c1 46261,N1(C(C(C)C2CC2)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46262,c1(NC(=O)C(=O)N(C2CC(n3cncn3)C2)C2CCSC2)ccccc1 46263,N1(C(CN(CC(C)C)C)=O)CCN(C(=O)CC(=O)NCCN(C)S(N)(=O)=O)C2CC12 46264,c1(C(N2CC(NC(COCCOC)=O)C3C2C3)=O)ccc2cnccc2c1 46265,c1(C(=O)O)cc2cc(CNc3ccc(C(F)(F)F)cc3F)sc2s1 46266,Cc1oc2c(F)c(F)c(F)c(F)c2c1CNS(=O)(=O)c1ccc(C(C)C)cc1 46267,N1(C(COC2(C)CN(C(C3N(C)C(=O)OC3)=O)C2)=O)CCc2n[nH]cc2C1 46268,C1(CC(=O)NC)CN(C(=O)CC(C)(C)OC)CCN1C(=O)CC1CC(C)(C)C1 46269,c1(CC)ncccc1NC(=O)CCC1(NC(=O)CCCF)CCC1 46270,C(=O)(C1CCCc2ncccc21)N1CC(NC(C2(C)CC(O)C2)=O)C1 46271,c1(C(n2cc(Br)cn2)C)c(C)nc2ncnn2c1Nc1ccccc1 46272,CN1CC(C(=O)NCC23COC(CNC(C4CCCC4F)=O)(C2)C3)CC1=O 46273,N1(C(Cc2n(C)ncc2)=O)CC2CC2(C(=O)NCC(F)CO)C1 46274,CC1CCN(C(=O)CC(C)C2CCCO2)C(C)C1NC(c1ccccc1Br)=O 46275,c1(OC)cccc2c1CCN(C(=O)COc1cc(-c3ccc(F)cc3)ccn1)C2 46276,c1(N2CCC(F)(C(=O)Nc3nccnc3F)C2)ncnn2cc(Br)cc12 46277,C1(C)(C(N2CCC(C(C)NC(CSC(C)(C)C)=O)C2)=O)CCS(=O)(=O)CC1 46278,CCC1CC(=O)N1C.C(=O)(CCCN(C)C)NC(C)CCC 46279,N1(C(C2(CC)CCCN2C(=O)C(C2CCCCC2)C)=O)CC2CCCC(C2)C1 46280,C1(C(=O)OC)CCC2C(CCN2C(c2cc3c(C(F)(F)F)cccc3s2)=O)C1 46281,C1(C(=O)NC2C(C(=O)OC)C2)CCCCC1(C)NC(=O)CC1(O)CCOCC1 46282,c1(-n2c(-c3c(CC)ccs3)nc(-c3ccoc3)n2)nc(Cl)sc1CC 46283,C1(C(=O)NCCC(C)NC(c2ncccn2)=O)(COC)CCOC1 46284,CC1C(C(=O)N2C3CCC2CC(C(=O)Nc2ccc(F)cc2)C3)=NOC1C 46285,c1(CC)cc(C(=O)NCC2(NC(c3cncnc3)=O)CC2)cs1 46286,c1(C(=O)NCC2C(NC(c3cnns3)=O)CCCC2)c(F)ccc2nc[nH]c12 46287,C1(CNC(c2n(CCC)ncc2)=O)CCN(C(C2CCCCO2)=O)CC1(F)F 46288,N1(C(C2CCC(CC)CC2)=O)CC(CNC(c2cncn2C)=O)CC1(C)C 46289,N1(C(c2nc(SC)oc2)=O)CCOC(CC(N2CCC(CCCO)CC2)=O)C1 46290,c1(C(=O)NC2C(NC(C(C)Sc3ccccc3)=O)COC2)ccnc(S)c1.C1(C)CC1 46291,c1(C(C)N)nc(C(=O)NCC23CCCC2C3)c(C)o1 46292,Cc1cc(C(N2CCC(C)(CNC(C3CCS(=O)(=O)N3)=O)C2)=O)n(C)n1 46293,N1(C(C=C(CC)CC)=O)CCC2CN(C(C3C(C)(C)C3(C)C)=O)CCC12 46294,C1(C)(CC)CCN(C(=O)C(C2CCCN(C(=O)C(C)C3CCC3)C2)C)CC1 46295,C(=O)(N1OC2CCC1C2)C1(NC(=O)C(C2CCCCC2)O)CCC(C)C1 46296,c1(C(=O)NC(c2ccc(Cl)s2)C)cncc(CNC(c2nccnc2Cl)=O)c1 46297,N1(C(CC(C)F)=O)CCCCCC1CNC(=O)Cc1n[nH]cc1Br 46298,S(=O)(=O)(c1c[nH]c2ncc(F)cc12)NC1CC2(CC(C(=O)O)C2)C1 46299,c12ccc(cc1)C(=O)NC2.C(CC(=O)NOCc1ccccc1F)OC(N)=O 46300,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46301,C(=O)(C(O)CCNC(=O)CN1CC2CC2C1)NC(C)C(=O)NC(C)(C)C 46302,c1(C(=O)NCC=C(C(N2C(CCC#C)CCC2)=O)C)c[nH]c2ncccc12 46303,c1(C(C(=O)NCCC#N)N(C2C3CCCC23)CC)cc(C)nnc1C 46304,N1(C(CCNC(C)=O)=O)CCN(C(C2CCCSC2)=O)CC(C)(F)C1 46305,c1(C(N2CCC(NC(C3CC(C)(CC)C3)=O)C2)=O)ccn2ncnc2c1 46306,c1(N(CCCNC(C2(C(=O)N(C)C)CC2)=O)C)ccccc1 46307,N#Cc1ccccc1CC(=O)NCC1CCCCN1C(c1coc(C2CC2)n1)=O 46308,Cc1cccc(C(N2CCC(N(C)CCOC)C2)C(=O)Nc2nnn(C)n2)c1Cl 46309,N1(C(CCCc2ccc(C)s2)=O)CC2CC(C1)CN(C(=O)C(C)C(C)O)C2 46310,C(=O)(C(C)(CC)CO)NCC1N(C(c2ncn(CCC)n2)=O)CCOC1 46311,C(CCC(C(=O)NCc1cccc(C)c1F)NC(C1CCCOCC1)=O)OC 46312,N1(C(CCOC(C2CN(C(=O)NC)C2)=O)=O)CC2(CC(CC(=O)NC)CO2)C1 46313,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46314,c1(C(=O)NCCC2(C(=O)NCCCCC)CCCC2)nc(=N)cc[nH]1 46315,c1(C(=O)NC(C)CN(C)C(c2ccc(-c3cccs3)[nH]2)=O)ncc(F)cc1N 46316,C1(NC(C2(F)C(C)C2)=O)CCC(F)(CNC(c2ccc(Cl)cn2)=O)C1 46317,c1(C(N2CC(NC(c3cc(CC)no3)=O)C(C)C2)=O)c(C)nc2sc(C)cn12 46318,O=C(C1CCc2ccccc21)N1CC2CC1CN2C(c1cc(F)cc(F)c1F)=O 46319,C(CCCCCCCO)=CC(=O)NCC1CCN(C(C23CC(C)C2C3)=O)C1(C)C 46320,N1(C(C(C)c2cccs2)=O)CCC(O)CC1C(N1CCC(c2ccco2)C1)=O 46321,C1(C(=O)NC2(CCNC(C(C)C)=O)CCCC2)CN2CCC1CC2 46322,N1(CC(C)NC(C2CC(F)(F)C2)=O)CCN(C(=O)C(c2ccnn2C)C)CC1 46323,N1(C(C(CCNC(C)=O)O)=O)CC2CN(C)CC2(NC(=O)OC(C)(C)C)C1 46324,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)CN1CCCC1 46325,c1(C(=O)NCC(CNC(C(CC)N(C)C)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46326,Cc1oc(C(=O)NCC2CC(C)CCN2C(C2CC2C)=O)cc1S(N)(=O)=O 46327,c1(C(=O)OC)c(C)cc(C)nc1Cl.c12nn(cc1I)CC(=O)N2 46328,C=CCCCCC(=O)NC(C(=O)NC1CC12CCC2)c1ccco1 46329,C(=O)(C#CC(C)(C)O)N1C(C(N2C(CC(C)C)CC2)=O)CC=CC1 46330,N1(Cc2cccc(OCCC)c2)CCC(NC(C2CC(C)C2)=O)C(F)C1 46331,c1(N2CCCC(N(C(N(C)C)=O)C)C2)nc(=NCC#CC2CC2)[nH]c2c1CCCC2 46332,NC(=O)CCCCC(=O)N1CCCC(O)(CCNC(=O)CC2CS(=O)(=O)C2)C1 46333,c1(C(=O)NCC2CCC(NC(C(CN(C)C)OC)=O)C2)cc2c(cc1N)OCO2 46334,C1(CN(C(=O)CC2C=CCCC2)C)CCCN1C(c1nocc1Br)=O 46335,CCCCC(CNC(=O)CC1(NC(=O)C(C)n2ccnc2)CC1)CCC 46336,C(=O)(C1=Cc2ccccc2C1)NCC1C2(CCN(C(COCC)=O)CC2)CCC1 46337,CCCCCS(=O)(=O)CC(=O)NC(C)CN(C(=O)CC(C)O)CC 46338,N1(C(CCOC(C)C)=O)CCCC2(CCCCC2NC(c2cccs2)=O)C1 46339,C1(NC(C2(CC)CCOC2)=O)CC1C1CCN(C(=O)C(C)CC(C)C(C)=O)CC1 46340,C1(Cc2ncc(C)cn2)CCN(N(Cc2ccc(Cl)cc2)CF)CC1 46341,C(=O)(CCCF)N1C(N(CC(C)(C)C)C(CN(C)C2CC2)=O)CC1 46342,C1(NC(c2ncc(OC)cn2)=O)CCOC2(CCN(C(C3CCO3)=O)CC2)C1 46343,CP(C)(=O)C1(O)CCN(C(C2CC=CCC2)C(=O)NCc2ccccc2Cl)CC1 46344,C1(NC(C2CC2F)=O)CC2CC1CN(C(=O)C1=C(Cl)CC1)C2 46345,c1(C(CC)(C)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)ccccc1Cl 46346,C(C(CS(C)(=O)=O)CS(C)(=O)=O)N(C(CC1CCCC(C)C1)=O)CC(=O)O 46347,Cc1ccc(C)n1CC(N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O)=O 46348,N1(C(CCSCC)=O)CC2(CCN(C(=O)C3=CCCCC3)C2)C1 46349,c1(CSCC(=O)NC(C)CCNC(c2coc(=O)[nH]2)=O)ccc2ccccc2c1 46350,C1(C(N(CCN(C(C)C)C(c2ccsc2)=O)C)=O)CC(C)=NO1 46351,c1(OC)cccc(CNC(=O)C(C)(O)C2CCN(C(=O)C(C)(C)C#N)C2)c1 46352,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1C=CCC1 46353,C1(NC(=O)Cn2cccn2)CC2(C1)CN(C(c1cc(O)ccc1I)=O)C2 46354,C1(CC)(NC(=O)Cc2ccoc2)CN(C(=O)CC(C)n2cccn2)C1 46355,c1(C(N2CC3CCN(C(CCC=C)=O)C3C2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] 46356,C(=O)(C(C)(C)C(=O)N1CCCC(N(C(=O)CC2(C#N)CCC2)C)C1)OC 46357,C1(N(C(=O)Cn2cccn2)Cc2cc(Cl)ccc2F)CCC12CCNCC2 46358,CC1CC(C(=O)NCCOC(=N)O)CN(C(c2ncc(F)cn2)=O)C1 46359,N1(C(CC)=O)CCCC(COC)(NC(c2cc(-c3ccccc3O)[nH]n2)=O)C1 46360,N1(C(CSC)=O)CC(O)CC1CNC(=O)CCC(=O)C1CC1 46361,C(=O)(C(F)CC1CC1)NCCN(C(C(C)=C1CCCC1)=O)C1CC1 46362,c1(C(=O)NC(CNC(C(C)OC)=O)CCOCC(F)(F)F)ncnc2sccc12 46363,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2n1CCN(Cc1ccc(C#N)s1)C2 46364,c1(C(=O)NCCN(C(C2C(C(C)C)C2)=O)C2CC2)cccc(O)c1F 46365,C(C(C)C)(C(O)C(=O)NCC1(C(N2CC(N3CCN(C)CC3)C2)=O)CCC1)OC 46366,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CC 46367,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)CN1CCC(=O)CC1 46368,c1(C(=O)NCC(CC)NC(=O)C=Cc2ncc[nH]2)cc2nc[nH]c2cn1 46369,C1(C(=O)NCCC(=O)OC)CN(C(c2ccc(Br)s2)=O)CC2(CCC2)C1 46370,CC(C(=O)NCCOCCOCCCNC(=O)CNc1cnoc1C)C(C)O 46371,C=CC1(NC(=O)CCC(C)NC(C2CC(N=[N+]=[N-])C2)=O)CCOCC1 46372,c1(COCCCNC(C(=O)NC(C2CCCCC2)c2ncc[nH]2)=O)ccc(F)cc1 46373,C1(C(=O)N)CC(F)(F)CN1C(=O)CCCC1CCC1.C(=O)CCc1ncco1 46374,c1(C(=O)NC2(C)CN(C(c3sc(Cl)cc3Cl)=O)C2)cn2c(n1)CCC2 46375,Cc1nc2cc(C(N3CC(CNC(=O)CN(C)C(=O)C4CC4)C3)=O)c(F)cc2[nH]1 46376,N(C(=NCCc1ccc2c(c1)CCC2)N1CCN(CCF)CC1)C(C)C1CC1 46377,c1(CC(=O)NCC2CN(C(c3ccccc3)=O)C3CC23)cnc2c(=O)[nH]ccn12 46378,N1(C(C(CCC)NC(C)=O)=O)CCOC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 46379,C(C(C)CC(=O)NC(C)CC(C)NC(=O)CN1CCS(=O)CC1)OC 46380,N1(C(C(C)C2CCC2)=O)CC(NC(=O)CCc2ncccn2)C2(CCOCC2)C1 46381,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46382,N1(C(CCC(CC)C)=O)CCC2(CCC(NC(=O)C(F)CC)CC2)CC1 46383,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46384,Cc1nn2cc(C(N3CC(CNC(c4cc(C(N)=O)no4)=O)C4CC34)=O)nc2s1 46385,N1(C(c2nnn(CC)c2C)=O)CC(CNC(=O)CCNC(=O)CO)C2(CC2)C1 46386,C1(C(=O)NCCC(C)N(C)C(C2CCOC2)=O)CC(C)N(C)C1 46387,N1(C(c2cnc(C(C)C)[nH]2)=O)CC(CNC(=O)CCc2cscn2)C(O)C1 46388,c1(C(=O)NCC(C(=O)NC2(C)CCC2)OC)cccc(F)c1C 46389,c1(OC)ncc(C(N2CC(CNC(C3CCC(C)O3)=O)C2)=O)cc1C 46390,c1(C(C(C)NC(=O)C2CC2)=O)occc1CNC(CC(CCO)N(C)C)=O 46391,C1(CNC(c2cnc(Cl)cn2)=O)CN(C(=O)CC2CCCCC2)CCC12CCC2 46392,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(NC(=O)Cc3cscn3)C2C1 46393,c1(Oc2c(C(=O)OC)nccn2)cc(C(=O)OC)c(F)c(F)c1 46394,CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC(CNC(=O)C(=Cc2cscn2)F)O1 46395,C1(N(CC#C)C(c2nocc2Cl)=O)CCN(C(C2(O)CCC2)=O)CC1 46396,N#Cc1ccc(C(O)C(=O)NCCC2CCC2c2ccccc2)cc1 46397,O=S(=O)(c1ccc(Br)cn1)N1CCC(N2CCN(c3ccccc3)CC2=O)C1 46398,N1(C(C2C(C)(NC(C3CN(C)C(=O)N3)=O)CCCC2)=O)CCCC(C2CC2)CC1 46399,c1(NC(=O)CNC(C2CC2CNC(=O)C2CC2)=O)snnc1-c1ccccc1 46400,c1(C(N(CCNC(c2cccc(N(C)C)n2)=O)CC)=O)ccc2nc(S)[nH]c2c1 46401,c1(C(=O)NCCCN(C(C2CCC(CC)O2)=O)CCO)cc(OC)cnn1 46402,N1(C(C(CO)N(C)C)=O)CCOC2CN(C(C3C4CC5C(C4=O)C35)=O)CC12 46403,CC1=C(CNC(C2CCN(C(c3cc(C#N)[nH]c3C)=O)C2)=O)CCCC1 46404,N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(C23CC(C2)C(C)O3)=O)CC1 46405,N1(CC(=O)N(CCCNC(=O)CCc2cn[nH]c2)C)CCC(C)(C)CC1 46406,C1(=O)C(C(C)C)CN1.C1(CNC(CC)=O)CCC(NCC)CC1 46407,N#CC1(C(=O)NC2CCCCCN(C(c3cccnc3)=O)C2)CC12CCOCC2 46408,c12c(ccc3c1CCC3)-n1nc(C3CCCN(C)C3)nc1-2.CO 46409,N1(C(Cc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCN2CCCC2)CC1 46410,C(=O)(CC1COc2cc(O)ccc21)NC(CC(C)(C)C)Cc1ccccc1 46411,C(=O)(C1=CCC(NC(=O)CC2COCC(C)O2)C1)NC(CSC)(C)C 46412,c1(NCC(=O)NC2C(CNC(C3(CCCC)CCCC3)=O)C2)ccc(Cl)cc1Cl 46413,CC1CCC(C(=O)NCC=CCC(=O)NC2(c3nc(O)n[nH]3)CC2)C1 46414,C1(C(N2CCC2CNC(C2(F)CC3(CCC3)C2)=O)=O)CN2CCCC2CO1 46415,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46416,C1(CN(C(CC2(OC)CCC2)=O)C)CN(C(c2sc(CO)nc2C)=O)CC12CC2 46417,C12(CNC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1(NC(C)C)CC1)=O)C2 46418,CCC(O)C(C)C(=O)NC1(CNC(=O)COCc2ccccc2)CCOCC1 46419,N1(C(=O)NC(c2nc(CCC(=O)OC)[nH]n2)C)CCC(F)(C#N)C1 46420,CCCCC(CNC(=O)CCC1CCC(C2CC2)O1)NC(=O)CN1CCOCC1 46421,c1(CNS(c2ccc(OC)cc2F)(=O)=O)cc([N+](=O)[O-])cc2c1OCOC2 46422,Cc1cc(C(N2CCC(F)C(NC(c3ccc(Cl)o3)=O)C2)=O)n2nccc2n1 46423,c1(C(=O)NC2CCCN(C(=O)C=C(Cl)Cl)CC2)ccc(=O)n2c1CCC2 46424,Cc1cc(C(=O)N(CC(C)NC(=O)COC2(C)CCC2)C)n2nccc2n1 46425,C(=O)(C(F)(F)C(F)(F)F)NC1CC(CNC(C2=NOC(C(C)(C)C)C2)=O)CC1O 46426,CC1CCCC(CC(=O)NCC(C2CC2)NC(=O)C(n2cc(Br)cn2)C)O1 46427,CC(C)C(O)CC(=O)N(CC(=O)Nc1ccc(COC)cc1)C1CCC1 46428,C1(N(C(=O)CCC2CCCCO2)C)CCCN(C(=O)COCc2nncs2)CC1 46429,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)OCCO2)=O 46430,C(=O)(C(C)CCCc1ccccc1)N(C(CCC=C(C)C)C)C1CCCC1 46431,c1(CC)cc(C(N2CCC2CNC(=O)C(F)(F)c2ccnn2C)=O)oc1COC 46432,Cn1ncc(CN2CCN(C(=O)NC3CCNC(=O)C3)CC2)c1-c1ccccc1 46433,C(=O)(C#CC1(C)CC1)N(C1CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)C1)CC 46434,N1(C(c2c(C)csc2)=O)CC2COCCC2(NC(c2nc(O)nc(O)c2F)=O)C1 46435,C1(C(C(=O)OC)NC(=O)CCc2cncs2)CCCCC12CC2 46436,c1(C(N2CC(C(=O)NCCOCCO)C(O)C2)=O)cccc2cnsc12 46437,c1(C(N2CC(C(=O)NC3(CO)CCCC3(C)C)(SC)C2)=O)cc2ccccc2[nH]1 46438,c1(C(=O)NCC(CNC(CS(CC)(=O)=O)=O)(C)O)cc2ccccc2nc1CC 46439,C1(CNC(C(C)=C2CC2)=O)CCN(C(=O)CN2CCC(C)C2)C1(C)C 46440,C1(CC(=O)NC2C(=O)N(Cc3ccc(Br)cc3)CC2)CCC2(CCNC2)CC1 46441,c1(CC(=O)NC(c2cccnc2)C(=O)NC(CSCC)CO)cn(C)cn1 46442,CCC(CC(=O)NCC1CCN(C(=O)CC2CN(C(C)=O)C2)CC1)C1CC1 46443,CC1OCCC1OCCC(=O)NCC(=O)NC1CCCC1 46444,C1(CN(C(C)=O)C(c2c(F)ccc(I)c2F)=O)CCC2(CCC2)CN1C 46445,C=CCCC(F)(F)C(=O)NC1CN(C(=O)Cn2cnnc2O)CC2(CC2)C1 46446,C1(NC(c2cc(C(C)C)c(C)o2)=O)CC2CN(C(=O)C=CC(=O)N(C)C)CC12 46447,CC1=NOC(=O)C1CC(=O)NC1CCC(C(=O)Nc2nncs2)C1 46448,O1NC(=O)C(C)(C)C2CCCN(C2)C(=O)C1.CC(C)(C)OC(N)=O 46449,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46450,N1(C(C2C(N(C)C(c3cc(C4CC4)no3)=O)C2(C)C)=O)CCC2CC12C 46451,c1(NC(C2CSCCN2Cc2scc(Br)c2Br)=O)ccc(O)cc1Br 46452,c1(C(N2C(C)CC(CNC(=O)CSc3ccccn3)C2)=O)ccc2c(c1)CCN2 46453,C1(CN(C(=O)CC(O)c2ccccc2)C)COCCN1C(=O)C=CI 46454,c1(C(=O)NCC2CCC(NC(c3cc[n+]([O-])cc3)=O)CC2)ccc2c(c1)COC2 46455,N1(C(c2nnn(CC)c2C)=O)CCCC(C)(NC(=O)CCc2cc(Cl)cs2)C1 46456,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(O)CC(F)F)cc1OC(F)F 46457,N1(C(c2ccc(CC)o2)=O)CC2CCOC2(CNC(=O)CC(C)P(C)(C)=O)C1 46458,c1(NC(CC)C2CCC2)ncnc(N2CC3CC2C3)c1C 46459,c1(N2CCCC(OCC)C2)cc(NCCC2CC(O)C2)nc(CC)n1 46460,C1(NC(c2scc(C)c2)=O)CC(CNC(=O)Cn2nc(C)nc2C)CC1O 46461,N1(C(CC(=C)Br)=O)CC(OC)C(NC(=O)C(C)CC2CCC2)C1 46462,C1(OC)CN(C(=O)CC(C)O)CC1NC(c1cc(C(N)=O)no1)=O 46463,N1(C(CCSCC)=O)CCOCC(CNC(c2cc(Cl)cn2C)=O)C1 46464,C1(CN2CC3(OCCC(N)C3)C2)CCC2(CCCCC2)CC1 46465,CC1CCCC1C(=O)NCC(C)(C)CNC(c1ccn(Cc2ccccc2)c1)=O 46466,c1(C(=O)NCC(CN(C(COC(CC)C)=O)C)O)csc(O)n1 46467,Cc1ccc2[nH]c(C(=O)NC(C3CCN(C(=O)CO)C3)(C)C)cc2c1Br 46468,c1(C(C)=O)cc([N+](=O)[O-])c(N2CC(C)(NC(=O)C(C3CCC(=O)N3)C)C2)cc1F 46469,C12(CC)CCC(C(=O)NC3CCC(NC(=O)CCc4ccn(C)n4)CC3)(CO1)C2 46470,C1(C(N2CC(C(C(N3CCC(CN=[N+]=[N-])C3)=O)OC)C2)=O)CC=CC(O)C1 46471,c1(N(C)C)ccc(NC(=O)NC(=O)CCC2CCC2)cc1.c12ccc(cc1)CN2 46472,N1(C(c2cccc(CC)c2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC(O)C1 46473,c1(C(=O)OC)ccc(Cn2cc(C(N3CCC3CCCC(=O)OC)=O)nn2)cc1 46474,C(=O)(CC(C)C(C)(C)NC(c1cc(Cl)ns1)=O)N1CC(CC)N(C)CC1 46475,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46476,c1(OC)cc(C(=O)NC(c2ncc[nH]2)C)cnc1-c1cnnc(C)c1 46477,c1(C2C(C)C2)ncc(C(=O)N(C)CCOCCCNC(=O)C(C)(C)F)s1 46478,C1(CC(=O)NC(C(=O)N(CCCC)CCO)c2ccoc2)CCCOC1 46479,C(C(=O)NC1CC1C(=O)OC(C)(C)C)(C(C)(C)C)NC(NNC(=O)OC1CC1)=O 46480,N(C1CCCc2c[nH]nc21)C(C(c1cccs1)NC(c1cncs1)=O)=O 46481,C(C(C)(CC)C(=O)NC1C(=O)OCC1CO)NC(CC(CC)C1CC1)=O 46482,C12(C(=O)NC(C3(O)CCN(C(C4(C)C(C)(C)C4(C)C)=O)C3)C)CCCC1C2(F)F 46483,C1(=O)CCCCCN1.C(=O)(CC(C)(C)C)NC(C)C(C)NC(=O)C1=CCC1 46484,C(C(=O)NCC1CCC(NC(c2nccn2CC)=O)CC1)(C(C)C)SCC 46485,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OCF)cn1)=O 46486,N1(C(C(C2CCC2)OC)=O)CCC12CN(C(=O)CCCSc1ccccc1)C2 46487,c1(C(N2CCCC(CN(C(C3C(C)C3)=O)C)C2)=O)ccc(F)c2occc12 46488,C(=O)C1CCCc2nn(C)cc21.C1(C)CC1C(=O)NCCN(CCOC)OC 46489,C(=O)(C(F)(F)C(C)(C)O)NC1C(NC(c2n[nH]c(C)c2C(F)(F)F)=O)CCCC1 46490,c1(C(=O)NC2CC(C)CN(C(C3CC4C(C3)C4(C)C)=O)C2)coc2c1CCCC2 46491,C1(CNC(c2c(C)ocn2)=O)CC2CC2N1C(=O)C#CC(C)C 46492,C1(C(=O)OCC)CC(C)(C)CN1C(=O)CN(CC)Cc1ccc(CC)nc1 46493,c1(C(N2CC(C(C)NC(C3CCCS(=O)(=O)C3)=O)C2)=O)ccc2c(c1)C=CCC2 46494,C1(C)(C(N(CC(C)C(=O)NCc2cccnc2O)C)=O)COCCO1 46495,c1(C(=O)OC)[nH]c(C)cc1NC(N1CCOC(CCC(F)(F)F)C1)=O 46496,N1(C(C=CCOC)=O)CCC2(CC2C(=O)NCC(C)(C)CO)C1 46497,C(=O)(C(C)CCCOC(C)=O)NCc1cccc(C(N2CC(CC#C)OCC2)=O)n1 46498,C(C(CSC)C(F)(F)F)NC(=O)C(O)C(C)C.N1(CCC)CCCC1C=O 46499,C1(CNC(C(c2cccc(C)c2)C)=O)CCCN(C(C2CCCC2(C)C)=O)CC1 46500,CC1CC(NC(C2CN(C(=O)C(C)(C)c3ccccc3)CCS2)=O)CCO1 46501,c1(C(=O)NC(C=CC(=O)N(C)Cc2cn(CC)nc2)(C)C)cc(F)n(C)n1 46502,c1(C(N2CC3C(C2)N3C(c2coc(Cl)n2)=O)=O)ccc2sccc2c1O 46503,C1(C(N2CC3C(NC(CN(C)S(N)(=O)=O)=O)(C3)C2)=O)CCN2CCCCC12 46504,C#CCCCC(c1nnnn1CC=C)NC1CCCN(C(=O)NC)C1 46505,c1(C(N2CCC(NC(c3cnc(-c4ccsc4)s3)=O)CC2)=O)cnn2c1OCC2 46506,c1(C(N2CCc3nc[nH]c3C2)C(=O)NC(C)C)cc(F)c(Br)cc1F 46507,C1(COC)CCC(C)CN1C(C1CCN(C(=O)C(C)=C2CC2)C1C)=O 46508,CCC(CC(=O)NC(Cn1ccnn1)C(=O)Nc1cc(C)nnc1O)C(C)C 46509,c1(CN(C2(O)CC2)C(=O)NCc2ccc(Cl)cn2)ccc(Br)cc1C(F)(F)F 46510,c1(C(=O)NC2CCN(C(CC(CC)OC)=O)CC2(C)C)cc2c(C)cccn2n1 46511,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)CCSc2ccccc2)CC1C 46512,C1(N(C(=O)CC2COC(=O)C2)C)CCN(C(c2cnc[nH]2)=O)CC1 46513,c1(C(=O)NCCNC(C(C2CCOC2)OC)=O)cn2cccnc2n1 46514,N1(C(CCC#C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46515,c1(CSCC)ccccc1SC(C)C(=O)NCCCCCC(F)(F)F 46516,C1(C(=O)N(C)CC2C(C)(C)C2(C)C)(NC(CC(C)SC)=O)CCC(C)(C)C1 46517,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46518,c1(C(C)C)cn2c(n1)CC(C(=O)OCCc1ncco1)CC2 46519,C1(NC(Cn2cc(CN(C)C)nn2)=O)COCCN(C(C2CCCCC2O)=O)C1 46520,N1(C(c2cc(CC)nc(O)c2)=O)CCC(CNC(=O)C(C(C)C)SC)C(O)C1 46521,Cc1cc(CC(=O)N(N2CCN(CC(c3ccc(Cl)cc3)O)CC2)C)cc(C)n1 46522,CCCCC(CC)C(=O)NCC12CC(NC(=O)C=CC(CC)=CC)(CO1)C2 46523,C1(NC(Cc2cc(C)no2)=O)CN(C(=O)C(=O)N(C)C)CC1C1CC1 46524,N1(C(c2c(OC)csc2)=O)CCN(C(C2CCC(Cl)CC2)=O)C(C2CCC2)C1 46525,Cc1nc(C(=O)NC2CCC2NC(c2csc(Cl)c2)=O)c(C)s1 46526,C#CC1(C)COCCN1C(=O)CC1CCN(C(c2cnn3c2OCC3)=O)C1 46527,N1(C(c2n(C)nc(O)c2)=O)CCCC2(CCCCC2NC(=O)C(F)=C2CCC2)C1 46528,CN1CCCC(Oc2ccoc2CCn2ccnc2)C1.C12CCN(CC1)C(=O)N2 46529,C1(CC(N2CC=CC(NC(c3c(C)c[nH]n3)=O)C2)=O)CCCC(F)(F)C1 46530,C1(C(N2C(C)CC(CNC(CCC(C)N(C)C)=O)C2)=O)CC2(CCO1)CC2 46531,C1(CNC(C(CC)OCC)=O)CCC2(CCN(C(=O)C(F)C(C)C)CC2)CO1 46532,CC1CN(C(=O)C(CNC(=O)CC2C=CCC2)N(C)C)CCS1=O 46533,C1(O)(CNc2c(OC)n[nH]c2)CCCN(C(c2cc(Cn3cccn3)on2)=O)C1 46534,C1(N(C(=O)CC2CC(O)C2(C)C)CC=C)CCC(CC(=O)NCCNC(C)=O)CC1 46535,C1(N(C(C(C)SC)=O)C)CCC(NC(c2nnsc2SC)=O)CC1 46536,C12CC(=NO1)C(=O)NCC(C)(C)CNC(=O)CCN2C.c1(S)ccccn1.CS 46537,c1(OC)cccc(CC(=O)NC2CN(C(C3(C#N)CCCOC3)=O)CC2C)c1C 46538,CC1(CC(=O)NC2CCOC2C(=O)N(CCCO)CCCO)OCCO1 46539,Cc1cccc(C(=O)NCC2CN(C(c3cn(C4CC4)cn3)=O)CC2C)c1 46540,C12(C(N)=O)CC3CC1C2C3O.C12(CNC(C(c3ccnn3C)C)=O)CN(C1)C2=O 46541,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46542,CCC(C)C(C(=O)NC1(C)CSC1)NC(C1CCCSC1C)=O 46543,C1CCCNC(C#C)C2CCN12.N1(C(C2CCC2)C)CCCC1 46544,c1(C(C)C)cnc(C2CC2)[nH]c1=NC(=O)C1(CN2CCOc3c(Cl)cccc32)CC1 46545,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)cc(C(C)C)n(C)n1 46546,c1(C(N2C(C)(CNC(CC(C)F)=O)CC(F)(F)C2)=O)nc2c(s1)COCC2 46547,CN1CCc2cc(C(N3CC(NC(C4CC4F)=O)CC4(CCC4)C3)=O)sc2C1 46548,c1(NC(C2CCN(C(C3(C)CCCCC3)=O)C2)=O)cc(Br)c(F)cc1Br 46549,C1(C)(NC(C(CCCC)NC(C2CCC2CCOCC)=O)=O)CCC(C)=C(C)C1 46550,C12(CCNC(c3c(SC)nc(C)nc3)=O)CCC(C1)N(C(=O)C(C)(C)C)C2 46551,C1(C(=O)NC(C)CNC(C)=O)CCN(C(C2(SC)CCC2)=O)CC1 46552,C12(C(N3CC(CCC)C(NC(c4cn[nH]c4)=O)C3)=O)CCC(CC1)CC2 46553,C1(C(=O)NCC2CC(NC(C(COC)O)=O)C2)Cc2cc(C)ccc2S1(=O)=O 46554,c1(C(=O)NC(C)CCF)ccc(CNC(=O)CCSC2CCCC2)nc1 46555,C1(CNC(CCSC)=O)CC(C)N(C(=O)CN(C)C(N)=O)C1 46556,C12(NC(c3ncn(C(C)(C)C)n3)=O)CCN(C(=O)C(Cl)=CCl)CC1C2 46557,C(=O)(C1OC(=O)c2ccccc21)N1CC(NC(CCC)=O)C(C)(C)CC1 46558,CCCC(CNC(=O)C(CC)OC)C(=O)N(C1CCN(CC)C1)C 46559,c1(NC(=O)NCC(C(CC)C)OC)cnc(C)c2c1COC(C)(C)O2 46560,C(CC(C(N)=O)NC(=O)C(C)N(C)C(C)C)OC 46561,C1(NC(C(=O)N(C)C)=O)CC2CCC1N(C(c1ccccc1Cl)=O)C2 46562,c1(CC)ocnc1C(=O)NCC(CNC(=O)Cn1cnnc1O)OC 46563,N1(C(c2c(CC)csc2)=O)CCCC(NC(=O)CN2CCCCCC2=O)C1C 46564,C1(C)(NC(c2cc(C)n(C)n2)=O)CCCCC1C(=O)N(C)Cc1cn(C)nn1 46565,S(=O)(=O)(c1sc(O)nc1C)N(C1CC2CC1CC2(O)C(F)(F)F)CC 46566,C=C(C)CCN=c1[nH]c(=NCC2(CF)CCOCC2)[nH]c2cccc(F)c12 46567,c1(CC)cc(NCC(CC(C)C)NC2CC2N(C)C)nc(C)n1 46568,NC(=O)C(N)CCC(=O)N1CCOCC(CNC(c2ncon2)=O)C1 46569,CC1CCN(C(C2(CCF)CCC2)=O)CC1CNC(=O)CCC(C)(C)F 46570,C1(C(=O)NC2(C)CN(C(c3cnn(C)c3C3CC3)=O)C2)CC2CCCCN2C1 46571,Cc1c(C(N2CCC(NC(c3cncc(Cl)c3)=O)C2C(C)C)=O)ccn1C(C)C 46572,C(c1ccc(OC(C)C(C)(F)F)c(OC)c1)=Cc1ccc(C)cc1 46573,CCC(C(=O)OC)C(=O)NCc1cc(C(=O)N(CC)CC)on1 46574,c1(C2C(C(=O)NC3C(NC(c4c(C#C)c[nH]n4)=O)C3)C2)ccc(Br)cc1C 46575,Cc1csc(CCC(N2CC(O)(CN(C(=O)C=CC(c3cn(C)cn3)=O)C)C2)=O)n1 46576,Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NC1CCN(C(=O)C=CC=C(Cl)Cl)C2CC12 46577,c1(CC)nc(C)c(C(N2CC(O)(CNC(=O)Cn3nnnc3C3CC3)C2)=O)o1 46578,C1(C(N2CC(C(C)NC(=O)C=Cc3cn(C)nn3)C2)=O)CCCCC1(C)C 46579,c1(C(=O)NCCCOCCCNC(COCC)=O)cc(Cl)c([N+](=O)[O-])[nH]1 46580,C#CCC(C)(C(=O)NCC(O)C(=O)Oc1ccc(C#N)cc1)NC(N)=O 46581,N1(C(CCc2n(C)c(S)nn2)=O)CCCN(C(=O)Cc2cccnc2O)CC1 46582,C1(CC(=O)NC2CCC(NC(=O)CCC3CCC(=O)N3)C2)CCC(=O)NC1=O 46583,N1(C(CSC(C)C)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 46584,N1(C(C(CC)(C)C)=O)CCC2CN(C(c3c(OC)ccnc3F)=O)CCC2C1 46585,C(CC(C)C)(C(=O)OC)N(C(c1ncoc1C)C(=O)NCC=C)C 46586,n1(CC)nc(C(=O)NC2CC2CNC(=O)CCc2cc(C)n(C)n2)cc1C 46587,N1(C(CC2C(C)OC(C)C2)=O)CC2CC1CCC2NC(=O)Cc1nncs1 46588,c1(CC)nn(C)c(N2CCCC(C)(NC(c3ccn(CC)n3)=O)C2)c1[N+](=O)[O-] 46589,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46590,c1(C(=O)NC23CC(NCc4cc(Br)cs4)(C2)C3)cc(Cl)cnc1O 46591,c1(SC)cc(N)c(OC)cc1N1CCCC1C(=O)NCc1cscn1 46592,c1(N(CC(C)NC(CCc2c(C)cccn2)=O)C)ncc2c(n1)CCCCC2 46593,N1(C(C2(c3n(C)ncc3)CC2)=O)CCC(NC(C2CCCCC2O)=O)CC(O)C1 46594,C1(NC(=O)CCCn2ccccc2=O)CN(C(=O)Cn2nccn2)CCC1CO 46595,c1(C(=O)NC2C(CCNC(c3c(OC)ccc(C)c3)=O)C2C)nc2cccnc2s1 46596,C(=O)(C(O)CCCNC(=O)CC1CCOC1=O)N1CC(C(C)OC)C1 46597,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(C(=O)Nc3cc(I)cnc3Cl)C2)C1 46598,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CCOCC3)CC2C)cc(O)cc1N 46599,N1(C(C2(C#C)CCC2)=O)CCOC(CN(C(=O)C(c2ccc(C)cc2)C)C)C1 46600,c1(CC)ncc(C(=O)NCCOC2CCN(C(C3CC3(C)C(F)F)=O)C2)c(O)n1 46601,c1(C(N2CCC(CN(C)C(C3(C)CCOCC3)=O)CC2)=O)cc2ccnn2cn1 46602,Cc1nnc(N2CCC2C2CCCCN2C(c2ccn(C)c2)=O)nc1C 46603,c1(OC)cc(C(=O)NC(C2CCCC2)CNC(C2C=CCC2)=O)ccc1Br 46604,N1(C(C2(CC=C)CCCC2)=O)C2CCC1C(CNC(c1cc(C)ns1)=O)C2 46605,c1(C(N2CCCC(CC(=O)NCC(CCCC)O)C2)=O)cccc(Cl)c1Cl 46606,CCCC(C(=O)NCC(CO)NC(c1c[nH]nc1-n1cnnn1)=O)N(C)C 46607,CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC2C=CC1O2)C 46608,c1(CCC(=O)N(C(CCNC(C(CC2CCC2)OC)=O)C)C)cnc(C(C)C)o1 46609,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(NC(C2CCC2(C)C(=O)OC)=O)C1 46610,c1(C(=O)NC2(C(NOCCC#CC)=O)CC2(C)C)cnn2c1CCC2 46611,CN1CC2CCCC(C1)N2C(c1sccc1CNC(C1CC1Cl)=O)=O 46612,c1(OC)ccc(C(N2CCC(O)(C(C)NC(C3C4CCCC34)=O)C2)=O)cc1 46613,C(=O)(C(F)CC(C)(C)C)N1CCC(N(C(CNC(CC(CC)SC)=O)=O)C)CC1 46614,c1(C(N2CC3C(CNC(c4cccc(N)c4F)=O)C3C2)=O)nc2c(s1)COCC2 46615,C1(C(=O)NCC(CCOC)NC(CC(C=C)(C)C)=O)CCC2(CC1)CNC(=O)C2 46616,c1(C(=O)NC2CCN(CC(=O)NCC)CC2C)c[nH]c2c(Cl)cccc12 46617,C1(C2CCC2)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnc(O)c(C)c2)=O)CC1 46618,C1(CNC(c2ccccc2F)=O)C2CN(C(c3nc(C4CC4)cs3)=O)CC12 46619,C(c1cncnc1O)=CC(=O)NCC1(C(C)NC(=O)C2=CCSC2)CC1 46620,c1(C(=O)NCCNC(c2cc(OC)c(O)c(I)c2)=O)cc2n(c1)CCCC2 46621,CC(CCCCNC(C1CCN1C)=O)NC(c1ccc(OC2CCCC2)nc1)=O 46622,CCCC(CCCNC(=O)Cc1nonc1C)NC(c1c(C)nn(CC)c1C)=O 46623,N(C(=NCCC(O)C(F)(F)F)NCC(C)(C)C(=O)OC)CC1CC(C(=O)OC)C1 46624,c1(N(C)Cc2nc(CC)sc2)nc(=NC)[nH]c(=NCCCC(=O)N(C)C)[nH]1 46625,C(=O)(CCC(=O)c1cncnc1)NCCCNC(c1c(CN(C)C)ccs1)=O 46626,C1(NC(c2cn(CC)nn2)=O)COC2(C1)CN(C(c1c(C)cnn1C(C)C)=O)C2 46627,C(CC(=O)N1CC2CC1CN2C(=O)CC(C)(C)C(F)F)(C(F)(F)F)OC 46628,c1(SC)cc(C(=O)NCCC(c2ccccc2F)N(C)C)ccc1[N+](=O)[O-] 46629,C=CC(C)(CC)C(=O)NCC1CCOC(C)C1 46630,c1(NCCn2ccc(C(=O)OC(C)C)c2)cccc(C(=O)O)c1 46631,c1(C(C)=O)cc(C(=O)NCC2CN(C(C3CCC3)=O)CC23CC3)c(C)nc1C 46632,N1(C(c2c(C)cnn2C)=O)CC(C)(C)CC1CC(=O)NCCc1nc[nH]n1 46633,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)N(CC(C)CO)C 46634,C1(NC(CS(=O)(=O)NCC)=O)CCCC12CN(C(=O)CC1CCCCN1C)C2 46635,C(=O)(C1=NNC(=O)CC1)NC1CCC(NC(c2cnc(C(C)O)s2)=O)CC1 46636,C(=O)(C1=CCC(C)(C)CC1)NC1CCC(F)(CNC(C2(CCC=C)CC2)=O)C1 46637,c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46638,C=C(C)C(CC(=O)NCc1ccsc1C(=O)NC(C)CSC(F)F)OCC 46639,C(CCCO)N(C(C1CC1CNC(C1CC1Cl)=O)=O)CC 46640,c1(C(N(CCCNC(CSCC)=O)CC)=O)ccc(SCc2ccccc2)cc1OC 46641,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)C3CC23)c1 46642,c1(OCC(=O)NC(C)CNC(C2CC2C(F)(F)F)=O)cc(C(N)=O)ccc1O 46643,C1(C(C)(C)N(CC(N2CCSCC2)=O)C(=O)CC2CCO2)CCCCC1 46644,C(=O)(C(C(=O)NC(C(=O)NCCCC1CC1C)C1CC1)OC)OC 46645,C(C(C)(CNC(=O)CC)NC(CN(CCC#C)C)=O)NC(C)=O.C(C)(CC)O 46646,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2(CC(NC(=O)CC3CC34CC4)C2)C1 46647,C(=O)(C1OC(=O)c2ccccc21)NC1(CN(C)C(C2CCC=CO2)=O)CC1 46648,N1(C(c2n(CC)c(O)nc2)=O)CCC(C)(NC(=O)CCCOC(C)=O)CC1 46649,N1(C(C2(F)CC2)=O)CC2CCC(C1)N2C(C1C2CC2C2CC12)=O 46650,c1(C(C(=O)N(CCCN(C(Cc2c(C)cc(C)s2)=O)C)C)O)ccc(Cl)c(Cl)c1 46651,c1(C(=O)NC2(CC(=O)N(CC(C)CO)C)CCC2)cnn(C(C)C)n1 46652,C1(C=O)CCN(C)S1(=O)=O.n1(C(C)C)cnc(C(N2CCC(N(C)C)C2)=O)n1 46653,CCC(CC)(CC)C(=O)NCCCN(C(=O)Cc1cncs1)Cc1ccccc1 46654,N1(C(c2cc(C)c(Cl)cc2C)=O)CCn2c(C(F)(F)F)nnc2C1 46655,CC1CN(C(=O)CC2CCCNC(=O)C2)CCCN1C(C1CN(C2CCC2)C1)=O 46656,C(C1CCc2ccccc21)N(C(CC)C(C)(F)F)C 46657,c1(C(=O)NCC2(O)CN(C(CCN(C)CC)=O)C2)cc(C(C)=O)c(C)o1 46658,CCCC(C(O)C(=O)NC(C(C)C)C1CC1)NC(=O)CCCn1ccnc1 46659,N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2n[nH]c(CC3CC3)n2)=O)CC(CO)C1 46660,c1(OC)cc(C)cnc1C(N1CCC(C)(NC(c2cncs2)=O)C1)=O 46661,c1(C(=O)OCC)cccc(CS(=O)(=O)NCC(C)(C)F)c1 46662,c1(CNC(C2(CC)CCCCC2)=O)ccc2c(c1)CN(C(=O)CCC(C)SC)C2 46663,c1(NC(CC(CNC(CCc2ccc(C)o2)=O)C2CCC2)=O)nc(C)ccc1C 46664,CCC(C)C(C)C(=O)N(C)CCN1CCN(C(c2ccnc(N(C)C)c2)=O)CC1 46665,N1(C(c2cc(CC)no2)=O)CC2CC2(CC(=O)NC2CCCN(CC)C2)C1 46666,c1(C(=O)NC(C2CN(C(C3C(OCC)C3)=O)C2)C)nccn2ccnc12 46667,C1(N(C(CCOCCOC)=O)CCF)CCCN(C(=O)CC2(C#N)CCC2)C1 46668,N1(CC)CCCC(C(=O)NCC(O)CN(C)C(C2CCNC(=O)C2)=O)C1 46669,C(CN=c1nc(N2CCC3(CCCO3)C2)cc(C)[nH]1)(C(C)(C)C)SCC 46670,C(CCO)(C(=O)N1CCCC(NC(=O)CN(C)CCN(C)C)C1)N(C)C 46671,C1(N(C(COCC#C)=O)C)CCCC(N(C)C(c2cc(CC)[nH]n2)=O)C1 46672,c1(C(N(C)CC2CCCN2C(C2CCCC2(C)C)=O)=O)cc2c(s1)CCC2 46673,c1(CNC2CC(C(=O)NCc3csc(C(F)(F)F)n3)C2)ccnc([N+](=O)[O-])c1 46674,C1(C(N2CCC(CO)C2)=O)Cc2nccnc2CN1C(=O)C1=COCCC1 46675,C(=O)(C(C)(C)CC(C)(C)C)NCCN(C(=O)Cc1csc(N2CCNC2=O)n1)C 46676,N1(C(C)=O)CCCCC1c1n[nH]cc1C(=O)NCCCO.n12cc(nn1)CCC2 46677,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)NCCN(C)C(N)=O 46678,C(=O)(CCCCCn1cnnn1)NC1CCCN(C(c2ccc(OC)cc2)=O)C1 46679,c1(C(N(C2CCC(CNC(=O)C(O)C(C)C)CC2)CC)=O)cc(P(C)(C)=O)ccn1 46680,c1(C(=O)NC(C)CNC(=O)CCF)occc1CN(C)C 46681,N1(C(Cc2c(C)ncs2)=O)CC(NC(=O)C(C)C(C)(F)F)CC2(CC2)C1 46682,CC1CCN(C(=O)COC2CCC2)C1C(=O)NCc1ccc(F)cc1 46683,c1(C(=O)NC2CC(C)(C)CN(C(=O)CCF)C2)cc(Br)c2nccn2c1 46684,C(=O)(CCCC(=O)N1CC2(COC)CC1(CC)C2)OCC.C(=O)(C1CC1)NC 46685,c1(C(=O)NCCC(=O)N(CCNC(C2(C)C=CCC2)=O)CC)ccc(F)c(F)c1 46686,c1(C(=O)NC2C(C)CCN(C(c3cccc(Cl)c3F)=O)C2)c(F)ccc(F)c1N 46687,N1(C(c2n(CC)cc(Cl)c2)=O)CCN(C(C2CCC(OC)CC2)=O)C(CO)C1 46688,C1(C(=O)NCCC2CN(C(C(c3ccc(F)cc3)(C)C)=O)C2)CCC12CCCO2 46689,c1(C(N2CCC(NC(CC(CC)C(C)C)=O)C(O)C2)=O)cccc2c1ccn2C 46690,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cccs1)=O 46691,CN(C1CN(C(=O)CCCC2CCCO2)CCc2ccccc21)C(=O)C=C1CCC1 46692,C(=O)(C(C)(C)CC(C)(C)C)NCc1ccc(C(C)NC(c2nccc(C)n2)=O)cc1 46693,CCC(N=c1cc(NCCOCC2CCCCO2)nc(C(F)(F)F)[nH]1)C(C)C 46694,c1(N2CCN(C(C)CO)CC2)nc(N(C)CC2CCCO2)c2cnn(C)c2n1 46695,C(=O)(C(F)n1ccnc1)N(CCN(C(c1cnn[nH]1)=O)CC)CC 46696,C1(CNC(=O)C#CC2CC2)COCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)O1 46697,N1(C(C2(CCN=[N+]=[N-])CCC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 46698,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 46699,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)O)=O 46700,c1(C(N(C(C)CNC(C2CCN2C(C)(C)C)=O)C)=O)c[nH]nc1C(C)(F)F 46701,N1(CC)CC(NC(=O)Cn2cc(CNC(c3nc(C)c(C)s3)=O)nn2)C(C)C1 46702,C1(NC(c2cc(CC)[nH]n2)=O)CCCCN(C(c2cnc(C)cc2Cl)=O)C1 46703,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(F)c2)c1 46704,Cc1cn2c(n1)C(C)N(c1nc3c(c(=NCc4cnn[nH]4)[nH]1)COC3)CC2 46705,c1(C(=O)NCCN(CCC)C(C)C)cnn(CCNC(=O)CCN2CCCC2)c1 46706,N1(S(C)(=O)=O)CCCN(c2cccc(-c3nc(C)n(CCF)n3)n2)CCC1 46707,N1(C(CCC(=C)C)=O)CCC(C)N(C(=O)CC2CC(C)(C)C(=O)N2)CC1 46708,C1(C(N(C2CC(NC(=O)CNC(=O)C(C)(C)C)C2)C)=O)CCCC(C)CC1 46709,c1(C(N2CCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ncc(Br)cc1F 46710,C1(CNC(c2c(C)ccs2)=O)CN(C(c2ccsc2C(F)F)=O)CCC1C 46711,c1(OC)cc(F)cc(C(=O)NCCCCNC(C2(C)CC(F)C2)=O)c1N 46712,c1(C(C)NC(c2nnc(OC)s2)=O)ccc(Cl)c(C)c1O 46713,N1(C(c2cc(OC)n[nH]2)=O)CC(NC(C2(CO)COC2)=O)CC12CCOC2 46714,CC(C(=O)N1CC(CN2C(=O)CC2)C1)C(C)(C)C.c1(SC2CCOC2)ccccn1 46715,c1(NC2CCCN(C)C2)cccc(S(=O)(=O)N(C)CC2CC(O)C23CCC3)n1 46716,C(CCCC(CO)NC(=O)C(C(C)C)N(C)C)NC(Cc1c(SC)cccc1)=O 46717,N1(CCN(c2cncnc2)C(=O)NCCC2CCCO2)CCOCC1 46718,Cn1nc2c(c1C(N1CCCC(CNC(C3CCSC3)=O)C1)=O)CS(=O)(=O)CC2 46719,c1(CNC(CCn2cc(C3CCN(C)C3)nn2)=O)ccc2c(n1)OCCO2 46720,C#Cc1ccnc(C(=O)NCC(O)CNC(=O)COCC2CCCCO2)c1 46721,c1(CCC(=O)NC(C)CCCNC(=O)C=CC2CCCO2)c(F)cccc1Cl 46722,CC1CN(C(=O)CCCn2cc(Cc3ccccc3)nn2)CCN1c1nccs1 46723,C1(C(=O)NCCCN(C(C(CC=C)CC=C)=O)CC)CC(C)(C)SC(C)(C)C1 46724,C1(C(=O)NC)CCN(C(=O)Cc2cccnc2)C1.c12sccc1CNC2=O 46725,CC1CCCC1C(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 46726,c1(C(=O)NC2(CC)CN(C(=O)C#CC3CCOC3)C2)cc(OC)c(C)c(OC)c1 46727,C1(OC)CCC(CC(=O)NCC23CC(CN2C(c2c[nH]nc2C(F)F)=O)C3)CC1 46728,C(=O)(C1Cc2c(Cl)cccc21)NC1C(S(N)(=O)=O)CN(C(=O)CCN2CCCC2)C1 46729,c1(C(C)=O)c[nH]nc1-c1ccc(-c2nccn2CCn2nccn2)s1 46730,C(C)(C)(CC(=O)N(C1CCCC1)CCCNC(=O)Cc1cc(C)ns1)OC 46731,C1(NC(=O)CCC2CC2)CCN(C(c2cnc3n(c2=O)CCS3)=O)CC12CCC2 46732,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 46733,N#Cc1cccc(N2CCN(C3CCN(C(=O)COCC4CC4)C3)CC2)c1 46734,CC1(NC(c2cc(C(F)(F)F)on2)=O)CCN(C(C2CCC(=O)C2)=O)C1.C=O 46735,c1(C(=O)NC2CCN(c3nc4cccc(F)c4o3)C2)cc2cc[nH]c(=O)c2s1 46736,N1(C(CNC(C(C=C)C)=O)C(F)F)CCN(C(=O)CC2CC2CN(C)C)CC1 46737,C1(NCCOC(C2(n3cncn3)CC2)=O)CC(C(=O)NC2CCOC2)C12CCC2 46738,N1(C(c2c(C)c(-c3ccccc3)on2)=O)CCC2C(NC(=O)CNC=O)C2CC1 46739,N1(C(CC(=O)NCC)=O)CCC(NC(C2C=CC(C(N)=O)C2)=O)C12CC2 46740,N1(C(c2ncn(C)c(=O)c2)=O)CCC(CNC(=O)CC2COCCO2)C(F)(F)C1 46741,c1(N2CCCC(C(=O)OC)C2)cc(Oc2ccccc2)cc(Br)c1C 46742,CC(C)CCC(C(=O)NCC1CCSC1)NC(C1CC2(CCCO2)C1)=O 46743,C1(NCC=CC(=O)NCCOCCOCC)CCCC1C(N)=O 46744,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 46745,c1(CC)cscc1C(=O)N(CCOCCNC(=O)CCCC1CCCC1)CC 46746,c1(N2CCC(NC(C(CC)C)=O)C(F)C2)nc(C)nc(C)c1F 46747,c1(NCC=CCOC)c(F)cc(F)cc1Br 46748,C1(C(=O)OCC(c2ccc(C(C)C)cc2)C)(OC)CCCC(C)(C)C1 46749,CCC(Cn1cncn1)N=c1[nH]c2c(c(=NCCCCCO)[nH]1)CSC2 46750,Cn1c(C(=O)NCC2COCC2NC(c2c[nH]nc2C(F)F)=O)nnc1S 46751,N1(C(C2CCC(C)O2)=O)CC(C)(C)CC1CNC(c1cnc(C2CC2)nc1O)=O 46752,C(=O)(CC1=CCCC1)N1CCC(CCCNC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1 46753,c1(OC(C)C)ccc(C(=O)N(C(C)CN(C)C(c2ncn(C)c2C)=O)C)cc1 46754,c1(C(N2CC(C)C(CNC(c3cnc4ccccn34)=O)C2)=O)cc(F)c(F)c(F)c1 46755,C(=O)(CN=c1cc[nH]cc1)NC1(CNC(C(C)Oc2ccccn2)=O)CC1 46756,c1(C(N2CC(OCCNC(C3=C(C)CCC3)=O)C2)=O)cc2ccc(O)nc2s1 46757,C1(NC(C2(OC)CCC2)=O)CN(C(c2cnc3[nH]ccc3n2)=O)CC1C1CC1 46758,c1(C(=O)NC2CC(CNC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 46759,CCCCCCCC(O)CC(=O)N1CCNC(=O)CC1.N12CC(C)CC1C2=O 46760,CCC(CC)CC(=O)N1CCC(CNC(=O)C(O)CCSC)C1 46761,c1(NC(N(CC(COC)C)CC)=O)cccc2c1OCO2.C12CC(C1)O2 46762,C12(CNC(c3c(COC)cccn3)=O)CCC(CC1)N2C(C1CCCC1(F)F)=O 46763,c1(NC(CC2C(C)(C)CC2)=O)ccc(F)cc1-c1cn(C(C)(CO)C(=O)O)nn1 46764,C1(C)(CC)CC(C(=O)NC2CCC(C(F)(F)F)CC2)CN1C(=O)CC1CN(C)C1 46765,CC(CC(=O)NCC1CCCC1NC(=O)CN1CCN(C)CC1)CC(F)(F)F 46766,N1(C(C(CC(=C)Cl)NC(=O)COCC2CC2)=O)CCC2C(CCN2C)C1 46767,CCC(CC(C)C)C(=O)N1CC(c2ccccc2)C(C)(C)C1 46768,C1(NC(C(C)C#N)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 46769,C(=O)(C1=CC2(CCNC2)C1)N1CCC(C(=O)NCCCSC)CC1 46770,C123CC(CCO1)N(C2)C(=O)C(CC)CN(C)C3=O.CCCCCSC 46771,c1(C(=O)NC2CN(C(CC#C)=O)C2)ccc(-c2ccc(C#C)cc2)cc1F 46772,N12CCC(O)(C1)C2=O.N1(CC(=O)NCC2(C)CCC2)C(=O)CSC1=S 46773,c1(C(N2C(C)(CNC(C3CC(C)OCC3)=O)CCC2)=O)cn2ccccc2n1 46774,N1(C(C(C)NC(=O)NC2CNC(=O)N2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1 46775,c1(OC)cc(NC(=O)CC2(N(C)C(c3sccc3C)=O)CC2)ccc1F 46776,OC1CC(c2nnnn2C2CC2)(NCc2ccccc2)C1 46777,C=CC1(c2cn(Cc3cccs3)nn2)COCCN1C(=O)C(=C1CCCCC1)F 46778,C1(N(C(C(c2ccc(F)cc2)C)=O)C)CN(C(=O)C=CBr)CC12CC2 46779,c1(CC)sc(C(=O)NCC(C(C)C)NC(=O)CCCCN(C)C)cc1C 46780,C1(NC(=O)Cc2ccc(Cl)nn2)CCCN(c2ccccc2)C1 46781,C1(NC(C2CC3(CC3)C2)=O)CCC2CN(C(=O)Cc3ccoc3)CCC2C1 46782,c1(OC)ccc(CC(N2CC(CNC(C3(CO)CC3)=O)C(F)(F)C2)=O)cc1Cl 46783,C(CNC(C1C=CCCC1)=O)(CC(=O)N(C)Cc1ccsc1)OC 46784,N1(C(c2cnc(OC)s2)=O)CCC(NC(c2ccn3nccc3n2)=O)C2(CC2)C1 46785,[N-]=[N+]=NCCCCCC(=O)NCC12CC(CO1)N(C(c1cnco1)=O)C2 46786,CC1(C)CCC(C(=O)NCCCC2CN(C(c3cccnc3O)=O)CCO2)CC1 46787,CCC(C(=O)N(C1CCCN(C(c2csc(C(N)=O)n2)=O)C1)C)C(C)C 46788,C1(O)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)C(C)SCC2CCCO2)CC1 46789,C(CC1c2ccccc2CCN1C(=O)C#CC1CC1)NC(c1coc(Cl)n1)=O 46790,C(=O)(CCCC(=O)NCC(C)NC(C1CSCCS1)=O)Nc1nc(C)[nH]n1 46791,CCC(C)(CCC(C)C)C(=O)NCCNC(c1ccc(-c2cccs2)nc1O)=O 46792,CC(O)CCCCCC(=O)NNc1ccc(N(C)C(C)C)c(F)c1 46793,C=C(C)CCCC(=O)N(C1CCN(C(c2ccncc2N)=O)CC1)CCO 46794,CC(C)(C)C(CO)C(=O)NCC1CC1C(=O)NCc1nccs1 46795,c1(CNCc2cccc(-c3cccc(O)n3)c2)cnn2c1OCC2 46796,CC1=C(C(=O)N2CC3(CC3)CC2CNC(=O)COC2CCOCC2)CCS1(=O)=O 46797,S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1C(NC(CCc2c(C)noc2Cl)=O)C1 46798,Cc1c(C(=O)N(C)CC2CCCCN2C(=O)CCc2cc[nH]n2)nn(C)c1N 46799,N1(C(C(F)=CCC)=O)CCC12CN(C(=O)COc1c(C)cccc1Br)C2 46800,C(CCCCC(=O)N1CCCC1CF)NC(C(C)CC1CCC1)=O 46801,CC1COC2(C1)CN(C(=O)C(C1CC=CCC1)NC(c1nnc(S)n1C)=O)C2 46802,N1(C(C(C2OCCO2)NC(CN(C(=O)OC)C)=O)=O)CC(C)C1C(=O)OC 46803,c1(C2C(C(=O)NC(C(C)C)CNC(C3(C#N)CCCOC3)=O)C2)cc(F)ccc1F 46804,CC1(C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CC2)CC1(F)Cl 46805,C1(C(N(CC(=O)OC)Cc2cccc3ccccc23)=O)CNc2ccccc2O1 46806,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 46807,C(=O)(CCCCCNC(c1cc(O)nc(Cl)c1)=O)N(C)CC1CCCCC1 46808,c1(OC)c(C(=O)NCC(C)NC(c2cnc(Cl)s2)=O)csc1C 46809,c1(SC)c(C(=O)NC2COCC2CNC(C2Cc3cscc3C2)=O)cccc1F 46810,C(=O)(C(C#N)C(C)(C)C)N1CCC(CC)(OC)C1.C1(=O)CCOCCN1 46811,C1(CNC(C2(CC)CCCO2)=O)CC2CN(C(C3(n4cccn4)COC3)=O)CC12 46812,C(=O)(CC(O)c1ccccc1)N(CCCNC(=O)COCC(F)F)CC 46813,C1(NC(C(F)=CC)=O)CCC(C)N(C(=O)CC(=O)Nc2ccc(C(C)=O)cn2)C1 46814,S(=O)(=O)(c1ccc2nc(C)nn2c1)C(C1CCCCCC1)(c1n(CCC)nnn1)C 46815,C(=O)(C(O)C(F)(F)F)N1CC(O)(CCNC(c2ccc(C#C)o2)=O)C1 46816,C(CN=c1[nH]c(=NCc2cc(C)on2)c2sccc2[nH]1)C1C(C)C1 46817,C(C(=O)N1CCCc2nccn21)C1(C(CC2C(C)(C)C2)=O)CC1 46818,c1(-n2cc(CSCCOC)nn2)cccc(C)c1Br.C12(C)CC1C(=O)N2 46819,C(=O)(CC(CCCC)NC(C1OCCC1C)=O)NC(C=C)COC 46820,C1(C(=O)NC2CC(NC(=O)C(C)(C)C)C2)CC=CCN1C(=O)C.CC 46821,C1(NC(c2n(CC)ncc2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 46822,Cc1csc(=NCC(=O)N2CC3C(CNC(C4(C)CNC(=O)C4)=O)C3C2)[nH]1 46823,C1(NC(c2cc(C3CC3)oc2C2CC2)=O)CCN(C(C23CCC2C3)=O)CC1F 46824,c1(OCCCNC(N(C2CC2C2CCC2)C)=O)ccc(C(=O)OC(C)(C)C)cc1 46825,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 46826,C1(C(N(C2CC(OC)C2)C)=O)C2CCC1(c1cccnc1)C2 46827,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CC(C)C3CCCO3)O2)C1 46828,CS(=O)CCCCNC(C1(CCNC(=O)Cn2cccc2)CCCC1)=O 46829,C#Cc1cnc(NCC(=O)OCC(Cc2ccccc2C)CO)nc1 46830,c1(C(=O)NCC2CN(C(C(C(C)C)F)=O)CC2C)ccc(C(N)=O)c(F)c1 46831,C(C1=CCN(C(=O)OC(C)(C)C)CC1)NC(c1nccc(C(C)C)n1)=O 46832,C(C(C)C(F)C(=O)Nc1cccc(Cl)c1)NC(c1c(OC)nn(C)c1)=O 46833,Cc1ccnc(C(=O)NCC(C2CCCC2)NC(c2conc2C(C)C)=O)c1N 46834,C(CCC(O)C(=O)NC(C)C(O)C(F)F)NC(COCC)=O 46835,C1(CNC(CCN(C(=O)CCNC(C2CC2)=O)C)=O)CC2(CCCO2)C1 46836,N1(c2n(Cc3nn(C)c(Br)c3)c(C3CCOC3)nn2)CCC2(CCCCO2)CC1 46837,Cc1cc(C(N2CC(CCO)(NC(=O)C(C)SC(F)(F)F)C2)=O)cnc1C 46838,C(C(C)CC(=O)N(C1CCCCC1)CCO)NC(Cc1c(C)ocn1)=O 46839,C1(CC=C)(NC(=O)C(Cc2cn[nH]c2)NC(C2CCC(=O)NC2)=O)CCOCC1 46840,c1(C(=O)NCC2CCC(NC(C3N(CCC)CCC3)=O)C2)c(C)ccc(F)c1N 46841,C1(CC(=O)NC2(COc3ccccc3)CC2)CCN(CC(F)F)C1 46842,CCCCCCCCC(C)CC(=O)NC1CCC1(C)C 46843,n1(C)cnc2ccccc12.n12cc(nn1)CN(C(CC)=O)CC2C.SC 46844,C(=O)(C(C)P(C)(C)=O)N1CCC(CC2(O)CN(C(CC(C)OC)=O)C2)CC1 46845,c1(C(=O)NCCC(C)N(C(c2cncc(CC)c2)=O)C)cc(C)cc(C)n1 46846,C1(CC(N2CC(NC(c3cn(CC)nc3C)=O)(COC)C2)=O)CC2C=CC1CC2 46847,N(C)(S(=O)(=O)N(C)C)CC(N1C(CCNC(c2ncn(C(C)C)n2)=O)CCC1)=O 46848,Cc1cccc(N)c1C(=O)NCC1CCCCN1C(=O)CCNC(=O)CO 46849,c1(C(=O)NC(CNC(CCC(C)(C)F)=O)C2CC2)ncc(Br)cc1C#N 46850,CC(C)CCCC(=O)NCC(CC(=O)Nc1cscc1C1CC1)C1CCC1 46851,C(=O)(CC(O)CC1CCNCC1)N(c1ccccc1)CCCOCCC(C)C 46852,Cc1cncc(CCC(=O)NCCC(C(C)C)NC(C23COCC(C2)C3)=O)c1 46853,N1(CCOCC)CCCN(C(=O)CONC(C2CCOC(CC)C2)=O)CC1 46854,CCC1=NOC(C(=O)NC2CC(NC(C3(CC(=O)N(C)C)CCCC3)=O)C2)C1 46855,c1(C(=O)NNC(=O)c2occc2F)c[nH]c2ccc(F)cc12 46856,N1(C(c2c(OC)ncnc2C)=O)CCC(C)N(C(c2cc[nH]c2)=O)CC1 46857,Cc1ncc(C(N2CC(C(=O)NC3(C(F)F)CCCC3)C3(CC3)C2)=O)cc1C#N 46858,C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCCCC2N1C(C1CCSC1)=O 46859,C1(C(N(C2CCCCN(C(=O)Cc3ccc(Cl)s3)C2)C)=O)CC2CCCCCC12 46860,C=CCC(C)C(C)(c1nnnn1CC1CC1)NCCc1cc(F)ccc1OC 46861,CC1CCN(C(=O)C(=O)NCC2(CCCNC(=O)Cc3cccnc3)CC2)CC1 46862,C(C1=NOC2CN(C(=O)CC3OCCO3)CC12)NC(c1cc(C)nnc1O)=O 46863,c1(CC(N2CC(N(C(C(C)c3cncs3)=O)C)C(O)C2)=O)cn2ccsc2n1 46864,N1(C(c2ncc(Br)cc2F)C(=O)Nc2ccccc2)CCCC2(CC2)C1 46865,C1(C(N(CC(=O)OCC)CC)=O)CCCC(NC(=O)CCn2cncn2)CC1 46866,C#CC1(C(=O)OCC)CCCC1.C(=O)(C(CCC1CCC1)OC)N1CC(C)(C)C1 46867,C1(C(=O)NCC2C3CN(C(Cn4nnc(C)n4)=O)CC32)CCN2CCOCC12 46868,c1(OC)cc(Cl)cnc1C(=O)OCCCC1CCCCO1 46869,CC1CC(C(C(=O)NC2CCCC2)N(C)CCN2CCOCC2)CCO1 46870,N1(C(C(=O)NCC)=O)CC(C(=O)N(CCCOC)C)C(C2CC2)C1 46871,CCC(C(=O)N1CC2CC1(CNC(c1cccc(F)c1C)=O)C2)C(C)O 46872,c1(C(C(=O)NCCC)N(C(C)C(C)C)C)ccc(OC)cn1.c1(CN)nnn(C)n1 46873,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(C)O)CC1C 46874,N1(C(c2nncc(OC)c2)=O)CCC(NC(=O)CSc2cnn(C)c2)C(C)C1 46875,C1(CC(=O)N(CCNC(=O)Cc2nnc(O)s2)C2CC2)CCCC2(CCC2)O1 46876,N1(C(C2(CC=C)CC=CC2)=O)CCC(F)(F)C(CNC(C2(C(F)F)CCC2)=O)C1 46877,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 46878,N1(C(c2cc(F)c(C)c(F)c2)=O)CC2(C1)CN(C(=O)C(C)S)CC2C(=O)O 46879,C(CN=c1[nH]c(=NC)[nH]c(=NCCCCOC(N)=O)[nH]1)CN(CCCC)C 46880,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(CNC(c2cc(Cl)n(C)n2)=O)C1 46881,c1(OC)cccc(=NC(=O)C(=O)Nc2ccc3c(C)[nH]nc3c2)[nH]1 46882,c1(OC)ccc(OC)c(CC(=O)NCC(C)(O)COCc2nnnn2CC)c1 46883,C(N=c1[nH]c(N2CCCOCC2)nc2ccc(-c3ccccc3)cc12)C1C(C)C1 46884,n1(C(CC)C)ncc2cc(C(=O)NCC3CCN3C(c3ccncc3)=O)cnc12 46885,CC1CCN(C(=O)C(c2ccccc2)O)C1CNC(=O)C(F)(F)c1ccccc1 46886,CCCCCCCC(=O)N1CCCC1C(C)NC(c1c(Br)c(C)nn1C)=O 46887,C1(C(=O)NC23CC(CNC(=O)CCF)(C2)C3)CCC(S(N)(=O)=O)CC1 46888,C1(C(N2C(C)CCC23CC3)=O)CC2CCCC2N1C(C1CC(C)(C)CCO1)=O 46889,C1(NC(CSCCC)=O)CCC2(CC1)CCN(C(c1csc3cncn13)=O)C2 46890,C(C(O)C(F)(F)F)N(C(C(C)N(C(CNC(=O)OCC)=O)C)=O)C 46891,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 46892,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 46893,C1(C(N(CC#C)CC#C)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 46894,N1(C(CCC2CCC(NC(C3CCN(C)CC3)=O)C2)=O)CCCC(F)CC1 46895,C(=O)(C1=NOC(C(C)(C)C)C1)N1C(C(=O)OC(C)C)CCCC1.C1(=O)CO1 46896,N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(=O)CCc2ccsc2)C1 46897,C=C(C)CCCC(c1nnnn1-c1ccc(OC(F)F)cc1)NCCOCCCN 46898,c1(C(N2CCC(NC(c3cn(CC)nc3C)=O)C2C)=O)ncc(F)c(OC)n1 46899,N1(C(C(=O)NCCOCCCC)=O)CCCC(N(C(C2(CC)CCC2)=O)CC)C1 46900,c1(CC)cc(C(=O)N(CC(C)CNC(=O)CC(CC)C2CCC2)C)ccn1 46901,Cn1ncc(C(=O)NC2CCCCC2NC(=O)CCc2nnc(S)n2C)c1Cl 46902,c1(N(CC=C)CCOC)nnc(-c2ccc(Br)cc2)n1CCC 46903,C1(C(=O)NCC2CC(NC(C(C)OCCC=C)=O)C2)CC(c2ccccc2)=NO1 46904,c1(C(=O)NCCOCC(N2C(COC)CC2)=O)cc(C)oc1C 46905,c1(CNCC(N2CC3CN(C(COC)=O)CC23)=O)nsc2ccccc12 46906,N1(C(C(CC)Oc2ccccc2F)=O)CC(OC)C(NC(=O)C=C(C)C(C)C)C1 46907,c1(C(=O)OC)coc(C=CC(=O)N(C2CCC(NC(c3snnc3C)=O)C2)C)c1 46908,C1(CN(C)C(c2cn(CCc3csc(C(C)(C)C)n3)nn2)C)CCCN1CC 46909,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C1C2 46910,c1(CC(=O)N(CCNC(C(C)SCCCC)=O)CCC)ccccc1 46911,C12CCC(CC1)OC2.CC(C)(CNC(=O)NCCOC(F)(F)F)CN 46912,c1(CSC)cn(CC(C)(C)CNC(=O)Cn2ccc(C(F)(F)F)n2)nn1 46913,N1(C(=O)NC2CC2)CCC(CC(=O)NC2CCCN2C(=O)C(F)C2CCOC2)CC1 46914,CCN=c1[nH]cc(C(=O)N(CCCN(C)C(C2CC2[N+](=O)[O-])=O)C)s1 46915,C1(N(C(CCOc2cccc(C)c2)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC12CC2 46916,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 46917,c1(C(N2CC(O)(C(C(=O)NCC34CCC(CO3)C4)F)C2)=O)cccc(CO)c1 46918,C12CCOCCN1C2.c1(C(C)O)nc(Cl)cs1 46919,c1(OCC)ccc(CNC(C23CC(C2)C3)=O)c(F)c1F.N12CCC(CC1)C2 46920,C1(CC=C)(C(N2CC(O)(C(C)NC(=O)COc3cccnc3)C2)=O)CC=CC1 46921,N1(C(C(C)NC(C2CCC2)=O)=O)CCCC(C)(CNC(=O)Cn2nccn2)C1 46922,c1(OC)ccnc(O)c1C(N1CC(NC(=O)Cc2cnsc2)C(C)C1)=O 46923,Cc1cc(C(N2CCN(C(=O)C(C)O)CC2)C(=O)NCC2CCCO2)cc(F)c1 46924,C1(S(C)(=O)=O)(CNC(=NCCSC)NCc2ccc(F)cc2)CCC1 46925,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1 46926,c1(C(N(C2CCN(C(C(CCC)O)=O)C2)CC)=O)cc(OC(F)(F)F)ccc1F 46927,C(=O)(C(C(C)(C)O)NC(C1CC1(C)C(F)F)=O)N1CC(C)C(O)C1 46928,CCC1=C(C(=O)NCC(C)(O)CNC(=O)CN=S(C)(C)=O)SCCO1 46929,C1(C(=O)NC2CC(NC(c3ccc(=O)oc3)=O)C2)CCN(C2CC2)C1=O 46930,n1(CC(=O)NCC(C)CN(C(C23COCC2C3)=O)C2CC2)ccc(C2CC2)n1 46931,c1(C(C(=O)NC(C2CN(C(Cn3nnc(C)n3)=O)C2)CN(C)C)C)cc(C)oc1C 46932,c1(CC(N2CC(O)(C(C)NC(=O)CCc3cnoc3)C2)=O)cncc(F)c1 46933,CCCC(C(=O)N1CC(=O)CC1C(=O)NC(C)(CO)C1CCCC1)OC 46934,c1(C(N2CCC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)noc2ncccc12 46935,c1(C(N(C(C(=O)NCC2(CCC)CC2)C)C)=O)cn(CC)nn1 46936,c1(OC)ccc(C(=O)NC(c2ccccc2)(C)CNC(=O)CCNC(N)=O)cn1 46937,c1(C(C(=O)N(C)CC2CCN(C(CNC(=O)NC)=O)C2)O)ccc(F)cc1 46938,CN1CCC(C)(C(=O)NCC(CC(F)(F)F)NC(=O)C(C)(C)CC2CCC2)C1 46939,Cc1ccc(C(N2CCC(CO)CC2)C(=O)NCc2ccnn2C)c(F)c1F 46940,C12(CNC(=O)Cn3ncc(Br)n3)CC1CN(C(=O)COc1ccccc1)C2 46941,C1(N(C(c2ccon2)=O)OCC=C)CCN(C(c2n[nH]cc2Cl)=O)CC1 46942,C#CC1(C(=O)NCC(C(C)C)OC)CCN(C(=O)CCCN(CC)CC)C1 46943,Cc1ccc(C2CC2)cc1C(N1CCSCC1CCNC(=O)C(F)=CCCF)=O 46944,N1(C(c2ccc(OC(F)F)cc2)=O)CCC(F)(F)C(Sc2ncc3c(n2)CCC3)C1 46945,C=C(C)CC(C(=O)NC1CCCCC1(C)C)NC(c1cncc(O)c1)=O 46946,c1(-c2ccc(Br)cc2)noc(C2c3ccccc3CCC2(C)C)n1 46947,CN1N=C(C(=O)N(CCCC(=O)NC2(c3cccc(F)c3)CC2)C)CCC1=O 46948,N1(C(C(C)Cc2ccccn2)=O)CCC(CF)(NC(=O)CCSCC(N)=O)C1 46949,C1(O)(CNC(C2C(c3n(C)cnc3)C2)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC1 46950,N1(C(C(C)OC(F)(F)F)=O)CC2CCCC(C1)N2C(=O)CC1CCOC1 46951,N1(C(CCOCCNC(c2ccnnc2O)=O)=O)CCc2ccccc21 46952,N1(c2ncnc(OC)c2OC)CCc2cc(C(N3CCS(=O)CC3)=O)ccc2C1 46953,C=C(C)c1ccccc1NC(=O)CC1CN(C(=O)C(C)NC(N)=O)C(C)(C)C1 46954,c1(NC(c2cccn2C)CNCc2cccc(C)c2)ncc(C)c(CO)n1 46955,c1(CC(=O)NCC(CC=C)NC(c2ccc(F)n2C)=O)ccc(OC)c(F)c1F 46956,Cc1c(CC(N2CCC2CNC(=O)C(C)C2CC2)=O)c(O)nc2[nH]nc(O)c12 46957,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C#N)CC3)cc2)=O)C1 46958,N1(C(c2c(C)ncs2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 46959,c1(C(N2C(C)CCC(C(=O)NC(c3nncs3)C)C2)=O)cccc2c1CCC2 46960,C12(C(N3C(C)CC(NC(C(C4CCCCC4)C)=O)C3)=O)CCC(F)(CC1)CC2 46961,CC(C)CC(C)(CNC(c1cccc(O)c1)=O)NC(c1ccn(C2CC2)n1)=O 46962,N1(C(C(c2cccs2)NC(C2CCSCC2)=O)=O)C2CCCC1COC2 46963,CC(C)(C)CC(=O)N1CCC(C(=O)NOCC2(C#N)CC2)CC1 46964,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 46965,c1(N(CCCN(C(c2nc(C)n(C)n2)=O)C)C)nc(Cl)ncc1Cl 46966,Cc1cc(-n2ccnc2)ccc1C(=O)NCCN(C(=O)C(F)C(F)(F)F)C(C)C 46967,C1(OC)CCCCCC1NC(=O)C(=O)NCC(c1ccc(Cl)c(F)c1)=O 46968,c1(C(=O)NCCCNC(=O)Cc2cnoc2)ccccc1SC1CCC1 46969,Cc1cc(=NCC2(CCCO)CCCC2)[nH]c(NC(c2cccnc2)C)n1 46970,CN1CCC(n2cc(C3CCCN3C(=O)CCn3cnc(C(N)=O)n3)nn2)C1=O 46971,CC(CNC(=O)Nc1ncc(C(=O)OC(C)(C)C)s1)(CO)CO 46972,C1(C(N2CCC(N(C(c3ncsc3C)=O)CC)C2)=O)CCCC2CC12 46973,N1(C(C(CC)OC)=O)CCC2(CCN(C(c3occc3C3CC3)=O)C2)C1 46974,c1(OC)ccc(F)c2c1CN(C(C)C(NCC1(C)CCOCC1)=O)CC2 46975,c1(C(=O)NCC2C(NC(CC3(CC)CCC3)=O)C2)cn(C2CCCC2)nn1 46976,c1(OC)cccc(S(=O)CC(=O)NC2(CN(C(=O)CNC(N)=O)C)CC2)c1 46977,C1(C)(CNC(CCC=C=C)=O)CN(C(=O)CC(C(C)C)OCC)C(C)(C)C1 46978,C1(NC(C2C(=C)C2)=O)CCN(C(c2ccc(C3CC3)o2)=O)C1 46979,C1(C)(C(=O)NC(CCCNC(c2n(COC)ncc2)=O)C)CCC(=O)C1 46980,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 46981,C1(NC(C(CCC)OCC)=O)CCCN(C(C2C3CC4C(C3=O)C24)=O)C1C 46982,N1(C(C2CC3CCC2O3)=O)CCOC2(CCN(Cc3nc(C4CC4)no3)C2)C1 46983,CC(C)C(CN(C)C)N=c1nc(N2CCC3(CCN(C)C3)C2)c2c([nH]1)CCS2 46984,Cc1nc(Cl)[nH]c(=NC2CC(NC(C3CC3c3cccnc3)=O)CC2)c1F 46985,Cn1nc(C(N2CCC(NC(c3cc(F)cs3)=O)C23CC3)=O)ccc1=O 46986,CC(CC(C(=O)N1Cc2cncnc2C1)NCCC1(C)CC1)C(C)(C)C 46987,C1(C(N(CCNC(CCCCC(C)C)=O)C2CC2)=O)CCCC2(CCOCC2)O1 46988,C1(OC)CN(C(=O)CC2CC(F)C2)CC1NC(C1(c2ccccc2Br)CC1)=O 46989,c1(CCNC(C2C(C)CNCC2)=O)csc2ccc(O)cc12 46990,Cc1cnc(NC(C2CSCCN2Cc2c(C)cccc2Br)=O)c(Cl)c1 46991,c1(C(=O)OCC)cc2n(n1)CC(C)N(C(c1cc3occc3[nH]1)=O)C2 46992,C(C(CC1CC1)C(=O)N1CCC(O)C1)NC(=O)Cc1ccns1 46993,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 46994,N1(C(CC(=O)OC)=O)CCCC(C(=O)NCC(F)(F)C(C)C)C1 46995,C1(C)(C(N(CCN(C)C(C2(C(=C3CCCCC3)C)CC2)=O)C)=O)CCC(=O)NC1 46996,CCC(C(C)O)NC(=O)CCC1CC(NC(c2cccn2C2CC2)=O)C1 46997,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(F)(F)C(O)C2CC2)CC1C1CC1 46998,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 46999,CS(=O)c1cccc(NC(c2noc(CC3CC3)n2)C(=O)OC)c1 47000,C=CC1(C2(C(N3CCC(CNC(=O)CCC(C)(C)[N+](=O)[O-])C3)=O)CCC2)CCC1 47001,C(c1cccnc1C)=CC(=O)NCC(C(C)C)NC(C(CC)c1ccccc1)=O 47002,CC1CC(NC(c2cncc(O)c2)=O)CCN1C(c1cccnc1Cl)=O 47003,Cc1[nH]c(C#N)cc1C(N1CC(CC(N2CC3(CCC3)C2)=O)C(C)C1)=O 47004,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)NCCC(O)C(C)C)CC1 47005,c1(N(C2C(C)CCNCC2)C(=O)C=Cc2ccoc2)ccc2cnccc2c1 47006,c1(OC)ccc(OCC(N2CC(CNC(=O)CN3CCCC(O)C3)C2)=O)cc1C 47007,C#CCCCCCCC(=O)N1CCN(C(=O)CCC(=O)N(C)C)C2CC12 47008,N1(C(=O)Nc2c(OC(C)(C)C)cc(CN)cc2)CCC2(CC=CCO2)CC1 47009,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47010,N1(C(c2c(C)cn(C)c2)=O)CCC2(NC(=O)C=CCOC(C)(C)C)CCCC12 47011,Cc1nn(C)c(C)c1S(=O)(=O)NC1CCN(C(=O)CC2NC(=O)NC2=O)CC(O)C1 47012,c1(OCC)ccc(CN(C2(SCC(=O)OC)CN(C(=O)CC)C2)CCO)cc1 47013,c1(C(=O)NC2C(NC(c3c(C)cncc3)=O)CCC2)ccc2cn(C)nc2c1 47014,c1(C(=O)NC(c2ccccc2)CNC(C2CNC(=O)C2)=O)cc2cccnn2n1 47015,C1(C(C(=O)O)SCC(=O)NCC(=O)N(C)C)CC2CCC1C2.c1ccccc1 47016,C1(C2(NC(C3CC3F)=O)CC2)CCCN1C(C1COCCO1)=O 47017,CC(C(=O)NC(C(C)(C)C)c1ncc[nH]1)N1C(=O)COc2cc(Br)ccc21 47018,Cn1cnc2c1CCCC2C(=O)NCC1(F)CN(C(=O)CCC2CCOC2)C1 47019,C1(C)(CC(=O)NC2(C#C)CC2)CCN(C(=O)C(F)OC(F)(F)F)C1 47020,Cc1cc(C(F)F)nn1CC(N1CC(NC(=O)Cc2cccs2)CC1C)=O 47021,C=Cc1cnn(C)c1C(N1CCC1CNC(c1cnccc1N(C)C)=O)=O 47022,c1(C(=O)NCC2(O)CCCN(C(CCSC)=O)C2)nc2ccccn2c1F 47023,C1(C(=O)NCc2c(C(=O)OCC)cc[nH]2)CCCN(C2CC(=O)NC2=O)CC1 47024,N1(C(C(CCN(C)C)(C)O)=O)CC2CC(C1)CN(C(=O)CC1CC3(CCC3)C1)C2 47025,C1(NC(=O)C=CC2CCOC2)CC2(C1)CC2C(=O)NC1CCOC1 47026,C(CC(O)CC(=O)NC1CCC(NC(=O)C(C)(C)n2cnnn2)CC1)SC 47027,N1(C(c2c(C)nccc2)=O)CCC(O)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 47028,c1(Cn2cc(CC)nn2)cccc(C(=O)NCCSC2CCOCC2)c1 47029,N1(CC(c2ccc(C)cc2)(C)C)CCCC(C(N2CC(O)C2)=O)CC1 47030,C1(C(=O)NCCc2ncn(C)n2)CC(O)CN1C(=O)CCN1CCCC1 47031,c1(C(C)=O)cc(C(=O)NCC23COC(CNC(=O)CCC4CCOC4)(C2)C3)n(C)c1 47032,N1(C(c2oc(C)c(CO)c2)=O)CC2(NC(C3CC3C(C)(F)F)=O)CCC1CC2 47033,C1(CCC(=O)NCCN(C(C)C)C(C2(c3ccsc3)CC2)=O)CCC(=O)NC1 47034,C1(NC(CCCC#N)=O)CC(F)(F)CC1NC(C1CC1(Cl)Cl)=O 47035,C1(NC(=O)C=CCNC(=O)CC2CC=CCC2)CCC(C2CC2)O1 47036,CCC(N)CCC(=O)N1CCC1(C(=O)OC(C)(C)C)C(C)C 47037,C1(N)CCN(C(c2csnc2NC(CCCNC(=O)CC(F)(F)F)=O)=O)CC1O 47038,c1(C(=O)NCCCN(C)C(c2ccn(C3CC3(F)F)n2)=O)ccc(F)cn1 47039,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2CCC(NC(C3CC(C)(C)C3)=O)C2C1 47040,C1(NC(C(C)NC(=O)NC)=O)CN(C(=O)C(C)CC(C)C)CC1(C)C 47041,c1(OC)ncc(C(=O)NCCC2(NC(=O)C(CC)OC)CCCC2)s1 47042,N1(C(c2ccc(I)cc2)CNC(=O)C(=O)NCC=C)CCC(C)CC1 47043,C1(CC(C)O)CCCCN1C(=O)COCCNC(=O)Cn1ccnn1 47044,CC12CC(C(N3CC(CNC(=O)CC4CCCC(C5CC5)O4)C3)=O)(C1)C(C)(C)O2 47045,N1(CCCNC(C(C)(C)C2CCCCC2)=O)CCN(C(=O)C(O)CC2CC2)CC1 47046,C1(C(=O)NCCN)CN(c2ncccn2)CCN1C.Cc1onc2c1C(=O)NC2 47047,c1(NC(C2CC(NCCCC#C)C2)=O)ccccc1Oc1ccccc1 47048,CCCCC(O)C(C)C(=O)N1CC2CCC(C1)C2NC(C1CCOCC1)=O 47049,c1(C(C(=O)NCCN(C(C(C)C)=O)CCCN(C)C)C)cncnc1 47050,c1(CNC(Cn2cc(CCCC=C)nn2)=O)cc(C)ccc1Cl 47051,C=CCCC(C(=O)NOCCC)NC(C1CC=CCO1)=O 47052,C(=O)(CC(C)(C)C(F)(F)F)N1C2(CN(C(c3nc(CC)oc3)=O)C2)CC1 47053,S(=O)(=O)(C(F)(F)F)NCCC(=O)NC1CSCCN1C(=O)C(Cl)(Cl)Cl 47054,N1(C(Cc2c(C)nn(C)c2)=O)CCC(C)C(CC(N2CCC(C3CC3)CC2)=O)C1 47055,N1(C(C(COC)O)=O)CC2CC(C(=O)NCC(=O)NCCOC)C(C2)C1 47056,N1(C(C(C2CCN(C(c3c(C)nc(Br)cc3)=O)CC2)C)=O)CCC(=O)N(C)CC1 47057,C12(C(N3CC(C(N)=O)(CNC(=O)Cc4nccn4C)C3)=O)CC(CF)(CO1)C2 47058,N1(C(c2cc(SC)ncn2)=O)CC(CNc2cncc(C(F)(F)F)c2)CC(C)C1 47059,C1(OC)CCCN(C(c2cc(CNC(C3CC3C3CCC3)=O)on2)=O)C1C 47060,C(CNC(=O)CCCc1cnn[nH]1)(CC(=O)NC(C)C)OC 47061,C1(NC(c2c(CC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47062,Cc1sc(C)c(S(=O)(=O)NC2CC(C)CCC2C(C)C)c1Br 47063,N1(C(=O)CCCNC(=O)NCCCc2ccccc2)CCC(CO)(CO)C1 47064,Cc1cc(C(N2C3CCC2CN(C(=O)CC(F)(F)Cl)CC3)=O)nc2ccccc12 47065,N1(CCC)C(=O)CCC1CC(=O)OCC1(C)CC1(C)C 47066,C(CNC(c1cccnc1)=O)(C(C)C(C)C)NC(c1c(C)nn(CC(F)F)c1)=O 47067,C(=O)(C(CSC)NC(=O)CN(C)C)NC(CCSCC)C 47068,c1(C(N2CCC(CNC(c3cc4n(c3)CCSC4)=O)C2)=O)ccc2cncn2c1 47069,C(C)(C(O)C(=O)NCC1CCC(NC(c2n[nH]cc2Br)=O)CC1)OC 47070,N1(C(c2c(C)[nH]nc2Cl)=O)CC(C2(NC(=O)C(F)C(C)(C)O)CC2)C1 47071,CCCCC(O)C(=O)N1CC2C(C(=O)NCCCn3cccc3)C2C1 47072,C1(c2ccccc2)(C(N(C)CCNC(C2CC(Cl)(Cl)C2)=O)=O)CC(O)C1 47073,c1(C(=O)NC2CC(C)(CNC(c3sc(C)c(O)n3)=O)C2)c(O)cccc1Cl 47074,c1(NCC(C2CC2)NC(c2ccncc2F)=O)ncc2scc(Br)c2n1 47075,N1(Cc2nc(-c3ccc(OC)cc3)sc2)CC2C3C=CC(CC3)C2C1 47076,N1(C(C=C(CC)CC)=O)CCCOC(CNC(C2CCCN2C2CCCC2)=O)C1 47077,C1(C(=O)NCC2(F)CC(NC(C(C)OCCC=C)=O)C2)CCCC(=O)N1C 47078,N1(C(C2(CO)CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CC2COCC(C2)C1 47079,O(C1CCSc2ccccc21)C(C1C(N)CCCC1)=O 47080,c12ccnc(n1)N(C)C2=O.C1(COC)CCCCN1C(=O)Cc1ccc(Cl)cn1 47081,S(=O)(=O)(CC(=O)NC(C1CN(C(=O)CSCCc2ccccc2)CC1C)=O)NCC 47082,C(CCCCCC(=O)N(CCCCCO)C)n1cc(CC)nn1 47083,C1(NC(CCNC(C)=O)=O)(CO)CCCN(CCC(C)C)C1 47084,C1(C(N(C2CN(C(C3CCC(=O)O3)=O)CC2(C)C)C)=O)COC(C)(C)CO1 47085,C1(NC(C2CC2(F)F)=O)CCCN(C(c2cnn(-c3ccccc3)c2)=O)C1 47086,Cc1cc(-c2nn[nH]n2)cnc1COCC(=O)NC(c1ccccc1O)C 47087,N1(C(C=O)=O)CCC2(C(F)(F)F)CC2C1.c1(C(N(C)CC2CC2)=O)ccnn1C1CC1 47088,N1(C(Cn2ncc(CC)c2)=O)CC(O)CCC1C(=O)Nc1ccc(F)c(CO)c1 47089,c1(C(N2C(CNC(CCN(C(CCC)C)C)=O)CCC2)=O)ccc2nonc2c1 47090,CC(C(O)C(F)F)NC(=O)C(c1cnn(C)c1)NC(=O)CC(C)(F)F 47091,CC(C)C(O)CNC(C1CCC1CNC(c1cc(CO)[nH]n1)=O)=O 47092,C(=O)(CC(O)C(C)C)NC1(COC)CCN(C(c2ccccc2NC(C)C)=O)C1 47093,N1(C(C(C=C)(C)C)=O)C2CCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)CC2 47094,C1(NC(C(CSC)C)=O)COC2(CNC(c3ccc(F)cc3N)=O)CC1C2 47095,N1(C(C2CCCO2)=O)CCCC2C1CCCCN2C(=O)COc1cccnc1 47096,N1(C2CCCN(C(CC(=C)C)=O)C2)CCN(c2ccnc(N3CCC3)n2)CC1=O 47097,C1(C(=O)NCC2(F)CC(NC(c3cc(C(=O)OC)sn3)=O)C2)CCS(=O)(=O)C1 47098,C1(NC(CCc2cn(C)nc2)=O)CN(C(=O)CSc2nncn2C(C)(C)C)CC1O 47099,C1(C(N2CCCC(N(C)C)CC2)=O)CCN(C(=O)CC2COC(=O)N2)O1 47100,c1(OCCN2CC3(C(C(=O)Nc4ncon4)C3)C2)cccc(Br)c1Br 47101,N1(C(C(C)(C)F)=O)CCC2(NC(=O)CSC3CCCC3)CCCCCC12 47102,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47103,N1(C(c2occ(C)c2C)=O)CCC2(NC(C3CCN3C3CCCC3)=O)CCCC12 47104,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47105,C1(CC)(N)CCN(C(=O)C(C)CC(=O)NCC2(CC)CCOC2)CC1 47106,C(=O)(CCC(C)C#N)N(C(CCNC(c1c(C)nc(Cl)s1)=O)C)C 47107,Cc1conc1C1CN(C(C2(CO)CCOC2)=O)C1.C1(C(=O)N)C2CCCC12 47108,C#CCCCC(C)C(=O)N1CCC(CCNC(C2(C#N)CCC2)=O)C1 47109,C1(C)(CCNC(c2cc(COC)sc2)=O)CCN(C(c2cnn[nH]2)=O)C1 47110,C(CCCCC(=O)NC1(C)CCCC1C)NC(CN(c1cn[nH]c1)C)=O 47111,C1(OC)CC(C)(C)CCC1NC(c1cc(C2CC2)cs1)C(=O)OC 47112,C12(CNC(CC3N(C)CC=CC3)=O)CCC1CCN2C(=O)CC1=CCCC1 47113,c1(OCC(=O)NC2CCN(C(C3CCC(F)CC3)=O)CC2O)ccccc1[N+](=O)[O-] 47114,c1(CC)ncoc1C(=O)N(CCCC(=O)NCC(c1ccccc1)F)C 47115,c1(C(N2CC(C)N(C(C3CCCCC3C3CC3)=O)CC2)=O)cc(=O)n2ccsc2n1 47116,C12(c3ccon3)CCN(CC1)C(CCCC#N)C(=O)N2.C1(C)(CC)CC1 47117,C(=O)(CS(=O)(=O)CCCC)N(CCNC(C1(n2cccn2)CCC1)=O)CC 47118,C1(CNC(C(c2cncnc2)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C1 47119,C1(NC(C2CCCC3(CCC3)O2)=O)Cc2ccccc2N(C(c2ccno2)=O)C1 47120,N1(C(=O)CC2CCOC2)CCN(CCNC(C2CC3CC3C2)=O)C2(CCC2)C1 47121,C(=O)(CCCC(F)(F)F)N1CC(C(=O)NCCCOCC2CCC2)CC(C)C1 47122,C(CCC(C)C)(C(=O)N(C)CCc1cccnc1)NC(C1CC=C(C)CC1)=O 47123,C1(C(N2CC(SC)C(CO)C2)=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 47124,C1(CNC(CCC(=O)NC)=O)CCN(C(=O)CCSc2nnnn2C)C12CCC2 47125,c1(CNCC=C2CCN(C(c3nnnn3C3CCC3)C)CC2)n[nH]c2c1CCOC2 47126,c1(OC)cc(C=CC(=O)N(C2CCN(C(=O)C(C3CC3)N(C)C)C2)CCO)sn1 47127,C1(CN(C(C(=O)N(C2CC3CCC(C2)N3)CC)C)C(C)=O)CC12CCCCC2 47128,N(C1CCc2cccnc21)C(C(c1ccoc1)C(=O)NCC1CN2CCC1C2)=O 47129,C1(NC(COCC(C)C)=O)CCC(NC(c2scnc2C2CCC2)=O)C1 47130,c1(OC)cccc2c(C3(c4c(C(=O)OC)ccc(F)c4)CC3)cccc12 47131,C1(NC(CC2(NC(C)=O)CC2)=O)CCSC12CN(C(=O)CC1CCCCC1F)C2 47132,C(=O)(C(C)CC(C)C)N(CCCC(=O)N(CCC)CCC)C 47133,c1(C(c2n(CCCOC)nnn2)NCCN=S(C)(C)=O)ncc(Br)cc1N 47134,c1(CC)nsc(CNC(=O)C(C2CCN(C(C3CCSCC3)=O)C2)C)n1 47135,C=CC(C)(O)C(=O)N1CCC(O)(CCNC(=O)CC(c2ccccc2)C2CC2)C1 47136,C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(NC(=O)CCc2ccccn2)CCCC1 47137,N1(C(C2(C)CC2(F)Cl)=O)CCC2(CCCC2NC(c2cnc(O)nc2O)=O)CC1 47138,C=C(C)C1OCCC1C(=O)NC1CC(CCNC(C2CCC(=O)N2C(C)C)=O)C1 47139,C(CCC(C)CC(=O)NC1CCC(NC(=O)CCc2nc[nH]n2)C1)=C(C)C 47140,c1(CC(C)C(=O)N2CCC(CN(C(=O)CC(=O)C3CC3)C)C2)cccc(Cl)c1 47141,CC1CN(C(C2CCC(CNC(=O)Cc3ccn(C)n3)CC2)=O)C(C)CO1 47142,N1(C(CCC2(NC(C3(CC=C)CCOC3)=O)CCCC2)=O)CC2(CCC(=O)O2)C1 47143,C#CCCCC(C)C(=O)N1CCC(C)(CNC(c2c(F)ccc(OC)c2F)=O)C1 47144,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47145,c1(CN(C)C)ccc(C(=O)NCC2CCCCN2C(C2CC3CCC2O3)=O)cc1 47146,c1(OC)ccc(C(N2CC(NC(=O)C(=O)NC(C)C)C2)=O)c2ccoc12 47147,N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(=O)CN2CCN(C)CC2)CCC1C 47148,C12(NC(C=C(CCN(C)C)Cl)=O)CCN(C(c3cc(Cl)n(C)n3)=O)CC1C2 47149,Cc1c(C(=O)NC2(CNC(c3cnn(CC(F)(F)F)c3)=O)CCC2)cnn1C 47150,C(=O)(Nn1cccn1)c1c(=N)[nH][nH]c1.c1(SC2CCC2)ccccc1F 47151,C(=O)(C(C#N)C(C)C)NCCNC(C(c1c(C)ccnc1)(C)C)=O 47152,c1(NC(C2N(C(c3ccc(Cl)cc3)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47153,Cc1ccc2c(C(N3CCCC(C)(NC(=O)CC(O)C(C)(C)C)C3)=O)c[nH]c2c1 47154,c1(C(=O)NC(C2(CNC(=O)COc3ccccc3)CC2)C)c(Br)cnn1C 47155,N1(C(CSCC=C)=O)CCCCC12CC(NC(c1ncsc1C(C)C)=O)C2 47156,N1(C(C2ON=C(C)C2)=O)CCC(NC(c2ccc(C(C)C)nc2)=O)C12CC2 47157,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47158,N1(c2n(C)c(C3CCC(=O)N3)nn2)CCC2(CCCCO2)C1 47159,N1(C(c2c(N(C)C)ccnc2)=O)CC(NC(=O)CCCN=[N+]=[N-])C(N=[N+]=[N-])C1 47160,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47161,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47162,Cc1cc(=O)cc(-c2cn(CCC3CN(C(C4OCCC4C)=O)C3)nn2)[nH]1 47163,C1(NC(CCC(CC)C)=O)CC(O)(C2CCN(C(=O)Cn3nnc(C)n3)CC2)C1 47164,N1(C(c2nc(C)sc2)=O)CC2(CNC(C3CN4CCN3CC4)=O)CCC1C2 47165,n1(CC(=O)Nc2c(C#C)cccc2)ccc(=NC(=O)c2cc(CC)no2)nc1O 47166,c1(C(N(C2CCN(C(c3cc(C(N)=O)ccc3O)=O)C2)C)=O)cn2c(n1)CCC2 47167,C1(C(N2CCC(OCCNC(C(C=C)O)=O)CC2)=O)CCCC2CC(O)CCC12 47168,N1(C(C(CC#C)(C)C)=O)C2CCC1C1CC1(NC(C1CCC(=O)N1C)=O)C2 47169,c1(CC(=O)NC23CN(C(C(C)O)=O)C(C2)C3)cc(F)ccc1F 47170,c1(SCC)nc(Br)c(NCc2ccc(Cn3cc(Br)cn3)o2)n2ccnc12 47171,C1(C(=O)NC(Cc2ccco2)CO)(NC(Cc2c(C)ccs2)=O)CCCCC1 47172,C1(NC(=O)C=CC=Cc2ccoc2)CCC12CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 47173,N1(C(CC(=O)NCC)=O)CC2(CCCC2)C1C(=O)NC(c1ncc(C)s1)C 47174,C1(c2cn(CC(=O)NCC)nn2)CCCCN1C(=O)CSC1CCCO1 47175,S(=O)(=O)(c1cc(C)cnc1NCC(O)CF)NC(CCCC(=C)C)C 47176,C(=O)(CN=c1cc[nH]cc1)NC(C(=O)N(CC(CCC)C)C)CC1CC1 47177,C1(N(C(=O)CC2COCCO2)C)CN(C(c2cc(Br)cn2C)=O)CC1F 47178,C(C)(C)(CC(=O)NCCC(N1CCC(CO)(CO)C1)=O)OC 47179,C1(C(N(C)CCN2CCN(C(c3cnn[nH]3)=O)CC2)=O)CC12CCCCC2 47180,c1(C(=O)NCCC2CCN(C(c3c(CC)nns3)=O)C2)cc(OC)cnc1O 47181,c1(CN(C(=O)CC2CCCN2C(C2(C)CCN(C(C)C)C2)=O)C)cn(C)nc1O 47182,c1(C(=O)NC(CNC(c2nc(CC)[nH]n2)=O)C(C)C)cnn2ccnc(N)c12 47183,N1(C(C2CCC(C)(C)O2)=O)CC2=C(C1)CN(C(c1ccc(F)c(Cl)c1F)=O)C2 47184,C1(C(=O)OCc2cc(C#N)[nH]c2)CC2(CCC(F)(F)CC2)CO1 47185,C(=O)(C#CC1CCCOC1)N1CC2CCC(NC(c3cc(C)nnc3O)=O)C2C1 47186,c1(C(=O)NCC2CN(C(Cn3ccc(C)c3)=O)CC2C)c[nH]c2ccc(F)cc12 47187,C#CCC(C)(C(=O)NCC(=O)NOC)NC(C1CCC(CC)C1)=O 47188,C1(NC(C=C(COC)C)=O)CC2(C1)CC(NC(=O)CCC1CCOC1)C2 47189,CC1CCc2[nH]nc(C(N3CCN(CCNC(c4cnn(C)c4)=O)CC3)=O)c2C1 47190,C(=O)(C1CCCn2cnnc21)NCC1CN(C(C(CC=C)C)=O)C(C)CC1 47191,c1(CCC(=O)NC2CC(NC(C(C)CN3CCOCC3)=O)C2)ccc(O)nn1 47192,Cc1ccc(N)c(C(N2CC(C)CCC2CNC(c2cc(C)c(C)s2)=O)=O)c1 47193,C(=O)(C(C)(C)C1=CCSCC1)N1CCC(C)C(N(C)C(C2CC(F)C2)=O)C1 47194,c1(N2c3ccc([nH]3)CCC2=O)cccc(Br)c1Cl.N(CCCOC)CC 47195,C1(CC=CNC(C=CCC)=O)CN(C)CCN1C(C1CCCN1C1CCC1)=O 47196,N12CCc3c(cccc3C1)OC(=O)C2=O.c1(CN(C)CC#N)ccccc1 47197,c1(CC(=O)N(C2CN(C(=O)Cc3cn[nH]c3)C2)C)ccc(S(N)(=O)=O)s1 47198,c1(C(C)NC(C=CCCC)=O)cnn(C)c1.C1(C2CCCO2)C(=O)N1CC 47199,CCC(F)(C(=O)OC)C(=O)N1CCOC(C(C)NC(=O)Cc2cnoc2)C1 47200,CC(N=[N+]=[N-])C(=O)NC(CC1CCC1)C(N1CCCCC1CF)=O 47201,S(=O)(=O)(CCCCCl)NCc1c(C)n[nH]c1.C12CCCC1N2 47202,c1(SC)cn(C)nc1C(=O)NC1CCCCC1CNC(C12CCCN1CC2)=O 47203,c1(CCCC)ccc(C(=O)N(CCC)CCNC(=O)C(C2CCOCC2)C)s1 47204,C1(NC(C2(C#N)CCC2)=O)CCN(C(c2ccc(F)s2)=O)C(C2CC2)C1 47205,c1(C(=O)NC(CNC(CC(CC)C(C)C)=O)C)c(O)cnc2ccc(F)cc12 47206,CC(C)(O)C(F)(F)C(=O)NC1CCCC(NC(c2sc3cnccc3c2O)=O)C1 47207,N1(C(C(C)CSC(F)(F)F)=O)CCC(CF)(NC(=O)C(=O)NCC(F)F)C1 47208,c1(C(CCC=C)=O)ccc(CC(=O)NCC)c(F)c1.C1(C)C(=O)NCC2(CC2)O1 47209,N1(C(CC2(OC)CCC2)=O)C(CC(=O)N(C)C2CC2)CCC1C1CCCC1 47210,C(=O)(CC(=O)NCC)N.c1(CCC(N2CC=CC2CF)=O)n[nH]cc1OC 47211,C(=O)(C(CO)C(C)(C)C)NCC1COCCN(C(C2CCCN(C(C)C)C2)=O)C1 47212,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NCC(F)(F)F 47213,Cc1ccc(NC(C2CCCCN(C(=O)NC3(n4cccn4)CC3)C2)=O)cc1Cl 47214,C1(C)(C(N(C(c2ccccc2)CNC(c2cnsc2)=O)C)=O)CC(=O)N(C)C1 47215,C1(C(=O)NCCN(C(=O)C(O)Cn2cncn2)C)CCCN1S(C)(=O)=O 47216,N1(Cc2cn(-c3cc(C)c(O)cc3)nn2)CCCCS(=O)(=O)C1CO 47217,C1(NC(Cc2c(OC)cccc2)=O)CCCCCN(C(C2CC2C(C)C)=O)C1 47218,C1(C(=O)NC(c2cn(C)nc2)C(F)F)CN(C(c2ccnnc2O)=O)C(C)(C)C1 47219,CC1CCCC=C1C(=O)NCCCN(C(c1scc(CC)c1)=O)C1CC1 47220,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47221,c1(CN2CCC(C(C(=O)NC(CCC)C(=O)OC)(C)C)C2)cc(O)ccc1C 47222,CCC(C(=O)N1CCC(C(=O)NCC(CC2CC2)OC)C1C(C)C)C(C)C 47223,N1(C(CS(CC)=O)=O)CCC2(OC)CCN(C(C3CC4(C3)CC(O)C4)=O)CC2C1 47224,C(C(C)(C(=O)NCc1cccc(Cl)c1)NC(c1ccc(F)cc1)=O)SC 47225,C1(N(C(CN(C)C(=O)C2CC2)=O)C)CN(C(=O)CC(C)(C)O)CCC1O 47226,CC(C)(O)CCC(=O)NCCCN1CCN(CC2CC2)CC1 47227,c1(C(=O)NCC2CN(C(CC3CCCC(C)C3)=O)C2)n[nH]c2ccccc12 47228,C(CCN(C)C(C12CCCC1C2(F)F)=O)(C(C)(C)C)NC(c1c(C)csc1)=O 47229,c1(C(=O)NCCNC(C2CCOC(C3CC3)C2)=O)ccc2c(c1)C(=O)CCCC2 47230,c1(C(=O)N(C2CCC(C(=O)O)C2)C2CC2)cn(C(F)F)c2c1CCCC2 47231,C1(C(=O)NC(C#C)CCC)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47232,C(=O)(CCCCCCCC(=O)NCCNC(c1ccc2cn(C)nc2c1)=O)OC 47233,C(CN=c1[nH]cc(CC)cc1C)N(C(C1C(CCC)CCC1)=O)C 47234,C1(NC(c2nc(C)n(C)c2)=O)CC12CCN(C(=O)C=CC1CCCC1)C2 47235,C(C1=NOC2CN(C(c3ocnc3CCC)=O)CC12)NC(CCCC(=C)C)=O 47236,C(=O)(CC(C)(O)C1CC1)NCCNC(C(c1ccccc1F)(C)OC)=O 47237,Cc1[nH]c(CCCCCCl)c(C)c1C(=O)NCc1ncccc1Nc1cnc[nH]1 47238,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cn(C(C)(C)C)nc2C)=O)C1 47239,c1(C(=O)NCC(CNC(C=CS(C)=O)=O)(C)O)c(N)cccc1[N+](=O)[O-] 47240,N1(C(CC(C)CN(C)C)=O)CCCCC(N(C)C(c2cn3ccnc3s2)=O)C1 47241,c1(NCCN(C(C(CC)C)=O)CCO)cccc(-c2ccco2)n1 47242,n1(CC2CCCN2NC(C2CC(CF)C2)=O)cc(C2(C3CC3)CC2)nn1 47243,C1(C(=O)NC(C2CCCC2)CNC(C2(CCCC)CC2)=O)CC12CCCCCC2 47244,c1(NC(=O)COC2CCN(C(C3CCC3(F)F)=O)C2)cncc(SC2CC2)n1 47245,C(=O)(C(C)(F)C(=O)NCC(C1CCCCC1)NC(c1cc(C)n(C(F)F)n1)=O)OC 47246,Cc1ccc(C(=O)NC2CC2NC(c2cccc(F)c2O)=O)c(C)n1 47247,C(=O)(CC1=CCOCC1)NCc1cc(C(=O)NCC(C(C)O)O)no1 47248,CCC(C)C(CC(=O)Nc1cc(C)cnc1OC)NC(=O)CCN(C)CC 47249,Cc1nc(O)sc1C(N1C(C(=O)NCCC(C)N(C)C)CC1C)=O 47250,n1(CC)cc(Cl)c(C(N2CCC(O)(CN(C)C(C3(C)CSC3)=O)C2)=O)n1 47251,c1(C(N2C(CNC(CC3(OC)CCOCC3)=O)CCC2)=O)cnc2[nH]nnc2c1 47252,c1(C(=O)NCC=CCNC(C(CC)(C)C#N)=O)nc2ccc(Br)cn2c1F 47253,C1(NC(C(CC=CC)NC(=O)Cc2ccccc2)=O)CC2C(C1)C2(C)C 47254,C12(NCC3(C)CCC3)CCCCC(CNC1)C2(F)F 47255,c1(NC(C)=O)ccc(Cl)c(NC(=O)NCC2CCCOC2(C)C)c1 47256,CCCC(C(=O)N1CC2CC1C2C(=O)NC(C)CCSC)OC 47257,C1(C(=O)NCCCCNC(C(CC=CC)CC)=O)OCCOC12CCC2 47258,N1(C(C2(CC#C)CCN(C(c3cnc(C)cn3)=O)C2)=O)CCC2(CCO2)C1 47259,C1(CC(=O)NC2CCC(CNC(Cc3nc(C)sc3C)=O)C2)CCCN(C)C1=O 47260,c1(C(N(C2CN(C(=O)COCCCF)CC2F)C)=O)cccc(Cl)c1F 47261,c1(C(=O)OCC)cncc(C2CCCN2C(c2[nH]nnc2C2CC2)=O)n1 47262,C1(NC(C=CCN(C)CC)=O)CCN(C(C2CCCCN2C(C2CCC2)=O)=O)CC1 47263,c1(C(N2CC3C(NC(C4CN(CC)C(=O)C4)=O)C3C2)=O)ccc(=N)[nH]c1Cl 47264,C1(NC(c2c(C)c[nH]c2)=O)CCCC2CN(C(c3nc4c([nH]3)CCCC4)=O)CC12 47265,N1(C(CCCC#C)=O)CCC2(NC(c3n[nH]cc3COC)=O)CCCCCC12 47266,c1(C(=O)NC(c2cccnc2)C(=O)N(CC#C)C)cc(C)sn1 47267,N1(C(c2nc(CCCC)sc2)=O)CCC(NC(=O)C(O)C2CCCC2)C(C)C1 47268,c1(CC)ncc(C(=O)NC(C)CC2CCN(NC(C)=O)CC2)c(C)n1 47269,CC1CCC(NC(=O)NCS(N)(=O)=O)CN1CCOCCO 47270,c12cc(Cl)ncc1C(=O)N2.C1(C2OCCO2)(NC(=O)NC2CC2)CCCCC1 47271,C1(CC)CN(C(c2scc(C)c2Cl)=O)CCC1NC(=O)CCc1cccnc1Cl 47272,Cc1cnc(CN(C)C(C2C3CN(C(=O)CCCC4CC4C)CC23)=O)cn1 47273,c1(C(N(C2CC(NC(C(C)=C3CC3)=O)C2)C)=O)c[nH]cc1-c1cnn(C)c1 47274,N1(C(C2C(C)OCCC2)=O)CCC(NC(c2cc[nH]n2)=O)C(C)(C)C1 47275,CC1(C)CC(NC(C23CSC(C2)C3)=O)CN1C(C1CN(c2ccccc2)CCO1)=O 47276,C1(C2CC2)(NC(c2cc(C)c(F)cc2)=O)CCN(C(=O)C2=CS(=O)CCC2)C1 47277,N1(C(C2C(NC(C(C(C)C)C3CCC3)=O)COC2)=O)CC(N(C)C)C2(CC2)C1 47278,Cn1nc2c(c1C(=O)NC1CN(C(C3(C)CS(=O)(=O)C3)=O)CC1C1CC1)CCC2 47279,C12(CC(=O)NC3CN(C(c4nnn(CC)c4C)=O)C3)CCC(CC1)CC2 47280,CON1CCC(C(=O)NC2CCC(CC(=O)NC(C3CCOCC3)C)C2)CC1 47281,C(=O)(C(C)(C)C(=O)NCCOC(C)(C)CNC(=O)C(c1ccccn1)O)NC 47282,c1(C(C)NC(=O)C(N2CCN(C(=O)CS(N)(=O)=O)CC2)=O)nc2ccccc2s1 47283,N1(C(C(=O)NCCCCCC)CCCSC)CCc2nnc(Cl)cc2C1 47284,C1(CC(=O)NC(c2cccnc2O)C)CCCC(NC(=O)C(C2CCOCC2)F)C1 47285,C1(CC(=O)N(CC(C)NC=O)C)CC=CCN1C.N1(CC=O)CCCC1=O 47286,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC(O)C3)=O)CCC2C1 47287,c1(COC)cccc(C(=O)NC(C2CCN(C(C3(C)CCC(C)C3)=O)CC2)C)c1 47288,c1(C(N(C2CCS(=O)(=O)C2)CCC)=O)ccc(Br)cc1Cl.C(=O)(C(C)C)NCC 47289,N1(C(C2(N(C)C(C3(C#N)CCCC3)=O)CC2)=O)CC2CC(C)C2C1 47290,c1(C(=O)NC2C3CN(C(C(C(=O)OC)C)=O)C2CC3)cc2c(F)cccc2[nH]1 47291,C1(OC)(CNC(=O)Cc2ccc(F)cc2F)CCN(C(=O)CSSC)CC1 47292,CC(CN(C)C)C(=O)N(C)CCOCCNC(C1CCC(C)O1)=O 47293,C(=O)(CC(C(C)(C)C)NC(=O)Cc1ccc(O)cc1)NC(CCC)C(F)(F)F 47294,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOC(c2ccccc2)C)C1 47295,CC#CCC(C(=O)NCc1ccccc1)NC(=O)CCCOC 47296,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47297,N1(C(C2OCCN(C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC(CO)C1 47298,N1(C(COCCC)=O)CCC2CC2(C(=O)NCCC2CCN(C)C2)CC1 47299,CN1CC=C(CCNC(=O)C(C2CCCO2)NC(=O)Cn2cccn2)CC1 47300,c1(NC(CCNC(CCC)=O)=O)ccc2c(c1)OCCO2 47301,C1(C)(C(=O)NCC2CN(C(CNC(C)=O)=O)C2)CCCO1 47302,C1(O)(C(=O)NC2COCCN(C(c3cnc(C)s3)=O)C2)CCCC(C)CC1 47303,N1(C(CN(C(c2cc(CC)on2)=O)CC)=O)CCCC2(CC2)C1.CCS 47304,CC1CCCN(C(=O)C(N2CC(NC(C3CC(CN(C)C)C3)=O)C(C)C2)=O)C1 47305,C1(CNC(Cc2c(C)ncs2)=O)CCCN(C(C2CCC(C(C)C)CC2)=O)C1 47306,c1(C(N(C2CN(C(=O)CC3CCC3(C)C)C2)C)=O)ccc(N)cn1 47307,c1(C2CC(C(N3CCC(N(C)C(C4(C)CC4(C)C)=O)CC3)=O)C2)ccc(Cl)cc1 47308,C1(CC#C)(C(=O)NCCC2(O)CN(C(=O)Cc3cncc(O)c3)C2)CC=CCC1 47309,C1(NC(CN(CC(CCNS(CC)(=O)=O)O)C)=O)CCCC(F)(F)C1 47310,C1(C)(C(N(C)CC2(NC(C3C4CCC(=O)C34)=O)CC2)=O)CCC2(CC1)OCCO2 47311,c1(NC(C2(CC)CCCN2C(=O)CC2(C)CC2)=O)ccc2ccoc2c1 47312,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47313,S(=O)(=O)(c1cccnc1NCC1(CSC)CC1)N(CCC(N)=O)C 47314,C1(C(=O)NCC(CC)NC(=O)Cc2sc(=N)[nH]c2C)CC2C=CCC(C1)C2 47315,c1(C(n2cc(CS(C)(=O)=O)nn2)C(C)C)cccc(C(=O)NCc2ccsn2)c1 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47385,CC1CCCCC1C(=O)Nc1ccsc1CNC(=O)CSc1nncn1C1CC1 47386,C1(C2CCC2)(C(=O)NCC(C)(C)OCCNC(C2CCC(F)(F)C2)=O)CCC1 47387,C(C(C)(C)CO)N(C(=O)C(O)C1CN(C(=O)CCN(C)C)C1)C 47388,c1(C(=O)NCC=CCNC(=O)CC23CCCC2C3)cc2cccnc2o1 47389,C1(NC(C2(CC)CC2)=O)CC=C(C(=O)NC2CC3C(C2)C3(F)F)C1 47390,CC1CCc2[nH]nc(C(=O)NC3CN(C(c4coc(C(F)F)n4)=O)CCC3C)c2C1 47391,C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cnsn3)=O)C2)C1 47392,Cn1cc(Cl)c(CC(=O)NCC2CC(F)CN2C(=O)C(F)CC2CCCCC2)n1 47393,N1(C(C2C(C(C)(F)F)C2)=O)CCC2CN(C(c3ccc(Br)cc3)=O)CC12 47394,CCC(C)(C(=O)Nc1cccnc1OC1CCOC1)C(F)F 47395,N1(CC)CCCCC1C(N1CC(F)(C(=O)NCCOC(C)COC)C1)=O 47396,c1(C(C)=O)ncccc1C(=O)NCCC(O)CNC(=O)CCc1nncs1 47397,c1(C(=O)NC2CC(NC(C=CCOC)=O)C2)cc2c(nc1O)CCSC2 47398,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3conc3C)=O)C2)C1 47399,C1CCC(C2CC2)NC(=O)C(CO)NC(=O)NC(C)C(=O)N1.C1(OCC)CCC1 47400,c1(CC)nc(Cl)c(F)c(=NC(CNC(C2(CO)CC2)=O)(CC)CC)[nH]1 47401,c1(OC)ccc(C(=O)NCC2(C3CCCO3)CCC2)c(Cl)n1.C12(CCC1)C(=O)N2 47402,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1O)=O)C2 47403,c1(C(=O)NCC(CCNC(c2c(C)cccc2O)=O)O)ccc2nnc(O)n2c1 47404,C#Cc1nccnc1NC(C1(C)CCN1C(c1cnc(Cl)c(I)c1)=O)=O 47405,C(=O)(C(O)C(F)(F)F)N1C(C(N2CCC(C(C)C)C2)=O)C(C)C1 47406,CC(C)CC(C(N)=O)NC(c1n[nH]c2c1CCC2)=O 47407,CC1CN2CCN1C(C(=O)NCCCCNC(=O)CCCN1CCCC1)C2 47408,c1(OC)ccc2c(c1)CCN(C(=O)CC1CCCCC1OC(c1nonc1N)=O)C2 47409,CCC(C)(O)C(=O)N1CCN(CC(C)(C)NC(=O)C=CC2CCOC2)CC1 47410,CC1CC(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)Cc2ccn(C)n2)C1 47411,C(=O)(C#CC1CC1)NC1CCN(C(CCN(C)CCO)=O)C1 47412,N1(C(CC2N(C)CCCC2)=O)CCN(C(C2CC2c2cc[nH]n2)=O)C(CO)C1 47413,C(C(C)N=c1[nH]c(=N)[nH]c(=NCCc2cnn(C)c2C)[nH]1)(c1ccccc1)OC 47414,c1(C(N2CC(C)C(CNC(C3CC34CC(O)C4)=O)C2)=O)ccc(F)c2c1OCC2 47415,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47416,N1(C(C(CSC)C)=O)CCC2(CCCN2Cc2cncc(N(C)C)c2)CC1 47417,C1(NC(c2cnc(CC)s2)=O)CC(CNC(c2cn(C)nc2C(C)C)=O)C1(C)C 47418,C1(C(=O)NCC=CCNC(c2cc(C)on2)=O)CCn2nccc2C1 47419,Cn1ccc2cc(C(=O)NC3(CCNC(C4CC(F)(CO)C4)=O)CCC3)cnc12 47420,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47421,N1(C(CCCCC#C)=O)CC2(CC(NC(c3c(OC)ccnc3F)=O)CO2)C1 47422,c1(C(=O)NCC(C)(C)NC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47423,c1(OC)ccc(C(N2CCCC2C(C)(C)NC(=O)CC2CCCC2C)=O)cc1 47424,C1(NC(C(CSC)OC)=O)CN(C(=O)COc2cc(C)on2)C(C)(C)C1 47425,C1(C)(C(N2CC(C(C)(C)O)(CNC(C(C)OCCC=C)=O)C2)=O)CC2CC2C1 47426,C12(C(=O)NCC3(F)CC(CNC(C=C(C)c4ccco4)=O)C3)CCCC1C2(F)F 47427,CC1(C(=O)NC2CC(O)C2CC(=O)NCc2cnc(C(F)F)s2)CCCOC1 47428,c1(OCC)cc(CNCC(c2cc(C3CC3)n[nH]2)=O)c2ccccc2n1 47429,C1(C(=O)Nc2ccc(OC)cc2)CCN(Cc2cn(C(C)O)cn2)S1(=O)=O 47430,C1(c2n(CCC)nnn2)(NC(CC)C2CCC2)CCCN2CCCCC12 47431,c1(C(N2C(C)CC(NC(c3nn[nH]c3Cl)=O)C2)=O)nccc2ncccc12 47432,c1(C(=O)NC(C(=O)NC2(C(N)=O)CC2)(C)CO)c[nH]c2cccnc12 47433,c1(-c2c(CNC(c3ccc(OC)o3)=O)cccc2)cnc(CO)cc1OC 47434,C1(CNC(C2CCC(CC)O2)=O)CCCN(C(=O)Cc2cncnc2O)CC1 47435,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47436,C1(F)(CNC(C2(C(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47437,N1(c2n(C)nnn2)CC23CCCC2(CN(C(c2cnc4c(c2)CCC4)=O)C3)C1 47438,C1(C#N)(C(N2CCC(NC(C(C)n3cncn3)=O)(CF)C2)=O)CC2CCC1CC2 47439,C12(CNCC3CCC(C)SC3)CC3CC(C1)CC(Br)(C3)C2 47440,C(=O)(C(C#N)C(C)C)NCC(C)(C1CC1)NC(c1c(C)scn1)=O 47441,C1(C#N)(C(=O)NCC2(NC(C(CC=C)CC)=O)CC2)CC2CCC1CC2 47442,N1(C(c2cnc(OCC)s2)=O)CCC(CN(C(=O)COc2cccnc2)C)CC1 47443,CC1CC(C)C(C(=O)N(C2CCN(c3nccc(-c4ccccc4)n3)CC2)C)O1 47444,N1(C(c2c(C#C)c[nH]n2)=O)CC(=O)NCC1C(=O)NC1CCCC12CC2 47445,S(=O)(=O)(c1c[nH]c2ccncc12)NC(CC1CC(C)N(Cc2ccccc2)C1)=O 47446,N1(C(c2ccc(S)cc2)=O)CC2(CCN(C)CC2)C1.CC1CC2(CC2)C(N)CO1 47447,CN1CCC2C(CCCN2C2CCN(c3ccc(F)cc3F)C2=O)C1 47448,C(c1cc2ccccc2n1CC(=O)NC(c1ccsc1)CO)=CC 47449,C(=O)(C(C)(C)S(C)(=O)=O)NC(C1CCCN(C(=O)COC(F)F)C1)C 47450,C1(NC(C2(C)CC2(F)F)=O)CCC(NC(=O)C(c2ccccc2)=O)CC1 47451,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CC3(F)F)=O)c12 47452,CCC(CC(=O)N1CC(F)CC1CO)N(C(=O)C=Cc1cn(C)cn1)C 47453,CC1CCCN(CCNC(C2(C)CN(C(c3cccs3)=O)C2)=O)C1 47454,c1(C(=O)OCC)ccc(-c2ncnn2CC)cc1.C12(c3nn[nH]n3)CC1C2 47455,c1(C(C(=O)NC(CC)CNC(=O)C(C)SC2CC2)C2CCCC2)ccc(F)cc1 47456,C(CC(C)CN=C(NCc1nsc(CC2CCCCO2)n1)NC1CC1)OC 47457,C(=O)(CC(C(F)(F)F)NC(c1snc(C)c1N)=O)NC(c1ccc(O)cc1)CC 47458,c1(CC(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47459,c1(NC2(CNCC)CC2)cc(C2CCC2)[nH]n1 47460,CN1C(=O)OCC1C(=O)NC1CCCCC1NC(C1(Cc2cccnc2)CC1)=O 47461,N1(C(C(CCCC)F)=O)CC2CCC1C(N(C(=O)C(C(=O)OC)OC)CCC)C2 47462,C1(NC(Cc2cc(COC)on2)=O)CC1C1CCCN(C(c2ccoc2C)=O)C1 47463,C1(NC(CN(C(C(C)C)=O)C)=O)CC(=O)NC1=O.C12CCN(C1)C2=O 47464,C(=O)(CC(C)CNC(=O)OC(C)(C)C)N(CC(C)N(C)C(c1cc[nH]c1)=O)C 47465,c1(OC)ccc(SCC(=O)N(CC(C)NC(C2(C)CCCC2)=O)C)cc1C 47466,c1(C(=O)NCC2(F)CCN(C(C3CCCOS3)=O)CC2)cnc2ccnn2c1O 47467,C1(CNC(C2(CC)CCC2)=O)CC(CNC(=O)C(C)OCCOC)CO1 47468,N1(Cc2nccc(NC)n2)CCCc2cc(OC)cnc21 47469,N1(C(c2c(C)n(C(C)C)cc2)=O)CC(NC(=O)C(C)(F)c2ccon2)C(C)(C)C1 47470,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47471,C12(C(N3CCCC(NC(c4cccc(N(C)C)c4)=O)C3)=O)CC(N=[N+]=[N-])C1C2 47472,C=CC(F)(F)C(=O)NCC(CNC(=O)C(C)c1cccs1)OC 47473,C(=O)(CS(=O)(=O)C1CC1)NCC1C(NC(C(C)Cc2ccncc2)=O)C1 47474,C(CN=c1nc2ccccc2c(N2CCc3nc(O)ccc3C2)[nH]1)C1CN(C)C1 47475,N1(C(C2(C=C)CCCC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47476,C1(NC(=O)C=C(Cl)Cl)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47477,CCCCCC(=O)NCCCCN(C)C(c1ccnc(N2CCCC2)n1)=O 47478,c1(NC(C2C(NC(C(C)O)=O)C2)=O)nc(Cl)ccc1F 47479,N1(C(c2c(CC)c(C)sc2)=O)CCN(C(c2c(C)ccn2C)=O)CC1CO 47480,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)N(C1CC1)Cc1ccco1 47481,C(=O)(C(C(C)NC(=O)CCC(C)CC)C(C)C)NCCCCC#CC 47482,C1(c2n(-c3ccc(CC)cc3)nnn2)(NC2CCC2C)CC2CCOC12 47483,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(=O)C3CC3)CC12 47484,CC1COCC(CC(=O)NCCSCC(=O)NCCC(C)(O)C2CCC2)O1 47485,C(=O)(C1=CC2(CCOC2)C1)NCC1CN(C(C(n2cnc(C#N)n2)C)=O)CC1O 47486,c1(C(N2CCC(NC(c3c(CC)oc(C)c3)=O)C2)=O)onc2c1CCCC2 47487,CCC(C)CC(=O)C(=O)NC(c1cccc(Cl)c1)Cn1cc(-c2nccn2C)nn1 47488,C(CC(=O)NCC1=CCN(C(c2ccn(CCF)n2)=O)CC1)(C(N)=O)NC(C)=O 47489,c1(NC(C2(C)CC=C(C)CC2)=O)cc2c(C)cccn2n1.C12CC(O)CN1C2=O 47490,N1(C(COC(C)=O)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)CC1 47491,Cc1cc(NC2CCC3CC23)ccc1-n1cnnn1.C1CO1 47492,c1(NCC)ccc(C)cc1C(=O)NCCC(C)NC(=O)Cn1nc(C)n(C)c1=O 47493,CC1CN(c2nnnn2CC2CCC(CN)C2)CCCO1 47494,Cc1cccc(COC(C)C(=O)NCC(C)(CO)NC(c2c(C)cnn2C)=O)c1 47495,C(=O)(CCCCC(=O)NC(C1CCCN(c2ccnc(SC)n2)C1)C)NC 47496,N1(C(c2cnc(C)nc2C)=O)CC(NC(C2(Cl)CC2)=O)C(N=[N+]=[N-])C1 47497,c1(C(=O)NCC2(C)C(C)CN(C(c3nnc(S)n3C)=O)C2)cc2ncccn2n1 47498,c1(C(N2C(C)CC(NC(C3CCC4(CC4)C3)=O)CC2)=O)c[nH]c2ccc(Br)cc12 47499,N1(c2nc(C3CC(C)(O)C3)on2)CCCc2ncc(F)cc21 47500,C=CCC(C)(C)CC(C(=O)Nc1ccccc1Br)N1CCC(C(C)(C)O)C1 47501,C12(C(N(C)CC3CCCN3C(=O)CCc3nncn3C)=O)CC1COC2(C)C 47502,C12CC3CC(C1C3)NC(=O)C1(CC1)C(=O)N2.c1(C2(C)CC2)cncc(F)c1 47503,c1(C(=O)NC2CCN(C(c3cc(O)cc(O)n3)=O)CC2CO)cc2occc2s1 47504,C1(CNC(=NC)NC2CCC(N(C)C)C2)CNCC(C)(C)O1 47505,C1(C(N2CCC(CNC(C(C)OCCCC)=O)C2)=O)(CC)CCCC1 47506,CC(c1cccnc1)=CC(=O)NCC1(CO)CCCO1 47507,C(=O)(C1=Cc2ccccc2C1)NC1C(C)(C)CN(C(c2nocc2Cl)=O)CC1 47508,C(=O)(CC1=CCCCC1)NC1(C)CCCN(C(c2cncc3nc[nH]c23)=O)C1 47509,C1(C(=O)NC(C(C)NC(=O)Cc2nnn(C(C)(C)C)n2)CO)CC12CCCCC2 47510,CC1(C(=O)Nc2ncccc2SC(F)(F)F)CCCN(C(C2CCOC2)=O)C1 47511,C(=O)(C1=NOC(CNC(=O)C(C)=C(C)CC)C1)N1CC(C#C)C1 47512,C(CC1=CCN(C(C2CCNC2=O)=O)CC1)NC(c1n(C)c(Cl)cn1)=O 47513,C1(CCCNC(=O)CCCF)CCCCN1C(c1cc(Cl)c(Cl)s1)=O 47514,c1(C(N2C(C3(NC(CN(C)C4CC4)=O)CC3)CCC2)=O)ccc(S(C)=O)cc1 47515,c1(CC(N2C(CN(C)C(C3CC3(Cl)Cl)=O)CC(F)C2)=O)ccc2c(c1)COCC2 47516,C1(NC(C2N(CCC)CCC2)=O)CC2(CCN(C(=O)Cn3nc(C)nc3C)C2)C1 47517,c1(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)OC)ccn2cncc2c1 47518,c1(C(=O)NCc2ccc(C(=O)NC(C)Cc3cccs3)o2)cccc(F)c1O 47519,CCCCC(CC)C(=O)N1CCC(CO)C(NC(c2ccnc(CC3CC3)c2)=O)C1 47520,N1(C(c2c(C)coc2)=O)CCC(N(C)C(c2nn(C)c(Cl)c2Cl)=O)C(C)C1 47521,O=C1CC(C2CC2)(C(=O)NC23CCC(C2)N(C(c2nnc(O)cc2O)=O)C3)C1 47522,C1(C(=O)NCCCOCCCO)(CNC(=O)Cn2cccc2)CCCO1 47523,c1(NC(c2ccn(C)n2)CC)cc(NCCC(O)C(C)C)ncn1 47524,C(=O)(C(F)(F)C(C)(C)O)NCC(=O)N(C(C)C(=O)NCC1CC1)CC 47525,C(=O)(CC(O)CC(C)(C)C)N(CC(=O)OC1CCOC1=O)C 47526,n1(CCOC)cc(CC(C2CCCCC2)NC(C2(c3cccnc3)CC2)=O)nn1 47527,c1(CN(CC)Cc2cccc(Cl)c2)cccc(F)c1C(=O)OC 47528,N1(CCN2CC(CCCCNC(=O)OC(C)(C)C)C2)CCCC1CC(=O)O 47529,c1(OC)nccc(I)c1CN1CCN(C(c2cnc(F)c(C3CC3)c2)=O)C2CC12 47530,N1(C(CC(=C=C)C)=O)CC2CCN(C(c3ccn(C(CC)CC)n3)=O)CC2C1 47531,C1(C(=O)NC(C2(O)CCN(C(=O)CC(C3CC3)C3CC3)CC2)C)CCCC(C)(C)C1 47532,C1(CC(=O)OC)C(C)OCCN1C(CCC1CCC1)C(=O)NCc1ccccc1 47533,c1(CNOc2cccc(C3(COC)CC3)c2Cl)ccc(N2CCCC2)cc1Cl 47534,Cc1nc(C(=O)NCCn2cc(C(=O)N(CCCN(C)C)C)cn2)sc1C 47535,n1(CC#C)cccc(C(N2CCNC(CC)C2)C(=O)NCC=C)c1=O 47536,Cc1nn(C)cc1CNC(=O)C(=O)N(CCCCC(=O)O)C 47537,C1(C(=O)OC)CC(C(N2CCN(C(c3cc(COC)c[nH]3)=O)CC2)=O)C12CCC2 47538,C(=O)(CCCCCCCC1CC1)NCCC1(O)CN(C(C2CC(N(C)C)C2)=O)C1 47539,c1(-n2c(CN(CC(C)C)CCC)ccc2)cccc(-c2cccn2CC(C)C)c1 47540,N1(C(CC2(N(C)C)CC2)=O)CCCCC(C(N2CC(c3ncc[nH]3)C2)=O)C1 47541,C1(C(N2C(CSC)CC2C)=O)CCCN(C(=O)COc2ccsn2)C1 47542,Cc1cc(C(=O)N(CCCNC(C2CCCC(F)(F)C2)=O)C)cc(C)c1O 47543,c1(OC)ccc(F)c(C(=O)NCC23CCC(CN2C(c2ccccn2)=O)C3)c1Cl 47544,C1(COC)CN(C(c2ccc(-c3ccncc3)cc2Cl)=O)CC(C)O1 47545,C1(COC)(NC(c2cc(C3(C)CC3)n[nH]2)=O)CCN(C(C2CC2F)=O)CC1 47546,Cc1ccc(C(=O)NC2CC(NC(=O)C(C)(C)c3ccno3)C(O)C2)c(F)c1C 47547,C(CCSC)(C(=O)NC1CCN(CC2CC2)C1)NC(C1CCC(CC)CC1)=O 47548,N1(C(c2cn(C)nn2)=O)CCC2(CC1)CN(C(C1CC3CC3C1)=O)C1COCC21 47549,N1(C(C(CC(C)C)C)=O)CCC(C2CCCN(C(C3SCCCS3)=O)C2)C1 47550,C1(C(N(C2CCCN(C(Cc3nnc(C)s3)=O)C2)C)=O)CCc2nc(C)nn2C1 47551,CC(CN=c1[nH]c(=NCC2CC(F)(F)C2)[nH]c2c1CCC2)n1ccnc1 47552,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cn2nc(C)cc2C)CC1SC 47553,C(=O)(CCC(=O)C(C)(C)C)NC1CCC(CCC(=O)NCC(N(C)C)C2CC2)C1 47554,Cc1ccccc1OCC(=O)NC1COCC1C(=O)NC(CO)C(C)C 47555,C(=O)(C(CC(C)C)C(C)C)NCCNC(=O)NC.C12(C)CCN(C1)C2=O 47556,c1(C(N2CCC(O)(C(C)NC(CNC(=O)NC)=O)C2)=O)cc2c(nc1O)CCC2 47557,C=CCCC(O)CNC(C1CN(C(C2CCOC2CC)=O)CC1C(C)C)=O 47558,CCCC(CCCO)C(=O)N1CCN(C(=O)CC2CCN(C(C)C)CC2)C(C)C1 47559,CN(S(N)(=O)=O)CC(=O)NCCCC1(NC(c2ccn(CCOC)n2)=O)CC1 47560,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47561,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47562,Cc1nc(F)ccc1NC1(c2nnnn2C2CCC2)CCN(c2ccccc2)C1 47563,C1(CNC(C2(OCC)CCCC2)=O)CCCC(NC(=O)CSCCC(C)C)C1 47564,N1(C(C(C)(C)C2CCCO2)=O)CC2CCCC(NC(C3CC3F)=O)C2C1 47565,c1(C(=O)NCC23C(CN(C(c4cn(CC=C)nn4)=O)C2)C3)cccn2cnnc12 47566,CCC(C)C(C)C(=O)N1CC(CNC(c2csc3nnsc23)=O)C(C)C1 47567,C(CC(C(=O)NOC(CO)C(C)C)NC(C1CC(C(C)C)C1)=O)=CC 47568,CCC(C(=O)NCC(CNC(=O)CC1(C)CC1)OC)Sc1nc(=N)[nH][nH]1 47569,N1(SCc2ccc(-c3cccs3)o2)CC(=O)N(C(C)(C)CC2CCCCC2)C1=O 47570,c1(C(C)(C)C)cc(NCC2(C3CCCOC3)CC2)n2ncc(C#N)c2n1 47571,C1(NC(c2nc(OC)c(F)cn2)=O)CCN(C(C2CCN2C(C)=O)=O)CC1C 47572,C12C3CCN(CC13)N1C(CC1)C(=O)N2.C1CCCC1.C(=O)CNC=O 47573,C1(NC(C(CC)NC(N)=O)=O)CC2CCC1C(NC(C1CC(O)C1)=O)C2.CC 47574,C(C)(C(C)(C)NC(c1ccn(C(C)(C)C)c1)=O)NC(C1CC(C)C1)=O 47575,c1(CS(C)(=O)=O)cc(-c2cc(NC(c3ccc(O)c(Br)c3)=O)n[nH]2)ccc1F 47576,CC(C)C(C)CC(=O)NCCC1(C(=O)NOC2CC2)CN(C(N)=O)C1 47577,C(c1ccc([N+](=O)[O-])cc1)=CC(N1C(CNC(C(C)C(C)(C)C)=O)CCC1)=O 47578,Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(c1cnoc1C(C)C)=O 47579,c1(C(=O)NCCCCCNC(Cc2cc(C)sc2)=O)coc2ccccc12 47580,N1(CC(C)O)CCN(C(c2nccn2CCC#N)C(=O)NC2CCC2)C1 47581,CCC(CC(=O)NCC1CN(C(=O)CCCCC(C)C)CCO1)C(C)C 47582,N1(C(=O)CCc2cnco2)CCCCC2(CCN(C(C3CCOCC3)=O)C2)C1 47583,C1(C(C)(C)C)CN(C(=O)C=CC2CCCO2)CCN1C(=O)C(Cl)=CCl 47584,CC(CN(C(=O)C(CCN(C)C)NC(C1CC(O)C(F)C1)=O)C)C(C)(C)C 47585,c1(C(=O)NC2CCN(C(C3(C(C)N(C)C)CC3)=O)C2)cc(C(C)C)oc1C1CC1 47586,N1(C(C(C)(C)N(C)C)=O)CCC(C2CCCN(C(C3CC3C(C)(F)F)=O)C2)CC1 47587,c1(CC)cc(-c2cncc(NC(=O)Cc3ccccc3Br)c2)cc([N+](=O)[O-])c1 47588,C1(CNCc2cccc(OCCCC)c2)CCCC1C1CC1 47589,c1(C(=O)NC(CC)CNC(C2(SC)CC2)=O)sc(C2CCCN(C)C2)nc1C 47590,N1(C(CC(CC(C)C)O)=O)CCC2CCC(C1)N2C(c1cccc(CN(C)C)n1)=O 47591,N12CCc3ccccc3C1CNC(=O)C2=O.Cc1cc(O)nc(C)c1C(N)=O 47592,C(CC1c2ccccc2CCN1C(=O)Cc1ccon1)NC(=O)C(C1CC1)C1CC1 47593,CC1CN(C(C2CCOCN2C(=O)CCS(C)(=O)=O)=O)CCS1=O 47594,c1(N(C)C)cc(NC(=O)NCC2CCC(C(C)(C)C)CC2)ncn1 47595,C1(OC)CN(C(C2SCCCS2)=O)C(C)(CNC(=O)COCC(=O)N(C)C)C1 47596,CCCC(CC1CCCCC1)C(=O)NC(CNC(c1c(C)cccc1F)=O)CC 47597,c1(CSC(C2C=CCC2)=O)ccccc1CN(C1CCC1)C 47598,C1(CN(C(=O)C(=O)Nc2cocn2)C=O)CCC(C(F)F)CC1 47599,Cc1ncc(C=CC(=O)N(C)CC2CCCN2C(=O)COc2cnn(C)c2)s1 47600,c1(CC(=O)NCC(C)NC(=O)CC2CCCOC2)ccc(N2CCOCC2)nc1 47601,C1(CCNC(C=CC(C)(C)SC)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 47602,CC(C)C(O)C(C)(C)C(=O)NCC1CCC(NC(=O)CSc2nnnn2C)CC1 47603,Cc1cc(CC(=O)NCC(C)CN(C(=O)CC(c2c(C)n[nH]c2C)C)C)ccn1 47604,c1(NCC(CC)C)ncnc(NC(COCC(F)(F)F)C(C)C)c1C 47605,C1(NC(c2ncc(CC)s2)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1C)=O 47606,N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CCC2 47607,C1(NC(C(C)(C)OC(C)C)=O)CCN(C(C2C(C)C2C)=O)C1C(C)(C)C 47608,c1(CC=CC(C(=O)O)NC(=O)OC(C)(C)C)cc(Cl)ccc1Cl 47609,O=C1CNC(=O)N1CCC(=O)NC12CC1CN(C(c1ccoc1C1CC1)=O)C2 47610,c1(NC(C=CC)=O)ncc(-c2c[nH]c(=N)c(C)c2)cc1O 47611,C1(N2CCOCC2)(CC(=O)N(c2ccccc2)CC)CCN(C(=O)C(=O)N(C)C)C1 47612,c1(NC(C2CC(NC(c3nc(N(C(C)=O)C)sc3)=O)C2)=O)c(C)[nH]c(C)c1C 47613,c1(C(=O)NCCCN(C(CC(c2c(C)n[nH]c2C)C)=O)C)cnc2nncn2c1C 47614,N1(C(CSc2ccc(OC)cc2)=O)CCCC(C)C1CNC(c1cc[nH]n1)=O 47615,CN1CCN(C(c2ncncc2F)=O)C(CNC(C2(F)CCC2)=O)C1 47616,Cc1nccn1CCCC(=O)NCC1CCN(Cc2cnn(C)c2)C1 47617,c1(Cc2ccc(COC(=O)Nc3cnc(SC)nc3)cc2)cnc(CO)nc1C 47618,Cc1nccn1CC(=O)NC(C(=O)NC(c1nc[nH]n1)C)C1(O)CCC1 47619,Cc1nc(C(=O)NCC2C=CCN2C(c2nscc2C)=O)c2ccccn12 47620,c1(CC2CC2)cnc(C)c(NCC(=O)N(C2CCN(C(=O)CO)C2)CC)c1 47621,C1(C(C)NC(=O)C(C)n2cccc2)CCN(C(=O)C(C)(C)C2CCCCC2)C1 47622,N1(C(CCCCCC)=O)CC(NC(=O)CC2CCCNC2=O)CC2(CC2)C1 47623,c1(NSc2scc(C)n2)nc(N2CCC(O)(CCN(C)C)C2)nc2ncn(C)c12 47624,c1(CCC(N2C(CCNC(C(C)n3ccnc3)=O)CCC2)=O)ccc(N)c(F)c1 47625,CC(C)CC(CNC(C1CCC(=O)N1)=O)C(=O)NC1CCN(C(C)C)CC1 47626,c1(OCC)ccc(S(=O)(=O)N(c2cc(C(C)(C)C)nn2C)C2CCC(N)C2)cc1Cl 47627,c1(C(N2CC(F)CC(C(=O)NCc3cccs3)C2)=O)cc(F)cc(F)c1I 47628,c1(N(CC(CN(C(C(C)CN(C)C)=O)C)O)C)cnc(C#N)cn1 47629,N12CCCC(C1)N(C1CN(C(C3CC34CC(O)C4)=O)C1)C(=O)CC2.C(C)(C)(C)OC 47630,C1(NC(CSCC(C)C)=O)CCN(C(C2CN(n3ccnn3)C2)=O)C(C)C1 47631,C(=O)(C(CC1CCCCO1)NC(C1CC2CC2C1)=O)OC 47632,C(=O)(CCCC(=O)NCC1CC1C(=O)NCC(F)CC1CCCC1)OC 47633,C(CCc1cn(CCNC=O)nn1)(C(=O)O)NC(C(C)(C)c1sccc1Cl)=O 47634,C(C(CNC(C1(C(=O)N(C)C)CC1)=O)C(F)(F)F)NC(C1(C)C(C)(C)C1)=O 47635,c1(C2(c3ccc(NC(C4C(C)C4)=O)o3)CC2)ccccc1S(C)(=O)=O.C12CC1C2 47636,c1(C(=O)NC2CC(CNC(C3C(C)C3C)=O)C2)cnc2ccc(F)cc2c1 47637,CC(C)CS(=O)(=O)CCC(=O)N1CC(CC(C)NC(=O)CCn2ccnn2)C1 47638,N1(C(C2CC(C(C)C)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1C 47639,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(CO)C1 47640,C1(NCC(F)(F)F)CCCCC1(C)C.c12ccc(cc1)NCC(N)C2 47641,C1(NC(CN(C(=O)Cn2c(C)ccc2C)CC#C)=O)CCn2ncnc2C1 47642,c1(OC)ccccc1CCN1CCOCC1c1cn[nH]c1.N12CCN(CC1)CC2 47643,N1(C(c2cc(CC)nn2C)=O)CC(C)(C)CC1C(=O)NCC1CCCN(C)C1=O 47644,c1(CCC(=O)NC(C2CN(C(c3n[nH]c(CC)c3C)=O)C2)C)nnc(O)nc1O 47645,C(C(C)(C)CC(=O)N1CCCCC1C(=O)NC1CCN(C(C)C)CC1)OC(C)=O 47646,c1(C(=O)NCCCCC=CCNC(C2CN(C)C(=O)N2)=O)ccnc(Cl)c1O 47647,CCC(C)C(O)CNC(C1CCCN(C(=O)Cc2c(C)noc2C)C1)=O 47648,N1(C(CCCc2ccc(C)nc2)=O)CCN(C(C2OCCCO2)=O)C2CC12 47649,c1(C(=O)NC2C(CNC(c3n[nH]c(C(C)C)c3Br)=O)C2)cc(F)c(F)cc1O 47650,CON(C)C(=O)CN=c1[nH]c(=NCc2cccc(C(C)C)c2)[nH]c2c1SCC2 47651,C1(CNC(=O)CN2CCN(C(=O)Cc3ccsc3)CC2)COCCOC1 47652,c1(CC)c(C(=O)NCC(C(C)C)NC(=O)CCC(C)(C)C#N)cnc2ncnn12 47653,c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CCC3)=O)C2)nn(C)c(C)c1Cl 47654,C1(CNC(c2noc(CC)c2C)=O)C(C2CC2)CCN1C(=O)C(C)=C1CC1 47655,C=CCCC(F)(F)C(=O)N1CC(NC(=O)CC(C)(C)COC(C)=O)C(CC)C1 47656,N1(C(COCCC)=O)CCC(NC(=O)C(O)CC)CC1(C)C 47657,N1(C(Cc2cncc(C)c2)=O)CCN(C(C2CCOC(=O)CC2)=O)C2COCC12 47658,C(CNC(C1CCNC1=O)=O)(CC(=O)N1CC(F)(CF)C1)OC 47659,N1(C(C(C)N(C)C)=O)CCC(CNC(C23CC(CO2)C3)=O)C1 47660,c1(N(C(C(N2CCCC(C)C2)CC)=O)CCCCC2CNC2)ncc(C)c(C)n1 47661,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)cc1)=O 47662,C1(C(=O)NC(CCCC)C2CC2)CCCCN(C(=O)C(C)OCOC)C1 47663,C1(CNC(c2cn(C3CCC3O)nn2)=O)CN(C(C2(CF)CCC2)=O)CC1O 47664,C(=O)(CC(C)(C)N(C(=O)CCn1cc(Br)c(C)n1)C)NCC(C1CC1)OC 47665,Cc1cc(N2CCNC2=O)ccc1NC(=O)C=C1CCC1.C12CCN(C1)C2=O 47666,C1(CC)C(NC(c2ccc(SC)o2)=O)CCCN1C(C1(CN(C)C)CC1)=O 47667,c1(C(=O)NCC(C)NC(c2coc(N(C)C)n2)=O)cnn2cccnc12 47668,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 47669,Cc1cc2ncc(C(=O)NCCC3CC(NC(C4(C)CC4(Cl)Cl)=O)C3)c(C)n2n1 47670,CC1(C(=O)NOCc2cccc(F)c2)CCN(C(c2nccnc2N)=O)CC1 47671,C(=O)(C1=CCC(C)(C)CC1)NC(CCC)C(=O)Nc1ccsc1C#N 47672,C=C(Cl)CC(C(=O)NC1CC(C)(O)C1O)NC(c1cc(Cl)cn1C)=O 47673,N1(C(Cc2cn(C)nc2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 47674,CCC(C)C(C(=O)NC(c1cncn1C)CO)N(C(=O)C#CC(C)(C)C)C 47675,Cc1ccc2c(C(=O)NC(C3CCN(C(c4occc4F)=O)C3)(C)C)c[nH]c2c1 47676,C1(NC(C2N(CC)C(=O)CC2)=O)CCC12CN(C(c1cnc(S)[nH]1)=O)C2 47677,N1(C(C(C)NC(=O)NC)=O)CCC2=C1CN(C(C13CC4CC1C3C4O)=O)CC2 47678,CCCCC(CCC)NC(C1(N(C(=O)CC2CCOCC2)C)CC1)=O 47679,N1(C(c2c(C)cccc2Cl)=O)CC(NC(=O)C=CC2CCCO2)CC2(CCC2)C1 47680,c1(CC2CCN(CCNC(C(CC)C(C)C)=O)CC2O)cc2oc(C)cc2[nH]1 47681,C1(C(=O)NC(C=C)C2CC2)CCC(C)(C)N(C(=O)CCC(C)CN(C)C)C1 47682,CCC1C(=O)NC2CC(C2)OCC(=O)N1.c1(CC(C)N(C)C)nc[nH]n1 47683,N1(C(c2cc(CC)sn2)=O)CCC2(C(=O)N(c3ccc(C)c(C)c3)CC)CC2C1 47684,C=C1CCN(C(=O)C(C)CN(C)C(C2(C)CC=CCC2)=O)CC1 47685,c1(SC)ccc(C(=O)NCC2CN(C(=O)C(C)SC)CC2c2cncn2C)cc1 47686,N1(C(c2ccc(C)cn2)=O)CC(C)CCC1CNC(=O)C(C1CCC1)C1CCC1 47687,C1(C(=O)NC2CCC(F)(CNC(CCOCC(C)C)=O)C2)CCc2ccnn2C1 47688,C(C(N=c1ccnc(NCCCn2cccnc2=O)[nH]1)C1CCCO1)N(C)C 47689,C1(NC(C(C)=C2CC2)=O)CC(C)(NC(=O)CC(C)N(C)C)C1 47690,CCC(CN=c1ccc(Br)c(S(=O)(=O)Nc2cc(C)cc(C)c2)[nH]1)OC 47691,C(CC(C(=O)NCC1CCC1C)N(C)C)NC(CC(C)C)=O 47692,c1(C(=O)NCC2C3COCC23)ccccc1OCc1ncoc1C 47693,CCCC(CCCNC(=O)COc1ccsn1)NC(=O)C=Cc1c(C)coc1C 47694,N1(C(C2C=C(C)CS2)=O)CCC(NC(C2CCCCS2)=O)C1c1ccccc1 47695,CC=C=CCCN=c1ccc(S(=O)(=O)N2CC34CCC3(COC4)C2)c[nH]1 47696,CC1CCC(c2nnnn2C2COC2)(NCCc2cnc[nH]2)C1 47697,c1(C(=O)NC(C)CN(C)C(C23CCC2C3)=O)cc(F)c(F)cc1F 47698,n1(CC(=O)NC2C(C)N(C(=O)C=CC3CC3)CC2)sc(=O)c2ccccc12 47699,c1(CC)cc(C(=O)NCCCN(C)C(C2CCCCN2N=O)=O)ccc1Cl 47700,N1(C(CC2(OC)CN(C(C3C=CCS3)=O)C2)=O)CC(CO)OC(C)C1 47701,C1(CC(C)C)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 47702,C1(NC(C2(CCC=C)CN(C(c3cc[nH]c3)=O)C2)=O)CCn2cncc2C1 47703,c1(CCC(=O)NCC(C)N(C(=O)CSCc2ccncc2)C)cncnc1O 47704,C1(C(=O)NCCC(=O)NCC#C)COC2(C1)CN(C(c1cnc(OC)nc1)=O)C2 47705,c1(C(=O)NC2C(C)CCN(C(c3nc(C)oc3C)=O)C2)c(C)nc2sc(C)cn12 47706,N1(C(C2C(C)(Br)C2)C(=O)NCc2cccs2)CCCC2C(=O)NCCC12 47707,c1(C(N(C2CCN(C(C(=Cc3ccco3)C)=O)C2)C)=O)cc2c(ccn2C)[nH]1 47708,C1(CC(C)C)(NC(=O)CN2OC(C)CC2=O)CCNCC1 47709,C(=O)(C(F)C(C)CNC(=O)Cc1cccnc1)N(CC(C)OC)C 47710,C12(CNC(C=CC)=O)CCC1CCN2C(=O)C1CC1 47711,C(=O)(CC(O)C(Cl)(Cl)Cl)NCC=CCNC(=O)Cc1cc(C(F)F)on1 47712,N1(C(C2N(CC)CCC2)=O)CCC(C)(CNC(c2sncc2C)=O)C1 47713,C1(CC(=O)N)(N(C)C)CCCC1.n1(CCNC(C(=O)NCC)=O)cnc(CN)n1 47714,c1(OC)c(OC)cc(C(C)NC(=O)NCCC2CCS(=O)(=O)CC2)cc1Br 47715,c1(C(N2C(CN(C(CC(C)C3CC3)=O)C3CC3)CCC2)=O)c(C2CC2)cnn1C 47716,C1(C(N(C)CCNC(=O)CCOc2cccc(Cl)c2)=O)CCN(C2CC2)C(=O)C1 47717,C(CC(O)CCO)NC(C(C)(C1CCC1)NC(CC(C)F)=O)=O 47718,[N-]=[N+]=Nc1ccnc(C(=O)NCC=CCNC(C23CCC2C3)=O)c1 47719,c1(C(=O)NCCCC(CCC)NC(=O)Cn2ncnn2)cnc2ncccn12 47720,Cc1nc2ccc(C(N3CCN(C(C4CCn5nccc5N4)=O)CC3)=O)cn2n1 47721,C(C)(CNC(c1ccncn1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 47722,N12CCC(O)C(C)(C1)C2.c1(-c2n(C)cnc2)csc(=NCc2cc(I)cnc2Cl)[nH]1 47723,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 47724,Cc1cc2c(C(N3CCC(CNC(=O)CSC(=N)N)CC3)=O)cccc2[nH]1 47725,C1(C)(CC(=O)Nc2c(C(=O)OC)n[nH]c2)CCCN(c2ccnc(C)n2)C1 47726,c1(-c2cn(CCC(N3C(CC)COCC3)=O)nn2)cc(C)cnc1F 47727,n1(CCOCC)c(N2CCOC(C)C2)nnc1C1(OC)CC1 47728,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 47729,CC1(F)CN(C(=O)COc2ccccn2)CCN(C(=O)Cc2nnn(C(C)(C)C)n2)C1 47730,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 47731,Cc1ncc(N)cc1C(=O)NCC(C)NC(=O)C(c1cscn1)N(C)C 47732,Cc1cccc(Br)c1CN1CCNC(=O)C1c1cccc(Cl)c1 47733,CN1C(=O)CCC1CC(=O)NCC1CN(C(=O)C(C)(C)n2cnnn2)C1 47734,c1(OCC)ccc(Oc2ccc(CCCC#N)cc2)cc1.N12CCCC1C2=O 47735,Cc1nsc(C)c1C(=O)NCC1CCCC1NC(c1cncc(N(C)C)n1)=O 47736,C(CC(=O)NCCS(C)(=O)=O)(C(F)F)NC(Cc1cc(C)n(C)n1)=O 47737,C1(O)(C(C)NC(C2(CC#C)CCOC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 47738,c1(C(C2CCOC2)CSC)nc(-c2cccs2)nn1-c1ccnc(F)c1 47739,C(=O)(C(F)(F)CC(C)C)NC1(COC)CCN(C(=O)Cn2cc(Cl)cn2)C1 47740,C1(CCC(=O)NC(C(=O)NC2CCN(CCF)C2)C2(O)CCC2)CCCOC1 47741,C(CS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CC(F)C(=O)N1)=O)OC 47742,N1(C(C2C(CC)C2)=O)CC(CNC(c2cccc(C(C)C)c2N)=O)CC12CCC2 47743,c1(CN(C)C)cnc(O)cc1C(F)(F)F.C12CC(C1)NC2=O 47744,C(C(C)(C(=O)NC(C1CCN(C(=O)C=Cc2ccncn2)C1)(C)C)OC)OC 47745,N1(C(COC2(C)CCC2)=O)CC(CNC(C2(C)CC2c2ccccc2)=O)C(O)C1 47746,C1(C(=O)NCC2C(NC(CCOCC)=O)C2)CC=CCC1 47747,CCC1=NOC(C(=O)NCC(CO)NC(c2cccc(C3CC3)n2)=O)C1 47748,N12CCC(C)(C1)C2=O.c1(N(C)C)cccc(OC(F)(F)F)c1 47749,Cc1nc(CN2CCC(C(=O)Nc3cccc(-n4cccn4)c3)CC2)c(C)s1 47750,C1(NC(=O)C(C)OC2CCCC2)CN(C(=O)CCc2cnc(C)s2)CC1CCC 47751,c1(CC(C)C)c[nH]c(C(=O)NCC2CCC2NC(=O)CCc2ccsc2)c1 47752,c1(C(c2n(CC(=C)C)nnn2)NC2CNC(=O)C2)cc(C(F)(F)F)ccc1F 47753,c1(C(=O)NCCC2CC(NC(C(C)(C)SC)=O)C2)cc(C(C)C)nc(O)c1 47754,O=C(C(O)C(F)(F)F)NC1CCC1CNC(c1cccc(C(F)(F)F)c1Cl)=O 47755,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 47756,Cc1ncnc(C)c1C(N1CC(NC(=O)C(C)C2CCOC2)C(C)C1)=O 47757,C(N=c1[nH]c(N2CCC(N3CCC3)C2)nc2c1COC2)c1c(Br)cncc1 47758,c1(C(=O)NCC(c2cccc(C)c2)NC(=O)C=C(Cl)Cl)c(C)[nH]c(C)c1C 47759,c1(CC)c(C(N2CCCC2CNC(c2[nH]cc(C)c2C)=O)=O)cnn1C 47760,c12ccc(cc1)C(=O)NC1CC21.CC(C(=O)N(C)C)c1ccco1 47761,CC1CCCN2C1C2.C1(C(=O)OC)CCCCNCC1 47762,N1(c2cc(N(C)C3CC3)ncn2)CCCC(C)(C#N)C1.c12cc(cc(F)c1)N2 47763,C(CCCCC(=O)NC(CC)C(C)(F)F)N(C(c1cc(C(=O)OC)[nH]c1)=O)C 47764,N1(C(CN(CCC)C)=O)CC(C)C(NC(c2nccc3ccsc23)=O)C(C)C1 47765,N1(C(C(CC)C2CCC(=O)N2)=O)CCN(C(=O)CCCCCOC)CC2(CC2)C1 47766,N1(C(C2CCC(N)C2)=O)CCc2c(C(=O)Nc3cc(Br)cc(Cl)n3)n[nH]c2C1 47767,Cc1cc(F)sc1C(=O)NC1CCC(NC(=O)CCC2CC(C)(C)CO2)CC1 47768,C1(CNC(=O)CC2C(NC(=O)CCC3CCOC3)CC2O)CCCCCCC1 47769,N#Cc1cncc(C(N2CCCCC(C(N3CC(CO)C(O)C3)=O)C2)=O)c1 47770,c1(CC)ccccc1CC(=O)N(C)CCOCCCNC(=O)C(C)c1cncs1 47771,C1(CCC)(Nc2nn(C)c(C)c2Cl)CCN(C(=O)CCc2nc(C)cs2)CC1 47772,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 47773,c1(CN2CC(CNC(C3CCC(C4CC4)CC3)=O)OCC2)ccc(Cl)nc1Cl 47774,C(=O)(CCCCCOC)NCC1(CCNC(c2ccnc(C(C)C)n2)=O)CC1 47775,Fc1cccc2c1OCC2n1c(=O)n(Cc2ccc(F)cc2)c2ncc(Br)cc12 47776,c1(NC(=O)Nc2ccc(N(C(C)=O)C)cc2)ccc(F)c(C#N)c1C 47777,c12ncc([nH]1)C(c1nnnn1CCCF)N2C.C(CNC(N)=O)NCCO 47778,Cc1ccc(C(=O)NC(c2ccccc2)CNC(=O)CCOCC(C)C)nc1O 47779,c1(C(=O)OC)cccc2c1OCCN(C(=O)Nc1cc(I)n(C)n1)C2 47780,C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N2C(C1CNC(=O)N1)=O 47781,Cn1cnc2c(NC3(C4CN(C(C5(C)CCCCC5)=O)C4)CC3)ncnc12 47782,c1(COC)ncsc1C(=O)NCC1(CC(N2CCCC2CSC)=O)CCC1 47783,C1(NC(C=CCOC)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(C2CC2)C1 47784,CC1CC(C(=O)NC2CCCCC2NC(=O)C(=O)NC2CC2)CN1C 47785,C(=O)(C(O)C(F)(F)F)NCCC(CNC(c1n(CC)ncc1)=O)O 47786,N1(C(c2c(C)c(F)ccc2)=O)CCCC12CCCN(C(c1cnn(C3CC3)c1)=O)C2 47787,c12ccc(cc1)CN(CC)CC(C)NC(=O)CC2.C1(C)(C(=O)OC)CC1(F)F 47788,c1(OC)ccc(NC(=O)CCn2cc(C3CCCOCC3)nn2)cc1 47789,C1(C(=O)NCCCC(C)NC(C(C2CCCCC2)OC)=O)CN2CCCN1CC2 47790,C1(CC)(CNC(C2CN(C(c3sncc3CC)=O)CC2C)=O)CCC(=O)N1 47791,c1(C(=O)NC(C(CO)NC(C(CSC)C)=O)C)ccc(Br)c(SC)c1 47792,C1(C(=O)NCCSC(C)C)CC(=O)N(c2cn[nH]c2)C1 47793,N#Cc1ccnc(CNCCN(C)CCOC(=O)CC2COCCO2)c1[N+](=O)[O-] 47794,c1(CS(=O)(=O)NC2(C(F)(F)F)CC3CC3C2)ccc(F)cc1 47795,Cc1ncc2cc(C(N3CC4CC(N(C(=O)CCCC5CC5)C)C3C4)=O)ccn12 47796,C1(C2CC2)(CNC(C(COCC)C)=O)CCN(C(c2ccc(C#N)o2)=O)C1 47797,C1(CNC(=O)CSC(F)(F)F)CN(C(=O)CC2CCCCC23CC3)CC1(F)F 47798,c1(OCCOC)ccc(C(=O)NCCNC(C2CC(OC)C2)=O)cc1C 47799,N1(C(C2CCC(=O)NC2)=O)CCOC2CN(C(c3cnc4ccccn34)=O)CC12 47800,c1(C(=O)NCC2OCC(CNC(CCC)=O)C2)cc2cccc(Br)c2cn1 47801,N1(C(C2(CSC)CC2)=O)CC2C3CCC(C2C1)N(c1nc(Cl)ncc1C1CC1)C3 47802,c1(NC(c2n[nH]cc2I)=O)ccc2c(c1)CN(C(c1cncnc1)=O)C2 47803,C1(C)(C(=O)NC2CCC(NC(C3(OC)CCC(C)C3)=O)CC2)C(C)(C)C1(C)C 47804,Cc1cccc(CC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)c1 47805,C(=O)(C(CO)C(F)(F)F)N1CCC(NC(=O)CC2CCC2)C1c1ccccc1 47806,C(=O)(C(CC(C)C)C(C)C)N(CCOC)CCNC(C1CC12CCC1(CC1)CC2)=O 47807,C1(CNC(C(C)N(C(C(c2cnn(C)c2)C)=O)C2CC2)=O)CNC(=O)C1 47808,c1(C(=O)NCC2N(C(C3CCC(CCC)CC3)=O)CC2)c(F)ccc(CC)c1F 47809,N1(C(CN(C)S(N)(=O)=O)=O)CCC(NC(C2CCC(=O)N2)=O)CC1C1CC1 47810,c1(CNC(C2(C(=O)OCC)CC2)=O)cccc(OC)n1.N1(C2CC2)CCCCC1 47811,C1(CSC)CCCN1C(=O)C(Cc1cc[nH]n1)NC(=O)Cc1ccsn1 47812,Cc1nc(S)nc(C)c1CCC(=O)NCC1CC1CNC(C1CCN(C)C1=O)=O 47813,C1(C(C#C)C)CCN(C(C2CCC2CNC(=O)Cc2ccoc2)=O)CC1 47814,C(=O)(C(C)C(C)C)N(CCC(=O)NC1CCN(C2CC2)C1=O)CCOC 47815,N1(C(CNC(CC)=O)=O)CC2CC(NC(c3ccn(C4CCCC4)n3)=O)C(C2)C1 47816,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC1CN(C(c2cn3cccnc3n2)=O)C1 47817,c1(NC(C(C2(O)CN(C(C(COC)OC)=O)C2)(F)F)=O)ccncc1[N+](=O)[O-] 47818,N1(C(C(F)OC)=O)CCC2CCN(C(=O)CC3CN4CCN3CC4)CC12 47819,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 47820,C1(C(=O)NC(C2CCOCC2)C(=O)NCCc2n(C)ncc2)CC(C2CC2)C1 47821,c1(C(=O)OC)cc(=NCC2CCC(NC(c3cc(C(C)(C)C)on3)=O)C2)[nH]cn1 47822,C1(CNC(C(C)(C)C)=O)CC2CCCCC2N1C(c1nccnc1C(N)=O)=O 47823,c1(C(C)NC(c2c(COC)scc2)=O)ccc(F)c(N(C)C)c1.C12CC1NC2=O 47824,C(CCCCCCC(=O)NC1CCC1CNC(c1cncc(N(C)C)c1)=O)SC 47825,CCC(CC)C(C)C(=O)NCC1(C)CCCN(C(C2(C3CCC3)CCC2)=O)C1 47826,C#CC1(C(N(C)CP(C)(C)=O)=O)CCN(C(=O)Cc2nonc2C)C1 47827,N1(C(C2(CC#C)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 47828,N1(C(C(c2ccccc2)C)=O)CC=C(CC(=O)N2CCC3CC23)CC1 47829,c1(C(CC)(C)C)nnc(N2CCOCC2C(=O)NC2CCCCC2)n1CC1CC1 47830,c1(C(=O)NCC2N(CC(=O)NC(N)=O)CCC2)ccn2ccnc2c1 47831,C1(CC(=O)NC(C=C)C)CCCN(C(=O)C(CCSC)NC(N)=O)C1 47832,c1(OCC)ccc2c(c1)OC(CC(N1CC(C(F)(F)F)OC(C)(C)C1)=O)O2 47833,c1(OC)cc(N)ccc1C(=O)NC1C2CN(C(C3CC3C3CC3)=O)CC12 47834,C1(CC)(NC(=O)CC2(O)CCOCC2)CCN(Cc2ccsc2C(F)(F)F)CC1 47835,c1(C(N2CC(NC(C3(C)CCC3)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 47836,c12cc(F)c(c(F)c1)[nH]c2=O.c1(N2C(C(=O)OC)CC3CC32)ccnc(SC)n1 47837,CCCCC(O)C(C)C(=O)NCCC1CCCCN1C(c1cccn1CC)=O 47838,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2cscn2)n[nH]1 47839,N1(C(c2cccc(CC)n2)=O)CCC2C(CCCN2C(=O)Cc2cncnc2)C1 47840,N1(c2n(CC(C)C)c(COCC(F)(F)F)nn2)CCC12CCC(C)CC2 47841,C1(F)(CNC(c2n(CC)ncc2Cl)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 47842,c1(CC(=O)NC2(C)CN(C(CSc3c(C)cccc3)=O)C2)nc([N+](=O)[O-])n[nH]1 47843,N1(C(C(C)n2ccnn2)=O)CC2(CCC(CNC(=O)CCF)O2)C1 47844,C(=O)(C1CCCc2nncn21)NCC1C(CC)CCN1C(=O)C(=O)N(C)C 47845,C1(CNC(c2on(C)c(=O)c2)=O)(CO)CCN(C(=O)Cc2cnns2)CC1 47846,C(=O)(C1=NOC(C)C1C)NCCC(N1CC(OC)C(CC2CCCC2)C1)=O 47847,c1(C(=O)NC2CC(NC(=O)C=CC3CCCCCC3)C2)ccc2nnn(O)c2c1 47848,C1(C(N2CCOCC(F)(CNC(CCCC#C)=O)C2)=O)CC2(C1)CC21CCC1 47849,CC(CNC(=O)C(CC1CCC1)NC(=O)COC1(C)CCC1)C(F)(F)F 47850,C1(C(=O)NC(C)C(CO)NC(c2cnncc2O)=O)CN(C)CCN(C)C1 47851,CC1=C(C(=O)N2CCC(NC(C3(CCF)CC3)=O)C(C)C2)CCCO1 47852,Cc1nc(Cl)nc(N2CCCC(C(C)NC(=O)C=Cc3ccncc3)C2)c1F 47853,CCS(=O)(=O)CC(CO)NC(=O)NCCCc1scnc1C 47854,C1(C(N2CCC(C(C)CNC(C3CC3C(F)F)=O)C2)=O)CCC2(CC1)OCCO2 47855,Cn1cncc1C=CC(=O)NCCN(C(C1CC1c1cccnc1)=O)C1CC1 47856,C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC(CNC(Cc1ccc(C)s1)=O)C 47857,Cc1ncccc1OCC(=O)NCc1cc(C(=O)NOCCF)co1 47858,N12C(=O)CCC(C1=O)C2=O.c1(SCC)ccccc1CN1CC2C(C)C2C1 47859,c1(C(=O)NC2C(NC(C(C)(C)n3cc(Cl)cn3)=O)C2)cc(F)c(Cl)cc1Cl 47860,N1(C(c2[nH]cc(CC)c2)=O)CCCC(C)C1CCNC(c1cn(C)c(O)n1)=O 47861,CCCCC(CC)CC(=O)NCC1CCC2CN(C(c3ncc[nH]3)=O)CCC2C1 47862,C1(O)(CN(C(=O)COC2CCCC2)CC)CN(C(=O)CCC2CC2(F)F)C1 47863,CC(C)C(O)C(=O)N(C(C)CCNC(=O)CCc1cnco1)C 47864,C(C)(CCC(=O)NCCn1cnc(C(=O)NC(C)C(C)F)c1)SC 47865,C1(CNC(c2ccc(C)c(O)n2)=O)CC2COCC2N1C(=O)Cc1cccnc1 47866,c1(OC(C)C)ccc(C(N2CC(NC(c3coc(Cl)n3)=O)CC(O)C2)=O)c(Cl)c1 47867,C12(NC(C34CC(C#N)(C3)C4)=O)CCCN(c3ccn4nccc4n3)CC1C2 47868,Cc1cccc(CC(=O)NC2CCN(C(C)COc3cccc(Cl)c3)C2)c1C 47869,n1(C(=O)NC2C(SC)CN(C(C3(C(F)(F)F)CCCC3)=O)C2)nc(C)c(Cl)c1C 47870,CC1CC(C(N2CCCCC2CC2CCOCC2)C(=O)NC2CCOC2)CC(C)C1 47871,Cc1nc(O)c(C(=O)NCC(C)NC(c2c[nH]c(=O)cn2)=O)cc1Br 47872,N1(C(C(C(=O)OC)OC)=O)CC(NC(=O)CCc2cccc(F)c2Cl)C2(CC2)C1 47873,c1(C(=O)NC2CCN(C(c3cscc3C3CC3)=O)C2)ccc(SC(F)(F)F)nc1 47874,c1(OC)cc(Br)c(-c2ccc(C3OCCO3)cc2)cc1NC(N1CC(O)C1)=O 47875,C1(N(C(=O)CC2CCCC(=O)C2)C)CCN(C(=O)C(Cl)=CCl)CC1 47876,N1(C(CC(C)C2CC2)=O)CC(C(=O)Nc2cccc(O)c2)CC12CCC2 47877,Oc1cncc(Sc2ccc(SCc3ccnc(C4CC4)n3)cc2)c1 47878,N1(C(C(N2CC(C)CC(C)C2)=O)=O)CCn2c(cnc2C(N2CCOCC2)=O)C1 47879,N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)C=C1CCSCC1)C1CCC1 47880,CCC1(C(=O)NCC(O)CN(C(=O)Cc2cnc[nH]2)C)CCCc2ccccc21 47881,Cc1nn(CC(=O)NCC2(O)CCN(C(=O)CC3(C)CCC3)C2)c2ncccc12 47882,C1(C(=O)NC2C(CNC(c3cnoc3C3CC3)=O)C2)CC2(C1)CC2(F)F 47883,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)F)cc(Cl)c2n[nH]cc2c1 47884,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 47885,CC1CCC1C(=O)NC(C(=O)NC1CC(CCC(N)=O)C1)C1CCCO1 47886,c1(C(=O)NC(CC=C)CNC(=O)CC(=O)OC)ccc(Br)c(OC)c1 47887,CCCCCC(O)CC(=O)NC(CC(C)(C)C)C(=O)NCc1conc1C1CC1 47888,c1(OC)ccc(F)cc1CC(=O)NCC(C)(CO)NC(=O)CC1CC2(CCC2)C1 47889,Cc1ccc(CC(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)cc1Cl 47890,C1(CC(=O)NCCN(C(C)C)CC)CCCC1NC(c1sncc1C)=O 47891,Cc1cccnc1C(=O)N(CC(O)CN(C)C(c1cc(CC(C)C)nn1C)=O)C 47892,CC1(C(=O)Nc2cc(=O)n(CCF)[nH]2)CCN(C(C2CC2c2ccccc2)=O)CC1 47893,c1(C(=O)NC(C)CN(C)C(c2ccns2)=O)cc(S(=O)(=O)N(C)C)oc1C 47894,C1(CNC(CSC(C)C)=O)CC(F)(CNC(C2(CF)CCC2)=O)C1 47895,N1(C(C(=O)NC2CC2)=O)CCCC(F)(C(=O)Nc2cccc(CO)c2Cl)C1 47896,c1(CCC(=O)NCCCCNC(C2CCC2C2CC2)=O)c(Cl)cccc1Cl 47897,c1(C(=O)NCCC2CN(C(C3=C(C)OCC3)=O)C2)cc2c([nH]1)CCOC2 47898,N1(C(c2nc(COC)oc2)=O)CCC2CCN(C(=O)C(=O)NC3CC3)C2C1 47899,C(=O)(CS(=O)(=O)CCOC)N1CC(Cn2cc(CCCCCCC)nn2)C(C)C1 47900,C1(C=C)(C(N(C(C)COC)CC=C)=O)CCN(C(=O)Cc2ccsn2)CC1 47901,c1(C(N(C)CCN(C)C(c2snnc2C2CC2)=O)=O)cccc(S(C)=O)c1 47902,N1(C(c2c(CC)cccc2)=O)CC2CCCN(C(=O)C(C)c3ncco3)C2C1 47903,CN1CC(C(=O)NCC(C2CC2)NC(=O)Cn2ccnn2)NC1=O 47904,C(C(=O)NNC(=O)OC(C)(C)C)(C(C)(C)C)C(N(C)CC1CSC1)=O 47905,C12(NC(=O)Cc3cc[nH]n3)CC3CCC(C1C2)N3C(c1cc(Cl)cnn1)=O 47906,N1(C(C2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 47907,c1(C(=O)NC2CN(C(c3ccco3)=O)C3CCCC23)cc2ccnc(Cl)c2s1 47908,Cc1nc2cc(C(=O)NC3(CNC(C4CCN(CC(F)(F)F)C4)=O)CC3)[nH]c2s1 47909,c1(C(N(CCCCNC(c2cc(C(C)=O)on2)=O)C)=O)cc(C)c(Cl)cn1 47910,c1(N2CCC(F)(CNC(CC(C)(C)SC)=O)CC2)ncc(C#N)cc1F 47911,N1(C(=O)CCc2ccnn2C)CCCCC1CNC.C(=O)C1=CCCC1 47912,c1(CNC(C2CC(NS(=O)(=O)Cc3ccc(Cl)s3)C2)=O)ccccc1 47913,CCC(CNC(=NC)NC1CC2CCC1O2)(CC)c1ccccc1 47914,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 47915,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 47916,c1(C(=O)NCC2(N(C)C(C3CC3F)=O)CC2)cnc(C2CCC2)s1 47917,c1(CN2CCC(C)(C(=O)Nc3cnc(Cl)cc3C(N)=O)C2)ccc(F)c(C#N)c1 47918,C1(CNC=O)CCCCC(CNC(=O)CCSC)C1.CC(=O)COCC.C(C)(C)C 47919,c1(OC)ccccc1C(=O)NC1CCC(NC(c2cccnc2SC)=O)C1 47920,N1(C(c2c(COC)n(C)nc2)=O)CCCC2(NC(C3CCOC(C)C3)=O)CC2C1 47921,c1(C(N(C2CN(C(=O)CCC3CC3(C)C)CCC2O)C)=O)ccc2cccnn12 47922,c1(C(=O)NCC2(O)CCN(C(CC=CC=C)=O)CC2)cnc2c(C)cccc2c1 47923,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 47924,C1(C(=O)NC2CC2C)CC12CCN(C(=O)Cc1cccc(Br)c1)CC2 47925,N1(C(CC2CCC(C)O2)=O)CC2CCC1CN2C(=O)CCCC1CCOCC1 47926,C1(NC(CC2CC(CC)C2)=O)C2CC(NC(c3cc(C(N)=O)cs3)=O)CC12 47927,C1(C(=O)NCC2N(C(C(c3cccnc3)C)=O)CCCCC2)CCCCC1(F)F 47928,c1(C(=O)NC2CC(CNC(c3c(C)n(C)cn3)=O)C2)cccn2c(C)cnc12 47929,CC1(CCC(=O)Nc2cnn(C3COCC3N)c2)CN(N2CCOCC2)C1 47930,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 47931,C1(CNC(C(CC)(CC)CO)=O)CCN(C(C2(C(=O)OC)CC2)=O)CCC1(F)F 47932,CCCCCCC(C)C(=O)N1CCN(c2nc(-c3cc(Cl)cc(C)n3)no2)CC1 47933,Cc1nc[nH]c1CC(N1CCC(NC(c2ccc(C(F)(F)F)o2)=O)C1)=O 47934,c1(CN2CC(NC(CC(C)(C)O)=O)C(C)(C)CC2)ccc2cccnc2c1 47935,C12(CNC(C3CCN3C3CCCC3)=O)CCCC1N(C(C1OCCO1)=O)CCC2 47936,N1(C(c2c(C)sc(O)n2)=O)CCN(C)C(CNC(=O)C=CC(=O)NC(C)C)C1 47937,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2ccc(OC)nn2)=O)C1 47938,N1(C(C2CC3(CSC3)C2)=O)CCC2C(CCN2C(=O)CC2CC(F)(F)C2)C1 47939,CCCC(CNC(=O)CC(C1CC1)C1CC1)NC(c1ccccc1)=O 47940,C1(NCCC(=O)OCC(=O)OC2CCCCC2)CCCC(N2CCCC2=O)C1 47941,N1(C(C(CNC(C(C=C=C)C)=O)C)=O)CCN(C)C(C)C1 47942,c1(C(=O)NCC2(C)CCN(C(c3[nH]cnc3C#N)=O)C2)cnc2ccc(C#N)cn12 47943,Cc1cc(N(C2CCCCCC2)C)ncc1C(F)(F)F 47944,C(=O)(CC(C1CC1)C1CC1)NCC1CC1C(=O)NC(C1CCCCO1)C 47945,C1(C(=O)NCCP(C)(C)=O)CCC(C2CC2)N1C(C1CC(O)C(F)C1)=O 47946,N1(C(c2cn(CC)nn2)C(=O)NCCCC2CC2)CC2(CO)CC2(C(F)(F)F)C1 47947,C1(C(=O)NC2C(NC(C3(C)CCNC3=O)=O)CCCC2)CC12CCSCC2 47948,N1(C(C(CC)(C)C)=O)CCC(C2CC2)C1CNC(=O)CSc1ccccc1 47949,N1(C(c2c(C)nc(CC)s2)=O)CC(C2CN(C(C34CCC(O)C3C4)=O)C2)C1 47950,c1(CN2CC(CC(N3CCOC4CC34)=O)C2)cccnc1F 47951,C(=O)(C(C)CC(C)(C)C)N1CC(CNC(c2ccc(OC)nc2C)=O)N(C)CC1 47952,C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(C1CS(=O)C1)=O 47953,c1(CNC(C=C2CCC(C)CC2)=O)nc2c(s1)CCN(C(=O)Cc1ncc(Cl)s1)C2 47954,C(CC1CCC1)(C(=O)NCC1CCC1)N(CCCF)C 47955,N1(C(CCCCOCCC=C)=O)CC2CCN(C(c3cn(C4CC4)nn3)=O)CC12 47956,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 47957,C1(OC(C)C)CCCN(C(C2CCN(C(C3CCN(C)CC3)=O)C2)=O)C1 47958,C(=O)(CCCCCCC(=O)NCCCCCNC(c1ccc(Cl)cn1)=O)OC 47959,C1(NC(c2c(C)cc(C(N)=O)s2)=O)CC2CC(NC(=O)C(O)CC(C)C)CC2C1 47960,C1(NC(c2nn(C)c(-c3ccccn3)c2)=O)CC2CCC(C1)N2C(=O)C(Cl)(Cl)Cl 47961,C1(CNC(c2c(OC)c(O)nc(O)n2)=O)CCC2C(CC1)C2(F)F 47962,N1(C(c2cc(C)ncn2)=O)CCC(C2CCN(C(=O)Cc3ccccc3C)C2)C1 47963,C(=O)(N1CCCc2nncn21)C1N(C(=O)CCc2nccs2)CCOC1 47964,C1(CN=c2nncc[nH]2)N(NC(C2CCCN(S(CC)(=O)=O)C2)=O)CC12CCCC2 47965,Cc1n[nH]c(C)c1C(C)C(N1CCC(C)(CNC(=O)COCCN(C)C)C1)=O 47966,C1(CNC(Cn2nc(C)oc2=O)=O)CC(C(=O)NCC(C)F)=NO1 47967,CCC(C)(COC)C(=O)NC(C)C(CO)NC(=O)Cn1cccc(C)c1=O 47968,c1(C(=O)NC2CCC(CNC(c3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 47969,S(=O)(=O)(c1cc(Br)cc2c1OCC2)NCC1C(NC(Cc2ccc(C)cc2)=O)C1 47970,Cc1ccccc1CC(=O)NC(C1(O)CCN(C(=O)C#CC(=O)N(C)C)C1)C 47971,CC(C(=O)N1CCCN1C(=O)CC1CCCNC1)c1cc(F)cc(F)c1 47972,C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(CC(C=C)C)=O)C1 47973,C12(CCNC(=O)CCc3ccccc3)CCC1CN(C(=O)COC1CCOC1)C2 47974,c1(N(C)CC)nc(=NC)nc(N(CC(=O)Nc2cnc(CC(C)C)s2)C)[nH]1 47975,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 47976,O=C(C#CC1CCOCC1)N1CC(CNC(C2COCC2Oc2ccccc2)=O)C1 47977,c1(C(=O)NCC(C2CC2)NC(C(C(=O)OCC)OC)=O)cc(S(C)(=O)=O)oc1C 47978,C1(CC)CN(C(C2(NC(=O)C(C)(C)OC)CC2C)=O)CCC1CO 47979,c1(OC(C(=O)NC(CC)CCCNC(c2coc(Cl)c2)=O)C)ccc(Cl)cc1C 47980,CCCCN=C(NCC1CC(F)(F)C1)N1CCC(OCc2ccsc2)C1 47981,S(=O)(=O)(c1cc(-c2ccc(F)cc2)no1)N1CCC(c2cn(C)nc2)C1 47982,C#Cc1cccc(C(=O)NC(c2sc(C(C)C)nc2C)C(C)C)c1C 47983,c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc(C2(Cl)CC2)n(C)n1 47984,C(=O)(C(C)(C)C(=O)NCCC(C)(C)NC(=O)Cc1ncccc1C)N(CC)CC 47985,S(=O)(=O)(c1ccccc1COC)NCc1c(C(=O)OCC)c(Cl)nc(SC)n1 47986,CC(C)CC(O)C(=O)N1CCN(C(=O)Cc2cnc(F)c(Cl)c2)CC1C 47987,CC(C)CC(C)(O)CNC(=O)CC1(N(C(=O)C(c2ccn(C)n2)C)C)CC1 47988,c1(C(=O)NCCN(CC(C)O)C(c2ccc([N+](=O)[O-])[nH]2)=O)ncn2c1CCC2 47989,CCCC(CNC(c1coc(C(C)C)n1)=O)C(=O)Nc1cn(C)nc1O 47990,C1(CNC(COCCC#C)=O)C(C2CC2)CCN1C(c1cnc(CC)nc1O)=O 47991,C1(NC(=O)NCCOC2(C#C)COC2)CCC(N2CCN(CC)CC2)CC1 47992,C=CCCCCCCCC(=O)N1CC2(CCCC(CNC(C3(O)CCC3)=O)O2)C1 47993,Cc1cc(Br)ccc1-n1nnnc1C1(NCCCc2ccsc2)CCC(C#N)C1 47994,C(=O)(C1CCc2c(Cl)cccc21)NC1CN(C(C=C(CC)CC)=O)CC1C 47995,c1(COC)nc(CC(=O)NC(C2CCN(C(C3CC3(C)C)=O)C2)C)cs1 47996,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C)c(F)ccc(F)c1O 47997,N1(C(C2(CC(C)C)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 47998,C1(C)(C(=O)NC(C)(C)CNC(c2cnn(-c3ccccn3)c2)=O)CC=CCO1 47999,N1(C(C2C(C)C2C)=O)CCC(N(C(=O)Cc2nc(C3CC3)no2)CCO)CC1 48000,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48001,C1(NC(CCCOCC(C)C)=O)CCCC(C(C)(C)C)CC1 48002,C(C(=O)N1CCC(NC(c2cnccc2Br)=O)C1)(C(C)(C)C)NC(C)=O 48003,N1(C(Cc2ccn(CC)n2)=O)CC(C(=O)NC(C)(CO)C(C)C)C2(CCC2)C1 48004,C(CO)(C(=O)NC(C)C=CC(=O)NCCNC(C)=O)N(C)CC 48005,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48006,C1(CC)CN(C(C2CCN2C(=O)COCC2CCCO2)=O)CCO1 48007,C1(Cl)(C(=O)NCCN(C(c2nocc2C2CC2)=O)CC)CC12CCC2 48008,N1(C(CC(C)c2ccco2)=O)CC2(CCCC(CNC(C3(C)CC3)=O)O2)C1 48009,c1(C(=O)NCC2(F)CCCN(C(C3CC4CC3CN4)=O)C2)cc2n(n1)CCCC2 48010,C=CCC(CC)C(=O)NCC=CCNC(C1CCCN1C(c1ccc(C)cc1)=O)=O 48011,c1(CC(=O)OCCC(CCC)C)ccc(C(F)(F)F)c(F)c1 48012,c1(OCC#C)ncccc1C(=O)NC(C)C(CO)NC(c1[nH]c(C)nc1C)=O 48013,Cc1nccc2c(=O)c(C(=O)NCC3C(C)CCN3C(=O)CC(C)C)c[nH]c12 48014,c1(C(=O)NCC(C)NC(=O)CCCN(C)C)cccc2cncn12 48015,c1(CC)nc(C)c(C(=O)OCCCCCCC2CN(C(=O)CN3CCCC3)C2)o1 48016,C(N=c1[nH]c(=NC(C)Cn2ccnc2)c2c(ncn2C)[nH]1)c1cccc(C)c1N 48017,C1(CCNC(CC2C(C)C2(F)F)=O)CN(C(c2cnn(C)c2C2CC2)=O)CCO1 48018,Cc1cn2c(n1)CCC(CNC(=O)NC(c1ccccc1)C(N)=O)C2 48019,C(=O)(CN=c1cc[nH]cc1)NC1(C2N(C(c3c(C)snn3)=O)CCC2)CC1 48020,C(CCCC(=O)NC1CCOC1C(=O)NOCCC(C)O)(OC)OC 48021,c1(C(N(CCCNC(=O)CCCC2CC2)C(C)C)=O)c(F)ccc2cnn(C)c12 48022,C=C1CCC(C(=O)NCC2CC2NC(c2ccsc2-n2cnnn2)=O)CC1 48023,Cc1csc2c(N3CCC(O)C3)ncnc12.N1(C(=O)NCC)CCOCC1C1CC1 48024,C(=O)(C(O)CCC(F)(F)F)NC1C(CC(N2C(C(=O)NC)CC2)=O)C(O)C1 48025,C1(C(=O)NCCCOCCCNC(CSC(C)C)=O)CCc2nncn2CC1 48026,C1(C(=O)NC2(C)CCC2)CC12CCCCC2.O1NC(=O)C2CC(C2)C1 48027,c1(OC(C(=O)NCC2(CNC(C=CC)=O)CCCCC2)C)cccc(Cl)c1Cl 48028,C1(N(C(C(C2CN(C=O)C2)OC)=O)C)CCCC(=O)C1.C(CCN=[N+]=[N-])N 48029,N1(CC(COCC(C)C)O)CCC(C(N2CCCC2)=O)CC1 48030,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(c2c(C)coc2)=O)(CF)C1 48031,C(C1CCCCCC1)=CC(=O)NC1CCN(C(CC2CCCN(C)C2)=O)C1 48032,N1(C(CCOC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48033,Cc1ccc(C)c(C(=O)NC(C23CC(C(=O)O)(C2)C3)C)c1O 48034,c1(C(=O)NCC2C(C=C)OCC2)c(C)sc2c(Br)cccc12 48035,c1(NCCC)ncccc1S(=O)(=O)NCCC(c1ccccc1F)CN(C)C 48036,CC1(CNC(C2CC(C#N)(OC)C2)=O)CN(C(=O)CC2CCC3CC3C2)CCO1 48037,C1(C(=O)NC2(CNC(C3CC3C(F)F)=O)CCCCCC2)C2CCC3C(C2)CC13 48038,c1(C(=O)CF)ccc(CNC(=O)C(c2cnn(C3CC3)n2)=O)cc1 48039,C12(C(N)=O)COC(CCN1Cc1n[nH]c3cccnc13)C2 48040,c1(C(N(C)CC2CN(C(C3C4COCC34)=O)CCO2)=O)ccc2c(c1)CCN2C 48041,N1(C(CC(CCC)O)=O)CC2CCC(C1)C2NC(c1csc(C)n1)=O 48042,c12cnc(F)c(c1)-c1nn(C3CC3)cc1C(=O)O2.c1(OC)cccc(CSC)c1 48043,C1(N(C(c2c(CC)ccs2)=O)C)CCCCN(C(=O)Cc2ccnc(O)c2)C1 48044,Cc1ccc(F)cc1NC(=O)C(C1CCCN(C(=O)CCc2ccnn2C)C1)C 48045,N1(C(c2cc(OCC)n[nH]2)=O)CCCC(NC(c2cc(OC)ncn2)=O)C1C 48046,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC1C(NC(C(C)O)=O)COC1 48047,C1(CC)CN(C(=O)CCC(C)(C)C)CCC1NC(C1CCCC1OC)=O 48048,CCC(C)(COC)C(=O)NC1CC(O)CN(C(=O)CCC(=O)c2ccccc2)C1 48049,c1(N2CC(COC)OCC2)nc2c(c(=NCCCC3CC3)[nH]1)CCCCC2 48050,C1(NC(C2CCc3c[nH]nc3C2)=O)CCN(C(C2C=CC=CC=C2)=O)C12CCC2 48051,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48052,c1(NC(C2CCCN(C(CCCCOC)=O)C2)=O)nccc(Br)c1O 48053,C(=O)(C(C)CS(C)(=O)=O)N1CCC(O)(C(C)NC(CC(=O)NCC)=O)C1 48054,c1(C(=O)NCC2CCN(C(CCC(CC)OC)=O)C2(C)C)ccc(F)c(C)c1O 48055,N(C1CCCc2c[nH]nc21)C(C(CC1CC1)NC(c1cccc(OC)c1)=O)=O 48056,C1(CNC(C2(C)CCCO2)=O)CC2(CC2)CN1C(c1ccc(N)cn1)=O 48057,c1(N2CCC(C)(CC)C2)ccc(Br)c(S(=O)(=O)NCC2C=CCC2)n1 48058,N1(C(=O)OCC)CCCC(NC(C2CC(NC(c3ccncc3)=O)C2)=O)C1 48059,CS(=O)(=O)c1nc(Cl)cc(=NC2CCCCC2NC(C2CCCOCC2)=O)[nH]1 48060,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48061,C(=O)(C(F)C(F)(F)F)NC1(C(F)F)CC(NC(C2C(C)CCO2)=O)C1 48062,c1(C(N(C)CCNC(=O)Cc2ccc(CO)cc2)=O)sccc1S(C)(=O)=O 48063,C1(NC(c2nncs2)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48064,CCCC(CC)C(=O)N(CC(=O)Nc1ccc(O)cc1Cl)C 48065,c1(C(N2C(CN(C(C(C)n3ccnc3)=O)C)COCC2)=O)ccn2c1CCCC2 48066,N1(S(=O)(=O)c2cccnc2)CCC2(CC1)CN(CC1Cc3ccsc3N1)CCC2O 48067,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CC2CCN(C)C2)C12CCC2 48068,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(=O)CC2CCOC2)C1 48069,N1(C(C2(CNC(c3c(CC)c[nH]c3)=O)CCCCC2)=O)CCCC1(C)C=C 48070,C1(C(=O)NC(CNC(Cc2cnc(C)s2)=O)C)CCc2nnc(O)n2C1 48071,C(CC(O)C(=O)NCCC1CCN(C(=O)CCOC2CCN(C)CC2)C1)SC 48072,C(=O)(C(O)C(C)(C)C)N1CCN(C(CNC(C(C2CCC2)OCC)=O)C)CC1 48073,c1(OC(C)C(=O)NC(CO)C(C)NC(C2CC2(F)F)=O)cccc(CO)n1 48074,C1(C(=O)NCC(C)(F)CNC(C2CC(F)C2)=O)CCOC1(C)C 48075,CC(C)(C)CC(C)(C)NC(C1CC(O)(CNC(=O)Cn2cccn2)C1)=O 48076,C1(C(=O)Nc2cc(C)sc2)CN(C)CCN1C(C1CC(C2CC2)=NO1)=O 48077,c1(OC)cc(NC(C2(F)CCN(C(c3scc(C)c3C)=O)C2)=O)cc(C)n1 48078,C(=O)(CCC(=O)C1CC1)N(CCC(=O)NCCC1CCCOC1)CC 48079,C(=O)(C(CSc1ccccc1)Cc1ccccc1)N(CCNC(C(CC)O)=O)C 48080,c1(OC)cc([N+](=O)[O-])ccc1NC(=O)NC1(C(C)Sc2ccc(OC)cc2)CC1 48081,N1(C(=O)NOCc2cn(CCc3ccccn3)nn2)CCOC(c2ncc[nH]2)C1 48082,C1(NC(CN(CCC)C)=O)CCN(C(c2cccc(N)c2C)=O)CC1O 48083,CN1CC=C(CC(=O)N2CCC3CCN(C(c4cc(C(N)=O)co4)=O)CC23)CC1 48084,c1(C(C)OC)nc(CCc2ccc(OC)cc2)n(-n2c(C)ncn2)n1.c1ccccc1 48085,C1(CNC(c2ncc(CC)s2)=O)CC2CCCC2N1C(c1cc(C2CC2)ns1)=O 48086,N1(C(C(CSC)OC)=O)CCC(C2CCN(C(c3cnc(C(C)C)s3)=O)CC2)C1 48087,N1(C(C2(C)C(CC)CCC2)=O)CCCCC(CNC(=O)Cc2nnc(S)n2C)C1 48088,C(=O)(CC(O)CN(C)C)NCC(CNC(Cc1cnc(C)s1)=O)(C)F 48089,C(CC(N)=O)(c1ncccn1)N(C)C(=O)Nc1csc(C(N)=O)c1 48090,N1(C(C(CCOC)C)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)C12CCC2 48091,C1(COC)(NC(=O)CNC(c2cccs2)=O)CN(C(c2cocn2)=O)C1 48092,NC1(C2CCN(C3CCN(C(C4CCCCC4)=O)C3)CC2)CC1 48093,C(=O)(CCS(=O)(=O)N1CCOCC1)N(C1(C)CN(C(=O)C=CC=C(Cl)Cl)C1)C 48094,C1(CC)CCCCC1CNC(c1cn(C)c(O)n1)=O 48095,c1(C(=O)NC2CCC(CCNC(Cn3c(C)ccn3)=O)C2)ccnc(C(C)C)c1 48096,C1(C(=O)NC2(C)CN(C(c3cc(C)on3)=O)C2)Cc2cc(F)cc(F)c2O1 48097,C(CC(C)C)(CS(C)(=O)=O)N.n1(CCCN(CC)CC)cc(C(F)(F)F)cn1 48098,C1(NC(c2c[nH]nc2-c2ccncc2)=O)CCCCN(C(=O)C(F)(F)CF)C1 48099,Cc1ccc2c(N(CC(=O)N(C)C)C)nc(=NCCn3cccn3)[nH]c2c1 48100,CC#CCC(C(=O)NC1(C)CC(=C)C1)NC(c1ccc(Cl)cc1)=O 48101,c1(C(=O)Nc2c(C(N3C(C(=O)NC)CCC3)=O)scc2)cc(=O)n(C)cn1 48102,c1(C(=O)OC)c(C(=O)NCCCN(C(=O)CN(C)C(C)=O)C)n[nH]c1C 48103,C1(OC)CC(CNC(C2(C)CC(C)(C)C2)=O)N(C(=O)CC2CCOCC2)C1 48104,N1(C(Cn2ccc(C)n2)=O)CCCC12CCCN(C(=O)C(C)CC(C)C)C2 48105,C12(C(N(CCCC=C)C)=O)C(NC(C3CCN(C(C)=O)CC3)=O)C3CC1C2C3 48106,c1(C(=O)NCC2(O)CCCN(C(COC(CC)(C)C)=O)C2)ccc(C#N)c(O)c1 48107,C=CC(C)(C)C(=O)N(CCCNC(=O)C(N1CCCCCC1)C)C 48108,Cc1nc2ccccc2cc1C(N1CCC1NC(c1ccc(N)c(C)c1C)=O)=O 48109,CN1CCCC(CCC(=O)NC(C)(C)CN(C)C(c2cc(Cl)ns2)=O)C1 48110,c1(C(=O)OC)ccc(NC(c2ccc(Cl)o2)=O)cc1O.C12CC13CCN(C3)C2=O 48111,C1(F)(CNC(CSC)=O)CCCN(C(c2ccc(F)cc2F)=O)CC1 48112,Cc1cc(C(=O)N(C(C)(C(=O)N2CC(OC(=N)O)C2)C2CC2)C)nn1C 48113,n1(CC(=O)NC(CN(C(c2cnn(COC)c2C)=O)C)C)nc(C)c(Cl)c1C 48114,C1(C(=O)NC(COC)CCO)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48115,N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(=O)C(c1ccc(Cl)cc1F)(C)C)C2 48116,C12(COC)CC(CN1CC1C(O)CCN1C(=O)OC(C)(C)C)C2 48117,C=C(CNC(C1CC(C)CO1)=O)CCNC(=O)COCCCOC 48118,N1(C(C2C(C)(C)NC(=O)C2)=O)CCC=C(C(=O)NC2CCCC2(F)F)C1 48119,Cc1ccc(F)c(C(N2CC(F)(F)CC2CNC(C2CC(C)(C)CN2C)=O)=O)n1 48120,C1(C(NOC(c2nc[nH]n2)=O)=O)CCCCCN1C(C12CCCCC1C2)=O 48121,c1(C(=O)NC2C(NCCCC(=O)OC(C)(C)C)CCCC2)ccc(F)c(Br)n1 48122,C1(CC(=O)N(CC(C(=O)NCC(C(=O)NC)O)C)C)NC(=O)NC1=O 48123,CC1=C(C(=O)NC2CCCCC2N(C)C(C2CCOC2(C)C)=O)CCS1(=O)=O 48124,C12(C(N3CC=C(CNC(=O)CCC4CCOCC4)CC3)=O)CCCN1CC(O)C2 48125,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48126,c1(C(=O)NC2C(C)(C)CN(C(C3(F)CCOC3)=O)C2)c(F)ccc2occc12 48127,C(C(C)(CC(C)C)NC(=O)C(C)N(C)C)NC(C1(CC)CC1)=O 48128,Cc1c(C(=O)NC2CC2NC(c2ccc(C(F)F)o2)=O)cnn1C1CC1 48129,c1(C(=O)NC(C(=O)NCC2(N(C)C)CC2)C2CCOC2)ccc(C#N)cc1 48130,C=C(CNC(=O)C(CC(F)F)NC(c1cccc2occc12)=O)C1CCOCC1 48131,C12(C(=O)N(CC(=O)NCC(O)C3CCC3)C3CC3)CCC(CO)(CC1)C2 48132,N1(C(C23CC(F)(C2)C3)=O)CCC12CN(C(C13CC(O)C1C3)=O)C2 48133,N1(C(c2n(C)ccn2)=O)CCC(C2CCN(C(c3cnco3)=O)CC2)C1 48134,N1(C(=O)NC2C(C)CC(Cc3cccnc3)C2)CCCCC12CC2 48135,C1(C(=O)NC2CCC(N(C)C)C2)CCC2(CC2)N1C(c1nc(CO)n[nH]1)=O 48136,N1(C(C(=O)NCCc2cc3c(cn2)OCCC3)=O)CCC2(CC1)OCC1CC21 48137,c1(N2CCC(CNC(CNS(NC)(=O)=O)=O)CC2)nccc(CN2CCCCCC2)n1 48138,c1(OCCC)cccc(NC(=O)C(N2CCCCC2CNC(C2(C)CC2)=O)=O)c1 48139,c1(C(=O)NC(CN(C(=O)C(C)(C)CF)CC)C)c[nH]c2cc(F)ccc12 48140,CN=c1nc(N2CCC(c3ccc(C(=O)NC(C)CC#N)cc3)CC2)cc(C)[nH]1 48141,N1(C(C2CC(=C)C2)=O)CCC2OCCN(C(c3ccc(SC)cc3)=O)C2C1 48142,N1(C(C=CC)=O)CCCC2(CCC2NC(C2CCCCO2)=O)C1 48143,c1(C(C)OC)nc(C(N2CCC(NC(c3ncoc3C3CCC3)=O)C2)=O)cs1 48144,c1(C(N2CC(C)C(CNC(=O)C(F)n3cccn3)CC2)=O)cncc([N+](=O)[O-])c1 48145,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48146,N1(C(c2c(C)occ2)=O)CC2C(NC(C3(c4ccc(F)cn4)CC3)=O)C2C1 48147,C1(C(=O)NCCC(C)OC)CCN(C(c2cn[nH]c2)=O)C12CC2 48148,C1(c2n(CC(C)(C)SC)nnn2)(Nc2cncn2C)CCOCC1 48149,C1(=O)C(Cc2ccoc2)NC(=O)C(F)=C(C)CN1.C(CCO)CC#C 48150,c1(CC)nnc(N2CC(O)(C(C)NC(C3(C)CC3)=O)C2)c(C#N)c1CC 48151,C1(CNC(C=CSC)=O)CC2CCC(C1)N2C(C1(C(N)=O)CC1)=O 48152,CC1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CN(C(c2cccnn2)=O)CCO1 48153,c1(C)ccccc1C.c1(CC(=O)NC2CCC(CN(C)C=O)C2)cn(C)nn1 48154,c1(C(=O)NCC(CC2CN(C(CCCCC)=O)C2)(C)C)ccc2oncc2c1 48155,c1(N(C(C=CCOCCOC)=O)C2CC2)cc(C)ccc1C.C1CCO1 48156,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)CC(O)C1 48157,C1(CNC(C(C)NS(C)(=O)=O)=O)C2CC2CN1C(=O)Cc1ccccc1 48158,N1(C(C2(C)CCN(C(Cc3nc(CCCC)[nH]c3Cl)=O)C2)=O)CC2CCC2(C)C1 48159,C1(C(N2C(C)C(NC(C3C4COCC34)=O)CCC2)=O)CCC(C2CC2)CC1 48160,S(=O)(=O)(c1ccc(NCCC(O)C2CCC2)c(C#N)c1)N1C(C)CN(C)CCC1 48161,CC1CSCCN(C(=O)CC2CCCC(NC(=O)C(c3ccnn3C)O)C2)C1 48162,C1(NC(C2(NC(C3CC(C)OC3)=O)CC2)=O)CC(C)(C)C12CCC2 48163,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48164,c1(OC)cc(C(=O)NC2CN(C(c3cocc3C)=O)CC2F)cc2nc(O)[nH]c12 48165,c1(C(=O)NC2CC3(C(NC(CC4N(CC)CCC4)=O)C3)C2)ccn2c1CSCC2 48166,c1(NC(C2NCCN(C(c3ccc(SC)s3)=O)C2)=O)cc(C)cc(Br)c1F 48167,Nc1ccc(C(=O)NC2CCN(C(c3ncc(F)cc3F)=O)CC2CO)nc1Cl 48168,C=Cc1cnn(C)c1C(N1CCN(C(C2(C)CC2(Cl)Cl)=O)C(C)C1)=O 48169,N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)CC2CC(C)C2)C2COCC12 48170,N1(C(CSCC)=O)CCC(NC(C2CC(c3ccccc3)CNC2=O)=O)C(O)C1 48171,CC1CN(C(=O)Cc2ncn3c2CCC3)CCCN1C(=O)Cc1cccc(Cl)c1 48172,N1(C(C2OCCN(CC)C2)=O)CCN(C(c2scc(C)c2C)=O)CCC1C 48173,C(=O)(C1=C(Cl)CCCC1)NCC1N(C(C2(N(C)C)CCCCC2)=O)CCC1 48174,CCCC(C)(O)CC(=O)N1CC(O)CCC1C(N1CCCC(N(CC)CC)C1)=O 48175,N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NCCC#N)CCC=C(C(=O)OC)C1 48176,c1(-c2c(OC)ccs2)nc(CCCO)nn1CCCO 48177,c1(CNC(CCC2N(C(Cc3nc(=N)[nH][nH]3)=O)CCC2)=O)cccnc1F 48178,N1(C(C=C(CCC)C)=O)CC2C(NC(=O)Cc3coc(-c4cccs4)n3)C2C1 48179,Cn1nnc2c(Cc3cn(CC4CCC(F)CC4)nn3)ccnc12.C12CCN1C2 48180,c1(C(N(CC(CC)NC(c2cocc2C(N)=O)=O)CC)=O)c(C)cccc1Br 48181,N1(C(CSCC#C)=O)CCC(F)(CNC(C2CC2OC(C)(C)C)=O)CC1 48182,Cn1nc(Br)cc1CC(=O)NCC1CCCN1C(c1n[nH]cc1F)=O 48183,C(N=c1[nH]c(=NC(C)C(C)CC)c2c(ncn2C)[nH]1)c1n(CCC)ncn1 48184,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48185,C1(OCC(=O)Nc2ccsc2C(=O)O)CCS(=O)(=O)C1 48186,C1(C)(NC2(CO)CN(C(c3cc(OC)ncn3)=O)C2)CCC(=O)NC1 48187,c1(NC(=O)NCCC(C)CCC2CC(OCC)C2)cc(C)nc2c1nc(C)n2C 48188,c1(C(N2CC(OCCNC(CC3C(C)CCC3)=O)C2)=O)nccc(F)c1Cl 48189,C1(N(C(C2(C#C)CN(C(C3CC(C)(C)C3)=O)C2)=O)C)CCOC(C)(C)C1 48190,C(C1OCc2ccccc21)Sc1ccc(F)c(F)c1F.O=C1CCN2C(=O)N1C2 48191,C1(CCOC)(NC(c2cc[nH]c(=N)c2)=O)CCN(C(=O)CC2CCOCC2)CC1 48192,C1(NC(c2ccc(C)cc2F)=O)CCC2CCN(C(C3CC4(CC4)CO3)=O)C2C1 48193,c1(NCC(=O)OC2CCSCC2)cccc(-n2nnnc2O)c1 48194,N1(C(C2C(C(=O)OC)C2)=O)CC2CCN(C(=O)CC3CCC(F)(F)C3)CCC2C1 48195,CC1(NC(c2nccnc2Cl)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 48196,C12(C(N3C(CCNC(c4cnc(COC)s4)=O)COCC3)=O)CCCC1OCC2 48197,C1(CCC#C)CCCN(C(=O)C(CO)NC(C2C=CCCC2)=O)C1 48198,N1(C(COC(C)(C)C)=O)CC(C(=O)NCC2CCOC2=O)CC12CCC2 48199,c1(C(=O)OC2CCN(CC(=O)N(CC(C)C)C)CC2)sc2cc(F)ccc2c1C 48200,c1(CC(=O)NC(C)C(CO)NC(=O)Cn2nnc(=O)[nH]2)coc2ccc(F)cc12 48201,c1(C(=O)NC(C2(O)CCN(C(C3(CF)COC3)=O)C2)C)ccc2c(c1)CCCO2 48202,N1(C(CC=C=C)=O)CC(NC(=O)C(CC)CC)C(S(C)(=O)=O)C1 48203,CCCCCC(C)(C)C(=O)NC1CN(C(=O)Cc2c[nH]c3cccnc23)CC1O 48204,CC1CN(C(C2CCC(NC(C3CN(C4COC4)C3)=O)C2)=O)CCS1(=O)=O 48205,c1(OC)ccccc1NC(=O)CC1(C)CN(C(C2(c3ccncc3)CCC2)=O)C1 48206,C(=O)(CCCCCC(C)C)N1C(C)CCC(NC(C2(CC)CC(C)(C)C2)=O)C1 48207,N1(C(COCC)=O)CCc2nc(C(=O)NCC3CCC3)cn2CC1 48208,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48209,Cc1cc(C(=O)NCC2(C)CC(NC(=O)C=CC(=O)N(C)C)C2)sc1Br 48210,Cc1ccc(C(N2CCN(C(=O)C(C#N)CC3CC3)C(C(C)C)C2)=O)nc1O 48211,Cn1ncc(SC2CC2)c1C(N1CC=CC(NC(C2(C(F)F)CCC2)=O)C1)=O 48212,C1(CC2(NC(=O)OC(C)(C)C)CCCCC2)CCN(C(=O)OC(C)(C)C)CC1(C)C 48213,c1(N2CCN(CCF)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48214,c1(C(N2C3CN(C(c4c(F)ccc(C)n4)=O)C(C3)C2)=O)c(N)cc(Cl)cc1Cl 48215,C1(F)(C(N2CCC(NC(Cc3c(C)con3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 48216,C(=O)(C#CC1CCCOC1)N1CC(C)C(CNc2ncnc3[nH]cnc23)CC1 48217,Cc1cc(F)sc1C(=O)NCCCC(=O)NCC(C)CC1CCCC1 48218,C1(NC(=O)CSC2CC2)CN(C(=O)C(O)CC2CCOCC2)Cc2ccnn2C1 48219,c1(OC)ccc2c(c1)N(C(c1cnn(C)c1)C(=O)NC(C)(C)C)C(C)(C)C2 48220,c1(C(=O)NCC2CC(NC(c3nnc(C)s3)=O)C2)cnc2c(c1)CCC2 48221,c1(CCC(=O)N(CC(C2CC2)NC(C2CCO2)=O)C)cncc(O)c1 48222,N1(S(CC)(=O)=O)CCCC1C(N1CCC1CNC(=O)CCOCCN(C)C)=O 48223,CCCCCCC(=O)N(CCCN(C)C(c1sccc1CN(C)C)=O)C 48224,C(=O)(CCCc1cc[nH]n1)NC(C1CCCN1C(=O)Cn1nccn1)C 48225,Cc1cc(C(=O)NC2CCCC(NC(=O)CCCN(C)C)CC2)c(O)c(C)c1 48226,c1(OC)cccc(C)c1C(N1CC2C(NC(=O)CCN3CCN(C)CC3)C2C1)=O 48227,N1(C(COCC)=O)CCCC2(CCC(NC(=O)COC)C2)C1 48228,C1(NC(C(CC)OC)=O)CCN(C(c2scnc2C(C)C)=O)C12CCC2 48229,n1(CC(=O)OC(C2CC(O)(C(=O)O)C2)=O)ccccc1=O 48230,C(C)(C(C)(C)C(=O)NCC1(n2ccnn2)CC1)NC(Cn1c(C)nnn1)=O 48231,C1(OC)(CNC(C2(Nc3cccc(Cl)c3)CC2)=O)CCN(C(=O)CCCSC)C1 48232,c1(C(N(CCN(C(c2cc(C)[nH]n2)=O)C)C(C)C)=O)ccnc(C(C)C)n1 48233,c1(C(N(C(C(CCC)C)=O)c2cncnc2C(F)(F)F)=O)ccc(Cl)cc1Br 48234,c1(C(=O)NCCCN(C(=O)COc2cccnc2)C)ccc2cccnc2c1O 48235,CC1CN(C(c2nnn(C)c2C(F)(F)F)=O)CCC1NC(C1CS(=O)C1)=O 48236,C#CC1(O)CCN(C(C2CCCC(NC(=O)CNC(=O)NC)C2)=O)C1 48237,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48238,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1ccc(CO)cn1)=O 48239,CC(C(C(=O)Nc1ccccn1)NC(=O)OC(C)(C)C)NCC1CCCS1 48240,C=CCC(CC)C(=O)NC(CCN(C)C)C(=O)NCCN(CCC)C1CC1 48241,c1(N(CCOC)CC)ncnc2c1ncn2CC(C1(O)CCCCC1)(C)C 48242,C12(C(=O)OC)CCCC1(C(=O)O)CN(CC(=O)N(C(O)CC(C)C)CCO)C2 48243,c1(C(C(=O)NCC(C)(O)CNC(C2(CC)CC2)=O)O)cccc([N+](=O)[O-])c1 48244,CC1CCCCCCC1NC(=O)CN(C=O)C.C(C)(=O)ONC 48245,c1(C(=O)NC(C)CNCCCC(=O)NC23CCC2C3)ccc(N(C)C2CC2)cc1 48246,c1(C(=O)OCC)cn(C)[nH]c1=NC(=O)CN(C)Cc1cccc(Br)c1 48247,c1(CNC(N2CC3C(C(=O)OC)C3C2)=O)c(-c2ccccc2)nn(C)c1C 48248,N1(C(COC)=O)CC(CNC(c2c(F)ccc(Br)c2F)=O)C2(CCC2)C1 48249,c1(C(N2CC(CN(C(=O)CSCC(N)=O)C)C2)=O)cnc(C(F)(F)F)c(F)c1 48250,C(=O)(C1=CCN(C(C2CCN(C)C2=O)=O)CC1)N(C(C)C1CC1)C1CC1 48251,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48252,C(=O)(CC(CC)C(C(=O)COC)CC)N(CCC)CCN(C)CC 48253,C12(CC(F)(F)C1)CN2.c1(C(N2CC(CNC(CSC)=O)C2)=O)nc(C)sc1C 48254,CCC(CCOC)C(=O)N1CC(CC(C)NC(=O)CC2CCC2OC)C1 48255,N1(c2cc(COC)ncn2)CC2(C1)SCCC2NC(=O)Cc1cnns1 48256,c1(CC)ccc2c(c1)NC(=O)NC1(CCC1)C(=O)OCC2.OC 48257,C1(C)(CC)COCCC1n1cc(CS(=O)(=O)CCCNC(=O)CN(C)C)nn1 48258,N1(C(C(CC#C)(C)C)=O)CC2CCC(CNC(=O)C(CC)SC)C2C1 48259,c1(C(N2CCOCC(O)C2)=O)cccc2c1CCN(c1ncnc3[nH]ccc13)C2 48260,c1(C(=O)NCCCNC(=O)CC2CC(C(F)F)(OC)C2)c(C(=O)OC)cnn1CC 48261,Cc1cc(=NC(=O)CCNC(c2cc3ccccc3o2)=O)[nH]n1CCO 48262,C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(c2ccccn2)=O)C13 48263,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)CC(F)(F)C2)cnc2ncnn2c1C 48264,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48265,CCC(C)(C(=O)N1CCC(N(C(=O)C(O)CC2CCOCC2)CCO)C1)OC 48266,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(Cl)ccc(OC)c2)=O)CC1 48267,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(C(F)F)nc1)=O 48268,C1(=CCNCC(C)Cc2ccc(C(C)(C)C)cc2)CCN(C(=O)C(C)(C)C#N)CC1 48269,C1(C(N2C(C)CCN(C(C3CCC(=O)N3)=O)CC2)=O)CC(F)(F)CCC1(C)C 48270,N1(Cc2ccccc2)CCN(CCc2nnnn2CC2CC2)CC1.c1(CC)ccccc1 48271,C1(C(N(C)Cc2cscn2)=O)CCCCC1NC(C1CNC(=O)C1)=O 48272,c1(C(=O)NC23CC(CNC(C(C)(C)SC)=O)(C2)C3)ccnc2nc(=N)[nH]cc12 48273,N12CCC3(CC1)CC(C)N2C3.c1(C=O)ccccc1SC(F)(F)F.CSC 48274,C(=O)(C(C)CC(C)CC(C)C)NC1CN(C(C(C(CC)(C)C)O)=O)CC(C)C1 48275,CCC(CC(=O)NC1CC(NC(c2cc(COC)[nH]n2)=O)C(O)C1)C(C)C 48276,CC(C(=O)NC1CC(N(C(=O)CCS(C)=O)C)C1)C(=O)N1CCS(=O)(=O)CC1 48277,C1(NC(C(C2CCC2)NC(c2ccc(C(C)C)o2)=O)=O)C2CCN(CC2)C1C 48278,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48279,C(C1CSc2ccccc21)NC1CCC(Cn2cc(CCC(=O)NC)nn2)C1 48280,c1(CNC23CCC(NC(C=CC)=O)(CC2)C3)cc(F)cc([N+](=O)[O-])c1 48281,C(C)(C(=O)N(CCC(=O)NCC(C)Cc1cn[nH]c1)C)OCCOC 48282,C=CCC(CNC(c1cc(Cl)no1)=O)C(=O)NCc1cc(C)cc(O)c1 48283,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48284,Cc1cn(C(C)C)cc1C(=O)N(CCC(C)NC(=O)CCC1CC(C)(C)CO1)C 48285,c1(C(CNC(C)=O)NC(C2(NC(C)=O)CCOCC2)=O)cc(F)c(Cl)cc1F 48286,Cc1cc(C(N)=O)sc1C(N1CC(C)C(F)C1)C(=O)Nc1ccccc1 48287,Cc1ccnc2c1OC(C(N1CC3(CCN(C(c4ncc[nH]4)=O)C3)C1)=O)C2 48288,C1(CC(N2CC(CC(C)(C)CNC(=O)Cn3cnnc3O)C2)=O)CCC=CCC1 48289,Cc1ccc(-c2ccc(NCc3scnc3C)cn2)cc1Br 48290,C1(NC(c2ccc(C#C)nc2)=O)CN(C(C2(C)CCC2)=O)CC12CCC2 48291,N1(C(=O)NCc2ccc(OC(C)C)nc2)CCC(O)C2(CCC2)C1 48292,Cc1ccc(C)n1CCC(N1CCC=CC1C(=O)NCc1cnsc1)=O 48293,N(C(=NCC1(NCc2ccon2)CCC1)N1CCC(N2CCCC2)C1)C(C#C)C 48294,c1(CNC(=O)NC(COCC(=O)OC)=O)cn(CCc2ccccn2)nn1 48295,N1(CC(=O)NCCCC(C)NC(c2sccc2F)=O)CCCC(N(C)C)C1 48296,CC1CCC(C)N1CC(=O)NC1(C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 48297,N1(C(C(C=CC)O)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC(F)(F)F)C2)C1 48298,CC(C)CCCCCCNC(C1CC1C1CN(C(=O)CC2CC(=O)NC2=O)C1)=O 48299,c1(CN(C)C(c2cnnc(O)c2)=O)ccccc1CNC(C1CC2(CCO2)C1)=O 48300,CCC(CC)(C(=O)Nc1ccc(OC(c2ccncc2)=O)c(Cl)c1)OC 48301,N1(C(Cn2nc(C)n(C)c2=O)=O)CCN(C(=O)CSc2nnc(S)s2)C(C)C1C 48302,CC#CCC(C(=O)N(CC(O)COC)C)NC(=O)Cc1cccs1 48303,C(CCCCC(=O)NC(C(=O)NCCCc1ncc(C)o1)C1CCCO1)OC 48304,c1(NC(c2c(C)ccnn2)=O)cnc(Cl)cc1C(N1CCNC(=O)CC1)=O 48305,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48306,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CC(O)CCN(C)C)CCC1 48307,c1(CC(=O)N2CC2)n[nH]c2cc(-c3cccc(Cc4ccc(Cl)cc4F)c3)ccc12 48308,C1(N(C(CCC2CCN(C)CC2)=O)C)CN(C(=O)C(=O)NCC2CC2)CC12CC2 48309,C(=O)(C1(C)CCc2ccccc21)NC1CC1.CC1C(CO)CCN1C(=O)CNC(=O)N 48310,C(=O)(CCC(=O)NN(C)C)NC(CC#CC)C(=O)NCc1oc(C)nc1C 48311,N1(C(CCCCCCC)C(=O)NC(C)(C)CC)Cc2ccccc2CC1(C)C 48312,CC1(C)CC(CNCCc2c(F)cccc2F)CCO1 48313,Cc1ccc(C(N2CCCC(NC(=O)Cc3csc(NC=O)n3)C2CO)=O)c(Cl)c1 48314,C(CCCN=c1[nH]nc(-c2ccon2)s1)OC(c1c(OC)ccc(OC)c1)=O 48315,N1(C(C)(C)C)CC(F)(c2c(-c3sc(C)c(Br)n3)nn[nH]2)C2(COC2)C1 48316,C1(NC(C2(CC)N(C(CC(=C)C)=O)CCC2)=O)CNC(=O)C12CC2 48317,CCC(CC(=O)NCC1c2cccc(c2)OC(=O)C(=O)NC1)C(F)F.CC#N 48318,c1(C(N2CCCN(C(C(CC)C#N)=O)CC2)=O)cccc2c3c([nH]c12)CCC3 48319,N1(C(C(CNC(C2CN3CCN2CC3)=O)O)=O)CC(=O)NCC12CC2 48320,S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC(=O)NCC(=O)OC2CCCC2)COCC1 48321,n1(CC)ncc(C(=O)NCc2ncoc2CCNC(C2CC23CC(O)C3)=O)c1C 48322,CC1=C(C)CC(C)(C(=O)NC2C=CCN(C(c3ncsc3S(N)(=O)=O)=O)C2)CC1 48323,C=CCCCCC(=O)NCC1CCC(C(N2CCC2C2CCCCC2)=O)O1 48324,C(=O)(C1=CC2C=CC(C1)C2)NCCC(CC)(C)NC(c1ccncc1OC)=O 48325,N1(C(c2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCOC(C)(C)C)C1 48326,C1(NC(CN2CCN(C(=O)OCC)CC2)=O)Cc2cccc(Cl)c2CN1 48327,C(=O)(CCCCC(N)=O)N1CCC(NC(C(C)(C2CC2)NC(C)=O)=O)C1 48328,Cc1ccc(C(=O)NOCC(=O)NC(c2snnc2C)C)cn1 48329,Cc1cccc(C)c1OCC(=O)NC1CCN(C(C2CCO2)=O)C1C(C)C 48330,C1(CC(=O)NC2(CNC(c3snc(O)c3Cl)=O)CCC2)SC2=NCCN2C1=O 48331,c1(C(N2C3(CN(C(C(Cc4ccsc4)OC)=O)C3)CC2)=O)n[nH]c2cccnc12 48332,c1(O)ccc(Cl)cc1.C1(OCC)CCN(c2nnc(N)s2)C1 48333,C(CCCC(=O)NCCCc1nncn1C)NC(Cc1n(C)ccn1)=O 48334,c1(C(N2CC(CNC(Cc3cn(C)nc3)=O)N(C)CC2)=O)ccc2cnoc2c1 48335,C1(C(C)(C)CNC(=O)CCF)CC2(CCN(CC3CCC(O)C3)CC2)C1 48336,CC1COCCC1NC(=O)CCN(C(=O)CCC1CCC(=O)C1)C1CC1 48337,N1(C(C2Cc3ncncc3C2)=O)CCCCC(C2CNC2)C1 48338,N1(C(C=C(C)Cl)=O)CCC(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)CC2)CC1 48339,c1(C(=O)NCC(NC(C(CC)OC2CCCC2)=O)SC)ccc(NC)c(C)c1 48340,c1(OC)cnc(C(N2CC3C(CNC(C4(CO)CC4(F)F)=O)C3C2)=O)nc1 48341,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48342,c1(C(=O)NCC(=O)NC(C2(C)CN(C(=O)CC3CCCCC3)C2)C)ccc(Cl)cc1 48343,C1(NC(CC(CN(C)C)(C)C)=O)C2CC(O)C1N(C(C1CSCCS1)=O)C2 48344,N1(C(C2N(C(C(C3CCC3)OC)=O)CC=C2)=O)CCN(C)C(=O)CC1 48345,n1(CC)ncnc1C(c1nnnn1CCC1(C)CC1)NCc1ccc(C)o1 48346,N1(C(C(c2c(C)cccc2)C)=O)CCC(CNC(c2snnc2C)=O)C12CC2 48347,C(=O)(C(C)=CC(C)(C)C)NCC(C1CC1)NC(CC1C(=C)C1)=O 48348,n1(CC(=C)C)nnnc1CNC(c1nc(C2CC2)cs1)C1(CC)CC1 48349,C12CCCCC1N2.c1(C(C)NC(=O)CN(C)C(C2CCCCS2)=O)ccccn1 48350,n1(CCC)nc(C)c(C=CC(=O)NCC(C)C(=O)OC(C)(C)C)c1Cl 48351,C1(CCNC(COCCOCC)=O)C(C)CCCN1C(c1cccc2c1CC2)=O 48352,Cc1cnoc1C(=O)NC1CC(CC(C)C)C1.C12(CCC1)C(=O)NC2 48353,N1(C(C(CC)O)=O)CCC(C(N2CCCC(CCOC)C2)=O)C(C)(C)C1 48354,C1(C(N2CC(CC(C)C)OCC2)=O)CC(O)CCN1C(c1cc(O)cc(F)c1)=O 48355,N1(c2ncc(CCCNC(=O)OC(C)(C)C)cn2)C2CCC1C(CO)C2.CNC 48356,C(CC(CNC(=O)C(C1CCCC1)C1CCCC1)NC(=O)C=CCOC)OC 48357,N1(C(CCC=CC)=O)CCC(NC(=O)CSCC(F)F)CC(O)C1 48358,Cc1cc(C(N2CC(N(C)C(c3cccc(O)n3)=O)C2)=O)cn1C(C)C 48359,c1(OC)cccc2c(C(=O)NC(C)CCNC(=O)C(c3cncn3C)O)csc12 48360,S(=O)(=O)(c1ccc2c(c1)CC(CO)C2)NC(N1CCOCC1C(C)(C)C)=O 48361,c1(NC2CCC3(CN(C(CCCNC)=O)C3)C2)cccc2cnccc12 48362,c1(NC)cc(Cl)ccc1C(=O)NCC1C#CC(NC(=O)C(CC)(CC)OC)C1 48363,C1(C(NOC(CC)C)=O)CC2CN(C(c3nc(C)oc3C)=O)CC2C1 48364,CN1CC(NC(C2C3CC3CN2C(c2nn(C)cc2Cl)=O)=O)CC1=O 48365,C1(CNC(CCCCC=C)=O)CCN(C(C2(OC)CCOCC2)=O)CCC1(F)F 48366,C(=O)(CCCC(=O)N1CC(c2cnc(F)cc2C)(O)C1)N(CC)CC 48367,C1(OC)CCCC(C(=O)NC2CCCC2CNC(=O)C=CSc2nc[nH]n2)C1 48368,N1(C(C(C)Cn2ccnc2)=O)CC2CC(CNC(C3COC3)=O)C2C1 48369,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2CCN(c3ccc(Cl)cc3)C2=O)c1C 48370,c1(C(N(CCCN(C(C(C)OCCOC)=O)C(C)C)C)=O)cc(O)ns1.C1(CO)CC1 48371,C(CC(C(=O)N1CCC(N(CCO)C(C2CCN(C(C)C)C2)=O)C1)NC(C)=O)SC 48372,C1(NC(CCSCCC)=O)CCCC(NCc2cn(CC(N)=O)nn2)C1 48373,C1(C)(CNC(CCc2n(C)ncc2)=O)CCN(C(C23CCCCC2C3)=O)CC1 48374,CC1CC(NC(=O)CC2CCN(c3nccs3)CC2)CN1C(C1CC2CC2C1)=O 48375,N1(C(COC(C)(C)C)=O)CCC(CN(C(=O)CC2C=CCCC2)C2CC2)C1 48376,c1(OCC)ncc(C(N2CC(NC(=O)CCCC3CC3)CC(C)C2)=O)cc1Cl 48377,N1(C(c2nc(CC)oc2C)=O)CCCN(C(=O)CC(C)O)CC1c1ccccc1 48378,C1(C#N)(C(=O)NCCCOCCNC(C(C)(O)C2CC2)=O)CCCCC1 48379,C1(N(C(C2C(NC(C(C3CCC3)OCC)=O)C2(C)C)=O)C)CCOC(C)C1 48380,CCC(C)CCC(=O)NC(C)C(C)(C)C(=O)NCCN(CC(F)F)C 48381,C1(N(C(C(C)=C2CCC2)=O)C)CCN(C(=O)Cn2ncccc2=O)CC1C 48382,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48383,N1(C(CN(S(=O)(=O)C2CC2)C)=O)CCCC12CCN(C(C1CC3CCC1O3)=O)C2 48384,C1(C)(C(=O)NC(CC2CC2)CO)CCCCO1.Cn1cc(C2CC(=O)N2)cn1 48385,c1(C(N2CC3(CCC(C(F)(F)F)O3)C2)=O)cc2ncccn2n1 48386,CC(CNS(C)(=O)=O)CC(=O)NCC1CC(NC(=O)C(c2cnn(C)c2)O)C1 48387,Cc1cc(Br)ccc1COC(c1cc(C2CCOCC2)on1)=O.C1CO1 48388,C1(C(=O)NCC2CCCN(C(C3(N(C)C)CCCC3)=O)C2)CCC2(CCCC2)C1 48389,CCC(CCCC(=O)NC1CCCC1)NC(=O)CN(C)CC 48390,c1(CC)cc(C)c(C(=O)NCCNCCCOC(=O)C2=CCCC2)o1 48391,N1(C(CN(C(C(C)C)=O)C)=O)CCC2(NC(c3cc(CO)[nH]n3)=O)CC2C1 48392,C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NC(C)Cc1nn[nH]n1)C 48393,C1(O)(CNC(CC2(CS(C)(=O)=O)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48394,C1(CC(C)NC(=O)CC(C)(F)F)CCN(C(C2CCCCN2C)=O)CC1 48395,c1(C(C)C(=O)Nc2cc(Cl)c(Br)cc2O)cc2ccccc2nc1O 48396,n1(C(C)C)cccc(C(=O)NCCn2cc(CNC(C3CC(F)C3)=O)nn2)c1=O 48397,c1(SC)ccc(Cl)c(C(N2CCC(CC(C(=O)CCS(C)=O)=O)CC2)=O)c1 48398,CCC(C)C(C(=O)NC1COCCC1NC(c1sc(O)nc1C)=O)N(C)C 48399,c1(SCC)ccc(C)c(C)n1.N12CCN(CC1)C1CN(C1)CC2=O 48400,N1(C(C2C(OC)CC2)=O)CCC(CO)(CNC(c2cc(C(F)F)ncn2)=O)CC1 48401,C1(C(=O)NCCCN(C(=O)CC(C)(C)F)C)CCCCC1(C)C 48402,C1(NC(CCCSC)=O)CN(C(=O)C(C)(C)C2CCOC2)CC1C 48403,N1(C(c2c(OC)scc2)=O)CCCCCC(NC(=O)Cc2cnc[nH]2)C1 48404,N12CC(CC(F)(F)C1)C2=O.c1(NCc2ccc(F)cc2Br)ccn2nccc2c1 48405,C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(c1c(C)cc(C)[nH]1)=O 48406,N1(C(C2C(C)=C2)=O)C2CCCC1CC(NC(=O)Cc1c(C)[nH]c3ccccc13)C2 48407,c1(NC(=O)NCCOCCOCCOC)c(C)cccc1[N+](=O)[O-] 48408,CCCC(CCCN)C(=O)N1CCC(CN(C)C)C(C)C1 48409,N1(C(C2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCOC1)OC)CCO2 48410,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48411,C(=O)(CCC(C)(C)C(=O)NCC(CO)NC(C1CCCc2ccnn2C1)=O)OC 48412,N1(C(Cn2c(C)cc(C(F)F)n2)=O)CC2(C1)CN(C(=O)CCOC1CC1)CCO2 48413,C1(C(N2CCCC(CN(C)C(c3ccc(Cl)[nH]3)=O)C2)=O)COc2ccccc2C1 48414,c1(CSCc2ccc(C)s2)ccccc1C(=O)NOC(C)(C)CO 48415,c1(CC(=O)NC(CNC(CCNS(CC)(=O)=O)=O)C)csc(CSC)n1 48416,N1(C(CC(C)C)=O)CC2CCC(N(C(=O)CCc3ccccn3)C)C2C1 48417,C1(NC(c2cnc(OCC)nc2)=O)CC2CN(C(=O)C(F)(F)CO)CC2C1 48418,CC(C)C(C)C(=O)NC(CC1CCC1)C(N1CCC(OCCF)CC1)=O 48419,N(C(=NCc1ccccc1)N1CCOC(c2cnn(C)c2)C1)CC(CC)(C)C 48420,C1(NC(c2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48421,c1(CC(=O)N(c2cc(OCC)ncn2)C2(C)CCC(N)C2)cc(C)cc(C)c1 48422,Cc1ccnnc1C(CC(=O)NCC1CC1)N(C1CCSC1)C 48423,c1(C2(NC(c3noc(-c4ccccc4)n3)=O)CC2)nnc(N2CCC3CC23)o1 48424,c1(C(=O)NC(CC)CN(C)C(c2cnnn2C)=O)ccc(C)c(F)c1F 48425,Cc1scc(C(=O)NCC2OCCC2C(=O)NCCc2ccccc2F)c1C 48426,C1(NC(C2(C(F)(F)F)CCC2)=O)CCCCN(C(=O)Cc2cn(C3CC3)cn2)C1 48427,CCC(CC(=O)NCCCNC(=O)CC1CC2(CC2)C1)C(C)C 48428,CC1CCC(=O)N1.C12(CC1C)C(=O)NC2.C1(C(=O)OC(C)(C)C)(COC)CC1 48429,CC1CCCC1(C)C(=O)NC1CC(CNC(c2nc(C(C)(F)F)cs2)=O)C1 48430,C1(C(=O)NC(CC)CNC(C2(CC)CC2)=O)CCc2cc(OC)ccc2C1 48431,C1(C(C)NC(C2CC2(C)C)=O)CCCN1C(c1ccncc1)=O 48432,N1(C(C(=O)NC(C(CC)C)C(N)=O)=O)CCCC1C1CCC(C(=O)OC)O1 48433,CC(C)C(C)C(CNC(=O)CCS(C)=O)NC(C1(CCOC)CC1)=O 48434,N1(C(C(CC(=C)C)C)=O)Cc2ccnn2CC(NC(c2cc(CC)oc2C)=O)C1 48435,O=C1NC2(C(=O)NCCC3(O)CCN(C(C4CCCS4)=O)CC3)CC3CC1C2C3 48436,c1(C2(CNC(=O)Nc3cccs3)CC2)ccc(Cl)nc1 48437,C1(C2CC2)(NC(C(C)OC)=O)CCN(C(=O)CCCc2sccc2C)C1 48438,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48439,c1(C(=O)NCC2N(C(Cc3c(C)occ3)=O)CC(F)C2)cc(Cl)cc([N+](=O)[O-])c1 48440,N1(c2cccc(NC(=O)C(F)(F)C(C)(C)O)n2)CC(C(=O)OC)c2ccccc21 48441,Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NCC(CO)NC(C1(C#N)CC2(CC2)C1)=O 48442,C=CC1CCCN(c2nccc(NS(=O)(=O)Cc3sc(Br)nc3C)n2)C1 48443,C1(=CC(=O)NCCCC2(NC(CC3C(C)C3)=O)CC2)CN2CCC1CC2 48444,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48445,Cc1nc(NCc2cccc3c2CN(C)C3)cc(=NCc2ccnc(CO)c2)[nH]1 48446,c1(CC(=O)Nc2nc(C)nn2C)cc(F)cc(Cl)c1 48447,c1(C(=O)NC2CCCN(C(CC(CCC)CC)=O)CC2)cccc2c1CC(C)(C)C2 48448,C1(NC(c2c(COC)ccs2)=O)CC(CNC(c2cn(C)cc2C)=O)C12CCC2 48449,N1(CC)CCCCC1C(=O)NC1CCN(C(=O)CN(C)CC2CCCC2)C1C 48450,C1(C(N(CCCNC(CNC(COCCOC)=O)=O)C)=O)OCCOC1(C)C 48451,c1(C(=O)N)ccc(S)o1.C1(SC(C(=O)NC2(C)CC2)c2ccoc2)CCCO1 48452,Cc1oc2cc(C(=O)N(CCCNC(C3(O)CC3(C)C)=O)C)[nH]c2c1C 48453,N1(C(CNC(C)=O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)c(F)c(Cl)c3)c2C1 48454,C=CC1(C(=O)NCC(N2CCCC2C)C)CCN(C(=O)COCCCF)C1 48455,C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CN(C(c2c(OC)nsc2)=O)C1 48456,CC(C)CC(CCO)NC(=O)CC1CCC(NC(c2csnc2Cl)=O)C1 48457,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48458,N1(C(c2ccc(SC)s2)=O)CCN(c2ncc(SC)cn2)CC1C(F)(F)F 48459,N1(C(C(C)CO)=O)CCC(NC(C2(C)CC(F)(F)C2)=O)CC1 48460,c1(C(N2CCCN(CNCC)CC2)C(=O)NCC(C)C)c(F)cc(Br)cc1F 48461,N1(C(C(CC)C)=O)Cc2ccccc2C1C(=O)Nc1nc2ccccc2nc1OC 48462,C1(C(=O)Nc2ccc(F)nc2C)CCC(O)CN1C(C12CC(C(=O)OC)(C1)C2)=O 48463,C1(CN(C)C)CC(O)CN1C(c1ncoc1CNC(c1ncncc1N)=O)=O 48464,CC(F)(F)CC(=O)NCC1(CCNC(C2COCC2c2ccccc2)=O)CC1 48465,C1(CC)CCCCC1C(C(=O)NCC(O)C(C)(C)C)NC.C(C(C)C)N 48466,C(CN=C(NCC1CCC(OC)O1)N1CCC(c2ccc(F)cc2)C1)OCC=C 48467,C1CCC(C)(C)C(=O)N1.C1(C)C(=O)NC2(CC2)CC(=O)N1C.C(C)(=O)OC 48468,C(=O)(CCCCCc1ccccc1)NCC(CNC(C1CC(C)(C)O1)=O)OC 48469,N1(C(C(CC=C)(F)F)=O)CCCC2(CCC(NC(c3nc(C)nn3C)=O)C2)C1 48470,CC1CC2(CCN(C(=O)CSc3ccccc3Cl)CC2)CN1C(C1CC1C)=O 48471,CC(CC(=O)NCc1cc(C(=O)NCc2ccn(C3CC3)n2)cs1)C1CC1 48472,Cc1n[nH]c(C)c1SC(C(=O)N1CC(NC(C)C)C1)(C)C.C12(CCCCC1)C(=O)N2 48473,CC1(NS(=O)(=O)CC2CCCC2(F)F)CC2(C1)CC(F)(F)C2 48474,C#CCC(CC#C)C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C 48475,N1(C(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1c(Cl)sc(C)c1C)=O 48476,N1(C(COC(C)(C)C)=O)CCC=CC1C(N1CC(CO)C1C(=O)O)=O 48477,Cc1cc(C)cc(CN2CCCCC2C(=O)NC(c2cccs2)C)c1O 48478,C1(C(N2C(C(=O)NC)CCC2)=O)(OC)CCN(C(c2sncc2C)=O)C1 48479,N1(C(C2ON=C(C)C2)=O)CCCC(CCNC(C23CCCC2(C(N)=O)C3)=O)C1 48480,N1(C(C2N(C)CSC2)=O)CC2CCC(NC(=O)CC3(CO)CCCC3)CC2C1 48481,Nc1cc(C(=O)NC2CC(F)(CNC(C3CCC(=O)O3)=O)C2)cnc1N 48482,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CCCC12CC2)=O 48483,C=CCCCCC(=O)NCC1CC(O)CN(C(=O)CCc2ccccc2N)C1 48484,Cc1ccc(F)cc1NC(C1CCCC1(C)CNC(C1NC(=O)C2CCC12)=O)=O 48485,C(c1cccc(Cl)c1)=CC(=O)NCC1(O)CCN(C(CSCC=C)=O)C1 48486,c1(C(=O)NCC2(CNC(c3ccc(N)c(F)n3)=O)CC2)cnc2[nH]nc(O)c2c1 48487,c1(C(N2CCC(CNC(C3(CC)CCCC3)=O)C2)=O)cn(C)nc1-c1ccoc1 48488,N1(C(=O)C=CC2CCC2)CCC2(CCN(C(=O)C(O)Cc3ccccc3)C2)C1 48489,C#CCCCCC(=O)NCc1cc(C(=O)NCC2(C3CC3)CCCO2)n(C)n1 48490,c1(C(N2CC(C)N(c3ncncc3C#N)CC2)=O)n[nH]c2cccnc12 48491,C1(C(N2CC(C(=O)NC3C(C(C)C)CCC3)(CO)C2)=O)Cc2nccn2C1 48492,C=C(Cl)CC(C(=O)N1CCN(C)CC1)NC(c1ccncc1NC(N)=O)=O 48493,c1(CNC(C2CC3CC3C2)=O)nc2c(s1)CN(C(C1(C(F)F)CCC1)=O)CC2 48494,c1(C(N2CC(NC(c3cccc(F)n3)=O)C(F)C2)=O)nccc2nc[nH]c12 48495,C1(N(C(C)=O)CC)CCN(C(c2ccc(C)s2)C(=O)NCCCF)CC1 48496,C(=O)(C#CC1(C)CCCO1)NCCC(C(=O)NC1CCC2(CC1)CC2)OC 48497,CCC(C)C(C(=O)N(C(C)CC(=O)NOCc1cccnc1)C)SC 48498,c1(NC(c2c(OC)ncc(-c3ccc(C#N)s3)c2)=O)cccc2ncsc12 48499,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48500,C1(NC(C)=O)CCCCC1NC(=O)Cc1c(Br)cnn1C 48501,C12(Nc3nc(C)c(C)s3)CCCC1CN(C(=O)CC(N)c1ccncc1)C2 48502,c1(CNC(COCC#C)=O)ncccc1C(=O)NC1(C(O)CO)CC1 48503,CCCCC(F)C(=O)N(C1CCCN(C(=O)CN(C)CCO)C1)C 48504,N1(C(C(CCC)(C)C)=O)CC2(C(=O)NCc3nc(C)no3)CCC1CC2 48505,c1(OC)nsc(OC)c1NC(=O)C(N1CCCCC1CN1CCOCC1)=O 48506,C1(C(=O)NCCSCCC#C)(SCC)CCCN1C(=O)C=CCF 48507,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)Cn1ncn(C)c1=O 48508,C(CCCCC(=O)NCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48509,CCC(CNC(=O)C(C1CCOCC1)O)(CC)NC(c1cnn(C)c1C1CC1)=O 48510,C(=O)(CC(C)CC(=O)NCC1(F)CC(NC(c2cncc(OC)c2C)=O)C1)OC 48511,c1(COC)cc(C(=O)NCCCN(CCO)C(C2SCCC2C)=O)no1 48512,C1(CCNC(C2CC(OCC)C2)=O)CCCCN1c1nccc(SC)n1 48513,C(C)(CCC(=O)N1CC2C(NC(C3CC(=O)N(C4CN(C)C4)C3)=O)C2C1)SC 48514,CCC(C)(CNC(c1cnco1)=O)C(=O)N(C1CCCC1)C 48515,C(=O)(C1CCCn2nccc21)NCCN(CCc1ccc(F)cc1F)CC 48516,N(C1CCc2cccc3cccc1c23)C(=O)NCC(c1n[nH]c(-c2cccs2)n1)C 48517,c1(OC)c(C)cc(-c2cc(CNC(=O)CCc3c(C)noc3C)ccn2)cc1C 48518,C1(O)(Cn2cc(CC(=O)OC)nn2)CCN(C(=O)CC2CCC(=O)N2)CC1 48519,c1(C(N(C2CCN(C(c3cc[n+]([O-])cc3)=O)CC2)C)=O)ncc(N)cc1Cl 48520,CCCC#CC(C)(C)NC(c1oc(CNC(c2ccncc2Cl)=O)cc1C)=O 48521,c1(C(=O)NC(c2ccccc2)CNC(C2(C3CCCO3)CC2)=O)cnn(C2CC2)c1 48522,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)C(c1ccc(OC)cc1)O 48523,N1(C(CC(=O)NC)=O)CCC2(CCC(CNC(C3CC3c3cnc[nH]3)=O)O2)CC1 48524,C1(NC(C(C)CO)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC2CCCC12 48525,c1(C(=O)NCC(CNC(C=C(C)C(C)(C)C)=O)O)cncc2nc(O)[nH]c12 48526,c1(CC)cc(C(=O)NC2CN(C(C3(N4CCCCC4)CCCC3)=O)C2)nn1C 48527,C1(CNC(CC)=O)CCN(C(C2C=CC(NC(=O)COC)C2)=O)C12CCC2 48528,CCCCCCC(=O)NC(C1CCCN1C(C1(C(F)(F)F)CC1)=O)C 48529,N1(CC(C2(c3nnnn3CC(F)F)C(C)(C)OC2)=O)CCC(C2(C)CC2)CC1 48530,C1(C(C)NC(C2(C3CCCO3)CC2)=O)CN(C(=O)CCCF)CCO1 48531,c1(C(=O)OCC)noc2c1CCCCC2.N12CCC(C(=O)OCC)(C1)OC(=O)C2 48532,c1(C(N(CCNC(c2cccs2)=O)CC)=O)ccc(F)cc1F.C1(=O)CC(C)N1 48533,C1(O)(CCNC(C2COCCC2(F)F)=O)CCCN(C(=O)CCc2cnoc2)C1 48534,C1(NC(Cc2ccc(C)nc2)=O)CCN(C(=O)CC2OCCCO2)CC1F 48535,c1(-c2cn(C3CN(C(C(C)=C4CCCO4)=O)CC3C)nn2)cccc(CO)c1 48536,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48537,C(=O)(C(F)(F)C(F)(F)F)N1CC(N(C(C2CCC(C3CC3)O2)=O)CC)C1 48538,CC(C)C(C(=O)NOCCCF)C(C)NC(=O)C(C)N(C)C 48539,C(=O)(C(F)(F)CO)NC1(CC=C)CN(C(c2n[nH]cc2C2CCC2)=O)C1 48540,C=CC(C)(CC)C(=O)NCC(C)N(C(C1CCCN(C(C)C)C1)=O)CC 48541,C1(NC(=O)C(=O)Nc2ccccn2)CC2CN(C(c3csc(Cl)c3)=O)CC12 48542,N1(C(C(=O)NCC)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(C)(C)C1 48543,c1(CCC)cc(C(N2CC(C(C)(C)O)(CNC(C3(F)CC3C)=O)C2)=O)no1 48544,c1(C(=O)NCC2(C)CCN(C(CC3CC(C)C3)=O)C2)cn(C)n2cccc2c1=O 48545,C#CCCC(O)C(=O)N1CCCN(C(=O)CC2CCOC2)CC1 48546,Cc1cc(C(N2CCC(C(F)(F)F)(C(=O)O)C2)=O)nc(O)c1 48547,C1(CCNC(=O)CCn2cccn2)COCCN1C(=O)CCN1CCCCC1 48548,C#CCCCC(C)N(C(=O)CCn1cc(C(C)OC)nn1)CC.N1(CCO)CCCC1 48549,C1(CC=C)(C(=O)NCCOC(C(=O)NCCCSC)C2CC2)CCOC1 48550,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)cc2)=O)CC2CC12 48551,N1(C(=O)Nc2cnn(CCO)c2)CCC(n2cc(Cl)cn2)CC1 48552,C1(C(=O)NCCN(CCC)C(c2cc(N)ccn2)=O)(CC)CC(C)(C)C1 48553,c1(C(N2CC(CC(=O)NC3(C(=O)NC)CCC3)C(C)C2)=O)cc(C#N)[nH]c1C 48554,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1C 48555,N(C(=NCCCF)NC1CCCCC1)CC(c1c(Cl)ccc(OC)c1)(COC)C 48556,C=C=CCCC(=O)N(C)CC1CN(C(c2nnn(C(C)C)c2C)=O)C1 48557,c1(CC)nc(N2CCN(C(N3C4CCC3CN(C)C4)=O)CC2)c2ccsc2n1 48558,N1(C(C2C(OC)CCOC2)=O)CCC(NC(c2cc(Cl)nnc2Cl)=O)C(CO)C1 48559,CCCCCC(O)CC(=O)N1CC2CC2(NC(=O)C(C)n2cncn2)C1 48560,C1(NC(C2(CNC(=O)COC(F)F)CC(=C)C2)=O)CCC2(CCC2)C1 48561,Cc1cccc2c1C(NC(C1(CCO)CCS(=O)(=O)CC1)=O)CC2 48562,c1(C(C)(C)C#N)ccc(C(N2CC(NC(C3(Cl)CC34CCC4)=O)C(O)C2)=O)cc1 48563,c1(C(=O)NCC(C2CCN(C(c3n[nH]cc3Cl)=O)CC2)C)nc(Cl)c(=O)[nH]c1N 48564,C1(C(=O)OCC)CCCCN1C(C1CCCN1C(c1cccc(SCC)c1)=O)=O 48565,c1(OC)cc(C(=O)NCC(CC(C)C)NC(c2n[nH]cc2C2CCC2)=O)n(C)n1 48566,N1(C(C2CCN(C3CC3)CC2)=O)CCCC(NC(C2CC3CC3C2)=O)CC1 48567,N1(C(=O)CC2(NC(=O)CN3CC4CC4C3)CCC2)CCc2ncncc2C1 48568,c1(C(=O)O)cn2c(n1)CCCN2c1nc(-c2ccccc2)ns1 48569,CC(C)CCCCC(=O)N1CCCC1CC(=O)N(C)Cc1cnccn1 48570,C1(SC2CCN(C(=O)Cc3ccc(C(N)=O)cc3)CC2)CCC2(CCCC2)O1 48571,C#CCC(C)(CC)C(=O)NC1CC=CCC1C(=O)N(C)CC1(C)CC1 48572,Cc1cc(NC(C2COCCO2)=O)ccc1NC(=O)CNS(=O)(=O)C1CC1 48573,C(=O)(CCC1=CCCCC1)N1CCCC(N(C(C2CC(SC)C2)=O)CCO)C1 48574,c1(OC(C)C(=O)NCCC(C)NC(=O)CNc2cccnc2)ccccc1Cl 48575,C(=O)(C1CCc2nccn21)NC1(C)CC(NC(c2cc3ncccn3n2)=O)C1 48576,N1(C(=O)CCC2CCOC2)CCC(NC(c2cc(C3CC3)on2)=O)CC(O)C1 48577,C(CCCC(=O)NON(C)C(c1ccc(F)c(O)c1)=O)N(C)C 48578,C(=O)(CCC(F)(F)F)N1CC(C(N)=O)(CNC(C2CN(CCOC)C(=O)C2)=O)C1 48579,C1(NC(Cc2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C)CCCS1)=O 48580,N1(C(C(C(C)C)NC(C)=O)=O)CC2(CCN(C(c3cnc(S)nc3)=O)CC2)C1 48581,O=S(=O)(c1cnccc1N1CC2C3CCC(C3)C2C1)NCc1cncs1 48582,C1(NC(CC2COCC(C)O2)=O)CC(C(=O)N(C)Cc2cnn(C)c2)=CC1O 48583,c1(NC(=NCC)NCC(C)COC)ccc(S(=O)(=O)c2ccc(Cl)cc2)cc1 48584,Cc1ccc2occ(C(=O)NCC3CN(C(C4CC(O)C4)=O)CC(C)(C)O3)c2c1 48585,N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(=O)C(O)C(F)F)C2CCCC12 48586,c1(C(=O)NC2C(OC)CN(C(=O)CC3OCCCO3)C2)ccc2nc(O)sc2c1 48587,C1(NC(C2(C(=O)NC)CC2)=O)CCC(CCC(c2cnccn2)NC(=O)C2CC2)C1 48588,C(C)(CC(=O)N(C1CCN(C(=O)Cc2csc(NC=O)n2)C1)CCO)OC 48589,Cc1snnc1C(=O)NC(CN(C)C)C(=O)NCCC1(O)CCOC1 48590,C(=O)(CN1C(=O)CCc2ccccc21)NC(C)CCN(C)C(c1ccnnc1)=O 48591,CC1CCCn2ncc(C(=O)NCC3(O)CC(NC(c4ncc[nH]c4=O)=O)C3)c21 48592,N1(C(CCCOCCC)=O)CCC(C)(CCNC(c2ccoc2CC)=O)C1 48593,C#Cc1ccc(OC)c(C(N2CCC(CCNC(=O)C(C)CS(C)(=O)=O)C2)=O)c1 48594,CCCCCCCCCC(O)C(=O)NC12CC(NC(C3(CCOC)CC3)=O)(C1)C2 48595,c1(C(CN)NC2CCN(c3ccccc3)C2=O)ccc(Cl)cc1Cl 48596,CCCC(CCCNC(=O)CCNC(C1CCCO1)=O)NC(=O)C=CCF 48597,C1(C(=O)NCC(C=C)O)CCC(C)N(C(c2cnc(CC)cn2)=O)C1 48598,c1(CC)cccc(NC(C2(C)CCCN2C(=O)C(c2ccc(C)o2)C)=O)c1F 48599,N1(Cc2n(CC)ncn2)CCCCC(NC(=O)Cc2ccc(Cl)s2)C1 48600,C12(NC(c3ccncn3)=O)CCN(C(c3ncoc3-c3ccccc3)=O)CC1C2 48601,C1(C)(C(=O)NC(C=C)C)CC12CCN(c1nnnn1C(c1ccccc1)C)CC2 48602,N1(C(c2scc(COC)c2)=O)CC2CCN(C(=O)CCCCCF)CC2C1 48603,N1(C(C=C(C)Cl)=O)CCCC(C(C2C(C(N(C)Cc3ccccc3)=O)CC2)=O)C1 48604,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48605,N1(Cc2n(C)c(S)nn2)CCC2(CC1)CC2(C)C(=O)NCCSCCO 48606,C12(NC(c3c(C)n(C4CC4)cc3)=O)CC(CNC(=O)C(C)CN(C)C)(C1)OC2C 48607,C(=O)(CCCCCC(F)(F)N1CCOCC1)O.c1(C(C)C)cc(S)ncn1 48608,C(=O)(C(F)C1=CCCCC1)N1CCCC(CN(C)CC2CCCCCC2)C1 48609,c1(CC)cccc(NC(=O)C(Cn2cncn2)NC(c2nonc2N)=O)c1C 48610,C(c1cc2ccccc2o1)=CC(N1CC(N(c2cc(CC)ncn2)C)C1)=O 48611,O=C(C(=O)C(F)(F)F)NCCOC1CCN(C(c2ccc(C3CC3)c(Cl)c2)=O)C1 48612,N1(C(C=CC(C)C)=O)CC2(C)CC(NC(C3CCC(CO)CC3)=O)C=NC=CN2C1 48613,CC(C)(C)COCCC(=O)N(CCCN(C(=O)CSC(=N)N)C)C 48614,C1(CC(=O)NC2CCC(CNC(C(CC)n3cncn3)=O)C2)CCCOCC1 48615,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CC2)C2(CCC2)C1 48616,N1(C(C(CN(C)C)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCc1cn[nH]c1)C2 48617,C(=O)(C1(C)CCOc2ccccc21)N(C)CCNC(c1cc(C(F)F)on1)=O 48618,C1(CC)CC(CO)N(C(c2cc(C(=O)O)c(C(F)(F)F)[nH]2)=O)C1 48619,C(=O)(CCCCCNC(=O)CC(C)C(C)C)NCc1c(C)nc[nH]1 48620,Cc1nc(C(N2CCCC(CNC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)cn1C(F)F 48621,C#Cc1ccc(-c2cc(C(=O)NC3CC(C(=O)OC)CCC3O)ccn2)cc1 48622,C#CCCCCCC(=O)NCCCCN(CCCNC(C1(F)CC=CC1)=O)C 48623,N1(C(=O)NCC)CCC(C(=O)NC2C(C(N3CCC(N(C)C)C3)=O)C2(C)C)CC1 48624,C12(C(=O)NC3C(C(=O)NC4CC(N(C)CC)C4)CC3)CCC(OC)(CC1)C2 48625,NC(=O)N(NC(=O)c1cc(F)ccc1F)c1ccccc1OCC(F)F 48626,n1(CC)ncc(-c2nc(C(=O)Nc3ncccc3C(F)F)cs2)c1C 48627,Cn1nc(-c2nc(-c3cccnc3)no2)c2c1CCN(C(=O)OC(C)(C)C)C2 48628,N1(C(C(C)=CC)=O)CC2COCCC2(NC(=O)Cc2c(C)nc(O)nc2O)C1 48629,N1(C(Cc2cccc(SC)c2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48630,c1(OC)ccc(F)cc1C(CNC(=O)CCC1CC1)NC(c1cccc(Br)c1)=O 48631,CC1CN(C(=O)C(N2CCCC(C(c3ccccc3)=O)C2)=O)CCC1C(=O)O 48632,n1(CC=C)cccc1C(=O)NCCCCNC(=O)Cc1ccoc1C 48633,Cc1noc2nc(C(F)(F)F)cc(C(=O)N(CC(Cl)Cl)C)c12 48634,C1(NC(C2CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(c1cccn1C)=O 48635,C1(NC(c2c(OC)n[nH]c2)=O)CCCCCN(C(c2ccnc(F)c2F)=O)C1 48636,c1(C(=O)NCC2(C)CCCN2C(=O)C2=C(Cl)CCCC2)cc(F)cc([N+](=O)[O-])c1 48637,c1(C(N(C(C)CNC(=O)C(F)Cc2ccccc2)C)=O)cccn2ccnc12 48638,CN1CC(C)(C(=O)NCCCN(C(c2ccccc2SC(F)F)=O)C2CC2)CC1=O 48639,n1(CC)ncc(CNC(C2(C)CCN(C(=O)C(=O)C(C)C)C2)=O)c1C 48640,CC(C)(CCCF)NC(=O)CC=C(Cl)Cl.C123CC(C1)(C2)C(=O)N3 48641,C1(C(=O)NCC(=O)OCCCC)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48642,c1(C2(C)N=N2)cc2scnc2[nH]1.C1(O)(C(=O)N)CCN(C(=O)N)C1 48643,Cc1ccc(C(C)NC(c2nnnn2CCCF)Cc2scnc2C)s1 48644,N(C(=NCCOC1(c2ccc3ccsc3c2)CCC1)NCCC1CCCO1)C 48645,C1(CO)(CF)CCN(C(=O)Cc2ccnc(Oc3cn[nH]c3)c2)C1 48646,CC1CCCC1(C)NC(C1(C(C2CC2)NC(=O)CC2CCCCC2O)CC1)=O 48647,C1(=O)CCCCC(C(F)(F)F)N1.O=C(C(=O)N(C1CC1)CC1CC1)NCC(F)F 48648,N1(C(c2cn(CC)nc2)=O)CCCN(C(=O)CSCCC(C)C)CC1C(F)(F)F 48649,C#Cc1ccccc1CC(N1CC(CNC(=O)CC(=C)Br)CC1C)=O 48650,c1(CN(CCCNC(c2ncccc2C2CC2)=O)CC)ccc2n[nH]cc2c1 48651,NC(CCc1ccccc1)C(=O)NCC1CC1Cc1ccccc1F 48652,Cn1cc(C(=O)NC2(CCNC(C3CCCC(C(F)(F)F)C3)=O)CC2)c(O)n1 48653,C1(NC(C2N(C)C(=O)CC2)=O)CC2CN(C(C3CCOC(=O)CC3)=O)CC2C1 48654,C(C(C)(C)CC(=O)N(CCCNC(C1CCCN1S(C)(=O)=O)=O)CCO)OC 48655,c1(N(C(=O)CCC2CN(C(=O)C=CC(C)C)CCO2)CCCC)c(C)cccc1Br 48656,c1(C(N(C2CCOC2CNC(C)=O)CCC)=O)ccc(F)cc1C 48657,n1(CC)c(C(=O)N(C(C(=O)NC2CCCCC2)C)CC(=O)N(C)CC)cnc1O 48658,C(=O)(C(C(C)C)C(C)C)NCC(C1CC1)NC(c1c(C)cc[nH]1)=O 48659,N1(CC(=O)NCC2ON=C(C)C2)CCN(C(=O)C=C(Cl)Cl)CC1 48660,C(C#CCN=c1[nH]c(N2C3C=CCC2CCC3)nc2cc[nH]c12)OC 48661,Cc1cc(Br)c(NC(=O)CN(C2CC2)CC2COC2)c(Br)c1 48662,CC1ON=C(C(=O)NC2CN(C(=O)C(CO)N(C)C)CC(C)(C)C2)C1C 48663,c1(C(=O)NCC(C2CCN(Cc3nccs3)CC2)C)cc(Cl)c(Cl)c(Cl)c1 48664,N1(C(C(C)C2CCC2)=O)CC2CCC(C1)C2CNC(=O)C(O)CC(F)(F)F 48665,C1(C(=O)NCc2c(COC)noc2)CCCCCC1NC(C1OCCOC1C)=O 48666,C12(NC(c3cc(C(C)=O)oc3)=O)CCCC1N(C(c1cscn1)=O)CC2 48667,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(C1(c3ncccc3F)CC1)=O)C2 48668,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc3nc[nH]c23)=O)C1)C)C(C)C 48669,N1(CC(=O)NCC2CC(NC(c3c(C)[nH]nc3C(C)C)=O)C2)CCC(=O)NC1=O 48670,C1(SCC)CCCC1C(=O)NCCN(C(=O)CCCSCCC(N)=O)CC 48671,C1(C(=O)NC2C(NC(c3ccn(C)c3C3CC3)=O)CCCC2)Cc2ccccc2S1 48672,CC1CN(C(=O)CCC=CCN(C)C)CCC1N=c1[nH]c(Cl)ncc1[N+](=O)[O-] 48673,C(CN=c1ccnc(N(C)Cc2nc(CC)co2)[nH]1)c1ccc(OCC)cc1F 48674,c1(C(N2CC(C(C(N3CCCCC3CO)=O)OC)C2)=O)cc(C)nnc1O 48675,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 48676,C1(N(C(=O)C(C)(C)CF)C)CCCCN(C(c2ncccc2F)=O)C1 48677,C(=O)(C(C)(C)C#N)NC1CC(C(C(=O)N(C(C(C)C)CO)C)F)C1 48678,c1(C(N(C2CCCC(NC(=O)C(C)(C)C)C2)C)=O)cc(C2CC2)cc(Cl)c1 48679,C(c1c(Cl)cccc1Cl)=C(C(=O)NCC1(F)CN(C(C(=O)NCC)=O)C1)C 48680,Cc1nn(CC(N2CC3CC2CC3CNC(c2csnc2Cl)=O)=O)cc1[N+](=O)[O-] 48681,C(CCCCC(=O)NCC1CCN1C(C1CC(OC)C(OC)C1)=O)=CC 48682,C(C(C)CNC(=O)COCc1cccnc1)NC(COCCCC)=O.S(C)CC 48683,CC(N=[N+]=[N-])C(=O)N1CC(CC(F)C(=O)N2CCCC2)C1.[nH]1cncn1 48684,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 48685,c1(OC)cc(C(=O)NC23COC(C2)C(NC(c2coc(C)n2)=O)C3)cc(OC)n1 48686,c1(C(N2CCC(N(C(=O)CCSCCC)CC)C2)=O)ccc(F)cc1C(F)F 48687,N1(C(C2N(C(Cc3c(C)nccc3)=O)CC2)=O)CCC2(CCCO2)C1 48688,C=CC1(OC)CC1.C1C(=O)N(C)CC(=O)NCC(=O)N1C 48689,C(CCC(C)C)(C(=O)N(C)Cc1nncs1)NC(C1C(CCC)CCC1)=O 48690,CCS(=O)(=O)C=CC(=O)N1CCC(C)(C)C(CNC(=O)CN2CCCCC2=O)C1 48691,C1(OCC)CC(CN(C(=O)CNC(c2cc[nH]n2)=O)C)C1 48692,C(c1cn(C)cn1)=CC(=O)N(CC(CN(C(CCc1onc(C)n1)=O)C)O)C 48693,C(=O)(N1CC(C)(O)CO1)N1CCC(O)(NC(C(C(CC)C)=O)=O)C1 48694,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 48695,C(=O)(NNC(=O)C1CCC(=O)N1)NCc1cc(C)[nH]n1 48696,C1(S(N)(=O)=O)(C(=O)NCC2CC(NC(c3cncc(C(C)C)c3)=O)C2)CCCC1 48697,N1(C(C(CC)(C)C#N)=O)CCCCC2(C1)CN(C(c1coc(Br)n1)=O)C2 48698,c1(C(=O)NC(CCNC(C(CCCC)O)=O)(C)C)cc(=O)c2cc(F)ccc2o1 48699,C1(C2CCCN(C(c3ccccc3Cl)=O)C2)(NC(C#CC(=O)O)=O)CC1 48700,Cc1cc(=NC2CCOC(CCN(C)C)C2)[nH]c(=NCCCN2CCCC2)[nH]1 48701,N1(C(CC2(CSC)CC2)=O)CCOCC(CC(N2CCC(C)(C)C2)=O)C1 48702,C1(C(=O)NC(C2CCN(C(=O)Cc3ccccc3)C2)C)C2CC3C(C2=O)C13 48703,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(=O)CC1(C#N)CCC1 48704,c1(C(N(C2CCCN(C(c3cc[nH]n3)=O)C2)C)=O)ccc(N)c(Br)n1 48705,CCC(C)(CN(C(C)CSC)C)C(=O)NC(C)C 48706,C=CC(CCC)CC(=O)N1CCC(O)(C(C)NC(=O)Cc2cc[nH]c(=N)c2)CC1 48707,N1(C(C(c2n(C)ncc2)O)=O)CCOCC(CNC(c2cnns2)=O)C1 48708,c1(OC)ncc(Br)cc1CN(C1CCN(C(=O)CC2CCN(C)C2)C1)C 48709,C=CCC(CC(C)C)C(=O)N1CC(NC(c2ncccc2Cl)=O)CC(C)(C)C1 48710,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCOC(C)C)=O)CC(O)C2)CC1 48711,N1(C(C=C(C)C2CC2)=O)CC(=O)NCC1C(=O)N(C)CC1(C)CC1 48712,C(=O)(CCCCN=[N+]=[N-])NC(C)CC(=O)NC1(C)CCC(CO)CC1 48713,CC(C)(C(=O)NC1CCCC1n1cc(C(C)(C)C(=O)N2CC2)nn1)c1ccccc1 48714,c1(C(=O)NCC2(OC)CN(C(C3CC4CC4C3)=O)C2)cnc2ncnn2c1C(C)C 48715,C1(C(=O)OCC)CNC(=O)CN1C(c1sccc1Br)C(=O)NC1CCOC1 48716,c1(C(=O)NCCCN(C(C)C)C(C2CCCCC2(F)F)=O)cccc2occc12 48717,C(C(CO)NC(=O)Cn1cccn1)NC(C1C(CC(C)C)C1)=O 48718,N1(C(C(=O)N)=O)CCOC(F)(F)C1.Cc1cnc(CC2(c3ccccc3)CC(F)C2)s1 48719,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 48720,CCC(CC(=O)NC1CCCC1NC(c1c(C)cnnc1O)=O)C(C)(C)C 48721,C(=O)(CC(C)C)NC(C(=O)NCCCN(CC)CC)c1cccs1 48722,C1(NC(C(CO)N(C)C)=O)C=CCN(C(c2ccnn2-c2cccnc2)=O)C1 48723,N1(C(=O)OC(C)(C)C)CCCC1Cc1cn(CCN2CC(CNC(=O)CO)C2)nn1 48724,c1(-c2nnc(N3CCC(C(F)F)(C(=O)OC)C3)n2CC(=O)OC)c(F)cccc1Cl 48725,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(=O)CC2(O)CCCOC2)C3)n1 48726,C(=O)(C#CC1CCCC1)NC1C(C)CN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1 48727,C1(CNC(=O)CCCc2cc[nH]n2)CC2(CCC2)CN1C(=O)Cc1ccncc1Cl 48728,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1C)=O 48729,c1(C(N2CCC(C)(CCNC(CCNC(C)=O)=O)C2)=O)cnc2ccncc2c1 48730,n1(CC(=O)NC23CC(NC(CC4CCC(C)O4)=O)(C2)C3)cc(S(N)(=O)=O)cn1 48731,C(=O)(C1=CC(O)C(NC(=O)CC(F)(F)F)C1)NCc1c(C)cccc1 48732,c1(CNC(c2csc(CO)n2)=O)cccc(NC(C2COC2)=O)c1 48733,N1(CC)CCOCC1C(=O)NCC(=O)NCC(=O)NC.N12COCCC1C2=O 48734,CS(=O)(=O)c1cscc1C(=O)NCC(CO)NC(C1(F)CC=CCC1)=O 48735,c1(C(N2CCCN(C(C(CC=C)C)=O)CCC2)=O)cnn2cc(OC)ccc12 48736,c1(C(C)=O)cc(S(=O)(=O)NCC2CCCC(C)(C)C2O)cc2ccccc12 48737,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 48738,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 48739,c1(OC)ccc2c(c1)C(NC(=O)NCC1(CC)CCCC1O)CCC2 48740,CCC(C#N)C(=O)NC(C)(C)C(=O)NC(N1CC(NC(=O)NC)C1)=O 48741,C(=O)(C(CN(C)C)c1ccccc1)NC(CNC(C(C)N(C)C)=O)CO 48742,CC1(C(N2CCCC(O)C2)=O)CCCN(Cc2ccccc2-c2ccc(F)cc2)C1 48743,c1(C(=O)NC(CN(C(c2c(CC)non2)=O)CC)CC)coc2ccccc12 48744,c1(SCC(=O)NC(CC)CN(C)C(c2ncc(Cl)s2)=O)ccc(C#N)cc1 48745,c1(NC(N(C(C(=O)NC)C)C)=O)ccc2cc(C)sc2c1 48746,n1(CC)cc(C(N2CCC(CNC(=O)CS(C)(=O)=O)C2)=O)c(C)n1 48747,c1(C(N2C(C(=O)NC3CCCN(CC)C3=O)CCC2)=O)ncc2ccccn12 48748,C1(CN(C(COCC(=C)C)=O)C)C2CN(C(C3CC3c3ccc(Cl)cc3)=O)CC12 48749,N1(C(C2C(SC)C2)=O)CC(CNC(=O)COC(F)F)C(O)C1 48750,C(CO)(C(C)NC(=O)C(C)c1ccsc1)NC(CN(CC)CC)=O 48751,c1(C(N2CCC(C(N3CCC(C#C)C3)=O)(CC=C)C2)=O)ccc(C#C)cc1 48752,C#CCC(O)C(=O)NC(C)(CO)C(=O)NCCc1cnns1 48753,c1(C(=O)NCCNC(CSCC=C)=O)cc(OC)cc(C(F)F)c1 48754,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(c2c(C)ncs2)=O)C(C)C1 48755,C(=O)(C(C)(C)C(C)O)NC1C=CC(CC(=O)NC(c2cccnc2F)C)C1 48756,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 48757,C#Cc1ccc(C(N2CCN(C(=O)C(C)c3cc[nH]n3)CC2C2CCC2)=O)nc1 48758,C#Cc1ccc(C(=O)N(C(C)CCNC(C2C(c3ccc(F)cc3)C2C)=O)C)cc1 48759,CCCCCS(=O)(=O)CC(=O)N1CC(C(=O)O)C(OC(N2CCCC(C)C2)=O)C1 48760,O([Si](C)(C)C(C)(C)C)CCCN(C)C(c1cn2ccsc2n1)=O 48761,CCCCC(CNC=S)CC.c1(-c2cnoc2C)nnc(-c2cnccn2)n1CC(C)C 48762,C(=O)(CS(=O)(=O)C(C)C)NC(C1CCN(C(c2c(CCC)nco2)=O)CC1)C 48763,N1(C(COCCCCC)=O)CCN(C(=O)Cn2ccc(C3CC3)n2)C(C)C1C 48764,C(N(C)N1CC2(CNC(=O)OC2)C1)c1ccc(N2CCN(C)CC2)cc1 48765,c1(OC)ncc(C(=O)NCC(C2CCCCC2)NC(=O)CCCCSC)nc1C 48766,c1(C(=O)NCCCCC(CO)NC(CC2(OC)CC2)=O)cccc2c1OCC2C 48767,C1(NC(=O)C(F)OC(F)(F)F)(CO)CCCN(C(=O)CCc2cncs2)C1 48768,c1(C(=O)NC(C(=O)N(CC(=O)N(C)C)C)Cn2cncn2)c[nH]nc1[N+](=O)[O-] 48769,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 48770,NCC(Cc1ccccc1)C(=O)N1CCCCC1CN1CCCC1 48771,N1(C(C2CC(C)NC(=O)C2)=O)CC2CCOC2(CNC(=O)C#CC2CCC2)C1 48772,Cc1nc(C(=O)NCC(CO)NC(C2CCC(=O)N2)=O)co1 48773,N1(C(=O)CC2(c3ccon3)CC2)CCC2(NC(C3CC3F)=O)CCCC12 48774,c1(OC)ccc(C(N2CCC(NC(c3ccnc(Br)c3)=O)C(O)C2)=O)cc1O 48775,C(=O)(CC(O)CNC(C1(C)CCC(C)C1)=O)N1CCC(NC(C)=O)C1 48776,C1(C(C)NC(c2cccc(C3(OC)CC(OC)C3)c2)=O)CC(C)(C)CO1 48777,c1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)nnc2n1CCCCC2 48778,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC12C(CN(C(c3ccc(N)c(Cl)c3)=O)C1)C2 48779,C(C(=O)NNC(=O)N1CCC1c1ccccc1Cl)N(c1ccccc1)C 48780,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(C1CCCN1C1CC1)=O 48781,N1(C(C=CSC)=O)CC(N(C)C)C(CNC(c2cc(CF)on2)=O)C1 48782,c1(NCC2C(O)COC2)ccccc1SCC1CCCCC1 48783,C1(NC(C(C)OCCN(C)C)=O)CN(C(=O)CCN(C)C)CC1C(F)(F)F 48784,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(=O)Cc1ccncc1Cl)C2 48785,CC1CC(CNC(=O)CCc2cn(C)nn2)CN(C(C2(C)CCSCC2)=O)C1 48786,C(CCCCCCCCO)N(c1cccnc1)C(C1N(S(C)(=O)=O)CC1)=O 48787,N1(C(=O)CC2CCCCN2C(=O)Cc2cccnc2O)CC2CC(O)CC2C1 48788,N1(C(C(CC)C)=O)CCN(C(C23COCC(C2)C3)=O)CC1CC1CC1 48789,c1(CC)cc2c(CC(=O)NCCOCCCNC(=O)C=C(Cl)Cl)csc2s1 48790,c1(NCC2CCCN(CCC(=O)OC)C2)cc(OC)ccc1[N+](=O)[O-] 48791,C1(N(C)CC2CCC2(C)C)CCCN(C(=O)CCc2ccoc2)CC1 48792,C1(CNC(C2CCC(C)C2)=O)CCC(NC(c2scnc2C2CCCC2)=O)CC1 48793,c1(C(N2C(CN(C(C(COCC)C)=O)C3CC3)CCC2)=O)csc([N+](=O)[O-])c1 48794,C(=O)(C1CCSc2ccccc21)NC(CN(C(=O)CCCC(=O)OCC)CCC)C 48795,C(=O)(CCC(C)(C)C)NC1(C)CCOCC1.CC1CN2CC1C2=O 48796,C(=O)(C#CC1CCOC1)NC(C)C(C)NC(c1ncsc1Br)=O 48797,c1(C(=O)OC)ncc[nH]c1=NCC1(CNC(c2cnc(C(C)O)s2)=O)CC1 48798,C1(C(=O)NCC2CC(SC)C2)(CNC(C2CC(OCC)C2)=O)CCCCC1 48799,c1(C(=O)NC(CNC(C(CCC)(C)C)=O)(C)C(C)C)nc2ccccc2cc1Cl 48800,c1(C(N(CCOC)CCNC(C2CC(C)(C)C2)=O)=O)cc(F)ncc1OC 48801,c1(C(=O)NCC(CC(=O)NCCN2CCCC(C)C2)C)occ2c1CCC2 48802,c1(NC(C(c2ccco2)NC(COC(CC)CC)=O)=O)ccc(F)cc1O 48803,N1(C(C(C)C2CCC2)=O)CCCC(CN(C(c2cnc(Cl)s2)=O)C2CC2)C1 48804,C1(C)(C(=O)OCC)CCCN1C(C1(n2cc(C(C)(C)O)nn2)CC1)=O 48805,Cc1[nH]c(C#N)cc1C(=O)NCCCC1CCCCN1C(=O)C=CS(C)=O 48806,c1(NC)cnc(C(=O)NC2CCCC2NC(=O)CC(O)c2ccccc2)cn1 48807,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(=O)Cn1ccc(C2CC2)n1 48808,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 48809,c1(-c2cn(Cc3nc(CNC(=O)CC4CCOC4=O)sc3)nn2)cnccc1Cl 48810,Cn1nnc2cc(C3CC3Nc3ccc4c(c3)OCO4)cnc12.C1C(=O)N1 48811,CCC(CC)(CC)C(=O)NC1CN(C(=O)C(O)C2=CCCCC2)CC1C 48812,CC1(C)C(CC(=O)N(C2CCCC2)CCO)CC1c1cn(C2CCOC2)nn1 48813,C1(C(N(C)Cc2cnc(C)s2)=O)CCC(C)(C)N(C(c2c[nH]nc2Cl)=O)C1 48814,N1(C(c2cc(C)on2)=O)C(C(=O)NCCF)CC2CC12 48815,C(=O)(CC(F)(F)C(F)(F)F)NCC(C)(C)CNC(c1cccc2c1OCCO2)=O 48816,C1(CNC(c2cc(CC)c(C)s2)=O)N(C(=O)CSC(C)(C)C)CCCC1(C)C 48817,C12(CNC(c3n(CC)c(O)nc3)=O)CCCN(C(c3c(C)cnnc3O)=O)C1C2 48818,C(=O)(C(O)CC(C)(C)C)NCC(=C)CCNC(c1ncc(C)cc1OC)=O 48819,C12(CNC(c3ccc(OC(C)C)cc3)=O)CCC1CN(C(=O)C(F)=CCCF)C2 48820,CCC(C)C(O)C(C)C(=O)N1CCN(CC(=O)NCc2ccc([N+](=O)[O-])o2)CC1 48821,C#Cc1cnn(CC(N2CCC(NC(=O)Cc3n[nH]c(=N)s3)C2C(C)C)=O)c1 48822,C1CC(C)N1.C(CCCC)N(C(=O)NC1C(=C)C1)C 48823,C=C(C)C(CC(=O)N1CCCCC1CNC(c1cnn(CC2CC2)c1)=O)OCC 48824,C(=O)(C(CN=[N+]=[N-])NC(C12CCCC1C2(F)F)=O)N(C1CC2(CCC2)C1)C 48825,Cc1cncc(C(=O)NCCC2CC(NC(C3CCCC3CC(C)C)=O)C2)c1 48826,O=C(CC1CN(C(c2ccc([N+](=O)[O-])cc2)=O)C1)N=c1cc(C2CC2)[nH][nH]1 48827,C(CC(C)C)(C(=O)N1CC(O)(C(C)NC(c2cc(C(C)C)[nH]n2)=O)C1)OC 48828,C(=O)(C1CCc2ccccc21)NCc1c(NC(c2c(C)con2)=O)c[nH]n1 48829,N1(C(C2CCC(C)CC2)=O)CCN(C(c2ccccc2F)=O)CC(C)(F)C1 48830,C1(C(=O)NCc2c(C(=O)NC3(CC#C)CC3)c[nH]n2)CCNC(=O)C1 48831,c1(NC(c2cccc(OCCC)c2)C)cc(C)c(NC)cn1 48832,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(CC2CC2)CCC1)=O 48833,Cc1cccnc1C=CC(N1CC(O)CC1CNC(=O)C#CC1CCC1)=O 48834,CS(=O)c1ccc(C(N2CCC(C)(C)C2CNC(=O)Cc2nc[nH]n2)=O)cc1 48835,C1(CC(=O)NC2CC(NCc3cccc(-n4cccc4)c3)C2)CC2(CC2)CO1 48836,C(=O)(C1COc2ccc(Cl)cc21)NCC1CN(C(c2ccn(C)c2)=O)C(C)(C)C1 48837,CC(C)(O)CCCNC(C1CCN(C(C2(N(C)C)CC(O)C2)=O)CC1)=O 48838,c1(OCC)ccc(CC(=O)NCC2(NC(C3(C)CCCCC3)=O)CCOC2)cc1 48839,C(C1CN(C(C2(COC)CC2)=O)Cc2ccccc21)NC(C1(OC)CCCC1)=O 48840,c1(CC(N2C(CN(C)C(c3cnc[nH]c3=N)=O)CCC2)=O)ccc(Cl)nc1 48841,C1(C(N2CC(N(C)C)C2)=O)CC(N=[N+]=[N-])CN1C(c1sccc1Cl)=O 48842,NS(=O)(=O)CCCC(=O)NCC1CCCCO1.C12CCCCN(C1)C2 48843,N1(C(C(CC)F)=O)CCOC(CN(C)C(c2csc(-c3ccsc3)n2)=O)C1 48844,C(=O)(CCCC(=O)OC)N1CCN(C(C(CN(CC)CC)F)=O)CC1.C(N)=O 48845,C(C1CCS(=O)(=O)c2ccccc21)OC(c1c[nH]c(=O)c2ccncc12)=O 48846,C(F)(F)(C(=O)NOCC1CCCC1)C1CCN(C(=O)NC2COCCC2O)C1 48847,CN1CC(C)(C(=O)NCCC2CN(C(=O)Cc3cnc[nH]3)CCO2)CCC1=O 48848,C(N=c1[nH]cnc2c(Br)cccc12)C1(O)CN(C(c2cc(C3CC3)ns2)=O)C1 48849,C1(NC(c2cncs2)=O)CCCOC12CCN(C(c1cc(Cl)nnc1Cl)=O)CC2 48850,n1(C2CCC(NC(=O)NCc3nnc(CSC)s3)C2)ccc(O)nc1=O 48851,C(C)(C)(CCC(=O)N(CC(N1CCCC(CN=[N+]=[N-])C1)=O)CCF)OC 48852,N1(C(CN(C)C)=O)CCN(C(=O)CC2CC2)CC1C(F)F.C1CCNCC1 48853,C1(C(=O)NCCC(CC)CO)CN(C(C2CC(C)CCO2)=O)CC(C)(C)C1 48854,c1(OC)ccc2cc(C(=O)N(CC(=O)N(C(C)(C)C)C)C)[nH]c2c1 48855,Cc1c(-c2cnccc2CCNS(=O)(=O)c2cccc(Cl)c2)cccc1[N+](=O)[O-] 48856,C1(CNC(c2cc(C)ncc2C)=O)CN(C(=O)C(C)N(C)C)C2(CCC2)C1 48857,O=C1Cc2cc(C(=O)NC3CC34CC(NC(=O)Cc3cncs3)C4)c(Cl)cc2N1 48858,c1(C(N2C(C)C(NC(=O)C(C)Cc3cnc[nH]3)CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 48859,CC(C)C(C(=O)NCc1nc(C(=O)O)cs1)c1ccnc(C(=O)O)c1 48860,Cc1nccnc1N1CCN(c2nnc(-c3ccnn3C)n2C2CCCC2)CC1 48861,C(C(CC(F)(F)F)NC(=O)Cc1cncnc1O)NC(c1n(CC)nnc1)=O 48862,C1(NC(CC=C=C)=O)CC(O)CN(C(c2ccc(C3CC(F)(F)C3)cc2)=O)C1 48863,CC(C)(C)C(CCOC(=O)Cc1ccc(Br)c2cccnc12)C(F)(F)F 48864,C1(=O)C(C)(C)CC2(C3CN1C3)CC2.C(C)(C(=O)N(C(C)C)C1CC1)OCOC 48865,C1(NC(C2C(C)C2(F)F)=O)CCCN(C(C23CCC2CC3)=O)C1 48866,N1(C(CC(C=C)(C)C)=O)CCC(NC(=O)C2=C(C)CCCC2)C(F)(F)CC1 48867,c1(-c2cn(CCN(C(=O)C(c3cccnc3F)(C)C)C)nn2)cnccc1Cl 48868,c1(C(N(CC(N2CCN(C3CCOC3)CC2)=O)CCOC)=O)cc2ncccc2o1 48869,c1(C(=O)NC(C2CN(C(c3cc(CC)c(CC)o3)=O)C2)C)c(N)ccc(F)c1C 48870,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3ccco3)=O)C1C2 48871,C(C)(c1ccc(C)cc1)=CC(N1CC(N(C(c2ccc(CCC)[nH]2)=O)C)C1)=O 48872,C(c1ccccc1Cl)=C(C(N1CC(CNC(CN(C2CC2)CC)=O)OCC1)=O)C 48873,CCN=C(NCc1ccc(C)cc1)NC1CSCC1C 48874,CSC1=C(C(=O)N2CCN(C(=O)CCC#N)CC2C2CC2)CCCC1 48875,C1(CNC(c2ccn(C)c2)=O)CCCC(C)O1.C12CN(C1)C(=O)C=CC2C 48876,c1(NCCC(CNC(=O)OC(C)(C)C)OC)ccc2occ(C)c2c1 48877,N1(C(C(C)(C)C)=O)CCC(NC(=O)CC2COC(=O)C2)C(F)(F)CC1 48878,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 48879,N1(C(CCSCC)=O)CCN(C(C2(C)CC2)=O)CC1c1cnn(C)c1 48880,C1(OC)CC(CNC(=O)C(C)C)N(C(C2CCN(c3ccncc3)C2)=O)C1 48881,N1(C(Cn2ncc(C#C)c2)=O)CCN(C(=O)C2=CC(C)C2)CCC1C 48882,C(CCCC(=O)NC12CCC1CN(C(=O)CCN(C)C)C2)(OC)OC 48883,N1(C(C2(O)CC(C)(C)C2)=O)CC2=C(C1)CN(C(c1ccc(NC=O)cc1)=O)C2 48884,N1(C(c2ncn(C)n2)=O)CC(F)CC1CNC(=O)CC1CCC2CC12 48885,c1(C(=O)OC)ncc(SC)cc1F.C12CCN(C1)C(=O)CO2 48886,c1(C(=O)NCC(CCCC)NC(=O)CC(=O)N(C)C)cc(F)c(F)cc1Cl 48887,c1(C(N2CCN(C)C(CO)C2)=O)cc2ccccc2s1.C1(=O)NNC(=O)C2CCN12 48888,c1(OC)ccc(C(=O)O)c2c1CNCC2.c12ccc(cn1)CNC2 48889,c1(C(C(=O)NC2CCC2)N(C(C=C)C2CC2)C)cccc2nn(C)nc12 48890,N1(C(C2(C(C)=O)CC2)=O)CCC2(CC1)CCN(C(c1c(C)ccnc1C)=O)CC2 48891,n1(CC(=O)N(CC(CN(C(CC(C)n2ccnc2)=O)C)O)C)cnc([N+](=O)[O-])c1 48892,c1(CNC(C2(CC)CCOC2)=O)ccc(NC(=O)C(C)CC2CCCC2)cc1 48893,c1(CSC)ccc(NC(=O)C(C(C)SC)c2ccccc2)cc1Cl 48894,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cncs3)=O)c2[nH]1 48895,N1(C(CCCCOC)=O)CCCC(O)(Cn2cc(COC(=N)O)nn2)C1 48896,C1(NC(CC2CC(CC)OCC2)=O)CN(C(=O)C=CC(C)(C)SC)CC2(CCC2)C1 48897,c1(N(C)Cc2c(N)cn(C(C)C)n2)cc(F)ccc1C(F)(F)F 48898,[N-]=[N+]=NC1CCCC(NS(=O)(=O)Cc2ccc(F)c(F)c2)C1 48899,N1(C(c2cc(CCC)on2)=O)CCC2C(NC(=O)CCN(C)C(C)=O)C2CC1 48900,C1(C(=O)NCc2cnc(C)s2)CN(C(=O)CC2CCOC2)CC1(F)F 48901,c1(CC(=O)NCC(=O)NCC2(C)CCN(c3cc(C)on3)C2)c(C)ncnc1O 48902,c1(C(=O)NCC2CCCN(C(CSCC(C)C)=O)C2)ccc([N+](=O)[O-])c(F)c1 48903,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N2Cc1ccns1 48904,C1(NC(c2cccc(C)n2)=O)CC2CCC1CN2C(c1ccn(C(C)(C)C)n1)=O 48905,Cc1cc(Cl)c(C(=O)NCc2ccc(NC(C3(Cl)CC3)=O)cc2)s1.C12CCC1C2 48906,CCCCCC(=O)NCC1(CO)CCN(C(c2nn(CC)nc2C)=O)C1 48907,N1(C(c2cnc(SC)s2)=O)CC2(CC(NC(=O)C=C(C)C(F)F)C2)C1 48908,C1(F)(CNC(COCCC=C)=O)COCCN(C(=O)CCC(C)(F)F)C1 48909,c1(C(N2C(CNC(=O)C(Cl)=CCl)CCC2)=O)ccc2ccnn2c1 48910,CC1CCC(C)(C(=O)NC2CC3(C2)CN(C(c2cnc(C(F)F)s2)=O)C3)C1(C)C 48911,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(c2sccc2OC(F)F)=O)C1 48912,C(=O)(C(C(C)(C)O)NC(C1CCCN(C)C1)=O)NCC1C(C)C1 48913,C(=O)(CCCC(F)(F)F)N1C(CCC)CN(C(=O)COC2CCCC2)CC1 48914,CCCC(CC(=O)N(C)CCN1CCCCC1)NC(=O)CC(O)C(C)C 48915,N1(C(c2c(CNC(C(C)SCC)=O)nccc2)=O)CCC2(CNC(=O)O2)C1 48916,c1(C(=O)NCCC(=O)N(C2CCC2)CCOC)ccnc(C)n1 48917,N1(C(CC=CC=C)=O)CC2(CCN(C(C3CCC(=O)N(C(C)C)C3)=O)C2)C1 48918,N1(C(C(Cc2cccc(OC)c2)N)=O)CCOC(C)(CNC(=O)C(C)(F)F)C1 48919,C1(NC(=O)CCc2coc(CN)n2)CN(C(=O)Cc2cccs2)C2(CCCCC2)C1 48920,c1(CC(=O)NCC2C(CNC(C=CCN(C)CC)=O)C2)cncn1C 48921,c1(C(=O)NCC(Cn2cc(-c3cccc(OC)n3)nn2)(C)C)cc(N)c(F)cn1 48922,C12(C(=O)NC(C)C(C)(C)C#N)CCC(CN(C(=O)CC(C)C(F)(F)F)C1)C2 48923,C1(C(=O)NCC(CC)N(C)CC)CCN(C(=O)CC2(C)CC2)O1 48924,C(=O)(C(C(C)(C)C)OC)N1CC(N(C(CSCC)=O)C)C(c2ccnn2C)C1 48925,N1(C(CN(C(=O)C(C)CCO)CCC)=O)CCCCCC1 48926,CCC(C)(C)CCNC(=O)CC(CNC(C1CCCS1)=O)C1CCC1 48927,C(=O)(C1CCc2c[nH]nc21)N(C)CC1(NC(c2cccc3c2CNC3=O)=O)CC1 48928,c1(C(N2CCC3(NC(COc4cn(C)nc4)=O)C(C2)C3)=O)c(Cl)ccc(F)c1Cl 48929,CC1CC(C)OC1C(=O)NC(C)CCNC(c1ccsc1-n1cnnn1)=O 48930,C(CC(C(=O)NCC(C)NC(=O)CC1CC(C)(C)C1)NC(=O)OC(C)(C)C)=CC 48931,c1(CN(C2CCN(C(c3cc(CCOCC)on3)=O)CC2)C)cccc(F)c1C 48932,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 48933,C(C(CNC(=O)CSc1cnn(C)c1)CO)NC(C1(CCC)CCC1)=O 48934,c1(C(=O)NC2CCC2CNC(C2CC2C(F)(F)F)=O)ccc(F)c(Cl)n1 48935,C(=O)(C1CCCc2nn(C)cc21)NCCCNC(C(C)CC1CCC1)=O 48936,C(CC(C)(C)CC1CC1)NC(C1(C(C)(C)OC)CC1)=O.C1(=O)C(C)N1 48937,c1(C(N2C(CNC(CC(CCSC)O)=O)CC2)=O)[nH]nc2ncnc(O)c12 48938,C1(N(CCC)C(c2ccc(OC)c(Cl)c2)=O)CCC2CC1C2(C)C 48939,CN1C(=O)CCC1C(=O)NCC1CCCC(CNC(c2cscc2Br)=O)C1 48940,C1(NC(C(C)(F)F)=O)CC2CC(NC(C3(c4cncc(F)c4)CCC3)=O)C1C2 48941,N1(Cc2ccc(N(CC)CC)cn2)CCC(NC(=O)CC(F)(F)F)C(O)C1 48942,C(=O)(CCCCCN(C)C)NC(C(N1CC=C(C)CC1)=O)CN(C)C 48943,c1(CN(C(=O)C(=O)N(C)CCN2CCNCC2)C)nnc(O)cc1O 48944,C(C(=O)NCCN(C(=O)COCC1CCC1)C)(C(C)C)NC(C)=O 48945,C1(NC(C2C(CC)C2)=O)CCC(NC(=O)CCOc2ccc(Cl)cc2)CC1 48946,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 48947,CC1CCC(NC(c2csc3cncn23)=O)CN1C(=O)C=CC1CCOC1 48948,c1(CC)ccc(OC(C)C(N2CCC(COC)(NC(c3ccns3)=O)C2)=O)cc1 48949,C(=O)(C1=CC(O)CCC1)NC1CCN(C(C2CC(C)(C(=O)OC)C2)=O)CC1 48950,Cc1csc2c(NCC3CCN(C(c4cc(Cl)cc(Cl)c4O)=O)C3)ncnc12 48951,c1(OC)cccc(C(=O)NCC2(O)CCN(C(c3ncccc3N)=O)C2)c1 48952,C1(NC(c2cn(CC=C)nn2)=O)CCN(C(=O)CC2(C(F)F)CC2)CC1C 48953,N1(Cc2cnc(C)s2)Cc2ccccc2C1C(=O)Nc1ccc2nncn2c1 48954,c1(CNC(c2cnc(Br)n2C)c2n(CC=C)nnn2)cccc(COC)c1 48955,c1(NC(C(C=C)O)=O)cccc(NC(=O)NC(C)C)c1 48956,N1(C(c2c(C)c(F)c(F)cc2)=O)CCC2CN(C(c3coc(Cl)c3)=O)CC2C1 48957,C(=O)(CCCC(F)(F)F)NCc1cc(C(=O)NC(CC(C)O)C)sc1 48958,c1(C(N2C(NC(=O)NCC3CCCC(OC)C3)CCC2)=O)cc2c[nH]cnc-2n1 48959,Cc1c(C(N2CCC(C(=O)NCCc3noc(=O)n3C)(C(C)C)C2)=O)nnn1C 48960,Cc1cc(C(=O)NC(C)CCNC(=O)C2=CCCC2)cc(Cl)c1 48961,c1(C(=O)NC(CC)CNC(c2cn(C)c(C)n2)=O)ccc(C(=O)OC(C)C)cc1 48962,C(=O)(C(C)(C)C1=CCSCC1)NC1CC(OC)CN(C(=O)Cc2nc[nH]n2)C1 48963,c1(C(=O)NCc2cccc(F)c2)ccc(F)c(S(=O)(=O)N2CCC2)c1 48964,N1(C(C=CC=CC)=O)CC2CC(NC(c3cc[n+]([O-])cc3)=O)CC2C1 48965,C1(C(=O)NC2(CC=C)CN(C(C3(CF)CC3)=O)C2)CCCCC1C1CC1 48966,c1(C(N2CCN(C(Cc3scc(CC)n3)=O)C3C2C3)=O)ccc2n[nH]cc2n1 48967,CC1CC(CNC(=O)COC2CCC2)CCN1C(c1ncoc1-c1ccco1)=O 48968,C(=O)(C(F)CCC(C)C)NCC(CC)(CC)C(=O)NCC1CC=CCC1 48969,C1(CC)CN(C(=O)C(O)C(F)(F)F)CCC1NC(c1cc(O)ccc1C)=O 48970,N1(C(C(=Cc2ccco2)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 48971,C1(NC(c2c(C)scn2)=O)CCCC(N(C(=O)CC2CCC(C)CC2)C)C1 48972,C1(C(=O)NC2CC3C=CC2C3)CCCN(C(=O)CN2CC(=O)NC2=O)CC1 48973,c1(CNC(C2CC(O)CN2CC2(CN)CC2)=O)ccc(-n2ccnc2)c(F)c1 48974,c1(C(=O)NC2(C)CCN(C(C3CC(C4CC4)=NO3)=O)C2)csc(=NC2CC2)[nH]1 48975,Cc1cnc2cccc(C(N3CC(NC(=O)COCCCF)CC(F)C3)=O)n12 48976,CC(C)(C)CCC(N)CNCCc1cnccc1Cl 48977,C(=O)(CCCS(C)(=O)=O)NC1CC(F)(C(=O)OCc2c(C)cccc2)C1 48978,c1(OC)cc(F)ccc1C(=O)NNC(=O)N1CCCC1(c1ccc(F)cc1C)C 48979,N1(C(CCCO)C(F)(F)F)CCc2cc(CC(c3ccccc3)=O)ccc21 48980,CC1=C(C(=O)N2CCC(C)C(CNC(c3nccnc3N)=O)C2)CCS1(=O)=O 48981,C1(C#N)(C(=O)NCc2cc(C)n(-c3ccc(F)cc3)n2)CCCCCCC1 48982,c1(C(=O)NCCOC2CCN(C(C(C)SC)=O)C2)nn(C)cc1Br 48983,Cc1cn(C)cc1C(=O)N(CC(=O)NCCOCC(N)=O)C1CC1 48984,N1(C(CCn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CCNC3=O)=O)CC2C1 48985,C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(=O)Cc2cnnn2C)C12CCCC2 48986,C(=O)(C1=NN(C(C)C)C(=O)CC1)N1CC2C(C#C)(CC2)C1 48987,CC(C(=O)NCCC1CC(NC(=O)CSc2cccc(Cl)c2)C1)C(F)F 48988,N1(C(CC2CC(=C)C2)=O)CC2(NC(c3cnc(CC4CC4)s3)=O)CC1C2 48989,c1(OC)ccc(CC(=O)NC2CCCC2NC(C2CN(C)CCO2)=O)cc1Cl 48990,CCC(C(=O)N1CCN(C2CN(C(c3nncs3)=O)C2)CC1)C(C)C 48991,C(C(=O)NOCCC(F)F)(C1(C(N)=O)CC1)NC(C(C)N(C)C)=O 48992,c1(C(N(CCNC(CC(c2ccc(F)cc2)C)=O)C)=O)cnc2cccc(C)n12 48993,C(=O)(CC(C)(C)C(F)F)NC1C(NC(C(C)S(N)(=O)=O)=O)CCC1 48994,CN1CCN(C(c2ccc(O)cc2)=O)C(CNC(c2cc3ccsc3s2)=O)C1 48995,Cc1nc(Cl)[nH]c(=NCC2CN(C(C3(C)CCC(=O)N3)=O)CC2C)c1F 48996,N1(CC(=O)N(C(CC)C(=O)OC)CC)CCN(C(C2CCC3(CCC3)O2)=O)CC1=O 48997,C#CCCCCCC(=O)N1CC(C)(C)CCC1CNC(c1cnn(C)c1Br)=O 48998,N1(C(CC(=O)N(C)C)=O)CC2CCC(C1)C2CNC(C1CCCC2CCCN12)=O 48999,c1(C(N(CC(C)NC(C(C)NC(=O)OC)=O)C)=O)c(C)nn(C)c1OC 49000,c1(CN2C(CNc3cc(C(=O)OC)cc(Cl)c3)CC3CC32)c(F)cc(O)cc1F 49001,Cc1cc(C)c(C(=O)NCC(C)N(CCCCNC(=O)NC(C2CCC2)=O)C)s1 49002,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49003,c1(NC(=O)OC(C)(C)C)cnc2nncn2c1NC(C1CCCO1)=O 49004,C(CC(=O)N1CC(n2cnnn2)C1)(C(F)F)NC(CC1C=NN(C)C1=O)=O 49005,C1(O)(CNC(c2cc(CCNC(=O)Cc3ccc[nH]3)on2)=O)CCCCC1 49006,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(CO)CCC2CC2)C)nn1C 49007,C(C)(CCC(=O)NCC1CCC(F)(Cc2cccc(F)c2)C1)OCC.C1(=O)CN1 49008,C(=O)(CC(C)P(C)(C)=O)NC1CCCC(C(=O)NCCCCC(C)C)C1 49009,C1(CC(=O)NCCOCCNC(C(C)NC(CC)=O)=O)C(=O)NN=C1C 49010,C(=O)(C(C)C(F)(F)F)NCCN(C(=O)C(C)COC)CCC=C 49011,c1(C(N2CCC(O)(CCNC(CC3(C)CCC3)=O)C2)=O)ccc2nn[nH]c2c1O 49012,C1(CCOC)CN(C(c2cnc(O)n2C)=O)CCN1C(c1[nH]cnc1C)=O 49013,N1(CC(=O)NCC2C(N(C(=O)CCCc3cccs3)C)CCC2)CCCOC1=O 49014,C(=O)(CC(=O)N(CCNC(=O)C(C)(C)C1CC1)CC)OCC.O 49015,C1(C(=O)NC23C(CN(C(c4[nH]cc(C)c4)=O)C2)C3)CCc2ccc(F)cc2C1 49016,c1(C(=O)NC(CC)CNC(c2csnn2)=O)cc(N)c(N)cc1F 49017,N1(C(COCCCCC)=O)CCN(C(c2cn[nH]c2)=O)CC1C1CC1C1CCOC1 49018,c1(C(N2CC(CC(C)NC(C3CCCN3N=O)=O)C2)=O)ccc(C#N)nc1O 49019,c1(C(N2C3(CNC(C4C(C)(C)C(O)C4)=O)CC(C2)C3)=O)cc(S(C)(=O)=O)co1 49020,CC(C)(C)C1=NOC(C(N2CC(NC(c3snnc3C3CC3)=O)CC23CCC3)=O)C1 49021,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49022,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49023,C12(C(=O)NC(C3CCCO3)CC)CCC(CC1)N(C(=O)C(=CC1CCCC1)C)C2 49024,C(=O)(CCC(=O)N1CC(N2CC(NC(C3CC3(Cl)C(C)C)=O)CC2)C1)NCC 49025,S(=O)(=O)(CC(=O)NC1CC(CCNC(C2CCN(CC(C)C)CC2)=O)C1)NCC 49026,C1(C(=O)OC)CC(n2cc(C3CCOC3)nn2)CN1S(=O)(=O)CC.C1(O)COC1 49027,c1(OC)cccc(C=CC(=O)N(C2CCC(NC(=O)C(N)=O)C2)C)c1OC 49028,c1(C(=O)NC2CC(CC(=O)NC(C=C)(C)C)C2)cn(C)nc1SC 49029,c1(C(=O)NC(CNC(=O)CN(CCCCOCC)C)C)cccc(C(F)F)c1F 49030,c1(C(C)C)nc(C(N2CC(CO)(NC(C3CCC3CF)=O)C2)=O)co1 49031,C(C)(C)(CCC(=O)N1CCN(C)CC1CNC(C1(c2cc(C)no2)CC1)=O)OC 49032,c1(C(=O)NC2C(C(=O)NCc3nnc(C#N)s3)CCC2)cccc([N+](=O)[O-])c1 49033,c1(C(=O)OC(C(=O)NC2(SCC)CC2)(C)C)nc2ccccc2cc1Cl 49034,C1(C2(O)CN(C(=O)C(C)=CC(C)(C)C)C2)(CNC(C(C)N(C(C)=O)C)=O)CC1 49035,C1(C(=O)NCC(=O)NC2CCOCC2)CCCN1C(=O)C(C1CCCCC1)F 49036,c1(C(N2C(CNC(C3C(OC)C3)=O)CC2)=O)nnn(-c2cccc(Cl)c2)c1C 49037,C1(NC(c2cncc(OCCOC)c2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1F 49038,C1(C(N(c2cccc(-n3cccc3)c2)C)=O)C=CCCN1C(=O)C(C)CO 49039,N1(C(c2nc(NC(=O)OC(C)(C)C)sc2)=O)CC2C(CC1c1ccco1)N=N2 49040,c1(OC)cc(NC(=O)CC2CC(Oc3cn(C)nc3)C2)ccn1 49041,C(N=c1[nH]ccn2cnnc12)c1cn(-c2ccc(F)cc2)nn1 49042,C1(CNC(=O)CSC2CC2F)CCN(C(C2(c3nc[nH]n3)CCC2)=O)CC1 49043,C=Cc1cnn(C)c1C(N1CCN(C(=O)C(N2CCOCC2)C2CC2)CC1)=O 49044,CC1CC2CN1NC(=O)C(=O)NC2.C1(C(=O)N(C)C)(CNC2CC2)CC1 49045,Cc1ccc2c(c1C)N(C(C1(C(=O)O)CCCCC1)=O)CCC2 49046,C(CCC(O)C(=O)Nc1ccc(C)nc1)NC(C(C)=C1CCCC1)=O 49047,n1(C2CC(C)C2)ncnc1Cc1cc(C)sn1 49048,c1(-c2ccc(C)nn2)ccc2cc(CNC(C3C4COCC34)=O)[nH]c2c1 49049,C1(C(N2CCC(N(C)CC)C2)=O)CC(F)CCN1C(=O)CCC(C)OC 49050,C#CCC(C(=O)NCC(C)NC(c1csc(Cl)n1)=O)C1CC1 49051,N1(C(c2nc(C)c(C)s2)=O)CCC2(NC(=O)CCc3cccnc3Cl)CCCC12 49052,c1(C(C)NC(CSCCC)=O)nocc1C(=O)NCC(F)CO 49053,c1(C(N(C2CCN(C(C3CCSC3)=O)CC2)CCO)=O)cnc2c[nH]nc2c1 49054,C1(C(=O)NC(c2nc[nH]n2)C)CC(NC(=O)Cc2ccoc2)CCO1 49055,N1(C(C2(F)C(C)C2)=O)CCC2(CCC2CNC(c2nncs2)=O)CC1 49056,CC(C)CC(F)(F)C(=O)NCC(C)(C)CN(C)C(C1CC1C)=O 49057,CC(C)CCCOCC(=O)NC(C1(C(=O)N(C)CCN(C)C)CC1)C 49058,C1(OC)CCC12CC(C(N1CCN(C(C3CCC(=O)N3C)=O)C(C)C1)=O)C2 49059,c1(C(=O)NCC2CC3(CC(NC(COC(C)(C)C)=O)C3)C2)cnc2n1CCCC2 49060,CC(C)(C(=O)NC1CCCC1)NCCn1ccc(C(=O)C2CC2)c1.c1(S)cc[nH]n1 49061,c1(CNC(C(N2CC(CC)C(O)C2)c2ccc(F)cn2)=O)ccc(Cl)cc1F 49062,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49063,c1(OC(C)C(=O)NCC(=O)NCc2nc(-c3cccnc3)no2)ccccc1F 49064,N1(C(C(n2c(C)ncc2)C)=O)CC2CCC2(CCNC(c2cc(Cl)n(C)n2)=O)C1 49065,C1(C)(NC(N(n2ccnc2)CCOCCOC)=O)CCOC1C 49066,c1(CNC(=O)NCCCN2C(C)CCCC2)ccc2n[nH]cc2n1 49067,c1(C(=O)NC(CC)CNC(=O)CCCOCCOC)cnc(Cl)n1C 49068,n1(CC)nncc1C(=O)N(C(C)CN(C(=O)C(c1ccccc1)N(C)C)C)C 49069,N1(C(c2c(C)nn(C)c2Cl)=O)CC(C)(C)OCC1CNC(C1CCC(=O)N1C)=O 49070,C1(CNC(C2(CCCC)CC2)=O)CCC(C)(C)CN1C(=O)CC1CCC(=O)N1 49071,C=CCC(C(=O)NC1CCSC12CN(C(c1ccc(Cl)o1)=O)C2)C(C)C 49072,N1(C(c2ccn(COC)n2)=O)CCc2sccc2C1CNC(C1CCC1)=O 49073,C1(c2c(OC)cccc2)CCCN(C(=O)C(C)C(=O)OC(C)=O)CC1 49074,C1(NC(c2nnn(C)n2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)CC12CCC2 49075,C(=O)(C(C)(C)CCCF)N(CCCCCNC(C(C(C)C)OCC)=O)C 49076,CC12CCC(C(=O)NCCCNC(=O)C(C)(C)c3cnc[nH]3)(CC1)CO2 49077,C1(C(=O)NC2(C)CN(CC(F)(F)F)C2)C2CN(Cc3ncccc3F)CC12 49078,N1(C(c2ccn(CCCC)n2)=O)CCC2CN(C(C3CC4(CC4)CO3)=O)C2C1 49079,C1(NC(C=C(C)C(C)C)=O)CCN(C(C2CNC(=O)C(C)(C)C2)=O)CC1(C)C 49080,c1(C(=O)NCC2CN(C(C(CCC#C)O)=O)C2)ccc(Br)c2nccn12 49081,c1(CNC(=O)OCC#C)ccccc1COC(=O)C=Cc1cccs1 49082,N1(C(C2SCCS2)=O)CCCC1C1CCCN1C(C1CC(F)(F)C1)=O 49083,C1(C2N(C(C(C3CCOC3)NC(C(C)O)=O)=O)CC2)CC(F)(F)C1 49084,C1(CNC(C)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49085,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49086,CCCC(C)CC(=O)NC1CCCC(NC(c2cccn2C)=O)C1 49087,C(=O)(C(O)C(C)(C)C)N(C1CCN(C(=O)C2=CCCCC2)CC1)CC(C)C 49088,c1(C(=O)NCC2CN(C(C3N(S(CCC)(=O)=O)CCC3)=O)C2)nccc(C)n1 49089,C(=O)(C1=CS(=O)CCC1)NCCCN(C(C)C)C(C1CCCN1N=O)=O 49090,CCC(C)(COC)C(=O)NCc1ccccc1CN(C(=O)C(C)C(F)F)C 49091,c1(C(N2CC(N(C(c3n(CC)ncn3)=O)C)C(F)C2)=O)ccc2c(c1)COC2 49092,c1(C(=O)OCC(C)CCO)ccc2c(c1)OC(F)(F)O2 49093,N1(C(C(c2cnn(C)c2)C)=O)CCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 49094,c1(OCCC#C)ccccc1C(C)N(C)Cc1sc(Br)cc1Br 49095,CCCCC(C)C(=O)NCC(C1CC1)NC(=O)C(F)(F)c1nc(C(F)(F)F)cs1 49096,C1(NC(=O)Cn2ncnn2)CCC(NC(c2ccnn2CCF)=O)C1 49097,CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)COc1ccc(Cl)cn1 49098,C1(CNC(C2(COC)CC=CC2)=O)CN(C(=O)OC(C)(C)C)CC12CCC2 49099,C=Cc1ccc(NC(N2CCSC(C(F)(F)F)C2)=O)cc1 49100,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC(C)(N(C)CC)C2)=O)C1 49101,CN1CCCC(CCC(=O)N(C)CC2CCN(C(C3(O)CCC3)=O)CC2)C1 49102,c1(OCC(=O)OC2CC(C(=O)OCC3N(S(CC)(=O)=O)CCC3)C2)cccc(C)c1 49103,C#Cc1ccc(C(=O)N(CC(C)O)CCNC(c2ccc(C#N)o2)=O)cc1C 49104,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49105,c1(C(=O)NCC(C(=O)N(C2CCC(C)(C)C2)C)N(C)C)ccc([N+](=O)[O-])o1 49106,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(CO)C(N)=O)C(C2CC2)C1 49107,C1(C)(C(=O)NCCN(C(C(CC)F)=O)C2CCCC2)C(C)(C)C1(C)C 49108,Cc1cc(C(N2CC3C(N(C(=O)CC4CCC(C)(C)C4)C)C3C2)=O)n(C)n1 49109,CCC(C(F)(F)F)NC(c1ccn(CCNC(C2COCC(C)O2)=O)c1)=O 49110,CC(C)C(C(=O)NC(C1(CNC(C2CCO2)=O)CC1)C)n1ccnc1 49111,c1(CN(C)C(=O)Nc2ccc(-c3ncon3)cc2)ccc(F)c(Cl)c1F 49112,c1(C(=O)NCC23CC2CN(C(C2CN(C4COC4)C2)=O)C3)ccc2snnc2c1 49113,c1(OC)ccc(C(=O)NC(C2CCCN2C(c2coc(O)n2)=O)(C)C)c(O)c1F 49114,CCC(C)(C)C(=O)C(=O)NCC(C1CCCC1)NC(=O)Nc1ccnc(OC)c1 49115,C1(SC)CN(C(c2noc(C3CC3)c2C)=O)CC1NC(C1CC12CCOC2)=O 49116,C1(C(N2C(CN(C(Cc3ccc(C)nc3)=O)C)COCC2)=O)CN(C)CC(C)O1 49117,N#Cc1ccc(C(N2CC(CF)(NC(=O)C=Cc3cscn3)C2)=O)s1 49118,C1(NC(C2(CC)CNC(=O)C2)=O)CC(C(=O)NCC2CNC(=O)CO2)=CC1O 49119,c1(CC(=O)NCCCC(C)N(C)C)ccccc1C(=O)OC.C(=O)(CC(=O)N(C)C)N 49120,C1(C(=O)NCC(CNC(=O)CCCC2CCCC2)F)CCCC(C(=O)OC)C1 49121,c1(C(=O)OC)cc(CC(=O)NC2CC2NC(=O)CC2(C)CCCCC2)ccn1 49122,C1(NC(c2cnc(C(C)(C)C)o2)=O)CCC(O)CN(C(=O)CCCCCC#N)C1 49123,C(=O)(CC(C)CCC)NCC1N(C(CN(CC=C)C(=O)OC)=O)CC1 49124,CCC(CC(=O)NC(CC1CC1)C(=O)OC)NC(=O)CCc1cn(C)nn1 49125,C1(CCC)(NC(=O)CC2CC3C=CC2CC3)CCCN(C(=O)Cc2nc[nH]n2)C1 49126,CCCCC(CNC(C1CCOC1CNC(C1(F)CCC1)=O)=O)CC 49127,C1(C(=O)NC(C)Cn2cc(C3(C)CNC3)nn2)CCC2CCCC12 49128,c1(OC)cccc(CNC(=O)CCNC(=O)C(F)(F)Cl)c1Oc1ccc(F)cc1 49129,c1(COC)nc(NCCC2CC(=O)N(C)C2=O)cc(=NCc2cccs2)[nH]1 49130,c1(C(=O)OC)ccnc(CC(N2CCC2CNC(C2(OC)CC2)=O)=O)c1 49131,S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)N1CC2CN(C(CCC=C)=O)CC2C1 49132,c1(OCC(Cc2ncn(C)n2)O)ccc(-n2cccn2)cc1 49133,c1(CC(=O)N(c2ccsc2)C2CC2)ccn(C2CC2)n1.C12CCN(C1)C2=O 49134,N1(C(c2cc(-c3cccnc3)on2)=O)CC2(CCN(C(C3(CCF)CC3)=O)C2)C1 49135,C1(CC(N2C(C(=O)NC3CN(C(C)C)C(=O)C3)CCC2)=O)Cc2ccccc2C1 49136,C1(N(C)C(c2cnc[nH]2)=O)CCN(C(=O)CCF)CC1 49137,N1(C(c2n(C)cc(Br)c2)=O)CC2(CCC2)CC1CNC(=O)C=CS(C)=O 49138,c1(C(N(C2CN(C(=O)C(F)OC(F)(F)F)C2)C)=O)cc(-c2cccs2)[nH]n1 49139,C1(C2CCN(C(=O)C=CC3CCC3)CC2)(NC(c2cc(OC)no2)=O)CC1 49140,C(=O)(CCCCCC)NC(CNC(C12OCC(COCC)(C1)C2)=O)CC(C)C 49141,c1(CC(N2CC(C)C(NC(C3(C)CNC(=O)C3)=O)C2)=O)ccc(F)cc1C(F)(F)F 49142,C(=O)(CCC(=O)c1cc(C)sc1C)NCCN(C(=O)CC1CCS(=O)(=O)C1)CC 49143,CC(C)CC(F)(F)C(=O)N(C)CCNC(=O)C(c1ccc(Cl)c(F)c1)O 49144,O=C(CC(C(F)F)NC(C1(F)CC1)=O)NCC1(F)CCOCC1 49145,CN1CCCC(F)(C(=O)NCC2(NC(c3cccc(F)c3O)=O)CCC2)C1 49146,C1(C(=O)NCCCN(C(C(c2ccccc2)OCC)=O)C2CC2)CCCC1F 49147,C(=O)(N1OC2CCC1CC2)C1(F)CCN(C(C(CO)N(C)C)=O)C1 49148,C1(NC(c2c(C)cno2)=O)CN(C(C2CC2c2ccccc2F)=O)CCC1C 49149,C1(C)(C(=O)NCC2(OC)CCN(C(c3cc(=O)n(C)cn3)=O)C2)CC(=O)N(C)C1 49150,C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CN1CCC(C)C1)C2)c1c(OC)cccc1 49151,C(=O)(CCC(F)(F)F)NC(c1cccnc1)C(=O)NCc1ncc(COC)o1 49152,C(=O)(C1CCSc2ccccc21)NCC(CNC(=O)CSCC(N)=O)OC 49153,N#Cc1c(C(=O)NCC2(O)CCN(C(=O)CCC(=O)NC(N)=O)C2)cccc1F 49154,c1(C(=O)NCC(C)C(=O)N2CC=CC2CF)cn(C)ccc1=O 49155,N1(C(C=CC)=O)CCC(C)(CNC(c2ccc(N(C)CC)nc2)=O)C1 49156,Cc1cc(F)c(C(c2nnnn2C2CCCCC2)NC2CC(C)C2)c(Br)c1 49157,c1(OC)ccc(CC(=O)NCCC2CCCN(C(C3(CC(C)=O)CC3)=O)C2)cn1 49158,C(=O)(CCS(N)(=O)=O)NCC1(C)N(C(c2nccnc2OCCOC)=O)CCC1 49159,C(=O)(CCCCC(C)(C)C)NC(CC#C)(C)C(=O)N(C)CCC1CC1 49160,CCCCC(CNC(=O)C#CCNC(=O)CNC=O)CC 49161,C1(C(=O)NC2CCN(C(c3snc(O)c3Cl)=O)C2)CCc2c[nH]nc2C1 49162,Cc1cc(O)ncc1C(=O)NC1C2CC1N(C(c1sccc1OC(F)F)=O)C2 49163,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc(O)ncn2)=O)CC1C 49164,C1(NC(CCS(CC)=O)=O)CCC(O)CN(C(=O)Cn2nnc(C3CC3)n2)C1 49165,C(=O)(CCC(=O)N(C)C)NC(C)C(c1cccc(O)c1)NC(c1nccs1)=O 49166,N1(C(CC(C)CF)=O)CCN(C(=O)CCC2OCCO2)C(CS(C)(=O)=O)C1 49167,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49168,c1(OC(C)C(N2CCC(C)C2C(=O)Nc2ccc(O)nc2)=O)cc(Cl)cc(Cl)c1 49169,Cn1cc(C(F)=CC(N2CC(NC(=O)CNC3CC3)C3(CC3)C2)=O)cn1 49170,C(=O)(C(CC(C)C)C(C)C)NC(C1OCCN(C(C2CCC(CC)O2)=O)C1)C 49171,c1(OC)ccc(OC)c(CN2CC3C(C2)N3C(c2ccn(C3CCCC3)n2)=O)c1 49172,c1(C(=O)NCCC2N(C(Cn3ncc(C)c3)=O)CCC2)cncc2cnccc12 49173,C12(C(=O)N(CC=CC(=O)NCCC3CCC3)CC3CC3)CCC(O)(CC1)C2 49174,CCCCCC(F)C(=O)N1CCC(c2cn(Cc3n[nH]cc3C)nn2)CC1 49175,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(CF)C2)=O)CCO1 49176,C1(CNC(c2c(C)nc[nH]2)=O)CN(C(=O)C(C(C)C)n2cncn2)CCN1C 49177,C#CC1CCCN(C(=NCCO)NCC(CC=C)CC)C1.C1(C)CC1 49178,C1(CCC)CN(C(=O)C(C)OCC)CC1NC(=O)C(c1ccc(F)cn1)(F)F 49179,C=CC(C(=O)NCC1CCCN1C(C1CC1CC(C)C)=O)c1ccccc1 49180,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NC(c2nc[nH]n2)(C)C)C1 49181,c1(OC)ccc(CC(=O)N(C)CC2CN(C(=O)Cc3ccsc3)CCO2)c(F)c1 49182,c1(C(C)OCC)nc(CN(CC(C)NC(=O)C=C(C)Cl)C)cs1 49183,C(=O)(NNC(=O)NC(F)(F)CF)c1c(C)ncs1 49184,N1(C(c2c(CC)n[nH]c2)=O)CC2=C(C1)CN(C(C1OC3CCC1C3)=O)C2 49185,C1(C)(C=O)CCCN(C(c2cccnc2Br)=O)C1.C1(NC(C)=O)(C)CC1 49186,N1(C(CCNC(=O)OC)=O)CCC2CCN(C(C3C4CN(C)CC34)=O)CC2C1 49187,c1(C2(C(N3CC4CCN(C(=O)C=CCO)C4C3)=O)CC2)nccc2ccccc12 49188,C(C)(CCCCNC(=O)CC1(O)CCC1)NC(C(c1ccc(F)cc1)OC)=O 49189,C1(CNC(C(C)OCC)=O)CC2(CCN(C(=O)Cc3ccnc(Cl)c3)CC2)CO1 49190,c1(C(=O)OCCOC(N(C(=O)CCC2CCCO2)C)=O)ccc2cnn(C)c2c1 49191,CC1(C(N2CC(CO)C3(CC3)C2)=O)CC2C=CC1C2.N12CCC(C=CC1=O)CC2 49192,CON(C(=O)c1cc(Cl)cnc1Cl)C1CCCC1 49193,c1(C(=O)NCC23OCC(NC(CNC(=O)OC)=O)(C2)C3)cc(SC)ccc1Cl 49194,Cn1ccc2c(C(N3CC4CCC(NC(c5cnc(O)s5)=O)C4C3)=O)ncnc12 49195,N1(C(c2cnc(C(C)(C)CF)o2)=O)CCN(C(C2C=CCC2)=O)CC1 49196,C1(N(C(=O)CCF)C)CCCC2CN(C(c3coc(C(N)=O)c3)=O)CC12 49197,n1(-c2cn(CC)nc2)nc(CC2CC2)nc1-c1coc(CNC(C)=O)n1 49198,C(=O)(C(C(C)CC)NC(=O)C(C(CC)CC)OC)NCC(C)OCC(=O)OCC 49199,C1(CNC(c2cc(CCC)ncc2)=O)CCN(C(=O)C(C2CC2)OC)CC1O 49200,c1(N2CCC(C(=O)NC3(O)CC(C)(C)C3)CC2)nc(Cl)nc2c(F)cc(F)cc12 49201,Cc1ccnc(CNC(=O)C(O)CCNC(C2CCCCCN2C)=O)c1F 49202,Nc1nc(Cl)ccc1C(N1CCOC(CCNC(C2CCOC2C2CC2)=O)C1)=O 49203,C(=O)(C(O)CC(F)(F)F)N1CCCC(N(C(COCc2ncc(C)o2)=O)C)C1 49204,c1(OC)cccc(OCC(=O)NC2CC2NC(c2coc(Cl)c2)=O)c1 49205,C1(C(N2C3C(NC(c4c[nH]c(Br)c4)=O)C(C3)C2)=O)CN2CCN1CC2 49206,N1(C(C(CC=C)C)=O)C2CCC1CC(C(=O)NC1(C(=O)OC)CC1)C2 49207,c1(C(=O)NCC2CC(NC(c3cc(C4CC4)cs3)=O)C(O)C2)ccnc2c1CCC2 49208,C1(C(=O)Nc2ccc(C#C)cc2)CN(C(=O)CC2CCCCCC2)CCC1(C)C 49209,C1(C#N)(C(N2CCC(C(=O)NC(C)Cn3ccnc3)C2)=O)CC(F)(F)C1 49210,CN=c1nc(N2CCC(C3CCSC3)C2)[nH]c(N2CCOCC(C(C)(C)C)C2)n1 49211,N1(C(c2c(CC)ocn2)=O)CCCC(NC(=O)C(C)(O)c2ccccc2)CCC1 49212,CCC(CC(=O)NCC1CC2CC2C1)NC(=O)C=Cc1cn(C)nn1 49213,C1(CNC(C(C)C)=O)COCC2(CCN(C(C3CC4CC4C3)=O)CC2)O1 49214,c1(OC)cc(C(=O)NCCN2CCCC2)ccc1Cl.C12C3CC1N(C3)C(=O)CS2 49215,Cc1cnc(Cl)c(C(=O)NC2CN(C(c3ccc(OCCF)cc3)=O)C2)c1 49216,N1(C(C2N(C)CCOC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)C(C2)C1 49217,N1(C(C(=O)NCc2cc(C)nc(C)c2)=O)CCNN(c2ccccc2Cl)CC1 49218,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49219,N1(C(CN(S(C)(=O)=O)C)=O)CCC2C(NC(c3sc(F)cc3Cl)=O)CC12 49220,C(=O)(C(C)(F)C(=O)NCCC(C)CCNC(=O)C(O)C(C)C)OCC 49221,c1(SC)cn(C)nc1C(N1CCCC(C(C)NC(C2(O)CCOCC2)=O)C1)=O 49222,N1(C(CC2(C)CC2)=O)CC2CCN(C(=O)CC3CC4C=CC3CC4)CCC2C1 49223,N1(C(C(C)NC(CC)=O)=O)CCC(NC(c2cccc(C3CC3)n2)=O)CC1C 49224,c1(C(N2CCC(F)(C(=O)NC3CCC(F)(F)C3)C2)=O)cc(F)ccc1[N+](=O)[O-] 49225,C(=O)(CCCC1CCCC1)NC(C1CCN(C(c2ccon2)=O)C1)C 49226,Cc1ccc2cc(C(=O)NC3CCCC34CN(C(C3CC3[N+](=O)[O-])=O)C4)[nH]c2c1 49227,C1(C(=O)OC2(CSC)CCC2)CC(C)(NC(=O)CC(=O)OC(C)(C)C)C1 49228,CC(N=c1cccc(S(=O)(=O)N2CCC(O)CC2CO)[nH]1)c1ccc(Br)c(F)c1 49229,N1(C(CCN(CCCCC)CC)=O)CC=CC1CNC(=O)CCN1CCC(F)C1 49230,Cc1ccn2ncc(C(=O)NC3CN(C(=O)CC4CC=CCC4)CC3(C)C)c2n1 49231,c1(C(=O)NCC2C(NC(C3C(C(=O)OC)C=C3)=O)C2)n[nH]c2nccc(Cl)c12 49232,CC1CNCCC1NC(C1CC(CNC(=O)COC2CCC2)C1)=O 49233,N1(C(C=CC2N(C(COCC)=O)CCC2)=O)CCN(C)C(=O)C1C 49234,c1(NC(C(C)OCc2ccccc2)=O)c(C(F)(F)F)ccc(Cl)c1Cl 49235,C(C(N=[N+]=[N-])C(=O)NC1CC(CNC(c2c(CO)cccc2)=O)C1(C)C)OCC 49236,C(=O)(CCS(=O)(=O)N(C)C)NCCC(=O)NCCC1CN(C)CC1O 49237,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(=O)CCc4ccncn4)C3)(C1)C2 49238,c1(C(=O)NCC2CCCCN2C(=O)C=Cc2ccncc2)cnc2c[nH]nc2c1 49239,C1(NC(=NCCCSC)NCC2(C)CC2(Cl)Cl)CCOC2(CCOCC2)C1 49240,c1(CCC)cccc(C(N2CCCCC2c2cc[nH]n2)=O)c1 49241,N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCN(C)CC2)=O)C(CF)C1 49242,c1(CC(N2CCN(C)CC2)=O)c[nH]c2ccc(-c3ccnn3CC#N)cc12 49243,c1(C(N2CC(CCCCNC(C3CCC(OC)C3)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 49244,C#Cc1ccc(F)c(C(N2CC3CCC2CN3C(=O)C(CCC)N(C)C)=O)c1 49245,C1(CC2CCN(C(C)C)C2)CCCCN1C(=O)Nc1ccn(C(F)F)n1 49246,O1N(C)CCCCNC(=O)C1.C(=O)(C(C)CO)N(CC(=O)OC)C 49247,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49248,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49249,c12n[nH]c3c1CN(CC3)C(=O)N2.c1(CCC)ccc2cc1O2.C1(C)CCOC1 49250,c1(C(N2CCC(CC(=O)Nc3nc(CCC)oc3)C2)=O)c(O)cccc1Cl 49251,c1(C(=O)NC2C3CN(c4ncnc5c4CCC5)CC23)cc(=O)c2ccccc2o1 49252,c1(OC)ccc(C2(CNC(=O)NC3(C)CCCNC3=O)CCOCC2)cc1OC 49253,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)ns2)=O)CC1F 49254,N(C1CCOc2ccccc21)(C(=O)CC1CCOC1=O)C1CC1.C1(=O)C(F)(F)N1 49255,CC1C(NC(C2CCCN(C(N)=O)C2)=O)CCCN1C(=O)C(F)=CC1CC1 49256,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49257,C1(C(C)N(CCCO)C2CC2)CCC2CC12 49258,c1(C(=O)NCCC2(O)CCCN(C(=O)C=CBr)C2)cn2cccc(F)c2n1 49259,Cc1cc(Cl)c(Br)cc1CNC(C1CC(O)CN1c1nc(C#N)c(C)s1)=O 49260,C=CC1(C(N2CCC(O)(C(C)C)C2)=O)CCN(C(=O)C(C)N=[N+]=[N-])C1 49261,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49262,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49263,c1(NC(C2CC2NC(N2CCc3n[nH]cc3C2)=O)=O)cccc2nc(Br)sc12 49264,C1(CC)(NC(=O)C=CC2CC2)CCN(C(=O)C(C)OC)CC1 49265,n1(CC)ccnc1C=CC(=O)NC1CC1CNC(C1COCCO1)=O 49266,c1(OC)ccc(CCC(=O)NCC2CCC2NC(C2CC3C=CC2O3)=O)c(F)c1 49267,N1(C(c2cnc(OCC(F)F)c(Cl)c2)=O)CCC2C(C1)CN2C(=O)CCC1CC1 49268,c1(NC(C=CC(=O)OC)=O)nc(C)c(CNC(=O)CS(=O)(=O)N2CCCCC2)s1 49269,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49270,C1(CNC(CC2ON=C(C)C2)=O)CN(C(c2cnccc2Cl)=O)C2(CCC2)C1 49271,c1(C(=O)NC(C(=O)N(C23CC2CNC3=O)C)CCOCCO)cccc(O)c1 49272,C1(C(C)C)C(NC(=O)CCOc2cccc(F)c2)CCN1C(=O)CCCC1CC1 49273,N1(C(CC)=O)CCN(C(c2nncn2CC)=O)CC1c1cnn(C)c1 49274,C1(NC(c2c(CC)non2)=O)CCC(O)CC1.c12cc(n[nH]1)C(=O)N(C)C2 49275,CCCC(C)(O)C(=O)Nc1cccc(NC(C2CC(OC)C2)=O)c1 49276,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCN(C)CC2)C1 49277,C12(C(=O)Nc3cccc(CNC(c4ccc(SC)s4)=O)c3)CC=CC(C1)OC2 49278,c1(N(C)C)cccc(C(N2CC3C(NC(=O)CN4CC(C)(C)C4)C3C2)=O)n1 49279,CC1=C(C(=O)N2CCC(C3CCCO3)C2)CCO1.c12nnc(s1)C(C)N2 49280,CCCC(CCO)NC(=O)C(CC)NC(=O)C#CC(C)C 49281,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49282,N1(C(C=CCC)=O)C2CCC1CC(N(C)C(c1ccncc1Br)=O)C2 49283,S(=O)(=O)(c1c(C)noc1C)NCC(N1C(CNC(C(CC)COC)=O)CCC1)=O 49284,c1(OC)c(C(=O)NC2CCC(NC(C3(C)CCC3)=O)C2)cccc1C(F)(F)F 49285,C1(C)(CNC(C(C2CCCOC2)OC)=O)CCN(c2nc(Cl)ns2)CC1 49286,C1(CCOC)(NC(=O)CC2CC2CO)CCN(C(C2CC2C(C)O)=O)CC1 49287,N1(C(C(COC)OC)=O)CC(CC(N2CCC2(C)COC)=O)C2(CC2)C1 49288,c1(CNC(=O)C(C2CCN(C(c3ccnn3C(F)F)=O)C2)F)cccc(CO)n1 49289,CC(C)C(O)CCNC(=O)CC1CN(C(=O)CCCCC2CC2)CCO1 49290,C(C(CNC(=O)CN1C(=O)CCC1=O)C(F)(F)F)NC(c1c(SC)nn(C)c1)=O 49291,Fc1cccc2nc(N3CCC(C4CC4)C3)[nH]c(=NCCc3nccs3)c12 49292,n1(CCOC)cc(C(=O)N(CCNC(C2CCC(C(=O)OC)C2)=O)C)cn1 49293,c1(OCC(=O)NCC2CCN(C(=O)Cc3cccnc3O)CC2)cc(F)cc(Cl)c1 49294,CCC(C)C(=O)NC(C1(O)CN(C(C2C=C(C)CS2)=O)C1)C 49295,c1(C(N2C(C)C(NC(C3CC4(C3)CC4F)=O)CCC2)=O)cnc2c(c1)CNC2=O 49296,Cc1ccc(-c2nn[nH]n2)c2c1N(CC1(OC)CC3CCC1CC3)CCC2 49297,c1(NC2CC(C=C)C2)[nH]c(=NC2CC3(CCCC3)C2)nc2scnc12 49298,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC=CC=C2)=O)CC1 49299,N1(C(C2C(C=C)CC2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49300,N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCCC(CNC(=O)C(C)CF)CC1 49301,CC1=C(C(=O)NC(CNC(c2ccc(C(C)C)cc2)=O)CC(F)(F)F)CCCO1 49302,N1(C(C2(CCCC)CC2)=O)C2CCC(C2)C1CNC(C1CNC(=O)N1)=O 49303,N1(C(c2ccc(C(C)=O)cc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49304,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)N(CC(=O)NCC)C)C2C1 49305,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49306,C1(NC(C2CC2F)=O)CCN(C(=O)C(c2cccs2)C2CCCC2)CC1 49307,N1(C(C2CC(CCC)C2)=O)CC2CC2(C(=O)Nc2cccc(C(=O)NC)c2)C1 49308,C1(CC(N2CC(C)C(NC(=O)COc3cnn(C)c3)C2)=O)CCC(C)(C)CO1 49309,c1(C(=O)NC2(CNC(C(C)SC)=O)CCOC2)cc2c(C)c(Cl)ccc2[nH]1 49310,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2C)=O)CC1C 49311,c1(OC)cc(N)ccc1C(=O)NCCC(C(C)C)NC(C1CCC(C)(C)CO1)=O 49312,C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49313,c1(OC(=O)CC(C2CN(C(=O)OC3CCCO3)C2)C)ccc(F)c(F)c1F 49314,c1(C(C)(C)C)conc1C(=O)NCCCNC(C1CC(C#N)C1)=O 49315,C1(C2CCN(C(=O)CCC3CCCC3)C2)CCCCN1c1nnco1 49316,CC1CCN(CCCN2CCC(C)(c3ccccc3)C2)CC1C 49317,CC1=NOC(C)(CNC2(c3ccccc3)CC2)C1 49318,C1(CN2C(CC(=O)N(CC(=O)N(C)C)C)COCC2)CN2CCN1CC2 49319,Cc1ccc(N2CC(C(=O)NCC3(N4CCCC4)CCCC3)CC2=O)cc1 49320,c1(N(CC(C)(C)N(C)C)C)nc(N2CCCC(NS(C)(=O)=O)C2)nc2scnc12 49321,CC1CC(=O)NC1C(=O)N(CCCNC(c1cnn(CC2CCCCC2)c1)=O)C 49322,CC1CC(NC(c2cc(C(C)(C)C)on2)=O)CN(C(=O)C2CC2)C1 49323,C12(CNC(c3c(C)n(C4CC4)cc3)=O)CCC1CCN2C(=O)CC1(C)CC1 49324,CCCC(C)(O)CC(=O)NC1CC(C(C)(C)C)CN(C(=O)CCC(C)COC)C1 49325,Cc1oc(C(=O)NC2CCCC2CNC(c2ccc(C(N)=O)cn2)=O)cc1CO 49326,C#Cc1ccc(CC(N2CCOC(C)(CNC(c3cnnc(O)c3)=O)C2)=O)cc1 49327,c1(C(N2CC(C(C)N(C(CCC3C(C)C3)=O)C3CC3)C2)=O)ncsc1C(C)C 49328,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49329,CC1CC(C)(C)CN1C(c1cn(CC2CCOC2)nn1)C(=O)NCC1CC1 49330,C1(NC(C(C)=C(C)C)=O)CCCC(NC(=O)C(F)(F)c2ccnn2C)C1 49331,c1(C(=O)NCC2(OC)CCN(C(=O)CNc3nccs3)C2)ccc(F)c(CO)c1 49332,N1(C(C2CCC(NC(c3n(C=C)ncc3)=O)C2)=O)CCC2(CCC2)C(O)C1 49333,N1(C(Cc2c(C)n[nH]c2)=O)CCC2C(C1)CN2C(c1ccc(NC(N)=O)cc1)=O 49334,c1(N2CCCC(NC(C)=O)C2)ncnc(NCC2CCCC2(C)C)c1C 49335,C1(C(N2C(CNC(C(C)SC)=O)CCC2)=O)CCN(C(c2c[nH]nc2F)=O)CC1 49336,C1(N(C)C(C2(C)CC3(CCC3)C2)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49337,C1(c2nn[nH]n2)(NC(c2c(Br)cnc(SCC)n2)=O)CC(C2CCC2)C1 49338,N1(C(C(C)C2CCOC2)=O)CCOC2(CCCN(C(=O)Cn3cnnc3O)C2)C1 49339,C1(NC(c2cnsn2)=O)CC12CCC(NC(c1cccc(F)c1Cl)=O)CC2 49340,Cc1cnc(C(=O)N(C(c2ccccc2)C(N2Cc3ncsc3C2)=O)C2CC2)c(F)c1 49341,Cc1oc(C(C)(C)C)cc1SCC(=O)Nc1cccc(OC(F)(F)F)n1 49342,CN=c1nc(N2CCN(CCF)CC2)[nH]c(N2CCCC(C)(CO)C2)n1 49343,c1(C(=O)NCCC(C)NC(=O)Cc2ncncc2Cl)cnc2nccn2c1 49344,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49345,c1(CCNC(C2(CNC(=O)COC3CCOC3)CC(=C)C2)=O)ncc(C)cn1 49346,C#CCC(C)(C)C(=O)NCCC1CCC(NC(c2n[nH]cc2OCC)=O)C1 49347,N1(c2nnc(C(=O)OC)s2)CC2CCCC1C2CNC(c1cc(Cl)ccc1F)=O 49348,c1(C(=O)NCC(C)(C2CC2)NC(C(N2CCNC2=O)C)=O)ccc2cc[nH]c2c1F 49349,O=C(CCCCCCCO)NC1CC(CNC(c2nnco2)=O)C1 49350,c1(C(=O)NC(C)CCNC(C2(F)CCCC2)=O)cc(Cl)cc(Br)c1N 49351,N1(C(CCC2N(C(c3cn(CCC)nn3)=O)CCC2)=O)CC2CCC(O)CC2C1 49352,C(=O)(CCN(OC)C(=O)Cn1ccnc1)N(CC=C)CCC 49353,C1(N(C)C(C2CC3CC3C2)=O)CCCCN(C(c2n[nH]cc2I)=O)C1 49354,C(=O)(CC(C)(C)C(=O)NC1CCCCC1NC(=O)CC1CCSCC1)OC 49355,c1(CCC)onc(C)c1C(=O)N(C1CN(C(=O)CCc2ccc(OC)cc2)C1)C 49356,C1(NC(CN(C)C(c2ccsc2)=O)=O)COCCN(C(C2CC3(CCC3O)C2)=O)C1 49357,C=C(C)C(CC(=O)NC1CN(c2cc(O)nc(SC)n2)CC1C#N)OCC 49358,C12(CNC(CC(=C)C)=O)CC(CNC(=O)CCCCc3ccc(Cl)cc3)(CO1)C2 49359,c1(SC)cccc(C(=O)N(C(C)CNC(C2(Br)CC2)=O)C)n1 49360,C(CCCC(C)(C)C(=O)NNC(=O)C(C)CC=C)NC(C(CC=C)C)=O 49361,N1(C(COC(CC)C)=O)CC2CCC(NC(C3CCc4cncn4C3)=O)CC2C1 49362,CC1CC(C)CN(CCNC(=O)CCN2CCCCC2C)C1 49363,C(=O)(C(O)CC(F)F)NC(CC)CNC(=O)Cc1cc(-c2ccccc2Cl)on1 49364,c1(C(=O)NCc2cn(-c3cccc(SC)c3)nn2)cc2ccccc2s1 49365,C(=O)(C1=C(F)CN(C(=O)C=CCF)CC1)NC1CCN(OCC)CC1 49366,N1(C(c2c(OCC)scc2)=O)CCN(C(=O)CC2COCC2(C)C)C(C2CC2)C1 49367,C=CCCCC(=O)N1CCC(n2cc(CNC(C34CC(F)(C3)C4)=O)nn2)C1 49368,C1(NC(C(C)N(CCC)C(c2ccc(O)cn2)=O)=O)CCCC(C2CC2)C1 49369,c1(OC)cnc(F)c(C(=O)NCC(C2CCCCC2)NC(=O)C(F)(F)CF)c1 49370,Cc1ccc2c(C(N3CC(CC(C)NC(C4(S(N)(=O)=O)CC4)=O)C3)=O)coc2c1 49371,C1(C(N(C2(CC(=O)N(CC(COC)(F)F)C)CC2)C)=O)CCCC(C)C1 49372,c1(NC(C=CCC)=O)ccc(NCCN(C(=O)C(C)=C2CC2)C(C)C)nc1 49373,C1(CCO)(CC)CN(C(=O)C(CC2CCCC2)NC(=O)Cn2cc(C)cn2)C1 49374,c1(C(N2C(NCCNC(c3c(CC)ocn3)=O)C2)=O)ccc(F)c(OC)c1 49375,n1(CC(N2CC3C(NC(c4c(C)ncs4)=O)(C3)C2)=O)nc2n(c1=O)CCCCC2 49376,C(CC(C)C(=O)NC1CCC(CN(C)C(c2cc(Cl)cs2)=O)CC1)=CC 49377,C1(C(=O)NCC23OCC(NC(c4cnco4)=O)C(C2)C3)CCc2nncn2CC1 49378,C1(C(=O)NCCNC(C(C)=C2CC2)=O)CCCN(C(N2CCOCC2=O)=O)C1 49379,CCC(C)(COC)C(=O)NC1(C)CCCN(C(c2cccc(CCOC)c2)=O)C1 49380,c1(C(=O)NCC2CC2NC(C2(c3ncco3)CC2)=O)cccc(-n2cccn2)n1 49381,CC12CCC(C(=O)NCCC3CN(C(C4CCCCCC4)=O)C3)(CC1)CO2 49382,c1(C(C)C)ccc(F)cc1C(N1CC2C(C1)N2C(c1coc(Cl)n1)=O)=O 49383,c1(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)cc(F)ccc1Br 49384,C1(CC(=O)NCCCOCCC(=O)N2CC(c3ncc[nH]3)C2)CCCSC1 49385,N1(C(c2cc(C)cc(F)c2F)=O)CCn2nc(C(=O)OCC(C)(C)C)cc2C1 49386,C1(NC(CC)=O)CC2CCC1(C(N1CCN(c3cnc(O)nc3O)CC1)=O)C2 49387,C(=O)(CCN(OC)C(=O)C(C(C)O)N(C)C)OC1(C(=O)NCC)CCC1 49388,N1(C(CCN(CCC)C)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49389,c1(OCC(=O)N(CCCNC(=O)CC(C)n2ccc(C)n2)CC)ccc(C)cc1 49390,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49391,N1(C(=O)NCc2c(OCCOC)cccc2)CCCC(CN)CC1 49392,C(=O)(C(CNC(=O)Cn1ccnn1)N(C)C)N(C(C(C)SC)C)C 49393,N1(C(C(C)n2cccn2)=O)CCSC(C)C1C.C1CS1 49394,c1(-c2cc(CN3C(C(=O)OCC)CC3C)no2)cc(F)ccc1Br 49395,Cn1cccc1C=CC(=O)NC1(CC(=O)NC2CCOC2=O)CC1 49396,OC1C2COCC1CC(N=c1[nH]c(=NCc3nncn3CC3CC3)c3sccc3[nH]1)C2 49397,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49398,N1(C(C(c2ccc(F)cc2F)=O)=O)CC(NC(C2CC3C=CC2CC3)=O)CC(O)C1 49399,C1(CNC(=O)OC(C)(C)C)CC2(CC(NCC3CCCOC3C(C)(C)C)C2)C1 49400,C(CCCCCNC(=O)Cc1cccnc1Br)NC(C(CC)=CC)=O 49401,C(=O)(CCCN(C)N=O)N1CC(C(C)NC(CCC2CC(OC)C2)=O)OCC1 49402,c1(CC)cnccc1C(=O)NC1CC(C(=O)NCC(c2ccccc2)F)C1(C)C 49403,N1(C(C23CC(NC(c4c(C)con4)=O)(C2)C3)=O)CCC2(CC(F)C2)C1 49404,C=CC(CCC)CC(=O)NC(C(=O)NC1CCCCCCC1)C(C)(C)C 49405,N1(C(c2cn(CC(=O)OC)nc2)=O)CCCC(CNC(c2c[nH]nc2OC)=O)C1 49406,c1(OC)cc(C(=O)NC23CC2CN(C(C24CC(C2)C4)=O)C3)c(OC)cc1I 49407,c1(C(=O)NC2C(CNC(C3N(C=O)CCC3)=O)C2)cc(Cl)c(Cl)c(Cl)c1 49408,N1(C(c2cc(C)nc(O)n2)=O)CC23CCCC2(C1)CN(C(C1(C)CCCO1)=O)C3 49409,N1(C(C2(C(C)=O)CC2)=O)CC2(COC(CNC(c3ncoc3C)=O)C2)C1 49410,NCCCC(C(=O)NC1(CO)CCSC1)c1ccccc1 49411,C(=O)(CC(F)(F)C(C)(F)F)N1CC(N(C(=O)C(F)n2cccn2)C)C2(C1)CC2 49412,N12Cc3n[nH]cc3C1C(=O)N1CCCC1C2=O.c1(NC(N)=O)nocc1C(C)=O 49413,c1(N2CCN(C)CC2)nc2c(c(=NCCSc3ccccc3)[nH]1)CSC2 49414,C1CC(C)(C)NC(=O)N1.C(N)(=O)OC(C)(C)C.CC(C)C(=O)C 49415,C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(c2nn(C)cc2O)C)(CC)CCC1 49416,Cc1nc(C2CCC2)sc1CC(=O)N(CCCNC(C1(CCO)CC1)=O)CCO 49417,N1(C(CCC(CC)=O)=O)CC2(CCCC2NC(=O)C=CC2CCCO2)C1 49418,c1(C(N(CC(CC)NC(=O)C(C2CCCCC2)F)C)=O)cc(C(N)=O)co1 49419,CC(CCCNC(=O)C(O)Cc1ccccc1)NC(c1sccc1C1CC1)=O 49420,C1(NC(C2(C)CCNC2=O)=O)COCCN(C(=O)Cc2ccccc2)C1 49421,N1(C(C=CC)=O)CC(F)(n2cc(C(=O)NCC(C)C)nn2)C1 49422,n1(CC(N)=O)cc(C(=O)NCC(C)(C2CC2)NC(=O)CCC2CCC(=O)N2)nn1 49423,N1(C(c2nnn(C)n2)=O)CCC(O)(CNC(=O)CCCN2C(=O)CNC2=O)CC1 49424,C1(NC(=O)NC2(CF)CC(OC)(OC)C2)CCC2(CCOCC2)CC1 49425,c1(-c2cccc(C(=O)OC)c2)c(OC)nc(Cl)nc1NC(=O)CC(C)SC 49426,c1(OC)ccc(C2CCN(CCn3cccn3)C2)c2ccccc12 49427,C=Cc1ccc(CN2CCN(Cc3cccs3)CC2)cc1 49428,CC1OCCCC1C(N1CCC(CCC(=O)NCCCN2CCOCC2)CC1)=O 49429,C1(C2CC2)(C(=O)NC(C2CC2(C)C)C)CN(C(C2CCCSC2)=O)C1 49430,c1(C(N2CC(CC=C)(NC(C3CC=C(C)CC3)=O)C2)=O)ccnc(OCC)c1F 49431,n1(CC)ncc(C(=O)NC(C)SCC(N2CCC(CNC(C)=O)C2)=O)c1C1CC1 49432,C1(NC(C2C(C)(C)CC2)=O)(CNC(=O)C=CCOc2cccc(O)c2)CCOCC1 49433,c1(NCc2nc(CC)sc2)cc(=NCCCOC2CC2)[nH]c(CC(C)C)n1 49434,Cc1nn2ccc(C(=O)N(C(C)(C)C)C)nc2n1.C123COC(C1)(C2)COC3=O 49435,N1(C(CC2CCC(=O)N2)=O)CCN(CCOCCOC2CC(CCO)C2)CC1 49436,n1(CCC)nnnc1C(c1ccc(C(F)(F)F)s1)NCc1ccon1 49437,c1(C(=O)NC(C)CNC(=O)Cc2ccc(F)cc2)c(F)ccc(Cl)c1Cl 49438,CC1CN(C)C(C)CC1N.c1(-c2cncs2)ccc(Cl)cc1Cl.c1(=O)ccc1=O 49439,c1(OCC(=O)NC(C)C(CO)NC(c2ccc(C(F)F)cc2)=O)ccc(Cl)cn1 49440,c1(CC(N2C(CNC(=O)C=Cc3ccccc3)CCCC2)=O)cc(F)ccc1O 49441,Cc1cccc2c(C(=O)NCc3cccc(CNC(C4CC4(F)F)=O)c3)n[nH]c12 49442,N1(C(C2C(C)OCC2)=O)CCC2(CCCN(S(=O)(=O)C(C)C)C2)C1 49443,c1(C(N2CC(NC(=O)CNc3ccc(Br)cc3)C2)=O)ccc2nncn2c1 49444,N#Cc1cc(CNC(=O)Nc2ccc(C3(C(F)(F)F)CC3)cc2)ccn1 49445,C1(CNC(C2C(C)OC(=O)N2)=O)C(C2CC2)CCN1C(=O)Cc1ccn(C)n1 49446,C1(C(=O)NCc2cnc(CC)[nH]2)C2CC3C(C2NC(=O)C(C)SC)C13 49447,N1(C(Cn2c(C)ncc2)=O)CCC(CNC(c2csc(CO)n2)=O)C12CC2 49448,CC1(C)COC1C(N1CCC(n2ccnc2)C1)=O 49449,CN1CC=C(C(=O)N2CCC2CC(=O)N(CCN(C)C)C2CC2)C1 49450,C1(C(=O)OC(C)(C)C)COC2(C1)CC1(CN(C(C3(C)COC4COCC34)=O)C1)C2 49451,N1(C(C2C(NC(C(C)=C3CCC3)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49452,Cc1cccc(CC(C(=O)NC2CC(N(C(=O)CC3CC34CC4)C)C2)NC(N)=O)c1 49453,c1(NC(c2cn(CCOC)nc2C)=O)ccc2ncc(I)n2c1 49454,c1(C(C)(F)F)csc(C(=O)NC2(CO)CN(C(c3csc(Cl)c3)=O)C2)n1 49455,N(C(=NCC1CC1)NCc1ncc(C(C)C)o1)C(CCC)C 49456,c1(C(=O)NC2C(NC(CCOC)=O)CCC2)cc2c(cc1Br)OCO2 49457,c1(CNC(N2CCCC2)=O)ccc(OCC23COCC2C3)c(F)c1 49458,N1(C(c2cc(C3CC3)nc(O)c2)=O)CC2CC1CN2C(C1C=CCS1)=O 49459,CC1CC=C(C(=O)NCC23CCC(CC2)N(C(C2CC4CC2CC4(F)F)=O)C3)CC1 49460,C(=O)(C1=C(c2ccccc2)CCC1)NCC(CC)NC(c1cnnc(C)c1C)=O 49461,CC1CCC(CCNC(=O)C(Cc2ccoc2)NC(C2CCC(O)C2)=O)CC1 49462,C(C)(CCC(=O)N(CCCNC(=O)Cc1cnc(C)[nH]1)C)SC 49463,c1(C(=O)NCCCOCCNC(CCCCSC)=O)ccc(C(C)(C)C)cc1C 49464,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49465,CN1CC(F)CC1C(N1CCC(CC(=O)NC2CC(CCF)C2)C1)=O 49466,Cc1cnc(CNC(=O)C(C2CCCCC2)c2cncn2C)c(C)c1 49467,N1(C(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)CCc2nnnn2CC1 49468,CCC(CNC(=O)CSc1cnn(C)c1)N=c1[nH]c(C(C)CC)nc(C)c1C 49469,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1c[nH]c2ccncc12)=O 49470,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)O)C2)cc1C 49471,CC1CCC(CC(=O)NCC2(NC(=O)C=Cc3ccc[nH]3)CCC2)C1 49472,c1(C(CN(CC#N)C(=O)Nc2ccc(C(=O)NC)cc2)C)cc(F)cc(F)c1 49473,C1(C(N(CC)Cc2ncc[nH]2)=O)C2CC3C(C2NC(=O)C(C)(C)CSC)C13 49474,C1(C)(CC)CC(NC(c2[nH]nnc2-c2cccs2)=O)CN1C(=O)CC1CCC1 49475,c1(C(N(C(CNC(CCc2ncc(C)[nH]2)=O)C2CC2)C)=O)ncccc1C(F)F 49476,Cc1nnn(C)c1C(N1CCC(C)(CNC(=O)Cc2ccccn2)C1)=O 49477,c1(C(=O)NC2CCN(C(C(C#N)C3CC3)=O)C2C2CC2)cnn2cccc(Cl)c12 49478,C1(C(N2CC3(CN(C(c4n(C)nc(C(N)=O)c4)=O)C3)C2)=O)CCC2(CCOC2)O1 49479,C#CC1CN(C(=O)C(C)OCC2CC2)CCN1C(C1(C2CC2)CC(=O)C1)=O 49480,N1(c2c(C#N)nccn2)CCCC(C2(NC(C3CC3Cl)=O)CC2)C1 49481,CC1(C(=O)N(CC(O)CO)CC2CC2)CCN(C(=O)C(=O)NC2CC2)CC1 49482,CC(O)C(C(=O)NC(c1cn(C)cn1)C)NC(=O)C(C1CC2C=CC1C2)=O 49483,CC(C)(C)C(CNC(C1CC1Cl)=O)C(=O)NCC1(c2ccon2)CC1 49484,C1(NC(c2cc(C)[nH]c2)=O)CC2C1CCN2C(c1cnn(C(C)C(C)C)c1C)=O 49485,c1(C(N2C(C)(CNC(CC(CC)OC)=O)CCC2)=O)ccc2c(c1)CNC2=O 49486,Cc1cc(C)c(C(N2CC(NC(=O)C(C)OCCN(C)C)C2)=O)c(O)c1 49487,N1(C(C=C(C)F)=O)CCN(C(c2nccc(CO)c2Cl)=O)C(c2ccccc2)C1 49488,C1(COC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(C(C)C)cn2)=O)C1 49489,CC1CC(CNC(c2cc(CCCO)on2)=O)CN1C(=O)C(F)C1CCOC1 49490,N1(C(Cc2c(C)nn(C)c2C)=O)CC(C)OC2(CCN(C(=O)C3CC3)CC2)C1 49491,Cc1ccc(C2CCCN2C(=O)Nc2cnn(C(C3CCN(C)C3=O)C)c2)cn1 49492,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3F)=O)CC2C1 49493,C1(CNC(=O)C(F)C(F)(F)F)CC2CCC(C1)N2C(c1ccc2c[nH]nc2n1)=O 49494,S(=O)(=O)(c1ccc(S(=O)(=O)NCCCNCC2CC23CCC3)cc1)NCC 49495,C1(CNC(C2(CO)CCCC2)=O)CCCCN1C(C1CCCCO1)=O 49496,N1(C(C2C(C(C)C)CCO2)=O)CCCC(C(=O)Nc2cnn(C(F)F)c2)CC1 49497,C1(n2cc(-c3c(C)nccn3)nn2)CC2CCC1(NC(=O)CCn1cc(Cl)cn1)C2 49498,N1(C(c2c(OC)ccc(Cl)c2)=O)CCC=C(C(=O)NCCc2ccncc2)C1 49499,N1(C(Cn2cc(C(=O)OCC)nn2)=O)CCN(CCNC(=O)CSC(=N)N)CC1 49500,C12CN(C3(CCC3)C1)C(=O)c1[nH]nc(c1Cl)C(=O)N2.C1(CC)C(F)(F)C12CCC2 49501,C#CCC(C(=O)NC)NC(c1cc(CNC(c2nccnc2C)=O)ccn1)=O 49502,C1(O)(C(N(CCN(C(CCN(CC)CC)=O)C)C)=O)CCOC1 49503,C1(C2CC2)(NC(c2c(C)con2)=O)CCN(C(=O)CC2OCCOC2(C)C)C1 49504,c1(OC)cccc(N2CCC(C(=O)NC3CC(CNC(=O)C(C)SC)C3)C2=O)c1 49505,CC1(C)CC(F)(F)CCC1C(N1CCOC(CNC(=O)CCCCC2CC2)C1)=O 49506,n1(CC)cc(C(=O)NCCCC2CN(C(=O)C(C)c3cc[nH]n3)CCO2)c(C)n1 49507,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49508,C1(C(=O)NC(CN(C2CCSC2)C)=O)CCC(CN2CC(O)CC2C(N)=O)CC1 49509,Cc1cc(C(N2CCCC(CNC(=O)CC3OCCCC3(C)C)C2)=O)ccc1N 49510,C1(CNC(c2c(C)cn(C)n2)=O)C2CCC(C2)N1C(C1(CC(C)C)CC(=O)C1)=O 49511,C1(NC(C2(COC)CN(C(=O)CC(C)C)C2)=O)CCCCCC1(C)C 49512,c1(C(N(CC(C)NC(C2CCC3(CCC3)O2)=O)C)=O)csc(S(C)(=O)=O)c1 49513,CC1(C(=O)NCC2CCN2C(c2cncc(C#N)c2)=O)CCc2ccccc21 49514,C1(C(N2CC(F)(CNC(C(C)(C3CC3)OC)=O)C2)=O)CCC(C)(C)OC1 49515,c1(C(N2CCC(NC(C=CSC)=O)C2)=O)c(C)nn(C)c1Cl 49516,N1(C(c2cnc(C(=O)OC)o2)C(=O)NCCC)CCOC(C)(C2CC2)C1 49517,C1(n2cc(CNC(C)=O)nn2)CCN(C(c2occc2Br)=O)CC1 49518,c1(C(=O)OC)nc(=NC2CCCN(C(=O)Nc3nc(C)c(C)[nH]3)C2)c(F)c(Cl)[nH]1 49519,C1(CNC(CC2CCC(C)CC2)=O)C(C)CCCN1C(C1CC1(F)F)=O 49520,c1(C(N(CC(CC)NC(CC2(OCC)CC2)=O)C)=O)cnn(CC)c1 49521,N1(C(c2c(C)scc2)C(=O)Nc2nnn(C)n2)C2CCCC1COC2 49522,C=CC1(CC)COCCN1C(c1ncc(Br)cc1Cl)C(=O)NCCC#N 49523,Cc1ccc(CC(N2CC3(NC(=O)COc4cccnc4)CCC2C3)=O)cc1F 49524,Cc1cc(-c2cn(C3CCC(=O)C3C)nn2)cc(F)c1 49525,N1(C(CN(CC(C)(C)C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49526,c1(C(=O)NCC(C)(CCn2cncn2)NC(=O)CNC=O)coc2c1COC2 49527,N1(C(c2cnn(C)c2CO)=O)CC2(COC(CNC(=O)C(=O)NCC(F)F)C2)C1 49528,N1(C(c2c(OC)cccc2Cl)C(=O)NCC(F)F)CCC(C)(C)CC(C)(C)C1 49529,N1(Cc2cccc(C)c2I)CCC2CN(c3ncc4[nH]ncc4n3)CC2C1 49530,C1(NC(C2(CSC)CCC2)=O)CCN(C(=O)CCCc2ccccc2)CC1O 49531,N1(C(C2C(=C)C2)=O)CCN(C(c2ncc(I)cn2)=O)C2(CCC2)C1 49532,c1(CC)cccc(F)c1C(=O)NC1CCN(C(=O)CC#N)CCO1 49533,c1(C(=O)NC2C(NC(c3cc(C)nn3C)=O)CC2)c(C)nc(O)nc1C 49534,C1(CC)(NC(=O)CCC2CCCOC2)CCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C1 49535,c1(C(CCOC)N(C)C)cc(C2CC2)ccc1SC.c1(=O)c(=O)[nH]1 49536,c1(OC)cc(C=CC(=O)NCC23CC(CN2C(c2cnoc2C)=O)C3)ccc1F 49537,c1(C(=O)NC(C)CCN(C)C(c2ccco2)=O)nccc(Cl)c1Cl 49538,c1(NC(C2CSCCN2Cc2cc(F)c(O)c(Br)c2)=O)ncc(Br)cc1[N+](=O)[O-] 49539,C(=O)(CCCn1cccn1)NC(C(=O)NC1(CN(C)C)CCC1)C1CCCO1 49540,C1(C(N2CC(C)N(C(c3ccn(C4CC4)n3)=O)CC2)=O)CN2CCCCC2CO1 49541,c1(C(=O)NC2(C)CCC(NC(C3CCC34CCC4)=O)CC2)scc2c1OCCO2 49542,c1(C2(NC(C3CC(CCN(C(CC(C)C)=O)C4CC4)C3)=O)CC2)cc(Cl)ccc1F 49543,c1(C(=O)NCC2C(NC(C(C3CC3)COCC)=O)CCCC2)cnc(O)c(C)c1 49544,C1(C(N(CC(CC)(C)OC)C)=O)C2CCC(C2)N1C(C1C=CCC1)=O 49545,c1(CCC)ccc(C(=O)NCCC(C)N(C(=O)C(N2CCNC2=O)C)C)[nH]1 49546,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1(CS(C)(=O)=O)COC1)=O)C2 49547,Cc1cc(Cl)c(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)cc1N 49548,N1(C(c2ccc(CC)o2)=O)CCC(NC(=O)Cc2sc(C)nc2C)CC1C1CC1 49549,N1(C(CCC=CC)=O)CCN(CCN(C)C(C2(C)CC=CCC2)=O)CC1 49550,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1[nH]cnc1C#N)=O)C2 49551,c1(C(=O)NCC(CCNC(c2c(C)nn(CC)c2Cl)=O)O)cccc2c1CCN2 49552,c1(C(C)NC(=O)CN(C(=O)CCC2CC2(F)F)C)nncn1C 49553,C(CC(C)(C)CNC(=O)CC1CC(NC(=O)CSC(F)F)C1)OC 49554,C1(C(=O)NCC(C(C)C)NC(=O)CCn2cccn2)CCC2(CC2)C1 49555,c1(C(=O)NCC2(C)CCCN(C(C(C)OCCC#C)=O)C2)nc(O)nc(O)c1N 49556,c1(CC(C(=O)NC2(CNC(c3c(C(C)C)[nH]cn3)=O)CCC2)C)ccc(O)cc1 49557,c1(C(=O)NC2(CCOC)CCN(C(C3(O)CC3(C)C)=O)C2)ccc(=O)n(C)n1 49558,N1(C(C2(CCOC(C)C)CCC2)=O)CCCC1CNC(c1ccccc1)=O 49559,C(CC(F)F)(C(=O)NC(=O)CN1CC=CC1)NC(CN1CC(=O)C1)=O 49560,C(C(=O)N(CCCCCCNC(=O)C=C1CCC(C)C1)C)(C(C)C)OCC 49561,C1(C)(C(=O)NCCN(CCC)C(c2ccc(Cl)o2)=O)SCCCS1 49562,C1(C(=O)NCCCOCCN(C(C2(C)CC(C)C2)=O)C)CCCC(C(=O)N(C)C)C1 49563,Cc1nn(C)c(Cl)c1C(=O)NCC1CCCC1C(=O)NC1(C)CC(F)(F)C1 49564,c1(N2CC(C)NC(=O)C2)nc(N2C3COCC2C3)nc2c1COC2 49565,c1(N2CC(NC(c3c(C)cc(OC)cc3C)=O)C(C)C2)ncnc2cc(C)[nH]c12 49566,C1(CC)CN(C(c2scnc2C)=O)CCN1C(c1nocc1Br)=O 49567,C#Cc1cnc(C(=O)NC(CC2CCOCC2)C(=O)N(CCC=C)C)c(C)c1 49568,C1(CCOC)CN(C(c2cnc(Br)s2)=O)CCN1C(=O)CCCSC 49569,C(=O)(CC(CC1CC1)NC(C1(CC)CCOC1)=O)NCC(CC)O 49570,N1(C(C2CCC(C)C2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)CC2CO 49571,c1(C(N2CCC(N(c3cc(CC)ncn3)C)C2)=O)cc(C#N)cn1C 49572,C1(OC)CN(C(=O)Cc2c(Cl)cccc2Br)CCC1NC(C12CCCC1C2)=O 49573,C12CCC(C1)n1cc(nn1)CCCN(C1CC1)C2=O.C(=O)(COC)OCC 49574,N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)CCC3CCC(C)O3)CC12 49575,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49576,N1(C(CC2C(C)(C)C(O)C2)=O)CC2(CC(C(=O)N(C3CCOC3)CCO)CO2)C1 49577,N1(CC2N(CC)CCC2)CCCC(C(=O)N(C)CCc2nncn2C)CC1 49578,C(C(C(=O)N(C(C)C(C)O)C1CC1)NC(c1ccc(CC)s1)=O)OCC 49579,c1(C(N(C2CN(C(CSCC(C)C)=O)CC2O)C)=O)cccc2c1OC(F)(F)O2 49580,c1(C(N2CCC(F)(CO)C2)=O)cnc2ncc(-c3cc4ccccc4s3)cn12 49581,CC1CC2(CC(C(=O)NCCC3CCC(NC(=O)CCN4CCCCC4)C3)C2)C1 49582,N1(C(=O)NC2(c3ccc(C(F)(F)F)cc3)CC2)CCOCC(C(=O)O)C1 49583,c1(C(=O)NC2CCN(C(C3CC3CN(C)C)=O)C2)ccc(F)c(F)c1F 49584,CC(C)C(O)C(C)(C)C(=O)N(CC(C1CC2CCC1C2)O)C 49585,Cc1ccc(F)c(C(=O)N(CC(C)N(C)Cc2nnnn2C2CC2)C)c1Br 49586,c1(OC)ccc(CC(=O)N(C(c2cn(-c3ccccc3)nn2)(C)C)C2CC2)c(C)c1 49587,C(N=c1ccnc(CNCCNC(=O)C(C)(C)C)[nH]1)c1c(N(C)C)cccc1 49588,C1(CNC(c2c(C)scc2)=O)CCCCN1C(=O)CC1C=NN(C)C1=O 49589,C(=O)(CCCCCC(C)(C)C)N1CCC(C)(CNC(c2ccc(C)cc2C)=O)C1 49590,c1(CC(=O)NC2CC3CC(C2)N(c2ncncc2C#N)C3)nc(F)c(F)cc1F 49591,N1(C(CCCCCC#N)=O)CCCC(C2(NC(=O)C=C3CCC3)CC2)C1 49592,CN1CCN(C(c2ccc(F)cn2)=O)CC1C(=O)NCCC1CCC(C)(C)O1 49593,c1(C(N(C(CC)C(=O)NCCOC(=N)O)C)=O)cccc2cc[nH]c12 49594,C(=O)(C1=CCCCCC1)NC1(CO)CCN(C(C(CC)N(CC)CC)=O)CC1 49595,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCCC1 49596,C(=O)(C(F)(F)C(O)c1ccccc1)NC1C(NC(=O)CNc2nccs2)COCC1 49597,c1(OCC)cccc(NC(=O)C(C2CCCC2)NC(c2csnc2OC)=O)c1C 49598,N1(C(C2(C)CC2)=O)CC2CCCC2(C(N2CCCCC(CO)C2)=O)C1 49599,c1(C(=O)NC2C(C)CN(C(=O)COCCN(C)C)C2)cc2ccccn2c1 49600,c1(NCCNCC(CNC(CCSC(C)(C)O)=O)CO)cccnc1-n1cccn1 49601,C1(NC(CCOCCC)=O)CC(C2CCN(C(c3cc(O)nc(C)n3)=O)C2)C1 49602,c1(NC2CC(CSC)C2)[nH]c(=NCc2cc(C(F)(F)F)n[nH]2)nc2c1cnn2C 49603,C(C(F)(F)C(F)(F)F)N(C(COCCCC#C)=O)CC1CC1.C1C(=O)N1 49604,c1(C(=O)NCCCCCCNC(=O)CC2CC(=O)NC2=O)cnc2[nH]cncc1-2 49605,c1(NC2C(C)CCCN2Cc2cc3cnccc3o2)cnc(C#N)c(C#N)n1 49606,CCCC(CC)C(=O)NC1CCCC1NC(c1cc(F)ccc1OC(C)C)=O 49607,C1(CNC(CC(C=C)C)=O)CCN(C(c2cc(C)ccn2)=O)CC1(F)F 49608,c1(OC)ccc(C(=O)NC(C)(CNC(=O)CC(C)(C)O)C(C)C)cc1C 49609,N1(CC)CCCC1C(=O)NC1CN(C(C)C)C1=O.C1(COC)CCCCC1 49610,C1(OC)(OC)C(C(=O)NCCNC(C2(C)CCC2)=O)CC1(F)F 49611,c1(CCC)ccccc1NC(=O)CC1CCCC1.c12ccc(cn1)[nH]c2=O 49612,Cc1cncc(C(=O)N(C2CCCN(CC=Cc3ccccc3)C2)C)c1Cl 49613,S(=O)(=O)(c1ccccc1C(F)(F)F)NC(COCC)CN 49614,c1(SC)ccc(N)cc1C(N1CCC(N(C(=O)Cn2cnnc2)C)C1)=O 49615,Cc1nc2sccn2c1C(=O)NCCC1CC(F)(F)CN1C(=O)C(O)C(C)(C)C 49616,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1ccnn1)C2 49617,C1(C(=O)NCC2CC(NC(=O)Nc3cccnc3)C2)CC(=O)N(CC(F)(F)F)C1 49618,C(CC(C)C)(C(=O)C(=O)OC(C)(C)C)N1CC(OCCN)C1.N1(C)CCCN(C)C1=O 49619,CCCC(CCC)CC(=O)NC1CCCOC12CCN(c1ncc(C)cn1)CC2 49620,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ccc(F)c2[nH]1 49621,c1(CCC(C)C)nc(-c2ccc(CCSC)cc2)n(C2CCCSC2)n1 49622,C1(NC(C(CCC)O)=O)CC1C1CCCN(Cc2c(OC)ncnc2O)C1 49623,c1(N(N(C(C=COCC)=O)CCCC)C)nc(=NCC2COCOC2)[nH]c2c1SCC2 49624,CC1(C)CCN(C(C2C3CCC(F)C23)=O)C1C(=O)Nc1ccc(F)nc1 49625,CCCCC(O)C(=O)NC(CNC(C1CCCSC1)=O)C(C)C 49626,Cc1cc(C(=O)N(C)CCN(C)C(c2cc(Cl)c[nH]2)=O)c2ncccc2c1 49627,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49628,c1(OCC)cc(Cl)ccc1CNC1CC2(C1)CC(C(=O)NC1CCOCC1)C2 49629,CC1(C(N2CCC(CNC(C3(N4CCCC4)CCCC3)=O)CC2)=O)CCCCC1 49630,c1(OC(C2CC2c2ccc(F)cc2)=O)c(F)ccc(C2CC2)c1F 49631,c1(C(c2n(CC=C)nnn2)Nc2cc(C#N)ccc2C)cc(Cl)cc(Br)c1F 49632,C(=O)(CS(=O)C(F)(F)F)NC(CC)CNC(=O)Cc1ccno1 49633,CCC(C)(C)CNC(=O)C(C1CCCC1)NC(=O)C=CC(C)(C)SC 49634,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49635,C(=O)(C(O)CC(C)C)N1C(C)(CC(N2CCCC(=C)C2)=O)CC1 49636,C1(NC(c2c(C)nc(C3CC3)nc2)=O)CCCC12CN(C(c1cccnc1)=O)C2 49637,c1(OC)ccc2c(C(=O)NCC(C)CNC(C(C)C(F)(F)F)=O)c[nH]c2c1 49638,C(CC(=O)NOCC)N(C(COC(=O)Oc1cnn(CC2(C)CC2)c1)=O)C 49639,N1(C(C(c2ccc(C)o2)C)=O)CC2(CCCC2)C1C(=O)N(CC1=CCCOC1)C 49640,C1(CNC(=O)CCC2CCC(O)CC2)CC(O)CN1C(=O)C=Cc1ncc[nH]1 49641,N1(C(c2n[nH]c(CC)c2Br)=O)CCC2(CCC2CNC(=O)C(C)O)CC1 49642,c1(CCC)sc(C(=O)NCC2(CN(C(=O)C(C)(C)O)C)CC2)cc1CC 49643,c1(CN2C(CCC(=O)NCCSC)CCC2)ccc(C2=COCC2)cc1 49644,c1(C(N(CC(C)NC(=O)C(F)n2ccnc2)C)=O)cccc(N2CCOC2=O)c1 49645,c1(C(N2CCN(C(CSCC(=O)OC)=O)C3C2C3)=O)ccc2ncn(C)c2n1 49646,N(C(=NCC1CCCSCC1)NC1CCC1)C(C1CCC1)C 49647,CON(CCC(=O)N1CCCC(CC2CC2)C1)C(=O)C=C1CCCCC1 49648,C(=O)(CCS(C)=O)NCCC(=O)N(c1ccoc1)CC 49649,CCCC(CCCNC(=O)CCCOC)NC(C1(C)CCN(C)C1=O)=O 49650,N1(C(CC2CC(SC)C2)=O)CC(NC(C2(C)CCCOC2)=O)CC(C)C1 49651,N1(C(C(CCC)CC)=O)CC2(CCCN(C(C3COCC(C)(C)O3)=O)C2)C1 49652,Cc1cccc(Br)c1C(C(N1CCC(CO)CC1)=O)NC(c1cnn(C)c(=O)c1)=O 49653,c1(C(=O)NC2CCCN(Cc3ncc(C)nc3)CC2)cccc2nccnc12 49654,C(=O)(C(C)C(C)S(C)(=O)=O)NCCC(C)NC(=O)C=Cc1ccn(C)c1 49655,CC(C)C(C(=O)N1CCC(C(F)(F)F)CC1CNC(=O)CNC1CCC1)C(C)C 49656,c1(CC)ccc(C(=O)NCC2CC(F)CN2C(=O)CSCc2ccccc2)cn1 49657,c1(C(=O)NC2(CC=C)CN(C(=O)CCS(C)(=O)=O)C2)c[nH]c2cc(OC)ccc12 49658,C1(NC(C(CC)n2cncn2)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 49659,CC1(C(=O)NCC2CC3CCC2N3C(C2(CO)CCC2)=O)CCCNS1(=O)=O 49660,C1(NC(=O)C=CC=C(Cl)Cl)CC2CC1N(C(C1CC1c1cncc(F)c1)=O)C2 49661,N1(C(c2cnc(C3(N)CCC3)s2)=O)CCC2CC2C1 49662,C1(C)(CNC(C(CC)=CC)=O)COCCN(C(c2cc(Br)c(C)cc2C)=O)C1 49663,C1(NC(c2c(CCCC)ocn2)=O)CC(NC(=O)CCC2OCCO2)C12CCC2 49664,Cc1cccnc1CC(=O)NC1CC(C)N(C(=O)CN2CCOCC2)C1 49665,N1(C(=O)NCCOCCOCC(N)=O)CCOC2CC12 49666,C1(CC)C(NC(=O)COc2cccc(F)c2)CCN1C(=O)C(C)NC(C)=O 49667,c1(CC)ncc(C(N2CCN(C(=O)CCn3cccn3)C(CC)C2)=O)c(O)n1 49668,C(=O)(C1=NNC(=O)CC1)N1CCCC(C)(NC(C2CCC3CC3CC2)=O)C1 49669,c1(OC)nn(C)cc1C(N1CC(CNC(C2(C#N)CCC2)=O)C(C(F)(F)F)C1)=O 49670,c1(C(N(CC(C)NC(C2CCCN2Cc2nnn(C)n2)=O)C)=O)ccc(Cl)cc1 49671,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 49672,N1(C(C2(C=C)CN(C(=O)CP(C)(C)=O)C2)=O)CCN(CCCC)C(=O)C1 49673,c1(-c2cnc(COCC)nc2)cc(C2CC2)nc2ccccc12 49674,N1(C(C(CC)=CC)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)CCC12 49675,CCC(CCCC(=O)N(CCC1CC1)CC)NC(c1cc(C)c(F)cn1)=O 49676,N1(CCC2N(C)CCCC2)CC(=O)N(CC(N2CCCCCC2)=O)C1=O 49677,CCCC(C)(CC)C(=O)NC1(CNC(c2nn(C)cc2C)=O)CC1 49678,Fc1cccc(CN=C(NCC2CCOCC2)NCC2CC=CCC2)c1F 49679,c1(C(N2CCC3CCN(C(CC(C)O)=O)C3C2)=O)c[nH]c2ccccc2c1=O 49680,Cc1ccc(CCC(=O)N(C(C)CCNC(=O)CC2CCCC(C)C2)C)cc1 49681,c1(CCC)nc(=NCC(c2ccccc2F)C(=O)NC2(C3CCC3)CC2)s[nH]1 49682,C1(C(N2CC(C)(NC(=O)Cc3cnn(C4CC4)c3)C2)=O)CC2(CCCC2)CO1 49683,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 49684,c1(OCC(N2CCC(N(C(=O)CO)C)CC2)=O)cc(F)ncc1Br 49685,N1(CC(=O)NC(C(=O)N(CC(F)F)C)C2(O)CCC2)CCSCC1 49686,C1(CN2CC(C(F)F)NCC2)CCOC12CCC2 49687,C(C1CN(C(=O)CC2CC(F)(F)C2)CC1C(=O)NCC1CC12CCC2)=CC 49688,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)C1 49689,C(CCN(C)C(c1ccc(CC)s1)=O)(C(C)C)NC(c1cc(CCC)[nH]n1)=O 49690,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCn2cc(C)cn2)C(C)(C)C1 49691,c1(CN(C(=O)CC(C)F)CC)ccc(CNC(=O)Cn2ncnn2)cc1 49692,C1(C(c2ncc(CC)[nH]2)NCc2nnnn2Cc2ccccc2)C2CCCCCC12 49693,C12(CC)CC(CNC(CC3(C)CCCN3C(c3ccn(C)c3C)=O)=O)(C1)OC2C 49694,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 49695,c1(-c2ccc(CNc3c(CC)nccc3)cc2)cc(OCC)cc(O)c1 49696,c1(N2CC(CSC)OCC2)cc(Br)ccc1S(=O)(=O)NCC1(CC#N)CC1 49697,C1(N(CC#CCC)CCOC)CCN(C(C2C(C)CC2C)=O)C1 49698,C(CCCC(=O)N1CC2CC2(CNC(c2cccnc2OC(C)C)=O)C1)OC 49699,c1(C(=O)NCC(C2CC2)NC(c2c(C)cn(C)c2)=O)cnc2ccnn2c1C 49700,N1(C(c2c(CC)csc2)=O)CCC12CN(C(=O)C(C)Cn1cccn1)C2 49701,C1(C(N(C(C(=O)NCCN(C)CC)C)C2CC2)=O)C(C(C)=O)C1(C)C 49702,C(CCCCC(=O)NC1CCC1O)N(C(=O)Cc1cncnc1)C 49703,N1(C(c2coc(OCF)n2)=O)CCCCCC1CNC(c1ccccc1F)=O 49704,CC1=C(C(=O)NC2COC3(C2)CN(C(c2scnc2C)=O)C3)CCS1(=O)=O 49705,c1(C(=O)NC(CC=C)CNC(C2(C)CCOCC2)=O)cc(C)cc2c1NCCC2 49706,CC1CC(CC(=O)NC2CCCN(C(=O)C(CN(C)C)N(C)C)CC2)CC(C)(C)C1 49707,C(=O)(CC(C1CC1)NC(=O)CCNC(=O)CC1CCC(C)O1)OCC 49708,CC(C(=O)N=c1ccn(C2CCCN2C(c2ccc3occc3c2)=O)[nH]1)C1CC1 49709,c1(NC(=O)C(n2cc(Cl)cn2)C)nccc(CO)n1.CC1CCN1 49710,CCCCCCN(C(=O)CCN(C(=O)CC1CSCCO1)C)CCOC 49711,C(C(CC(=O)N(C)CC)C1CC1)NC(COCCCOC)=O 49712,N1(CC2(C(N3CCC(NC(=O)CCC4CC4(F)F)C3)=O)CCC2)CCCC1CO 49713,C#Cc1ccc(CC(N2CCC(NC(=O)C(C)N3CCCC3)CC2C)=O)c(F)c1 49714,C#Cc1ccc(C(=O)NCC(CCNC(C23CCC(OC)C2C3)=O)OC)cn1 49715,CCCCC(C)CCC(=O)N1CCC(NC(=O)Cc2cn(C)nn2)CC1C 49716,c1(C(=O)NCC(C)NC(c2cnc(C3CCOCC3)o2)=O)cccc(C(N)=O)c1 49717,n1(CC)nnc(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)N3)=O)C2)c1C 49718,C1(C(=O)NCc2n(C)ccn2)CC2CCC1N2C(=O)C(C)(O)C1CCC1 49719,n1(CCC(=O)N(C2CCCC(NC(C=CC)=O)C2)C)ncc2ccccc12 49720,CON1CCC(CC(=O)NC2(C(=O)NC3CCOCC3C)CCCCCC2)CC1 49721,C1(C(=O)NCC2(C)CCN(C(CCCOC)=O)C2)CCC2(CCC2)O1 49722,Cn1cnc2[nH]c(C(N3CC4(CCC4NC(=O)CCc4ccncc4)C3)=O)cc12 49723,c1(C2(C(N3CC(CCNC(C4(CC)CC4)=O)C3)=O)CC2)cccc(F)c1 49724,c1(SC(C)C(=O)N(C)CCOCCN(C(=O)CC2CCC(=O)N2)C)ccccc1 49725,CC1CCC(C(=O)NCCCCCCF)CN1C(C1CCC(O)CC1)=O 49726,C1(N(C(C(=O)NCC(F)F)C2CCCO2)C)CC=CCC1 49727,c1(-c2nc(C(C3CC3)OC)nn2C(C)C(C)C)ccc2c(c1)COCC2 49728,Cc1ccc(C(N2CC(F)(F)CC2C(=O)NCCC(C)C)=O)c(O)c1 49729,C1(C(c2n(CCC)nnn2)NC(c2ccncc2)C)CC2CCC1O2 49730,N1(CC)CCC1C(=O)C1CC1.C(CNC(C1(COC)CC1)=O)N 49731,N1(C(c2nc(C(C)OC)sc2)=O)CC(NC(=O)C2=CCCO2)C(C)(C)C1 49732,CC1(C)CC(NC(c2ccc(Cl)cc2N)=O)CN1C(C1CS(=O)C1)=O 49733,Brc1cc(CN2CCCC2c2cccc(Br)n2)c(C2CCCN2)s1 49734,c1(OC(C)=O)ccc(C(N2CCNCC2C(=O)Nc2c(C)cccc2F)=O)cc1Cl 49735,N1(C(C2CC(=O)NC2)=O)CCCC(C2CCN(C(=O)CCc3ccc[nH]3)C2)C1 49736,C1(NC(C(CCC)NC(N)=O)=O)CN(C(c2cccc(N)c2N)=O)CCC1CO 49737,C1(CNC(C2(C)CC2)=O)CCN(C(=O)CCc2ccncn2)CC1 49738,c1(C(=O)NC(COC)C)cn2c(n1)CCCC2C.c12cccc(c1C)C(=O)N2.C(C)(=O)O 49739,N#Cc1cc(C(N2CCOCC2C(=O)NC2CC3C=CC2C3)=O)c[nH]1 49740,N1(C(C2(COC)CC=CCC2)=O)CCCCCC1CNC(=O)CC1CC=CC1 49741,CCCC(O)CC(=O)N(CCCN(C)C(c1occc1-c1ccc(F)cc1)=O)C 49742,N1(C(C2(CC)CCCCO2)=O)CCN(C(=O)CCc2cncn2C)CC(CO)C1 49743,N1(C(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC(O)C1 49744,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2c(Cl)cnn2C(C)C)=O)CCN1C 49745,N1(Cc2cccc(OCC3C(F)(F)OC3)n2)CC2CC3CCCN3C2C1 49746,C12(NC(=O)Cc3cc[nH]n3)CCCC1CN(C(c1c(F)cncc1Cl)=O)C2 49747,Cc1cn2ccnc(C(=O)NC(C3CCN(C(=O)Cc4cc[nH]n4)CC3)C)c2n1 49748,c1(COC)ccc(-n2ccnc2)cc1.C12CCC1CNC2=O.C12CC1C(=O)O2 49749,C1(CNC(=O)Cc2ccn(C(F)F)n2)CC(O)CN1C(=O)Cn1ccnn1 49750,C1(C(=O)NCCC2C(C)(C)CC2)CCC(F)(F)C1O 49751,C1(CNC(CC(C)SC)=O)CCCCCN1C(c1cc(F)cs1)=O 49752,c1(N2CCC(CNC(C34CCC(C(=O)O)(C3)C4)=O)CC2)c(Br)cccc1[N+](=O)[O-] 49753,c1(OCC)ccc(CCC(=O)NC(CNC(c2cc(C)no2)=O)C(C)(C)C)cc1 49754,Cc1nsc(C(=O)N(CCCN(C(=O)C(C)Cn2ccnc2)C)C)c1Br 49755,CC(C)(C#N)CCC(=O)NC(CC(N1CCS(=O)CC1C)=O)C1CC1 49756,c1(CC)cnccc1C(=O)NCC1CCN(C(C2C=CCC2)=O)C1 49757,CC(C(=O)NC(C1CCCN1C(=O)C(F)C1(O)CCC1)(C)C)C(F)(F)C(F)F 49758,C(C(C)(C)NC(c1c[nH]nc1F)=O)(C1CCC1)NC(C(C)NC(C)=O)=O 49759,C1(NC(c2cccc(COC)c2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CCC1(F)F 49760,c1(CC(=O)NC(C(C)C)CNC(c2ncsc2C2CC2)=O)ccc(Br)cn1 49761,C(C(O)C(=O)NC1(CNC(C2(OC(C)C)CCC2)=O)CCOC1)OC 49762,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]cc2C(F)(F)F)=O)C)cc1Cl 49763,C12(C(=O)NCC3CCN(C(C(C(C)C)F)=O)C3)C3CC(CC13)C2(F)F 49764,c1(C(=O)NCC2C(CNC(c3cc(SC)oc3)=O)C2)cnc2n1CC(C)CC2 49765,CC1(C)OCC(C(F)(F)C(=O)NCCn2cc(CCCCCO)nn2)O1 49766,C(C(C(=O)N(C)CCF)C(C)(C)C)NC(C(C)SCCN(C)CC)=O 49767,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(C(c2ccccc2)C)=O)C)C(O)C1 49768,C1(CNC(C2CCN(C)C2)=O)CC2COCC2N1C(=O)Cn1cc(F)ccc1=O 49769,N1(CC)CCN(C(c2cnn(C(C)(C)C)n2)C(=O)NCCSC)CC1 49770,CCCC(C)(CCC)C(=O)NCCN(C(=O)C(=Cc1ccncc1)C)C 49771,N1(C(CSS(C)(=O)=O)=O)CC2CCC1(CNC(=O)C(O)CF)CC2 49772,c1(CCC(=O)NCCOCCOCCOCC#C)ccccc1Cl 49773,C1(COC)CC(F)CN1C(=O)CNC(=O)CCn1ccnc1.C1(=O)CN1 49774,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(c1cc(C2CCC2)[nH]n1)=O 49775,CCC(C(=O)OC)NC(C1CC1CNC(C1COCC1O)=O)=O 49776,C1(C(N(CCCNC(C2(C)CCN(C)C2=O)=O)CC)=O)COCCN1C=O 49777,C(C(CC(C)C)C(=O)NCCC(=O)N1CC(Cn2ccnn2)C1)NC(=O)OC 49778,S(=O)(=O)(c1ccnc(C(=O)O)c1)NC(c1cncc(N2CCN(C)CC2)n1)C 49779,C1(CNC(CSCCCC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 49780,CC(CC(=O)NCc1cc(C(=O)NCCOC2(C)CCC2)co1)CC(C)(C)C 49781,CC(C)CCC(C(=O)NC1CC1)NCCN(CC(F)F)C 49782,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 49783,CCCC(CC)CCC(=O)NCC1CN(C(c2ccc(N)c(F)n2)=O)CC1O 49784,C(=O)(C(C)(C)Cc1ccccc1)OCc1nnc(C)s1 49785,c1(C2(NC(N(CC(C)(C)OC)C)=O)CCCC2)ccc(Br)cc1 49786,C(=O)(C(C)CC(F)F)Nc1cc(NC(N2C(CCC#C)CCC2)=O)ccn1 49787,C(c1cnc(OC)nc1)=C(CC)C(=O)NC1CC(C)OC(C)C1 49788,C#CCCC(C(=O)NCC(F)(F)Cl)NC(c1cnc(O)cc1C)=O 49789,c1(OC)cccnc1C(=O)NC1CCN(C(C2CCOC2c2ccco2)=O)CC1 49790,c1(C(c2n(CCOC)nnn2)NCC2(OC)CCC2)c(Cl)cnc(F)c1Cl 49791,C1(CNC(COC)=O)CC2(CCN(C(=O)Cc3ccc4sccc4c3)CC2)CO1 49792,N1(C(C(C)CN(C)C)=O)CCC(C)(C)C1C(=O)NCc1cccnc1Cl 49793,N1(C(c2ccccc2)=O)CC2(C1)CN(C=O)CC2CO.C1(CO)CCC(=O)N(C)C1=O 49794,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 49795,C1(OC)CN(C(=O)C=CCF)CC1NC(=O)C(CO)N(C)C 49796,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 49797,n1(CCC)nnnc1C(CCCc1ccccc1)NCCC(C)C 49798,c1(C(=O)NC(CN(C(COCC(=C)C)=O)CC)C)ccc2n[nH]cc2n1 49799,CCC(C)(Cl)CNC(=O)Nc1cc(O)ns1 49800,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(N)=O)=O)CCO1 49801,N1(C(=O)C(c2cccc(Cl)c2)(F)F)CCCC(NC(C2CC(F)(CO)C2)=O)CC1 49802,c1(C(N(CCN(C(COCC=C)=O)C)C)=O)cnsc1 49803,CC1CC(NC(=O)C(C)(C)c2ccn(C)n2)CN(C(=O)CCc2nccn2C)C1 49804,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 49805,CC1=C(C(=O)NCC2N(C(C34CCC(CSC)(CC3)CO4)=O)CCC2)CCCO1 49806,C=CCC(CNC(C1CCO1)=O)C(=O)N(C)Cc1cccc(F)c1C 49807,Cc1ccc2oc(C(=O)OCc3ccc(F)c(F)c3)c(C)c2c1 49808,C12COC3(CCN(CC3)N(C(C)C)C1=O)C2.c1(C(C2CC23CCC3)=O)nc[nH]c1OC 49809,C1(CNC(C(CCCC)=O)=O)CC2CCC(C1)N2C(=O)C(C)CC1CCC1 49810,c1(C(=O)NC(C)C(F)(F)F)cncc(CNC(C2CC23CCCC3)=O)c1 49811,Cc1c(C(=O)NCCC2(O)CN(C(C3SCCC3C)=O)C2)c[nH]c1C#N 49812,N1(C(C2CN(C)C(=O)N2)=O)CCN(C(=O)CCCC2CCOCC2)CC(O)C1 49813,N1(Cc2cn(CCN(C)C(c3c(Cl)nsc3Cl)=O)nn2)CCN(C)C(=O)C1 49814,[N-]=[N+]=NCC(C(=O)NCCN1CCC1)NC(c1nnsc1N)=O 49815,C1(NC(C2(CC#C)CC2)=O)CCC2CCN(C(=O)CCc3ccc(C)cc3)C12 49816,C1(N(C)Cc2n(CC)cnc2)CCCC(N)CC1 49817,N1(C(C(C)c2cccs2)=O)CC(NC(C2CCC2C)=O)C2CCCC12 49818,c1(C(=O)NC(CNC(C(C=C)(C)C)=O)CC(C)C)cc(C)ccc1C(F)F 49819,C(CCC(C(=O)N1CCC(N(C)C)CC1)NC(C1CC1(F)Cl)=O)OC 49820,N1(C(C(C2CCOC2)OC)=O)CC(NC(c2ccc[n+]([O-])c2)=O)C2CCCC12 49821,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3ccnc(C4CC4)c3)C2)C1 49822,c1(OC)ccc2[nH]c(CN3CCC(O)CC3C(=O)Nc3csc(C)n3)cc2n1 49823,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 49824,CC1CN(C(=O)C2=CCCC2)CC(C)N(C(c2cc(Cl)cc(Br)c2)=O)C1 49825,C=CCC(C)C(=O)N1CCC(C(N2CCC(CO)CC2)=O)C1 49826,C1(C(N2CC(OC)C(NC(C3CC4(CC4)C3)=O)C2)=O)CC2(CCCO2)C1 49827,Cc1cc2[nH]c(C(N3CC(C)(C(=O)Nc4csnc4C)C3)=O)cc2s1 49828,Nc1cc(C(=O)NCCCSCCCO)cc(F)c1 49829,S(=O)(=O)(c1ccccc1C(N)=O)NCCNC1(c2nnnn2C)C(C(C)C)COC1 49830,N1(C(C=C(CCC)C)=O)CCc2nc(CNC(C3(C)CC3(F)Cl)=O)sc2C1 49831,CC1CCN(C(C2CCCN(C(=O)CCc3ccc(C#N)cc3)C2)=O)CC(=O)N1 49832,c1(OC)c(C(N2CC3C(NC(c4c(C)cccc4Br)=O)C3C2)=O)cccc1F 49833,S(=O)(=O)(c1cccc(-c2ccc3scnc3c2)c1)NC1CC(=O)NC1 49834,c1(NCCC(C)F)[nH]c(=NC2CCSCCC2C)nc2c1ncn2C 49835,N1(C(C=C(C)C)=O)CCC2(NC(c3cncc(C(F)(F)F)n3)=O)CCCCC12 49836,C1(C(=O)NCCC2(NC(CNC(C(C)n3ccnc3)=O)=O)CC2)C(C#N)C1(C)C 49837,c1(OC)cnn(C)c1Cl.C1(NC2c3nc2cs3)CCN(c2ccccc2)C1=O 49838,C1(C(=O)NC2CC(C)(NC(C(CC)Sc3ccccc3)=O)C2)CC(F)CN1C 49839,C1(NC(C2CN(C)C2)=O)CCCC1CNC(C1CCCC1O)=O 49840,c1(C(N2C(CNC(=O)Cc3ccc(F)cc3F)CCC2)=O)ncnc2[nH]cnc12 49841,c1(CC)ccsc1C(=O)N(C)CC1CCN(C(C2CC3CC3C2)=O)C1 49842,Cc1nc(C(=O)NC2CC2CNC(C2(Oc3ccncc3)CC2)=O)c(=O)[nH]c1C 49843,N1(C(=O)C(Cl)=CCl)CCC(F)(CNC(c2n[nH]cc2OC)=O)CC1 49844,C1(CNC(C2(NC(c3cc(-c4cccc(F)c4)on3)=O)CC2)=O)CC12CC2(F)F 49845,CCCC(C)C(=O)N1CCC(N(C(=O)CC(C)(C)C)C)CC1 49846,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC(C(N3CC(CO)C4(CCC4)C3)=O)C2)C1 49847,C1(C#N)(C(=O)NC(C2CN(C(c3nc(C)[nH]n3)=O)C2)C)CCCC1 49848,CC1CCCCN1C(C1CC(NC(c2cc(Cl)cs2)=O)C(O)C1)=O 49849,CC1CC(=O)NCC1C(=O)NC1(CC=CC(N2CCN(C3CC3)CC2)=O)CCC1 49850,c1(C(=O)NCC(C2CCC2)NC(CC(CC)C)=O)cc2occ(C(F)(F)F)c2[nH]1 49851,C(C(CC)CCO)NC(CCN(C(c1cnc(Cl)s1)=O)CC)=O 49852,N1(C(CCC#C)=O)CC2(C1)CN(C(C1CCC3(CC3)C1)=O)CC2CO 49853,N(C(=NCC#CC1CC1)NCC1(CO)CCCO1)C(c1ccccc1)CC 49854,C1(c2nnnn2CCCOC)(NCC2C(C)(CC)C2)CC(C)(C)OC(C)(C)C1 49855,C1(NC(c2ccc(C#N)o2)=O)CC(C(=O)NCC2CCCC2O)C12CCC2 49856,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 49857,N1(C(c2cc(Cl)c3c(c2)OCO3)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 49858,C(=O)(CC1=CCOCC1)N1CCC(C(=O)NCC2CCCC(O)C2)(CC)C1 49859,CC#CCC(C(=O)NC1CCC12CCCC2)NC(C1CCC1CCOC)=O 49860,C(=O)(C(C)C(=O)NCCCN(CCCNC(C1CNC(=O)C1)=O)C)OC 49861,C1(NC(C23CCC(OC)C2C3)=O)CN(C(=O)CC2CC3(CCO2)CC3)CCC1O 49862,S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(c2cnn(C3CC3)c2)=O)cn1)NC 49863,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2ON=C(C)C2C)=O)CC1 49864,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 49865,c1(C(=O)NCC2(CNC(CCNC(=O)NC)=O)CC2(F)F)nc(C(C)C)cs1 49866,C(=O)(CCCCN(C(=O)C(C)SCC(C)C)C)NCc1ccc(CC)s1 49867,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 49868,Cc1nc(C(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 49869,c1(C(=O)NCC(C)NC(COC(C)=O)=O)sc(Cl)c(Cl)c1OC 49870,c1(CSCC(N2CCC(CNC(c3n(COC)ncc3)=O)C2)=O)ccc(F)cc1 49871,C1(C(C)NC(=O)CCN(CC(F)(F)F)C)CCCN1C(=O)CC1(C)CCCO1 49872,N1(C(C(=O)NC(c2cc(C)c(C)s2)C)=O)CC(C)(C)COC(C)C1 49873,CCCC(C)C(=O)NCC(C)(O)CNC(=O)CCc1cc[nH]n1 49874,CC1=C(C(=O)N2CCCC(C)(C(=O)Nn3cncn3)C2)CCC1 49875,C1(NC)CN(C(N(CC(C(C)C)C)C)=O)CC1CC(C)(C)C.C(C)(C)(C)O 49876,C(=O)(C(C)CCCOC)N1CCC(CN(C(C(CCC)O)=O)C)CC1 49877,Cc1c(Cl)c(NC(N2CC(C(c3ccccc3)=O)C(C)(C)C2)=O)nc2ccccc12 49878,CCCC(C)CCCC(=O)Nc1nnc(CN2CCCCC2)s1 49879,c1(OC)c(C(N2CCC(N(C)C(c3csc(SC)n3)=O)C2)=O)cccc1F 49880,c1(OCC)cccc(C(c2nnnn2C(C)C)Nc2cc(CO)on2)c1C 49881,c1(C(N2CCN(C(C3C(C)CC(=O)N3)=O)CC2)=O)ccnc(C#N)c1 49882,CCCC(C(=O)NCCN(C(=O)C=Cc1cnc(C(C)(C)C)nc1)CC)C(C)C 49883,N1(C(CCC(CC)C)=O)CCC2CN(C(C3CCCCN3C(C)=O)=O)CC2CC1 49884,N1(C(CC2=NC=C2C(=O)OC)=O)CCN(C(c2ccon2)=O)C(CC(F)(F)F)C1 49885,C(CCN=c1cc(Cl)nc(C2CCC2)[nH]1)N1C(C)CCCC1 49886,C(CCC(C)C(C(=O)NCC1CCCO1)N1CC(F)CC(F)C1)=C(C)C 49887,CC(CNc1cc(NCc2nccn2C)ncn1)CC(F)F 49888,c1(NC(C(c2n(C)ncc2)N(C2CC2)CC2OC3CCC2C3)=O)cccc(Cl)c1O 49889,c1(C(CC)=O)ccc(CC(=O)NCCCCN(C)C(c2cc[nH]c2CC)=O)cc1 49890,N(C(=NCCN1CC2CCC1C2)NCCN1CCCC1)Cc1scc(C#N)c1 49891,O=C(C1=CCC(NC(c2n[nH]nc2Cl)=O)C1)NCC(c1ccsc1)O 49892,CCCC(F)(F)C(=O)NCCC1(C)CCN(C(=O)C(C)c2cc[nH]n2)C1 49893,C(=O)(C(C)(C)C(=O)NCC1CC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1)OC 49894,N1(C(C2CC(CC(=O)Nc3n(CC)ncc3)C2)=O)CCNC(=O)CC1C 49895,C12(NC(CCCOC(C)=O)=O)CCC(CC1)N(C(=O)C1CC1)C2 49896,c1(C(N(C2CCCN(C(=O)CCc3cocn3)C2)CC)=O)cc(F)cnc1O 49897,C1(CNC(C(CCOC)C)=O)(NC(C2CCC(F)(F)C2)=O)Cc2ccccc2C1 49898,c1(N(CCC#C)CCNC(C2(N(C)C)CC2)=O)n[nH]c(C)c1Cl.C1C(=O)N1 49899,C12(NC(c3cc(C(C)C)no3)=O)CCC(CC1NC(c1csnn1)=O)C2 49900,c1(SCC(=O)NCC(CNC(CCOCCCC)=O)C)nnnn1C1CC1 49901,Cn1cc(CCC(=O)NCC2CN(C(C3(c4ccno4)COC3)=O)C2)nn1 49902,C1(NC(C2CC=CCO2)=O)CCC2CCN(C(c3coc(CC4CC4)n3)=O)C12 49903,CC(CC1CCC1)CN=c1[nH]c(=NCCN2CC(C)OC(C)C2)[nH]c2c1CSC2 49904,c1(C(N2CCC(N(C(C(C(CC)C)N(C)C)=O)CC)C2)=O)c(F)ccc(F)c1N 49905,C(CC(C(=O)NC1CC(O)C1)NC(=O)Cn1cnnc1O)SC 49906,CC1CN(C(c2cnc(O)nc2O)=O)CC(CCNC(c2ccncc2N)=O)O1 49907,CCCCC(CN(C(=O)NCc1ccc(Br)s1)CC1(C)CCC1)CC 49908,CC(C(=O)Oc1c(COCNCC(=O)NCc2ccccc2)cccc1)S(N)(=O)=O 49909,CC#CCCCC(=O)NNC(=O)Nc1ccc(COC(=O)C(F)(F)F)cc1C 49910,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(CC(C)C)n2)=O)CCC1C 49911,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 49912,CCCCC(C(=O)NC1CCCCCC1C)NC(=O)C=CCN1CCCC1 49913,C(=O)(CCC(C)S(C)(=O)=O)NCC1CC(NC(CC(C)C(F)(F)F)=O)C1 49914,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 49915,Cc1ncc(C(N2CCCC2C(=O)N(C(C)CCO)C)=O)c(=N)[nH]1 49916,c1(-n2c(C(C3CC3)C)nnn2)ccccc1C(=O)NC(C)C(=O)NCC1(C)COC1 49917,C(=O)(CCCCCC#N)N1CC(O)(C(C)(C)NC(=O)COCC2CCCC2)C1 49918,Cc1ccc2[nH]c(C(N3CC4CCC4(NC(C4CCC4(C)C)=O)C3)=O)cc2c1C 49919,N1(C(C2N(CC)CCC2)=O)CC2(NC(C3(N4CCOCC4)CC3)=O)CCC1C2 49920,C(CC(O)CNC(=O)CN1CSCC1=O)NC(=O)Cc1cnn(C2CCCC2)c1 49921,C1(CNC(C2CC(C(C)(C)C)C2)=O)CCCN(C(C2CCCCCC2)=O)C1 49922,C=Cn1nncc1NC(=O)C(=O)NCC(C)Oc1cccc(Cl)c1 49923,C(C(N=[N+]=[N-])C(=O)N1CC(O)CC1C(=O)NC(c1nnc(O)o1)C)OCC 49924,N1(CCNC(c2cccnc2Cl)=O)CCC(=O)N(CC23CCC(CC2)O3)C1=O 49925,N1(C(CC2CCC(OC)C2)=O)CCN(CCCc2ccsc2)CC1 49926,C1(CC)(NC(=O)CC2CCC(=O)O2)CCN(C(=O)CCCn2ccnn2)CC1 49927,C1(S(C)(=O)=O)(C(=O)NCC2C(CNC(CSC)=O)C2)CCCCC1 49928,c1(C(C(=O)OC)C(N2CC(C(CCC(=O)OC(C)(C)C)C)C2)=O)ccc(C)cc1 49929,C=CC1(C(=O)NCCC(C)N(C(=O)C(C)(C)NCC(F)(F)F)C)CCCCC1 49930,Cc1cccc2c(C(N3CCC(NC(=O)Cn4nnc(=N)[nH]4)C(C)C3)=O)n[nH]c12 49931,N1(CC)Cc2ccc(NC(C3(OC(COC)C(C)(C)C)CCCC3)=O)cc2C1=O 49932,N1(C(CCNC(N)=O)=O)CCC2(CCCCN(C(C3CCC4(CCC4)CC3)=O)C2)C1 49933,Cn1nc(C(N2CC3CC3(CNC(=O)CN3CCC(C(N)=O)CC3)C2)=O)cc1O 49934,C(=O)(C1c2c[nH]nc2CCC1C)N(C(CCNC(c1c(O)ccc(C)c1)=O)C)C 49935,C(=O)(CCCC1CCCO1)NCC1C(C(C)C)C1.C12CC(C1)C(=O)NCC2 49936,c1(-c2cn(CCC(N3CC(C)NC(=O)C3)=O)nn2)ccc2ncsc2c1 49937,C1(N(C(c2c(CC)csc2)=O)C)CN(C(=O)C(CC(C)C)NC(N)=O)CC1(C)C 49938,S(=O)(=O)(c1cc(C(=O)OC)c(C)c(Cl)c1)N1CCN(CCCOCC)CC1 49939,C(=O)(CS(=O)(=O)N1CCN(C(C2(C)CCN(C(=O)NC(C)(C)C)C2)=O)CC1)OC 49940,N1(NCCOCC(=O)Nc2cc(C)ncc2)CCC(C)CC1c1ccccc1 49941,C1(C)(C(=O)Nc2cn(CCC)nc2)CCN(C(C2CN(C)CCO2)=O)CC1 49942,CN1CC(C(=O)NCC2CC(O)CN2C(C23CSCC2C3)=O)CCC1=O 49943,c1(OC)c(C)nc(C2CC2)[nH]c1=NC1CC(NC(C2CCCN(C)C2)=O)C1 49944,C(=O)(CC(O)CC(C)C)N1CCC(C(NOC(CCCC)C(=O)NCC)=O)C1 49945,c1(SCCC(N2C(C)CC(CNC(c3c[nH]c(=N)s3)=O)C2)=O)ccc(F)c(F)c1 49946,c1(C(=O)NC2CN(C)C(=O)N2)cc(CC2CC2)cc(F)c1.C1(OC)CSCC1 49947,N1(C(c2cc(OC)n[nH]2)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 49948,c1(OC)cccc(C(=O)N(C)CC2CN(C(c3cnco3)=O)CCO2)c1OC 49949,CS(=O)(=O)c1ccccc1CC(N1CCC2CN(C(=O)C=CC3CC3)C2C1)=O 49950,C(=O)(C1CC(C(C)C)Cn2ccnc21)NCC1(NC(c2nc(CC)sc2)=O)CC1 49951,c1(C(=O)NC2CN(C(C)=O)C2)cc2ncsc2[nH]1.C12CCC(CC1)C(=O)N2 49952,C1(C(=O)NCCCNC(C2CCCC2C(F)(F)F)=O)CCS(=O)(=O)CC1 49953,C1(CNC(c2ccc(Cl)o2)c2nnnn2CC2CCCO2)CCCCCC1 49954,c1(C(N2CCC(N(C)C(c3cnco3)=O)C2)=O)ccc2c(n1)CCCC2 49955,c1(CC)cc[nH]c1C(=O)NC1CC(NC(=O)Cn2cnc(C(F)(F)F)c2)C1 49956,c1(NC(=O)Nc2cc(C)[nH]c2)cccc(OC2CCCCC2C)c1 49957,c1(C(=O)NC2(C)CCN(C(C(C)SCC)=O)C2)cc2c(Br)c(C)ccc2[nH]1 49958,c1(-c2n(CCC=C)ccn2)cccnc1-c1nccn1CCCS(N)(=O)=O 49959,N1(C(CCC(C)SC)=O)CCC(C)CC1CNC(c1ccc(C(F)F)c(F)c1)=O 49960,C1(NC(=O)COC2CCCOC2)CN(C(C2(Br)CC2)=O)CCC1CO 49961,C1(C(N2CC3CC3(C(N3CCC(n4ccnn4)C3)=O)C2)=O)CC2CC1CC2O 49962,c1(C(C)C)ccc(Br)cc1C(=O)NC1CC(NC(=O)C(C2CCOCC2)F)C1 49963,c1(N2C3CN(C(C(C(C)C)NC(C)C)=O)C(C3)C2)ccc(Cl)cc1Cl 49964,C1(NC(CCN(C)CC)=O)CCCN(C(c2cc(C)n(C3CC3)n2)=O)C1C 49965,CCCCC(C)CCC(=O)NCC1CC(NC(=O)CN(C)CC)CCO1 49966,Cc1onc(Cl)c1C(N1CC2C(CNC(c3snc(Cl)c3Cl)=O)C2C1)=O 49967,N1(C2CN(C(C3C(C)CCC3)=O)C2)CC(NC(=O)CSc2cnn(C)c2)CC1=O 49968,C1(NC(C=CC(C)C)=O)C2CC1N(C(=O)Cn1cc(Br)cn1)C2 49969,C1(C(N2CC(CC(=O)NC3(C4CC4)CC(=O)C3)(OC)C2)=O)CC2CCCC2C1 49970,c1(C(=O)NC2CCC(CCNC(C(C)(C)OC)=O)C2)cnc2sccn2c1=O 49971,N(S(=O)(=O)N1C(CC2CC(F)(F)CO2)CCN(C)C1)CCCOCC 49972,C1(C2CC2)(C(=O)NCCCN(C)C)CN(C(c2ccc(Cl)s2)=O)C1 49973,N1(C(CS(CC)=O)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2csc(C)n2)C1 49974,N1(C(C(C)OC)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 49975,C1(C(=O)NC(C2N(C(c3n[nH]c(CC)c3Cl)=O)CCC2)C)CCOC(C)(C)C1 49976,c1(C(C)OC)nc(C)c(C(=O)NCCCC2CCCN2C(=O)CN2CCC2)s1 49977,N1(C(c2c(C)c[nH]n2)=O)CC2CCC(Nc3ncc4c(n3)COC4)CC2C1 49978,C1(C(N2CC(OCCNC(C(CC)=CC)=O)C2)=O)COCC(=O)N1C(C)C 49979,C1(NC(Cc2nc(C)sc2)=O)(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CCCCC1C 49980,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 49981,CCCCC(CCCC)NC(C1CC2C=CC1N(C(C1CC1C(C)(C)C)=O)C2)=O 49982,N1(c2snc(OC)n2)CCC(C2(NC(=O)C(C)SC(F)(F)F)CC2)CC1 49983,c1(C(N2C(Cc3cn(CC(=O)OC)nn3)CCC2)=O)ccc2c(c1)CN(C)C2 49984,n1(CC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CCNC(=O)C2)c(C(C)C)n1 49985,C1(OC)CCCC(C(=O)N(C2CCCC2)CCCNC(c2cn(C)c(C)n2)=O)C1 49986,C(N=c1[nH]cnc(Cl)c1F)C1C(NC(Cc2c(C)ccnc2)=O)CCCCC1 49987,CCC(CC)CCC(=O)NCC1(C)CCN(C(=O)C(C)CNC(=O)OC(C)(C)C)C1 49988,C(=O)(C(F)C(=O)N(CCC(=O)N(C)CCN(C)C(C)=O)CC)OCC 49989,C(=O)(C(C)(CCC)CCC(C)C)NCC(CC)(C)NC(=O)CCc1cccc(Cl)c1 49990,N1(C(c2n(CC)nc(C)c2)=O)CCC2(CC2C(=O)NCCF)C1 49991,c1(C(N(CCNC(C=COCC)=O)C2CC2)=O)ccnc2ncnn12 49992,c1(OC)ncc(C(=O)N(CC(C)NC(C2CC3CC2C3)=O)C)cc1Cl 49993,Cn1nc(Br)c2c(NCC(O)CCNC(c3ccc(Cl)cc3F)=O)ncnc12 49994,C(=O)(CCCC(C)(C)C#N)N(CC(F)CN1C(=O)CCC1)C 49995,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C 49996,c1(CC)ncc(CN2CCCC(N3CCN(C4CCNC4=O)CC3)C2)c(=N)[nH]1 49997,c1(C(=O)NCCCN(C)C(c2ccn3ccsc23)=O)ccn2nccc2c1 49998,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCSC(C)C)CCO2 49999,N1(C(C(C)n2ccnn2)=O)CC(C(N2CCC(CO)C2)=O)(N(C)C)C1 50000,Cc1cnc(NC2CN(C(c3cnc4c(F)cccn34)=O)CC2C)c([N+](=O)[O-])c1 50001,c1(C(CC)NC(=O)N(Cc2ccsc2)CC2(C)CC2)ccccc1 50002,c1(C(N(C(C(=O)NC(C)Cc2nn[nH]n2)C)C2CC2)=O)ccnc(O)c1 50003,C1(C)(C(=O)NCCC(C)N2CCCC2)CCCN(C(C2CCOC2(C)C)=O)C1 50004,CC(C)C(O)C(C)(C)C(=O)NC1COCC1C(N1CC(C)(CCO)C1)=O 50005,c1(CC(=O)OC)cccc(CN(C(CC2N(C(C3CC3C)=O)CCOC2)=O)C)c1 50006,C1(NC(C=CC(C)NC(=O)CCCOCC(F)F)=O)CC(N(C)C)C1(C)C 50007,N12C3CCC1CC(C3)C2=O.C12(C(C)N(C(=O)CNC(=O)C3CC3)C)CCC(CC1)C2 50008,N1(C(c2cnn(CCO)c2)=O)CCC(C(C)NC(=O)CCSC)CC1C(F)(F)F 50009,C1(C(N(CC=CC(=O)N(CC(C)C)CC(C)C)C)=O)CC1C1CCCC1 50010,C(=O)(CCCCCCC(=O)N1CC2CC(NC(C3(OC)CCCC3)=O)C1C2)OC 50011,Cc1ccc(C(O)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50012,CC(CNC(C1C2(CC2)C12CC2)=O)CC(=O)N1CCC1C(=O)N(C)C 50013,N1(C(C(C)N(C(=O)CC2CSC2)C)=O)CCCCC1.C1(N)CC1 50014,c1(CN(C(C2CC2NC(CCNC(=O)OCC)=O)=O)C2CC2)ccnn1C 50015,C1(CC(Cl)(Cl)Cl)(C(=O)O)CCN(C(C2CC(O)CS2)=O)C1 50016,c1(C(C(=O)NCC)N(CCC(N)=O)C)nc(C#N)cs1.C1CN1 50017,Cc1cc(NCCc2nnc(C)o2)nc(C)c1.C12(CCC1)CC(=O)N2 50018,Cc1cnc2n1CCN(CCCSc1cc(C(N)=O)cs1)C2 50019,C(C)(C)(CC(=O)NCC1C2CC1N(C(=O)C(C)Cc1cccc(Cl)c1)C2)OC 50020,c1(C(N2C(CN(C(c3nccc(C)n3)=O)C)COCC2)=O)cc2c(ncn2C)[nH]1 50021,c1(C(=O)NC2C3CN(C(c4ccn(C(C)(C)C)n4)=O)C2C3)n[nH]c2c1COCC2 50022,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50023,c1(CC)nc(C(=O)N(CCOC)CC2CCOCC2)c(Cl)s1.C(C)(C)C 50024,c1(-n2cc(CN3CCCC(NC(c4ccns4)=O)C3)nn2)ccc2c(c1)CCO2 50025,C(=O)(C(C)(F)F)NCC(C)CNC(=O)CC(c1ccccc1)N(C)C 50026,CC1CN(C(c2csc(C#N)c2)=O)CCCN1C(c1cnc(Cl)[nH]1)=O 50027,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cscn1 50028,C1(C(=O)NC(C)CC(C)N(C)C)(NC(C)=O)CCCOC1.N12CC(C1)CC2=O 50029,C(C)(CNC(=O)COCc1nc[nH]n1)(C(C)C)NC(C(c1ccnn1C)C)=O 50030,c1(OC)ccc(N)c(C(N2CCOCC2CNC(=O)Cc2cc(Cl)cs2)=O)c1 50031,C1(NC(C(=O)NCCN2CCN(C3CCOC3)CC2)=O)CC12CCCCC2 50032,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50033,c1(C(=O)NCCN(C(C(CC=CCC)C)=O)CC)nn2cccnc2c1Br 50034,Cc1cnc(CNC(C2CCCN2C(=O)C(C)(F)F)=O)o1 50035,c1(C(=O)NCCNC(=O)CCc2cn[nH]c2)ccc(F)c2ncccc12 50036,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50037,CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1CNC(=O)Cc1ccc(O)cc1 50038,Cc1ccc(Cl)cc1OCC(=O)NC1COCCN(C(c2ccc(=N)[nH]n2)=O)C1 50039,C(=O)(C1=C(C)OCC1)NC1(C(=O)NCC(C#C)CC)CC1 50040,CN1CCC(C)(C(=O)NC(C2CCOC2)CNC(=O)Cc2csc(S)n2)C1 50041,CCCC(C)C(=O)NCC1CC(NC(=O)CN(c2ccc(Cl)cc2)C)C(O)C1 50042,C(=O)(CCC(=O)NCC(CC)NC(C1CCCN1c1ncccn1)=O)NCC 50043,C(=O)(C1=COc2ccccc2O1)N(C)CCN(C)C(=O)NC12CCCCC1C2 50044,c1(CCC)nnc(S)n1CC(=O)N(C)CCN(C(=O)CCOC(C)C)C1CC1 50045,CC1CN(Cc2nc(-c3ccc(F)cc3)n[nH]2)CCN1C(C1(C)CC=CC1)=O 50046,N1(C(CC2N(C(c3n(CC)c(O)nc3)=O)CC2)=O)CC(N(C)C)C2(CC2)C1 50047,C(C)(C)(C(c1nnnn1CC(F)F)NCC1C=CCC1)OCC 50048,c1(CCCC(=O)NC(Cn2cc(CC(CC)(C)O)nn2)C)c(C)nn(C)c1C 50049,C1(CC(=O)NCCN(C(=O)Cn2cc(C3CC3)cn2)CC)CCC(=O)NC1=O 50050,Cc1cc(I)c(C(N2C3CCC2CC(C(=O)NCc2cnccn2)C3)=O)cc1C 50051,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)N(C)C 50052,N1(C(C(C)=CC)=O)CCN(C(C2CCCS2)=O)C(c2ccc(F)cc2)C1 50053,CCCC(CNC(c1cc(CO)ccn1)=O)C(=O)NC1CCCC1CN=[N+]=[N-] 50054,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50055,C(=O)(CC(C=C)CCC)N(CCCCC(C)(C)C1CCC1)C(C1C(=C)C1)=O 50056,N1(C(CC(C)CNC(=O)CCc2ccc[nH]2)=O)CC2(CNC(=O)N2)C1 50057,C1(NC(CC(C)CF)=O)CN(C(c2cc(CCN3CCCC3)on2)=O)CC1(C)C 50058,CC1Cc2cc(N(C=O)C(c3ccc(C(C)C(F)(F)F)cc3)=O)ccc2O1 50059,CN1C(=O)CSC1=CC(=O)NCC1CC2CCC1N2C(=O)CN1CCCCC1=O 50060,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)nn4C)=O)CC23)=O)c(O)n1 50061,N1(C(c2ccc(C(N)=O)cn2)=O)C2CCC1CC(CNC(C1CSCCS1)=O)C2 50062,Cc1ccc(C)c(C(=O)NC2CN(C(C3CC3C(F)(F)F)=O)CC23CC3)c1O 50063,c1(CC(=O)NCC(C)N(C(=O)Cc2nccn2C)CC)ncc(F)cn1 50064,C1(C(=O)NCC2(CNC(C3(F)CCS(=O)(=O)C3)=O)CC2)CC(c2ccccn2)=NO1 50065,C1(C(=O)OCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCSC)C1(C)C 50066,c1(C(=O)NCC(CN(CCC)C(C)=O)C)ccc2c(c1)SCC(=O)N2 50067,N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)C=Cc2cnn(C)c2C)C2CC12 50068,N1(C(c2c(OC(C)C)nccc2)=O)CCC2(CC(NC(=O)CC(F)(F)F)CO2)C1 50069,c1(CCN=C(NCCOCC=C)NCCF)nnc2n1CCCC2 50070,c1(OC)ccc2c(c1)OCC2C(=O)N1CCC(C)C(F)(F)CC1 50071,C(=O)(CCC[N+](=O)[O-])NCC1(OC)CN(C(=O)CC2CCCOCC2)C1 50072,c1(C(=O)NCC(CC)NC(=O)CSC(C)=O)ccc2c(C)noc2c1 50073,CC1(N2CCCC2Cc2ccccc2Br)CS(=O)(=O)CCO1 50074,CS(=O)(=O)C1CCC(CNC(=O)C(=O)NC2CCC(O)C2)CC1 50075,C(CC(C)C)(C(=O)NCc1ccoc1C(N1CC(N(C)C)C(C)(C)C1)=O)OC 50076,CC(C)CC(C)(O)C(=O)N1CCN(CCNC(=O)CC(=O)NC2CC2)CC1 50077,c1(C(N2CCC(N(C(C(CCOC)C)=O)CCO)CC2)=O)c[nH]c2nccc-2c1 50078,CCC(CC(=O)N1CCN(C)CC(c2ccccc2)C1)C(F)F 50079,c1(CC)c(C(=O)NCC2CC(NC(c3ncn(CC)n3)=O)C2(C)C)cccc1F 50080,c1(OC)cc(C(=O)NC(CCN(C(=O)CC2CC2(Cl)Cl)C)C(C)C)ccc1C 50081,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)CN1CCCC1 50082,CC1CCN(Cc2ccccc2O)CC1.c12ccnc(c1)CN(C)NC2=O 50083,N1(C(C=C(C)C(C)(C)C)=O)CCOC(CCNC(=O)CN2CC(C)C2)C1 50084,Cc1cc(CC(=O)NC(C2CC(NC(=O)CCn3ccnn3)C2)C)nn1C 50085,c1(C(=O)NCC2CCN(C(C3(CC#C)CCCO3)=O)C2)cncc([N+](=O)[O-])c1 50086,c1(OC)nc(N2CCCCC(NC(=O)COC3CCOC3)C2)nc2ccccc12 50087,c1(C(N(CC(C)NC(=O)Cc2nnc(S)n2C)CC)=O)cc2cccnc2[nH]1 50088,Cc1nc(O)sc1CN(C(C1CCOC1c1nccn1C)=O)C1CC1 50089,Cn1c(C(c2nnnn2CC2CCOC2=O)NCCF)ccc1Cl 50090,c1(C(=O)NC2CN(C(C3(C=C)CCC3)=O)CC2C)ccc(OCC2CC2)cc1Cl 50091,c1(CC)ncc(C(N2CC(NC(=O)C(C)CSC)CC2(C)C)=O)c(C)n1 50092,C1(CN(C(C(CC#C)C2CC2)=O)c2cccs2)CN(C(c2ccc(Cl)[nH]2)=O)CC12CCC2 50093,CCC(C(=O)NC(C)(C)C=CC(=O)NC(CC1CC1)CC1CC1)n1cncn1 50094,c1(C(CC=C)OC)cn(C)nc1-c1nc(C2CC2c2ccoc2C(F)(F)F)no1 50095,CCC(C)CC(=O)C(=O)N(C(C)C(=O)NCCc1cc(C)on1)C1CC1 50096,C1(C(N2CC(COC)(NC(C3(F)CCOCC3)=O)C2)=O)(OC)CCOCC1 50097,C1(NC(c2cc(OCC)no2)=O)CC(NC(C2(CCOC)CCCC2)=O)C1(C)C 50098,c1(C(=O)NC(CNC(CN(C(C)C)C)=O)C(C)C)cn2c(n1)SCC2 50099,S(=O)(=O)(c1nc(N2CCC(C(C)(C)CO)CC2)ccc1Br)NC(CC)CO 50100,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50101,N1(C(CC(C)=C(C)C)=O)CCCCCC1CNC(c1cc(C(F)(F)F)nn1C)=O 50102,C1(CC(=O)NCCCNC(c2cc(Sc3cccs3)on2)=O)CCCCO1 50103,c1(SCC(=O)NCC(CC)NC(=O)CN2CCCNC2=O)ccccc1C(C)C 50104,c1(C(=O)NCc2c(C(=O)Nc3ccc(CCC)cc3)c[nH]n2)cc2occc2[nH]1 50105,c1(OC)ccccc1CCCC(=O)Cc1ccccc1.c1(=O)c(=O)o1 50106,C(=O)(C(C)C(O)CCCC)NCCC1N(C(c2n(C=C)ncc2)=O)CCCC1C 50107,Cc1ccc2nnnn2c1N(CC(C)C(F)(F)F)c1ccncc1 50108,CCCCCCC(CC)C(=O)N(CCNC(c1nnn2c1COCC2)=O)CC 50109,C1(C(=O)OC2CC(C(CC)CC)OCC2)CC2(CCOCC2)CCO1 50110,N1(C(c2ccccc2F)=O)CCC(C(=O)N(C23CCC2C3)C2CC2)CC1 50111,N1(C(CC(C)C)=O)CCN(C(=O)C(C2CCC2)C2CC2)CC1c1ccc(F)cc1 50112,N1(C(C(C)(CO)NC(CCCCC=C)=O)=O)CC(C)OC2(CCC2)C1 50113,C1(C(=O)NCCC2N(C)CCC2)CCCC(NC(C2(CO)CCCC2)=O)CC1 50114,N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2CCCCC2C)=O)CC(C)C1 50115,C1(C(N2C(C(N(CCn3c(C)ncc3)C)=O)C=CC2)=O)CCCC(C)(C)C1 50116,C12(C(=O)NC(CN(C(c3cc(C)nc(O)n3)=O)C)C)OCCCC1C2(F)F 50117,C1(COC)CCCCN1C(c1ccc(F)cc1)C(=O)Nc1ccc(C)nc1 50118,c1(C(=O)NC(C)CNC(=O)C=C2CCC2)cccc2cnnn12 50119,c1(C(N2CCC(NC(C3CC34CCC4)=O)(CF)C2)=O)cc2c(Br)cccn2n1 50120,N1(C(=O)C2=CS(=O)CCC2)CCOCC2(COCCN2C(C2CCSCC2)=O)C1 50121,CCS(=O)(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2F)=O)C1 50122,c1(N(C)Cc2ccn(CC(F)F)n2)cc2c(cc1Br)CCC(=O)N2 50123,N1(C(C2C(CC)C2)=O)CCC(O)(CCNC(c2ccc(CC3CCC3)cc2)=O)C1 50124,CC1CN(C(=O)CC2C(C)(C)C2(C)C)CC1NC(c1ccc(CO)cn1)=O 50125,c1(CC)cnccc1C(N1CCOC(C(=O)NCC2(C)CCCO2)C1)=O 50126,N1(C(COC)=O)CCN(C)CC1CNC(=O)CC(c1ccc(Cl)cc1)O 50127,c1(C(N(C)CC2CCCN2C(=O)CCOc2cccnc2)=O)cn2c(n1)SCC2 50128,CC1(C)CCCCC1(C)NC(c1ccc(CNC(C2(C#N)CCC2)=O)nc1)=O 50129,N1(C(C2OCCC(C)C2)=O)CC2CN(C)CC(C1)O2 50130,c1(CC(=O)NCC2C(NC(=O)CNC(C3CC(F)(F)C3)=O)CC2)cncc(O)c1 50131,CCN(C)N1CCNC(c2ccc(Cl)cc2)CC1 50132,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50133,C1(NC(=O)CCCC2CCCC2)CC2(C1)CC2NC(=O)CC1CC(CF)C1 50134,c1(C(=O)Nc2cc(F)cnc2Cl)cc2cc(-c3cccc4c3OCO4)ccn2n1 50135,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50136,C1(C(N2C(CC(=O)N(c3cnccn3)C)CCC2)=O)CCCN(C(C)(C)C)C1=O 50137,N1(Cc2cccc(OC)c2)C(=O)CN(CC(c2ccnn2C)O)C1=O 50138,CC1CN(C(=O)C(C)C#N)CC1CCNC(=O)C(c1cccc(O)c1)(C)C 50139,c1(OCC)ccccc1C(CC(=O)O)NC(=O)Cn1cccn1 50140,C(C)(CN=c1[nH]c2ccccc2cc1C#N)NC(Cn1ncc(C#C)c1)=O 50141,c1(NC(C(C2CCN(C(c3cocn3)=O)CC2)C)=O)cncc(Cl)c1 50142,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C(=O)CCSc1cccs1)C)(C)C 50143,c1(COC)nc(C(=O)NCC2(NC(=O)CCc3n[nH]c(C)n3)CCCC2)co1 50144,C1(NC(C(Cc2ccsc2)NC=O)=O)CC2CCC1N2C(=O)CC1COCCO1 50145,N1(C(CCCCOC)=O)CCC(C2CCN(C(=O)Cc3c[nH]ccc3=O)C2)CC1 50146,c1(C(=O)NC(C)CNC(=O)CN(C)CCO)cc2nc(O)[nH]c2cc1N 50147,Cc1ccn(C)c1C(N1CCC(C(N2CCCC2)=O)C1)=O.c12cnc(o1)[nH]c2=O 50148,CCC(CC)(C(=O)NCCCC(=O)N(C(C)CC1CC1)C)C(C)C 50149,Cc1ccc(Cl)c(C(N2CCC(O)C(NC(=O)C(C(C)(C)C)C3CCC3)C2)=O)c1 50150,C1(C2CCCN(C(c3c(F)ccc(F)c3F)=O)C2)(NC(C(CCSC)O)=O)CC1 50151,c1(C(=O)NC2C(C)CN(C(=O)C=CC(C)(C)C)C2)nn(C)cc1S(C)(=O)=O 50152,N#CC1(C(=O)N(CCCNC(=O)CCOC2CCOCC2)C2CC2)CCCCC1 50153,c1(CN(C(C2(SC)CCCOC2)=O)C2CC2)nc(O)c2sccc2n1 50154,c1(C(=O)NC(CN(C(=O)Cn2ncc(O)nc2=O)CC)C)ccc2cc[nH]c2n1 50155,C1(C(N2CCC(CNC(CCC#C)=O)C23CC3)=O)CC12CCC1(CC1)CC2 50156,c1(C(N2CC3C(NC(c4ccn(CC)n4)=O)C3C2)=O)ccc(O)nc1Cl 50157,C1(C(C)NC(C2(C(=O)N(C)C)CC2)=O)CCN(C(=O)CCc2nncn2C)CC1 50158,c1(CNC(C(=O)OC)CC2COC(C)(C)O2)ccc2c(c1)cc(C)n2C 50159,C(C1CN(C(=O)C(C2CC2)SC)CC1C(=O)NC1CCN(C)C1=O)=CC 50160,c1(NC(C2N(C(CCNC(C)=O)=O)CCC2)=O)nnc2ccc(Cl)nn12 50161,O=C(NN1CCCC1NC(C1CCCS1)=O)N1CCN(C2CCC2)CC1 50162,CCC(C)C(CC(=O)N1CC(O)C(C#C)C1)NC(C1CCCS1)=O 50163,c1(C(=O)NCC(C)(C)NC(C2CC3(CCC3O)C2)=O)cc(F)cc(F)c1O 50164,C(=O)(CCCC(=O)N1CC2(CNC(=O)CC3(C)CC(F)(F)C3)CC1CO2)NC 50165,c1(N2C(C)(C(=O)NCc3ccc(O)cc3O)CCC2)ncnc2sc(Br)cc12 50166,c1(C(=O)NC(CNC(c2cc(C)nn2C)=O)CO)cc([N+](=O)[O-])cn1C 50167,c1(C(=O)NC2CN(C(c3c(C)nns3)=O)C(C)CC2)cccc2nc(Cl)cn12 50168,c1(N2CCCC(NC(C(C)OCc3ccccn3)=O)CC2)ncc(C#N)cc1Cl 50169,N1(C(CN(CCOC)C)=O)CC2CC2(NC(=O)COC(C)(C)C(F)(F)F)C1 50170,Cc1cnc(C(F)(F)F)cc1C(=O)NC12CC1CN(C(C1(N(C)C)CC1)=O)C2 50171,C1(NC(=O)CCC2CCN(C(=O)CC3CC4C=CC3C4)C2)CCC(C2CC2)C1 50172,C1(O)(C(N2CC(CNC(C3N(CC)CCC3)=O)C2)=O)CCCC(C)(C)C1 50173,C1(OC)CCCC2CN(C(c3cnc(-c4nc[nH]n4)nc3O)=O)CC12 50174,C1(C(=O)NC2(C3CCC3)CN(C(C(C)(C)C3CC3)=O)C2)CCCCC1F 50175,N1(C(c2c(CC)scc2)=O)CCC(C(C)(C)NC(c2csc(C)n2)=O)CC1 50176,C1(CC=C)(C(=O)NCC2CCN(C(=O)C(c3ccccc3)O)C2)CCCC1 50177,n1(CC(=O)N(C)CCn2cc(C3(C)CNCCO3)nn2)cc2ncccc2n1 50178,N1(C(c2cncc(C)c2)=O)CCc2nc(CNC(C3CC(F)CN3C)=O)sc2C1 50179,C#CC(CC(C)C)NC(=O)CCN(C(=O)C(C)(C)CC)C 50180,CN1CCCC12CN(C(C1(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1)=O)C2 50181,c1(OC)ccc(C(N2CCN(C(C3CC(O)C3)=O)C3CC23)=O)c(OC)c1Cl 50182,C(CC(C(C)C)NC(c1cccc(C2CCC2)n1)=O)NC(C=CC)=O 50183,C(CN=c1nc(OC)[nH]c(NCC(=O)N(C)CCC2CC2)n1)c1cnc(OC)s1 50184,C(CCC1CCC1)(C(=O)NCC1CCC(F)(F)C1)NC(C(OC)OC)=O 50185,c1(CC)cccc(C(N2CCC(N(C)C)(CO)C2)C(=O)Nc2ccccc2)c1F 50186,c1(NC(C2C3CN(Cc4cc(OC)cc(F)c4)C2C3)=O)c(F)ccc(F)c1Cl 50187,N1(C(Cn2ccc(C)n2)=O)CC2(CC2)CC1C(=O)NCCC1OCCO1 50188,c1(C(=O)NCCCCC2CN(C(C3CC(CCC)C3)=O)C2)cc(C)nn1C 50189,C12(NC(c3[nH]c(=NC)sc3)=O)CCOC(CNC(=O)Cn3nccn3)(C1)C2 50190,c1(CNC(C2CN(Cc3scc(C)c3)CC2O)=O)ccc2cc[nH]c2c1 50191,C1(COC)CCN(C(C2CC(CNC(=O)C(C3CC3)SC)C2)=O)C1 50192,C1(CC(=O)NCc2ncccc2F)COCCN(C(c2n[nH]c3c2COC3)=O)C1 50193,c1(C(N(C)CC2(O)CN(C(CC3C(C)OCC3)=O)C2)=O)ccc(S(N)(=O)=O)cc1 50194,N1(C(COC)=O)CCN(C(c2cn(C3CCC3O)nn2)=O)CC1c1nccn1C 50195,c1(C(=O)NC(C)CC2CN(C(C3(C)COC3)=O)C2)ccnn1C1CCC1 50196,C1(C(C)C)CCCCC1C(=O)NC1CC(C)N(C(=O)CCOCC(F)F)C1 50197,C(C)(CCC(=O)NCc1ccsc1C(=O)NC1CCN(C(C)=O)C1)OCC 50198,N1(C(CC2(N(S(=O)(=O)C3CC3)C)CCC2)=O)CC(NC(=O)CO)CC(O)C1 50199,N1(C(c2nncc(N(C)C)c2)=O)CCCCC(NC(=O)C(O)c2ccsc2)C1 50200,N1(C(c2c(C)cn(C)n2)=O)C2CCCC1CC(NC(c1cn(C)n1C)=O)C2 50201,N1(C(CCc2cc(C)no2)=O)CC(=O)NCC1C(=O)NCCSC(F)F 50202,C1(CNCC2CCC(NC(=O)OC(C)(C)C)C2)CC12CCOC2 50203,N(C(=NCCC1(C)Cc2ccccc2C1)N1CCCC(O)CC1)C(C=C)C 50204,C(C(C)C(C)C(=O)N1CC(CNC(c2cccc(C)c2Cl)=O)(OC)C1)OC 50205,CCC(C)CCC(=O)NCC12CC1CN(C(=O)C=CSCc1ccco1)C2 50206,N1(C(c2c(C(C)C)ncnc2)=O)CC2CCN(C(=O)CC3CCC(=O)N3)CC2C1 50207,N1(C(c2c(CNC(c3c(C)n[nH]c3)=O)ocn2)=O)CCN2CCOCC2C1 50208,C1(CC(N2CCC(COC)(NC(=O)CCCF)C2)=O)CN2CCN1CC2 50209,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)Cc2cnccc2Cl)CC1C 50210,C1(CNC=O)(CO)CC12CCC2.c1(C(N(C(C(=O)OC)C)C)=O)cn(CCF)nc1C 50211,c1(C(N2CC(C3(NC(C4(C)CCC4)=O)CC3)C2)=O)ccc2sccc2c1 50212,C(C)(CS(=O)(=O)CCNC(=NCC)NC(C)CC(F)(F)F)OC 50213,Cc1c[nH]cc1C(N1CCC(C(N2CC(C(N)=O)C2)=O)C1)=O 50214,Cc1cnn2ccc(C(=O)NC(C)C(CO)NC(=O)Cn3nccc3C)nc12 50215,N1(C(C2(C)CC(C)=C(C)CC2)=O)CC2CCCC(NC(=O)COc3ccon3)C2C1 50216,C(N=c1[nH]cncc1Cl)C1CN(C(C(C)C)=O)C(C)C1 50217,C=C(C)CCC(=O)NC1CCC(CCNC(c2nccnc2C)=O)C1 50218,C1(CC)(CO)CCN(C(=O)NC2(CO)CC2c2ccncc2)C1 50219,n1(CC(N2C(CCCCNC(=O)Cc3ccccc3)CCC2)=O)cc(F)ccc1=O 50220,c1(CNC(C2(CN)CC2(F)F)=O)c(N)sc2cccnc12 50221,C=C(Cl)C(C)(C)C(=O)N1CCC(CNC(=O)Cn2nc(Cl)ccc2=O)C1 50222,c1(C(N2CCCCC(NC(CN(C)C3CC3)=O)CC2)=O)nc2n(c1Cl)CCCC2 50223,O=C1CC2(C1)CC1(CC(NC(C3CC4CCCCCCC34)=O)C1)C2 50224,N1(C(C=CCC)=O)CC2CCCC1C2CNC(=O)CNC(C1CCC1)=O 50225,Cc1occc1CC(=O)NC(Cn1cncn1)C(=O)NCC(O)CCC1CC1 50226,C1(CC)CCCN(C(c2cc(CNC(=O)C(c3ccnn3C)O)nn2C)=O)CC1 50227,c1(OCCC)ccccc1C(N1CCC(C)(NC(c2ccc(C(C)C)o2)=O)C1)=O 50228,C(=O)(C(C)(CO)NC(C1CCC(F)(F)C1)=O)N(CC(C(=O)NC)C)C 50229,N1(C(c2snc(C)c2N)=O)CCN(C(=O)C(F)C2CCCC2)CC12CC2 50230,N1(C(C2(COC)CCCCO2)=O)CCC2(CCC(NC(C3CCN3C)=O)C2)CC1 50231,N1(Cc2ccc(OC)cc2)CCC(F)(CN(C2CC2)Cc2ccc(F)c(F)c2)CC1 50232,c1(C(c2n(CCOC)nnn2)NCCP(C)(C)=O)ccc(Br)c(F)c1F 50233,n1(CC(=O)OC)cc(C(C2CCCO2)N(CCCOC(CC)=O)CCO)nn1 50234,N1(C(C(C)=CC=C)=O)CCOCC(C(=O)Nc2cccc(O)c2CC)C1 50235,c1(C(N(C(CNC(C2(NC(C)=O)CC2)=O)C2CC2)C)=O)cc2c(nn1)CCC2 50236,C1(C(=O)NC(COC)CO)N(C(=O)CCOC2COC2)CCCC1(C)C 50237,c1(C(N2C(CNC(C3(CCC=C)CC3)=O)CCCC2)=O)cc(Cl)c2ccccc2n1 50238,Cc1ccc(C(=O)NC2CC(C(=O)NC3(CO)CC(C)(C)C3)C2)n1C 50239,N1(C(C(NOC)=O)=O)CCC2(CCC(NC(c3c[nH]nc3C)=O)C2)CC1 50240,C1(CCNC(C2(C)CC3CCC2O3)=O)CCN(C(=O)Cc2cn[nH]c2)CC1(F)F 50241,c1(OC)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50242,C1(C(=O)NC(C(C)NC(CNC(=O)OC)=O)C)(NC(N)=O)CCCCC1 50243,CC1(C)CC(CCNc2cc(N3CCOC(C4CC4)C3)ncn2)CO1 50244,c1(C(C)NC(C(=O)Nc2cn(CC)nc2)=O)ccc(Br)cc1Cl 50245,C1(CCNC(c2c(CC)noc2C)=O)CCN(C(c2cn[nH]c2)=O)CCC1(F)F 50246,N1(C(CC(C)F)=O)CCCC(CNC(C2(F)CCCCC2)=O)CC1 50247,CC(CF)CC(=O)NC(CNC(=O)C(c1ccc(Cl)cc1)(F)F)CO 50248,c1(C(=O)NCC(C)NC(c2ncc(OC)cc2F)=O)ccc(F)c(C)c1N 50249,C1(C(=O)OCC)CCCN(C(CC2C=CCC2)C(=O)NC2(C)CC2)C1 50250,CCC(C)(C(=O)NC1CN(C(c2cccc(Br)c2)=O)C(CC)(CC)C1)OC 50251,c1(NC(N)=O)cccc(C(N2CC(NC(=O)C(O)C3CC3)C(F)C2)=O)c1 50252,c1(C(C(F)(F)F)NC(c2c(C)ocn2)=O)ccnc(Cl)c1F 50253,C(=O)(C(CC(C)C)N(C)C(C1C2CN(C(C3(CC)CCCO3)=O)CC12)=O)OCC 50254,c1(C(=O)NCC(CO)NC(c2cc(O)ncn2)=O)cc2n(c1)CCCC2 50255,c1(C(=O)NC2CCCC(NC(C3CC(C)(F)C3)=O)C2)ccc(Cl)c(F)c1N 50256,c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCN3CCCC3)CC2SC)o1 50257,CC(CS(C)(=O)=O)C(=O)NC(C)(CNC(c1cc2c(ccn2C)[nH]1)=O)CC#N 50258,C1(NCc2ccc(OCC)cc2)CC(NC(C2(C(=O)O)CC2)=O)C12CCOCC2 50259,c1(CNC(=O)NC2CN(C(=O)CCN3CCCC3)C2)cc2ccccc2o1 50260,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50261,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50262,c1(C(=O)NCC2CC(F)(CNC(c3cncs3)=O)C2)cc2cccnn2n1 50263,C1(CNC(C(CCC)NC(N)=O)=O)CCCN(C(=O)C2=NNC(=O)C2)CC1 50264,c1(OC)ccc2c(CNC(c3cnn(C(F)(F)F)c3)=O)c[nH]c2c1 50265,c1(CNC(=O)CCC2(NC(C3C(C)NC(=O)CC3)=O)CCCC2)cccc(F)c1N 50266,C1(C(=O)OC)CC(C)(NC(=O)C(n2cc(CCC3(O)CCC3)nn2)C)C1 50267,c1(CC(=O)NC(CNC(=O)Cc2csc(C(F)F)n2)CO)ocnc1C(F)(F)F 50268,C1(NC(c2cnc(C3CCC3)s2)=O)CC2CC1N(C(c1csc(Cl)c1Cl)=O)C2 50269,c1(C(N2CC=CC(O)(C(=O)O)C2)=O)cnc2[nH]ccc2n1 50270,N1(C(C2N(C(=O)C(F)C3CCCC3)CCC(=C)C2)=O)CCC(C)(C2CC2)C1 50271,N1(C(c2n(C)c([N+](=O)[O-])cc2)=O)C2CCCC1CN(C(C13CC(F)(C1)C3)=O)CC2 50272,Cc1cccc(C)c1C(=O)NCCOC1CN(C(c2ccnc(C)c2N)=O)C1 50273,C1(C(=O)NC2CC(C(C)(C)C)C2)(NC(=O)CC2(O)CCCC2)CC(F)C1 50274,C1(N(C(=O)CNC(c2ccco2)=O)C)CN(C(C2(C)CC2C(F)(F)F)=O)CC12CC2 50275,Cc1nc(-c2c[nH]c(C(=O)NCC3CCN(C(=O)C(C)n4cccc4)C3)c2)cs1 50276,N1(C(c2nc(C(C)=O)sc2)=O)CCN2CCN(C(=O)CCC3CC3C)CC2C1 50277,C1(CC(=O)NCc2c(CNC(C(CC)N(C)C)=O)n[nH]c2)CC2C=CC1C2 50278,n1(CC(=O)N(C(C)C(=O)NC(c2nn(C)cc2O)C)CCC)ccc(=O)cc1 50279,CC1CCC(C2CCCC2)CN1Cc1cn(Cc2cccnc2)nn1 50280,c1(OC)ccc(Cl)cc1NC(N1CCC(NC(=O)CN(C)C)C(O)C1)=O 50281,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 50282,c1(C(N(C2CCN(C(=O)C=Cc3cn[nH]c3)CC2)C)=O)cc(O)cc(C#N)c1 50283,COn1cnc(C)c1C(N1CC(C)(NC(c2ncncc2NC)=O)C1)=O 50284,C(=O)(CC(C)CC(C)C)NC1CC1.c12cccc(c1)NC(=O)C(=O)NCCS2 50285,C(=O)(C1CCc2c[nH]nc21)N1C(C(N(CC#C)CCO)=O)C2(C1)CCCC2 50286,N1(C(CCOC)=O)CC2CCC2(CC(=O)Nc2csnc2C)C1 50287,C(C(=O)NCCN(C(=O)C=C1CCC1)C(C)C)(C(C)C)OCC 50288,Cn1nc(-c2ccsc2)c2cc(CNC(c3ccns3)=O)cnc12 50289,C1(CNC(c2ccc(CC)[nH]2)=O)C(C)CCCN1C(C1CCCN(C)C1)=O 50290,C1(CNC(CCC2N(C)CCCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1O 50291,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50292,C(=O)(C(C(C)O)NC(=O)CC1CCCN(C)C1)N(C1CCC(C)C1)C 50293,C1(C(C(=O)NC(C)Cc2nn[nH]n2)NC(=O)COC2CCOC2)CC=CCC1 50294,Cc1noc2nc(C(=O)NC3CCCC(NC(=O)CC(C)O)C3)ccc12 50295,CC(c1ccccc1)=CC(=O)NC1CC1CNC(=O)C(C)n1ccnn1 50296,C1(NC(=O)CSC2CC2)CC2CN(C(c3cccc(-n4cccc4)c3)=O)CC12 50297,C1(CN(C)C(c2ncccc2F)=O)CN(C(C2CCCOCC2)=O)CC12CC2 50298,N1(C(=O)NC2(N3CC(C)(C)C3)CC2)CC(c2ccccc2)C(F)(F)C1 50299,c1(C2CC(F)(CNC(=O)NCC=Cc3cnc[nH]3)C2)cc(Cl)sc1Cl 50300,c1(-c2nc(C(N3CCC(C)(N(CC)CC)CC3)=O)c(C)s2)ccc(C#N)c(F)c1 50301,c1(N(CC(C)OC)C)nnc(CC(C)SC)n1CC1CCOC1 50302,c1(N2CCN(C)C(CNC(c3cn4c(n3)CCC4)=O)C2)ncnc2[nH]ccc12 50303,c1(C(=O)NCCN(C(COCC=C)=O)CC2CC2)ccccc1 50304,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50305,c1(NC(C(c2ccc(Cl)o2)N(C2CCSC2)C)=O)ccc(Nc2ccccc2)cc1 50306,CN(CCNS(=O)(=O)c1ccc(Cl)s1)N1CC(CO)OC2(CCC2)C1 50307,n1(CCOC)nc(CCCO)nc1-c1ccc(COc2ccc(Cl)cc2)cn1 50308,C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(=O)C=Cc1ccoc1)CC2 50309,N1(C(Cc2ccc(CCOC)cc2)=O)CC(O)C2(CCOCC2)C1 50310,c1(OCC)cc(NC(c2cnc(OC)c(-c3cncc(C#N)c3)c2)=O)ccc1Cl 50311,Cc1nc2cccc(C(N3CC(C(C)NC(c4cncc(N)c4)=O)C3)=O)c2[nH]1 50312,C12(CNC(C=CC)=O)CC1CN(C(c1ccn(CC(F)F)n1)=O)C2 50313,CCC(O)C(C)(C)C(=O)N(C)CC=CC(=O)NC1C2COCC12 50314,c1(NCCn2cc(C(=O)O)nn2)cccc(C(=O)NC2CC(SC)C2)c1 50315,c1(C(N(CCCO)C(C)C)=O)ccc2nc(-c3ccc(F)cc3)cn2n1 50316,CCN(NC(=O)C(O)CCn1cc(C(C)(C)CC)nn1)C(=O)NS(C)(=O)=O 50317,C1(C(=O)OCCCCc2ccc(F)cc2)(NC(=O)OC(C)(C)C)CCCC1C 50318,N1(C(c2c(Br)cc3ccccc3n2)C(=O)NC)CC2C(CO)CS(=O)(=O)C2C1 50319,CCCC(CNC(=O)Cc1nc[nH]n1)C(=O)NCCN(C)CCCC1CCC1 50320,C(=O)(CC(P(C)(C)=O)c1ccccc1)N(CC(O)CNC(C1(C)CCC1)=O)C 50321,C1(CCOC)CN(C(C2(CCN=[N+]=[N-])CC2)=O)CCN1C(=O)CCS(C)=O 50322,N1(C(=O)NCc2n[nH]c3cccnc23)CCN(S(=O)(=O)N2CCOCC2)CC1 50323,CC(C)(C)S(=O)(=O)CC(=O)NCC1CCCN1C(C1CCC(C(F)(F)F)CC1)=O 50324,C1(C(N2CCC(CC#C)C2)=O)CCCCCCN1C(=O)C(C)CC(=O)OCC 50325,CCCCCCN(C)C.C1(=O)C(=O)NCC(CNC(=O)CC2(CO)CC2)CN1 50326,C(C(C)NC(c1cccn1CC)=O)(C(C)C)NC(CCC)=O 50327,c1(OC)c(CNC(=O)C(C2CCN(C(=O)C=Cc3cnn(C)c3)C2)F)cnn1C 50328,C(c1ccccc1)=CCN1CC(C(C)NC(C2N(C(C)=O)CCC2)=O)C1 50329,C1(C(=O)NC23CC(C2)C3)CCC2(CN(C(c3ccccc3O)=O)C2)O1 50330,CCC(CC(=O)NC1(c2cn(-c3ccc(F)cc3F)nn2)CCC1)C(F)F 50331,N1(C(C(C)SC)=O)CC(O)(C(=O)NCCC2COCC2O)C1 50332,Nc1cnc(C(=O)NCCCCNC(=O)C=Cc2cnc[nH]2)c(Cl)c1 50333,C=CC(C)(O)CC(=O)NCCCC(c1ccccc1)NC(=O)CC(O)CN(C)C 50334,CC#CCC(C(=O)NCCC(O)CCO)NC(=O)C(C)OC1CCCC1 50335,c1(NC(C(C2CCN(C(c3nc(CC)sc3)=O)C2)C)=O)ccc(C)cc1CO 50336,N1(C(CCCOCC=C)=O)CCN(C(CNC(c2cc(Cl)cs2)=O)C(F)F)CC1 50337,C(=O)(CCS(=O)(=O)CC(C)C)NCC(CC=C)NC(c1cnn2c1OCCC2)=O 50338,c1(C(N2CCC(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(F)(F)C2 50339,c1(COC(C2C(=O)NC(C(F)(F)F)CC2)=O)cc2cccnc2c(F)c1 50340,Cc1c(NC(=O)C(c2ccc(O)nc2)N2CC(CO)C2(C)C)cccc1Cl 50341,N1(CCCCCOC)CCOCC(C(N2CC(C(=O)OC)C2)=O)C1.C(C)(C)(C)OC=O 50342,C(=O)(C(F)C(C)(C)O)NCC1(CNC(c2ccc(OCC#C)cc2)=O)CCCC1 50343,C=CCCCCCC(=O)N1CC2CC(NC(c3cc(C)oc3CC)=O)CC2C1 50344,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50345,c1(NC(C2(COC)CN(C(=O)CS(=O)CC)C2)=O)cnc(F)c(C)c1 50346,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50347,C(CNC(c1cccc(CS(C)(=O)=O)c1)=O)(CC(F)(F)F)NC(C(=O)NC(C)C)=O 50348,S(=O)(=O)(c1ccc(-c2ccc(N(C)CCO)cc2)s1)N(CC=C)CC 50349,c1(C(=O)NCC2CCCN(C(c3c(CC)n(C)nc3)=O)C2)c(C)cc(O)cc1C 50350,C1(NC(COCCCC)=O)CC(CNC(=O)CCc2cccnc2)C1(C)C 50351,c1(C(N2CCC(C(C(=O)N(CC#C)CCF)C)C2)=O)ccnc(Cl)c1 50352,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CCOC(C(C)C)C2)=O)C1 50353,c1(C(N2CC(C)C(NC(=O)CCCCC3CC3)C2)=O)ncc(C(N)=O)cc1Cl 50354,c1(NC2(C(C(=O)NC)C(C)(C)C)CCN(C)C2)nc2ccc(Br)cc2s1 50355,C(=O)(CCCCCSC)N1CCC(CCOC)(NC(=O)CN(C2CCCC2)C)C1 50356,C1(CCC)CCN(C(=NCCc2ccnc(F)c2)NCCNC(=O)OC)C1 50357,N1(C(Cc2c(C)ccc(C)c2)=O)CC(=O)N2CCOCC2(CNC(=O)C(C)O)C1 50358,c1(C(CC)(C)C)cccc(C(=O)NCC2CCCN2C(C2CN(C)CCO2)=O)c1 50359,C1(CCOC)(NC(c2c[nH]nc2C(C)C)=O)CCN(C(c2nnc(C)s2)=O)C1 50360,c1(CC(=O)NCC2CN(C(c3[nH]nnc3C3CC3)=O)CC2O)csc2ccccc12 50361,C1(C)(C(N2C(C(C)C)CCCC2)=O)CC12CCN(C(=O)Cc1ccccc1F)CC2 50362,c1(C(=O)NCCC(CNC(C2(CSC)CCC2)=O)O)ccc(-n2cnnn2)cc1 50363,N1(C(CNC(CCC)=O)=O)CCN(C(=O)C(C)OCC(C)C)C(CC(F)(F)F)C1 50364,CCCCCC(F)C(=O)N1CCCC1(C(N1C2CCC1CC2)=O)COC 50365,Oc1nccc(=NCCNC(c2ccccc2)Cc2ccccc2)[nH]1 50366,c1(C(C(=O)OC)(F)F)cc2cc[nH]c(=NCCc3cc(F)cc(F)c3)c2[nH]1 50367,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50368,N1(C(c2c(CN(C)C)occ2)=O)CC2(CC(NC(=O)CN3CSCC3=O)C2)C1 50369,c1(N2CCCC(CCC)C2)nc(=NCC2(CC(C)C)CN=N2)[nH]c2c1CCCC2 50370,c1(CN(CC(=O)NCC(F)CNC(=O)CCn2ccnc2)C)c(F)cccc1F 50371,CC(C)C(C)(C)C(=O)NCC=CCNC(c1ccccc1OC(C)(C)C)=O 50372,c1(C(N2CCCN(C(CSC(C)C)=O)CC2CO)=O)cnc2cc(O)ccc2c1 50373,C(=O)(C#CC1CCCCO1)NC1C(CNC(C2C(C=C(C)C)C2(C)C)=O)CCCC1 50374,c1(C(C)C)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50375,Cc1cccc(CCNC(=O)CCC2(C)CN(C(C3CC(C(C)C)C3)=O)C2)n1 50376,C(C(CO)C(C)(C)C)c1onc(-c2c(C)nccc2)n1 50377,C1(C(=O)NCCC(C)NC(C2CC3COCC3C2)=O)CCCC(F)(F)CC1 50378,C1(C#N)(C(=O)NCC2OCCN(C(Cc3nc(C(C)=O)sc3)=O)C2)CCOCC1 50379,S(=O)(=O)(c1nc(N2CCCC(F)C2)ccc1Br)NC(COC(C)C)(C)C 50380,C1(C(=O)NCCCN(C(c2cscn2)=O)C2CC2)CC2CCCCN2C1 50381,N1(C(C(CC)(F)F)=O)CCC(F)(C(=O)NCC2CCCC(C3CC3)O2)CC1 50382,C12(C(N(CCc3ccc(Cl)cc3)CC)=O)CCCC(CCC1)C2(F)F 50383,C(=O)(C(F)CC(CC)CC)NC(CC#C)(C)C(=O)NC1CC=CCC1 50384,O=C1CCC(CC(N2CCCC2CC(=O)NC2CC(N3CCCC3)C2)=O)N1 50385,c1(OC)c(F)ccc(F)c1C(=O)NC1CCCN(C(C2CCCOCC2)=O)CC1 50386,C1(C(N2CCN(CC(C)NC(C3(C)CC3(C)C)=O)CC2)=O)Cc2cscc2C1 50387,N#CC1CN(Cc2ccc(O)cc2)CC1NC(C1CCC2CC12)=O 50388,N1(C(CC2(NC(c3ncn(C)c3)=O)CC2)=O)CCC(O)C(F)C1 50389,Cc1ccccc1C(C)CC(=O)NCC(C1CCOC1)O 50390,N1(C(c2c(C(C)NC(c3ccc(CC)[nH]3)=O)noc2)=O)CC(COC)C1(C)C 50391,C1(NC(CCc2scc(C)n2)=O)CC2CC(C1)N(C(=O)CC(C)C(F)(F)F)C2 50392,c1(SCC)c(N2CCOC(c3nc[nH]n3)C2)nnc(Cl)c1C 50393,CCC(C)(C(=O)N(CC(C)C(=O)N(C)Cc1n[nH]c(C)n1)C)OC 50394,CC#CCCC(=O)NCCCCN(C(=O)COc1ccc(O)cc1)C 50395,Cc1cn(C)cc1C(=O)NCCCCNC(c1ccnnc1S)=O 50396,c1(C(=O)NCC2(C(=O)NC(C#C)CC3CCCC3)CCC2)cn(CCC)cn1 50397,CCC(C)(C(=O)N1CC(NC(=O)CCc2cnco2)C(C(F)F)C1)OC 50398,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50399,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CC(CO)C1)=O 50400,c1(OC)nc(Cl)ccc1C(c1nnnn1C)NCCOCc1ccc(Cl)cc1F 50401,c1(C2(C(=O)NC(c3ncc(Br)cn3)C)CNC2)cccc(F)c1 50402,N1(C(C=CC)=O)CC(CNC(c2cccn(C3CCSC3)c2=O)=O)CC(O)C1 50403,CC(C)(CC(N)=O)NC(C1C=CC(NC(=O)CCCC2CCCO2)C1)=O 50404,N1(C(c2ncc(F)cn2)=O)CCCC2(CCO2)C1 50405,CC(CC(=O)NCC(CO)NC(c1cnc(C(F)F)s1)=O)C1CC1 50406,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50407,N1(C(c2c(CN)ccs2)=O)CCc2cc(Cl)ccc21 50408,c1(C(=O)NCCCN(C(C2CCS(=O)(=O)N2)=O)CC)c[nH]c2ccc(Cl)cc12 50409,CCCCC(CNC(C12CCC1C2)=O)NC(c1cccc(OCC(F)(F)F)c1)=O 50410,CC1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C(=O)NC1CC=CCC1C 50411,CC1CN(C(=O)CS(C)(=O)=O)CC2(CCN(c3ccc([N+](=O)[O-])cc3Br)C2)O1 50412,N1(C(CCC2CCC(=O)N2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50413,N1(C(C2(C)CCC(=O)NC2)=O)CC2CCCC(C1)N2C(=O)C(c1cccnc1)O 50414,N1(C(C2CN(CC(C)C)C(=O)C2)=O)CCN(C(C2CSC2)=O)CC1C1CC1 50415,N1(CC(=O)N(CCC2(C)CC2)CCO)CCN(C(=O)Cc2cnoc2)CC1 50416,C(C)(CNC(C12CC(CO1)C2)=O)(CC(C)C)NC(C1(c2c(C)cccc2)CC1)=O 50417,C1(NC(C(C)C(F)(F)F)=O)CCC(C)(C)CC1CNC(c1cnc(N)c(N)c1)=O 50418,C(C(=O)NCCC1(C)CC1)(C(C)CCc1ccc(F)cc1)N(CC(C)(C)OC)C 50419,C1(O)(c2cn(CC(=C)CC)nn2)CCN(C(=O)CC2CCC(=O)N2)CC1 50420,C1(NC(c2cc(C)[nH]c2)=O)CC2CCC1N2C(=O)C(c1cccnc1)C 50421,N1(C(C(C)N(C(C)=O)C)=O)CCC(NC(C2CC(O)CN2C(N)=O)=O)C(C)C1 50422,S(=O)(=O)(c1ccc(N)c(NC(C2CC2C)=O)c1)N(CC)CC 50423,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50424,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50425,c1(C(N(CC(C)NC(c2cc(O)ccc2Cl)=O)C)=O)c[nH]cc(Cl)c1=O 50426,N1(C(C(CC)OC)=O)CC2(CNC(c3cc(OC)cc(F)c3)=O)CCC1CC2 50427,C1(SC)CN(C(=O)C(F)=CC2CC2)CC1NC(c1cc(Cl)no1)=O 50428,C1(C(=O)NCCNC(CC(C)F)=O)CC(c2cccc(Br)c2)=NO1 50429,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50430,c1(C(=O)NC2CC(C)(COC)N(C(=O)CCSC)C2)cnc(O)c2ccsc12 50431,n1(C(c2cc(C(=O)NC3CCCC3)cs2)CC)nnnc1CNCCOCC 50432,Cc1c(CNC2(C)CC2(C)C)cnn1-c1ccc(F)cc1 50433,c1(C(=O)NCCN(C(C(C)OCC)=O)CC(C)O)cc(C)c(O)c(Br)c1 50434,C1(C(C)C)N(C(=O)CN2CCNC(=O)C2)CC12CC(N)C(O)C2 50435,CC1(C)CN(C(=O)CCCC2CCCC2)CCN(C(C2CC2C(C)(F)F)=O)C1 50436,N1(Cc2ccccc2)CCC2C1CCCN2C(=O)C(CCO)NCc1cc(C)ns1 50437,C1(F)(C(=O)NCC2CC(C#N)C2)CCN(C(C2CCC2Cc2ccccc2)=O)C1 50438,CC1COC2(C1)CN(C(c1coc(CNC(C3CCC(O)CN3C)=O)c1)=O)C2 50439,C1(C)(NC(C(C)Cc2cnn(C)c2)=O)CCN(C(=O)CC2CCCO2)CC1 50440,Cc1sc(Cl)nc1C(=O)NCC1COCCN1C(=O)CCn1nc(C)nc1C 50441,N1(C(=O)COC2CCC2)CCC2(NC(c3cc(F)ccc3F)=O)CC2C1 50442,C1(NC(c2cccc(C(=O)NC)c2)=O)CN(C(=O)CC2(C)CCCO2)CCC1C 50443,C(C(C)C(F)C(=O)NCc1cccnc1O)NC(C1(CC#C)CC1)=O 50444,c1(NC(=O)C(c2cccc(C(F)(F)F)c2)N2CCC(O)CC2)cc(Br)cnc1O 50445,c1(C(N2CC(C)N(C(=O)C(C3CCOCC3)F)CC2)=O)noc2ncccc12 50446,N1(CC(=O)NCC(C)(C)NC(=O)CCCC2CCCC2)CCC(C)(C)C1 50447,N1(Cc2c(C)noc2)CCC2(NC(=O)C(=Cc3c[nH]cn3)F)CCCC12 50448,C1(C)(OC)CCN(C(C2C=CC(NC(c3cccc(Br)c3F)=O)C2)=O)CC1 50449,N1(C(CC(C)N(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50450,c1(OC)ccc(C(=O)N(CCCCN(C(=O)C(C)OC)C)C)nc1N 50451,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50452,N1(C(C)C(N)=O)CCC(C2CCN(C(=O)Cc3ccc(F)nc3)CC2)C1 50453,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50454,c1(OC)cc(C(N2CC(N3CCN(C(c4sc(C)nc4C)=O)CC3)C2)=O)ccn1 50455,c1(OC)cscc1C(=O)NCC1CCC1C(N1CCCC1C(C)(C)C)=O 50456,c1(C(N2C(C(C)(C)NC(C(CC)O)=O)CCC2)=O)cncc2cc(Cl)ccc12 50457,C(=O)(CCC(CC)CCC)N1CC(OCCNC(CC(=O)NC)=O)C1 50458,C1(CNC(Cc2cc(C)sc2C)=O)COCCN(C(c2cnn(C(F)F)c2)=O)C1 50459,c1(C(C)C(=O)NC2CCCC2NC(C2CCC2)=O)ccc2c(c1)OCO2 50460,C(=O)(C1CCCc2n[nH]cc21)NC1COCCN(C(CCS(C)(=O)=O)=O)C1 50461,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50462,C(=O)(C1=C(Cl)CCC1)N1C(CNC(c2ncccc2Br)=O)CCCC1 50463,c1(C(=O)NCCCC2(NC(C(CC)NC(N)=O)=O)CC2)nn2ccccc2c1C 50464,CC(C)(CC(=O)N1CCC(NC(c2conc2C2CCC2)=O)C1)c1cccs1 50465,C1(NC(c2ccnnc2Cl)=O)CCSC12CN(C(=O)CCC1CCOC1)C2 50466,c12cc(ccc1C)NC(=O)NC2.C1(N2CCOCC2)(CC)CCCOC1 50467,Cc1c([N+](=O)[O-])c(C(=O)NCC(C)(CO)NC(=O)CCC(N)=O)nn1C 50468,c1(COC(C)=O)cccc(-c2cn(C(C)C(=O)N(C)Cc3ccsc3)nn2)c1 50469,CC(O)CCN=c1[nH]c(=NCc2ccc(C)n2C)c2c(F)cccc2[nH]1 50470,N1(C(C2C(CCC)C2)=O)CCOCC(F)(CNC(C2C3CC4C(C3=O)C24)=O)C1 50471,CC(C)CCCCC(=O)NCC1CN(C(=O)CC2OCCC2(C)C)CC1C 50472,N1(C(C(CC)=CC)=O)CCC(C(C)C(=O)N(C2CCC(F)(F)C2)C)CC1 50473,N1(C(CC(C)NC(=O)Cn2cccn2)=O)CCC12CCN(C)C2 50474,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50475,C(=O)(CCCCC(N)=O)NCC1(C)C(C)CN(C(CCOCC#C)=O)C1 50476,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50477,N1(C(CCC(C)OC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C(C2CC2)C1 50478,c1(C(=O)NCC(C)NC(C(c2cnn(C)c2)OC)=O)cc2cccc(C)c2nn1 50479,C(C(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2cn(C)cn2)=O)CC1)OC 50480,C(=O)(C1=CCC(F)(F)CC1)N1C2(CN(C(c3ccc(C=C)cc3)=O)CC2CC)CC1 50481,C1(CO)CC2(CCC2)CO1.C(C1(C)C(=O)NCc2c(scc2)C(=O)N1)OC 50482,C(=O)(CCCC(C)(C)C)N1CCC(C)C1C(=O)NOCC(=O)OC(C)(C)C 50483,C1(CC)CN(C(C2CC2F)=O)CCC1NC(c1ccnn1C(CC)CC)=O 50484,N1(CC(=O)NCC(C)(CO)NC(C2CC2C(F)(F)F)=O)CCS(=O)CC1 50485,CC(C)C(O)C(C)C(=O)N1CC(C)(NC(c2ccc(F)cc2)=O)C1 50486,CC1CN(C(c2cc(N(C)C)ccn2)=O)CCC1CNC(=O)CCCC1(C)N=N1 50487,n1(CCN(C(c2cnc(Cl)[nH]2)=O)C2CC2)nccc1-c1cn(CCCOC)nn1 50488,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50489,c1(-n2cc(C(CC(N)=O)NC(c3cc(C)oc3)=O)nn2)ccc(F)cc1Cl 50490,C1(CC=C)(NC(=O)CC(F)(F)F)CCN(C(c2ccc(COC)o2)=O)C1 50491,C=C1CCN(C(=O)CSC)C(C(=O)OC(=O)NC(C)CCC)C1 50492,N1(C(C(n2cc(C3CCC3)nn2)C)=O)CCCC2(C1)C(O)CC2O 50493,N1(C(c2c(CC)ncc(Br)c2)=O)CC2CCC(C1)N(C(=O)C#CC(C)C)C2 50494,Cc1ccc(Cl)c(N)c1C(=O)NC1CC(C)N(C(=O)CN(C)C(=O)C2CC2)C1 50495,N1(C(CNC(C)=O)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50496,C1(C(N2CCC(CF)(NC(C3(C4CCCCO4)CC3)=O)C2)C)CCC(C)(C)CC1 50497,N1(C(CCC=CC(C)C)=O)CC(CNC(C2CCC(CO)CC2)=O)C(C)C1 50498,CC(C(=O)N(C1C2CN(C(=O)Cc3cccc(C(C)(C)C)c3)CC12)C)C(C)(F)F 50499,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50500,CCC(C)C(O)CC(=O)NC1C2CC(NC(C3(C#N)CC3)=O)CC12 50501,C1(CC)CN(C(=O)CN2CCC(O)CC2)CCN1C(=O)CNS(N)(=O)=O 50502,c1(C(=O)NC2C(C)(CNC(C(CC(C)C)C)=O)CCC2)cnc2[nH]c(O)nc2c1 50503,c1(OC)ncccc1C(N1CCCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50504,CCC(CC)C(=O)NCC1CC(F)(CNC(=O)C(c2cccnc2)C)C1 50505,C(CC(=O)N1CC(CSC)C2(CC2)C1)(C(F)(F)F)NC(C1C(CCC)C1)=O 50506,N1(C(c2c(C)c[nH]c2)=O)CC2C(CNC(c3ccnn3C3CCOCC3)=O)C2C1 50507,c1(C(=O)NCC(CO)NC(=O)CCOc2cccc(Cl)c2)cc2ccncc2[nH]1 50508,CCCCC(O)CC(=O)N1CC(C(=O)NC23CCC(CC2O)C3)C(C)C1 50509,CCCC(CCCNC(c1cnc(CC(C)C)[nH]1)=O)NC(C1CCC2CC12)=O 50510,Cc1ccc(C(N2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)=O)c(O)c1 50511,C1(CNC(C(C)NS(=O)(=O)C2CC2)=O)CC(=O)N(C2CCN(C)CC2)C1 50512,C1(NC(C(CC)OC2CCCC2)=O)CCN(C(c2cc(OC)cs2)=O)C(C)C1 50513,c1(C(N2CCC(N(C(C3CN(CC)C(=O)C3)=O)CC)C2)=O)cc(N)c(O)c(F)c1 50514,CC1CCC(CO)CN1C(C1CC(NC(c2cnn(C)n2)=O)C1)=O 50515,C(=O)(C(O)CCCNC(c1ccccc1)=O)N(CC)Cc1ccsc1 50516,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50517,c1(C(=O)NCC(C(C)C)NC(C2(OC)CC=CC2)=O)ccc(C(C)(F)F)nc1 50518,C=CCC(C(=O)NCCCN(C(C1CCC(C)(C)O1)=O)C1CC1)NC(C)=O 50519,C1(C(=O)NC(C)CCNC(=O)Cc2ccsc2Cl)CCC(C)(C)OC1 50520,CCCC(CCC)C(=O)NCCN(C(=O)C(C)C(O)C(C)C)CCC 50521,Cc1c(C(=O)NC2(C#N)CCN(C(c3ccon3)=O)C2)cncc1Br 50522,N1(C(C(C(=O)NC)(C)C)=O)CC2CC(NC(C3(n4nccn4)CC3)=O)CC2C1 50523,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50524,N1(C(CCc2cc(C)on2)=O)CC(N(C(=O)Cc2nn(C)cc2Cl)C)C(F)C1 50525,C(=O)(C(CCF)NC(=O)CC#N)N(CC(O)CO)C 50526,N1(C(CCOCC)=O)CC(CO)C2(C1)CN(c1cc(-c3ccccc3)ncn1)C2 50527,N1(C(CCCSC)=O)CC(NC(=O)C(C)(C)c2cccnc2)CC1C 50528,C1(C(N2CCC(C)(CC(=O)OC)C2)=O)CCCCCN1C.C12CCCC1NC2=O 50529,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(c1csnn1)C)C(C)C 50530,Cc1cc(Cl)nc(Cl)c1NC(c1cc(NS(=O)(=O)CCCCCl)cn1C)=O 50531,C1(C(N2CC(NC(CSc3ccc(C)cc3C)=O)C(C)C2)=O)CC2CCC(C1)C2O 50532,Cc1cc(C)c(C(N2CC=C(CNC(=O)C=Cc3cccnc3)CC2)=O)cc1N 50533,N1(C(c2cn(CCOC)nn2)=O)CCN(C(=O)CC23CCC2C3)CC1CO.C1CC1 50534,C(=O)(CC1CCCc2ccccc21)N(CCNC(C(CC#C)C)=O)C1CC1 50535,c1(CNC(C(c2ccccc2)C)=O)cc2n(n1)CCN(C(C1(C)CC1(F)Cl)=O)C2 50536,CC(C)CC(COc1ccc(Cl)cc1Cl)N=c1nc2c(ncn2C)c(N(C)C)[nH]1 50537,c1(C(=O)NC(CCNC(c2n(CCC)ncc2)=O)(C)C)ncccc1Cl 50538,c1(CSCC)nc(C(=O)NC2CC(C)N(C(=O)CCc3cn[nH]c3)C2)cc(=N)[nH]1 50539,CS(=O)(=O)CCC(=O)NCCCC1CCCN1C(=O)CCc1cncc(F)c1 50540,N1(C(C(C)SCCCC)=O)CC(NC(C2CN(C(=O)NCC)C2)=O)C2(CCC2)C1 50541,c1(CC#N)ccc(C(=O)NC2CCC(NC(c3ccc(CO)nc3)=O)CC2)cc1 50542,C1(C(N(CCN(C)C(c2ccn(C(C)(C)C)c2)=O)C)=O)CCc2nncn2C1 50543,c1(OC)ccc(C2(Cc3nc(-c4csnn4)n(CC4CCCC4)n3)CC2)cc1 50544,CC1(C)CN(C(=O)CCCCC2CCCCC2)CC1NC(C1CC1CF)=O 50545,C#CCCC(=O)N(C(C)C(=O)NC1CCOC1=O)CCC 50546,Cc1ccc(N(C)C(C2CCCC2CNC(c2ccc(CO)o2)=O)=O)c(C)n1 50547,C1(C(N(C2CCCCC2)CC#C)=O)(NC(=O)CN(C2CC2)C)CCCC1 50548,C12(CNC(CSCC#C)=O)CC1CN(C(C1C3CCCOC13)=O)C2 50549,C(CCC(C)C(=O)N(CCCCC(=O)N(C)Cc1ocnc1C)C)OC 50550,Cc1c(Cl)sc(Cl)c1C(N1CC(NC(c2nnn(C)c2C)=O)C(F)C1)=O 50551,Cc1cc(C(=O)N(CC(=O)NCC2CC(O)C23CCC3)CC2CC2)cnc1O 50552,N1(C(CCC(C)(C)C#N)=O)CCOC2(CCN(C(=O)C(C)(C)O)C2)C1 50553,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50554,N1(C(c2cn(CC)nn2)=O)CC(C)(C)CC1CNC(=O)C(C1CCCCCC1)F 50555,C1(N(C(C(n2cc(C)nc2)(C)C)=O)C)CN(C(=O)CN2CCCC2=O)CC1F 50556,C1(CNC(c2ccc(C(C)C)s2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50557,C1(C2CCCO2)(C(=O)NCC2CC(C)N(C(=O)Cc3ccnn3C)C2)CCCO1 50558,C1(NC(Cc2c(C)ncs2)=O)CCN(C(=O)CNS(N)(=O)=O)CC1C 50559,C(=O)(CC(=O)NCCC1(C(=O)NCCC(O)CO)CCCC1)N(C)C 50560,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)OC(C)(C)C 50561,Cc1cnc(C(=O)NC(CC2CC2)C(=O)NC2CCCCC2C#N)cc1C 50562,N1(C(CCC(C)(C)NC(=O)C=Cc2ccccn2)=O)Cc2ccccc2C1 50563,C1(CNC(CN(C)C(N)=O)=O)CC(F)(F)CN1C(c1cccnn1)=O 50564,c1(C(N2CC3C(N(C)C(c4cnns4)=O)C3C2)=O)ccc2c(c1)NCCC2=O 50565,C1(NC(c2c(C(=O)OC)nn(C)n2)=O)CN(C(=O)C=CCO)CCC1C(F)(F)F 50566,C(=O)(CCCCCC(C)O)NC1C=CCN(C(C(CC(C)C)O)=O)C1 50567,C1(C(N(C(=O)NC(CC=C)C)C)C)CC(F)(F)C1 50568,C1(C#N)(C(=O)NC2(C)CN(C(CN(CC(=O)NC(C)C)C)=O)C2)CCCOC1 50569,CN1CC(C(N2CCC(F)(C(=O)NCCC(F)=C(F)F)C2)=O)CC1=O 50570,C1(NC(c2nc(C)n(C)c2)=O)CCCC(C(=O)N(CC(Cl)Cl)C)CC1 50571,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1NC(=O)CCC12CCC(CC1)C2 50572,c1(CNC2(C(=O)Nc3ccncc3)CC2)ccc(F)cc1C(F)(F)F 50573,CCC(CC)CC(=O)NC1CN(C(=O)Cc2[nH]cnc2C)CC12CC2 50574,c1(NC(c2ccc(C(C)(C)C)s2)=O)cnc(O)c2ccsc12 50575,C1(C(N(C2CCOC2)CC#C)=O)CCC(NC(=O)C(C)=O)CC1 50576,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1C 50577,C1(ONC(CNC(CC(C2CCC2)OC)=O)=O)CCCC(CC(=O)N(C)C2CC2)C1 50578,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50579,C(=O)(C(C#N)CCC)N(C(CC=C)C(=O)NC12CCC(CC1)CC2)C 50580,CC(CCNC(=O)C(C)(C)n1cc(Br)cn1)CCNC(C1CCC1)=O 50581,N1(C(c2ccc(CSCC)o2)=O)CC2=C(C1)CN(C(C1CC(CC(F)F)C1)=O)C2 50582,C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)CN1CCCC1=O 50583,C(C)(CN=c1ccn2ncc(S(=O)(=O)N3CCC4(CCCO4)CC3)c2[nH]1)OC 50584,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50585,C1(NC(COCCC)=O)CC2(N(C)C(C3CCN3CC)=O)COC1C2 50586,C(C)(CO)(C(=O)NCCC(N)=O)NC(C(C)OCC=C)=O 50587,c1(NC(c2n(CCOC)nnn2)c2cc(COC)no2)ncc(F)cc1C 50588,CCC1=NOC(CC(N2CCCC2C2(C(=O)NCC3CCC3CC)CC2)=O)C1 50589,c1(C(=O)NCCNC(=O)C(O)(C2CC2)C2CC2)cc2sccc2s1 50590,C1(OC)CC(NC(=O)CC=C(Cl)Cl)C12CCN(C(=O)C1=CC(C)(C)C1)CC2 50591,c1(OC)cc(C(=O)Nc2ncc(C3CCOC3)s2)ccc1N 50592,CC1(NC(=O)CC2CC(F)C2)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1 50593,CC1CC(CNC(=O)CCCc2cnn[nH]2)CCN1C(C1CCCO1)=O 50594,c1(C(=O)NC(C2CCN(C(=O)C=Cc3cnc[nH]3)C2)C)coc2c1CSC2 50595,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50596,N1(C(C(COC)N(C)C)=O)CCC(CC(=O)N(CCC(C)C)C2CC2)CC1 50597,C(=O)(CCC(F)(F)F)NCCN(C(C1C(C=C)OCC1)=O)C(C)C 50598,N1(C(C(C2CC2)SC)=O)CCCCC(NC(=O)CC(C)N2CCCC2=O)C1 50599,C1(N(C(CCc2ccc(C)s2)=O)CC(C)C)CCN(C(C2CN(C)C2)=O)CC1 50600,Cc1c(O)ccc(CNC2CCC(C(=O)Nc3coc(C#N)c3)C2)c1O 50601,O=C(CC(C(F)(F)F)NC(=O)C(=O)NCc1ccccc1)NC1(C2CCC2)CC1 50602,N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CCCN(C)C(C)C)C(C)C1C 50603,C(=O)(C(C(C)CC)NC(=O)Cc1ccc(COC)cc1)Nc1c(CCC)[nH]cc1 50604,c1(CNC(=O)C)c(C(=O)NCC(N(C)C)C2CC2)cccc1F.C1(SC)CCCO1 50605,CN1CCC(C(=O)NCc2ccc(CNC(=O)C3=CCCC3)cc2)S1(=O)=O 50606,Cc1cnc(NCC2CCCCC2NC(c2ccncn2)=O)nc1O 50607,C1(OC(c2ccc(F)cc2Cl)=O)CC2(OC(F)(F)F)COC1C2 50608,N1(C(COCc2cccc(C)c2)=O)CCC(NC(=O)CCOC2CC2)C(O)C1 50609,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)CC1 50610,CC(C)C(C)C(CNC(=O)CN(C)C)NC(=O)CC(C)(C)c1cccs1 50611,c1(C(N(CCN(C(C(CCCC)CC)=O)C)C)=O)cccc([N+](=O)[O-])c1OC 50612,CC(C)C(C(=O)NC1CCN(c2ccnc(Cl)n2)CC1)c1cccnc1 50613,C1(NC(c2ccc(N(C)C)nn2)=O)CC2CN(C(=O)C3=CCCOC3)CC12 50614,C1(C(N(CC(C)NC(C2CC(Cl)(Cl)C2)=O)C)=O)CCCCC(=O)N1 50615,C12(C(=O)OCC)CC(c3nnc(-c4ccco4)o3)(OC(C)C(=O)OC)CC1C2 50616,C1(C2CCOCC2)(C(=O)NC2C(NC(C(C(C)C)NC(COC)=O)=O)CCC2)CC1 50617,C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(=O)C2=CCCSC2)C(CO)C1 50618,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50619,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50620,c1(CC)oc(C)cc1C(N1CCC(CCNC(c2cnco2)=O)C1)=O 50621,CS(=O)(=O)C(CNC(=O)Cc1cccc(Cl)c1F)CNC(c1cc(C#N)c[nH]1)=O 50622,c1(OCCOC)cccc(N(C)C(c2sccc2C(=O)OC)=O)c1.C1(C)C(=O)N1 50623,N1(CC)CCC(Nc2[nH]nc(C(F)(F)F)c2Br)CC1 50624,C(C(=O)N1CCCN1)OC(C1CC2CC1C1CC21)=O 50625,CC1CCN(C(=O)CCc2cncnc2)CCN1C(c1cccc(N(C)C)n1)=O 50626,C1(C(=O)NC(C)C(=O)NCC2COCCO2)CCCN1C(N)=O 50627,N1(C(c2cncc(CNC(CNC(C)=O)=O)c2)=O)CC2CCC(O)C(O)C12 50628,C(C(C)(CC(C)C)NC(c1ccc(C)c(O)n1)=O)NC(c1c(CC)cncc1)=O 50629,C1(C(N2CCC(C(=O)OCC)CC2)=O)CCN(C(=O)C#CC2CCOCC2)O1 50630,C1(CNC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCC2)C1NC(C1CCCC1)=O 50631,CC(C)CC(CN(C)C)N=c1[nH]c2c(c(=NCCc3cc(C4CC4)no3)[nH]1)COC2 50632,N1(C(c2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C=CCO)C(C)C1 50633,c1(C(=O)NC2(C3N(C(COCC#C)=O)CCC3)CC2)ccc(OC)cc1F 50634,C(=O)(C1COc2ccc(Cl)cc21)N1CCCC(CN(C)C(C2CCCN2C)=O)C1 50635,c1(CCNC(=O)NC(CC)CSC)cccc(Br)c1 50636,C(=O)(C(F)(F)CCOCc1cc(O)nc(C)n1)NC 50637,CC(C)C(F)C(=O)NCCC1CCC(NC(=O)CC2CC(=O)C2)C1 50638,N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC(O)C1 50639,C1(NC(C(c2cccnc2)N(C)C)=O)CCCC(NC(c2c[nH]cc2Br)=O)C1 50640,C1(NC(C=C(COC)C)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1N=[N+]=[N-] 50641,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 50642,c1(C(=O)NC(C2CCN(C(C34CC(C3)C4)=O)C2)C)cc(Cl)ccc1Cl 50643,C=Cc1ccc(C(N2CCCC(C)(CNC(=O)CSc3nncs3)C2)=O)cc1 50644,c1(CC(=O)NC23CCN(C(=O)CN4CCSCC4)CC2C3)ccc(Cl)cc1Cl 50645,N1(Cc2cc(OC(C)C)ncc2)CC2(CCN(S(=O)(=O)c3cnc(Cl)nc3)C2)C1 50646,c1(NC(=O)C(c2cc(Br)no2)N2CCNCC2)ccc(F)cc1 50647,c1(CNC(CC(=O)NC)=O)nn(C)c2c1CN(C(=O)C(c1cncn1C)=O)CC2 50648,CCC(C)C(C)C(=O)NCc1ccc(N2CCC(NC(=O)COC(=O)OC)C2)cc1 50649,c1(C(N(CCCN(C(c2scc(OC)c2OC)=O)C)C)=O)cnc2c[nH]nc2c1 50650,Cc1ccc(-c2cn(C3CCN(C(=O)CCCN(C)C)CC3)nn2)cc1N 50651,N(C1CC2(CN(C(=O)CC3CC4(CC4)C3)C2)n2ccnc21)C(C1ON=C(C)C1)=O 50652,C1(C(=O)NOC(c2cccc(F)c2)C)(CNC(C2CCC(C)O2)=O)CCCCC1 50653,c1(C(N2CCN(C(=O)Cc3nc[nH]n3)C(CO)C2)=O)nc(Br)c2n1CCCC2 50654,C1(C(=O)NC2CN(C(CC3CCN(C)C3=O)=O)CC2(C)C)CC2(CCCC2)CO1 50655,C1(CC(=O)NCCN(C(C=CC(=O)OCC)=O)CC)CCCCCC1.C1(N)CC1 50656,c1(C(N2C(C)(C)CC(NC(=O)C3=CSCCO3)C2)=O)cc(N)cc([N+](=O)[O-])c1 50657,c1(C(=O)NC(C2CCN(C(C3CC4CC4C3)=O)CC2)C)cc(C#N)c(F)cc1F 50658,N1(C(C(=O)NC(C2CCCOC2)C)=O)CN(C)CC1CO 50659,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 50660,c1(C(N(CC(CC)NC(=O)C(=O)NCC(F)(F)F)CC)=O)cc2c(s1)CCC(C)C2 50661,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N1CCOC2CC12 50662,N1(C(c2c(CC)csc2)=O)C(C(=O)NC2CCN(C3CC3)C2)CCC12CC2 50663,C1(NC(C2(N(C(C)C)CCO)CC2)=O)CN(C(=O)C=C(Cl)Cl)CC1(F)Cl 50664,c1(NC(C2C(CNC(=O)C=CCF)C2)=O)ccc(Cl)cc1O 50665,CC1CN(C(C(=O)NCC2CCCO2)C(C)CC2CCCCC2)CC(C)(C)C1 50666,c1(OC)ccccc1NC(=O)C(C)N(C1CCC1)C(c1n[nH]cc1C1CC1)=O 50667,C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 50668,N#CC1(C(=O)OCCc2cn[nH]c2)CC12CCCCC2 50669,N1(C(COC(C2(C)CC(=C)C2)=O)=O)CCN(c2ccc(-c3ccnnc3O)s2)CC1 50670,c1(C(=O)NCC2C(NC(CCCCSC)=O)C2)ncc(Cl)cc1Cl 50671,N1(C(c2ncn(CC)c2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CO 50672,N1(C(c2n(C)cnc2)=O)CCCC2(CCC(NC(c3coc(Cl)n3)=O)C2)C1 50673,C=CCC(C(=O)NCc1c(C(N2CC(C)C(C)C2C)=O)cnn1C)C(C)C 50674,CC1CN(C(=O)C(=O)N(C)C)CCC1CNC(=O)C(c1cccnc1)O 50675,C1(CC#C)CN(C(=O)C(CC2CCCC2)OC)CCO1.C12(CCOCC1)C(=O)N2 50676,C(CCNC(=O)C(C)n1ccnn1)(C(=O)NCCNS(C)(=O)=O)OC 50677,CCCS(=O)(=O)CCNC(=O)NC(Cc1ccccc1Br)CCO 50678,c1(OC(C)C)ccc(C(N2CC(NC(C3CCCO3)=O)C(F)C2)=O)cc1I 50679,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 50680,c1(C(N2CC3C(CNC(C(CC=C)CC=C)=O)(C3)C2)=O)ncccc1S(C)(=O)=O 50681,C(=O)(C(C)S(=O)(=O)N(C)C)N1CCC(C(C)NC(CCC(C)SC)=O)CC1 50682,C=C1CC(CC(=O)NC(C(=O)NC(COC)COCC)c2cccs2)C1 50683,CCCS(=N)(=O)NC(Cc1ccccc1)C(=O)N(C)C 50684,C=CC(CC)CC(=O)N(CC(=O)NC12CCN(CC1)C2)CCOC 50685,C=C(C)CCCC(=O)N1CC=CC(NC(c2cnc(Cc3cccc(C)c3)s2)=O)C1 50686,C1(C(N2CC(NC(CSCC(=O)OC)=O)C(O)CC2)=O)CC2(C1)CC1(CCC1)C2 50687,CC1(C)CN(C(=O)Cc2cn[nH]c2)CC(C)(C)C1NC(C1CC2(CCC2)CC1)=O 50688,c1(C(N(CC(C(=O)OC)c2nn[nH]n2)CCC(=O)N)=O)[nH]c(C)cc1C.CC 50689,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCNC2=O)C(CC(F)(F)F)C1 50690,C(C(COC)C(=O)NC1CC(NC(=O)CC2CCCC2(F)F)C1(C)C)OC 50691,C(C(=O)NCCCCC(C)NC(c1c(F)cnn1C(C)C)=O)(C(C)C)NC(C)=O 50692,Cc1cc(C(=O)NCC(C)NC(=O)C(N2CCCC2)C2CC2)c(N)c(C)c1 50693,CC1CC(NC(=O)CCc2cnn[nH]2)CN1c1nnco1 50694,c1(CC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccsn2)CC)cc1 50695,C1(O)(CC(=O)NC2C(C(=O)NCC(C(=O)OC)O)CCC2)CCCCC1 50696,CC1(C)C(C(N2CCCC2c2nccs2)=O)CC1O 50697,C=CC(CC(=O)N(c1ccccn1)CCNC(=O)COCCC)c1ccccc1 50698,Cc1ccnn1C(C)C(=O)N(C1CCCCC1)CCNC1CC(n2cnnc2)C1 50699,c1cn2c(n1)CCC(CNc1ccc(-c3ccc(C4CCCC4)cc3)o1)C2 50700,N1(C(c2cn(C3CCC3)nn2)=O)CCN(C(=O)CN2CCCS2(=O)=O)C2CCC12 50701,C(CC)(C(=O)NC(C1CN(C(=O)CC2CC2C(F)(F)F)C1)C)=CC 50702,N1(C(C2(CC(C)=O)CCOCC2)=O)CCN(C(=O)C=CC(C)C)C(C)C1 50703,c1(C(C)C)cccc2c1CCCC2N(C)C(=O)C(=O)Nc1ccn2ncc(Br)c2c1 50704,c1(OCC)ncc(C(C2CNC(=O)C3C(C3C)N2)=O)cc1Cl.C1CC1 50705,c1(C(N2C(C)CC(NC(c3ccc(=O)oc3)=O)CC2)=O)ccccc1[N+](=O)[O-] 50706,c1(C(=O)NCCC2CCN(C(c3c(C)coc3)=O)C(C)C2)cn2ccccc2n1 50707,c1(NC(c2ccccc2)CCN2CC(F)C2)ccccc1Br 50708,C1(C(=O)NCC2(CNC(C3(C(=O)NC)CC3)=O)CCCC2)CCCCN1C 50709,c1(-c2n(Cc3ccc(OC)cc3)c(N3CC=C(C)CC3)nn2)c(F)cccc1Cl 50710,N1(C(c2c(CC)nco2)=O)CCN(C(c2c(C)cc(C)nc2S)=O)CCC1C 50711,CCCCCCCN(C(=O)CN(c1ccccc1)C)CC1CC(C)(C)CO1 50712,N1(C(C(C)(C)c2cncnc2)=O)CCC(CC(=O)NCCOC2CCOC2)CC1 50713,C(Nn1cccn1)c1cn(C2CC(C(=O)O)C2)nn1 50714,c1(CCN2C(CC(=O)N(c3ncn(C)n3)C)CC(F)C2)c(F)cccc1F 50715,C1(C(=O)NCC2(O)CN(C(c3cnco3)=O)C2)(CC)CNC(=O)C1 50716,c1(C(=O)NCCC2CN(C(c3nc(C)nn3C)=O)C2)cnn2ccn(C)c12 50717,Cc1cccc(CC(=O)NCCCCNC(=O)C(N2CCC(C)C2)=O)c1F 50718,C#CC(N(C)N(C)Cc1ccc(-c2ccc(F)cc2)cc1)C1CC1 50719,Cn1cc(S(N)(=O)=O)c(C(=O)NC2CC(C)(NC(=O)CC3CCC(=O)N3)C2)n1 50720,CC(C)(C)C(CO)C(=O)NCC(CC1CC1)C(=O)NCCCn1cc(CO)nn1 50721,CCCC(C)(CC)C(=O)NCC(C1CC1)N.c1(C(=O)NC)cnc(OC)c(Cl)c1 50722,N1(CCC)C2CCC1CN(C(=O)C(C)Cc1cncc(-c3nn[nH]n3)c1)CC2 50723,Cc1csc(C(=O)NCCC(O)CNC(C2(O)CC(F)(F)C2)=O)c1C 50724,N1(C(C(CCCOC)(F)F)=O)CC(=O)NCC1C 50725,N1(C(C=CSC)=O)CCN(C(C2(CO)COC2)=O)CC1c1ccc(F)cc1 50726,C1(C(N2CCN(CCN(C(C(CC)=CC)=O)C)CC2)=O)CCC(C)(C)CC1 50727,c1(OCC)ccc2c(c1)CCN(c1nc(NC3CCOC3C)c3ccsc3n1)C2 50728,C=CCC(C)(O)C(=O)N1CCCC(CCNC(=O)CCn2cc(C)cn2)C1 50729,CCCC(CCC)C(=O)NC(CCN(C)C)C(N1CCC(C)(C)C1C)=O 50730,c1(-c2ccc(CN3CCC(C(=O)OC)(CC)C3)cc2)c(OC)cccc1Cl 50731,c1(CC)c(C(=O)NC(CNC(c2ccsc2C(F)F)=O)CO)[nH]c(C)c1C(N)=O 50732,C(C)(C)(CCCF)NC1CN(C(CNC(C(C2CCOC2)OCC)=O)=O)C1 50733,C1(CC)CC(C(=O)N(C2CCCC2C)C)CCN1C(c1nn(C)cc1Cl)=O 50734,N1(C(C2(C)CC(=C)C2)=O)CCC(C)(NC(c2ccn(C3CCCCC3)n2)=O)C1 50735,C1(OC)CN(C)CC1NC(=O)C(C1(C)CC1)NC(C1CC1(C)C(F)F)=O 50736,c1(C(C(=O)NCCOCC)N(C2CCCO2)CCOC)ccc(F)c(Br)n1 50737,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 50738,CC1(C)CCCC(C(=O)NCCC(O)CNC(C2C3CCCCC23)=O)C1 50739,C1(C(N2CC(O)(CN3CCCC3)C2)=O)(CC)CCCCC1.N12CCCC1CNC2=O 50740,C(=O)(C(CC)C(C)C)N1CC(C=C)(CC(=O)NC(CO)CCSC)C1 50741,N1(C(C2CCN(CC)C2)=O)CCC(C(C)CNC(=O)C(C)(C)SC)CC1 50742,c1(CNc2ccc(C3(N)CC3)c(F)c2)c2c(cc([N+](=O)[O-])c1[N+](=O)[O-])OCCO2 50743,N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)CSc2nc[nH]n2)C(COC)C1 50744,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 50745,Cc1nn(C)c2[nH]c(=NCCC3(C)CC3)cc(NCCc3nc(C4CC4)cs3)c12 50746,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 50747,CN1CCC(CCNC(=O)CC2C=CC(NC(c3cncn3C)=O)C2)C1 50748,Cc1cc(CC(N2CC(NC(=O)C=Cc3cc[nH]c3)C(C(F)F)C2)=O)ccn1 50749,C12(C(=O)NCCC(C)NC(=O)CC3CCC4CC4C3)CCC(N=[N+]=[N-])(CC1)C2 50750,Cn1nnc2cc(C(N3CCCC(CCNC(=O)CC4CC4(C)C)C3)=O)ccc12 50751,C1(NC(c2onc(COC)n2)=O)C2CCN(C(c3ccnnc3)=O)C12 50752,c1(CC)ccc(C(=O)NC2CCC(C(=O)NC3(CC)CCC(F)C3)C2)cn1 50753,C1(C(N2CCC(CCNC(c3ccc(C)s3)=O)C2)=O)C(Cl)(Cl)C12CC2 50754,N1(C(C=COCC)=O)CC(NC(=O)CCC2CCCCN2C)CC(C)(C)C1 50755,C(=O)(CCCCCCC(=O)OC)NC1CN(C(CCC(=C)C)=O)CC(F)C1 50756,Cc1ncc(C(=O)NCC(C)CNC(=O)CC(C)n2ccnc2)c(Br)c1Cl 50757,Cc1cccc2cc(NC(c3nnnn3CC3CC3)c3csnn3)cnc12 50758,C1(C(=O)NC2CC(NC(c3ccc(NC4CC4)nc3)=O)C2)CCC(F)(F)C1O 50759,C(CN=C(NCSCC(C)O)NCc1ccsc1)N1CC(C(=O)NC2CCC2)C1 50760,C1(NC(Cc2c(C)ccc(F)c2)=O)CCCC12CN(C(C1NC(=O)C3CC13)=O)C2 50761,CC(CC(=O)N1CCC(C2CCCN2C(=O)COC2CCC2)CC1)C(C)(C)C 50762,c1(C(N2CC(OC)(CNC(=O)Cc3nocc3C)C2)=O)n[nH]c(C(C)C)c1Br 50763,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 50764,CCCC(CCC)C(=O)NC(C)CN(C)C(c1onc(OC)c1Br)=O 50765,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 50766,c1(OC)ccncc1CC(=O)NC1CCN(C(=O)CCc2cc(Cl)cs2)C1 50767,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 50768,C(CN=c1ccc(C#N)c[nH]1)NC1(CCC)N(C(=O)OC(C)(C)C)CCC1 50769,Cc1ccc(C(=O)NC2CCCCC2NC(=O)COCCOCCOC)c(Cl)c1 50770,CC1CN(C(=O)CC2C3CCCC3N2C(=O)C=CC2CCC2)CCC1C 50771,C1(OC)CCC(C(=O)NC(C)CNC(c2sccc2C(C)(C)C)=O)CC1 50772,C(C)(C)(C(=O)CN(CCCNC(C1CC(F)C1)=O)C(=O)C1CC1)OC(C)C 50773,C1(C(N2CC(CC(=O)NCc3n(C)nc(CO)n3)C2)=O)C2CC3C(C2=O)C13 50774,CC1OCCC1C(=O)NC1(C(=O)N(C)C)CN(C(=O)C(C)OC2CCCCC2)C1 50775,N1(C(c2c(Cl)cnc(C(C)C)n2)=O)CC2CCC1CN2C(c1cc[nH]n1)=O 50776,CC1CN(C(c2nc(C(F)(F)F)cn2C)=O)C(C(=O)O)CC1C 50777,c1(CC(=O)NCCN(C)C(C2CC2(C)C(F)F)=O)cnn(C)c1 50778,C(=O)(C1CCc2c[nH]nc21)N1CCC(n2cc(C(C)(C)N(C)C)nn2)CC1 50779,C1(CC(=O)N(C2(N)C3CNCC23)c2ccc(CCN)cc2)NC2CCCC12 50780,C#CCC(CC#C)C(=O)NCC(C1CCC1)NC(=O)COCc1ccccc1C 50781,CC(C(=O)N1CC(NC(C2CNC(=O)N2)=O)C(O)C1)C(C)C1CCCCC1 50782,c1(CNC(C2C(CC)C2)=O)nnc2n1CCN(C(=O)C(C)(C)CF)C2 50783,C(C(=O)NCC1(NC(c2c(Cl)cnn2C)=O)CCC1)(C(C)C)SC 50784,C1(C2CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)(C(=O)OC)CC(F)(F)C1 50785,N1(C(=O)CC2CC2)CCN(c2cnn(C)c2)C(=O)CC1.c12ncc(o1)C(=O)NC2C 50786,c1(C(N2C(C)C(C(=O)NC(c3ccc(CC)cc3)=O)CC2)=O)cncc(Cl)c1C.CC 50787,Cc1ccc2c(c1)C(C(=O)NC(C)CC(C)NC(c1nc(C)no1)=O)CC2.CC1CC1 50788,CC1CN(C(=O)CCc2cccc(N(C)C)c2)CCCN1C(c1ccc(Cl)s1)=O 50789,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NCCC1CCC1 50790,CCC(F)(F)C(C)(C)C(=O)N1CC2CC1CN2C(c1ccc2oc(C)nc2c1)=O 50791,c1(NC(=O)Cc2ccc(F)cc2Cl)ccc(O)cc1Cl.N12CC3(CCC3C1=O)C2 50792,C12(C(=O)NC3CC(CNC(c4ncc(OC)cc4F)=O)C3)CCCCC1OCC2 50793,C#CC1CC2CCC1N(C(C1CCN(C(=O)CC3CCCN3C)C13CC3)=O)C2 50794,c1(CN(C)C)ccc(CC)cc1C(=O)NCCN(CCC)CC1CC1 50795,c1(C(=O)NCC2(OC)CN(C(C3CCC(C)O3)=O)C2)cc2ccccc2[nH]1 50796,c1(C(N2CCC(CCNC(C(C)SC)=O)C2)=O)cccc(=S)n1O 50797,CC(C)(C(=O)N(C1CCCC1)CCCNC(C1OCCOC1C(F)(F)F)=O)C(N)=O 50798,N1(CC)CCN(C(=O)C(c2csc(C)n2)=O)CC1CCO 50799,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(C(C)C)C2)=O)C1 50800,N1(C(CCC(=C)C)=O)CC(CNC(=O)C(c2ccc(C)cc2)(C)C)CC12CCC2 50801,c1(OC)ccc(Cl)cc1CC(=O)N(C1CC(NC(=O)CC2(O)CCCC2)C1)C 50802,c1(C(=O)NCC2CN(C(=O)CC3CC4C=CC3C4)CCCO2)cc2n(n1)CCC2 50803,C1(SC)CN(C(c2conc2C)=O)CC1NC(C1CC1c1cccc(O)c1)=O 50804,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(CCO)C1 50805,C1(C(=O)NC2CN(C(C=Cc3ccn(C)c3)=O)C(C)(C)C2)CC2C=CC1C21CC1 50806,c1(C(N2CCC(CNC(C(CC)(C)O)=O)C2)=O)cc2ccccc2cn1 50807,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1cc(-c2ccccc2)on1)=O 50808,N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C(F)F 50809,Cc1ccc(C(=O)NCC(C)(C)CCNC(C2CCCC2C(F)F)=O)c(F)c1 50810,c1(OC)cc(C)sc1C(N1CC(NC(C2(OC)CCOC2)=O)C(SC)C1)=O 50811,N1(C(CC=CC)=O)CCCC(N(C(=O)CCOc2cccc(C)c2)C)C1 50812,C1(C#N)(C(=O)NCC(C(=O)NC(CCOC)CO)C)CCCOC1 50813,N1(C(COCC(=O)NC)=O)CCC2CCCC12C(=O)NCCCCCO 50814,CCC(C)(C(=O)NCCC(O)CNC(c1cc(C(N)=O)co1)=O)C(N)=O 50815,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(=O)NCCOC)CCC1C 50816,N1(C(CN(C2CC2)CC)=O)CCCN(C(c2sc(=N)[nH]c2C)=O)CC1C 50817,N1(C(C2C(NC(c3c(COC)occ3)=O)CC=CC2)=O)CC(C)N(C)C(C)C1 50818,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 50819,c1(C(=O)NCCC(C)NC(CC=CC)=O)cnc2ccccn2c1=O 50820,Cc1ccc(C)c(C(=O)NC(c2ccccc2)C(C)NC(c2ccncc2)=O)n1 50821,c1(C(C(=O)NCCCC(C)NC(CCOC(C)=O)=O)C)ccc(F)cc1 50822,C1(C(C)C)CCC(NC(=O)C(=O)NCc2cccc(Cl)c2)CC1 50823,c1(NC2CC(C)N(C(c3cccc(F)n3)=O)CC2)ncc2c(c1C#N)CCC2 50824,C1(N(C(=O)C(c2ccccc2)N(C)C)CC#C)(OCC)CCCS(=O)(=O)C1 50825,c1(NC(C(C)C2CCCO2)=O)ccc(CN2CCC2)o1.C12CN(C1)C2=O 50826,N1(C(CCOC(C)=O)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2cnn(C)c2)C1 50827,Cc1cc(O)ncc1C(=O)NC(C)(CNC(=O)CC1CCC(=O)NC1=O)CO 50828,N1(C(C(C)Oc2c(F)cccc2F)=O)CC2(COC(CN(C)C)C2)C1 50829,Cc1ccc(C(=O)NCc2cccc(CO)c2)nc1C.N12CCC(C)(CC1)C2=O 50830,N1(Cc2ccc(OCCCC(C)C)cc2)Cc2ccccc2OC(C)C1 50831,C1(C(=O)OC)CCCN(C(=O)CC2CC2C)C1.N12CC(C1)C2=O.C1CC1 50832,Cc1ccc(C(=O)N(CCNC(=O)C(C)(O)C(C)C)C(C)C)cc1I 50833,c1(C(C)C)cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc(Br)c1 50834,C1(CC(C)C)CN(C(C2CCCN(Cc3cncc(Br)c3)C2)=O)CC(F)(F)C1 50835,CC(C)(CCNC(C1OCC1(C)C)=O)NC(=O)CC1(c2ccccc2)CCC1 50836,C1(C2(O)CCC2)(C(N(CC(C)N(C)C(C2CC3C=CC2C3)=O)C)=O)CC1 50837,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 50838,N1(C(C(CC#C)O)=O)CC2CC(C(N3CCCC4(C3)N=N4)=O)(C2)C1 50839,c1(C(N2C3C(NC(C(C(CC)CC)C)=O)C(C3)C2)=O)nc(N)cc2ccccc12 50840,N1(C(C(F)=CC)=O)CCC(C)C(NC(C2(SC)CCC2)=O)C1 50841,C1(NC(C2CCCN(C(Cc3c(C)cccc3)C)C2)C)CCC2CC2CC1 50842,C(=O)(CCC(C)(C)C(=O)Nc1cnc(Cl)cc1CNC(=O)NC1CC(CO)C1)OC 50843,C1(NC(CC2(C)CCCC2)=O)C2CCN(C(c3ccc(Cl)c(F)c3N)=O)CCC12 50844,c12ccc(cn1)c(=O)o2.c1(C(C(C)NC(N)=O)N)ccccc1 50845,CC1(C)CN=C(N2CCN(C(=O)CN(c3ccccc3)Cc3cccs3)CC2)S1 50846,c1(C(N2CC3C(CNC(CCCSC)=O)(C3)C2)=O)cnc(CO)nc1C 50847,CCC(C)C(C(=O)NCC1COCCN1C)NC(C1OCCC1C(C)C)=O 50848,CCCC(O)CC(=O)NC(C)(C)CN1CCN(C(=O)CCC(C)C)CC1 50849,c1(-c2ccc(C(=O)NC(CNC(C3CCSC3)=O)CO)s2)cccc(F)c1 50850,C1(CC(C)C)CCC(C(=O)N(CC(C)CNC(=O)COCCO)C)CC1 50851,C1(NC(C(C)OCCCC)=O)CCCC1CC(=O)N(c1ccn(C)n1)C 50852,C1(CC(=O)NCC2(CNC(C(c3n(C)ncc3)(F)F)=O)CC2)CC2C=CC1C2 50853,C1(CC(=O)NC2CC(N(C(CSCC(C)C)=O)C)C2)CN(C)CC1O 50854,O=C1NC(CCC(F)(F)F)C(=O)N1CCC(F)Oc1ccccc1 50855,C1(C(N2C(CCC(=O)NCCn3ccc(C4CC4)n3)CC2)=O)CC2CCC1C2 50856,CC(=O)N=c1nc(Cl)nc(C2CCN(C(=O)CC3CCCC(C)C3)CC2)[nH]1 50857,N1(C(C(C=CC)O)=O)CCCC(C)(C(=O)Nc2ccc(O)c(C)c2)C1 50858,C(C)(CCC(=O)N1CCCC1C(C)CO)ONC(CC1ON=C(C)C1)=O 50859,N1(C(C2CC2F)=O)CCC2(CCN(S(=O)(=O)c3ccc(O)cc3)CC2)C1 50860,c1(NC(=O)NC2C(CC)CCOC2)nc2cc(C(F)(F)F)ccc2s1 50861,Cc1cccnc1C(=O)NC1CC1NC(c1cnn(C)c1F)=O 50862,C1(C(=O)NC(C(=O)NCCOCC)(C)C)CCC(O)CN1C 50863,Cc1ccc(C(C)C(=O)Nc2nc(CNC(=O)CC3CCC3OC(F)F)cs2)cc1 50864,C1(C(C)NC(c2ccc(C)o2)=O)CN(C(=O)CC23COCC(C2)C3)CCO1 50865,c1(OC(C)C)cc(NC2CCCC(CNC(C3(C)C=CCCC3)=O)C2)ncn1 50866,C1(=Cc2cccc(OC)c2)CN(C(c2conc2C)=O)CCC1C 50867,C1(NC(CC(C)C2CCCO2)=O)CCC(C)N(C(=O)Cc2cnn(C)n2)C1 50868,N1(C(C=CC)=O)CCC(NC(C23CC(C)C2C3)=O)C1C1CC1 50869,O(NC(=O)C(c1cccc(Cl)c1)C1CC=CCC1)CC(=O)N(CCOC(C)=O)C 50870,Cc1nccn2c(C(N3CCN(O)C(=O)C3)=O)cnc12 50871,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 50872,c1(N(C)CC2(N(C)C)CC2)ccc(Br)c(S(=O)(=O)N2CC(CC)OCC2)n1 50873,c1(C2(NC(=O)NCc3cc(Cl)cs3)CC2)ccc(F)c(F)c1 50874,N1(CCc2nc(-c3ccccc3)on2)CCCC(O)(CO)C1.N12CCC(CC1)C2 50875,N1(C(CCC=CC)=O)CCOC(CNC(C2CCCN2C(=O)CSC)=O)C1 50876,C1(C(C)CO)COC(C)(C)CN1C(=O)C1=CCN(C(=O)CC2CCCCCC2)C1 50877,C1(CNC(C)=O)CCCCC1NC(=O)C(C)(C)c1ccn(-c2n(CC)nnc2)n1 50878,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(c2ccc(C(F)(F)F)[nH]2)=O)CC1 50879,N1(C(C(CC)F)=O)CC(C2CCCCN(C(C3CCc4n[nH]c(C)c4C3)=O)C2)C1 50880,c1(CC)cc(C(N2CC(F)(C(=O)NC3(c4ccncc4)CC3)C2)=O)nn1C 50881,C1(C(N2CCC(CC#C)CC2)=O)CCN(C(c2csc(C3CC3)n2)=O)C1(C)C 50882,C(=O)(C1=CCOC1)N(C(C1(CNC(C2C(OC(C)(C)C)C2)=O)CC1)=O)C(C)C 50883,c1(C(C(=O)NCC2NCCC2CC(F)(F)F)O)ccc(Cl)cc1 50884,c1(C(=O)NCCN(C(=O)C(O)C(C)N(C)C)C(C)C)cnc(N(C)C)nc1 50885,C1(C(N(C)CC2CCN(C(c3cncc(Cl)c3)=O)C2(C)C)=O)CCS(=O)(=O)CC1 50886,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)F)C2)ccc(C)c([N+](=O)[O-])c1 50887,C(CCC(C)(C)NC(=O)C=C(C1CC1)C1CC1)NC(CC(=C)C)=O 50888,c1(C(N2CC(C)(NC(C3CCS(=O)(=O)C3)C)C2)=O)cccc(SC(F)(F)F)n1 50889,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(C1(C)CCCC1(F)F)=O)C2 50890,Cc1cccc(C(F)(F)F)c1-n1nc(Cn2cnnc2)nc1CCCC(C)(C)C 50891,C1(C(=O)OC)CCN(C(c2n[nH]c(CO)n2)C(=O)NCCSC(C)C)C1 50892,c1(C(N2CC(C)C(CNC(c3cnn(C)c3N)=O)CC2)=O)ccn2nccc2n1 50893,C(CCCC(=O)N(C1CCC(F)(F)C1)C)N(C(C1N(CCOC)CCC1)=O)C 50894,CN1CCN(C(=O)Cn2cnnn2)CC1NC(C1CCSC1)=O 50895,C1(C(N2CC(O)(CNC(c3cnccn3)=O)C2)=O)CC2(C1)CC2(F)F.CN 50896,CCCC(C)(O)C(=O)N1CCC(O)(CNC(=O)Cc2cc(Cl)sc2Cl)C1 50897,CC1CC(NC(=O)CC2CCN(C(C3CC(F)CN3)=O)C2)C(=O)O1 50898,N1(C(C(C2CC2)OC)=O)CCN(C(c2cn3cccc(F)c3n2)=O)CC2(CC2)C1 50899,CN1CCC(C)(C(=O)NC2(C)CC(NC(c3cc(C(N)=O)co3)=O)C2)CC1 50900,C=CC(CC)CC(=O)NCC1CC(C)CCN1C(=O)C1=CCCCO1 50901,c1(OC)c(C(=O)NCC(C2CCCC2)NC(c2c(Cl)cnn2C)=O)ccnc1Cl 50902,Cc1ccnc(O)c1C(=O)NCC.C123CCC(C1C2)OC1(CO)CN(C1)C3=O 50903,Cc1c(C(N2CC(F)(C(=O)NC3(C)CCCC3(F)F)C2)=O)cccc1O 50904,C=CCCCC(C(=O)N(CCCCCO)C)NC(C1CC(CC2CC2)C1)=O 50905,[N-]=[N+]=NCCC(=O)NC1CCC(C(=O)NC2C3CCCCC23)C1 50906,C(C(CNC(=O)CCc1nncs1)C(F)(F)F)NC(C1CC12CCCC2)=O 50907,C1(C(N2CC(C(C)NC(c3ncoc3-c3ccon3)=O)C2)=O)C(C)(C)C1(C)C 50908,c1(OC)ccccc1SCC(=O)NC(C1CN(C(=O)CC2CCC3CC23)C1)C 50909,C=CC1(CC(N2CCC(C#N)C2)=O)CN(C(c2cc(COC)on2)=O)C1 50910,C(=O)(CC(C)CNC(=O)CCC1CCCOC1)NC1(COC)CCOC1 50911,CCCS(=O)(=O)CC(=O)NCC(C)(O)CNC(C1CC2(CCC2)CO1)=O 50912,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 50913,c1(CNC(C(C)=CC)=O)ccc(CNC(c2cc(=O)n(C)o2)=O)cc1F 50914,C1(NC(C2N(C(C(CC)NC(N)=O)=O)CC3(CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 50915,c1(C(N2C(CC)C(NC(=O)CC3CC3)CC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 50916,Cc1ccc2cccc(C(N3CC(CNC(C4CC4F)=O)CC(C)C3)=O)c2n1 50917,N12CC3COCCC3(C1)Nc1c(c(F)ccc1)C2=O.CC(C)(CO)c1nn[nH]n1 50918,c1(C(N(CCN(C(C2N(CC)CC2)=O)C)C(C)C)=O)c(C2CCC2)cccc1F 50919,N1(C(C2C(C(=O)OC)C2)=O)CCC(C2(NC(c3cc(C)ccn3)=O)CC2)CC1 50920,C(C(CC)CO)NC(CN(C(C=CCOCCOC)=O)C(C)C)=O 50921,c1(C=O)sc(C)nc1C.C1(OC)CCN(CCNC(=O)C(CC2CCC2)C2CC2)C1 50922,CCCCC(O)CC(=O)NCC1CCC1C(=O)NCc1ccc(F)c(O)c1 50923,c1(CCC(=O)NCC(O)CNC(C2(F)CCCC2)=O)ccc2c(c1)OCO2 50924,C1(C)(C(N2CCC(CCNC(C(CSC)O)=O)CC2)=O)Cc2ccccc2N1 50925,C1(N(C(=O)Cc2cccnc2)C)CCCC2CC1C2 50926,CC1CN(C(=O)C(C2CCCCC2)O)CCN1C(c1ccc(F)s1)=O 50927,c1(C(=O)OC)c(F)cc(Br)c(CS(C)(=O)=O)c1F 50928,c1(C(N2CC(C(C)NC(c3cnns3)=O)C2)=O)cc([N+](=O)[O-])c2nsnc2c1 50929,c1(OC)nccc(C(N2CC(OC)CC2)=O)n1.C1C(=O)N1C(C)C 50930,Cc1nn(C)cc1C(=O)N(CCNC(=O)CC1CCCN1CC(F)(F)F)C 50931,c1(OC(C)C)cncc(C(N2CC3CC3(C(N3CC4CC4C3)=O)C2)=O)c1 50932,c1(NC(C)Cc2nncn2C)cc(Br)ccc1S(=O)(=O)N.C1(N)CCCC(O)C1 50933,C#CCC(CC(=O)NCC(C)(O)CCC)NC(C1CCCN1C(=O)C1CC1)=O 50934,N1(C(C=NOC)=O)CCCCC1CCNC(=O)CCc1ncc[nH]1 50935,C(C(CC(=O)NC(CC1CCC1)CO)NC(C1(C)COC1)=O)OC 50936,C1(CNC(C(C)C)=O)COC(CNC(c2ccc(CN3CCCC3)o2)=O)C1 50937,c1(C(=O)NC(CCCNC(C(C(CC)C)O)=O)(C)C)cc2ncn(C)c2cn1 50938,CCC(COC)C(=O)NC1CN(C(c2ccc(-c3csnn3)cc2)=O)CC1C 50939,C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(=O)C=CCN2CCCC2)C1 50940,C1(C(NOCCC)=O)N(C(c2csnn2)=O)CCC1(C)C 50941,N1(C(=O)CCc2ccccc2)CCC(C2CCCN(C(c3ccco3)=O)C2)C1 50942,Cc1sc(-c2ccccc2)nc1C(N1CC(C(=O)CS(N)(=O)=O)C2CC12)=O 50943,c1(C(=O)NC2CC(CNC(C3(C)N(C)CC(O)C3)=O)C2)ccc2nc(=N)[nH]n2c1 50944,C1(NC(C(c2n(C)ncc2)O)=O)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 50945,C#CCC(C)(C)C(=O)NC1CC(NC(c2c(Br)ncn2C)=O)C12CCC2 50946,C1(C(=O)NCC2C(NC(C3CC(CCC)C3)=O)CCC2)CCc2nc[nH]c2C1 50947,CCCCCCCCCCC(O)CNCc1cc(CC)cc(CC)c1 50948,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)Cc2cccnc2Cl)C(F)C1 50949,Cn1cc(CC(=O)NC(C)(C)C(=O)NCCCC2(O)CCC2)nn1 50950,N1(C(COCCOCC#C)=O)CC(NC(c2cc(COC)cs2)=O)CC1C 50951,c1(C(=O)NC(CC(=O)N2CCC(CC#C)C2)COC)coc2c1COC2 50952,c1(C(N2CC3C(NC(c4nc(COC)sc4)=O)(C3)C2)=O)ccc(F)cc1C1CC1 50953,N1(C(=O)CCOCC2CC2)CCC(O)C(C(N2CCCC23CC3)=O)C1 50954,C1(O)(C(C)NC(C(=Cc2ccco2)C)=O)CCN(C(c2cc[nH]c2)=O)C1 50955,N1(C(c2ccc(OC)cc2)=O)CCCCC(CNC(=O)CCCCSC)C1 50956,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCOCC1 50957,CCC(C)(CCC(C)C)C(=O)N1CCOC(CC(N2CCC(F)(F)C2)=O)C1 50958,c1(NC(=O)NC2C(C#N)CN(Cc3ccccc3)C2)ccc2ccccc2n1 50959,CCC(CC(=O)N(CCCCCNC(=O)C=C(C)C(C)C)CC1CC1)C(F)F 50960,C1(CNC(COc2ccn(C)n2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC1(C)C 50961,N1(C(C2COCCN(C(c3c(CC)ncs3)=O)C2)=O)CCNc2ccccc21 50962,c1(C(N2CCC(NC(c3n(C)ccc3)=O)C(F)C2)=O)cncc2[nH]ccc12 50963,C1(C(N(C(C2CCOCC2)C(=O)NCCCCN2CCC2)C)=O)CCCOC1 50964,C1(CC)CC(C(=O)N2CC(NC(=O)CC(C)(C3CCC3)OC)C(C)C2)=NO1 50965,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3c(C)ncs3)=O)C2)ccc(N)cc1Cl 50966,c1(C(N2CC=CC(NC(=O)C3=CCC3)C2)=O)ccc2c(=O)ccoc2c1 50967,C(=O)(C#CC1(C)CCCO1)N1C2CC(CN(C(C3CCCN(CCC)C3)=O)C2)C1 50968,c1(C(=O)NCCCCC2CN(C(C(C(CC)O)C)=O)C2)ccc2nnc(O)n2c1 50969,c1(OC)cc(CCC(N2CCC(C(N)=O)CC2)=O)ccc1O.c12nnn(C)c1N2 50970,N1(c2cc(NCc3ccco3)nc(C)n2)CCCN(C)C(=O)C1 50971,c1(CC)noc2ncc(C(N3CCN(C(C4CCCSC4)=O)C(C)C3)=O)cc12 50972,c1(C(=O)NC2C=CCN(C(C3CC4(CC(OC)C4)C3)=O)C2)ccc2c(n1)CCC2 50973,S(=O)(=O)(C1(C(N2CCC2CNC(c2ccc(CN(C)C)o2)=O)=O)CCC1)N(C)C 50974,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)C)F)C1 50975,C1(=O)CCCCCN1.C(=O)(CCCOCC)N(CCOCCO)CC.C1(C)CC1 50976,c1(C(=O)OCCC=CCC)cc(C(C)=O)ccc1C 50977,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 50978,c1(OC)cccc(C(=O)NCC2CCN(Cc3nc(Cl)c(Cl)s3)CC2)c1O 50979,C1(C(=O)NC(C(C)NC(C(CC=C)(F)F)=O)CO)CN2CCN1CC2C 50980,Cc1nc(NC(c2ccc(F)cc2F)CF)ncc1Br 50981,C=CC(CCC)CC(=O)N1CCOC(C)C1C(N1CCC(OCC)C1)=O 50982,S(=O)(=O)(c1ccc(OC)cc1C)NCc1c(F)ccc(OC)n1 50983,N1(C(C(=O)NC(C2CCCC(C)C2)C#C)=O)CCC(C)(C)CC1 50984,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(=O)C(N2CCOCC2)C)CC(C)C1 50985,c1(OC)cc(N)c(F)cc1C(=O)NC(C1CCCN1C(=O)CCCSC)C 50986,Cc1ccc(Cl)cc1C(N1CCC(NC(=O)Nc2ncncc2I)CC1)=O 50987,C1(CCNC(c2n(C(C)C)ncc2)=O)CCCCN1C(=O)CNc1nccs1 50988,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 50989,c1(OC)n[nH]cc1C(=O)N(C)CCOCCCNC(=O)Cc1nnc(O)s1 50990,CC1C(NCc2ccccc2)C(C)CCN1Cc1cnc2cccnn12 50991,C1(NC(CC(C=C)C)=O)CC(C(C)(C)C)CN(C(=O)C(CC)(CC)OC)C1 50992,C=CC(C)(CC)C(=O)NCCCc1ccc(OC)cc1 50993,C1(F)(CNC(C)C(=O)NC2CCN(c3ccccc3)C2)CCN(C(=O)C2CC2)C1 50994,N1(C(CC(C(C)C)O)=O)CCN(C(=O)Cn2cc(Cl)c(O)nc2=O)C(C)C1 50995,C1(NC(C(=O)NC2CC2)=O)CCN(C2CCOCC2)C1=O 50996,c1(C(=O)OC)cncc(C(=O)NCCOCCNC(=O)CCc2cn(C)nn2)c1 50997,c1(OC)ccc2cc(C(=O)N(C)CC3(NC(=O)CC(C)C(F)F)CC3)[nH]c2n1 50998,c1(NC(CSCC)C)nc(N2CCCC(C(=O)OC)C2)nc2scnc12 50999,N1(C(c2cc(CCC)nn2C)=O)CC2(C(=O)NCCCCCCCO)CC1CO2 51000,c1(C(=O)NC2CC(C)(C(=O)NC3CCCCCC3)C2)sccc1C#N 51001,c1(C(=O)NCC(CC(F)CO)NC(C(C(=O)OCC)F)=O)c(F)ccc2c1OCC2 51002,C=Cn1nncc1C(=O)NC1CCC(NC(=O)CC2CC2(C)C)C1 51003,c1(OC)cc(C)c(C(N2CCCC(NC(c3ccc(C#N)cc3)=O)C2)=O)cn1 51004,n1(CC)nc(C)cc1C(N1CC(F)CC1CC(=O)NCC1C=CCCC1)=O 51005,C1(NC(c2cn(CCC)nc2C)=O)CCCN(C(=O)NCC2CC2)C1C 51006,N1(C(C(C)NC(=O)CC2SCCS2)=O)CC(O)C2(CCCC2)C1 51007,c1(C(N2C(C3CCN(C(C=CC(C)(C)SC)=O)C3)CCC2)=O)cc(C)c(C)o1 51008,CCC(C)(C)C(C(=O)NC1(CC(=O)NCC2(CO)CCCO2)CCCCC1)OC 51009,N1(C(CC(C)P(C)(C)=O)=O)C(C)CC2CN(C(c3nc[nH]c4nccc3-4)=O)CC12 51010,Cc1sc(C(F)(F)F)nc1C(=O)NCCC(C(C)C)NC(=O)C(c1cnn(C)c1)C 51011,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51012,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 51013,N1(C(c2cc(C)n(C)n2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)CC1C 51014,C1(C(=O)OC)CC2CC2N1C(=O)C(N1CC2CC2C1)C 51015,CCC(C)(C)C(=O)C(=O)N1CC(C(C)(C)O)(CNC(=O)C(F)C(C)C)C1 51016,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51017,c1(C(N(CC(C)NC(=O)C(C)(O)c2ccccc2)CC)=O)ccc(C)nc1OC 51018,Cc1ccc(C)n1CC(N1CCCC1C1(NC(=O)CCn2cnnn2)CC1)=O 51019,c1(C(=O)OCC)cc(C#N)cnc1NC1CCCC(NC(c2ccncc2)=O)C1 51020,c1(C(=O)NC2(C)CN(C(C3CC(C#N)C3)=O)C2)nnn2c1CSCC2 51021,c1(CC)ccc(C(=O)NCC=CCNC(c2cccc(OC)c2)=O)c(C)n1 51022,Cn1ncc2c(N3CCCSC3)nc(=NCCCOCc3ccccn3)[nH]c12 51023,C1(CC(N2C(C(C)NC(CCCC(=C)C)=O)CCC2)=O)C2CC3CC(C2)CC1C3 51024,c1(C(=O)NC(CNC(CC(CCC)O)=O)(C)CC)cc2ccc(F)cc2[nH]1 51025,C1(COC)(CNC(=O)C(O)Cc2ccccc2)CCCN1C(=O)C(F)=C(C)CCC 51026,C[Si](C)(C)CC(C(=O)O)NCc1ccc2c(c1)COC2 51027,CCCC(CCC)CC(=O)NCC1CCC(C)(C)CN1C(c1sncc1CC)=O 51028,CN1CCC(C(=O)NCC(C)(CO)NC(c2nn[nH]c2Cl)=O)CC1=O 51029,c1(C(=O)NC(CCCNC(C(CC)O)=O)c2ccccc2)cc2cccnc2o1 51030,CCCCCC(O)CC(=O)N1CCCC(C)(NC(C2CCCCO2)=O)C1 51031,CC(C)C(O)Cc1cn(C(C)COC(F)F)nn1.C1(=O)CN1C.C1C(=O)N1 51032,C1(NC(C(C)NC(C=COC)=O)=O)CC(N=c2[nH]c3c(C)cc(C)cc3s2)C12CCC2 51033,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51034,c1(C(=O)NC2C(NC(CCC(CC)C)=O)C2)c(OC)cc(OC)cc1OC 51035,C1(NC(=O)NC(c2ccccc2)C=C)CCC(C#N)CC1 51036,c1(C(=O)NC2CC(F)(CNC(c3c(CC)nn(C)c3)=O)C2)cc2occc2n1C 51037,N1(C(c2nc(C)c(C)s2)=O)CC2(CCC2)C1C1CCCO1 51038,CC(C)CC(C)NC(=O)CCN(C(=O)CC1OCCO1)C1CCC1 51039,CCC(CCCO)NC(c1ccc(-c2cccs2)o1)=O 51040,C1(N(C(=O)C(C)CC2CCCCC2)CC)CCN(C(C2CC2(Cl)Cl)=O)CC1 51041,C1(C(=O)NC(C2CC(NC(C3CC3C3(C)COC3)=O)C2)C)CCC(O)CN1C 51042,c1(C(=O)NCC2C(CNC(C3(C(C)C)CC3)=O)C2)cnc2[nH]ncc2c1 51043,N1(C(Cc2cc(=N)[nH]cc2)=O)CCCC(NC(c2cccc(CO)c2)=O)CC1 51044,c1(N(CCC)C2CC2)ccc2[nH]c(C)cc(=NCC3CCCC34CC4)c2c1 51045,CC(C1=CCCCC1)NC(C1C2CCC(C2)C1NC(=O)CC1CCCN1C)=O 51046,c1(N2CC(C)(C)C(NC(=O)COc3ccsn3)C2)cc2nncn2cn1 51047,c1(OC(C)C)nc(C(=O)N(C(C)CNC(C2CCC(=O)N2)=O)C)cc(O)n1 51048,N1(C(c2ncn(CC)c2)=O)CCC2(CC1)CN(C(C1COCCN1CCSC)=O)C2 51049,c1(NC(C(C)OC(CNC(C)=O)(C)C)=O)cc(C)ccc1Cl 51050,C=C1COCCN(C(C2CN(C(C3CCCC(C#N)C3)=O)CC2F)=O)C1 51051,Cc1nc(Cl)[nH]c(=NCC(CNC(c2ncccc2F)=O)C(F)(F)F)c1[N+](=O)[O-] 51052,c1(OC)ncccc1CO.c12nnc(s1)C1CN(C1)C(=O)NC2 51053,C1(C(=O)NC(CN(C)C)C(=O)NCC(N)=O)CCC2(CC2)C1 51054,Cc1ccccc1C=CC(=O)NC1C2CC3C1C3C2F 51055,c1(C(=O)NCC(CC)NC(=O)CCC2CCOC2)ccc(S(N)(=O)=O)c(F)c1 51056,C1(N2CC(CC(=O)O)C2)CC12CCN(C(=O)C(C)CC#N)CC2.CCC(F)F 51057,CN1C(=O)CCC1CNC(=O)CC=CCNC(c1ocnc1C(F)F)=O 51058,N1(C(c2cccc(OCC)c2)=O)CCN(C(=O)CSC)C(c2ccnn2C)C1 51059,c1(C(=O)NC(C2CCCN2C(C2CC2C2CCC2)=O)(C)C)ccc2cncn2c1 51060,C=CCC(F)(F)CNC(=O)CC1CCN1CC1(C(=O)NC)CC1 51061,C1(C(N(C(C)CC(=O)NCC2(F)CN(C)C2)C)=O)C2CN(C)CC12 51062,c1(C(=O)OC)ccc(Cl)c(C(N2CCOCC2CNC(c2cnnn2C)=O)=O)c1 51063,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51064,C=C(C)CC(=O)NCC(C)NC(=O)CC1(SCC)CC1 51065,C(=O)(CC(C)CC(=O)N1CCC(C)(C)C1C(=O)NCCc1cc(C)no1)OC 51066,c1(C(C)C)ccccc1C(=O)NCc1cc(C(=O)NC(C)(CO)CO)co1 51067,C1(NC(C(C)O)=O)CN(C(=O)C=CC2CCCCCC2)CCC12CCC2 51068,C1(C)(NC(C(C)=C2CC2)=O)CC(NC(C2CCC(Cc3cnn(C)c3)C2)=O)C1 51069,c1(C(N2CCC(NC(C3ON=C(C)C3)=O)C(O)C2)=O)cc2ccc(F)cc2s1 51070,c1(C(=O)NCC2(F)CC(NC(=O)CC3CC(F)(F)C3)C2)nccc(Br)c1O 51071,CC(C)C(CO)C(=O)N1CC(F)(F)CC1CCNC(c1ccccc1)=O 51072,CCCC(C(=O)N(CCCNC(C1CCN(C)C1C)=O)C1CC1)NC(N)=O 51073,c1(C(=O)O)ccc(NCC2(F)CCCC2)nc1.N12CC3CC3(C1)C2=O 51074,c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)C2)CCO)=O)ccc(F)c(C)c1N 51075,c1(-c2onc(C3(c4cn(C)nc4-c4ccnn4C)CC3)n2)ccc(F)c(F)c1 51076,CC1CN(C(C2CCN2C2CCCC2)=O)CC1(C)CNC(=O)COCC(F)F 51077,Cc1cnc2cccc(C(=O)NCCOCCC(C)(C)NC(C3(C)CC3C)=O)n12 51078,C1(CC(=O)NC2CC(C#C)C2)(CNC(=O)C(O)C=CC)CCCCC1 51079,c1(C(=O)NCC(CC)(CC)NC(=O)CN2CCOCC2=O)nc(Cl)ccc1N 51080,N1(C(c2cc[nH]n2)=O)CCCC(C(N2CCC2C2CC2)=O)CC1 51081,N1(C(C)C)CCN(CC2CCCOC2c2ccc(F)cc2)CC1C=O 51082,c1(CCC)cccc(C(N2CCC(C)(CNC(=O)CCS(C)=O)C2)=O)c1 51083,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51084,c1(CC(C(=O)NC2CC(CCNC(C3CC3C(F)F)=O)C2)O)ccc(F)cc1F 51085,C(c1ccccn1)=C(C)C(=O)NC(C)CN(C(=O)CNS(C)(=O)=O)C 51086,CCCCC(F)C(=O)NC(C)CCN(C(=O)CCc1ccc(C(F)F)cc1)C 51087,N1(C(C(=O)NC(C)C)=O)CCC2CC12C(=O)NC(CO)C(N)=O 51088,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CN1CCC(C)C1 51089,C(C)(c1cnccn1)=CC(N1CCN(CC2CN(C(C(C#C)(C)C)=O)C2)CC1)=O 51090,C(=O)(CC(CN(C)C)C(F)(F)F)NCCN(C(CCC1C(C)=NOC1=O)=O)C 51091,c1(C(N2C(CNC(C3(CSC)CC3)=O)CC2)=O)c(C)cc(C)cc1O 51092,C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CN2CCOC2=O)C1 51093,c1(NC(C2COCCN(Cc3cncc(OC)c3)C2)=O)cc(F)c(C)cc1Br 51094,c1(C(=O)NC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)ccc(=O)n2c1COCC2 51095,C1(C(N(CC(C)NC(C23CC(CO2)C3)=O)CC)=O)CCOC(=O)CC1 51096,c1(OCC)ccc(C(N2CC(N(C(=O)Cc3ccsn3)CC)C(O)C2)=O)cc1N 51097,c1(N(C)C)ccnc(C(N2CC(CF)(NC(=O)C(F)(F)CO)C2)=O)c1 51098,C1(NC(C2C(C)(CC)C2)=O)CC2CCC(C1)N2C(C1(SC)CC1)=O 51099,c1(C(=O)NC(CC=C)CNC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51100,C1(C(=O)NC2CC(NC(C(C)OCC=C)=O)C2)CCC2(CC1)CC2(F)F 51101,Cc1cc(C(=O)NCCC(O)CNC(=O)CCC2CC2)n(CCO)n1 51102,CCCC(C)(O)C(=O)NC(C1CC1)C1CC1NC(=O)Cc1ccc(Cl)cc1Br 51103,C1(CNC(CCc2ccc(OC)nc2)=O)(NC(=O)C(C)C#N)CCCCC1C 51104,N1(C(C2CCC(CCCCC)O2)=O)CC=CC(NC(=O)C(C)(Cl)Cl)C1 51105,CC1CN(C)CCN1C(=O)CC1CCCN1C(c1ccccc1)=O 51106,C(c1cccc(Br)c1)=CC(=O)NCC(C)NC(=O)Cc1ncn(C)n1 51107,C(CC(C)C)(C(=O)N1CC(c2ccn(C)n2)C1)ONC(C(C)SC)=O 51108,c1(SOc2c(NC)cccc2C)nn(C)c(Cl)c1I 51109,C(=O)(C(O)CC[S+](C)C)NC(CN(C(C1(C)C(C)C1)=O)C)(C)C 51110,Cc1nnccc1C(=O)NC(C1CCOC1)CNC(=O)CN1CCOCC1 51111,c1(OC)cccc(C=CC(=O)NC2CC2NC(=O)CCc2nnc(S)nc2O)c1 51112,Cc1c(C(=O)NCc2n[nH]cc2C(=O)NC2COCC2CO)nnn1C 51113,C12CC(F)CN(C1)C2=O.c1(NC(CC2C(C)CCC2)=O)cc(C(F)(F)F)ncn1 51114,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51115,C1(C(N(CC(C)C(=O)N(C)Cc2ccncn2)C)=O)C(C)(C)C1(F)F 51116,C1(F)(C(=O)NC2C(C(C)C)CCCC2)CCN(C(c2ccccc2)=O)CC1 51117,C1(CNC(=O)CSC(F)F)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51118,N1(C(c2cnc(CC)s2)=O)CC2(CC(CNC(C3CCCCO3)=O)C2)C1 51119,c1(OC2(CC(=O)NCCC(C)C3(c4ccccc4)N=N3)CC2)ccc(F)cc1O 51120,N1(C(C(C2CCC(=O)N2)C)=O)CC2(C1)CN(C(C1(c3ccsc3)CC1)=O)C2 51121,CC1(CNC(C2CC(CSC)C2)=O)CCCN1C(C1CCC(C(F)(F)F)O1)=O 51122,N1(C=O)CC2C(C(=O)CCN(C)C(=O)OC(C)(C)C)C2C1.C1(CCC)(N)CCCC1 51123,C1(OC)CCCC(C(N2CCC(NC(=O)Cc3cn(C)cn3)CC2)=O)C1 51124,c1(CN(C(C(=O)NC(C#N)C2CC2)C2CC2)C)ccc(F)c(F)c1 51125,C(=O)(C(CCNC(=O)CC1(C#N)CC1)OC)N1CCC(C(CC)CC)C1 51126,c1(C(=O)NC2(CCNC(c3ccc(N)c(F)n3)=O)CC2)cc2ccc(O)nc2s1 51127,CC1C(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CCCN1C(=O)CC1(C#N)CCCCC1 51128,Cc1nnc2n1CCCC2C(=O)c1nnc(-c2cc(F)ccc2F)o1 51129,N1(C(C(NOC)=O)=O)CCC(C=CC(=O)NC(C)CC(C)(C)C)CC1 51130,C1(CC(=O)O)CCCN(C(C2CCCN(Cc3cccc(Cl)c3)C2)=O)C1 51131,C1(N)CCCCN(CC(C(=O)C(C)C)=O)C1.C(=O)(C(F)(F)F)N(C1CCOCC1)C 51132,CCCCC(CC)C(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C2(CCC2)C1 51133,C1(O)(CN(C)C(c2ccnn2CC#N)=O)CCN(C(=O)COC2CCOC2)C1 51134,C1(C)(CNC(N2CC(n3cc(OCC)nc3)C2)=O)CSCCO1 51135,CC1CN(C(c2cscc2Cl)=O)CC1NC(c1cccc(OC(F)F)n1)=O 51136,c1(OCCC)c(F)cc(-c2cccc(C(N3CC4CCC3C(O)C4)=O)c2)cc1F 51137,C1(N(C(COCC(C)C)=O)C)CCN(C(=O)Cc2cncn2C2CC2)CC1 51138,N1(CC)CCCN(Cc2cc(C(=O)Nc3cnn(C(C)(C)C)c3)on2)CC1=O 51139,C(=O)(CS(=O)(=O)C1CC1)N1CCN(C(c2c(C)cc(C)nc2)=O)C(C2CC2)C1 51140,c1(C(=O)OCC)cncc(C(=O)NC2CN(C(c3cc(C)on3)=O)CC2C)c1 51141,c1(C(N2CCN(C(C)C)CC2)C(=O)NCCC)ccccc1SC 51142,C(CO)(CCCCNC(c1ccnn1C(C)C)=O)NC(c1c(CC)ncs1)=O 51143,N1(C(CN(c2ccccc2)C(C)=O)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51144,c1(C(=O)NC(c2cn(C(CC=CC)C(=O)NC3CC3)nn2)=O)nnc2n1CCC2 51145,C1(NC(c2nnc(O)nc2O)=O)CC=C(C(=O)N2CCCCC2CO)C1 51146,N1(C(C=Cc2ccn(C)c2)=O)CCC2(CC(NC(=O)CN=S(C)(C)=O)CO2)C1 51147,c1(C(N2CC(OC)CC2CNC(c2c(CC)n(C)nc2)=O)=O)n[nH]cc1[N+](=O)[O-] 51148,Cc1cc(Cl)cc(C(N2CC(NC(=O)CSc3ccncc3)CC(C)C2)=O)c1N 51149,C(=O)(CP(C)(C)=O)C1C(c2n(C)nnc2)C1.N12CCC(C1)C2=O 51150,c1(OC)cccn2ncc(C(=O)NC(C)CNC(=O)Cc3cc(F)ccc3O)c12 51151,c1(C(=O)OC)cc(C(=O)NC2(C)CN(C(=O)CC3CC3C)C2)cc(C)c1 51152,C(=O)(C(C)S(N)(=O)=O)NC1CCCN(Cc2ccc(C(=O)NCCOC)cc2)C1 51153,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51154,CCCCCC(CC)C(=O)NC1CN(C(c2nccnc2CC)=O)CC1N=[N+]=[N-] 51155,C1(C(=O)OC)(CNC(CCC)=O)CCCN(C(=O)CC2C(CO)C2(C)C)C1 51156,C1(C(N2CCC(C(C)NC(C=Cc3nc(C)sc3)=O)C2)=O)Cc2ccccc2O1 51157,c1(C(=O)NCC23CC(NC(c4c(OC)ccs4)=O)(C2)CO3)cccc(O)c1Cl 51158,c1(-n2cc(C(C)NC(c3cc[nH]c3)=O)nn2)cccc(Br)c1Cl 51159,CN1CCC(NCCCC(N2CCN(COC(N)=O)CC2)=O)CC1 51160,CC(C)(CC(F)(F)F)C(=O)NCC1CC1CNC(=O)CCc1ccc[nH]1 51161,c1(CS(=O)(=O)NC(c2cncc(NC)c2)=O)ccc(F)c(F)c1.C#CCNCC=C 51162,N1(C(C(C=C)O)=O)CC(OC)C(OC)C1CNC(=O)CCS(C)(=O)=O 51163,c1(OC)cc(C(=O)NC(C2CCCN2C(c2cnn(C)n2)=O)C)[nH]n1 51164,c1(CC(=O)N(C(C)C)CCN(C)C(C2CCOC2C)=O)cnc2n1CCCC2C 51165,C1(C(=O)NCCn2cc(CO)nn2)CC12CCN(C(=O)C=Cc1cscn1)C2 51166,Cc1cc(=NCCCN(N2CCCC2=O)C)[nH]c(N2CCCN3CCCC3C2)n1 51167,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51168,c1(CC(=O)NC(CNC(c2cc(OC)ns2)=O)C2CCC2)cccc(C#N)c1 51169,C1(NC(C(C(=O)OC)F)=O)CCCCN(C(=O)CNC(=O)C(F)(F)F)C1 51170,c1(NCc2cccc(C3(C)CC3)c2)nccc(=NC2CCCC23CCOC3)[nH]1 51171,C1(CN(C(=O)CCNC(C2CCO2)=O)C)CCOCC1 51172,N1(C(CCCOC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51173,N1(C(CSCC)=O)C(C(N2CSCC2CO)=O)CCC12CC2 51174,C1(C(=O)NC(c2ccc(Br)cn2)C)C2CCC(C2)N1C(=O)CN1CCOCC1C 51175,C=CCC(C(=O)NC1CC=C(C(=O)NC2COC(C)(C)C2)C1)C(C)C 51176,Cc1occc(=O)c1OCC(=O)Nc1cnc(-c2cncc(C(F)(F)F)c2)s1 51177,N1(C(c2c(C)nn(C)c2)=O)CCC2(CC(C(=O)N3CCOCC3C)=NO2)C1 51178,c1(C(C(=O)NCCC(=O)OC)NC(=O)Cc2nccn2C(C)C)c(C)cccc1Br 51179,N1(C(C2CN(OC)C(=O)C2)=O)C(C)CC2CN(C(=O)CCC(C)N(C)C)CC12 51180,C1(CC(=O)N(C(C)C(=O)NCCC2CCC2)C2CC2)CCN(C)CC1 51181,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51182,N1(C(c2c(OC)cncn2)C(=O)NCC2CCCO2)CC(CO)C(C2CC2)C1 51183,c1(COCCOC)cn(CC(=O)NC(C)C(=O)Nc2ccc(C(N)=O)o2)nn1 51184,C1(C(=O)NCC(CC=C)NC(c2cnc(C)[nH]2)=O)CCC(C(=O)OC)CC1 51185,c1(C(=O)NC2C(NC(CC(CC)C3CCC3)=O)CCCC2)ncnc(C)c1C 51186,C(CC(C)(C)NC(=O)CNC=O)NC(CN(c1ccccc1)C)=O 51187,C1(NC(=O)Nc2ccc(F)cc2)CCCCN(CC2(C3CCCO3)CCC2)C1 51188,N1(C(CC(C)O)=O)CCc2c(C(N3CC(CO)C4(CC4)C3)=O)csc2C1 51189,CCCCCC(O)CC(=O)N1CC2CCCC2(C(=O)NCC(C)C(C)(F)F)C1 51190,c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(Cl)nc3)CC2)ccc2c(c1)COC2 51191,c1(NC)cncc(C(N2CCCC(N(C(=O)Cc3occc3C)C)C2)=O)c1 51192,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CCc2nc(O)n[nH]2)CCO1 51193,C(CNC(=O)CNC(C1CCCCCC1)=O)(CC(C)C)NC(C=CCC)=O 51194,C1(N(C(c2ccc(C(F)F)cc2)=O)CC)CCCN(NC=O)C1.C(C(CCC)SC)O 51195,C12(CCNC(c3csc(CNC(c4ccc[nH]4)=O)n3)=O)CC(CO1)C2 51196,c1(C)ncc(Cl)n1C.c1(C(C(=O)NC(C)C)N(CC)C2CC2)cnc(N(C)C)nc1 51197,c1(C(=O)OCC)nc(NS(CCc2nc(COC)on2)(=O)=O)cs1 51198,c1(C(=O)OC)ncn2ccccc12.C1(=O)CC(=O)NCCCO1 51199,CC1CCC(C(=O)NCCn2cc(C(=O)NCC(F)(F)C(N)=O)cn2)CC1 51200,c1(C(=O)NCC(CNC(Cc2c(C)ccs2)=O)O)ccc2[nH]ccc(=O)c2c1 51201,C1(C(=O)NCC(C)(C2CC2)NC(C2(c3ccc(C)cc3)CC2)=O)CC2CCC(C1)C2 51202,C1(C)(CC)NC(=O)N(Cc2nc(C3(C)CN(C)C3)no2)C1=O.C(C)(C)(C)OC(=O)OC 51203,c1(C(N2CCC(CCCC)C2)C(=O)NCC)c(C)cccc1C.C(CO)N(CC)CC 51204,Nc1cccc(C(N2CCC(CNC(=O)CCc3ccc(O)nc3)C2)=O)c1 51205,c1(OC)noc(C)c1C(=O)NC1CCC(C(=O)NC(c2cncs2)C)CC1 51206,c1(OC)ccccc1CNC(C1CC1NC(c1ncc(OC(F)(F)F)cn1)=O)=O 51207,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3ccnn3)C(F)C2)=O)c1 51208,C(CC(C)C)(C(C(=O)NC1CCCCC1)N(C)CCC1CCOC1C)OC 51209,c1(C(=O)NCCCC2COCCN2C(=O)C(O)C2CC2)ccc([N+](=O)[O-])cc1 51210,c1(OC)cc(C)c(C(=O)COC2(c3ccc4c(c3)OCO4)CC2)c(C)c1C 51211,n1(CC(=O)OCCN(c2ccc(C)c3n2nnn3)CCO)nc(C)c([N+](=O)[O-])c1C 51212,c1(CN2CC(C)(CNC(=O)Cc3ccc(F)cc3Cl)C2)cccc2ccnn12 51213,c1(C(=O)NCC2C(C)CN(C(C3CCCC3C)=O)CC2)nc(Cl)c(=O)[nH]c1N 51214,C1(CNC(CC(C)OC)=O)CC(=O)N(C2CN(C(=O)CC3(C)CC(F)(F)C3)C2)C1 51215,c1(C(=O)NC(CNC(c2cnc(OCC)nc2)=O)CC(C)C)ccc(F)cc1C 51216,c1(C(=O)NC2CCC2NC(c2cnc3[nH]ccc3n2)=O)nc2cc(O)ccc2[nH]1 51217,N1(C(CCCCC#C)=O)CCS(=O)(=O)C(CCNC(=O)C(O)P(C)(C)=O)C1 51218,N1(C(C2C(OC)CC2)=O)CCC(NC(=O)CNC(c2cccc(C)c2)=O)C(C)C1 51219,C1(O)(C(=O)NC2CCC(CNC(C(N3CCOCC3)C)=O)C2)CCCC(C)(C)C1 51220,c1(C(N2CCNCC2C#N)C(=O)NCCCCCC)ccnc(C(F)(F)F)c1F 51221,S(=O)(=O)(c1cc(Br)c(Br)s1)NC1CCC(C(=O)NC2CCC(=O)NC2=O)C(O)C1 51222,C(=O)(C(CC1CC1)N(C(=O)CCc1cnco1)C)OCC.C1(=O)C(C)N1 51223,C1(CNC(c2nnn(CC)c2C)=O)C(C)CCCN1C(=O)C(C)OC1CCCC1 51224,c1(CC(=O)N(CC(O)CN(C)C(C2CC2OC)=O)C)csc(Cl)c1 51225,C(C(=O)N=c1cc(C)n(CCO)[nH]1)SCc1c(NCC)cccc1F 51226,C(C(CNC(=O)C(F)=CCCF)C(F)(F)F)NC(C1CCN(C)CC1)=O 51227,c1(NC(COC(CC(C=C)C)=O)=O)cc(C)cc2cccnc12 51228,C1(NC(c2nsnc2O)=O)C=CCCC1C(=O)NCCc1cnn[nH]1 51229,c12ccccc1Cn1cc(nn1)CO2.N1(C(C)=O)CCCC1CO 51230,c1(C(N2CCC(C(N3C(COCC#C)CCC3)=O)(CO)C2)=O)cccc(=O)n1C 51231,C(Cc1ccccc1)(CCCO)NC(=O)Nc1n(CC)cnc1 51232,c1(COC)ncc(C(=O)OC)s1.C12CCCN1CCCN(CCN(C)C)C2=O 51233,c1(SCC(N2CCN(C(C3CC(C)(C)C3)=O)CC2)=O)ccc(F)c(F)c1 51234,N1(C(C(c2ccc(C)cc2)CC)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 51235,N1(C(C2(SC)CCC2)=O)CCN2CCN(C(=O)C#CC3CCOCC3)CC2C1 51236,N1(C(c2c(COC)cccn2)=O)CCC(NC(=O)C(F)CC(C)C)C(C)(C)C1 51237,c1(N(C)CC2CN(C)C2)nc2c(F)cc(F)cc2c(=NCCC#CBr)[nH]1 51238,CC(O)C(F)(F)C(=O)N1CCC(CN(C(=O)CSCC(N)=O)CCO)CC1 51239,C1(CC(=O)NC2CC(C(C)C)C2)CN(C(=O)CC(F)(F)F)CC1CN(C)C 51240,C(=O)(CCCCCSC)NCC(CC)NC(c1ccc(CO)cc1)=O 51241,N1(C(C2(CC=C)CC2)=O)CC2CCN(C(=O)C=C(C)C)C2C1 51242,N1(C(c2c(CNC(C(CCCC)=O)=O)occ2)=O)CC(C)OC2(CCC2)C1 51243,C#Cc1ccc(C(N2CCC(CNC(c3cncc(C)n3)=O)CC2C)=O)c(F)c1 51244,CCC(C(=O)N1CC=CC1CNC(c1ccnn1C(C)(C)C)=O)NC(C)=O 51245,c1(C(=O)NCCN(C(C(CC)n2ccnc2)=O)C)cc(OC)c(Cl)cc1OC 51246,c1(C(N2CC(CCNC(Cc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51247,Cc1c(C(=O)NC2CN(C(=O)CC3CCCOC3)CC2O)oc2c(Cl)cccc12 51248,C1(NC(C2(SC)CC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 51249,N1(C(C(C)OCC)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51250,c1(C(C(N(C2(C(=O)NC(c3ccns3)C)CC2)C)=O)C)nc[nH]n1 51251,Cc1c(-c2cc(C(N3CCC(C)C(O)C3)=O)n[nH]2)cc(F)cc1F 51252,C1(COC)=NC2=CC(=NC3CCCC(C3)CN2)N1.C(C#CCCO)SC 51253,C1(C(C)NC(c2cc(C3CC3)[nH]n2)=O)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F 51254,N1(C(C=C(COC)C)=O)CCCC2(CC(NC(c3sc(C)nc3C)=O)C2)C1 51255,N1(C(C(C)CN(C(=O)Cc2ccc(F)nc2)C)=O)CC2CC1CO2 51256,C(CN=c1[nH]c(=NC2CSCCSC2)c2ncccc2[nH]1)c1ccc(OCC)cc1 51257,c1(C(C)C)c(C(=O)NCC(O)CN(C(=O)CC2CC=CCN2C)C)cnn1C 51258,C1(N(C(CCC#C)=O)C2CCOCC2)CC2CC1N(C(=O)CC(CC)C1CCC1)C2 51259,c1(C(=O)NCC2(COC)CN(C(c3cccnc3N)=O)C2)ccc2ccnn2c1 51260,C1(C2(O)CN(C(=O)CC3CCOC3C)C2)(CNC(CC(C)C)=O)CC1 51261,C(=O)(CCCC(F)F)N1CCC(N(C(C(C(C)C)C)=O)CCO)CC1 51262,C1(OCC)CCCC(C(=O)NOCc2cn(-c3c(Cl)cnn3C)nn2)C1 51263,N1(C(CC(C)OC)=O)CC(C)N(C(c2c[nH]nc2OC)=O)C(C)C1 51264,C(C(=O)N(OC)C1CCC1)N(CCC)C(C12CCCC1OCC2)=O 51265,c1(CC=C)ccccc1C(=O)NC1CCOC(C(=O)N(C(C)CC(C)C)C)C1 51266,c12ccnc(c1O)C(=O)N(C(c1cccs1)C)C2=O.C1(OC)CCCCC1 51267,C(N=c1[nH]c(=N)[nH]c(=NCc2ccccn2)[nH]1)C1(N(C)C)CCCC1 51268,C1(C(C)=O)CC1(Cl)C(=O)NCC(C1CCCC1)NC(=O)COc1cnsn1 51269,CCC(C)CC(C)C(=O)NCc1ccc(CNC(c2cc(C)c(C)cc2C)=O)cc1 51270,c1(NCCCC)ccc(C(=O)NC2CCC2NC(=O)CCC)c(C)c1 51271,N1(C(CCC2CC(OC)C2)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC1CO 51272,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2(N(C)C)CCCC2)=O)C1 51273,C1(NC(C(CC#C)NC(=O)C(C)CC2CC2)=O)CCCOC12CCC2 51274,N1(C(CCOCCC)=O)CCN(C(c2cn(C3CC3)cn2)=O)CCC1C 51275,C(C)(CC(C)C(F)F)NC(CN(C(c1cc(CC)[nH]n1)=O)C)=O 51276,C1(O)(CCNC(C(C)SC)=O)CCN(C(=O)CC=Cc2ccccc2)C1 51277,CC1=C(C(=O)Nc2cccc(-c3[nH]c(C)c(C)c3C#N)c2)SCCO1 51278,Cc1ccc2cc(C(=O)NC(C)(C)CNC(C3CCC4(CCOC4)O3)=O)[nH]c2c1 51279,C1(C(C)C)CCCC1C(=O)NC12CC(NC(c3cccn3C)=O)(C1)C2 51280,N1(C(Cc2n(C)cnn2)=O)CCC2CN(C(C3CC(C4CC4)=NO3)=O)C2C1 51281,C(C(C)(C)C#CC(=O)NCP(C)(C)=O)NC(C(CC)COC)=O 51282,C1(NC(C2CN(C(C)C)C2)=O)CC2(CCC(CNC(C3CC(CF)C3)=O)OC2)C1 51283,C1(C(N2CCC(C)(CCO)C2)=O)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 51284,N1(C(Cc2n(C)ccn2)=O)CC2(CC(CNC(=O)CC3OCCC3C)C2)C1 51285,c1(CN2C(C(=O)NC(C(C)O)CO)CC2)ccc(F)c(C#N)c1 51286,c1(C(N2CC(CCNC(=O)C(C)CC3CCCO3)(OC)C2)=O)ccc(=NC)[nH]c1 51287,C1(C(=O)NCC(CC)OC)CC(NC(=O)C(C)C2CCOC2)CCO1 51288,N1(C(C2CC(=C)C2)=O)CCC2(CC(NC(c3c(-c4ccccc4)coc3C)=O)C2)C1 51289,N1(CC(=O)NC2C=CCN(C(c3c(C(C)C)[nH]cc3)=O)C2)CCCCS1(=O)=O 51290,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51291,C1(C)(C(=O)NC2CN(C(c3sc(CC)c(C)c3)=O)C3C2C3)CCC(C)CC1 51292,C12(C(CN(C3CN(C)C(C)(C)C3)C)=O)CC3CC(C1)CC(N)(C3)C2 51293,N1(C(C)(C)C)CCC(C(O[Si](C)(C)C)=O)CC1.C1CS1 51294,CC(C)CC(=O)NCCCN(C(C1CNC(=O)N1)=O)C(C)C 51295,N1(C(C(C)OC)=O)CCN(CC2CCCCN2C(c2cc(C#N)no2)=O)CC1 51296,c1(C(N2C(C)CC(NC(CC(C)(C)OC)=O)C2)=O)cccc2[nH]cc(Cl)c12 51297,C(=O)(CC(O)C(C)C)NC(c1ccc(C)cc1)CNC(=O)Cc1ccccn1 51298,CON1CC(C(=O)NCC2CCCC2C(=O)NC2(C)CC=CC2)CC1=O 51299,C(C)(CCC(C)(C)C)(c1nnnn1C(C)(C)C)NCC1=CC(C)(CC)C1 51300,c1(N(CCN(C(C)C)C(c2csc(CO)n2)=O)C)nc(O)c2ccc(Cl)cc2n1 51301,N1(C(C(C)(C2(C)CC2)OC)=O)CC2CC(NC(c3cccs3)=O)CC1C2 51302,c1(OC)ccc(NC(C2CC(NC(=O)C3=CCCOC3)C2(C)C)=O)cc1C 51303,N1(C(CC(CC)OC)=O)CC(NC(=O)CC(=O)NCC2CC2)C2(CC2)C1 51304,c1(-c2c(F)ccc(C)c2)cc(C)c(C)cc1I.C12(CCOCC1)c1noc2n1 51305,O=C(CCCc1ccc(F)cc1F)NNC(=S)NCCc1ccccn1 51306,C1(CC(=O)NCCN(CCOC)C(c2n[nH]cc2Br)=O)CCCC(=O)N1 51307,Cc1cc(N(CC(C)CO)C)nc(=NCCc2ccc(C(F)F)cc2)[nH]1 51308,C1(C(N(CC(C)OC)CC)=O)(NC(C2CCCO2)=O)CCC1 51309,c1(C(N)=O)cc(C(=O)NC2CCCC2CNC(c2cnc(C3CC3)[nH]2)=O)co1 51310,C(CCCCC(=O)NCCn1cc(C(N2CCCC2C(=O)N(C)C)=O)nn1)OC 51311,N#CC1(C(N2CCOC(CNC(=O)CCC(N)=O)C2)=O)CC(F)(F)C1 51312,c1(C(=O)NC(C)CC(C)NC(C2CCCC2c2cnn(C)c2)=O)ccc(O)nc1 51313,C1(C(=O)NC(CN(C(c2c(C)nc(C)[nH]2)=O)C)(C)C)CC2COCC2C1 51314,C(CC(C)CC)(C(=O)NCC(C)(O)CC(C)C)NC(c1c(CC)nn[nH]1)=O 51315,c1(CNC(=O)NC2CCC3CC23)ccc(C2CCC2)cn1 51316,C1(C(=O)NC2(F)CN(C(C=C(C)C3CC3)=O)C2)CCCCC1O 51317,C1(C(C(C)NC(=O)NCc2ccccc2)C)CCCN1C(=O)CC1CC(F)(F)C1 51318,c1(CC)c(Cl)nc[nH]c1=NCC1CC(C)(C)CCC1NC(=O)C(C)SC 51319,N1(C(CCCOCC)=O)CCN(C(c2cc(OC)ns2)=O)CC1C1CC1 51320,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)n1nccc1C)CO2 51321,C1(C(=O)NCCC2CCN(C(=O)CC3COCCO3)C2)CCn2ccnc2C1 51322,c1(C(N2CCCC(NC(CCc3ncn(C)c3)=O)C2)=O)cc(O)cc(Br)c1 51323,Cc1cccc(CC(=O)NC23CC2CN(C(c2ccsc2C(F)F)=O)C3)c1Cl 51324,N1(C(c2ccccc2)CCOC)CCC(S(=O)(=O)C(C)C)C1 51325,N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 51326,c12cc3n(n1)CCCN(C3)C2=O.c1(CNC(=O)C(F)Cl)ccc2nc(O)oc2c1 51327,c1(CC(N2C(CC)C(NC(=O)CC#N)CCC2)=O)c[nH]c2cc(C)ccc12 51328,C12(CNC(CCOC(C)C)=O)CCCC1N(C(C1CC3(CCC3)C1)=O)CCC2 51329,N1(C(c2cccc(Cl)c2F)=O)CCOC2(C1)CN(C(C13COCC1C3(F)F)=O)C2 51330,N1(C(CS(C)(=O)=O)=O)CCN(C(c2cc3cccn3cn2)=O)C2CCCC12 51331,C12(C(N(CC(=O)NCC(C)OCC#C)CCC)=O)CC(C#N)(C1)C2 51332,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCN(C)CC2)C1 51333,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51334,c1(CNC2C(Nc3ccnc(SC)n3)CCCC2)cc(O)cc(O)c1 51335,c1(C(=O)NCCN(C(=O)C(O)C(F)F)C2CCCC2)cc(Br)cc2c1OCC2 51336,N1(C(CCCCC=C)=O)CCC2CN(C(=O)C(C)C(C)C)CCC12 51337,CC(CNC(=O)C(C)n1cccc1)CC(=O)NC1(C2CCC2)CC1 51338,c1(C(=O)NC(CCNC(c2c(C)snc2)=O)C)nn(C(C)C)cc1Br 51339,c1(OCC(=O)NCCOC)ccc(OC(=O)CC2(C)CCC2)cc1 51340,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2N)=O)CCC12CCC2 51341,c1(SC)ccc(C=CC(N2CC(C(C)NC(C3CCCCC3O)=O)C2)=O)s1 51342,C1(C(=O)NC2(C=C)CCC2)CCN(C(c2ncsc2NC)=O)C1(C)C 51343,c1(NC(C=C(C)CNC(=O)C(C)=C2CCCC2)=O)ccc(NC(C)=O)c(F)c1 51344,Cc1ccc(Cl)c(C(=O)NC(C)Cn2cc(CNC(=O)COC(C)C)nn2)c1O 51345,CC(O)C(C)(C)C(=O)N(CCC(C(C)(C)C)NC(=O)CN(C)C1CC1)C 51346,C1(OCC(N2CC(CC(C)N)C2)=O)CCCCC1.C1(O)(CC=O)CCOC1 51347,c1(C(=O)NCCC(=O)NCCC2CC(OC)CN2C(C)=O)c(F)ccc(F)c1Cl 51348,C12(CNC(C3(COC(C)C)CC3)=O)CCC(C1)N(C(=O)C(C)n1cccc1)C2 51349,C1(CC)(CC)CC(C(=O)NCC2(C(=O)NC3CCCC3C)CCCO2)C1 51350,c1(NC(CN(C(c2cn(C)nn2)C(=O)NC(CC)(C)C)C)=O)cncc(C)n1 51351,Cc1cc(C(=O)NC2CCCCC2N(C)C)c(Br)s1 51352,S(=O)(=O)(c1cccnc1NCCOC(CC)(C)C)N1CC(C)OC(C)C1 51353,C(=O)(C1CCOc2ccccc21)N1CC(NC(c2nocc2C)=O)CC(OC)C1 51354,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51355,C(=O)(C#CC1(C)CCCO1)NCC(C)N(C(c1cc(Cl)ccc1O)=O)CC 51356,c1(C(N2C(C)CN(C(=O)C(F)n3cccn3)CC2)=O)c(Br)ccc2c1OCC2 51357,CCCCC(O)C(=O)N1CC(CNC(c2cc(CO)oc2C)=O)C(F)(CO)C1 51358,C1(C(=O)NCCN(C(=O)CCCSc2ccccc2Cl)C(C)C)CC2C=CC1C2 51359,N1(C2(CCN(C)C)CC2)CCC2CCCC12C(=O)NCC1N(C=O)CC1.C1CC1 51360,c1(C(=O)NCC(C2CCCCN2C(=O)CC2CSC2)C)ccc(S(=O)(=O)NC)cn1 51361,C1(NC(C(=O)NCCC(CC)O)=O)CCC(C(C)(C)C)CC1 51362,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(C)C(NC(=O)CSS(C)(=O)=O)CCC1 51363,Cc1nn(C)nc1C(N1CCC(C(C)(C)NC(c2ccnc(OC(F)F)c2)=O)C1)=O 51364,CCC(CC(=O)N1CC(C)(C)CC1CC(=O)N(C)Cc1cnnn1C)CC(C)C 51365,CC(CC(=O)N(C)CCc1ccccc1)NC(=O)CC1(C#N)CC1 51366,C(CC(C)C)(C(=O)O)OCC(=O)NCC1CCC1(F)F.c1(OC)cccc(C)c1 51367,CCCCS(=O)(=O)N1CCCC(C(=O)N(CCC2(C)CCO2)C(C)C)C1 51368,C(=O)(C#CC1(C(F)(F)F)CC1)NCCOCCNC(=O)CCc1ccncc1 51369,CC1CN(C(=O)CN(C(=O)C(C)Cn2cccn2)C2CC2)CCN1C1CC1 51370,N1(C(c2onc(CNC(C3(C)C(C)C3)=O)n2)=O)CCC(C)(CCO)CC1 51371,c1(C(=O)NCC2(C)CCN(C(CN(S(CC)(=O)=O)C)=O)C2)ccc2snnc2c1 51372,N1(C(C(CCC)N(C)C)=O)CC(N(C(=O)C=Cc2cccnc2)C)C2(CC2)C1 51373,N1(C(c2cc(COC)cs2)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)C(C2CC2)C1 51374,C12(C(=O)NCC=CCNC(c3c(C)occ3)=O)COCC(C1)C2 51375,C(C(CC(C)C)C(=O)N1CCC(C)(C)C(O)C1)NC(COCCC=C)=O 51376,CCC(C)CCC(=O)NC1(CNC(=O)CCS(C)=O)CCCCC1 51377,C(=O)(C(C)CC(F)(F)F)N1CC(CC(=O)NCC(CC(=CC2CCC2)C)(C)C)C1 51378,C12(NC(CCc3onc(CC)n3)=O)CCC(CC1NC(c1oncc1C)=O)C2 51379,NS(=O)(=O)c1cc(NC(=O)Nc2ccc3c(c2)CC(=O)NC3)c(F)c(Br)c1 51380,c1(CNCCOCC(=O)OCC)cnc(COc2ccccc2)s1 51381,c1(CCC)cnnc(C(=O)NCCCCN(C(=O)CC2(CO)CC2)C)c1 51382,N1(C(c2c(C)scc2)=O)CCN(C2CCCN(C(=O)CSCCN(C)C)C2)C(=O)C1 51383,c1(OC)cc(NCC(C)CNC(=O)C(=O)NCC2CC2)ncn1 51384,c1(C(=O)NC2(CNC(C34CCCCC3C4)=O)CCC2)c[nH]c2nccc(Cl)c12 51385,C(c1ncc(C)[nH]1)=CC(=O)NC1CC(F)(CNC(C2N(CC)CC2)=O)C1 51386,C(=O)(CCC(=O)N1CCC(CCNC(=O)CNC(=O)C(C)(C)C)CC1)OC 51387,C1(NC(C=CCN(C)C)=O)CN(C(=O)CC2CC(C)(C)CO2)CC1C 51388,C(C)(C)(C(=O)NC1CC(NC(=O)Cc2ccnn2C(C)(C)C)C1)N(CCC)CCC 51389,CCCCC(C(=O)N1CCN(C(c2cnc(Cl)c(N)c2)=O)CC1CC)NC(N)=O 51390,c1(C(=O)NCCN(C(=O)C(CO)NC(N)=O)CC)cnn2cccc(Cl)c12 51391,N1(C(C2=C(C)CC2)=O)C(CC(N2CC3CCCCC23)=O)C2CCCC12 51392,c1(OC)nc(C)ncc1-c1nc(CCSc2ccc(F)cc2)no1 51393,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51394,c1(CNC(c2ccn(CCNC(CC3C(C)(C)C3)=O)c2)=O)csc(C#N)c1 51395,N1(c2n(CC)c(-c3coc(CC4CCC4)c3)nn2)CCN(C)C2(CCOC2)C1 51396,C=CCC(Cc1ccccc1)C(=O)NC1CC(CC(=O)NC)C(O)C1O 51397,c1(NC2CCC(C)(CN)C2)ccc(S(=O)(=O)NC(=O)CCC2CCCC2)cn1 51398,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)CSCc2c(C)noc2C)C(CO)C1 51399,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51400,S(=O)(=O)(c1ccc(F)cc1)C(N(CC(N)=O)Cc1cn(C(C)C)nn1)=O 51401,C1(NC(=O)C=C2CCCC2)CC(NC(c2cc(F)cc(F)c2)=O)C12CCC2 51402,C(C(=O)N(C(C)CCNC(=O)C(C)Sc1ccccc1)C)(C(C)C)NC(C)=O 51403,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3ccco3)CCC2)C(=O)C1C 51404,C#CCCCCC(=O)NC1CCC(N(C)C(c2ccnnc2OC)=O)CC1 51405,N1(CC)CC(C(=O)NC2CCCN(CC(=O)NC3CSCN3C)CC2)CCC1=O 51406,N1(C(CCCC=C)=O)CC2CCN(C(c3nc(C)oc3OC)=O)CC2C1 51407,C(C(C)(C)C(F)F)NC(C(C)NC(=O)C=Cc1ccccc1)=O 51408,c1(C(CC)N)ccc2ccccc2c1.c1(C2N(CC)CCC2)ccc(C(=O)O)s1 51409,N1(C(c2c(C)n(C)cc2)=O)CCC2(CCN(C(=O)C(C)CO)C2)C1 51410,N1(C(C(C)=C2CC2)=O)CCC(CNC(=O)C(C)CCc2ccccc2F)C12CCC2 51411,c1(OC)ncccc1CCNC(C1(n2cccn2)CC1)=O 51412,c1(C(=O)NC(C2CCCCC2)CNC(CC(C)SC)=O)cc2n(n1)CCCN2 51413,c1(C(=O)NC2C(CNC(COC3(C)CCOCC3)=O)CC2)ccc2snnc2c1 51414,C(c1ncccc1C)=CC(=O)NCCN(C(=O)C=CC(=O)NC1CC1)CCC 51415,Cc1cc(CC(=O)NCC(C2CC2)NC(c2nc(C(C)(F)F)cs2)=O)c(C)o1 51416,C1(NC(C(C=C)O)=O)COC2(C1)CN(C(c1cnc(C(C)C)[nH]1)=O)C2 51417,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)SC)CC(C)C 51418,CC(C)(C(=O)NCCC1CCCN(C(=O)COCC(F)(F)F)C1)C(F)(F)F 51419,C(N=c1ncc(C(F)F)c[nH]1)C1CCC(NC(CC(C)SC)=O)CC1 51420,N1(C(C(C(CC)O)(F)F)=O)CC2CCCC(N(C(=O)C(COC)OC)C)C2C1 51421,c1(C(=O)NCCC(CCNC(CC(CC)O)=O)C)coc2cc(F)cc(F)c12 51422,c1(OC)ncnc(OC)c1CN1CCCC1CC(=O)Nc1sccc1C 51423,CN1CCN(C(=O)CCCNC(=O)CCCc2ccc(F)cc2F)CC1CO 51424,CCCCCC(=O)NCC1CCCC1NC(c1cccn1Cc1ccccc1)=O 51425,C1(C(N(CC)Cc2ccc(C)cc2)=O)CCCN(C(=O)CCN2CCOC2=O)C1C 51426,CC(CC(=O)N1CC(C)C1C(=O)N=c1ccn(C)[nH]1)CC(C)(C)C 51427,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51428,c1(OC)cccc2c(C(N3CC(NC(C4CC4C(C)(C)C)=O)C(C)C3)=O)coc12 51429,C1(C(N(CCCNC(c2ccc(CC3CC3)s2)=O)CC)=O)CCCCCN1C 51430,C1(NC(c2c(C)ccs2)=O)CCCCN(Cc2cnc(C(F)(F)F)s2)C1 51431,C1(NC(c2c(CC)n[nH]c2)=O)CC2(CNC(=O)CCC3CCOCC3)CC1CO2 51432,C(=O)(C(C)C(F)(F)F)N1C(C(=O)NC(CCCCC)C)CCC1 51433,N#Cc1cc(C(=O)NC2CC(CNC(c3scnc3Br)=O)C2)co1 51434,c1(C(N2CC(NC(C3CCC4(C3)N=N4)=O)C2)=O)cccc(Br)c1F 51435,C(=O)(C1=CCC(F)(F)CC1)N1CCC(C2(NC(c3cc(C)no3)=O)CC2)C1 51436,C#CCCC(=O)NCCn1ccc(C(=O)NC2CCN(CCC)C2)c1 51437,C1(CNC(CNC(=O)OCC)=O)CC(NC(c2cc(CO)c[nH]2)=O)C1(C)C 51438,c1(NC(=O)Nc2nnc(SC3C(C=C)OCC3)n2C)c(OC)cccc1C 51439,c1(CCOC)c(O)nc(=O)n(CC)c1N.C12CCCN(C1)CCCC(=O)NCC2 51440,C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(N(C(C=CC(C)(C)SC)=O)C)C1 51441,C1(C(=O)NCC(C)(C)NC(C2CC3(CC3)CO2)=O)CCS(=O)(=O)C1(C)C 51442,N1(C(CCOCCOC)=O)CCOC2(CCN(C(C3(C)CCOC3)=O)C2)C1 51443,C(C(F)(C(=O)NCCC1CCCCO1)C(C)C)NC(c1c(C)nsc1C)=O 51444,CCC(CCC(=O)NC1CC2(C1)CC2C(=O)N(C)CCOC)OC 51445,N1(C(c2scnc2C(F)(F)F)=O)CCC2CCC(C1)N2C(=O)CC1CCSC1 51446,C12(NC(=O)Cn3nccn3)CCC(C1)N(C(=O)Cc1ccncc1)C2 51447,C1(CN(C)C)CCCN(C(=O)C(F)(F)CO)C1.C12CCC(O1)CNC2=O 51448,CON1CC(C(=O)NCC2(O)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O 51449,C1(CNC(CCOCCOCC)=O)(CC(C)C(N)=O)CCC(F)(F)C1.C(=O)(C=CCO)N 51450,c1(C(=O)NC2C(CNC(COc3ccc(OC)cc3)=O)CC2)cnc(Cl)c(N)c1 51451,C1(NC(C2CCS(=O)(=O)C2)=O)CN(C(=O)CCc2ccc(O)nc2)CCC1F 51452,c1(C(N2CCC(C)C2c2cn(-c3cc(C)ns3)nn2)=O)nn(C)cc1Cl 51453,c1(NC(C2CCN(C(c3n[nH]c(CC)c3F)=O)CC2)=O)ncc(C)cc1Br 51454,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51455,c1(C(C(=O)NCC)N(C)Cc2ncc(-c3ccccc3)o2)cc2n(n1)CCC2 51456,CCCC(CC)C(=O)NC(CC(=O)NCC1(C#N)CCC1)C(C)OC 51457,n1(C(C(C)C)C)nc(C2CSC2)nc1CC1CCC(O)C1 51458,c1(Nc2ccc(-n3ccc(C(=O)OCC)n3)cc2)cc(F)cc(O)c1 51459,Cc1cnn(CCC(=O)NCC(O)CNC(c2csc(Cl)c2)=O)c1 51460,C12(C(=O)NC(C(C)NC(c3cncn3C)=O)C)CC(CCO1)C2 51461,C1(NC(C(c2cnn(C)c2)OC)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51462,c1(OC)cccc(CCC(=O)NCC(C)CNC(=O)C(C)C(F)(F)F)c1F 51463,C12(NC(CC(CCC)O)=O)CC3CC(C1)CC(CNC(=O)C(C)C(=O)OC)(C3)C2 51464,c1(C(=O)NCCN(C(=O)CCCC2CC2C)CC)ccc2c(c1)CCOC2 51465,c1(CC(N2CC3CC(NC(C4(COC5CC5)CC4)=O)C2C3)=O)c(Cl)cccc1Cl 51466,Cc1[nH]ccc1C(=O)NC1CCC(NC(C2OCCCO2)=O)C1 51467,c1(C(CN(C(=O)C=CCOC(C)(C)C)C)NC(C(C)=C(CC)C)=O)ccccc1 51468,N1(C(c2nc(C)nn2C)=O)CCC2(CC1)CC2CNC(=O)CC(C)c1cccnc1 51469,C=C=CC(C)C(=O)NCC(C)C(=O)NCCCN(CC(C)C)C 51470,CC(C)CCCC(C)OC(C1CN(C(=O)CSc2cccnc2)C(=O)O1)=O 51471,C1(NC(c2cc(C3(CC)CC3)on2)=O)CC2CC(NC(=O)Cn3cccn3)CC12 51472,c1(CC(=O)NC23CC2CN(C(c2ccoc2)=O)C3)nnc(O)nc1O 51473,Cc1ccc(O)cc1C(N1CCC(NC(=O)C=C2CCN(C)C2)C(F)C1)=O 51474,C#CC1(C(=O)NCCSc2n[nH]c(C)n2)CCN(C(=O)CNC(=O)CC(C)C)CC1 51475,c1(C(N2CC(CC(=O)NCc3n(CC)ncn3)C2)=O)cc2cccnc2[nH]1 51476,N1(C(c2ccc(C)nc2)=O)CCC2C(CCCN2C(c2c[nH]cc2C(C)C)=O)C1 51477,c1(C(N(CC)Cc2cccs2)=O)nc2c(o1)CCSC2.C12(C)CCN(CC1)C2 51478,c1(C(=O)NC)c(C)[nH]c2ccc(C(=O)OC)cc12.C12C(C1C1CC1)CNC(=O)C2 51479,CCC(CC(=O)N1CC(C)(OCC(=O)NC2C(C)CC2(C)C)C1)CC(C)C 51480,N1(C(C2(C3CCCO3)CCC2)=O)CC(NC(c2ccn(CC)n2)=O)CC(F)C1.C=CC 51481,Cc1cnccc1C(C)Cc1cc(C(F)(F)F)n[nH]1.C12CC3(C1)CC3NC(=O)N2 51482,C#Cc1cccc(NC(C2CCOCC2COC)=O)c1.C12(CC1)CC(=O)N2 51483,c1(C(N2CC(CN(C)C(C3CCCS3)=O)C2)=O)csc2nccn12 51484,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CCCF 51485,C1(CC(=O)OC)(C(=O)OCc2nncc(OC)c2)CCC(C)(C)C1 51486,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(=O)CCc2nncn2C)CC(C)(C)C1 51487,C(C(C)(C(=O)N1CCC(CO)CC1)NC(C1CCCN1C(C)=O)=O)SC 51488,c1(NC(c2cnn(C(CC)C)c2C2CC2)=O)nc2ccc(Br)cn2c1F 51489,C(CC(C)C)(C(=O)N(CCC(=O)NC1CCC(C)(C)C1)C(C)C)NC(C)=O 51490,C1(CC)CN(C(C2(F)CCN(C(=O)CNC(N)=O)CC2)=O)CCN1C 51491,C12(C(N(CCC)CC3CC3)=O)CC(CN(C(=O)CCc3nc(C)no3)C1)C2 51492,N1(C(CCNC(C2OCCN(C)C2=O)=O)=O)CCC(=C(F)F)CC1 51493,C=CCCC(C(=O)NCc1ccccc1F)NC(c1cn(C)nc1OC)=O 51494,Nc1ccc(C(=O)NCC(=O)NCCC2CCCN2C(C2C3CCCC23)=O)cc1 51495,Cc1ncnc(N2CC(OC(F)F)(NC(=O)CC3(C(F)(F)F)CC3)C2)c1Br 51496,c1(C(N2C(CNC(C3C=CCS3)=O)CC2)=O)ccc2[nH]ccc2c1 51497,N(C(=NCC(C)C)N1CCC(n2cccn2)C1)C(c1ccccn1)C#C 51498,c1(C(=O)NCC(CC)NC(C2(C)CCNC2=O)=O)c(C)nc2ccccc2c1C 51499,c1(OC)cncc(C(=O)NC2CN(C(=O)CC(C)SC)CC2SC)n1 51500,C(=O)(CC(C)CNC(C1CCOC1NC(=O)C(C)C#N)=O)OCC 51501,N1(CC(N2CC(SC)C(NC(=O)CNS(=O)(=O)N(C)C)C2)=O)CCC(=O)NC1=O 51502,N1(C(c2c(C)ncs2)=O)CCN(C(C2CC3COCCN3C2)=O)C2COCC12 51503,C(C(C(C)C(C)C)NC(=O)CCn1cc(Cl)cn1)NC(C=C(CCC)C)=O 51504,C1(CC(=O)N(C2CCN(C(c3cnc4n3CCS4)=O)C2)C)CN2CCC1CC2 51505,n1(CC(=O)NCCN(C(C2CCC(=O)C2)=O)CC)c(C)c(C)sc1=O 51506,C1(CC)CCCN(CC(=O)N(CC(C)(C)CNC(C2CCC(C)(C)C2)=O)CC)C1 51507,C12(C(=O)NCC3CC(CNc4nccc(OC)n4)OC3)CC3CC(CC(C3)C1)C2 51508,CC(N=c1[nH]c(=NCc2cc(Cl)ccc2F)[nH]c2ccsc12)c1ncccc1F 51509,CCC(CC)C(=O)NCc1nnn(C)c1C(N1CCCCC1CC)=O 51510,C1(C(=O)NOCC2N(C(CCC(=O)NCC)=O)CCCC2)C2(CCC2)C12CCC2 51511,C(=O)(C(C(C)(C)O)NC(c1c[nH]c(=S)cn1)=O)N(C)Cc1ccccc1F 51512,n1(CC)nc(C)cc1C(=O)NC(C)C(C)(C)NC(C1CN(C)C1)=O 51513,C1(N(C(Cn2c(C)ccc2C)=O)C)CCN(C(C2CC(=C(F)F)C2)=O)CC1C 51514,N(C1CCCn2nccc21)C(C(C)(C1CC1)NC(C(c1ccccc1)OC)=O)=O 51515,c1(C(=O)NCC(CNC(C(C)OCC#C)=O)OC)cc(Cl)c(Br)cc1C 51516,C(=O)(CC1=CCOCC1)NCCC(=C)CNC(C1CC(C)OC(C)C1)=O 51517,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C2CCN(SC(F)(F)F)C2=O)C1 51518,N1(CC(=O)Nc2ccncc2)CC2CCN(C(c3cc4ncccc4[nH]3)=O)C2C1 51519,N1(C(C(c2ccoc2)NC(C(F)=CCC)=O)=O)CCN(CCO)CC1 51520,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)CSCC(F)(F)F)OC 51521,C(C(C(=O)Nc1cnn(CCF)c1)C(C)C)NC(c1c(C)n[nH]c1C)=O 51522,c1(N(C)C)ncc(Br)c(C(=O)OC2CN(C(=O)OC(C)(C)C)CC2C)n1 51523,N1(C(C(N2CCNC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51524,c1(C(N2C(C(=O)OCCC#C)CCCC2)=O)cc(C)cc(F)c1 51525,Cc1nc(CCC(=O)NCCC(C)(C)NC(c2coc(C(N)=O)c2)=O)[nH]c1C 51526,CC1(C)CCC(c2nnnn2C2CC(F)(F)C2)(NC2CC2CCOCCO)C1 51527,N1(C(C(C)(C)C2CCCCO2)=O)CCC12CN(C(c1ccns1)=O)C2 51528,C1(C(=O)NC2(CNc3c(C(=O)OC)ncs3)CC2)CCC(C2CC2)C1 51529,C1(C(N2CC(C(C)(C)O)(CNC(CCC(=O)NCC)=O)C2)=O)COC2CCCCC12 51530,N1(Cc2n(-c3c(C)cncc3)c(-c3cc[nH]n3)nn2)CCCC(O)(C2CC2)C1 51531,c1(C(CN(C(C)CNC=O)C)=O)ccc(CN2CCSCC2)cc1.c1(S)cnc[nH]1 51532,N1(C(C2N(C(=O)CCc3ccc[nH]3)CC=CC2)=O)CCCC(O)(CO)C1 51533,c1(OC)c(C)ccc(C(=O)NC2COCCC2NC(=O)CCc2cnoc2)c1F 51534,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(c3cn(C)cn3)=O)CC4)n21 51535,C1(CC=C)(NC(C2CCCN(CC)C2)=O)CCCN(C(=O)Cc2ccnn2C)C1 51536,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(=O)Cc1coc(C)n1)C2 51537,c1(C(c2n(CCC)nnn2)NCc2conc2COC)ccccc1OC1CC1 51538,c1(C(=O)NCCN(C(C(CCSC)O)=O)C2CC2)cccc2c1CCCN2 51539,S(=O)(=O)(c1ccc2c(=O)ccoc2c1)NC(c1cccc(CC)c1)C 51540,c1(C(=O)NC(CCOC)CNC(=O)Cc2cc(C)ns2)nccc2cc[nH]c12 51541,C1(CNC(=O)Cc2cccnc2)CN(C(=O)CCc2ccccc2O)CC1(F)F 51542,c1(CN(C(=O)C(N2CCCC2c2ccsc2)=O)C)cccc(Br)c1 51543,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51544,Cc1ccc(CCC(=O)N(C)CC2CCCN2C(c2cc(C)c(C)o2)=O)cc1 51545,N1(C(CCCCCCC)=O)CCN(C(c2cc(C3CC3)sn2)=O)CC2(CC2)C1 51546,CCC(CCC(=O)OCCSN)N(C)C 51547,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51548,C1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CCOC)CCC=CCCC1 51549,Cc1cccc(C(=O)NC(CNC(=O)C(N2CCOCC2=O)C)C(C)C)c1F 51550,c1(NC(C2OCCN(C(CC3(OC)CCCC3)=O)C2)=O)ccc(C)nc1C 51551,c1(C(N(C(CCO)C(F)F)C)=O)cc(=O)c2cc(C(=O)O)ccc2o1 51552,Cc1csc(C(N2CCCCC2CCN(C(=O)CC(C)F)C)=O)c1C 51553,CC(N=c1nn[nH]n1C)C1CCCCN1C(c1c(Cl)cnn1C)=O 51554,N1(C(c2c(CC)csc2)=O)CC2CC(C1)C2NC(c1cc(Cl)cs1)=O 51555,N1(C(C(C=C=C)C)=O)CCC(CC(=O)N(CC(C2CCCC2)O)C)C1(C)C 51556,CCC(CC(=O)NCC1CCC(CNC(=O)C=CC2CCCN2C)CC1)SC 51557,CN1CCC(NC(=O)C(N2CCNC(=O)C2CCF)=O)C(c2cnn(C)c2)C1 51558,N1(CCC(C)C)CC(C(C)C)C(O)C1.C1(C)(C)CNC(=O)N1 51559,C1(C(=O)NCCCCC2CN(C(C3(CC#C)CC3)=O)C2)CC2(CCCCC2)CO1 51560,c1(OC)ccsc1C(=O)NCC1CCCC1C(=O)NOCC(O)CO 51561,c1(C(N2CCC(NC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51562,c1(C(=O)NC2C(C)CCN(C(=O)CNC(=O)CN(C)C)C2)cc2ccccn2n1 51563,C1(NC(c2cc(C#N)no2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(O)C1 51564,C=CCC(CC(F)F)C(=O)N1CC(N2CCN(C(=O)C3=C(C)OCCC3)CC2)C1 51565,c1(C(=O)NCCNC(C=CC(C)(C)SC)=O)nccnc1O 51566,CC1CC(C(N2CCN(C(=O)CN(c3ncccn3)C)CC2)=O)CC(=O)N1 51567,N1(C(CC(C)(C)OC)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51568,C1(NC(C2CCC(CC)O2)=O)CCC2(CC1)CCN(C(C1C=CCC1)=O)C2 51569,c1(C(=O)NCCC(CNC(CC(COC)COC)=O)O)ncc2ccccn12 51570,CC1(C(N2CC3(CCC3NC(=O)Cc3ccccc3F)C2)=O)CCCCCC1 51571,CC(C)C(N=[N+]=[N-])C(=O)N1CSCC1C(=O)NC1CC2CC1CC2(C)O 51572,C1(C(=O)NCC2OCCN(C)C2)CC2(CO1)CN(C(=O)C(F)(F)C(F)(F)F)C2 51573,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1C(=O)NC1(C(O)C(F)(F)F)CC1 51574,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(C)O)CCCOC 51575,C=CCN=c1ccc(S(=O)(=O)N2CCCCC2c2ncc[nH]2)c[nH]1 51576,N1(C(c2cc(OC)nn2C)=O)CC(NC(=O)C(C)OC)CC1(C)C 51577,C1(CC(=O)NC(c2nccs2)CC)(CNC(=O)CC2(C)CCCC2)CCCCC1 51578,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC12CC(I)(C1)C2 51579,CCCCS(=O)(=O)CC(=O)NCC(CO)NC(c1csc(C)n1)=O 51580,Cc1ccc(C)c(C(=O)NC2CCCC2(C)NC(=O)CCCC2CC2C)n1 51581,C(=O)(C1=CS(=O)CCC1)NC1CN(C(c2ccc(CC)cc2N)=O)C(C)CC1 51582,N1(C(Cc2ccc(C)c(C)c2)=O)CC(CNC(c2nsnc2O)=O)C2(CCC2)C1 51583,C1(NC(c2nccc(C)c2)=O)CCN(Cc2cnc(C)nc2)CC1O 51584,C(C(=O)N(C)CCN(C(C1CCOC1C)=O)C(C)C)(C(C)(C)C)OC 51585,N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51586,c1(C(N(C2CCN(C(=O)C(C)N3CCC3)CC2)CCC)=O)cnc(C)nc1.C1CC1 51587,C(C(C)(C1CC1)NC(=O)CNS(C)(=O)=O)NC(COC(CC)C)=O 51588,c1(COC)csc(C(C(=O)NCC(F)F)N(C)Cc2ccsc2)c1 51589,Cc1cc(C)n(CCNC(=O)C(=O)Nc2cccnc2OC(F)(F)F)n1 51590,c1(-n2cc(C3N(C(C4C(C(C)C)CCC4)=O)CCC3)nn2)ncccc1O 51591,C1(NC(C=C(C)C(C)(C)C)=O)CC(F)(F)CC1NC(=O)CS(=O)(=O)NC(C)(C)C 51592,Cc1cc(CNC(=O)NCC(c2ccccc2Cl)O)ccc1-c1ccncc1 51593,C#CC1CC2CCC1N(C(=O)C(CC1CC1)NC(c1cnn(C(F)F)c1)=O)C2 51594,Cc1nsc(C(c2nnnn2CCN2CCOCC2)NC(C)CCc2ccco2)n1 51595,C1(CC)(CO)CCCN(C(=O)C(C)Oc2ccccc2)C1.C(=O)(CCO)NC.O 51596,C1(NC(CS(=O)(=O)NCC)=O)CN(CC2(C)CCC(=O)N2C)Cc2nccn2C1 51597,c1(CC)nc(C)c(C(=O)NC(C)CCNC(C2CC(O)C2CC2(C3CC3)CC2)=O)s1 51598,C(C1COc2ccccc21)NC(NC(C#C)CCc1ccc(C)cc1)=NCCF 51599,C(=O)(CC(=O)N=c1cc(-c2ccc3c(c2)OCO3)o[nH]1)NC1C(C)OC(C)C1C 51600,c1(NC(c2cc(C)c(C)c(C)c2)=O)ccc2c(c1)CC(c1ccccc1)OC2=O 51601,CCCC(C)(CCC)C(=O)N1CCC(NCNC(C2(CO)CC2)=O)C(COC)C1 51602,C1(C(=O)NC2CC(CNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51603,N1(C(=O)C=Cc2ccco2)CCCC2(NC(C3CC(O)C3)=O)CC2C1 51604,C(=O)(CCC(C)COCC)N(CCOCCNC(CCC=CC)=O)C 51605,N1(C(C(C)NC(CN(C(C)C)C)=O)=O)CCC(N(C)C)C(C)C1 51606,c1(OC)cnc(Cl)[nH]c1=NC1CC2CN(Cc3ccc(F)c(F)c3)CC12 51607,c1(C(N2CC(F)(C(=O)NCC3(CCO)CCC3)C2)=O)ncccc1Cl 51608,c1(C(=O)NC2CC2C(N2CC(=O)NC(C(=O)OC)C2)=O)c(Br)c(OC)nn1C.CC 51609,C1(CNC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CSCCS2)=O)CC1O 51610,c1(C(=O)NC2CC(CCNC(=O)C(Cl)=CCl)C2)cccc(C(F)(F)F)n1 51611,C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)ccc(Cl)c2)=O)CC(F)C1 51612,c1(CCNC(=O)NC2(C(F)F)CCC2)ccc2c(c1)OCCO2 51613,C1(CN(C(=O)CN2CCOCC2)CC)CCCN1C(=O)C(F)=C1CCC1 51614,N1(C(=O)Cc2cccc(O)c2)CCC(F)(F)C(CNC(=O)CCF)C1 51615,N1(C(C=NOC)=O)CCC(N(CCO)C(C2CC2OC(C)(C)C)=O)CC1 51616,CCC(C(=O)N1CCCC(O)(CNC(c2cnccn2)=O)C1)C(C)(C)CC 51617,CC1(C=CC(=O)N(C2CCCN(C(=O)CC3CC34CC4)C2)CCF)CCOCC1 51618,S(=O)(=O)(CCCC(F)F)NC(CC#C)C 51619,C(=O)(C(C)C(O)CCCC)N1CC(C#C)(C(=O)N(C2CC3(CCC3)C2)C)C1 51620,C(=O)(C(F)(CNC(c1coc(C(C)C)n1)=O)C(C)C)N(CCC)CC 51621,C1(CNC(C(CC)C2CCC2)=O)CCC2(CN(C(=O)CCC3CCC(C)O3)C2)O1 51622,c1(-n2c(C(C)Oc3cnn(C)c3)nc(-c3cccs3)n2)ccc(Cl)c(Cl)c1 51623,CCC(CC)C(C(=O)NC1(C(=O)NCC(C)CC2CC2)CSC1)OC 51624,C(N=c1[nH]cnc(Cl)c1F)C1CN(C(c2nc(CC(C)C)sc2)=O)CC1(C)C 51625,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)Cc3ncccn3)ccnc2[nH]1 51626,CC1CCCN(C(=O)C(=O)NC2(C)CN(C(=O)C3=CCCS3)C2)C1CO.C(C)(C)(C)O 51627,CCC(CC)CCC(=O)NC(C1CCCN(C(C2(CO)CC2)=O)C1)C 51628,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)CO)C3)=O)cccn12 51629,C1(C(C(=O)NC(c2cccnc2)C(=O)NCC2(C)CC2)C)CCOCC1 51630,c1(OC(C)C)cncc(C(=O)NCCCC(C)(C)NC(c2ccco2)=O)c1 51631,c1(OC)cc(Cl)c(Br)cc1CN=c1[nH]c(-c2cccnc2C)cs1 51632,c1(C(=O)NC2CCCCC2Nc2ncnc3scnc23)cc2c(nc1O)CCOC2 51633,N12CCC3(CCCC13)C2=O.c1(CC(=O)NC(C2(CO)CC2)C)cnoc1 51634,C(c1ccnn1C)=CC(=O)N(C(C(=O)NCc1n(CC)ncc1)C1(C)CC1)C 51635,c1(C(N)=O)ccc(C(=O)NCC2(F)CN(C(=O)CCc3ccco3)C2)o1 51636,CCCC(C(=O)N1CC2C(CNC(C3C4CC5C(C4)C35)=O)C2C1)NC(C)=O 51637,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51638,N1(C(C2N(CC)CCC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51639,C1(NC(c2cc(OC)nn2C)=O)CN(C(C2CCCCC2O)=O)CCC1CO 51640,CC1CCN(C(c2ccccc2CO)=O)CC1NC(c1ccc(Br)o1)=O 51641,c1(CN(C)C(=O)NCc2cncc(Cl)c2)nc2c(s1)CCCC2 51642,c1(SC)ccc(C(=O)NC(C2CCN(C(C3(C)CC3)=O)C2)C)cc1[N+](=O)[O-] 51643,c1(C(N2CCSC2c2ccc(Cl)s2)=O)cccnc1NC(=O)Cn1cccc1 51644,CC1CCCCN1C(=O)COC1CCOC1.C(=O)(CCn1cccn1)NC(N)=O 51645,C12(C(N3CCCC(CNC(=O)CCC4CCCCCC4)C3)=O)CCCC1C2(F)F 51646,n1(C(C)C(N2CCCC(Cc3ccccc3)CC2)=O)cc(C#N)c(O)nc1=O 51647,C(=O)(C(C)(C)C(C1CCCCC1)NC(C1CC(=O)N(c2cnn(C)c2)C1)=O)OC 51648,Cc1c(C(=O)NCC2CC(CNC(=O)CN(C)C)CO2)sc2ccc(F)cc12 51649,C(=O)(C(C)(C)C(=O)N1CCCC1CNC(=O)Cn1ncccc1=O)OCC 51650,C1(NC(C2C=CCC2)=O)CC2CCC1N(C(c1ccccc1-c1nc[nH]n1)=O)C2 51651,C1(F)(C(=O)NCC2(CNC(C(N3C(=O)CCC3=O)CC)=O)CC2)CC2(CCC2)C1 51652,c1(CC(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)ccc2nsnc2c1 51653,c1(C(=O)NCC(CN(C(CC(CCC)C)=O)C)O)cccc2nncn12 51654,N1(C(C(CC=C)(C)C)=O)CCN(C(=O)Cc2ccccc2C(C)C)CC(O)C1 51655,CC1(C)CCC=C1C(=O)NCCCNC(=O)Cn1ccc(=O)n(C2CC2)c1=O 51656,C(=O)(CC1COc2cc(O)ccc21)NS(CC)(=O)=O.C1CCNCCN1C(C)C 51657,Cc1nc(N2CCC(NC(=O)C(C3CC3)C3CC3)CC2C)cc(C#N)n1 51658,c1ccc2c(c1)OCCO2.C1(NCC=C)C2CN(C(=O)C(OCC)OCC)CC12 51659,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(C2C=CC=CC=C2)=O)CC1 51660,c1(NC(=O)CCCCN(C(=O)CCOC2CC2)CCO)c[nH]c2ncccc12 51661,c1(CNC(C(C)=C(C)C)=O)cc(OC2CCN(C(C3CCCO3)=O)C2)ccn1 51662,N1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCCCCC(N=c2cnc(F)c[nH]2)C1 51663,CCCCCC(O)C(=O)N1CC(C2CN(C(=O)C(F)CC)C2)C1 51664,N1(C(CC(C)(F)F)=O)CCOC2(CCN(C(c3sccc3C(F)F)=O)CC2)C1 51665,c1(C(N2CCC3(C(NC(c4nn(CC)c(C)c4)=O)C3)C2)=O)cn2ccccc2n1 51666,N1(C(C=CC(C)(C)C)=O)CCN(C2CCC(NC(=O)C(F)C3CCC3)CC2)CC1 51667,CCC(O)CC(=O)NCC1CCC(NC(=O)C(C)(C)C2(C)CC2(F)F)CC1 51668,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 51669,c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc2cnsc2c1 51670,N1(CC(C)NC(=O)CCc2ccc(C3CC3)cc2)CCN(C(=O)C=CCO)CC1 51671,c1(C(=O)NCC2(O)CN(C(C3(C)CC=C(C)CC3)=O)C2)cc2cn[nH]c2cn1 51672,C(=O)(C1CCCc2scnc21)NCC1N(C(COC(CC)C)=O)CCN(C)C1 51673,CC(C)(CO)C(=O)NC(C1CCN(C(C2CCCCS2)=O)CC1)CO 51674,N1(C(c2c(C(C)C)n[nH]c2)=O)CC(NC(C2CCC2CF)=O)C(O)C1 51675,C1(n2cc(CCCCNC(c3ccc(C=C)cc3)=O)nn2)CCn2nccc2C1 51676,C1(COC)(CNC(=O)C(C)n2cccn2)CCCN1C(C1CC(CCO)C1)=O 51677,N1(C(Cc2scc(CC)c2)=O)CC(C2(NC(=O)CCn3ccc(O)nc3=O)CC2)C1 51678,CC1CCOCC1C(=O)NCc1cccc(C(=O)NC2(CO)CCC2C)n1 51679,C=CC1(CC(=O)NC2(C)CCCC2NC(=O)C(C(=O)OC)OC)CCOCC1 51680,C1(C(N2CC(N(C(=O)CCCCCF)C)C(O)C2)=O)(COC)CCCNS1(=O)=O 51681,C1(C2(O)CCC2)(C(=O)NC2C(CNC(c3cnc(CC(C)C)[nH]3)=O)C2)CC1 51682,n1(CC(=O)NC(c2ncc(-c3ccccc3)s2)C)cc(CN(C)C)nn1 51683,c1(-c2cn(CC(N3C(c4n(C)ccc4)CCC3)=O)nn2)ncccc1C(=O)O 51684,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 51685,N1(C(c2c(CC)ccs2)=O)CCC(NC(=O)CN(c2ccccc2)CC)C(CO)CC1 51686,C(C(=O)C(C1(CCN)CC1)=O)(C1CCCC1)OC.C(C(C)O)N(C=O)C 51687,N1(C(c2c(C)c[nH]n2)=O)CCC(O)C(C(=O)NCc2ccccn2)C1 51688,c1(OC)ncc(CCNC(=O)C(C2CCC(=O)N2)C)s1 51689,Cc1cc(CC(=O)NC23CCCN(C(=O)CCn4cccn4)C2C3)ccc1F 51690,c1(C(C)(C)N(CCOCCn2cc(COC)nn2)C)ccc2c(c1)OCO2 51691,N1(C(CCC(=O)NC)=O)CCN(C)C(CNC(c2ncc(-c3ccccc3)s2)=O)C1 51692,c1(C(N(C2CCCC(N(C)C(c3ccoc3)=O)C2)C)=O)ccc2ccn(C)c2c1 51693,c1(OC)cc(CNC(c2ccc(-c3ccnn3C)cn2)=O)ncc1C 51694,c1(C(=O)NC2CCC(NC(=O)C(F)=CC3CC3)CC2)cc2c(cn1)OCCC2 51695,N1(C(CC)=O)CC2CCC(NC(=O)C(C)Oc3ccc(Cl)cc3Br)(C2)C1 51696,C1(C(=O)NCC(C)(C2CC2)NC(c2n[nH]cc2Cl)=O)CCN(CCF)CC1 51697,C1(NC(=O)CCCN2C(=O)CNC2=O)CC2CC(C1)N(C(c1nccs1)=O)C2 51698,C(C(O)CCNC(C1(n2nccn2)CC1)=O)NC(=O)C=CC(=O)NC1CC1 51699,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 51700,N1(C(c2ccn(CC)n2)=O)CCC(N(C(=O)C2=CCC2)C)C2(CC2)C1 51701,CC1CN(C(c2ccc(F)cc2F)=O)CCC1CNC(C1(C)C=CCCC1)=O 51702,C1(CNC(C(C)NC(N)=O)=O)CN(C(C2CC(F)(F)C2)=O)CCC1(C)C 51703,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2ccc(OC)nn2)=O)C2(CCC2)C1 51704,C=C(C)C(O)CC(=O)NC1CN(C(=O)Cc2cc(OC)ccc2F)CC1C 51705,CN1CCCC1(C)C(=O)NCC(O)C(=O)NCCCC1(O)CCC1 51706,Cc1ncc(C(N2CCC(C(C)C(=O)NCCSCCO)C2)=O)n1C 51707,Cc1cc(Cl)ncc1CC(=O)NC1CCC(F)(CNC(C2(N(C)C)CC2)=O)C1 51708,CC1(NC(=O)CNC(=O)C(F)C2CC(NC(C3CCSCC3)=O)C2)CCCC1 51709,C(C(CC(C)C)NC(=O)CC1CCC(C(C)(C)C)CC1)NC(CCCOC)=O 51710,c1(-c2nc(C(CC=C)C)n(CC(C)CO)n2)ccc(C)c(F)c1 51711,C=C=CCC(=O)N1CCC(C(C)C(=O)N(CCC)CC)C1 51712,c1(C(=O)NC)nccc2ccncc12.c1(C(N2CCC(N)C2)=O)nnn2c1COCC2 51713,c1(OCCN2C(NC(C3(C)CCOC3)=O)CC2)cccc(F)n1 51714,Cc1nc(C(N2CC3CC2C3CNC(C2CC(O)CN2C)=O)=O)ccc1[N+](=O)[O-] 51715,CCC(F)(F)C(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1 51716,c1(C(=O)NC2CCN(C(=O)C3=CCCCO3)CC2F)cc(Cl)cc([N+](=O)[O-])c1 51717,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)Nc2cccc(F)c2)C1 51718,C1(C(=O)NCC2N(C(c3ncc(CC)cn3)=O)CCC2C)CCn2nccc2C1 51719,C(=O)(C1=NOC2COCC12)NC(C(C)C)CCNC(C1CC(n2cnnc2)C1)=O 51720,C1(C(=O)OCC(C=C)(F)F)CC2(CCO2)C1 51721,N1(C(C(C)CC2CCCC2)=O)CCCCC(NC(c2cc(C(N)=O)ccn2)=O)C1 51722,c1(C(C(=O)NCC(=O)NCC2(S(C)=O)CC2)(C)C)ccc(O)cc1 51723,C1(CC(=O)NC(c2c(C)nns2)C)CC2(CC2)CN1C(c1nnn(C)c1N)=O 51724,C(=O)(C(C)(O)C(C)(C)C)N1CC2CC(CNC(C(CC)CCOC)=O)C2C1 51725,c1(C(N(C(CC)C(=O)N2CC(C)(CF)C2)C)=O)cc(=O)cc[nH]1 51726,C1(C(=O)NCCSC(C)C)CCCN(C(=O)CC(O)CSc2ccccc2)C1 51727,C1(NC(c2nc(CNC(C(C)C3CCOC3)=O)oc2)=O)CC2CCC1(CO)C2 51728,CN=c1cc(C(N2CCC(N(CCO)CCO)CC2)=O)cc[nH]1 51729,CC(C)(COc1ccccc1)C(=O)NC1CN(C(c2cccc(OCCF)n2)=O)C1 51730,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCN2CCCC2)ccc2c[nH]nc2c1 51731,c1(C(=O)NCC(CC=C)C(=O)NC2CN(C)CCC2O)coc2ccccc12 51732,C1(C(=O)NC2CC(N(C(c3n(CC)cc(Cl)c3)=O)C)C2)CCOC(C)(C(C)C)C1 51733,N12CCC(C)(CC1)C2=O.Cc1cncc(-c2cn(-c3cn(C)nc3C(F)F)nn2)c1 51734,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 51735,c1(OCCC)ccc(C(=O)NC2(CO)CCOC2)cc1OC 51736,c1(C(N2CCCC(O)(CNC(C(=O)NCC)=O)C2)=O)cnc2cc(OC)ccn12 51737,C1(C(=O)NCC(CCOC)NC(=O)Cc2ccc(N)cn2)CCc2nn[nH]c2C1 51738,c12sc3nccnc3c1NCCN(C1CC1)C2=O.C1(C)(C=O)CC1.CCO 51739,C(=O)(CCC1CCOc2ccccc21)NCC(C)CNC(c1cn(C)nc1O)=O 51740,C1(NC(C2CN(C(C)(C)C)C(=O)C2)=O)CN(C(c2cncc(Cl)c2)=O)CCC1F 51741,C(=O)(C1CCc2ccccc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C#C)CC2CC2)C1 51742,N1(CC)CCOCC1C(=O)NCCCCC(C)NC(=O)C(C)c1cccs1 51743,C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)C(CO)N(C)C)C(C)(C)C1 51744,CC1OCCCC1C(=O)NC1CCC(CNC(c2cc(Cl)ccn2)=O)CC1 51745,C(c1ccccc1)=CC(N1CC(CCCCNC(CC2C(C(C)=O)C2(C)C)=O)C1)=O 51746,C(=O)(C(O)C(C)(C)C)N1CCC(O)(C(N(CCCCCSC)C2CCCC2O)=O)C1 51747,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(C2CC2)C2CC2)C1 51748,C(=O)(C1=CCCOCC1)N1CC(CCOC)N(C(c2nc(C)ccc2F)=O)CC1 51749,CC1(C)CCC=C1C(=O)N1CCCCC1CNC(c1cn2cnnc2cn1)=O 51750,C(CC(F)(F)F)N(C(=O)CCC1CCC(NC(=O)CN2CCCCC2)C1)CC 51751,Cc1cccc(C(N2CCC(C(c3ccccc3)NC(c3ccon3)=O)CC2)C)c1 51752,c1(N(C(=O)Cc2ccc(CNSS(C)(=O)=O)cc2)CC)c(F)cc([N+](=O)[O-])cc1F 51753,c1(N2CCC(C=C)C2)ncnc(NC)c1C.c12ccccc1C(=O)N(CCCO)C2 51754,c1(CNC(c2n(CCCC)nnn2)(C)CCOCC2CC2)cc(C)cc(F)c1 51755,C1(NC(c2cnn[nH]2)=O)CN(C(=O)COC(F)(F)F)C2CCCCC12 51756,c1(C(C)C)[nH]nc(C(=O)NCCCNC(C2CC(C)CO2)=O)c1[N+](=O)[O-] 51757,c1(NC(CN(CC(=O)NCCCn2c(C)ncc2)C)C)ccc(C#N)cc1 51758,CC1CN(C(=O)C(C2CCOCC2)F)CC1(C)C(=O)NC1CC2(CCCO2)C1 51759,C1(CNC(Cc2c(C)nsc2)=O)CN(C(c2ccc(C(=O)OC)nc2)=O)CC1C 51760,CC(CCNC(=O)C(N1CCN2CC(C)CC2C1)=O)C(F)(F)C(F)(F)F 51761,c1(C(N)=O)cscc1C(=O)NCC1CCN1C(c1cncs1)=O 51762,c1(C(N(CCC)CCNC(C2(CC)CNC(=O)C2)=O)=O)cc2cscc2s1 51763,CC1CN(C(=O)C(C2CCOCC2)C)CC(C)N1C(c1ncncc1Cl)=O 51764,c1(C(=O)NCC2(C)CCC(NC(c3cccnc3Cl)=O)C2)cncc([N+](=O)[O-])c1 51765,C1(C(=O)NCC(CN(C(C2CCC(C(=O)OC)C2)=O)C)(C)C)Cc2nncn2C1 51766,C1(NC(c2n[nH]cc2Cl)=O)CCCCCN(C(c2cccc(C(F)F)c2)=O)C1 51767,c1(C(N2CC3C(N(C(c4cc(C)c(Br)s4)=O)C)C3C2)=O)c(C)[nH]c(C)c1C 51768,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 51769,C=CCN=C(NCc1cccc(C(=O)OCC)c1)NCc1cnccc1C 51770,c1(C(N2CCN(C(COCCC#C)=O)C(C(C)C)C2)=O)cc(Cl)cc2c1CCC2 51771,c1(C(N(CCCCCNC(C(CC=C)CC)=O)C)=O)ccc2c(c1)nc(C)n2C 51772,CN1C2CCC1CC(CC(=O)NCCOCCCNC(=O)CC1(C)CCOC1)C2 51773,C1(c2cncc(Cl)c2)(C(=O)OC)CCN(C(c2cc(C(F)F)cs2)=O)C1 51774,c1(C(=O)NC(C2(CCNC(COC(CC)C)=O)CCC2)C)nccnc1C 51775,C1(NC(CN2CC(C)(C)C2)=O)CCN(C(=O)CSc2nc[nH]n2)CCC1CO 51776,CCC(C(=O)OC)C(=O)NOCC(N1CC(CN(C)CC)C1)=O 51777,C(C1CCN(C(c2nccn2C2CC2)=O)CC1)=CC(=O)NCc1c(C)cnn1C 51778,c1(CNC(c2cnc(C)cn2)c2n(C(CC)(C)C)nnn2)nc(C)c(C)[nH]1 51779,CN1CCN(C(C2CC(F)(CO)C2)=O)CC1CNC(C1CSCCS1)=O 51780,N#CC1CCC(CNC(=O)C(CC(F)F)NC(=O)CCOCC(F)F)CC1 51781,C1(C(=O)NC2CC3(C2)CC3NC(CCC(=C)Cl)=O)(OC)CCCC(C)(C)C1 51782,c1(NCCNC(=O)NC2CCOCC2F)ccc(Cl)cc1 51783,N1(C(c2nc(C(=O)NCc3ccc(Br)cc3)sc2)=O)CC2CCC1CO2 51784,c1(CNC(=O)CCCCF)cnn2c1CN(C(C1CC(OC3CC3)C1)=O)CC2 51785,C(CC(C)(C)C(=O)N1CCCC(N(C(=O)C(O)C(C)C)C)C1)SC 51786,N1(C(c2cc(OC)ncc2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)CC1 51787,CN1CCN(C(C2CC(Cc3ncnn3C)C2)=O)C(C(=O)N(C)CC2CC2)C1 51788,N1(C(Cn2ccc(C)n2)=O)CC2(CC(NC(=O)CCCC(N)=O)CO2)C1 51789,Cc1cc(C(F)(F)F)sc1C(=O)NC1CCC(N(C(=O)CCF)C)C1 51790,C(C)(C(C)C(=O)NC(C)C)NC(C1(CCN2CC(SC)C2)CCC1)=O 51791,C(CC(C(C)(C)C)NC(c1ncccc1Cl)=O)N(C)C(c1cc(F)ccc1F)=O 51792,C1(C(=O)NC2C(C)C2(C)C)(NC(C=C(C)C2CC2)=O)CCCCC1 51793,C=CC1(C(N2CCCC(C)C2CCO)=O)CCN(C(c2c[nH]nc2CC)=O)C1 51794,C1(C(=O)Nc2n(COC)ncc2)(OC)CCN(C(=O)CN(C2CCCC2)C)C1 51795,N1(C(C2N(C(c3ccc(CC)o3)=O)CC(=O)NC2)=O)CCOC2CN(C)CC12 51796,O1NC(=O)CN=C2NC(=NCC(C)(C)C(C)(F)F)NC1=CC=C(Cl)C=C2.CCOCC 51797,CC(C)(C)C(CO)C(=O)NC1CCN(C(=O)CCCCCO)C1 51798,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 51799,c12ncccc1CNC(=O)C2C(=O)C1CC1.C1(C(OC)OC)(CSC)CCCC1 51800,CC(O)C(C(=O)NCC1(NC(c2csc(-c3cn[nH]c3)n2)=O)CCCCC1)N(C)C 51801,c1(C(N2CC3(CN(C(C)=O)C3)C2)=O)cc2cc[nH]c(=O)c2s1 51802,N1(C(C2(COC)CCC(=O)N2)=O)CCCN(C(C2CCN(OC)CC2)=O)C(C)C1 51803,c1(OC)c(Cl)cc(C(=O)NCC2CCN(C(=O)CC3CCCCO3)C2)cc1Cl 51804,CC1CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(c1cncs1)=O 51805,C(=O)(CC(F)(F)C(F)F)N1CCN(CCNC(CN(C2CCSC2)C)=O)CC1 51806,C1(CNC(C2CCC(CC)CC2)=O)CC(C)(C)CN1C(c1nc(C)oc1C)=O 51807,C1(C(N2CC(CC)C(NC(=O)Cc3cnns3)C2)=O)CN2CCCN1CC2 51808,C(N=c1cc[nH]cc1S(=O)(=O)NC1CN(C(C)(C)C2CC2)C1)C1CCC(C)O1 51809,c1(C(N(CCN(C(C2(CCC)CC2)=O)C)C)=O)nc(O)c(C)s1 51810,CCS(=O)(=O)CC(C)N(C(c1ccccc1)C1CCCCC1)CC1CCCCC1 51811,c1(NC(C2CCC(N3CCN(Cc4ccc[nH]4)CC3)CC2)=O)ccc(F)cc1 51812,c1(C(=O)NCC(CO)NC(=O)Cn2cc(C3CCC3)nn2)cc(CO)ccc1F 51813,Cc1nc(NC(=O)CC2CN(C(c3ccnc(Br)c3Cl)=O)CCO2)ccc1F 51814,c1(C(C(=O)N(CC(C)NC(=O)CC2CCC(=O)N2)CC)C)ccc(C(C)=O)cc1 51815,C1(N(C(c2c(C)nc(COC)o2)=O)C)CCN(C(=O)CC=C(C)C)CC1C 51816,c1(CC)cccc(C(N2CCOCC2CCNC(c2ncccc2F)=O)=O)c1N 51817,C1(C(N2CC(CC(C)NC(C=Cc3scc(C)n3)=O)C2)=O)CCCCN1N=O 51818,CCC(C(=O)N1CCC(C)(NC(c2ccoc2Cl)=O)C1)C(F)(F)F 51819,C12(NC(C3CC3c3cccs3)=O)CC(CNC(c3cnn[nH]3)=O)(C1)C2 51820,OC1CN(Cc2ccc(F)c(Br)c2)CCC1(F)F 51821,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 51822,c1(C(=O)N)sccc1NC(c1csc(C)n1)=O.C1(CC(=O)NC)(COC)CC1 51823,c1(C(C)NC(COC2CCN(C(c3c(C)noc3)=O)C2)=O)ccc(C)nc1 51824,CC1CCC(C)(NC(c2cccc(CNC(=O)CC3OCCC3C)n2)=O)C1 51825,c1(SC)ncc(CN2CCC(C(=O)Nc3nc(C(C)=O)cs3)C2)c(Cl)n1 51826,C1(CNC(C(C(CC)O)C)=O)CC2(CCC2)CN1C(=O)CC1(N2CCCC2)CC1 51827,c1(C(=O)NC2CC(CCNC(C3C(C)CCO3)=O)C2)cnn2ccccc12 51828,C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ncc3Cl)=O)C2)CCC2C1C2(F)F 51829,C1(C(=O)NCc2cc(CC)no2)CCN(C(=O)C2CC(N=[N+]=[N-])C2)O1 51830,N1(C(CCc2cc(C)no2)=O)CC2CCN(C(C34CCCC3C4(F)F)=O)CC12 51831,C1(c2n(C)cnn2)CCCN(C(=O)CN2C(=O)CC2=O)C1 51832,CC1(C)CCC(C(=O)O)C(C(=O)NCC23COCCC2C3)C1 51833,Cc1cc(C(N2CC3CC3C2C(N2CC3C(CO)C3C2)=O)=O)ncn1 51834,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 51835,n1(C(C)C)cnc2ccc(NC(=O)NCc3cccc4nc(Cl)ccc34)cc2c1=O 51836,c1(OC)ccc(I)c(CNC2CCC(C(N3CC(O)CC3C)=O)CC2)c1 51837,C1(NC(C(C2CC2)OC)=O)CCC(N(C)C(c2nnn(C)c2N)=O)CC1 51838,Cc1sc(O)nc1C(=O)NCC1C=CCN1C(=O)CCN1CCOCC1 51839,C(=O)(C1=CCC(C)(C)CC1)NC1(C(=O)NCC2(CCO)CCCC2)C(C)CCC1 51840,N1(C(CC2(OC)CCC2)=O)CCC2(CCC2)C(NC(C2(S(N)(=O)=O)CC2)=O)C1 51841,c1(CNC(C2(CO)CC(CNC(C3CC34CCOC4)=O)C2)=O)cnccc1Cl 51842,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 51843,c1(NC(=O)CCN2CCCCCC2)nc(-c2ccccc2)ncc1Br 51844,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 51845,C1(CC(=O)N(CC(C)NC(=O)Cc2cccc(N)c2N)C)CC2CCC(C1)C2 51846,c1(C(C2CC2)NC(C(=O)NC2C(C)C2C)=O)cccc(S(C)(=O)=O)c1 51847,CCC(CN=c1cccc(S(=O)(=O)NCC(CSCC)OC)[nH]1)OC 51848,N1(C(c2cc(C)ns2)=O)CCC(C)(C(N2CCC(F)CC2)=O)C1 51849,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 51850,c1(OC)nc(C(=O)NC(C2CCCCC2)CNC(=O)C(C)(C)CF)sc1C 51851,c1(CNC(CC)=O)nnn(C)c1C(=O)NC(COC)C(=O)OC 51852,c1(C(=O)NC2CCN(Cc3c(O)cccc3Br)C2)ccc(O)c([N+](=O)[O-])c1 51853,C1(CC(N2CCC(NC(CCOC)=O)C2)=O)CCCC(C)C1 51854,N1(C(=O)Cc2cnsc2)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC2C1 51855,c1(CC)ccc(C(=O)NCC(O)CNC(=O)COCCc2ccccc2)o1 51856,N1(C(Cc2ccc(CSCC)cc2)=O)CCC(O)C(NC(=O)CC(C)C(F)F)C1 51857,N1(C(CS(CC)=O)=O)CCC2(CC1)CC(NC(c1cnc(O)cc1C)=O)CO2 51858,C12(NC(C3(OC)CS(=O)(=O)C3)=O)CCCC(CN(C(=O)C(C)OC(C)=O)C1)C2 51859,C1(C(=O)NCC(=O)NCC=C)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 51860,C(=O)(CC(F)(F)F)N1CC(CC(CN(C2CCS(=O)(=O)C2)C)O)C1.C1C(=O)N1 51861,n1(CC)ccc(=NC(c2nc(C(=O)O)c(C)s2)c2nnnn2C2CCC2)[nH]1 51862,C1(C(N(CCN(C)C(C2CN3CCC2CC3)=O)C)=O)CCC2CC1C2(C)C 51863,CC1(C)COC(CCC(=O)NCCC2(O)CN(C(c3cc(O)cs3)=O)C2)C1 51864,c1(C(=O)OC)cccc(OCC(=O)NC2CCCC2NC(C2(C)CC2C)=O)c1 51865,CC1(C)COCC(NC(C23CC2CN(Cc2ccc(F)cc2)C3)=O)C1 51866,N1(C(c2nc(COC)sc2)=O)CCOCC1CC(=O)NCC1(C#N)CCCC1 51867,N1(CC(=O)NC2CN(C(CCCC#C)=O)CC2O)C(=O)NC(C)(CC)C1=O 51868,c1(OC)ncccc1C(=O)NCC1CC(NC(C2CC2C)=O)C1.C1(O)CCCCC1C 51869,N1(C(COCCCOC)=O)CC(O)CC1(C)CNC(=O)CSc1nnnn1C 51870,C1(C(=O)NCC2(CC(C)C)CCC2)CCOCCN1C(=O)CCN1CCOCC1 51871,C1(C(N2CC(C)(c3cn(-c4ccncc4)nn3)C2)=O)CC12CCCCC2 51872,N1(CC(C)CC(F)F)CC(=O)N(CCn2ccnn2)C1=O 51873,N1(C(CN(C(Cc2c(C)ccnc2)=O)C(C)C)=O)CCC2CCN(C)C2C1 51874,N1(C(C(CC#C)(C)C)=O)CCC(CNC(C2CC2=C)=O)C(F)(F)C1 51875,Cc1cc(-c2cn(C3CCN(CCCc4nnc(C)n4C)CC3)nn2)ccc1O 51876,C(=O)(C(C)(C)C(=O)NCc1c(Br)cnc(Cl)c1F)N(C)C 51877,CCCCC(CN=c1[nH]cnc(Cl)c1Br)NC(=O)C1CCc2cccnc21 51878,C(=O)(C(C)(O)CC(C)C)N1CCCC(F)(CO)C1.c1(N)cc(O)nc(O)c1 51879,CCCCCCC(=O)N(C)CC1CN(C(C2CC3(c4ccccc4)CC2C3)=O)C1 51880,C1(C(NOCC=C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 51881,C(=O)(CC(C)CC(F)(F)F)NCCC1N(C(c2nc(C)[nH]n2)=O)CCOC1 51882,c1(C(=O)NCC2CCN(C(C(C)CF)=O)C2)cnnc2ccccc12 51883,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 51884,Cc1ccc(N)c(C(N2CC(NC(c3cnn(CCO)c3C)=O)C3(CC3)C2)=O)c1 51885,N1(C(C(C)OCC(C)C)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CCC1C 51886,CCC(C)CC(C(=O)N1CCCC1CN(C)CC)NC(c1cccn1C)=O 51887,C(CC(C(=O)OC(C)(C)C)N1CCCC1CNC(=O)Oc1ccccc1)SC 51888,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 51889,CC1(C(=O)NC2CCCN(Cc3ccccn3)C2)CCCN(CCCl)C1 51890,c1(C(=O)NCc2occ(C(N(C)CC3C(C)OCC3)=O)n2)cc2ccccn2c1 51891,c1(C(C(=O)NCC)NC(CSCCc2nncs2)=O)cnn(C)c1 51892,CN1CC2CC1CN2C(C1CC(NC(c2ncn3c2CCC3)=O)C1(C)C)=O 51893,c1(C(c2nnnn2C2CC2)Nc2nccc(OC)c2C#N)ccc2c[nH]nc2c1 51894,C(=O)(C(O)CC(=O)OC(C)(C)C)NCC(C)(C)NC(=O)CC1CCCO1 51895,CN1CCC(CCNC(=O)CC2CNC(=O)O2)C1=O.C12CCCCC1C(=O)N2 51896,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)CCCn2cccn2)C2COCC12 51897,N1(C(C=C(C)c2ccccc2F)=O)CCNCCC12CCC2 51898,N1(C(C(C)n2cccc2)=O)CCCCC(C2CN(C(=O)CCC(C)(C)C)C2)C1 51899,C1(NC(c2c(OC)cccn2)=O)CCN(C(C2CC(O)C2)=O)CC1F 51900,Cc1cc2nc(N3CCC(NC(c4cnn[nH]4)=O)C3)cc(=O)n2o1 51901,c1(C(C(=O)NCC(CC=C)NC(=O)CCCOC)C)ccc(C(F)(F)F)cc1 51902,C1(C(C)C)CCCC1CC(=O)NCCCC(C)NC(=O)CCc1ccsc1 51903,N1(C(C(CC)(C)COC)=O)CCC(C2CCN(C(=O)C3=C(C)OCC3)CC2)CC1 51904,Cn1c(I)cc2c(N(C3CNCC3O)C(c3c(F)cc(Br)cc3Br)=O)ncnc12 51905,N1(C(c2nc(=O)o[nH]2)=O)CCC2C(C1)OCCN2Cc1cncs1 51906,C=CC1CN(C(c2ccc(OCCOC)cc2)=O)CC1NC(=O)CC1CC(=C)C1 51907,c1(C(N2CCCC(CNC(c3n(CC)c(O)nc3)=O)C2)=O)coc2ccccc12 51908,c1(C(=O)NCCN(C(C(CC=CC)C)=O)C)cc(OC)cc2ccoc12 51909,CC(C)(CC(=O)N1CCC(C2CCCCC2)C1)c1cn(CCCF)nn1 51910,C1(CC(=O)NCc2cc[nH]c2C(=O)NCC(c2ccccc2)O)CC(C2CC2)C1 51911,N1(C(c2c(OC)scc2)=O)CCC(NC(=O)CN(c2ccccc2)C)C(CO)C1 51912,C(=O)(CS(=O)(=O)C1CC1)N1C(N(CCC)CCCC)CCC1.C(=O)OCC 51913,CC(C)(CNC(=O)C1CC1)CC(=O)N1CCC(C#N)C1 51914,N1(C(CCN(C)C)=O)CCCCC(CNC(C2CNC(=O)N2)=O)C1 51915,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 51916,N1(C(N2CCC(C)=C(C)C2)=O)CC2(CCC2)CC1C=O.CCC1=NOCC1 51917,C1(NC(C(CC=C)CNC(C2(O)CCC(C)CC2)=O)=O)C2CCN(CC2)C1C 51918,C1(CNC(c2cc(CNC(C=CCC)=O)sc2)=O)CN(CC)C(=O)O1 51919,N1(C(Cc2n(C)ccn2)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 51920,CN1CCC(C(=O)NC2(CCNC(C3CCS(=O)(=O)N3)=O)CC2)c2ccccc21 51921,c1(C(=O)NCC2C(NC(c3c(N)c(F)ccc3)=O)C2)cccc2c1OC(F)(F)O2 51922,C(=O)(CC1=NNC(=O)C1)NCCOCCCNC(C1C(C(C)C)CCC1)=O 51923,C1(NC(CC)CN)CCCN(c2ccc(C)cc2)C1.C(=O)(N(CC)CC)NCC.C 51924,C1(c2onc(C)n2)CCCCN1C(C(=O)NC(C)(C)C)C1CC1C 51925,c1(C(N2CC3C(NC(C4N(CC)CCC4)=O)C2C3)=O)cc(OC)cc2c1CCC2 51926,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 51927,Cc1cccc(C(N2CCCC(CNc3nccnc3C#N)C2)=O)c1Cl 51928,C1(CCCNC(CCCOC(C)C)=O)CCN(C(=O)CC2CCOC2)CC1 51929,CCC(C)CC(C)NC(=O)CNC(C1(NC(=O)CN(C)CC)CC1)=O 51930,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)NCC=Cc3ccco3)C2)c1 51931,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 51932,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 51933,c1(C(=O)NC2C(NC(C3(CC)CCNC3=O)=O)CCCC2)cnc(Cl)cc1N 51934,C12(C(N3CCC(CNC(c4cnn(C(C)C)n4)=O)CC3)=O)CC1Cc1c[nH]nc12 51935,CCCCC(C)CCC(=O)NC(Cc1cnn(C)c1O)C(=O)N(CCCN=[N+]=[N-])C 51936,c1(COCC)nc(-c2cc(Cl)c(Cl)s2)n(C2CC(C(C)(C)C)C2)n1 51937,c1(SC)cccc(NCC2(NC(c3occc3Br)=O)CC2)c1[N+](=O)[O-] 51938,C1(C)(NC(C(CNC(CC(=O)OCC)=O)(F)C(C)C)=O)CN2CCC1CC2 51939,N1(C(=O)C=Cc2cn[nH]c2)CC2CCN(C(c3nc(C(F)(F)F)cs3)=O)C2C1 51940,C(=O)(CC(F)(F)C(F)F)NC(CC(C)C)CNC(c1cn(C)[nH]c1=N)=O 51941,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 51942,CCC(C)C(O)CC(=O)NC(C)(C)CCCNC(c1ccnc2ccsc12)=O 51943,O=C1CCCC(C(N2CCC(CCC(=O)NCC(c3ccccn3)O)C2)=O)C1 51944,C(CCO)(C(=O)NCCC1CCN(C)C1=O)NC(CN1C(C)CCC1)=O 51945,C(CCC(C)C)(C(=O)NC1CN(C)CC1C)NC(COCCCOC)=O 51946,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 51947,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 51948,c1(OC)cccc(N(C(c2cn(C)cn2)C(=O)OC2CCCCC2)C2CCC2)c1 51949,Cc1ncc(C#N)c(NC(C2CC3CC3N2C(C2CCC(=O)N2)=O)=O)n1 51950,C(CC(F)F)(C(=O)NC1COCCC1O)NC(C1CCC(=C)CC1)=O 51951,C1(C(N2C(CNC(CNS(CC)(=O)=O)=O)CC2)=O)CSCN1C(=O)C(C)(C)C 51952,N1(C(Cc2cc(OC)no2)=O)C2CCC(C2)C1CNC(c1cc(CO)ccc1F)=O 51953,C(c1cncn1C)=CC(=O)NC1CC(CNC(CSCCC)=O)C1 51954,CC(C)CCC(=O)NC1CCN(C(C2CC(n3ccnc3)C2)=O)C1 51955,n1(CC(N2CC(CC(C)NC(C3CC(C)(F)C3)=O)C2)=O)cccc(O)c1=O 51956,CCC(CN(C)C)CC(=O)NC(C)(CN(C)C)C(=O)N(C(C)C)CC 51957,CC1C2CC(C2NC(=O)OC(C)(C)C)N1Cc1c[nH]cc1-c1ccccc1 51958,C1(CNC(C2CCCCS2(=O)=O)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1O 51959,C1(C(=O)NCCCN(C(C(C2CC2)SC)=O)C2CC2)CC(O)C(F)C1 51960,N1(C(C(F)=C(C)C)=O)CCN(C(c2cccc(Cn3cccn3)c2)=O)CC1C 51961,N1(C(c2cc(C)ns2)C(=O)N(C)C)CCCC(C)(Oc2ccc(F)cc2)C1 51962,C1(C(=O)NC2CCCC(N(C(=O)C=CCF)C)C2)CC2(CCC2=O)C1 51963,C(=O)(C#CC1CCCCC1)N(C)CC1(N(C(=O)CC2C(C)(C)C2(C)C)C2CC2)CC1 51964,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(C1(n2cccn2)CCC1)=O)CO 51965,c1(CC)cnn(CC(=O)NC2(CC(=O)NCC(C)C)CCC2)c1.C1CC(=O)N1 51966,N1(C(C2CCOC2)=O)CCN(C(=O)CC2CC2)C2COCC12 51967,CCC(CC)C(C)C(=O)N(CCNC(=O)Cc1ccccn1)Cc1ccccc1 51968,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CC2CCC(=O)N2)CC1)[N+](=O)[O-] 51969,C1(COC(c2c(O)c(Cl)ccc2)=O)CCC2(CCC3(CC2)OCCO3)O1 51970,C=CC1(C(=O)N(C)Cc2cscn2)CCN(C(c2cc(CCO)on2)=O)C1 51971,N=c1cc(C(N2CCC(F)(CNC(C3CC3c3cccc(Cl)c3)=O)C2)=O)cc[nH]1 51972,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 51973,CC(CC(=O)c1ccco1)C(=O)NC1CCC(N(C(=O)CN(C)C)C)C1 51974,c1(CC)nc(C(=O)NCCCC2CCCCN2C(C2COCCO2)=O)c(N)s1 51975,c1(CNC(C(COC)NC(=O)CC2COCC2O)=O)cc(C)ccc1O 51976,N1(C(=O)COC2CC=CC2)CCOCC(CNC(=O)C=Cc2ccccc2)C1 51977,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2C)=O)c(Cl)c1 51978,C1(NC(CN(C2CCC(NC(CCC)=O)CC2)C)=O)CCn2ccnc2C1 51979,C1(F)(C(N2CCN(C(c3cc(Br)cnc3Br)=O)C3C2C3)=O)CCCCC1(F)F 51980,N1(C(CCC=CC)=O)CC(C)CCC1CNC(=O)CCc1cn(C)cn1 51981,C1(NC(c2ccncc2F)=O)CCCC12CN(C(c1sccc1F)=O)C2 51982,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 51983,N1(C(Cc2nnc(C)o2)=O)CC2CC(C)N(C(=O)Nc3c(C)cccc3C)C2C1 51984,CC1(C(N2CCC(N3CCC(NC(=O)CCC4CCC4)C3)CC2)=O)CC(C#N)C1 51985,C(=O)(C(C)(C)S(C)(=O)=O)NCC1CC(NC(C(c2c(OC)ccc(F)c2)=O)=O)C1 51986,C1(C)(COC(c2cc(OC)n(C)n2)=O)CCCN(C(c2cccc(OC)c2)=O)C1 51987,C(C(C)(C)C(=O)N)SCCOC(C)(C)C.C12(C=O)CC(C(=O)OC(C)(C)C)C1C2 51988,c1(CN(C)CCn2cnnn2)ncccc1Cl 51989,CC(C)CC(CNC(C1OCCCO1)=O)NC(c1cnoc1C1CCOCC1)=O 51990,N1(C(CN(C(C)=O)C)=O)CC2CC(C1)CN(C(=O)C(c1ccc(F)c(F)c1)O)C2 51991,c1(CC)cccnc1C(=O)NCC1C=CC(NC(=O)CC2CCSCC2)C1 51992,O=C(C(=O)N=c1ccn(C(F)(F)F)[nH]1)NCCCOCC1CCC1 51993,n1(C(C)C)cc(C(F)(F)F)c2ccccc12.c12cccc(c1C(=O)O)C(=O)N2 51994,c1(C(CN(C)C(C2CCSC2)=O)F)ccccc1F 51995,C12C(C1(C)C)CNC2=O.C(=O)(C(=O)NCCF)NC(c1nn[nH]n1)C 51996,c1(OC)cc(C)c2cc(C(=O)NC(C)CNC(c3cnn4c3OCC4)=O)[nH]c2c1 51997,CC1CC(C)N(C(c2cnn(CCF)c2)=O)CCN1C(c1nccc(N)c1Cl)=O 51998,n1(C(=O)NC2C(CC3CC(CNC(=O)CSC(F)F)C3)C2)nnc2c1CCCC2 51999,N1(C(COC)=O)CC(NC(c2ccc(-c3ccsc3)cc2)=O)C(SC)C1 52000,C12(C(N3CCC(F)(CNC(CCCC=C)=O)C3)=O)CC3CC(CC(C3)O1)C2 52001,O=C(C#CC1CCC1)NC1CC(C(=O)NCC(O)C2(O)CCC2)C12CCC2 52002,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52003,c1(C(=O)NCC(C2CCCC2)NC(C(N2C(=O)CCC2=O)C)=O)ccncc1F 52004,N1(C(Cc2ncc(C)s2)=O)CC2(CCN(C(=O)NC3CC(C(C)C)=NO3)CC2)C1 52005,C1(NC(C2(CC)CCN(C(c3n(CC)ccc3)=O)C2)=O)CCCC1C1CC1 52006,C1(CCNC(c2c(CC)nc[nH]2)=O)CC(F)(F)CN1C(=O)C=CC(=O)N(C)C 52007,c1(CNS(=O)(=O)CCc2cc(Br)cc(Br)c2)cc(F)c(Cl)cc1Cl 52008,CC(C)C(COC(=O)CCc1ccccc1)n1cncn1 52009,c1(C(N2C(CNC(c3coc(Cl)c3)=O)CC(F)(F)C2)=O)cn2c(n1)CCCC2 52010,C1(NC(=NC)NCC(C)Cc2cnn(C)c2)CCS(=O)(=O)CC1 52011,c1(OC)cc(C2CC2)ccc1C(=O)N(C1CN(C(=O)CCOC)C1)CCO 52012,N1(C(COCC(=O)OC)=O)CC2(CCC2NC(=O)C(F)C2CCC2)C1 52013,CC(C(=O)N(C)C)NCCC1(C(F)F)CCC1 52014,C12CCOCCN1C2.c1(C(F)(F)F)cccnc1Br 52015,c1(N2CCCC(CN(C(CCc3ccc(C)s3)=O)C)C2)ncnc(Cl)c1CO 52016,C(CCC(C)C(C(=O)NCCN1CCOCC1)N(C(CC(C)C)C(=O)OC)C)=CC 52017,c1(OC)ncc(-c2cnn(CCF)c2)cc1C(=O)NCCC#N.N1CCC(O)C(C)C1 52018,CCC(C)(C)CCCC(=O)NC(C)CC(=O)Nc1ccc(F)cc1 52019,N1(C(=O)CCn2ccnn2)CCCC(C2CN(C(c3cn(CCO)nn3)=O)C2)C1 52020,C(=O)(C1=CCC(C)CC1)NCC1CCN(CC)C1.C12CCC(CC1)CN(C)C2=O 52021,n1(C(C(=O)NC(CC)CNC(=O)CC2CC3(CC3)CO2)C)nc([N+](=O)[O-])cc1C 52022,c1(OC(C)C(N2CCC(CNC(C3C=CCCC3)=O)C2)=O)cccc(F)c1 52023,c1(C(=O)NC2C3(CC(NC(C(CC=C)C)=O)C3)C2)cnc2sc(C)cn12 52024,C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCCN(C(C(=O)OC)c1cncs1)CCF 52025,c1(C(N2CC(NC(C3CC4(C3)CC4F)=O)CC(C)C2)=O)cccc2cccnc12 52026,c1(C(N2CCC(C(C)NC(=O)CC3OCCCO3)CC2)=O)n[nH]c2c1NCCC2 52027,S(=O)(=O)(c1ccc2[nH]c(=NCCCCC(N)=O)sc2c1)NC1(COC)CC=CCC1 52028,c1(C(N2CC(CNC(c3ccc[n+]([O-])c3)=O)OCC2)=O)cc2[nH]ccc2cn1 52029,C=CC1CN(C(=O)Nc2c(C3CC3)nn(C)c2C2CC2)CC1O 52030,C#CCCC(O)C(=O)NC1(CCC)CCCN(C(=O)CNc2cnn(C)c2)C1 52031,C1(C(=O)NCCCOC(C)=O)CCCC1NC(=O)C(C)CC1CCC1 52032,c1(C(N2CC(NC(Cc3c(C)noc3)=O)C(C)C2)=O)cnc2sccc2c1 52033,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52034,C1(NC(Cn2c(C)cnc2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52035,C(=O)(CCCC(=O)N1CC(N(C(=O)C(CC)NC(N)=O)C)C(O)C1)OCC 52036,N1(C(=O)OC(C)(C)C)CCN(C(c2cc(C)c(N)cn2)=O)c2ccc(Cl)cc21 52037,N1(Cc2nc(C(C)OC)sc2)CCN(C(c2ccnc(N(C)C)c2)=O)CC1 52038,C1(C)(C(=O)NCC(C2(O)CCN(C(C(C)(C)OC(C)=O)=O)C2)C)CCCN(C)C1 52039,N1(C(CC(CN(C)C)O)=O)CC=C(C(=O)N2CCCC(N(C)C)CC2)CC1 52040,N1(C(c2ccc(NC)cc2)=O)CC2CCCC2C1C(=O)NCc1ccon1 52041,c1(NC(C)=O)ccc(NC(C2CCCN(C(c3ccncc3O)=O)C2)=O)cc1 52042,c1(COC(CNC(=O)NC(C)CCCl)(C)C)cnn(C)c1 52043,C1(C(=O)NCc2c(C(=O)NC(Cn3ncc(C)c3)C)scc2)CC2CCCC2C1 52044,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52045,C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(NC(c2cc(F)c(F)cc2O)=O)C1 52046,c1(OC)ccc(C(=O)N(CCCN(C)C(c2ccc(F)s2)=O)C)cc1OCCO 52047,N1(C(=O)C#CC2CC2)CCCC2(CC(C(=O)N3CCc4ccc(Cl)nc4C3)=NO2)C1 52048,c1(C(=O)NCC(CNC(C(=O)N(C)C)=O)CO)c(Cl)ccc(Br)c1F 52049,c1(C(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2C)ccn2ccnc2n1 52050,Cc1ccc(C(N2CCCC2CN(C(=O)CNC=O)C)=O)nn1.c1(C=O)cccs1 52051,C(=O)(CCCCCC(C)(C)C)NC1CN(C(c2c(C)oc(Cl)n2)=O)CC1C(F)F 52052,C1(CNC(c2nc(C(N)=O)sc2)=O)CC(F)CN1C(C1CC(N2CCOCC2)C1)=O 52053,N1(C(C(=O)NCCC)C)CCN(C(C2CC(F)CN2C)=O)CC1 52054,CC1(C)CN(C(c2csc(C(F)F)c2)=O)CC(C)(C)C1NC(C1CCC1(F)F)=O 52055,C#CC1CCCCN1C(C1CC(=C)CCN1C(C1CC2(C1)CC(O)C2)=O)=O 52056,C(=O)(CC1=CCOCC1)NC(CC(=O)NCC1(CCO)CCC1)C(F)F 52057,N1(C(CC2(CC)CC2)=O)CCC(O)(C(C)NC(C2CCCC(O)C2)=O)CC1 52058,N1(C(C(Cc2cnc[nH]2)NC(c2ccc(C(C)=O)[nH]2)=O)=O)CCC(C)(F)C1 52059,C=CCC(C)(C)CC(=O)N(CCNC(C1CC2CC1OC2)=O)Cc1ccccc1 52060,C(c1ccccn1)=C(C)C(=O)N(C)CC1(NC(c2ccnc(C)n2)=O)CC1 52061,C1(C)(NC(CCn2c(C)ncc2)=O)CCN(C(C2(C(C)C)CCCO2)=O)C1 52062,C(=O)(C#CC1CCCOC1)N1CC2C(CNC(=O)C=Cc3cc[nH]n3)C2C1 52063,C(=O)(C1CCCc2nncn21)N1CCN(C(C(CCCC=C)(C)C)=O)CC1C 52064,C1(CNC(CNC(C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CCC1(F)F 52065,C(=O)(CC(O)CC(C)C)NCCN(C(COCCOCC#C)=O)C(C)C 52066,N1(C(C(CC)C)=O)CCC2(CCCC2CNC(=O)CCOCC(F)(F)F)CC1 52067,C1(C(=O)NCCc2cccc(F)n2)C2CCC(C2)N1C(=O)CCc1ccccc1 52068,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(C=CC(=O)OCCCC)=O)OCCC1 52069,C1(=O)C(O)CCCN1C.C1(N(C(=O)C2CC2)CC)COCC1O 52070,n1(CC(=O)N(C)C2CC2)cc(C2(O)CN(C(=O)Cn3ccnn3)C2)nn1 52071,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52072,c1(-c2cccc(C)c2C(=O)OCC2CC3C=CC2C3)ccc(C)c2ccccc12 52073,Cc1nc(NCC(C)(C2CC2)NC(c2ccsc2C)=O)c(C)c(O)n1 52074,C1(NC(c2cnn(CC)c2C)=O)CCN(C(=O)Nc2c[nH]c(=N)nc2C)C12CC2 52075,n1(CC)ncc(C(=O)NCc2ocnc2C(=O)NC2(C)CCOC2C)c1C 52076,N1(C(CC(C)F)=O)CCN(CC(C)(C)NC(c2cc(CCO)on2)=O)CC1 52077,CCC(C)(C)C(O)C(=O)N1CC(NC(C2CCC(OC)CC2)=O)C(C)(C)C1 52078,c1(C(=O)NCCCCNC(C2CC(C)(O)C2)=O)cc2scnc2[nH]1 52079,C1(NC(C=CSC)=O)C(C)CCN(C(c2cnc(C3CC3)o2)=O)C1C 52080,CC1CCCCC1(C)C(=O)NC1CCCN(C(c2csc(O)n2)=O)CC1 52081,N1(C(c2c(C)cccn2)=O)CCCCC2(CCN(C(C34CSC(C3)C4)=O)C2)C1 52082,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52083,N1(C(c2c(CC)ncs2)=O)CCCN(C(c2ccc(O)c(C#N)c2)=O)CC1C 52084,C1(CCCC(N2CC(O)(NC(C(C)NC(COC)=O)=O)C2)=O)CCCC(=O)N1 52085,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52086,N1(C(C2OCCN(C)C2)=O)CCN(C(=O)CCc2cc(Cl)cs2)CC1CCO 52087,C1(C)(CNC(c2ccc(C)o2)=O)CCCN(C(C2CC3(CC3)CN2C)=O)C1 52088,C1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2)=O)CCC2(CCC2)O1 52089,C(=O)(C(O)C(C)(C)C)NCCC1(O)CCN(C(c2cc(C)c(Cl)s2)=O)C1 52090,c1(NC(=O)Nc2scc(C(C)N)n2)ccc2cc(I)cnc2c1 52091,Cc1cc(C(=O)NC(C(=O)N(C)Cc2nc[nH]n2)C2CCCC2)ncc1N 52092,N1(C(Cc2ccc(C)o2)=O)CCCCC12CC(NC(C1CN(C)C1)=O)C2 52093,CCCCC(CC(=O)NCC(F)(F)C(C)C)NC(c1cc(C)ncn1)=O 52094,C=CCCCCCCNc1nc(CS(C)(=O)=O)nn1-c1ncccc1F 52095,CCCC(CCCNC(=O)CC(O)C(C)C)NC(c1cc(C2CC2)nn1C)=O 52096,Cc1ncnc(C)c1CNC(C1(F)CCN(C(=O)C=CC(=O)N(C)C)C1)=O 52097,C=CC(CC)CC(=O)N1CCN(C(=O)C2=CCSC2)C(CCO)C1 52098,CC1(C)NC(=O)CCC1NC(=O)COc1cccc(Cl)c1 52099,CCCC(CC)CCC(=O)NCc1cc(C(=O)NCc2noc(C3CC3)n2)cs1 52100,CC1CN(C)CCN1C(C1(O)CCN(Cc2ncc(Cl)cc2Br)CC1)=O 52101,CCCCCC(=O)N1CC(NC(c2cncn2Cc2cccc(Cl)c2)=O)C2CC12 52102,O=C(C1=CCSC1)NC1CCC(NC(=O)CCc2ccccc2)C1 52103,C12(C(=O)NCCCNC(C(C(C)(C)C)SC)=O)CCC(C)(C(=O)O1)C2(C)C 52104,C(C1CCc2c[nH]nc21)N(C(=O)CC12CCC(CC1)C2)CCCN(C)CCF 52105,c1(CC(C)(C)C)ccccc1C(=O)NC1COCC1CNC(=O)COC1CCC1 52106,C1(CNC(C(C)c2ccco2)=O)CCC(NC(=O)CC2(O)CCC2)CC1 52107,C1(NC(CC2C(C)OCC2)=O)CC(OCCNC(CCN=[N+]=[N-])=O)C1(C)C 52108,Cn1ncc2cccc(-c3nc(CS(C)(=O)=O)nn3CCN3CCCCC3)c12 52109,N1(CCC(C)(C)C#N)C(=O)NC(CC2CCOCC2)C1=O 52110,N1(CC(=O)NCCC(C)N(C(=O)C(=O)N(C)C)C)CC(=O)N(C)C1=O 52111,c1(CNC2CC(CC(=O)Nc3cnc4cnccn34)C2)c[nH]c2nccc(Cl)c12 52112,C1(c2cn(CC(=O)OCC)nn2)CCCN(C(C2(Br)CC2(C)C)=O)CC1 52113,c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)C)=O)ccc2c(c1)CCCC2 52114,CCCCC(O)C(=O)NC(C1CCCC1)CNC(c1ncc(F)cn1)=O 52115,Cc1cnc2cc(C(=O)NCC3CC3)nn2n1.C1(C(=O)NC)CCC2(CCC2)C1 52116,CCC(CC1CCCCC1)C(=O)NC1CCOC(CNC(C2CC(C#N)C2)=O)C1 52117,N1(C(C(N2CCCC(C)C2)=O)=O)CCC2(CCN2C(=O)Cc2c[nH]nc2O)C1 52118,C(CCCCCC(=O)N1CC2(CCN(C(c3ccccc3C(C)C)=O)C2)C1)SC 52119,N12CCC(C1)C2=O.C1(CNC(C)=O)CCCC1NC(=O)CCC1CC(C)C1 52120,c1(NC(C(c2ccn(CCOCC)c2)NCCOC)=O)ccc(S(C)(=O)=O)cc1 52121,N1(C(CN(C(=O)Cc2ccc(C#N)cc2)C(C)C)=O)CCS(=O)C(C)C1 52122,c1(OCC=C)ccc(Cc2nc(-c3ccc(Cl)s3)nn2CC(C)C)cc1 52123,C1(NC(CC2(OCC)CCC2)=O)CCN(C(c2ccc(C(C)=O)cc2)=O)C(C)C1 52124,c1(C(N)=O)nccc(=NC2CCN(Sc3nnc4ccccn34)C2)[nH]1 52125,C1(CC(=O)NCCC2CCOCC2)CN(C(=O)CC2CCOC2=O)CCO1 52126,N1(C(CC2CCN(C(C(C)CO)=O)CC2)=O)CCCCCC1CO 52127,c1(C(CC)C)ccc(C#N)c(NCC(C)CNC(C2C=CC=CC=C2)=O)n1 52128,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cn2c(n1)CCCC2 52129,c1(C(=O)NCC2C(NC(CCNC(CC(C)C)=O)=O)C2)ccccc1C(F)(F)F 52130,Cc1ccccc1C(=O)NCCCCCNC(C1CCC(C(F)(F)F)C1)=O 52131,c1(C(=O)NC(CC2CC2)C(=O)NCCCCn2ccnc2)cccc[n+]1[O-] 52132,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)CCN(C)C)C(C)(C)C1 52133,c1(CCC)ccc(C(=O)NC2CN(C(=O)CCc3cnc(C)o3)C2)cc1[N+](=O)[O-] 52134,c1(C(=O)NC2CC(C)(CC)N(C(=O)CN(C)C(=O)C3CC3)C2)c(C)nc2sccn12 52135,c1(C(=O)NC(CN(C)C(C2CC(CC(=O)OC(C)(C)C)C2)=O)(C)C)cnc(Cl)s1 52136,c1(C(N2CC(NC(Cn3c(C)ncc3)=O)C(O)C2)=O)ccc(Cl)c2ccccc12 52137,C(=O)(CCCC(C)NC(=O)CC1(COC)CC1)N1CC(CC(C)C)N(C)CC1 52138,C(=O)(C(O)CCCNC(=O)CCCC1CC1C)N(CCC(=O)NC)CC 52139,C(=O)(C(O)CC(C)C)NCCN(C(c1nn(C)cc1C(F)(F)F)=O)CC 52140,CC1(C)CCCN(C(=O)C=Cc2cnc[nH]2)C1CNC(C1CCS1(=O)=O)=O 52141,c1(SCCOCCOCC)cc(N(C2CCSCC2)CCC)c2c(Br)cccc2n1.NCC 52142,n1(CC(C(=O)NCCN(C(=O)CCc2c(C)noc2C)CC)C)nc(C)cc1C 52143,c1(C2CCN(Cc3ccc(CC4CN(C)C(=O)C4)o3)CC2)cc2c([nH]1)CCCC2 52144,C12(C(=O)NCC3(NC(CCOCC#C)=O)CCCCCC3)CCCCC1C2(F)F 52145,c1(C(CN2CCC(NC(=O)NCc3n(C)ccn3)CC2)=O)c(Cl)cccc1Cl 52146,CN1CC(C)(C(N2CC(NC(=O)CSc3nncn3C)C2)=O)CCC1=O 52147,C1(NC(COCCC)=O)CC2CCC1(C(=O)NC1CC(CCC(C)C)C1)C2 52148,C1(CC(N2CC(N(C)C(c3ccncn3)=O)C2)=O)NC(=O)CN(C)C1=O 52149,N1(c2cccc(S(=O)(=O)N3CCC(C#N)(F)C3)n2)CCC(=O)N2CCCCCC12 52150,C1(CC)CN(C(=O)CC(F)(F)CC)CCN1C(=O)CNc1cc(F)ccc1F 52151,C1(C(=O)NC2(C(COC)O)CC2)C(NC(=O)C(C)N(C)C(C)=O)C1(C)C 52152,CCC(CC)C(=O)NC(Cc1cnn(C)c1O)C(=O)NCCc1noc(=O)n1C 52153,c1(SCC(=O)NCC(F)CNC(=O)CCN2CCOC2=O)ccccn1 52154,C1(NC(C=C(C)C)=O)CCC(C)N(C(C2C3COCC23)=O)C1 52155,C=C(C)C1OCCC1CNC(=O)CC1CC(NC(=O)CC2(C)CC2)C1 52156,C1(C(CNC(CSCCN(C)C)=O)(C)O)CCN(C(C2(F)CC2)=O)CC1 52157,Cc1ccn2c(C(N3CCOC(CO)CC3)C(=O)Nc3ccccc3)cnc2c1 52158,C1(C(=O)NC2C3(CN(C(=O)OC(C)(C)C)C3)CC2)CC2CCC1C21CC1 52159,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)F)c2)=O)C1 52160,c1(C(=O)NC2CC(C)N(C(c3cc4c[nH]cnc-4n3)=O)C2)cc(N)c(Cl)c(O)n1 52161,C(=O)(C1=NOC(C)(C)C1)N(C1CCCC(NC(c2c(CC)[nH]cc2)=O)C1)C 52162,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52163,C#Cc1ccc(C(=O)NCC(C)NC(c2cnn(CCC(C)C)c2C)=O)cc1 52164,S(=O)(=O)(c1cccc(NC(=O)C(C)SC)c1)NC1(C(=O)OC)CC(CO)C1 52165,C#CCCCC(C)C(=O)NC1CC(C(=O)NCCCN2CCCC2)C1 52166,Cc1cc(C(=O)NC23CC(CNC(c4csc(C(F)F)c4)=O)(C2)C3)cc2nn[nH]c12 52167,C1(NC(=O)C(=O)NC2COC3CC2C3)CCC2(CCOCC2)C1 52168,c1(C(=O)OCC)nc(NCC2CCCN2C(=O)C(C(C)C)SC)cc(O)n1 52169,C(=O)(C(C1CCOC1)NC(=O)CN(C)C)NCCOCC.C(C)(C)C 52170,N1(CC(=O)NC(C(C)C)CNC(=O)C(C)N(C)C)CCC(=O)NC1=O 52171,C1(NC(C(C=C)(F)F)=O)CCCN(C(c2cncc(OC)c2C)=O)C1C 52172,n1(CCC)ncc(C(=O)NCC2(NC(C3CSC3)=O)CCOC2)c1Cl 52173,C1(OC)(CNC(C2CC23CC3)=O)CCN(C(=O)CCn2nc(C)cc2C)C1 52174,C(=O)(CCCCCN1C(C(=O)NC)CCCCC1)NCCOC(CC)C 52175,CC1CC(NC(=O)C(C)(C)CC#N)CCN1C(c1ccn(-n2cccn2)n1)=O 52176,c1(CN(c2cc(Nc3cccc(C4CC4)c3)ncn2)C)ccc2nc(Cl)sc2c1 52177,c1(CN2CC(CNC(C(CC)C)=O)OCC2)nc2ccccc2[nH]1 52178,N1(C(C#CC(C)C)=O)CCCC(C2CC2NC(=O)CC2CCCCCC2)C1 52179,c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)c(O)nc(=O)n2c1CCC2 52180,n1(CC(=O)OC)cnc(C)c1C(=O)NCCCN(C(c1cccnc1C)=O)C(C)C 52181,c1(CNC(c2n(CC(=C)C)nnn2)C2(CC#N)CC2)c(Cl)ncn1C 52182,O=S(=O)(c1[nH]cc2c1CCS(=O)(=O)C2)N1CC(=Cc2cncs2)C1 52183,c1(-c2scc(C)n2)cccc(NC(=O)NC2CCC(SCC(C)C)C2)c1 52184,C12(N(C)C(C3CCCCC3(C)C)=O)CCC(CC1)N(C(C1CCCO1)=O)C2 52185,c1(CCN(CCCC(=O)OC)c2ccccc2)ncc(-c2ccccc2)cn1 52186,C1(F)(C(=O)NCC2C3CN(C(c4scc(C)c4)=O)CC32)CC2(CCC2)C1 52187,C(=O)(C(CCOC)NC(=O)CCn1ccnc1)NC(c1nc(C)no1)CC 52188,N1(C(C2CN(C(c3ccnnc3)=O)CCN2)=O)CCN2CC(O)CC2C1 52189,CC1CC(NC(=O)CNC(=O)COc2ccccc2)N(C2CCCC2)C1=O 52190,N1(C(C2(C)CC2Br)=O)CCC2(CCCCN(C(c3ccc4cnnn4c3)=O)C2)C1 52191,N1(C(c2cncc(SC)c2)=O)CCOCC(NC(=O)C(C)(C)N2CCOCC2)C1 52192,C(=O)(C(F)(F)C(F)(F)F)N(C1CCCN(C(C2(C)COC(=O)C2)=O)CC1)CCO 52193,C(=O)(CCCCCCS(N)(=O)=O)N1CC=C(C(N2CC(C)NC(=O)C2)=O)C1 52194,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52195,Cc1cc(C(=O)NCCCOCCNC(=O)C(O)CC(F)F)nc(O)c1 52196,C#CC1(C(=O)NCc2cc(C)c(C(=O)NC(C)C(C)C)o2)CCCC1 52197,C1(C(=O)NC)(N(C(=O)C=Cc2ccc(OC)cc2)C2CC2)COc2ccccc2C1 52198,C=CCCC(C(=O)N1CCC(CCO)C1)NC(c1ccc(C)cc1)=O 52199,CN1CC=C(B(O)c2ccc(NCC(c3cccc(C(F)F)c3)=O)cc2)CC1 52200,C1(CC(=O)NCC2(CC)CCCO2)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 52201,c1(C=O)cncc(N(C)C)c1.c1(C=O)ccncc1.C1C(O)CN(C)N1C 52202,c1(CCC(=O)NCC2C=CC(NC(C3CNC(=O)N3)=O)C2)cccc(C(F)(F)F)n1 52203,C1(C(N(CCN(C(=O)C(C2CC(F)(F)C2)O)C)C)=O)CCCN(C)C1 52204,CN1CC(C)(C)CC1C(=O)NC1CN(C(c2csc(C3CCCCC3)c2)=O)C1 52205,N1(C(CCC=CC)=O)CCC(C2CCN(C(c3c[nH]nc3C)=O)C2)C1 52206,C(=O)(C(F)(F)CN1CCCC1)NCCCN(C)C(C1(F)CCCCC1)=O 52207,c1(C(=O)NC2CCC(C)N(C(C3(C(N)=O)CC3)=O)C2)ccc2cnoc2c1 52208,N1(C(C=CSC)=O)CCC2CCC(C1)N2C(c1cccc(N2CCOCC2)c1)=O 52209,Cc1c(CC(=O)NC(C)CN(C(=O)Cc2ccc(F)cc2)C)cnn1C 52210,C1(CCNC(C2(C)C(C)C2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 52211,C1(OC)(OC)CC(C(=O)N(C2CCN(C(=O)CCC3CCCOC3)C2)CCO)C1 52212,c1(C(N2CC(O)(C(C)(C)CNC(=O)CCCCCF)C2)=O)ccc2n[nH]cc2c1 52213,C(=O)(C(CCF)NC(=O)CN(C)C(=O)C1CC1)NC(C)CCCO 52214,N1(C(C2CC(CC)C2)=O)CC2(C(=O)NCC3CCSC3)CC1CCO2 52215,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52216,C1(O)(CNC(c2cc(C)c(O)cc2)=O)CCCN(C(C2CNC(=O)C2)=O)CC1 52217,C1(NC(c2nc(C)sc2C)=O)CC2(CNC(=O)CC(O)C(C)C)CC1CO2 52218,n1(CC)cnc(C(=O)NC(C)C(C2CCCCC2)NC(C2CC(C)(F)C2)=O)n1 52219,N1(C(c2c(C)ocn2)=O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C2COCC12 52220,c1(C(N(CCC(=O)NCC(c2ccco2)O)C)=O)c[nH]c(=O)cn1 52221,N1(C(CC2(C=C)CC2)=O)CCC2(CCCN2C(=O)Cc2cnn3ccccc23)C1 52222,Cc1cccc2[nH]cc(CC(N3CCC(CN(C(=O)CN(C)C(C)C)C)C3)=O)c12 52223,c1(C(=O)NCC2C(CNC(CC3=NN(C)C(=O)C3)=O)C2)cnc2c(n1)CCCC2 52224,N1(C(c2c(CNC(c3c(C)coc3)=O)ccs2)=O)CC(=O)NC(C(C)C)C1 52225,CCCCC(=O)C(=O)NC(CN(C)C)C(=O)N(CC)Cc1ccoc1 52226,C1(C(N(C)NCC2CCN(C(CC3CC(=C)C3)=O)C2)=O)CCCN(CCCC)C1 52227,N1(C(c2cncc(N)c2)=O)C2CCCC1CN(C(C1(Br)CCC1)=O)C2 52228,C1(NC(C(C(C)O)(C)C)=O)CCCCN(C(=O)CC(=O)OC(C)(C)C)CC1 52229,CCC1=NOC(CNC(=O)CC(=O)C(C)(F)F)C1.C(C)(C)(CC1CCC1)O 52230,N1(C(COCC)=O)CC(C)(C)CC1CNC(=O)C(C1CC(F)(F)C1)O 52231,c1(C(=O)NCCCCC(C)C)n[nH]c2c1CC(C)CC2 52232,CCC(O)C(C)C(=O)N1CCCC(CCNC(c2cc(C3CC3)n(C)n2)=O)C1 52233,c1(C(N2CCCCC(CNC(CC3CN(C)C3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52234,N1(C(C(CC)C(C)C)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52235,C1(CNC(C(c2ccccc2)C)=O)CC(O)CN1C(=O)CC1CC(=O)NC(=O)C1 52236,C#Cc1cc(C(=O)NCCC(O)C(=O)N(CC)Cc2ccoc2)ccc1C 52237,C1(C2CCCN(C(C3CCCN3C3CC3)=O)C2)(NC(c2cn(CC)nn2)=O)CC1 52238,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52239,N1(C(COCCSC)=O)CCC(NC(C2Cc3cscc3C2)=O)C(C(C)C)C1 52240,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52241,CC1CN(c2ccccc2)C(C)CN1CC1CCCNC1=O 52242,C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC12CCC2 52243,c1(C(=O)NC)ccc(OCCCC(=O)NCCOCCOC)nc1.n12ccnc1C2 52244,c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)C23CC3)nc(C)c(C)nc1C 52245,N1(C(=O)C=CC2CCCC2)CCC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 52246,c1(C(N2CC(O)CC(NC(C(CC)N(C)C)=O)C2)=O)n[nH]c2c(C)cccc12 52247,C1(C(N(CC(N2CCCC2)=O)C)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)C1(C)C 52248,c1(C(=O)NCCN(C(c2coc(Cl)n2)=O)CC)nc(C)ccc1O 52249,CCC(C)C(C(=O)NC1C2CC3C1C3C2C(=O)N(CCCO)C)N(C)C 52250,C1(CN(C(CN(C)C(N)=O)=O)C)C2CN(C(=O)CCCn3cccc3)CC12 52251,c1(OC)ccc(F)cc1C(=O)N(CCNC(c1cn2ccnc2s1)=O)C(C)C 52252,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52253,CCC(C)C(C)C(=O)NCC1CN(C(=O)CCN2CCC(C(N)=O)CC2)C1 52254,C(=O)C(c1cnsc1)C1CC1C.C(=O)(COC(C)=O)N(C)CC 52255,N1(C(CCc2ccc(C)cc2C)=O)CC(CNC(C2(C)CC2F)=O)CC(C)(C)C1 52256,N1(C(C2C(C)CC(=O)CC2)=O)CCOCCC1C(=O)NC1CCC(F)CC1 52257,N1(C(c2ccc(C3CC3)nc2)C(=O)NC2CC(F)(F)C2)CCN2C(CNS2(=O)=O)C1 52258,CC(=O)C(C)(C)CC(=O)N1CC2(CC(C(=O)NCC3(C)CC3)CO2)C1 52259,N1(C(C2(CN3CCCCC3C3CCN3)CC(=C)C2)=O)CCC2(CCCCC2)CC1 52260,C1(c2noc(C3CC3)n2)(C(N2CCSCCC2CO)=O)CC2(CCC2)C1 52261,CC1(CC(=O)NC(CO)C(F)(F)F)CCN(C(c2nccnc2N)=O)C1 52262,CCC(C)CC(C(=O)NCC(O)C(F)(F)F)NC(=O)CN(C)CC 52263,C1(C(N(CCCNC(=O)Cc2ccnnc2O)CC)=O)CCC(C)NC1=O 52264,C1(=CCNC(C(C)(O)C2CCOC2)=O)CCN(C(=O)CSS(C)(=O)=O)CC1 52265,C1(OC)CC2CC(C1)N(C(C1CCC(CNC(c3cc(C#N)cn3C)=O)C1)=O)C2 52266,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)Nc1cnn(C(C)(C)C)c1 52267,C1(NC(C(=O)NCC)=O)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CC1C1CC1 52268,c1(CC(=O)NCC(=C)CCNC(c2cc[nH]n2)=O)nc(C2CC2)nn1C 52269,c1(-c2cn(C3CN(C(C4CCCSC4)=O)C3)nn2)cccc(Br)c1Br 52270,c1(C(=O)NCCNC(CN(S(C)(=O)=O)C)=O)cc2cc(Cl)ccc2s1 52271,C(=O)(C1=COc2ccccc2O1)N(CC(C)NC(C1(CCOC)CCC1)=O)C 52272,C(=O)(CCS(=O)(=O)CC(C)C)NCN=c1[nH]c(=NCC(C=C)OC)[nH]c2c1[nH]cc2 52273,C1(CN(C(C)C)C)CCCN(C(=O)CCOCCNC(=O)Cn2cnnn2)C1 52274,C1(NC(CCN(CCC)C)=O)CCCCCC1NC(=O)CC1CCC(F)(F)CO1 52275,c1(C(N(C2CCCN(C(C34CCC(C3)OC4)=O)CC2)C)=O)cc2ccccn2n1 52276,C(=O)(C(F)C(C)(C)O)NC(C(C)C)CNC(=O)C=Cc1ccccn1 52277,c1(CNC(C(C)c2ccsn2)=O)ncoc1CCNC(=O)COC(F)(F)F 52278,Cc1cc(F)ccc1C(=O)NC(C)CCc1ccc(F)cc1 52279,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(CNC(=O)C(C)CC2CCCO2)C1(C)C 52280,C(=O)(C=CS(C)=O)NCC(C(C)C)NC(c1cnn(C)c1)=O 52281,Nc1ccc(C(N2CCCCC(CNC(=O)COCC(F)(F)F)C2)=O)nc1F 52282,N1(C(c2oc(CC)c(C(=O)OC)c2)C(=O)NC(C)C)CCS(=N)(=O)C2(CCC2)C1 52283,N1(C(COCCCC)=O)CC2CCN(C(=O)CC3CCCC(C)(C)C3)CC12 52284,N1(C(C2CCC(C)CN2C(c2cc3n(n2)CCC3)=O)=O)CC(C2CCCC2)C1 52285,C1(CC(=O)N(C2CCN(C(C(COC)(C)C)=O)C2)CCO)C(=O)N(C)N=C1C 52286,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52287,C1(NC(c2cn(CC(C)C)nc2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52288,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2occc12 52289,c1(C(=O)NCC2(CN(C(=O)CC34CCCN3CCC4)C)CC2)ccc(F)cc1O 52290,N12CCCC1NC(=O)C1(CC1)CNC(=O)C2=O.c1(CN(C)C2CC2)cccs1 52291,C1(NC(C(C2CCN(OCCO)CC2)C)=O)C2CCC(C2)C1Cc1ccncc1 52292,C(CNC(c1ccc(C(C)=O)cn1)=O)(C(C)(C)C)NC(CCC1CC(OC)C1)=O 52293,C1(C(=O)C=CC2CCCO2)=NC2C(=C1)N=CN2CC1CC1 52294,C(=O)(C(C)Cn1ccnc1)N(C1CCCC1)C(CC1CC(C(=O)OCC)C1)=O 52295,C(c1cncn1C)=CC(=O)N(CC(C)O)CCNC(C(C1CCC1)OCC)=O 52296,c1(C(=O)OC)cc(C(=O)Nc2cccc(CNC(=O)Cc3coc(C)n3)c2)ccn1 52297,Cn1nc(Cl)c(C(N2CCCC2CNC(c2cnc3n2CCC3)=O)=O)c1Cl 52298,C1(S(N)(=O)=O)(C(=O)NCC(CO)NC(CC2N(C(C)C)CCC2)=O)CCCCC1 52299,C1(C(=O)NCCCC(C)NC(C(CCOC)OC)=O)CCCC(=O)CC1 52300,C1(n2cccn2)(C(N(CCCF)C)=O)CCN(C(c2ccc(Cl)cn2)=O)CC1 52301,C(=O)(C(C)(C)C1CCC1)NC(C(=O)N(C1(CC)CC1)C)C 52302,C1(C)(C(N(C2CCCN(C(C3(F)CCCOC3)=O)C2)CC)=O)CCCCC1 52303,CC(C(=O)N1CCC(C)(C(=O)NCCOC2CCCC2)CC1)S(C)(=O)=O 52304,S(=O)(=O)(c1ccccc1C(=O)Nc1cnc2ccnn2c1C(F)(F)F)NCC=C 52305,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52306,C#CCC(C)(C(=O)NCC1COC(=O)N1C)NC(c1cnc(OC)cn1)=O 52307,C1(NC(c2c(C)cccc2)=O)CN(C(=O)CC2CNC(=O)C2)CC(C)(C)C1 52308,C1(NC(C=CC)=O)CC2CCC1CC2NC(c1ccnn1CCC)=O 52309,N1(C(CSC)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52310,CC(C)C(C(=O)N(CC(C)O)CCNC(=O)C(F)(F)c1csc(Cl)c1)NC(N)=O 52311,C=CCCC(F)(F)C(=O)NCC1CN(C(=O)C(c2ccccc2F)F)C1 52312,C(=O)(C(O)CCSC)NCC1C(NC(CCc2onc(CSC)n2)=O)C1 52313,c1(C(=O)NCCCNC(C2C(C)(C)OC(=O)N2)=O)cnn2c(Cl)cccc12 52314,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)N(C1(C)CCCC1)CC1CC1)C2 52315,N1(C(C(C(C)C)O)=O)CC(CN(C)C(C2(C(F)F)CCN(C)CC2)=O)C2(CC2)C1 52316,Cc1ccc2c(C(=O)NC(C3CCCN3C(c3c[nH]c(=N)s3)=O)C)c[nH]c2c1 52317,C(CC(C)(C)C(=O)CNC(=O)CCc1cnco1)N(C)CCO 52318,C(=O)(C(C(C)C)C(C)C)N1C(CNC(C2CCCC(=O)N2)=O)CC(OC)C1 52319,CCCC(CCO)NC(C1CCCN1S(=O)(=O)CC1(C#N)CCCC1)=O 52320,N1(C(c2c(SC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52321,CC(CC(=O)NC(CC1CC1)CC(=O)NCCc1cocn1)C(F)(F)F 52322,C(C)(C)(CCC(=O)N(C1CCC(NC(c2cc(F)cs2)=O)CC1)C)N(C)C 52323,Cc1cc(C(=O)NCC(CNC(=O)C(F)C(F)(F)F)CO)ncc1S(C)(=O)=O 52324,c1(C(=O)NCC(CC)(CC)NC(=O)C2=C(C)OCC2)cnc2ncnn2c1O 52325,CS(=O)(=O)CCCC(=O)NC1(CNC(C2CC23CCOC(C)C3)=O)CCC1 52326,c1(C(=O)NCC2CCCCN2C(c2cn3c(n2)SCC3)=O)cc(F)c(Cl)cc1Cl 52327,CC(C(C)C(=O)N(C(C)C(=O)OC)C)N(C(c1nc(=N)cc[nH]1)=O)C.N(C)C 52328,c1(CN2C(C)(CNC(c3cncc(N(C)C)c3)=O)CC2)ccc(F)c(F)c1 52329,C1(NC(CC(OCC)OCC)=O)CCCCC1NC(=O)CCC 52330,Cc1ncc(C=CC(N2CCN(C(=O)CSc3nc[nH]n3)C3CC23)=O)c(O)n1 52331,C(CCCC(CO)NC(=O)CCC1CCC1)NC(C(C)N(C)C)=O 52332,Cn1ncc2c(N(CCF)Cc3cccc(Cl)c3)[nH]c(=NCC3=COCC3)nc12 52333,c1(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CCOC2)ccc(N)c(Cl)n1 52334,c1(CCCC)cccc(OCNCCOC)c1OC.C12CCC3(C1)CC3C(=O)N2 52335,Cc1ncc([N+](=O)[O-])cc1C(=O)N(C)CCNC(=O)CCC#N 52336,C1(CNC(N(C2C=CCC2)C)=O)CC(F)(CO)C1 52337,CC1C(=O)N(CC(N2CC(NC(=O)C=CBr)C3(CCC3)C2)=O)C(=O)C1C 52338,N1(C(COCc2cc(C)no2)=O)CCCC(NC(c2cncc(Cl)c2C)=O)CC1 52339,C1(NC(CC2(CC)CCOCC2)=O)COC2(CCN(C(C3(C)CC3)=O)C2)C1 52340,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)nc(O)nc1C)=O)C2 52341,c1(-c2n(-c3cccc(C)c3)nc(C3CCOC3)n2)cn(C)cc(Br)c1=O 52342,c1(NC(COCC)=O)ccc(NCc2cc(C(=O)C(C)(C)C)n[nH]2)cc1 52343,C(=O)(C1=CCCN(C(C2(C#N)CCCC2)=O)C1)NC(CC)CC(=O)OC 52344,N1(C(CCNC(C(C)(C)C)=O)=O)CC(O)(C2(CNC(=O)CC(C)(C)O)CC2)C1 52345,c1(NC(C)C)ccc(C(=O)NCCC2(O)CN(C(C3CC3C(C)C)=O)C2)cn1 52346,c1(C(N2C(CCNC(C3(O)C(C)(C)C3)=O)CCC2)=O)cccnc1OC(F)F 52347,c1(OC)cc[n+]([O-])c(C(=O)NCC2CCN2C(=O)C(C2CCC2)OC)c1 52348,C1(NC(c2cc(CC)sn2)=O)CC12CCN(C(=O)C(C)C1CCCC1)C2 52349,N1(C(C(N2C(c3ccc(C(=O)OC)n3C)COCC2)=O)=O)CC(=O)NCC1C 52350,N1(C(c2cc(C)n(C)c2)=O)CC(NC(=O)C(F)C2CCC2)C(N=[N+]=[N-])C1 52351,C(C(F)(C(=O)NC(C(N)=O)C(C)O)C(C)C)NC(c1c(CC)cco1)=O 52352,c1(N(CCCC(=O)NCC2(O)CC(C(N)=O)C2)C)cc2nncn2cn1 52353,n1(CCC(=O)N(S(C)(=O)=O)C)cc(CNC(=O)C(C)(C)O)nn1 52354,c1(-c2c(N(n3nccn3)CCO)cccc2)ccc(F)c(Cl)c1F 52355,c1(C(N2CCC(O)(C(C)NC(=O)C=CC3CCOCC3)C2)=O)cn2c(n1)CCCC2 52356,N1(C(Cc2c(CC)cccc2)=O)Cc2nccn2CC(NC(=O)C(C)CF)C1 52357,c1(C(N2C(CN(C(C(C)=CC3CC3)=O)C)CCC2)=O)ccc2ncn(C)c2c1 52358,C1(C)(CNC(C(C)CSC(F)(F)F)=O)CCN(C(=O)CN2CCCCC2=O)C1 52359,Cc1cc(NC(=O)C=CCOC)c(O)c(C)c1.S1(=O)(=O)CC(=O)NCC2(CC2)N1 52360,N1(CC(=O)NCCc2c(C(=O)NC3(C(C)C)CCC3)c[nH]n2)CCNC(=O)C1 52361,c1(OC)cc(Br)c(-c2noc(C3CC(C(C)C)N(C)C3=O)n2)cc1C 52362,c1(OC)ccc2cc(C(N3CCC4(CCN(C(=O)CC5CC5)C4)C3)=O)nnc2c1 52363,N1(C(c2c(C)nc(C3CC3)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52364,C1(CC(=O)NCCOCCNC(C2C(C(N)=O)C2)=O)CN2CCN1CC2 52365,C(=O)(CCCCC(F)F)N(C(C)CCNC(C1(CCF)CCOCC1)=O)C 52366,N1(C(C(CC2CC2)OC)=O)CCCC(C)(NC(=O)CC2OCCO2)C1 52367,CC1CC(NC(=O)Cc2ccnn2C)CN1C(=O)Cc1coc(-c2cccs2)n1 52368,N1(CC(=O)Oc2cc(CO)cc(OC)n2)CC2(CCC2)CC1C(=O)NCC 52369,C(F)(F)(C(F)(F)F)NS(=O)(=O)Cc1ccc(C(C(C)N(C)C)OC)cc1 52370,c1(C(=O)NC(CNC(CNC(=O)OCC=C)=O)C)ccc(N)c(C)c1F 52371,n1(CC)nc(C(N2CCC(NC(=O)CC3COC(C)(C)C3)C2)=O)cc1C 52372,Cc1[nH]nc(C(F)(F)Cl)c1C(=O)NC1CC(C)N(C(=O)CN(C2CCSC2)C)C1 52373,C1(C(=O)NCC23CC(CNC(C4CCC(F)CC4)=O)(OC2)C3)Cc2cscc2C1 52374,C1(NC(c2ccc(F)c(Cl)c2F)=O)CCC12CCN(C(C1CCCS1)=O)CC2 52375,c1(OCC(N2CC(CC)C(NC(c3coc(C)n3)=O)C2)=O)ccc([N+](=O)[O-])cc1 52376,CC(Cn1cccn1)C(=O)NC(C)CN(C(=O)Cc1ccn(C)c1)C 52377,C1(N(C(C(C)NC(N)=O)=O)C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1 52378,N=c1cc(CN2CCN(CCC(=O)Sc3ccnc(C(F)(F)F)c3)CC2)cc[nH]1 52379,C1(C)(C(=O)NCC2(C(N(C(C)CC3CC3)C)=O)CCCC2)SCCCS1 52380,C#CC1C(C(N2CCC2CNC(=O)CN2CCC(O)CC2)=O)C1(C)C 52381,C(=O)(CC(O)CC(C)C)NCC1(OCC)CN(C(c2n(CC)ncc2Br)=O)C1 52382,Cc1c(C(=O)NC23CCC2CN(C(c2cc(Br)c[nH]2)=O)C3)nn(C)c1N 52383,Cc1c(Br)cnc(O)c1C(=O)NCC(C(C)(C)C)NC(C1CCC(=O)N1)=O 52384,n1(CC(=O)NCC2C(NC(C(C)=C3CCC3)=O)COC2)ncn2nccc2c1=O 52385,N(C(=NCCN1CCOCC1)NC1CCC1C)C(c1cccc(OC)c1)COCC 52386,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)no1)=O)CC2 52387,c1(C(=O)O)ccn2ncc(-c3cn(C)nn3)c2c1.C(=O)(C(F)(F)C(O)C1CC1)N 52388,CC1(NC(C)(CCBr)c2nnnn2C2(OC(F)F)CCCC2)CCOC1 52389,N1(C(CCN(C)C)=O)CC2CC2(C(=O)Nc2sccc2I)C1 52390,c1(C(N(CCCCCNC(=O)C(C)c2cncs2)C(C)C)=O)ccc(Cl)cc1 52391,c1(SC)cc(C(=O)NCC2CCCN2C(c2cn(C(C)(C)C)nc2C)=O)ccn1 52392,c1(OCCC(=O)NCC2N(C(C(C)C)=O)CCCC2)c(Cl)cc(Cl)cc1Cl 52393,CCCC(C(=O)N1CC(NC(c2cc[nH]n2)=O)CC(O)C1)S(N)(=O)=O 52394,C1(NC(=O)C(O)C(F)(F)F)CN(C(C2CC3(C2)CC2(CC2)C3)=O)CC12CCC2 52395,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)CC1)=O)CC 52396,CC12CCC(C(=O)NCC3(C)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)(CC1)CO2 52397,CC1CC(C)C(NC(=O)C(=O)NCCNc2ccccc2)CN1C(C1CCCC1)=O 52398,c1(CNCc2cncc(F)n2)ccc(F)c(F)c1Br 52399,c1(OC(C)=O)cn(OC(c2n[nH]c(C)n2)=O)nc1C1CCCC1 52400,C(CC(=O)N(C)CC1CCCCC1O)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52401,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52402,C(=O)(CC(C)SC)N(CCC#C)CC.C(=O)(CC1CC1)NCC1CC1 52403,CN1CC(C=O)NC1=O.N1(N2CCC2)CCC(N(C(=O)C=C(Cl)Cl)CCO)CC1 52404,C1(NC(C(c2cccc(C)c2)C)=O)CCCN(C(c2cc(O)ncn2)=O)CC1 52405,O=S(=O)(c1cnc(NCC2CCOCC2)c(Cl)c1)N1CC2CC2(CO)C1 52406,c1(CC(N2CCC(CC=C)(NC(=O)C(C)N(C)C)C2)=O)ccc(C)c(OC)c1 52407,c1(Cc2nc(-c3ccc(C)cc3)on2)cnc(C2CC2)c(C)c1 52408,c1(C(F)F)cn(C)nc1C(=O)NCCC1CC(NC(c2occ(C(C)=O)c2)=O)C1 52409,c1(C(N2CCCC(CNC(C(C)SCCCC)=O)C2)=O)nnc(O)cc1O 52410,c1(SC)ccccc1C(=O)NCCOCCNC(c1ccc(C2CCOC2)s1)=O 52411,N1(CC(C)N(C)C)CCC2OC(=O)OC2C1 52412,N1(C(c2ncn(C)c2Br)=O)CC(C2CC2c2cn(C3CCC3)nn2)C1 52413,c1(C(=O)NCC2N(C(C(CCC)OCC)=O)CCC2)ccc2ocnc2c1 52414,c1(C(=O)NCC2(O)CN(C(C3(OCC)CCCCC3)=O)C2)cc2c([nH]1)CCOC2 52415,C(=O)(C1=CCCCC1C)NCC1CN(C(C2(C(=O)OCC)CCC2)=O)CC1O 52416,n1(CCCOC)c(N(CC(C)C2CC2)C)nnc1-c1nonc1C 52417,C1(C(=O)NC2CC2CC2CCCC2)(OCC)CCC(C)(C)CC1.C1(=O)CCN1 52418,CC1(C)CCN(C(=O)C=CC2CCC2)CC1NC(=O)CCCOCc1ccccc1 52419,O=C1CC(C(=O)NCCOCCCNC(c2coc(O)n2)=O)=NN1 52420,N1(C(c2ccc(C#C)nc2)=O)CCN(C(C2CC2(F)F)=O)CC(O)C1 52421,C1(NC(Cc2nc(C)[nH]n2)=O)CC(=O)N(C2CN(CC(=O)NC3CC3)C2)C1 52422,CN1CC(CC2C(C)(COC)C(=O)NCCOCCCNC2=O)C1 52423,CC(C)C(C(=O)N1CC(CO)(NC(=O)C(C)NC(C2CCOCC2)=O)C1)N(C)C 52424,Cc1ccc(CCCC(=O)N(C(CNC(c2cnc(S)n2C)=O)C2CC2)C)cc1 52425,C1(C(=O)NCc2nnn(C)n2)(NC(=O)C(F)CC2CCOC2)CC(F)(F)C1 52426,C12(NC(C(c3cnn(C)c3)C)=O)CC(CNC(=O)CC3(C(F)(F)F)CC3)(C1)C2 52427,CCCCCCCCC(CCCCCC)CCOC(=O)CC1(C#N)CCOCC1 52428,c1(C(N2C3CCC(NC(c4cc(F)n[nH]4)=O)(C3)C2)=O)ccc2cccnc2c1O 52429,C(=O)c1ccc(N(CC)C)cc1.N(S(=O)(=O)N(C)C)N1CCC(C)CC1 52430,N1(C(CC2CC(C)C2)=O)CCC2CN(C(=O)CCc3ccc(O)nc3)CC12 52431,c1(N(CC(CCC)O)C)ccc(S(=O)(=O)NC2CC3CC2CC3CO)cc1Br 52432,Cc1ccc(-c2cc(-c3nc(C(C)O)nn3CCC(C)C)on2)cc1C 52433,N1(C(c2cc(CC)ncn2)=O)CC(CNC(=O)C(C)=C2CCC2)C2(CC2)C1 52434,c1(C(N2CCC3C(NC(CS(CC)(=O)=O)=O)C32)=O)cc(C#N)cc(C)n1 52435,C=CCC(CNC(c1c(C)[nH]c(C)c1C)=O)C(=O)N1CCC(C)(CN(C)C)C1 52436,C1(CNC(C2N(C(CCC)=O)CCCC2)=O)(COC)CC2CCC1C2 52437,CN1CC(C(=O)NCC2CN(C(c3csc(-c4ccco4)n3)=O)CCO2)CC1=O 52438,Cn1ncc2c1CC(C(=O)NC(C)(C(N)=O)c1ccccc1)CC2=O 52439,CCC(C)(C(=O)NC1CCC(NC(c2ccnc(C)n2)=O)CC1)C(N)=O 52440,c1(C(N(C(CCNC(c2c(CC)nns2)=O)C)C)=O)ccc(C)n1C 52441,N1(C(CCC2C(C)=NNC2=O)=O)CCN(C(=O)Cc2ccc(C)c(O)c2)CC1C 52442,N(C1CCC=Cc2ccccc21)c1ncnc(NCC(=C)Cl)c1C 52443,C1(C(=O)O)CCCN(C(C2CN(C(=O)CC3CCCC4CC34)CCO2)=O)C1 52444,CC1(C)CC(CCNC(=O)C(N2CCCC2CCOc2ccccc2)=O)C1 52445,Cc1c(NC(C2(F)CN(C(C)C(=O)NC(N)=O)C2)=O)oc2ccc(Cl)cc12 52446,C(C)(C(CC)NC(C1(C(C)C)CC1C(F)(F)F)=O)SCC 52447,c1(OC)cnn2cccc2c1.C12CCN(C1C(C)C)C(=O)CONC2=O 52448,Cc1c(C(Cn2cc(CCN(C)C)nn2)NC(=O)C(C)O)oc2ccccc12 52449,C(=O)C1=CCCCC1C.C(=O)(C(C)CC1CCC1)N1C(CC(=O)NC)CC1 52450,N1(C(CCSCC)=O)CC2CC2(N(c2nnnn2C)C(=O)COC2CCCCC2)C1 52451,C1(NC(Cc2nc(C)oc2)=O)C2CC3C1C3C2C(=O)NC(CF)C(F)(F)F 52452,c1(OC)ccc(C(=O)NCC2(NC(=O)C=C(C)C)CC2)c(O)c1F 52453,C12(CCCN(C(=O)C(C)(C)CCOC)C1)C(=O)N2.C1(COC)(OC)CCCCC1 52454,N1(C(CSCC(C)C)=O)CCOC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 52455,c1(C(=O)NCC2(C)CC(NC(C=CC)=O)C2)c(C)c(C)nn(C)c1=O 52456,C=CCCCC(C)(C)C(=O)N1CC(OC2(CC(=O)OCC)CCC2)C(OCC)C1 52457,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52458,C1(NC(C=C(C)C)=O)CC2(CCN(C(C3CC3c3cccc(F)c3)=O)CC2)C1 52459,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2C3CCCC23)=O)CC1C 52460,N1(C(C2(c3cn(-c4cnn(CCF)c4)nn3)CC2)=O)CCOCC1CC(F)F 52461,N1(C(C2CCN(C(C=CCC)=O)C(C)C2)=O)CCCN(C=O)CC1 52462,c1(C(=O)NC(CC=C)CNC(=O)C(C)OCCN(C)C)ccc(O)nc1Cl 52463,N1(C(=O)C(n2cc(-c3cn(CCCCO)nn3)cn2)=O)CCCC(CO)CC1 52464,N1(C(C2C3CC2N(c2ncc(F)cn2)C3)=O)CC=C(c2cccnc2)CC1 52465,c1(N2C3CN(C(C(CC)(C)CC)=O)C(CC3)C2)ccc([N+](=O)[O-])c(O)n1 52466,c1(N2CCC(N(C(C3C=C3C)=O)CC)C2)snc(C)c1C#N 52467,N1(C(CCC=C)=O)CC(OC)CC1(C)CNC(=O)COc1ccc(C)cc1N 52468,N1(C(C(C)CO)=O)CCC(CNC(c2nccc(Cl)c2O)=O)C(C)(C)C1 52469,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2CN(C(C3(C(C)C)COC3)=O)CCC2C1 52470,c1(CN2CCCC(NC(=O)COC(F)(F)C(F)(F)F)CC2)cc2ccccc2o1 52471,N1(C(C(C(C)O)(C)C)=O)CCC2(CCC(NC(c3scnc3Cl)=O)C2)C1 52472,C(=O)(C1=CC2(CCOC2)C1)NC(CNC(c1cc(N)c(C)c(N)c1)=O)C 52473,CC(C)C(F)(F)CC(=O)N1CC(CNC(=O)CN(C)CCO)CC12CCC2 52474,c1(SCC(=O)NC2(C)CN(C(c3c[nH]ccc3=N)=O)C2)ccsc1[N+](=O)[O-] 52475,N1(CC(=O)N(CCC(=O)N(C)CC2CCCC2)CC#C)CCCC1C 52476,CC(C)CCCCC(=O)N1CCN(C(C2CN(c3nnnn3C)C2)=O)CC1 52477,CCCCC(O)CCC(=O)N1CC(NC(CSC2CCC(C)(C)OC2)=O)CC1C 52478,CCCC(O)CC(=O)NCCN(C(=O)Cc1ccc(CC)cc1)C 52479,N12CCC(CC1)NC2=O.C(CCOCCN(C)CC1CCC1)OC 52480,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(c2cscn2)=O)C1 52481,N1(C(c2c(C)cn(C)n2)C(=O)NCC(C)C)CCC(O)C(CO)C1 52482,C1(C(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)CCC2(CCC2)CO1 52483,C(=O)(C(CCOc1cnn(C(C)C)c1)SC)NC(c1ccsc1)CC.C1(=O)CO1 52484,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52485,c1(C(N(C2CCN(C(c3ccc(N)cc3Cl)=O)C2)CC)=O)cnc(O)n(C)c1=O 52486,N1(C(C(C)CC2CCCO2)=O)CCC(C2CC2)(CNC(=O)COC2CCOC2)C1 52487,Cc1c(C(N2CCN(C(=O)COC3CCCC3)C(C)C2)=O)cc(F)cc1Br 52488,c1(NCc2c(C3CN(C(c4cc(C)on4)=O)C3)ocn2)ncnc2sccc12 52489,C1(C(=O)NC2(C(C)(C)C)CC2)(NC(C2(F)CCOC2)=O)CCCC1 52490,Cc1nnc2cc(NCCCCNC(=O)C(c3cccc(Cl)c3F)(C)C)ncn12 52491,C1(NC(c2cc(C)sn2)=O)CN(C(=O)CC2CN3CCN2CC3)C2(CCOC2)C1 52492,C1(NC(C(C=C=C)C)=O)CN(C(=O)C=Cc2cccc(Cl)c2)CCC1O 52493,C1(NC(C2CCC(C(=O)OC)C2)=O)C2CC3CN(C(=O)CC4=CCCCC4)C1C3C2 52494,CC(CC(=O)NCC(C)NC(C1(CC(F)F)CC1)=O)C1CCCO1 52495,c1(CC(=O)NC2C(C)N(C(c3conc3C3CC3)=O)CC2)c[nH]c2ccccc12 52496,CC1(C)CC(NC(=O)COC2CC2)CN(C(c2coc(C3CC3)n2)=O)C1 52497,C(=O)(C1=CCCCC1P(C)(C)=O)NC1C(F)CCN(C(C2(C)CC2)=O)C1 52498,c1(C(=O)NC(c2cn(Cc3ccc(Cl)nc3)nn2)C)cn2ccccc2n1 52499,c1(NC(Cc2ccc(-c3ccc(C(C)(C)C)cc3)cn2)=O)ccc(C#N)c(F)c1 52500,C1(CNC(N(C)CC2CCCO2)=O)(NS(C)(=O)=O)CCCCC1 52501,C(CC1CCCCO1)(C(F)(F)F)C(N(CCC)CCO)=O.C(=O)C(C)(C)C 52502,c1(C(N(C(C(=O)NCc2nnc(CC)o2)C2CC2)C)=O)cc(C#N)ccc1N 52503,C1(C(N2C3CN(C(C4(Br)CC4)=O)CC3C2)=O)COC2CCCCC12 52504,N1(C(c2c(C)nc(CCC)s2)=O)CCC(NC(=O)C(C(C)C)SCC)C(O)C1 52505,CC1(C)CCC(CNC(C23CC=CCN2CCC3)=O)N(c2nccnc2F)C1 52506,C1(NC(C2(NC(=O)CC3CCOC3)CCC2)=O)CC12CCCCCC2 52507,Cc1ccc(F)cc1C(=O)NC1(C)CCN(C(C2CCC3CC23)=O)CC1 52508,n1(CCOC)ccc(C(=O)NCCCCNC(=O)CSCCOC)n1 52509,C12(CNC(CCCN(C)C)=O)CCC(CC1)CN2C(=O)C(c1ccc(F)cc1)O 52510,c1(CCC(=O)NCC23OCCC(NC(C)=O)(C2)C3)nc2ccccc2s1 52511,N1(Cc2cn(-c3c(Cl)ccc(C)c3)nn2)CCCC1C1CCCO1 52512,C(C(F)C(=O)NC1CCC(c2ccccc2)O1)OC(C)(C)C 52513,C1(C(=O)NCc2ccc(C3(C)CC3)cc2)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 52514,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)C)cc2c1 52515,C1(NC(C(C)OC)=O)CCN(C(=O)CCC2CCCCO2)C(C)C1 52516,c1(C(=O)NC(CC=C)CNC(=O)Cn2cnnc2O)ccc2nc(C)cn2c1 52517,C1(NC(C2C(C)CN(C(=O)C(=O)N(C)C)CC2)=O)CCc2ccccc2N(C)C1=O 52518,c1(C(=O)NC2(CC=C)CCCN(C(c3c[nH]c(=N)o3)=O)C2)cncc2ccsc12 52519,c1(N(C2CCC(C)(C)C2)C)ccc(N2CCCCC2=O)cc1Cl 52520,N1(C(c2c(CNC(=O)CCCCC3CC3)ccs2)=O)CCSC2CCC12 52521,c1(NC(c2[nH]cc(C(=O)OC)c2)=O)cccc(NC(C2(C)CCCC2)=O)c1 52522,N1(CCOc2ccc(CCC(C)C)cc2)CCOC(C(=O)O)C1(C)C 52523,c1(N2CCSCC(C)C2)nccc(=NC2CCCn3nccc32)[nH]1.N1CCOCC1 52524,N1(C(C2CCCN3CCCCC23)=O)CC2OCCN(C(=O)C(F)=CC3CC3)C2C1 52525,C1(C(=O)OC)CN(C(=O)CCC2(NC(C3(SC)CC(O)C3)=O)CC2)CCC1O 52526,C1(C(=O)NC(C)CC(C)NC(=O)COCCN(C)C)CC12CCC1(CC1)CC2 52527,c1(COC(C)=O)cccc(NC(=O)CN(S(C)(=O)=O)C(c2ccc(Cl)cc2)C)c1 52528,C1(NC(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)CN3CCCC(C)C3)CC12 52529,c1(OCC)ccc(NC(=O)CN2CCC(c3ccccc3F)C2)cc1 52530,C1(C(c2cccc(Cl)c2)NC(C(C)OCC2CC2)=O)CN(C(=O)C(C)(C)F)CCN1C 52531,N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CC(CO)c2ccccc21 52532,c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)C(C)C)cc2[nH]nc(C)c2cn1 52533,C1(C(=O)NC2(C#C)CC(F)(F)C2)C(C2CC2)CCN1C(=O)C=Cc1ccoc1 52534,N1(C(C2C(C)(C)CCCO2)=O)CCC2(CCCC2NC(C2SCCS2)=O)CC1 52535,C(C(CC(C)C)NC(=O)CCSC1CCCC1)NC(c1c(NC(C)=O)cccn1)=O 52536,c1(CCC(=O)NCC(C)NC(=O)C(F)(F)c2ncc[nH]2)nnc(C2CCCC2)o1 52537,C1(OC)CN(C(=O)Cc2cccc(Cl)c2)CC1NC(=O)CC1CCC(C(N)=O)O1 52538,C1(SCCNC(C2CCCC(C)C2)=O)CN(c2ccc(C#N)nc2)CCN1C 52539,N1(C(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(c3ccccc3)=O)CC2)C1 52540,C(C)(C(=O)NCCC(=O)NC(C)C=CC(N1CCCC1)=O)OCOC 52541,c1(NC(CC2N(c3nccc(OC)n3)CCOC2)=O)cc(Br)cnc1I 52542,c1(CNC2(C)C(C(C)O)C2)ccc(C2CC2)cc1 52543,C(=O)(CC1CCc2ccccc21)NC1(C2CN(C(C(C)n3cncn3)=O)C2)CC1 52544,C(=O)(CS(=O)(=O)C1CCCC1)N(CCNC(c1cc(C(=O)OC)n(C)c1)=O)C 52545,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52546,C(=O)(C(C)(C)CCCC(=O)NCC1(O)CN(C(c2c(C)nn(C)c2F)=O)C1)OC 52547,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52548,C1(CNC(Cc2c(C)n[nH]c2C)=O)CN(C(C2CCCOC2C)=O)C(C)(C)C1 52549,Cc1nc(C(N2CC23CN(C(c2c[nH]nc2C)=O)C3)=O)cc(O)n1 52550,c1(NC(=O)OCC(c2n(C)ccc2)=O)c(F)ccc(Cl)c1Br 52551,CC(N=c1ccc(Br)c(S(=O)(=O)NCCCS(C)=O)[nH]1)c1cccc(F)c1F 52552,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCC2(NC(=O)CC3CCCCO3)CC2C1 52553,N1(C(c2ccc3c(c2)OCC3)C(=O)NCC)CCC2(CC1)OC1(CCCOC1)O2 52554,C1(CNC(CCC)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52555,N(C(=NCCCF)NCc1ccco1)CCc1cc(OCC)c(C)cc1 52556,C#Cc1cccc(C(N2CCC(C3CCN(C(=O)CN(C)C)CC3)C2)=O)c1C 52557,c1(N2C3CC(CNC(c4c(C)cn(C)c4)=O)CC2CC3)cc2nnc(C)n2cn1 52558,C(=O)(C1CC(=O)Nc2cc(F)ccc21)NCCNC(CSC(C)C)=O 52559,CON(CCC(=O)N1CCCC(C)(C#N)C1)C(=O)Cc1c(C)nn(C)c1C 52560,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCC2(C)CCCC2O)nn1C 52561,C(CC(F)(F)F)(c1ccc(F)cc1)NCc1n(CCOC)ncc1 52562,C1(CC)COCC1NC(=O)C(C)(C)NC(=O)C(C)=CC(C)(C)C 52563,c1(C(=O)NCCC2CCN(C(C(CC)C(=O)OC)=O)C2)ccc([N+](=O)[O-])cc1CC 52564,N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)(CCNC(=O)CC2OCCO2)C1 52565,C1(NC(c2c(CC)cco2)=O)CC1C1CCN(C(=O)COCCCN(C)C)CC1 52566,c1(OC(C)C)nc(C(=O)NC(C)(C)C(C)NC(=O)C(O)CN2CCCC2)ns1 52567,C(=O)(CC(C)C(C)C(C)C)N(CC)CC.CCCCCCCNC(=O)C(=O)N(CC)CC 52568,C1(NC(Cc2ccc(OC)cc2)=O)CC2(C1)CC(N=[N+]=[N-])C2.c12nc(cs1)CO2 52569,C12(CNC(=O)Cc3ccco3)CC1CN(C(=O)C(N1CCCC1)C1CC1)C2 52570,c1(C(N2CC(NC(C(C)NC(C)=O)=O)C(F)C2)=O)cc(Br)c(F)cc1Cl 52571,c1(C(N2CCC(CC(=O)NCC(CC)(C)C)C2)=O)nn(C)cc1C 52572,C1(C(N2C(CO)CC(NC(=O)CCC3CCC(O)CC3)C2)=O)CC2C=CC1CC2 52573,c1(OC)ccc(Br)c(C)c1C(=O)NC1CCN(C(c2cc(C)c(C)cn2)=O)C1 52574,C(CN=c1cc(-c2cccs2)nc[nH]1)(N(C(=O)Cc1cnccc1Cl)C)C1CC1 52575,C1(C(N2C3CC(NC(c4occc4Cl)=O)(C3)C2)=O)CCCCC12CC2(F)F 52576,c1(COC)cc(CC(=O)NCC(C)N(C)C(c2c[nH]nc2C(C)C)=O)no1 52577,C(=O)(CC1=CCCCC1)NC1(C(N(C2CCN(CCCO)C2)C)=O)CC1(C)C 52578,c1(NC(CC=C)C)cc(N2CCCC(OCC)C2)nc(C(F)(F)F)n1 52579,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CNC(C1CC1(F)F)=O 52580,CC1CN(C(=O)C(=O)C(F)(F)F)CC2(CCN(C(C)C(=O)NCC(F)(F)F)C2)O1 52581,N1(C(N2C(CC(=O)N(C)C)COCC2)=O)C2CCC1CC1(C2)CC1(F)F 52582,C(=O)(CCCC1CC1)N(C(C)C(=O)N(C)CC1(CO)CCCC1)C 52583,CC(C)C(O)CC(=O)NC12CC(NC(C3(C)CC3(F)F)=O)(C1)C2 52584,c1(SCC)nc(=NC(CNC(=O)CCC2CCCCCC2)CO)s[nH]1 52585,CC1(CNC(=O)C(C2CC2)C2CC2)CCCN(C(C2C3CCC(F)(F)C23)=O)C1 52586,c1(C(N(C(CCC(=O)OC)(C)C)C2CC3CNC2C3)=O)cn2ccccc2n1 52587,c1(OCC2N(C(c3c(OCC)cccc3OC)=O)CC2)c(F)cc(OC)cc1F 52588,c1(C(C(=O)NCC(C2CC2)NC(C2(CC)CC2)=O)=O)cc(F)c(F)c(F)c1 52589,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52590,C1(CNC(c2cn(CCOC)nc2)=O)CN(c2ncncc2I)CCC12CCOC2 52591,C(=O)(NNc1cc(C(F)(F)F)cc(Br)c1)c1c(C)nn(C)c1C 52592,CC(C(=O)NC(C)(C)CCCNC(=O)C(C)(C)CC1CCOC1)C(C)(F)F 52593,C1(NC(c2nc(COCC)sc2)=O)CN(C(=O)CCc2ncc(C)[nH]2)CC1F 52594,c1(C(N2CCCC(CN(C(c3c(CC)nc[nH]3)=O)C)C2)=O)ccnc2[nH]nnc12 52595,c1(C(C)C)nn(C)c(Cl)c1C(=O)NC(C1CCN(c2nc(C(F)(F)F)ns2)C1)C 52596,Cc1cc(C(=O)NC2CC3CCC2(NC(=O)CC2CC(C)(C)C(=O)N2)C3)nc(O)c1 52597,O=C1CC(CC(=O)N2CCC3(CC2)CC3NC(c2ccsn2)=O)=NN1 52598,C1(NC(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CS(=O)(=O)C2)=O)C1 52599,N1(C(CCC=C(C)C)C(=O)Nc2cccc(Cl)c2)CCc2c(N(C)C)cccc21 52600,CC1=C(C(=O)N2CCC3(C2)CN(C(=O)CSc2nncn2C)C3)CCS1(=O)=O 52601,C1(CC(=O)N(C)CCOCCN(C)C(C2SCCC2C)=O)(CC)CCCC1 52602,C(=O)(CC(C)CN(C(c1cc(C)nn1C)=O)C(C)C)OCC 52603,C1(C(N2CC(C3(NC(C4N(CC)CC4)=O)CC3)C2)=O)COCCN1CC(F)F 52604,C1CCCCCNC(=O)c2cn1nn2.C1(C(=O)NC(C(=O)OC)C)OCCC1C 52605,c1(CC(=O)N(CCNC(=O)CCC2CCC2)C2CC2)ccc(Cl)nc1 52606,N#CC1CCCC1C1CCN(C(c2ncsc2C(F)(F)F)=O)CC1 52607,CC1CN(C(C23CC2COC3(C)C)=O)CCN1C(c1[nH]cnc1C#N)=O 52608,CCCCC(C)C(=O)N1CC2(CC2)CC1CNC(=O)CCCN1C(=O)CNC1=O 52609,C1(CC)CCCCC1C(=O)N(C)CCN(C(c1cc(Br)co1)=O)C(C)C 52610,C1(NC(C(C)=C(CC)C)=O)CC2CC1CC2C(=O)N(C)Cc1ccccc1O 52611,c1(NC(CCCCn2cc(NC(C(COC)C)=O)nn2)=O)ccc(F)c(Cl)c1 52612,C1(CNC(CSCC(C)C)=O)CN(C(=O)C(c2ncccc2F)(F)F)CCN1C 52613,Cc1cc(C(=O)NC2CCN(C(=O)CSc3n[nH]c(=N)s3)CC2C)nnc1C 52614,C(=O)(C1CCCc2nncn21)NCCN(C(=O)C(C)n1ccnc1)CC 52615,C1(NC(C2(CN(C)C)CCCC2)=O)CCCN(C(=O)CCC2CNC(=O)N2)CC1 52616,C1(NC(C2(C)C=CCC2)=O)CN(C(c2ccc(C(N)=O)c(Cl)c2)=O)CCC1CO 52617,C(=O)(C(O)CC(C)C)N1CCC(CCNC(Cc2c(C)cccc2)=O)C1 52618,C1(CNC(C(N2CCN(C)CC2)C2CCCC23CC3)=O)CN2CCC1CC2 52619,C1(N(C(CC2(OCC)CCC2)=O)C)CCC(NC(=O)C=Cc2nc(C)cs2)CC1 52620,C(=O)(C1CNC(=O)c2ccnn21)N(C(C)CNC(=O)CN(C)S(N)(=O)=O)C 52621,C1(N(C(=O)COC2CCCCC2)C)CCCN(C(=O)CCC2CC2(C)C)C1 52622,N1(c2n(C)nnn2)CC2CC(NC(C3CN(c4nncs4)C3)=O)C2C1 52623,C(=O)(CCCC(F)F)N1C(CNC(=O)CC23CC(C2)C3)CC(OC)C1 52624,c1(C(=O)NCC2N(C(c3ccc(C)nn3)=O)CC2)ccc2scnc2c1 52625,C(C)(C(O)C(=O)N1CCC(CNC(=O)C(=O)Nc2cccc(C)c2)C1)OC 52626,C1(CNC(C2(COC)CCOC2)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)CC1 52627,c1(C(=O)NCC(C)NC(C=CC=C)=O)csc(Cc2cccnc2)n1.C1CO1 52628,C1(C(C)C)CCCN(C(=NCC2CC3CC3C2)NC2CCC2)C1 52629,c1(CNC(c2c(CC)noc2)=O)cc(F)ccc1C 52630,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52631,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52632,N1(C(C(C)CN2CCOCC2)=O)CCC2CN(C(c3cc[nH]c3)=O)CC12 52633,c1(COCC)ccc(C(=O)NC(C)C(C(C)C)NC(c2ncccc2F)=O)cc1 52634,CCS(=O)(=O)CC(=O)NC(CCNC(c1cnc(CC(C)C)[nH]1)=O)C(C)C 52635,c1(CN(C)C)ccccc1-c1cnc(F)c(C(=O)NC2CCCC(F)C2)c1 52636,CC1CC(N(C)C(=O)CCN2CCN(c3ccccc3)CC2)C1(C)C 52637,c1(C(COC(C(C)=CC(C)(C)C)=O)=O)cc(C)ccc1C 52638,C1(C(CC)C(=O)N2CC(N(C)C(C3CCCO3)=O)C2)CCC(C)CC1 52639,C1(CN2CC(C(=O)OC)C(c3ccc(Cl)c(Cl)c3)CC2)C2Cc3ccccc3C12 52640,C1(C(=O)NC(C2(O)CCN(C(C3(C)CCCC3)=O)C2)C)CCCOCC1 52641,N1(C(CC2CCCN(C(CCCC(=C)C)=O)C2)=O)CCn2ccnc2C1C 52642,c1(C(c2n(CCOC)nnn2)NC2CC(CC(C)(C)C)C2)cccc(C)c1C 52643,c1(C(=O)NCC23CC(NC(=O)COc4ccccc4)(C2)C3)ccc(F)cc1F 52644,c1(C(N(C(CNC(c2csc(=N)[nH]2)=O)C2CC2)C)=O)cnc(-c2ccccc2)o1 52645,N1(C(C(Cc2ccc(O)cc2)NC(C)=O)=O)CC2CCC(C1)N2C(C1(F)CC1)=O 52646,C1(c2nnnn2C2CCCC2)(NC(c2ccn(C)n2)CC)CC2CCC2C1 52647,Cc1cc(F)c(N)cc1C(=O)NC1CC(F)CN(C(c2nnc(O)nc2O)=O)C1 52648,CC(C)CC(C)C(=O)N(CCCNC(=O)CCc1nnc(S)nc1O)C 52649,CC(C)C(C(=O)N(C)CC1CN(C(=O)COC2CCOCC2)C1)CC(F)(F)F 52650,N1(C(c2cn(CC)nc2C2CC2)=O)CCC(CO)C(NC(=O)C(Cl)=CCl)C1 52651,N1(C(C(CCC)NC(N)=O)=O)CCC2(C=C(C(=O)N(C(C)CSC)CC)C2)C1 52652,N(C(=NCCCCl)N1CC(C)(C)OC2(CCC2)C1)C1CC(C)OCC1 52653,CCCCC(C(=O)OC)NC(c1cc(C)[nH]n1)=O.C1(=O)CC2(CC2)N1 52654,CN1CCC(C(=O)N(C2CCCN(C(=O)CCc3nncs3)C2)C)C1=O 52655,S(=O)(=O)(c1cccc(F)c1C)CN(C(CC(=O)OC)CO)C1CC1.c12ccc([nH]1)C2 52656,C(=O)(CC(C)CC(F)(F)F)NCC1CN(C(C(C)=C(CC)C)=O)CC12CC2 52657,c1(CC)ccc(C(N2CCNC(=O)C2)C(=O)NCCC2CC2)nc1 52658,C1(NC(CCCC#C)=O)C2CC1CN(C(c1ccnn1CC(C)C)=O)C2 52659,c1(CCC(=O)NCC(CNC(CC2C(C)C2)=O)CO)cnc2ccccc2c1 52660,C1(NC(=O)CC(F)F)CC2CC(C1)CN(C(=O)CC1CCS(=O)(=O)C1)C2 52661,N1(C(C2N(C(C(CC)C)=O)CSC2)=O)CCC(O)(CC2(O)CCSCC2)CC1 52662,c1(C(=O)NCCC2CCCN(C(c3cc(OC)ncc3)=O)C2)cc(C#N)[nH]c1C 52663,c1(C(c2n(CCCC)nnn2)NCC=C)cc(C)ccc1C.C(C)CCCCO 52664,CN1CCN(C(c2ccn(C3CCC3)n2)=O)C(C(=O)NC2CCC2CCO)C1 52665,C1(NC(C(C)C)C(N)=O)CC2CCC(C1)N2C(=O)CN 52666,c1(COC)ccc(C(=O)NC2CN(C(=O)C(n3cc(Br)cn3)C)C2)o1 52667,c1(C(=O)NC(C2CCN(Cc3ccccc3Cl)C2)(C)C)cnc(C(N)=O)cn1 52668,c1(SC)cc(C(=O)N(CC(O)CN(C)C(c2ccc(C)cc2)=O)C)c(Cl)cc1Cl 52669,CCC(C)CC(C)N(C(=O)C(CCOCCO)NC(=O)C=CC(F)(F)F)C 52670,c1(CNC(C2CC(=C)CN2C(=O)Cn2cccn2)=O)cccc(O)c1F 52671,c1(C(N2CC(CC(C)NC(=O)CSCC(C3CCCC3)=O)C2)=O)ncccc1N 52672,C(CC(C)C(=O)N(C(CNC(c1coc(C(C)(C)C)n1)=O)CC)C)=CC 52673,C1(CN(C)C(C2(n3ccnn3)CC2)=O)CCCN1C(c1cnc(C2CCCO2)s1)=O 52674,N1(C(C(=Cc2ccco2)C)=O)CCCC2(C1)CN(C(=O)C(O)CCCC)C2 52675,C1(C(=O)OC)CCC(C(=O)OC(N2CCC2CO)=O)CC1.N1(C)CCCC1CO 52676,c1(CC(=O)NCC2(F)CCC(NC(C(CC)F)=O)C2)cc(OC)ccc1F 52677,CN1C(=O)Cc2c(C(N3CCN(C(C4COCCO4)=O)CC3CO)=O)cccc21 52678,c12ccccc1C(=O)N2.C1(C(=O)NCC=CCCC(C)C)CC1C1CCC1 52679,C(=O)(C(C)CC1CCCC1)NCC(CC)N(C(=O)C(C)OCCc1cccs1)C 52680,CCC(C)(C(=O)NCC1CN(C(c2cn(CCOC)nn2)=O)CC1O)OC 52681,n1(CC)cnc2c(N(C)CC3CCCC3(F)F)[nH]c(=NC3CCCSC3)nc12 52682,n1(C(C(=O)N(CCCNC(C(C)=C(C)C)=O)C2CC2)C)nc(C)cc1C 52683,O=C(CC1CCN1C(=O)C(F)n1cccn1)N=c1ccn(-c2ncccc2Cl)[nH]1 52684,C1(C(=O)NC(CN(C(=O)C=NOC)CC)C)CCN(c2cnccn2)CC1 52685,N1(C(c2nc(C(=O)OC)sc2)=O)CCC(NC(=O)CCc2cnn(C)c2)C1C 52686,c1(NC(N2CCCC(c3n(C)ncc3)C2)=O)ccc(F)c(Br)c1F 52687,c1(OC)cc(Cl)c(C)cc1CNC(=O)C(=O)Nc1cc(OC(F)F)cc(C)n1 52688,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(C)cc1C)=O 52689,C(Cn1cncn1)(C(=O)NC1CN(C2CCCCC2)C1)NC(c1ncc[nH]1)=O 52690,c1(OCC(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 52691,Cc1c(Cl)ccc(C(=O)NC2CCC(CNC(c3ccon3)=O)C2)c1N 52692,c1(CN(C(c2cnc(Cl)s2)C(=O)NCCC2CC2)C)cc(Br)cc(O)c1O 52693,Cc1nc2ccc(C(=O)NC(CNC(C3CC(=O)N(C)C3)=O)C(C)C)cc2s1 52694,c1(C(N2CCC(NC(CC3CC(C)(C)OCC3)=O)C2)=O)cc(Br)cn2ccnc12 52695,C12(NC(CC3(COC)CC3)=O)CCCC1N(c1nc(C(C)(C)C)ns1)CC2 52696,c1(NC2(C3CN(C(C(CC)CCNC(C)=O)=O)C3)CC2)[nH]c2cc(C)ccc2c1C 52697,C(CCS(=O)(=O)N(C1CCN(C(=O)C(C)N2CCCC2)C1)C1CC1)OC 52698,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 52699,N1(C(CCc2ccc(C)cc2)=O)CC2CC(C1)C2NC(=O)COC1CCCOC1 52700,CC(CCCO)C(=O)NC1CC(C)(NC(=O)CCCOCCOCC#N)C1 52701,c1(C(=O)NC2C(CNC(c3ccnc(-c4ccccc4)n3)=O)C2)cc(F)cnc1O 52702,C1(NC(C(c2ccc(OC)cc2)=O)=O)CCN(C(c2ccsc2Cl)=O)C(C)C1 52703,CC1(C)CC(NC(C2CC(F)(F)C2)=O)CN(C(c2ccoc2Cl)=O)C1 52704,Cc1cc(C(=O)Nc2nc(Cl)cc(Cl)n2)cc2nc[nH]c12 52705,c1(OCC)ccccc1C(=O)NC(c1ccccc1)CNC(C1CC12CCC2)=O 52706,c1(CC)cc(CC(=O)NC2(CCCNC(=O)C(C3CC3)C3CC3)CC2)n(C)n1 52707,c1(C(=O)NC2CC(C)(CC)N(C(=O)C(C)NC(N)=O)C2)ccc(OC)c(F)c1N 52708,n1(CC(=O)NCC(CNC(CCC(CC)C)=O)F)ccc(=O)c2ccccc12 52709,Cc1c(C(=O)NCCN(C(c2cnc3ccoc3c2)=O)C2CC2)cccc1C#N 52710,CC(C)(O)C#CC(=O)NC1CN(C(=O)CCNC(=O)C=CCl)CC1(C)C 52711,Nc1cc(F)c(C(N2CC=CC(NC(=O)C(O)CC3CCCC3)C2)=O)c(F)c1 52712,CC1(C)CN(C(c2ccn(C3CCCC3)n2)=O)C(CNC(c2ccsn2)=O)CO1 52713,c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)CC)coc2c(F)cccc12 52714,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(C)CC2)CC1)=O 52715,C(=O)(C1=CS(=O)(=O)CCC1)NCC1C2N(C(CCSC)=O)C(CC2)C1 52716,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 52717,c1(C(=O)NCCCC2N(C(c3cc(C(=O)OC)[nH]n3)=O)CCC2)n[nH]c(C)c1C 52718,c1(C(N2C(CNC(CC(=O)OC)=O)CC2)=O)cc(C(F)(F)F)ccc1Cl 52719,N1(CC(=O)OCc2ccccc2)CCN(CC2CCCC2)CC1 52720,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 52721,N1(C(C(C(C)C)NC(C)=O)=O)CCCN(C(c2sc(F)cc2Cl)=O)CC1 52722,c1(-c2n(C)ncc2)cccc(C(N2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)=O)c1 52723,C1(O)(C(C(=O)NCC2CCCOC2)(F)F)CCOCC1.O=C1CC2(CC2)CN1 52724,c1(OCC(=O)NC(C)C(CO)NC(=O)COCS(C)(=O)=O)cccc(C#N)c1 52725,c1(C(=O)NC(C)CC(C)(C)O)cc2c(s1)CCCC2 52726,Nc1ccc(C(=O)NC2CCN(CCCNC(c3ccc(F)o3)=O)C2)nc1N 52727,c1(NCc2c[nH]c(=NC)s2)ccc(-c2cn(-c3c(C)cccc3Cl)nn2)c(F)c1 52728,CC(CCO)C(=O)N1CCC(C(C)NC(=O)C(c2ccc(Cl)cc2)=O)C1 52729,C=CCC(CNC(c1ccc(C#N)cc1)=O)C(=O)N1CC(C)(COC)C1 52730,N1(C(C(=O)NCC)=O)CCC(NC(c2cn(CCF)nn2)=O)C(F)C1 52731,C(=O)(CC(C)CN=c1[nH]cnc(Cl)c1N)OCC 52732,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 52733,C1(C(C)C)CCCN(C(C2CCC=CC2NC(=O)CN2CC(C)(C)C2)=O)CC1 52734,c1(NC(CC2N(C(C(CC)CC)=O)CC(O)C2)=O)cc(C#N)cnc1C 52735,c1(C(N2CC(NC(c3cc(C)nn3C)=O)(CO)C2)=O)cccc(S(=O)(=O)CF)c1 52736,C1(CO)(NC(C(c2cnn(C)c2)OC)=O)CC(NC(C2CC2c2ccccc2)=O)C1 52737,C1(CCNC(CCNC(=O)NC)=O)CN(C(=O)Cc2ccnn2C)CCO1 52738,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)Cc2cccs2)C1(C)C 52739,C=C(C)CCCC(=O)N1CCN(c2cc(OC)nc(OC)n2)CC1 52740,c1(C(N(C2CC2)CC2CCN(C(COC(CC)(C)C)=O)C2)=O)cc(N)ccc1O 52741,S(=O)(=O)(CC(=O)NC1CN(C(=O)CC2(n3cccn3)CC2)CC1C)N(C)C1CC1 52742,c1(C(=O)NCC(CCNC(C(c2c(C)nn(C)c2)C)=O)(C)C)cn2c(n1)SCC2 52743,N1(C(c2c(CC)c[nH]c2)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 52744,N1(Cc2cc(C(N3CCCCC3)C)no2)CC(C)OC2(CCOCC2)C1 52745,C1(C)(C(N2CC(CN(C)C(C3OCC3(C)C)=O)OCC2)=O)CCCCNC1=O 52746,c1(C2CN(CCN(C)C(c3csc(C(C)(C)C)n3)=O)C2)ccc(Cl)cc1 52747,c1(C(=O)NC(CC)CNC(c2cc(C(C)(C)C)c[nH]2)=O)cc(SC)n(C)n1 52748,CC1=C(C)CC(C)(NC(c2cnc(CNC(=O)CC(C)OC)nc2)=O)CC1 52749,N1(C(CCCC=C)=O)CC2(CCN(C(C3CC3c3cscn3)=O)CC2)C1C(C)C 52750,Cc1c(C(=O)NCCc2cn(-c3cccc(F)c3)nn2)oc2ccccc12 52751,C1(C(=O)NC2CN(C(C3CC4(CC4)C3)=O)CCC2CO)OCC2COCCC12 52752,c12nc(co1)C1CN(C(=O)C(C)N3CCCC23)C1.C1(OC)CC(OC(C)=O)C1 52753,C(=O)(C(O)CC(C)C)N1CCC(CN2CCN(C(c3c(C)nns3)=O)CC2)C1 52754,C=CC(C)(C)C(=O)NCCN(C1CCCCC1)C(=O)CC1CC1C1CC1 52755,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 52756,C=CCC(CC)C(=O)NCC1CN(C(c2nonc2CC)=O)CC1C 52757,c1(C(N(C2CN(C(COCC(C)C)=O)CC23CC3)C)=O)cc(S(N)(=O)=O)cn1C 52758,N1(C(CC2CCN(C(c3c(CC)nccn3)=O)CC2)=O)CCc2ccsc2C1 52759,C1(CN(C)CCO)CCCCN1C(=O)CCC1CCCC(O)C1.C1CCN1.C(N)=O 52760,C1(C)(C(=O)Nc2c(C(=O)OCC)scc2)CCN(C(=O)Cc2cc[nH]c2)C1 52761,C1(C(=O)NCC(COC)C)CCN(C(=O)CC2C(C)(C)C2(C)C)CC1O 52762,C1(CNC(C(=O)N(c2ccc(C)cc2)CCN)=O)CC2CCC1N2C(=O)C1CC1 52763,c1(SC)nn(C)cc1C(=O)NCC1(O)CN(C(=O)C=C(C2CC2)C2CC2)C1 52764,C=CC(C)(O)CC(=O)NCCOC1CCN(C(C2CCC(=O)NC2)=O)CC1 52765,N1(C(C(CC)F)=O)CC(C)(C)OC2(C1)CN(C(c1nn(C3CC3)cc1Cl)=O)C2 52766,C1(NC(=O)CCn2cccn2)CCCCCN(C(c2cc(C(N)=O)co2)=O)C1 52767,Cc1ccc(F)c(C(=O)NCC2CC(C)N(C(=O)CSCc3ccncc3)C2)n1 52768,c1(SC)nc(NC(N2CCC(O)(c3cccc(C(F)(F)F)c3)C2)=O)c(C)o1 52769,c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)cnc2ncccn12 52770,C(CN=c1nc(N2C3CCC2CC3)c2cc(Cl)ccc2[nH]1)(OC)Oc1ccccc1 52771,c1(C(C)C)nc2cc(C(=O)NCCC(C)(C)C)cc(C(C)(C)C)c2[nH]1 52772,c1(OCC)ncc(NC(C2CC(CNC(c3cccc(Cl)c3Br)=O)C2)=O)cc1Cl 52773,N1(C(COC)=O)CCCCC2C1CCCN2C(c1csc2cc(C)ccc12)=O 52774,CCC(CC)C(F)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 52775,c1(OC)cnccc1C(C(=O)NCc1ccccc1F)N(C)Cc1occc1Br 52776,C1(C(C)NC(C2N(CC)CC2)=O)CCN(C(=O)CC2CCC(=O)C2)CC1 52777,C1(CS(=O)(=O)NC2CCCN(C(C)(C)C)C2)CC(c2ccccc2[N+](=O)[O-])=NO1 52778,C(C(=O)NNC(=O)C(C)(C)C)N1CCC(C)CC1 52779,C1(NC(CC=C)=O)CCC(NC(c2cc(C)c(C)s2)=O)CC1 52780,C(COC)(N=c1cc(C)nc(N2CCN(C)CC(CSC)C2)[nH]1)c1c(OC)cccc1 52781,N(C1CCc2c(Cl)ccc(F)c21)c1cc(CCN2CCN(C)C(=O)CC2)ncn1 52782,C1(N(C(C=CSC)=O)C)CCCC(N(C)C(c2cc(N3CCCC3)ccn2)=O)C1 52783,C(F)(C(=O)NC(CNC(=O)Cn1cncn1)C1CC1)=CC 52784,N1(C(=O)CC2CSCCS2)CCC2(C1)CN(C(c1ccc(Cl)c(F)c1)=O)CCO2 52785,c1(SC(c2cn(CC(c3ccccc3)=O)nn2)C)nc(C)ccc1F 52786,C1(SC)CCC(N=c2ccnc(N(C)Cc3cc(Cl)ncc3F)[nH]2)CC1 52787,c1(C(CC(=O)NC(C(C)NC(Cn2c(C)ccn2)=O)C)O)ccc(Cl)c(Cl)c1 52788,NS(=O)(=O)c1ccc(-c2nnc(N3CCCC4(CCO4)C3)n2CC2CC2)cc1 52789,C1(C)(C(N2CCOCC(NC(CSCCC)=O)C2)=O)CCCNS1(=O)=O 52790,C(=O)(C1CCCc2scnc21)N1CC(O)CCC(NC(c2n[nH]c(C)c2Cl)=O)C1 52791,N1(C(C(CC2CC2)OC)=O)CCCC(CN(C(=O)C(c2ccccc2)C)C)C1 52792,Cc1oc(Cl)nc1C(=O)N(CCCC(=O)NCC1CCN(C(C)C)C1)C 52793,C1(C#N)(C(=O)NCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 52794,c1(C(CNC(c2conc2-c2cccs2)C)(C)C)c(F)cc(F)cc1F 52795,C1(CC)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(=O)CCc1ncc[nH]1 52796,CC(C)C(F)(F)CC(=O)NC1CCCC1NC(c1cc(Cl)cn1C)=O 52797,c12cnc(OC)c(c1)C(=O)N1CC(CC1C)CNC(=O)C2.C1(COC)CC12CC2 52798,c1(OCC)c(C(=O)NC(Cn2cc(CCC3CC3)nn2)CC(C)C)cnn1C 52799,Cc1nc(CCC(=O)NCC(C)CNC(c2ncoc2-c2cnn(C)c2)=O)cs1 52800,c1(CC(C)NCCO)ccc2c(c1)O2.C1(OCCOC)CCCO1.N1(C)C(=O)C1 52801,C1(NC(c2n(C)nnc2)=O)C2CCN(C(=O)CCCC(=O)OC(C)(C)C)CCC12 52802,C1(CCC(=O)OC)CCCCN1Cn1c(C(N2C(CCC=C)CCC2)=O)cnn1 52803,CC1CN(C(=O)COC(C)(C)C)CC(C)C1NC(c1c[nH]nc1OC1CC1)=O 52804,N1(C(C(C)NC=O)=O)CCC(CCNC(c2cc(CCO)on2)=O)C1 52805,c1(C(N(CCCNC(C2C(CC)CCC2)=O)CCO)=O)ccc2nccn2n1 52806,n1(CC)ncc2c(N3CC(F)(CNC(=O)CC(C)(C4CCC4)SC)C3)ncnc12 52807,C1(C(N(C2CCN(C(COCCOCC#C)=O)C2)C)=O)CCCN(S(C)(=O)=O)C1 52808,N1(C(=O)OC(C)(C)C)CCC2CCN(C(=O)Cc3ncccc3Br)C2C1 52809,C1(O)(NC(C(=O)N(CCC)CC)=O)CC2CCC1C2 52810,C1(C(=O)NCC(CNC(C2(CC=C)CC=CC2)=O)O)CC(F)(F)C1(C)C 52811,c1(OCCOC)ccc(-n2nc(C)nc2-c2sc(Br)cc2Cl)c(F)c1 52812,c1(CNCC2=CCCN(S(CCC(=O)OCC)(=O)=O)C2)ccc(F)cc1Br 52813,c1(OC)cnc(C(N2CC(NC(=O)COc3ccsc3)C(O)C2)=O)cn1 52814,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCCC3)C2)=O)C1(F)F 52815,C1(NC(c2scc(OC)c2)=O)COCCN(C(=O)C(F)(F)c2ccccc2)C1 52816,C(=O)(C(O)C(F)F)NCCCC(=O)N(CCCN(C(CC(C)C)C)C)C 52817,N1(C(c2ccc(C(C)C)nc2)=O)CCCC(NC(c2ccn(C)c2)=O)C1C 52818,c1(N2CCC(CC=C)C2)nc(N(C)Cc2sccc2C)c2ncn(C)c2n1 52819,N1(C(C2=CCCC2C)=O)CCC(NC(C2CC3CC(OC)C3C2)=O)C12CCC2 52820,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccn2)nc1 52821,N1(C(CCc2cn(C)nc2)=O)CCCC1(C)C(=O)NCCCN1CCCC1 52822,C#Cc1ccc(C(=O)NCCC(C)CCNC(=O)CSc2ccccn2)c(C)c1 52823,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCCC(NC(C2(C)CC(C)(C)C2)=O)C1 52824,c1(OC)c(-c2cn(CC3CC(O)CN(C(CC(CSC)O)=O)C3)nn2)cnn1C 52825,C1(NC(C2(Cc3ccccc3)CCC2)C)CCCCC1(C)O 52826,N1(C(CC=C(C)C)=O)CCCC2(CNC(C34CCC(C)(C3)OC4)=O)CCCC12 52827,C(CO)(CCCCNC(=O)C(c1ccc(Cl)s1)C)NC(c1c(C)nc(CC)o1)=O 52828,Cc1ccc2c(N3CCCC3(C)NCc3ccc(Cl)cc3CO)ncnc2c1 52829,c1(C(=O)NC(C(C)C)CCNC(=O)C(C#N)C2CC2)cccc2nc(C3CC3)[nH]c12 52830,N1(C(C2CCC(NC(C3CC(C(C)C)C3)=O)C2)=O)CC(O)C12CCOCC2 52831,c1(-c2cc3cc(C(C)C)sc3cc2)cn2c(n1)CN(C(c1cn(C)cn1)=O)CC2 52832,C(=O)(CN=c1ccc(C#N)c[nH]1)NCC(C)(C1CCC1)NC(=O)C(O)CC(F)F 52833,c1(CN(C(=O)C(c2ccccc2)=O)C)ccc(CNC(C2(O)CNC2)=O)cc1F 52834,CCC(C)(C)C(C(=O)NCC1CC1CNC(=O)C(C1(CO)CCOCC1)C)OC 52835,c1(C(N2CCCCC2CNCc2ccc(O)c(O)c2O)=O)cc2ccccc2o1 52836,C1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)(C)C2)NC(=O)CN(C)C1=O 52837,C1(F)(CNC(c2c(C)nsc2)=O)CCCN(C(C2CNC(=O)CC2C)=O)CC1 52838,c1(N2CC3N(C)C(CC3)CC2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 52839,C1(C(=O)NCCOC2CCN(C(c3cscn3)=O)C2)CCc2nc[nH]c2C1 52840,N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC2CCCN(C1)N2C(=O)CC1CCCC1O 52841,Cn1cc(C2CC(C(N3CCC(N4CCOC4=O)CC3)=O)C2)c(C2CCC2)n1 52842,N1(C(COCOC)=O)CCCOC(CNC(=O)CC2CCCCCC2)C1 52843,N1(C(CC(C(C)C)C)=O)CC2OCC(C(=O)NCCC3(O)CCC3)C2C1 52844,c1(C(=O)NCC2(O)CC(NC(C3CC(F)(CO)C3)=O)C2)cc2ccccc2o1 52845,Cn1cc(C(C)NC(=O)CN(c2cccs2)C(c2cocn2)=O)cn1 52846,N1(C(c2cnc(OC)nc2)C(=O)NC2CCOC2)CCn2c(CCO)nnc2C1 52847,C(=O)(C(C(F)(F)F)=Cc1ccccc1)NC1CCN(C(CN(C)C2CC2)=O)C1 52848,c1(NC(c2cccs2)=O)ccc(C(=O)NCC2CCN(C(=O)CSCC(C)C)C2)o1 52849,c1(-c2c(C(=O)N(c3ncccn3)Cc3cnco3)occ2)ccc(Cl)cc1 52850,c1(C(=O)NC(C2(CNC(CCN(C(CCC)C)C)=O)CC2)C)csc(Cl)c1Cl 52851,c1(CC(C)C)ccc(C(C)C(=O)NCC(O)CNC(C2CCOC(=O)N2)=O)cc1 52852,Cc1cc(=NC(=O)C(=O)C(C)(C)C)[nH]n1CCNC(C1CCN(C)S1(=O)=O)=O 52853,N1(C(C2(CC=C)CC2)=O)CCCC(C)(CNC(C2(C)CCCCC2)=O)CC1 52854,c1(C(N2CC(CNC(C(CC)F)=O)C(C)C2)=O)cc2cc(Cl)cnc2[nH]1 52855,c1(C(=O)NCCC(C)NC(c2c(CC)ncnc2)=O)c[nH]nc1[N+](=O)[O-] 52856,C1(NC(C(CNC(CCOCC)=O)CC2CCCC2)=O)CCCCCCC1O 52857,C1(C(=O)OCC)(CN)CC2CCC1C2.c12cccc(c1)COC(=O)CCC2 52858,CC(CCOC(F)F)C(=O)N1CCC(N(C(=O)COCC(C)(C)C)C)C1 52859,C(C)(C)(CCCCNC(C1(CC)CCOC1)=O)N(CC=C)C.C12(CC1)C(=O)NC2 52860,c1(CC(=O)NCCC(C)NC(C2C(CC)C2)=O)cc(S(N)(=O)=O)cn1C 52861,C1(CNC2CCC(C#C)CC2)CCOCC12CCC2 52862,C1(C(=O)NC(CCN(C(c2cnc(C(C)C)s2)=O)C)C)CCC(=O)N(C)C1 52863,N1(C(c2cn(C(C)C)nc2)=O)CCC(C(=O)NCC2CC(C)(C)O2)C12CCC2 52864,N1(C(C(C)NC(CC)(C)C)=O)CC(C)CC1C(N1CC(OC)CC1CF)=O 52865,c1(OC)ccc(OCC(N2CC(NC(c3cnn[nH]3)=O)CC2CO)=O)cc1C 52866,N1(c2cc(C(=O)OCC)nc(COC)n2)CCC2CC(NCCOC)CCC2C1 52867,O=C1CC2CC(C(N3CCCCCC3C(=O)NC3(CC4CCC4)CC3)=O)C1C2 52868,CC1CN(C(=O)C(C2CC2)NC(=O)C(F)C(C)(C)O)Cc2c[nH]nc21 52869,CCCC(C)CC(=O)OCC1CCC(C2CC2)O1.c1(CC(=O)N)cc(F)ccc1Cl 52870,Cn1cc(C#N)cc1NC(N1CC2(CC(N)C2)C1)=O 52871,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3(O)CCC3)C2)=O)ccnc(C)c1O 52872,C1(NC(C(C)n2ccnn2)=O)CCC(C)(NC(C2COCCOC2)=O)CC1 52873,C1(CC)CCN(C(=O)CC2(C)CCC2)C(C(=O)NC2CC(C)C2)C1 52874,N1(C(c2c(C)ocn2)=O)CCN(C(c2ccnn2CCOCCO)=O)CC1 52875,c1(C(=O)NC2CCC2NC(C2CCSCC2)=O)cc(OC(F)F)ncn1 52876,C(=O)(C(O)C(F)(F)F)N1CC(OCC)C(CNC(=O)CCc2ccoc2)C1 52877,c1(C(=O)NCC2CC(O)CN2C(=O)Cc2csc(Cl)c2)cnn2c1OCCC2 52878,C1(N(C(CC2N(CCC(C)C)CCC2)=O)CCO)CCN(C(C2CCCO2)=O)CC1 52879,N1(C(c2cnc(CCC)s2)=O)CCCC(N(C)C(c2ccn(C(C)C)n2)=O)CC1 52880,C12(C(=O)NCCOCCOCCNC(CC(C=C)C)=O)C3C4C1C1C2C3C41C 52881,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 52882,Cc1ccc(C=CC(=O)NC2CCC(NC(=O)Cc3cc(C)no3)C2)nc1 52883,N1(C(C2C(C(=O)OC)CC2)=O)CCC(N(C(=O)Cc2cocn2)C)C1 52884,C(C(C(=O)NC(C)Cc1ccnn1C)C(C)C)NC(Cn1ccc(C)c1)=O 52885,Cc1c(C(=O)NC2C=CCC(C(=O)NC3(c4cccs4)CC3)C2)cccc1F 52886,c1(C(=O)NCCC(CNC(C(C)OCC)=O)=C)cc(N(C)C)ncn1 52887,CC1(C(=O)N(C2CC(=O)N2)CCO)CCN(C(CC(F)F)=O)C1 52888,C1(NC(=O)CCc2ccc[nH]2)CC2CN(C(c3cccc(Cl)c3Cl)=O)CC12 52889,C1(NC(C2CCN(C(c3cn(CCC)nc3)=O)C2)=O)CCN(C)CC1C#N 52890,C1(C(=O)NC(C2CCOCC2)C#C)CCC(C)N1C(=O)CC1CCOC1 52891,C(CCN=C(Nc1ccc2c(c1)OCO2)N1CCOC2(CCCCC2)C1)OCC 52892,c1(C(N2CC(NC(C(c3ccccc3)OC)=O)C(O)C2)=O)ccc2cc[nH]c2n1 52893,Cc1cccc(C(=O)NCC2CCCC2NC(C2(O)CCC(C)CC2)=O)c1N 52894,N1(S(CC(=O)OCC)(=O)=O)CC(C(=O)O)C2(CCN(CC3CC3)CC2)C1 52895,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 52896,C1(O)(C(C)NC(C2CSCCS2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 52897,C(c1cccnc1)=C(C(=O)NC(CCOC)CNC(=O)CCc1cc(C)no1)F 52898,C1(CC(C)NC(=O)CCN2CCC2)CCN(Cc2cn(C3CCCC3)nn2)CC1 52899,C1(C(=O)NCC(C)CC2CCC2)CCC2CCC1N2C(=O)Cn1cnnc1O 52900,c1ccc2c(c1)CCC(Nc1n[nH]c3c1CCC3)CC2 52901,CC(CC(=O)NOCC1CC1)N(C(=O)C(CO)NC(N)=O)C 52902,C(=O)(CC(C(=C)C)OCC)N(C1CCCN(C(CC2(C(=C)F)CCC2)=O)C1)CC 52903,N1(C(C2(CC#C)CCCCO2)=O)CCC(NC(=O)Cc2ccco2)C(F)(F)CC1 52904,C(=O)(C1=CC2CCCC12)NCC(C)CNC(c1c(O)cccc1Br)=O 52905,N1(C(C(CCF)NC(C(CC=CCC)C)=O)=O)CCCNC(=O)C1 52906,C1(C(=O)NCC2CC3CC2C2CC32)CCC2CN(CCCO)CC2C1 52907,N1(C(C2N(C(Cc3cccc(C#C)c3)=O)CCCC2)=O)CC(F)(F)CCC1C 52908,c1(OCCC)ccc(NC(=O)OC2CC2(F)F)cc1OCCCCl 52909,Cc1sc2ncnc(N3CCC4CCC(NC(C5CCC(C)C5)=O)C3C4)c2c1C 52910,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 52911,c1(NC(C(N2CC3C(C)C3C2)C2(CC)CCC2)=O)ccc(N(C)C)cn1 52912,Cn1cc2c(n1)CCCC2C(=O)NCC(C)(O)CNC(=O)CC1(O)CCC1 52913,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2ccnc(Cl)c2O)=O)C1C 52914,C#CC1(CC(=O)NC2CC(F)(F)C2)COCCN1C(C(=O)OC)c1cscn1 52915,C1(C(N2CCSCC2C2CC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 52916,N1(C(CC(CC)O)=O)CC(C)CN(C(c2cc(F)n(C)n2)=O)CC1C 52917,Cc1c[nH]c(=NCCC(C(C)(C)C)NC(c2cc(F)ccc2Cl)=O)nc1O 52918,C1(C(=O)NCC(CN(C(=O)C(C)(C)N2CCCC2)C)(C)C)CCCCC1C(F)(F)F 52919,c1(C(CNC(=O)C(O)CNC(C2C3CCC2CC3)=O)OC)ccc(CO)cc1 52920,CC1CN(C(c2cnc(C3CC3)s2)=O)CCCN1C(=O)CC1CCCCC1O 52921,Cc1sc(O)nc1C(=O)NC1CCOC1C1CCN(C(C2(C)CCOC2)=O)CC1 52922,C(=O)(CCCCC(N)=O)N(C)CC1CCCN1C(=O)C(C)N(CC(F)(F)F)C 52923,N1(C(CC2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 52924,C1(C(N(C)CCNC(c2cccc(=O)o2)=O)=O)CC(C)(C)OC1(C)C 52925,C(=O)(C(C)(C)S(C)(=O)=O)N(C)CC1N(C(c2c(OC)n(C)nc2)=O)CCC1 52926,CC(C)CCC(=O)NCCNC(=O)CN.C1(NC(=O)C2CC2)CC1CC=O 52927,C1(C#N)(C(=O)NC(C)(C)CNC(C2CCCN(CC(F)(F)F)C2)=O)CC12CCC2 52928,N1(C(c2c(C)cnnc2)=O)CCN(Cc2cccc(F)c2Br)C2CC12 52929,C1(C(N(CCC(C)C)CCNC(=O)C(C)O)=O)CC(C)(F)C1 52930,N#Cc1ccc(=NCC(=O)N2CCN(C(C3(CF)CC3(F)F)=O)CC2)[nH]c1 52931,C(CN=C(NCc1cc(Cl)ccc1F)N1CCC(C2CCOC2)C1)N(CC)CC 52932,N1(C(CCn2ccc(C)n2)=O)CCC2(C1)CN(C(c1cc(C)c(C)cc1F)=O)C2 52933,c1(N(C(CC(C)C)C(F)(F)F)c2n(CC(=C)C)nnn2)noc2ccc(O)cc12 52934,Nc1c(C(=O)NCC(=O)NCCC2CCOC2)cccc1F 52935,C1(OC)(CNC(C2(n3cccn3)CC2)=O)CS(=O)(=O)C1.C1(COC)CC(C(=O)CC)C1 52936,c1(-c2nc(OC)c(C)s2)cc(N)c(C(=O)O)cc1F 52937,c1(C(=O)NCCNC(C(CC)CC2CCCC2)=O)cnc2c(F)cccn12 52938,CC1(C)CCCCC1(CO)NC(C1CCC1C1CC1)=O 52939,c1(OCC)ccc(C(=O)NC2(C)CCN(C(C3(C4CCCO4)CC3)=O)C2)cc1Cl 52940,C1(C(N(C2CCN(C(C3CC3C#N)=O)CC2)CCC)=O)CN(C)CCO1 52941,c1(C(=O)NC2(c3nc(C45OC(C)C(CC4)C5)on3)COC2)cc2ccccc2s1 52942,c1(CC)ncc(C(=O)NCCC2COCCN2C(=O)C(O)CCN(C)C)c(O)n1 52943,Cc1nc(N2CCSCC2C(=O)NCCc2cc[nH]n2)c2c[nH]nc2n1 52944,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 52945,C1(C(N(c2cccc(O)c2)CC)=O)CCC2CCC1N2C(=O)C(O)CC(C)C 52946,C1(C(N2CCC(C(C)C(=O)NCCN(C)C3CC3)C2)=O)CCNC(=O)C1 52947,C(=O)(C(CC(F)F)N(C(=O)Cn1cnnn1)C1CC1)N(C1CC(C(=O)OC)C1)C 52948,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(CN(C)C)C1)=O 52949,C1(C(N(CCC(=O)N(c2cnn(C)c2)C)C)=O)CC2CCC1C2 52950,C1(CC(=O)N(CC(=O)NC23CCCC2C3)C(C)C)COCC(C)O1 52951,CCCCCC(=O)N1CCC(C)(NC(=O)C(c2ccc(Cl)cc2)OC)C1 52952,C(=O)(C1CCCc2cn(C)nc21)NCCN(C)C(c1cc2ccc(F)cc2s1)=O 52953,C1(NC(Cc2cnc(C)o2)=O)CCC(C)N(C(c2c(Br)nnn2C)=O)C1 52954,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(c2ccc(C(F)F)o2)=O)C1 52955,c1(C(=O)NCC23CCCC2CN(C(=O)C=CCO)C3)ccc2ncncc2c1 52956,N1(C(c2c(C)n[nH]c2C)=O)CCCOC(CNC(c2c[nH]nc2Br)=O)C1 52957,c1(OC)cc(C(N2CCC(CNC(=O)CC3CN(C)C3)(OC)C2)=O)cc(F)c1F 52958,CC(C)CCC(O)C(=O)NC1CCN(C(c2cc[nH]c(=N)c2Cl)=O)CCC1CO 52959,N1(C(c2c(C)con2)=O)CCCC2(NC(c3ccccc3Br)=O)CC2C1 52960,Cc1oc(Br)cc1C(=O)NC1CC(CNC(C2(C)CNC(=O)C2)=O)C1 52961,N1(C(C=COCC)=O)CCOCC1CN(C(=O)COc1ccccc1)C 52962,Cc1c(F)ccc(-c2ccc(C(=O)NCc3ccncc3F)nc2)c1Cl 52963,c1(C(N(CC(CC)NC(=O)CCCF)C)=O)cc(C)nc2c(F)cccc12 52964,C1(CNC(CC2(OC)CCC2)=O)Cc2ccccc2CN1C(=O)CC(C)(C)F 52965,N1(C(c2cn(C)nc2C(F)F)=O)CC2CCC(C1)N2C(=O)CC1CC1C(F)(F)F 52966,C1(C(=O)NC2(COC)CN(C(C3CC34CC4)=O)C2)CC2CCC1C2 52967,N12CCOCC1C2=O.c1(COC)ccc(C(=O)NC(C)C2CC2)o1 52968,Cc1coc(C)c1C(=O)NCc1csc(CNC(c2cn(C)nn2)=O)n1 52969,n1(CCN(c2nnc(-c3c[nH]c4nccc-4c3)n2C)C)c(=O)oc2ccccc12 52970,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)cc1 52971,c12nccnc1C(=O)NC(C)(COC)C(=O)N2.C=CCNC1CC1CC 52972,Cc1cn2c(C(=O)NC(C)CCN(C(=O)CN3CC4CC4C3)C)c(C)nc2s1 52973,N1(C(COCCCN(C)C)=O)CC2CCC(NC(c3c(C)csc3C)=O)(C2)C1 52974,c1(C(N2CCC(NC(c3n(C)c(Cl)c(Cl)c3)=O)C2)=O)nc2c(s1)COCC2 52975,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CC(C)(CNC(C(C)OCCOCC)=O)C1 52976,CC1(C)CCN(C(C2CCCN2C(C)C)=O)C1NC(C1CCCC(=O)N1)=O 52977,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 52978,C(=O)(C1=COCCC1)NCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 52979,N1(C(Cc2c(C)con2)=O)CC(NC(=O)CCC2CCC(=O)N2)C(C)C1 52980,n1(CC)nc2c(c1C(N1CC3(C1)CN(C(=O)C(F)CCC(C)(C)C)C3)=O)CCCC2 52981,CN1CCCC1(C)C(=O)Nc1nc(CC(N2CCCCC2)=O)cs1 52982,C1(OCC)CC(NCCN2CCN(C3CCCCC3O)CC2)C12CCOCC2 52983,C(=O)(C1=CCCN(C(=O)Cc2ncccc2F)C1)NCc1c(C)ncs1 52984,C1(C(=O)NC(c2ccn(C)n2)C)CN(C(=O)C(O)C2CCC2)CC12CCC2 52985,c1(OC)cc(NC(=O)CN(C(=O)CC(C)c2ccccc2)C)ccc1F 52986,c1(C(N(C)CCOCCNC(C2COCC2c2ccccc2)=O)=O)cn(C)c(O)n1 52987,N1(C(=O)CNS(=O)(=O)C2CC2)CCN(C(C2CC3CCCC(C2)C3)=O)C2(CC2)C1 52988,c1(N(CCC)CCNC(=O)CC2=NNC(=O)C2)cnc2cc(F)c(F)cc2n1 52989,n1(C(C(=O)NCCCN(C)CC)C)cc(CCC2CC2)nn1 52990,C1(OCCN(C)C)CCN(C(CC2CCCO2)C(=O)Nc2ccccc2Br)CC1 52991,C#CCC(C)(C)C(=O)N1CC(O)(C(F)C(=O)NCC(CC)C(C)(F)F)C1 52992,CC1=NN(C)C(=O)C1CC(=O)NC1(CN(C)C(C2(C)CC2)=O)CC1 52993,C1(C(N(C(C)CNC(=O)CC2COCCO2)C)=O)CCCCN1C 52994,N12CCC(CC1)CN(C1C(CO)C1(C)C)C(C1CC1)C2=O.CCCOCC 52995,C1(NCc2ccc(C(=O)O)cc2)CC2(C1)CC(C(=O)NCc1cccnc1)C2 52996,c1(OC)ccc(C(N2CCN(C(C3(NC(C)=O)CCOC3)=O)CC2)C)nc1 52997,C1(C(N2CCC(C(C)NC(=O)Cn3cnnc3O)C2)=O)CCCC(=O)C1 52998,c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)COC2CC=CC2)ccc1F 52999,N1(C(C(CN(CC)CC)F)=O)CCCC2(CCN(C(=O)CN(C)C(C)C)C2)C1 53000,c1(NC(CC2CCN(C(COC(CC)C)=O)C2)=O)cc(C)cnc1O 53001,C1(C(N2CC(NC(Cc3ncc(CC)[nH]3)=O)C(C)C2)=O)CC(NC)CCO1 53002,CC#CCCC(=O)NC(Cc1cc[nH]n1)C(=O)NCC1(SC)CCC1 53003,c1(C(=O)NC2CC(C(C)NC(c3cnc(Cl)s3)=O)C2)nnc2ccccc2n1 53004,N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CCNC(C1(CC(C)C)CCC1)=O 53005,Cc1cc2nc(C(N3CC4(CCC4NC(=O)C4=CCCC4)C3)=O)cn2cc1C 53006,N1(C(C2(C=C)CCC2)=O)CC=C(C(=O)N2CC3CC2C2CC32)C1.N 53007,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CCCC1 53008,c1(-c2scc(C(=O)NC)n2)cncc(NC(C2CCC(=O)CC2)=O)c1 53009,Cc1cc(=O)c(C(N2CCOCC2CN(C(=O)CSCC#N)C)=O)cn1C 53010,c1(OC)ccc2cc1-c1c(nnn1C)C2.N(CP(C)(C)=O)CC1CC1 53011,CC1=CCC(C)(C(N2CCOCC(NC(=O)C=Cc3ccccc3F)C2)=O)CC1 53012,N1(C(C2=NOC(C)C2)=O)C2CCC1CC(NC(=O)Cc1ccc([N+](=O)[O-])cc1)C2 53013,c1(C(C)=O)ccc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2cccnc2F)cc1 53014,C1(C(=O)NCC=C)CCC(C)(C)N(C(=O)C(C)OCC)C1 53015,N1(C(C(C)NC(CC)=O)=O)CCCCC1CCCCc1cccc(C)n1 53016,Cc1cc(NC(C2CC(CCNC(c3[nH]ccc(=O)c3C)=O)C2)=O)ccc1F 53017,C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1oc(SC)cc1C)=O)CC2 53018,N1(C(C2CN(Cc3ncc(OC)nc3)C2)=O)CCCC2(COC2)C1 53019,N1(C(C(=O)NCC)Cc2ccccc2)CCOCC1(C)C1CC1 53020,C1(C(C)C)CN(C(=O)CN2CC=CC2)CC1C(=O)N(C1CC12CC2)CCO 53021,c1(CNC(CS(CC)=O)=O)nn(C)c2c1CN(C(=O)Cc1cnc(C3CC3)[nH]1)CC2 53022,C1(CC)(NC(c2nc(C)n(C)n2)=O)CCCN(C(=O)CC2CC2(Cl)Cl)C1 53023,N1(C(CN(C)C)=O)CCN(C(C2C(C(F)F)C2(C)C)=O)C(C2CCCC2)C1 53024,C1(NC(C(C)NC(C2CCCC2)=O)=O)CCN(C(=O)CSCC#N)C1 53025,C1(COC)(NC(c2[nH]ccc2SC)=O)CCN(C(c2ccc(SC(C)=O)o2)=O)C1 53026,c1(CC)cn(CCCC(=O)NC(COCC2CC(C)C2)Cc2ccccc2)nn1 53027,C(C(CC(=O)NCCC1CCC(C)(C)O1)NC(=O)C(O)CCSC)OC 53028,N1(CC(=O)N(C2(c3nn[nH]n3)COC2)C)CCCC(C(C)(C)C)C1=O 53029,C(=O)(CCC(C)SC)N(CC=CC(=O)NCC1(COC)CCCO1)C 53030,c1(CC(N2CCCC(C)(OC)CC2)=O)ccc2c(c1)CC(C)O2 53031,C(=O)(CCP(C)(C)=O)N1CCC(N(CC#C)C(c2nc(C)oc2C)=O)C1 53032,CC1CCN(C(=O)COc2ccon2)C1C(=O)N(C)CCN1CCOC1=O 53033,C(C(=O)C(=O)C(C)C(=O)OC(C)(C)C)(C(C)(C)C)NC(CCSC)=O.C(C)N 53034,Cn1ccc(C(=O)NCC2CCCN(C(C3CCNC(=O)C3)=O)C2)cc1=O 53035,c1(C(C)(C(=O)O)N(CCN(C)C)C2CC2)ccc(F)cc1 53036,N1(C(C2CN(C(C(CC3CCC3)OC)=O)CC2(C)C)=O)CCOC2(CCC2)C1 53037,C(C(CC(F)(F)CNC(=O)CC1(C#N)CCCCC1)OC)OC 53038,n1(COC)cc(C(=O)NCC#CCNC(c2cc(C3CCCCC3)no2)=O)cn1 53039,N1(Cc2c(Cl)cc(F)cc2F)CCC(S(=O)(=O)C2CCCCC2)C1 53040,C1(C(=O)NC2(CCNC(c3ccc(F)cn3)=O)CCC2)CC2C=CC1C2 53041,N1(C(C2(c3cccc(OC)c3)CC2)=O)CC2ON=C(C(F)F)C2C1 53042,c1(C(=O)NCC2(O)CN(C(c3cnc4[nH]nnc4c3)=O)C2)ccc(Cl)c(F)c1F 53043,N1(C(C=C(CCC)C)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53044,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1C)=O 53045,N1(C(C(n2ccc(C3CC3)n2)C)=O)CC2CC(CNC(=O)CC(C)(C)CC)CC1C2 53046,CCC(CC(=O)NC(C)(CNC(c1nc(C(F)(F)F)cn1C)=O)CO)C1CC1 53047,c1(C(n2ccc(CCC)n2)N(C)C)ccccc1OCCOC 53048,C(=O)(C(O)CC(F)(F)F)N(CCC(=O)N)CCN1CCC1.C(CN)OC(F)(F)F 53049,Cc1cc(C(=O)O)c(Sc2cn(CC(C)O)nn2)cc1[N+](=O)[O-] 53050,CCC(CC)N(CCOCC)CC1CC1C1CCCO1 53051,C1(C(N2CC(N(CCC)CC)C2)=O)CCC(CNC(=O)CCCF)O1 53052,C1(N(CCC(CC)(F)F)C(C2CCCC2)=O)CCCN(C)C1c1ccnn1C 53053,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53054,c1(CNC(C2N(C(CC(C)O)=O)CC2)=O)c(Br)ccc2cccnc12 53055,C1(CC=C)(C(=O)NC2CCN(CC)C2)CCN(C(c2conc2COC)=O)C1 53056,N1(C(=O)Nc2c(C(N)=O)occ2)CC2CC2C2CC12.c12cccc(c1)OC2 53057,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53058,C(C1=NOC2CCCC12)NC(COC1CC(NC(C(N)=O)=O)C1)=O 53059,C1(O)(CC(N2CC(CNC(=O)C(O)C3CCC3)C2)=O)CCCOC1 53060,c1(N2CCN(C)CC2)cncc(C#N)n1.c12ccccc1OC(=O)CO2 53061,c1(C(N2C(C(N3CCN(C)CC3)=O)CC(C)C2)=O)ccc(N=[N+]=[N-])cc1 53062,C1(CC(C(=O)OC)Nc2ncnc(OC)c2C)CCC2COCCC2C1 53063,c1(C(=O)NCC2(NC(C(CC)F)=O)CCC2)ncn2ccc(C)cc12 53064,CCC(C)CCC(O)CC(=O)N1CCCCC1CNC(=O)CCc1cccnc1 53065,C1(CNC(C2CCCC2F)=O)C2CC1N(C(=O)COC1CCCC1)C2 53066,c1(C(N2C(C(=O)Nc3n(C)nc(CC)c3Br)CC3CC32)=O)nc2c(s1)COCC2 53067,C1(C(=O)NCC2(COC)CC2)C2CN(C(C3(n4cnnn4)CC3)=O)CC12 53068,c1(NC(c2ccc(Cl)cn2)=O)cc2sccc2[nH]1.CC1CN2CC1C2=O 53069,CCC(C)(C)C(C(=O)N(CCNC(c1coc(OC(C)C)n1)=O)C1CC1)OC 53070,c1(C(=O)NCC2=CCN(C(CCSC)=O)CC2)ccc(S(=O)(=O)C(F)F)cc1 53071,c1(C(=O)NC(C(C(C)C)NC(C2CC(OC)C2)=O)C)cncc(N)c1C 53072,C(=O)(CC(N)C(C)(F)F)NCC(C(=O)OC)(C)O 53073,N#Cc1ccc(N2CCCC2)cn1.c12cccc(c1)OC(=O)O2.C(C)(C)(C)O 53074,c1(C(=O)NC(COCC)C(=O)NC2CCCC2CC)ccc2cnccc2c1 53075,CC1(C#CC(=O)N2CCCc3[nH]ccc32)CN(Cc2ccccc2)C1 53076,c1(C(C(=O)NC2CCCCC2)N(CC(=O)OC)C(C)C)cc(F)c(F)c(Cl)c1F 53077,N1(C(C(C)N(C(C)=O)C)=O)CCCN(C(c2cnc(C(C)C)nc2)=O)CC1C 53078,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53079,C(=O)(C(F)C1=CCCCC1)NC1C(CNC(c2c(CC)n[nH]c2)=O)CC1 53080,c1(C(C(=O)NC)N(CC(F)(F)F)CC#N)cc(C(C)(C)C)no1 53081,N1(C(C(C)SCC)=O)CCCC(C)(CNC(=O)CCc2cc(C)nc(C)c2)C1 53082,C1(NC(CCN(C(C2(C(=O)NC)CC2)=O)CCOC)=O)CCCC2(C1)N=N2 53083,C1(NC(C(C=C)C)=O)CCCCC1NC(=O)CCc1cc(C)no1 53084,c1(NC(C2(C)CCCN(C(C34CC(C3)C4)=O)C2)=O)nc2c(s1)COCC2 53085,CC(C)CCC(O)C(=O)NC(Cc1ccoc1)C(=O)NC(C1CCCCC1)C 53086,c1(C(=O)NCC(CN(C(C2CC(OC(F)F)C2)=O)CC)(C)C)cn2c(n1)CCCC2 53087,O=C(N=c1cc[nH]c2cc[nH]c12)C12CC1CN(Cc1cncc(O)c1)C2 53088,N1(C(C2N(C(c3ccc(NC)cn3)=O)CC(C)C2)=O)CCC(C)C(C)C1 53089,c1(N(C2CCN(C(c3c(C)nc(C4CC4)o3)=O)C2)CO)c[nH]c2ccc(Cl)cc12 53090,c1(C(C(C)NC2(C)CC(NC(C3CCCSC3)=O)C2)=O)csc(Br)c1 53091,C1(CNC(C(c2cncnc2)C)=O)CC2CCC1N2C(c1ncccc1Cl)=O 53092,C(C(C)(C)CC(=O)NCC1CCC(C(N)=O)O1)NC(c1c(C)oc(COC)n1)=O 53093,CCCC(C)(C)CC(=O)N1CCC(NC(=O)C(C)(C)CC(C)C)C(C)C1 53094,c1(C(=O)NCC2N(C(=O)C(C)(C)CF)CCN(C)C2)cc2c(o1)CCCC2 53095,C1(NC(c2cc(N)ncc2)=O)CC2(NC(C3CC34CCCC4)=O)COC1C2 53096,CON=C(C(=O)NC(CNC(=O)C(C)(C)C1CCC1)C1CC1)c1ccco1 53097,N1(c2nc(N(C)Cc3ncco3)c3c(n2)scc3)CCC2(CCC(O)CC2)C1 53098,c1(CC(=O)NC2C(C)N(C(=O)Cc3cnoc3)CCC2)ccc2c(c1)ncn2C 53099,N1(C(C(C2CCN(C(CS(CC)=O)=O)CC2)C)=O)CCc2nn[nH]c2C1 53100,c1(C(=O)N(C)CCC2C=CCC2)cccc(NCC(C)CN(C)C)n1 53101,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53102,c1(C(N(C(C)CCO)C)=O)n[nH]c2c1CN(C(C1(C)CCC(=O)N1)=O)C2 53103,c1(OCC(=O)NCC(CNC(CCCOCC=C)=O)F)cc(Cl)ccn1 53104,c1(C(CNC(C2(O)CCCC2)=O)NC(C23CCC(CC2)C3)=O)cc(F)cc(Cl)c1 53105,N1(C(CC2(C=C)CC2)=O)CCC(NC(=O)Cn2ccc(C3CC3)n2)C12CC2 53106,C1(NC(C(CSC)O)=O)CCCC(C(=O)NC2COC(C3CC3)C2)CC1 53107,N1(C(C(C)CC2CC2)=O)CCC(OCCCNC(=O)CC2(C(F)(F)F)CC2)CC1 53108,c1(OC)ccc(C(C(=O)OC)NCc2cc(CNC(C)=O)on2)c(C)c1 53109,c1(C(=O)NC(CC)(C)CNC(C2(C)CC2(Cl)Cl)=O)ccc(F)cc1OC 53110,C1(NC(CN(C(C)C)C)=O)CC(NC(c2c(F)cncc2Cl)=O)C12CCC2 53111,C=CC(C)C(=O)N(CCC(=O)NC(C1CCC1)C)C 53112,C1(C(=O)NC2CCCN(C(CCc3cnc(C)s3)=O)C2C)CCS(=O)(=O)C1(C)C 53113,N1(C(C(C)(C)CC2CC2)=O)CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1 53114,Cn1ncc(C(=O)NCC23CC(c4ccccc4)C2C3)c1C1CCOCC1 53115,Fc1cncc(NC(c2nc(Br)cs2)c2nnnn2C2CCCCC2)c1 53116,C(N=c1[nH]cnc(=N)[nH]1)C1C(C)CN(C(C2OCC2(C)C)=O)CC1 53117,C1(C(=O)NC(c2nc(CC)[nH]n2)C)CN(C(c2ncn(C)c2C)=O)CC(C)O1 53118,C1(CNC(C2(N(C)C)CCC2)=O)CC2(CCC2)CN1C(=O)CCC1CC(F)(F)C1 53119,C12(CO)CCCN(C1)C(c1nncn1C)C(=O)N2.n1(CC)cc(CSC)cn1 53120,C(=O)(C(C)P(C)(C)=O)NCC(C)N(C)C(c1occc1Cn1cccn1)=O 53121,C1(C)(CCNC(CC(=O)NCC)=O)CCN(C(c2[nH]nnc2C)=O)C1 53122,N1(C(CC2N(C)CC2)=O)CCOCC1CNC(c1cc(-c2ccco2)no1)=O 53123,C=CCC(C)(C)CC(=O)N(C1CCCC(NC(C2(C)CC=CC2)=O)C1)C 53124,c1(-c2ccc(N)s2)cc(OC)cc(F)c1F.CCOC 53125,n1(CC)nc(C(N2CC(O)CC2C(=O)NC(COC)CC(=O)OC)=O)c(C)n1 53126,CC(C)CC(O)C(=O)NCCCOC1CCN(C(=O)CSC(F)F)C1 53127,c1(OC)ncnc(N2CCOC(C(C)NC(c3cnccn3)=O)C2)c1OC 53128,N1(C(c2nccc(OC)c2)=O)CC2CCN(C(=O)CS(N)(=O)=O)C(C2)C1 53129,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C)CCN1C(=O)Cn1ccc(C(F)F)n1 53130,N1(C(=O)NC(C(C(C)C)C)CN(C)C)c2ccc(Cl)cc2OCC1C 53131,N1(C(C2CC(CC)N(C(C3CCCC3F)=O)CC2)=O)CC2CCCCC2C1C 53132,C12(C(N3CCCC(NC(CSCCCC)=O)(CO)C3)=O)COCC1CS(=O)(=O)C2 53133,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53134,CC1(C(N)=O)CCN(C(=O)CCC2CCOCC2)C1.c12cc(cs1)CNC2=O 53135,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53136,C1(C#N)(C(=O)NC2CCCC(CNC(c3ccc(CC)s3)=O)C2)CCSCC1 53137,c1(C(N2CC(CCCNC(=O)C=CC3CC3)OCC2)=O)cccc2[nH]cc(Cl)c12 53138,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)N(CCC)CC 53139,C1(C(N(C)CC2CCCCO2)=O)CC1C1CN(C(=O)CC23CCCC2C3)C1 53140,c1(C(=O)NC2(C)CN(C(C(CCC)CC)=O)C2)cc2c(C)cccc2[nH]1 53141,N1(C(CC(C)(C)C)=O)CC(NC(=O)CCCc2nc3ccccc3s2)C(C2CC2)C1 53142,N1(C(C(C)N=[N+]=[N-])=O)CC2COCC2(C(N2CCSC(C)C2)=O)C1 53143,C(=O)(C1OCCc2ccccc21)NCC(CN(C(c1c(COC)nn[nH]1)=O)C)O 53144,CC1(C)CC(C(N2CC(NC(=O)CCC=CBr)CC(F)C2)=O)OC1=O 53145,N1(C(C=C(C)C(C)(C)C)=O)CC=CC(NC(=O)C(c2ccc(F)cc2)N(C)C)C1 53146,CCCCCCC(CNC(c1nc(C)c(C)nc1C)c1nnnn1CCCF)CC 53147,CN1CCN(C(=O)CCc2nccs2)C(C(=O)NC2C3CCC(F)(F)C23)C1 53148,c1(N2CCC(NC(c3c(C)nco3)=O)C2)cc(-c2ccc(Cl)cc2)ncn1 53149,c1(C(=O)NCC2N(C(CCCC#N)=O)CCC2)n[nH]c2c1CC1CC21 53150,C1(NC(=O)CN(C)C(=O)OC(C)(C)C)CN(C(C2CC(=C)C2)=O)CC2CCCC12 53151,c1(CNC2C(C(=O)Nc3c(C(=O)OC)ccnc3F)C2)cc2cc[nH]c2cc1F 53152,N1(C(C(C=C)O)=O)CC2(CC(NC(=O)Cc3c(C)cc(C)nc3O)CO2)C1 53153,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53154,C(=O)(C(CCC(C)C)NC(=O)C(=O)NCC1CC1)NC1C(CC=C)COC1 53155,C1(NC(C2OCCN(C)C2=O)=O)CCCC12CN(C(=O)C=Cc1ccccc1F)C2 53156,Cc1cncc(C(=O)NC2C=CCN(C(C3(CC#N)COC3)=O)C2)c1 53157,C(C(C(F)(F)F)n1cccn1)OCCl.O=CCCCn1ccnc1 53158,N1(C(Cc2c(C)ncs2)=O)CCC(C(=O)Nc2ccccc2F)C(C)(C)C1 53159,c1(C(=O)NC(C2CCOC2)Cn2cc(CC(OC)OC)nn2)cc(Br)sc1Cl 53160,Cc1cccc(C)c1OCC(=O)NC1CC(Cn2cc(-c3cncnc3)nn2)C1 53161,NC1CN(C(c2cc(-c3cnc(F)nc3)[nH]n2)=O)CC1F 53162,C1(C(=O)NC2CCN(C(C(C)=C3CCCC3)=O)C23CC3)CCn2nccc2C1 53163,C1(NC(C(=O)OC)=O)(CNC(C2CCC(C)S2)=O)CCC(F)(F)CC1 53164,c1(C(N2C(C(=O)NCc3cnc(C)nc3)CC3CC32)=O)ccc(Cl)c(Br)c1 53165,c1(C(C)NC(=O)NC2C(C(C)C)CCO2)ccccc1OC(F)F 53166,CC(C)C#CC(=O)N1CCC(O)(N(C(=O)C(C(=O)OC(C)(C)C)OC)C)C1 53167,C1(CCC(=O)NC(C(C)NC(CCCCCC)=O)CO)CCc2cnn(C)c2C1 53168,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC2CC2)C(C)C1)=O 53169,c1(C(=O)NCCCN(C(C2(n3nccn3)CC2)=O)CC)ccc[nH]1 53170,C(C(F)(F)C(=O)NC1CN(C(=O)C(c2cccc(Cl)c2)C2CC2)C1)NC 53171,CN=c1[nH]nc(CC(=O)NCC2(O)CCN(C(C3(F)CCCC3)=O)C2)s1 53172,C1(CC(=O)N(CCN(C(=O)OC)C)C(C)C)CC(C)CCN1C(=O)C(C)NC=O 53173,N1(C(c2c(C)n(C3CC3)cc2)=O)CCN(C(=O)CSCCN(C)C)CCC1C 53174,c1(CN2C(C(=O)NCC=CCN3CCCCC3)CSCC2)c(Cl)ccc(F)c1F 53175,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1N(C(Cc2cccc(SCC)c2)=O)CCC1 53176,N1(C(C(C)OCOC)=O)CC2(CCCC2)C1C(=O)NC1CCCCCC1OC 53177,N1(C(c2ccc(C(F)(F)F)nn2)=O)CC2(CCC(NC(C3(Br)CCC3)=O)C2)C1 53178,C(c1ccc(N)c(N)c1)=CC(=O)NC1(CNC(c2cccc(CC)n2)=O)CC1 53179,n1(CC)nc(C(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)cc1C 53180,c1(C(=O)NCC(C)(C2CCC2)NC(c2ccc(OC)s2)=O)nn(C)c(C)c1Cl 53181,N1(C(C#CC(=O)O)=O)CCC2CN(C(=O)Cc3ccc(C(F)(F)F)nc3)CCC12 53182,c1(C(=O)NC(CC)(C)CNC(=O)C(O)CC2CC2)cc2c(cn1)NC(=O)CO2 53183,N1(C(C(C)C)=O)CC(C(C)(C)O)(N(C(=O)COC(C)(C)C)Cc2cnn(C)c2)C1 53184,c1(C(N(C(C)CCNC(=O)CC2CN(C)C2)C)=O)n[nH]c2ccccc12 53185,C1(O)(C(=O)NCCOC(CNC(C=CC=CC)=O)(C)C)CCCC(C)CC1 53186,C1(O)(CN(C(CCC=C)=O)C)CCCN(C(C2(F)CC=CCC2)=O)C1 53187,N1(C(CS(CC)(=O)=O)=O)C(C)CC2CN(C(=O)Cn3nccc3C)CC12 53188,CC#CCC(C(=O)N1CCC(C2(C)N=N2)C1)NC(=O)Cc1csc(C)c1 53189,C1(C(N(C2CCN(C(=O)C(C)N3CC(C)C3)CC2)CC)=O)CCC(F)CC1 53190,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53191,N1(C(c2c(CC)ccs2)=O)CC2CCC(CNC(c3cncnc3CC)=O)(C2)C1 53192,N1(C(c2cc(C)cc(N)c2)=O)CCN(C(=O)C=C2CCC2)C2CCCCC2C1 53193,N1(C(C(C)N2CCCC2)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53194,N1(C(c2c(=N)[nH][nH]c2)=O)CC2CCOCC2(NC(=O)C(=Cc2cccnc2)F)C1 53195,CC(C(=O)NOCc1cn(C(c2ccccc2)(C)C)nn1)n1cncn1 53196,C(=O)(C(C)(O)C=C)NCCOCCNC(C1(CC=C)CC1)=O 53197,Cc1ncc2c(n1)CCC(C(=O)NCC1CN(C(=O)C#CC3(C)COC3)C1)C2 53198,N1(C(c2cc(C3CCOCC3)[nH]n2)=O)CC2OCCN(C(C3CCOC3)=O)C2C1 53199,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53200,C(=O)(CC(C)(O)CCC)NC1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1 53201,c1(C(=O)NCC(CC)(C)NC(C2(COC)CCOC2)=O)cccnc1C 53202,N1(C(CC=CC)=O)CCCCC(C2CN(C(c3cncn3C3CC3)=O)C2)C1 53203,N1(C(CCCC=C)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53204,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53205,c1(C(=O)Nc2cc(Cl)cc(Cl)n2)ccc2c(c1)CCN(c1ncc(Br)cn1)C2 53206,c1(CCN(C(C(c2ccoc2)N(C)C(C)N(C)C)=O)C)nc(O)c2c[nH]nc2n1 53207,c1(OCC(N2C(C)CC(NC(=O)CCc3ccon3)C2)=O)nc(O)nc(O)n1 53208,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53209,CCCCCCNC(=O)C(c1ccc(C)o1)N(C1CCCCC1)CC 53210,Cc1cc(C(=O)NC2CN(C(c3cc(Cl)cnc3Cl)=O)CC2C#N)cc(C)c1Br 53211,C(=O)(CCN(OC)C(=O)c1cccc(F)c1)NCC(C(CC)C)O 53212,c1(C(N(C2CN(C(C=C(CCC)C)=O)C2)C)=O)ccc(C(C)C)c(Cl)c1 53213,c1(CC)c(OC)ccc(S(=O)(=O)N2CCNC3COCCC23)c1OC 53214,c1(NC(CCNC(C(C)CSC(F)(F)F)=O)(C)C)ncnc2ccc(Cl)cc12 53215,C#Cc1cnn(CC(=O)NC(Cn2cccn2)C(=O)NC2CC(C(=O)OC)C2)c1 53216,c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)ncc(Br)cc1N 53217,Cc1ccc(-c2cc(C(=O)NC(CNC(=O)C(C)NC(N)=O)CO)n[nH]2)s1 53218,CCCC(C#N)C(=O)NCCCCCNC(c1conc1-c1cccc(Cl)c1)=O 53219,c1(NC(=O)NCc2cc(Cl)ccc2I)cc2ccc1-2.Cc1cc(C(F)(F)F)ncn1 53220,c1(C(=O)NCCNC(C(C)(C)c2cncs2)=O)cncc(C2CCC2)c1 53221,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53222,c1(C(N(CC)CC2CCCCN2C(=O)CC(C)(C)O)=O)cc(Cl)cc(Cl)c1 53223,N1(C(c2n(CCC)ccc2)=O)CCC(C)(C)C(CNc2cc(O)nc(=O)n2C)C1 53224,C1(C(C(=O)NCC2CC2c2ccco2)F)CCN(C(=O)CC2CCOCC2)CC1 53225,C(CC(CC)C(=O)NC1CC(C)(NC(=O)C(CC)C(=O)OCC)C1)=CC 53226,c1(CNC(C(C)N(C(=O)CN2C(C)CCC2C)C)=O)ccc(F)c(O)c1 53227,C(=O)(CCCCCCC(=O)N1CCN(C(=O)C2=CCCCCC2)C2CCC12)OC 53228,Cc1cc(C(=O)N(CC(C)N(C)C(c2ncn(C(C)(C)C)n2)=O)C)cc(O)n1 53229,C1(=O)C(C(C)C)N1.C1(CCOC)CCN1C(=O)Cc1cnoc1 53230,N1(CC(=O)NCCCC(C)(C)OC(C(=O)OC)C2CCCC2)CC(=O)N1 53231,Cc1nc(=O)c2c(C)c(C(=O)OCCC(C)NC(=O)OC(C)(C)C)sc2[nH]1 53232,C1(CC)(CNC(c2cncnc2C)=O)CCN(C(C2CCCSC2C)=O)C1 53233,C(=O)(CC(C)CNC(c1ocnc1C(C)C)=O)N(CCC(=O)OCC)C 53234,Cc1oc(C#N)cc1C(N1CCCC(C(=O)NC2(CO)CCOCC2)C1)=O 53235,c1(-n2c(C)ncc2)ccc(C(=O)NC2(CNS(C)(=O)=O)CC2)cc1 53236,C(=O)(N=c1[nH]onc1C1CC1)C1CCCC(CNC(CCC(=O)N(C)C)=O)C1 53237,C(N=c1[nH]c(C)ncc1F)C1C(C)CCN(C(c2cc(SC)ncc2)=O)C1 53238,CC12CN(C(=O)CO)C(CNC(=O)Cc3cnns3)(C1)C2c1ccncc1 53239,c1(OC)cncc(C(N2CCCC2CCNC(C2(C)CC3CC3C2)=O)=O)c1 53240,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53241,CS(=O)(=O)c1cc(OC(F)F)ccc1NS(=O)(=O)C1CC1F 53242,N1(C(CC=CC=C)=O)CCN(c2ncncc2C)CC1C 53243,C1(C(=O)NCCNC(c2c[nH]nc2C(C)C)=O)(OC)CC1(C)C 53244,C(=O)(C1CCCc2scnc21)NC1CCC(CNC(c2coc(Br)c2)=O)C1 53245,C(=O)(CCS(N)(=O)=O)NC(C1CCN(C(c2cc(Cl)nnc2O)=O)C1)C 53246,C(=O)(CC(O)CNC(=O)NC(C)Cc1cc(Br)no1)NC 53247,C1(NC(C2(O)CCCC2)=O)CCC(CCNC(=O)C(C2CCOCC2)O)C1 53248,N1(C(C(C)(C)F)=O)CC(NC(c2cc3n(n2)CCC3)=O)C(C#N)C1 53249,c1(C(=O)NC2CN(C(C(C)(C)c3ccc(Cl)s3)=O)CC2F)ncc(F)cc1F 53250,C1(NC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(C)(C)c1ccn(C)n1 53251,N1(C(C2CC(C(C)C)C2)=O)CCCCC1CN(C)C(c1cncn1C1CC1)=O 53252,N1(C(c2nc(C)[nH]n2)=O)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)C2 53253,c1(NC(N2CC3C(CC(=O)Nc4ccc(Cl)cc4)(C3)C2)=O)ccccc1[N+](=O)[O-] 53254,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53255,c1(C2CC(C(N(CC(C)Cc3cccs3)C(=O)C3CC3)=O)C2)cccnc1 53256,C(=O)(C#CC1CCCCC1)NC(c1nc(C(N2CCC(C)C2C(N)=O)=O)co1)C 53257,N1(C(c2c(CC#N)ccs2)=O)CC(NC(C2CCCC2)=O)CC(F)(F)C1 53258,N1(C(c2n[nH]c(CC)c2C)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53259,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53260,C1(CC)CN(C(=O)C(C)(C)CSC)CCN1C(C1CCC(N(C)C)CC1)=O 53261,N1(C(COC)=O)CC2(C1)CN(C(c1cccnc1C(F)F)=O)CC2CO 53262,CC(C)CC(C)(CNC(=O)CCc1cnc(O)[nH]1)NC(c1cnn(C2CC2)c1)=O 53263,c1(C(N(C(C(=O)OC)C(C)C)C)=O)cnn2c(Br)cccc12 53264,C(=O)(C(C)C(O)CCCC)NCCC1CCN(C(C(CC=C)OC)=O)C(C)C1 53265,N1(c2n(Cc3cc(C)on3)c(-c3nc(Br)cs3)nn2)CC2C=CCOC2C1 53266,Cc1cc(N(C)C(=O)NCCN2CCCC(C)C2)ccc1N1CCOCC1 53267,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CCN(C(C2CCC2)=O)C(C2CC2)C1 53268,c1(CN(c2ccnc(CC3CCCO3)n2)C(C)C)cc(Cl)ccc1Cl 53269,Cn1cncc(C(=O)NC2COCCN(C(c3cnc(CC4CC4)s3)=O)C2)c1=O 53270,N1(C(c2c(C)n[nH]c2)=O)CC2CN(C(c3coc(C(C)(C)C)n3)=O)CCC12 53271,Cc1cc(C(=O)NCC2CC3CC3N2C(c2ccc[nH]2)=O)c(C)cc1Br 53272,CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2cc3ccc(O)nc3s2)=O)C(O)C1 53273,c1(OC)ccc2[nH]nc(C(=O)NCC(O)CNC(=O)C(C#N)C(C)C)c2c1 53274,c1(C(=O)NC2C(NC(c3cccc(C4C(C)C4)n3)=O)CCC2)cc(F)ccc1Cl 53275,N1(c2nccc(N3CCC(C)C3)n2)CCCC2(CC=CCO2)C1 53276,c1(C(=O)NCCN(C(=O)CCn2ccnn2)C)ccc2cc(F)c(F)cc2n1 53277,C1(CC(N2C(CNC(=O)COc3ccsn3)CC2)=O)CCCC2(CCC2)O1 53278,C1(NC(c2c(C)coc2)=O)CC(C)N(C(=O)C(C)O)C1 53279,c1(C(=O)NCCC(C(=O)N2CC(C#N)(CCF)C2)OC)ccc2nccn2c1 53280,c1(C(=O)NC2C(CC)N(C(=O)Cc3ncccc3C)CC2)cnn2c(C)cccc12 53281,c1(NC(=O)NC(c2nscn2)C)oc(C(N)=O)nc1-c1ccccc1 53282,c1(C(N2CCCC(C(C)NC(=O)Nc3cnc(Cl)nc3)C2)=O)ccc(I)cc1Cl 53283,C(=O)(CCCC(F)(F)CO)N1C(CNC(c2cc3n(n2)CCCCO3)=O)CCC1 53284,C(CCCCC(=O)N1CCCc2nccn21)NC(=O)C1CCCc2c[nH]nc21 53285,c12cccc(c1)N(C)C(=O)C2=O.c1(NC(C)=O)cccc(NC(C2CC2CN)=O)c1 53286,c1(C(=O)NC2CCN(C(c3c(OC)scc3)=O)C2C)ccn2ncc(C)c2n1 53287,C1(C2CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CN(C(=O)CC=C(Cl)Cl)CCO1 53288,C1(C(=O)NC(C)(CNC(c2cocn2)=O)C2CC2)CC1[N+](=O)[O-] 53289,CC1CC(C)CN(C(N2CCCC(C(=O)OC(C)(C)C)N2C(=O)C(C)COC)=O)C1 53290,C(=O)(C(F)(F)CC=C)N1CCC(C(CNC(CC2(CSC)CC2)=O)F)CC1 53291,N1(C(C2C(CC)C2)=O)CCCN(C(c2c(OC)cccc2C)=O)C(C)C1 53292,O(C1CCc2ccc(C(=O)O)cc21)C(c1cccc(C(C)(C)C)c1)=O 53293,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 53294,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53295,Cn1[nH]nnc1=NC1CC2CN(C(c3nnn(C(C)(C)C)n3)=O)CC12 53296,C1(NC(C2CN(C(C)C)C2)=O)CC2CCC1N(C(c1cnc3ncccn13)=O)C2 53297,C1(NC(=O)CC2CCC2)CC(NC(c2ccccc2-n2cccn2)=O)C12CCC2 53298,c1(CN(CCCOCC)CC)ccc([N+](=O)[O-])o1 53299,C1(NC(c2ccc(F)nc2)=O)CCOC(CNC(c2ccoc2C2CC2)=O)C1 53300,C(CCCC(C)(C)C(=O)NNC(=O)C(C)(C)S(=O)(=O)c1ccccc1)NC(C)=O 53301,CCC(CC(=O)NCC1COCCN1C(C1CCOC(=O)CC1)=O)C(C)(C)C 53302,N1(C(C2C(C)N(C)CC2)=O)CCCC(C)(NC(=O)CCc2ccc(Cl)nc2)C1 53303,Nc1c(-c2ccc(-c3nccn3CC(O)CO)cc2)cnn1CC1(O)CCC1 53304,C(C(O)C(=O)N(C)CC1CCCN1C(c1cc(C(C)(C)C)on1)=O)SC 53305,N1(C(CC2(OC)CC2)=O)CCC(C2CC2C(=O)NC2(CC(F)(F)F)CC2)CC1 53306,N1(C(Cc2c(CC)cccc2)=O)CC(C)CN(C(=O)CC(F)(F)F)C(C)C1 53307,C1(c2cn(C3(CC)CC3)nc2)CN(C(c2cccnc2)C)CC1C 53308,c1(NC(C(CCC)C)=O)cc(S(=O)(=O)NC(C)C)ccn1 53309,c1(C(=O)O)cc(Cc2cn(C3CN(NC(C4(C5CC5)CCC4)=O)C3)nn2)ccn1 53310,C1(CNC(C2(C(=O)NC)C(C)(C)C2)=O)CCCS1(=O)=O.C(CC(=O)O)COCCOCC 53311,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(C(=O)NC)CC2)CC(C)C1 53312,C1(C(C(=O)N(CC)CC2CC2)F)CCCN(C(C)C(=O)Nc2ccc(F)cc2)C1 53313,C1(C(N(C)CCNC(=O)Cc2cscc2Br)=O)CCN(CC(F)(F)F)C1=O 53314,C1(C)(COC)CC(NC(=O)Cc2ccnn2C)CN1C(=O)CCc1nncn1C 53315,C(C(CCCC)SC)Nc1cc(NC(CC(C=C)O)=O)ncn1 53316,S(=O)(=O)(CC(=O)NC1(C)CN(C(=O)C(C)(C)N2CCCC2)C1)NC 53317,c1(CNC(C(C)c2ccsn2)=O)cnn2c1CN(CCC1(N(C)C)CCC1)CC2 53318,N1(C(c2ccc(COC)nc2)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53319,CCCCC(C(=O)NCC1(CN(C)C(C2(CC(F)F)CC2)=O)CC1)N(C)C 53320,Cc1cc(C(=O)NC(C)CCNC(C2C3CCCOC23)=O)cn1C(C)C 53321,C(=O)(C(F)C(=O)NC(CO)C(=O)C(C1C(CO)C1(C)C)=O)OCC 53322,c1(C(N2C(C)CCC(NC(C(CO)OC)=O)C2)=O)sc2cc(F)ccc2c1C 53323,c1(N2CCN(C(C3CCn4cc(nn4)CC3)=O)CC2)nc2ccccc2[nH]1 53324,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CNC(c3ccccc3F)=O)CCCCC12 53325,Cc1ccc2ccnc(N3CC(c4nc(N(C)C)no4)C3)c2c1 53326,CON=Cc1ccc(C(=O)N(C(C)CCNC(c2cncc(Cl)c2)=O)C)cc1 53327,c1(CC(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)ccc2c[nH]nc2c1 53328,N1(C(=O)C=CCN2CCCCC2)CCC(c2ccccc2)C1CO 53329,C(=O)(C(O)C1=CCCCC1)N1CC=C(CNC(CC(CCCCC)O)=O)CC1 53330,C1(C(N2CCC(NC(CCC(=O)NC)=O)C2)=O)CCC(=O)C(C)C1(C)C 53331,c1(C(N(CC(C)N(C(C(C)n2ccnc2)=O)C)C)=O)cc(S(N)(=O)=O)sc1Cl 53332,C12(CNC(C(C)=CC3CC3)=O)CCCC(CN1C(=O)C(O)C(F)(F)F)C2 53333,C1(CC)CCCCCN1C(=O)CC1CCCCN1C(c1cncc(C(C)=O)c1)=O 53334,N1(C(C(CC)OC2CCCCC2)=O)CCCC2(CCCN2C(C)=O)C1 53335,C1(NC(c2ccc(F)cc2O)=O)C2COCC1CC(NC(C1CCCCS1)=O)C2 53336,c1(CNC2C(c3nnnn3CCCF)(OCCOC)CC2)cccc(C)c1C 53337,C1(CCC)(NC(C2COCCO2)=O)CCN(C(C2CN(C(C)C)CCO2)=O)CC1 53338,N1(C(C(CC2CCCC2)OC)=O)C2CCC1CC(CNC(C1(CO)CCC1)=O)C2 53339,C1(CCNC(CSc2cn(C)nc2)=O)CCCN(C(=O)CCOC2CCC2)C1 53340,N(C(=NCCC1CCCO1)NCc1ncccc1N1CCCC1)Cc1ccc(Br)o1 53341,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2C(C)O)=O)CC1 53342,CC1(CCCC(=O)NCC2(O)CCN(C(=O)Cc3ccco3)C2)NC(=O)NC1=O 53343,c1(C(C(=O)NC(CNC(c2c[nH]c(=NC)s2)=O)C)C)cccc([N+](=O)[O-])c1 53344,C12(C(N3CC(NC(CCc4ccc(C(C)(C)C)cc4)=O)C3)=O)CC(C)(C1)OC2(C)C 53345,C1(NC(c2c(CCC)nco2)=O)CC2(C1)CC2C(=O)NC1(C(F)(F)F)CC1 53346,C1(NC(c2nnc(C)s2)=O)CCC12CN(C(C1CCN1C1CCCC1)=O)C2 53347,C(=O)(C(F)CC(CC)CC)N1CCCC(C(=O)NC(CCC)(C)CO)CC1 53348,N1(C(Cc2ccc(OC)cc2)=O)CC2CC(C)N(C(=O)C(C3CC3)SC)C2C1 53349,N1(C(C(=O)N(C(C(=O)OCC)C)CC)c2cnsc2)CCN(c2ccccc2)CC1 53350,c1(CCC)cc(C(=O)NCCNC(=O)C(C)NC(=O)OC)no1 53351,C1(CC(=O)OC)CCCCN1C(=O)CC=CCNC(=O)C(C)N1CCCC1 53352,c1(C(C(N2CC3C(C(=O)OC)(C3)C2)=O)NCC2CCCO2)ccc(OC)c(F)c1 53353,CC1c2ccccc2CC1NC(C1(CNC(c2cccc(Cl)c2N)=O)CCC1)=O 53354,Cc1cc(C)c(OCC(N2CCC2CNC(=O)C(F)(F)C(C)O)=O)c(C)c1 53355,Cc1nncc(C(=O)NC(C2CCCCN2C(=O)CSc2cn[nH]c2)C)c1C 53356,N1(C(C(C)(C)CF)=O)CC(CNC(C2CC3CCC2CC3)=O)C2(CC2)C1 53357,c1(C(=O)NC2C3(CN(C(Cc4cncc(C)c4)=O)C3)CC2)cc2nccnc2[nH]1 53358,CCC(CC(=O)NCc1cc[nH]c1C(=O)NC12CCN(CC1)C2)C1CC1 53359,C(=O)(C(C)CC(C)(C)C)NCCn1cc(C(=O)N(CC2=CCCC(C)C2)CC)nn1 53360,N1(C(c2cc3n(c2)CCSC3)=O)CCC2CN(C(=O)C3=CCOC3)CC2C1 53361,c1(C(=O)N(CCn2cc(C3(C4CC4)CC3)nn2)C2CC2)cn2cc(F)ccc2n1 53362,C(C)(C(=O)N1CC(O)(CC(=O)NCC2(SC)CC2)C1)(OC)SC 53363,C(CC(C(C)(C)C)NC(=O)Cc1nc([N+](=O)[O-])n[nH]1)N(C)C(C1CCSC1)=O 53364,CC1(C)CC=CCN(C(C2(NC(C3CC3(C)C(F)F)=O)CCOCC2)=O)C1 53365,C12(C(=O)OC)CCC(C(=O)N(C3CN(C(=O)Cc4sccc4C)C3)C)(C1)C2 53366,C(N=c1ccnc(N2CC(CO)OC(C3CCC3)C2)[nH]1)c1ccc(C#N)cc1 53367,C1(CONC(=O)Oc2cnsc2)CCCCO1 53368,c1(C(C(=O)NCCCCCNC(=O)CSC(C)(C)C)N(C)C)ccccc1Cl 53369,N1(C(CCCOC)=O)CCC(N(C(=O)CN2CC3CC3C2)C)C2(CC2)C1 53370,c1(OC)cccc2cc(-c3ccc(OC(F)F)cc3C(=O)O)oc12 53371,C1(C2CC2)(CNC(CC2CCC(C)(C)CO2)=O)CCN(C(=O)C(Cl)=CCl)C1 53372,C(C1=NOC2CN(C(c3cnn[nH]3)=O)CC12)NC(c1ccc(C(C)(C)C)cn1)=O 53373,C(=O)(CC(C)C(C)C)NC(C(=O)NCCCC(=O)N1CC(CC)C1)CO 53374,CCC(C(=O)OC)C(=O)N1CC(c2ccccc2)(NC(C2CC(F)CN2C)=O)C1 53375,C1(C(=O)NCC(C)NC(=O)CCc2ccn(C)c2)CCC2(CC1)NC(=O)NC2=O 53376,CC1(C(=O)N(CCNC(C2CC2CCOCCO)=O)C2CC2)CC2(CC2)C1 53377,C1(NC(c2c(C)csc2)=O)CC(C2CCN(C(C3(O)CCCC3)=O)C2)C1 53378,c1(NC(CCO)C2CC2)nccc(N2CCOC(c3cccc(F)c3)C2)n1 53379,N1(C(c2ncn(C)n2)=O)CCCC2C1CCCN2C(c1csc(CO)n1)=O 53380,n1(CC)cccc1C(=O)N(CC(=O)N(C1(CC)CC1)C)C(C)C 53381,C1(CCC(=O)N(C(C)CN(C)C)C)CCCCN(C(=O)C=CC2CC2)C1 53382,c1(NC(=O)NCC2C(CC)CC2)ccc(OCC(C)OC)cc1 53383,C12COC3(C1)CN(C3)C2=O.c1(NC(C(N2CCC(C)C2)=O)=O)ccc(C#N)[nH]1 53384,C(=O)(C1=CC2C=CC1C2)NCC#CCNC(Cc1c(O)ccc(C)c1)=O 53385,C1(NC(=O)NC2CC(F)(F)C2O)CCc2nc(C(F)(F)F)[nH]c2C1 53386,N1(C(C2CC23CC(F)(F)C3)=O)CCOCC(CNC(=O)CC(=O)NC2CC2)C1 53387,C(CCF)(C(=O)NCCC1CC(C)C1)NC(C1CC(OCC)C1)=O 53388,C1(C(N2CC(O)(C(C)NC(c3cnc(C)s3)=O)C2)=O)CC(C2CC2)=NO1 53389,c1(CC)cc2c(CC(=O)NC3CC(CCNC(C4CCOCC4)=O)C3)csc2s1 53390,N1(C(C2(C#N)CC(=O)C2)=O)CCC(C2(NC(C3CC3C3CCCC3)=O)CC2)CC1 53391,C12CCCN(C1)C2.c1(CC(=O)NCCNC(c2cncs2)=O)cccc(F)c1 53392,c1(C(=O)NC2CC(c3ccccc3)(CF)C2)cc(Br)c(C(F)(F)F)cc1F 53393,c1(CC)ccc(C(=O)NC2CC2NC(C2(c3ccno3)CCOCC2)=O)cc1N 53394,CCCC(C)CC(=O)N(CCNC(C1CCCCC1(F)F)=O)CCOCCO 53395,N1(C(C2C3CC2N(C(C2CCO2)=O)C3)=O)CCC2(CCCO2)C1 53396,N1(Cc2n(CC)ncc2)CC2CC1CN2C(C1CC1C)=O 53397,C(CC(N)CC)N(C(c1nc(-c2ccccc2)cs1)=O)CC 53398,C1(NC=O)CCCN(C(=O)Cc2cscc2Br)CC1.C1CCCC12CC2 53399,C(CCC(=O)NC1CCC(CCNC(=O)C(C)(C)C2CCOC2)C1)OCC=C 53400,c1(CC)ccc(C(=O)NCCN(C(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53401,C1(CNC(c2cnc(C(N)=O)o2)=O)CCCN(C2CCCc3ccccc32)CC1 53402,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cnn(C)c2C2CC2)=O)C1 53403,C(=O)(CCC(=O)NCCCCCN(C)C(C1(F)CC1C(=O)OC)=O)NCCC 53404,CC1CCN(C(=O)C(N)=O)CCN1C1C2CCC1(c1ccccc1)C2 53405,C(C(=O)NNC(=O)CCOCCO)NC(c1n(CC)nnn1)C1CC1 53406,C1(N(C(CN(C(c2cnc(CC)o2)=O)C(C)C)=O)C)CCC(F)(F)C1 53407,N1(C(c2nccc(SC)n2)=O)CCN(C(C2CCC(C)=C(C)C2)=O)CC(C)(F)C1 53408,c1(C(=O)NC(CNC(C2C(=C)C2)=O)C(C)C)ccc(OC)c(S(=O)(=O)NC2CC2)c1 53409,CCC(CC)C(F)C(=O)N1CC(O)CC1Cn1cc(CC(O)C2CC2)nn1 53410,c1(CNC2CCC(C(=O)NCCCCO)C2)cnc2c(Br)cc(Cl)cn12 53411,c1(C(=O)NCC2COCCN(C(C3CCCS3(=O)=O)=O)C2)ccnc2c1CCO2 53412,C1(CC)(NC(=O)CN2CCCNC2=O)CCCN(C(=O)CC(C2CC2)C2CC2)C1 53413,C(=O)(C(C)C(C)COCC)N(CCCNC(C(COCC)C)=O)C 53414,c1(NC(=O)C(C)(C)C2CCOC2)ccccc1F.CCC1CNC(=O)CO1 53415,C(c1cnn(C)c1)=CC(=O)NC1(CO)CN(C(c2c(OC)csc2)=O)C1 53416,c1(OC)ccc(OC(C)C(N2CCCC2C2CCN(C(C3CC3C)=O)C2)=O)cc1 53417,C12CN(CCC1CO)Cc1cn(nn1)CC(=O)N2.C1(C(C)=O)CCCCC1 53418,O=C1COC(CNC(=O)NC2CCC(CSC)C2)CN1 53419,c1(C(=O)NC2CC3(C(NC(C(CC#C)C)=O)C3)C2)cc(C(C)C)ccc1F 53420,c1(OCCC)ccccc1.N1(Cc2nc(C(=O)OC)sc2)CCC(COC)(C)C1 53421,N1(C(c2ccn(COC)n2)=O)CC(CNC(=O)CCc2cc(OC)no2)C2CC12 53422,c1(-c2scc(C(=O)Nc3c(OC)ncnc3OC)n2)n[nH]c2ccc(C)cc12 53423,C(=O)(CCCCC1CC1C)NCCNC(CCCOCCC)=O 53424,C(c1ncco1)=CC(=O)NC(C1CCN(C(c2nccn2C)=O)C1)C 53425,CC(C)(C)C1=NOC(C(=O)NCCOCCNC(=O)C(F)CC2CCOC2)C1 53426,C1(CCC)CN(C(=O)CC2CC2c2ccccc2)CCN1C(=O)Cc1nc[nH]n1 53427,Cn1cc(C(C)(C)C(=O)N(CCO)CCc2ccccn2)cn1.N 53428,C1(CC(N)=O)(NC(c2c(C)cc(C)o2)=O)CCN(C(C2CC(=O)C2(C)C)=O)CC1 53429,C1(C(=O)NCC2=CCCCC2)C2CCN(C(c3ccsc3Cl)=O)CC12 53430,C1(CC=C)(NC(c2coc(CC)n2)=O)CCCN(C(C2CSCCS2)=O)C1 53431,c1(C(C)C)ccc(CC(=O)NC(CNC(=O)CCC(F)F)CC(F)(F)F)cc1F 53432,C1(C(=O)NCC(C2CC2)NC(C(CN(CC)CC)F)=O)CCC(C)CC1 53433,N1(C(c2cnn(CCCC)c2C)=O)CCC(C)C(N(C)C(c2csc(=N)[nH]2)=O)C1 53434,NS(=O)(=O)CCC(=O)NCCNC(C1CCCN(C(=O)CN2CCC(O)CC2)C1)=O 53435,c1(C(N2CCC(CNC(C3CC4CC4C3)=O)C23CC3)=O)cc2c([nH]1)CCCC2=O 53436,C=C=C(C)CC(=O)NC1C2CCN(C(=O)C(C(=O)OCC)C3CC3)C12 53437,C#Cc1ccccc1SC.C12CCN(CC1O)C(=O)C(C)C(=O)N2C1CCCC1 53438,c1(C(=O)NCc2c(C(N(CC(CC)OC)C)=O)cco2)cncnc1C 53439,N1(C(=O)OC)CC2CCC(C1)C2NCC(C)Cc1ccc(Br)cc1 53440,c1(C(=O)OCC)ccncc1C(=O)NCc1ccc(SC)cc1 53441,N1(C(Cn2c(C(C)C)nnn2)=O)CCN(C(C2CCSCC2)=O)CC(O)C1 53442,Cc1ccc(C(N)=O)cc1C(=O)NCCCC(C)NC(C1COCC1(C)C)=O 53443,N1(C(CN(C(=O)CCC(F)(F)F)CC)=O)CCCC(C)(N(C)C)C1 53444,C1(N(c2nccc(OC)n2)C(C(C)NC(C)=O)=O)CC2(CCNCC2)C1 53445,N1(C(CCn2nc(C)c(C)c2C)=O)CC2(CCCCN2C(=O)C(C#N)C(C)C)C1 53446,C(CC(C(N)=O)NC(C1(NC(C2CC2(F)Cl)=O)CCOCC1)=O)OC 53447,N1(C(C2=CC(C)(C)C2)=O)C2CCC1CN(C(C1CCc3nnnn3C1)=O)C2 53448,c1(-n2cc(-c3n(C)ncc3)nn2)ncccc1Cl.C1(N)CCCNC1=O 53449,c1(C(=O)NCCCCCN(C)C(C2C=CCC2)=O)cnn2c1OCC(O)C2 53450,CCCCCC(F)C(=O)NC(C)C(=O)NOCCO 53451,Cc1nsc2cc(C(N3CC(NC(=O)CCCCCC#N)C4CC34)=O)ccc12 53452,c1(C(N2CC3C(CNC(COCC(C)C)=O)C3C2)=O)nn(C)cc1S(C)(=O)=O 53453,C12(C(=O)NCC(CN(C(=O)CCc3ccccc3)C)(C)C)CCC(F)(CC1)C2 53454,Cc1cc(C(=O)NCC2CCCC2NC(c2ccn(C)c2C)=O)cc(=O)n1C 53455,c1(C(=O)NCCCCC2CN(C(C(COCC)C)=O)C2)cc(Cl)c2n[nH]cc2c1 53456,C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(C(C2CCCO2)NC(C)=O)=O)CC1 53457,C1(C2CC2)(NC(C(F)OC)=O)CCN(C(c2nc3ncccn3n2)=O)C1 53458,CN1CCN(C(=O)CC2CC2C2CC2)C(CNC(=O)CC2CCCCC2(C)C)C1 53459,c1(C(C)C)nnc(C=CC(=O)NC2CCCC2NC(=O)Cc2ccon2)o1 53460,C12(CNC(CCCOCC=C)=O)CC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 53461,C(N=c1nc2scnc2c(N2CCN(CCF)CC2)[nH]1)C1C(C)(C)COCC1 53462,CC1(C)CCC(CNC(C2CCC(=O)NC2)=O)N(c2nnco2)C1 53463,c1(C(N(CCNC(=O)Cn2ccnn2)CC)=O)ocnc1C1(C(=O)OC)CC1 53464,CS(=O)(=O)CCCC(=O)NCC1(C(=O)NCC2(O)CCCCC2)CCCCC1 53465,N1(C(C(c2ccc(CCC(C)N(C)C)cc2)(C)C)=O)CC2C3CCC(C(O)C3)C2C1 53466,C(CCC(C)C(=O)N(CCCNC(=O)Cn1cnc([N+](=O)[O-])n1)C)OC 53467,c1(CN(C)C)ccccc1NC(=O)CCc1csc(Br)c1 53468,c1(C(c2n(CCCSCC)nnn2)NC(c2nc[nH]n2)C)cc(C#N)n(C)c1 53469,C1(NC(CCN(CC)CC)=O)CC(NC(=O)CCC(C)N(C)C)C1(C)C 53470,c1(OC)cc(F)cc(C(N2CCC(CNC(=O)C(C)=C(C)C)C23CCC3)=O)c1N 53471,c1(C(N2CCC3(NC(=O)CC4CCOCC4)C(C2)C3)=O)c[nH]c2nccc-2c1 53472,c1(C(=O)NC2(CCCC(=O)NCCC=C=C)CCC2)ccc(C)c(F)c1 53473,C(=O)(C(C)(C)C(C)O)N(CCC(=O)NCC1CN2CCC1CC2)CC 53474,c1(CNC(CC2(OC)CN(C(C3(C)CC3C)=O)C2)=O)nc(C)sc1C 53475,CC(C(=O)NC1COCCC1NC(c1cn(C(F)F)cn1)=O)S(N)(=O)=O 53476,C1(CN(C(c2n(C(C)C)ncc2)=O)C)CN(C(=O)CC2CN(C)C2)CCO1 53477,C(=O)(C#CC1CCCO1)N(C)CC1(O)CCN(C(c2nn(CC)c(O)c2)=O)C1 53478,Cc1ccc(-c2csc(SC3(C(=O)NC(CN)CO)CC3)n2)cc1.CC(C)C 53479,C(=O)(C(C)CC(C)(C)C)N1CC(C(C)NC(=O)C(C)(C)c2cc[nH]n2)OCC1 53480,C=CCCCCCC(=O)N(C1CCCCN(C(=O)C(C)(C)OCC)C1)C 53481,N1(C(C2(C)CCCC2O)=O)CC2(CC(CNC(c3nc(Cl)cs3)=O)C2)C1 53482,C1(NC(CCC)=O)CC1C1CCCN(C(=O)C(c2ccccc2OC)C2CC2)C1 53483,N1(C(c2c(CC)cno2)=O)CCC(C)C(N(C(=O)Cc2cn[nH]c2)C)C1 53484,c1(C(=O)OCC)c[nH]c(=NC2CCC3CCC23)cn1 53485,C1(C(=O)NC(CSCC)C(=O)N2CC=CC2)CCCCC1F 53486,c1(C(=O)NCCC(C)N(C(CC(C)F)=O)C)cc(N)c(Cl)c(O)c1 53487,N1(C(c2c(C)nc(C)o2)=O)CCCC(C(N2CCC(CC(F)F)C2)=O)C1C 53488,C(=O)(CC1=CCN(C)CC1)NCCCC(CCC)NC(C1CCC(C)=C(C)C1)=O 53489,Cn1cnc2[nH]c(C(N3CCC(NC(=O)CN4CCSCC4)C3)=O)cc12 53490,c1(NC(C2N(Cc3ccc(C)nc3)CCSC2)=O)cccc([N+](=O)[O-])c1F 53491,NC(=O)CCN=c1ccn2ncc(S(=O)(=O)N3CCN(CC(F)(F)F)CC3)c2[nH]1 53492,c1(N2CCC(C(=O)OC)C2C)ncc2[nH]ncc2n1 53493,C1(CN(C(=O)C(O)C2CN(C(=O)CSCC(F)F)C2)C)CCCOC1 53494,C1(C=O)CCN(C(=O)OC(C)(C)C)C1C.C(C)(C)(C)OC(=O)NC(C)C 53495,c1(C(N(CCCNC(C2(CCCC)CC2)=O)CC)=O)ccc2c(c1)N(C)C(=O)C2 53496,N1(C(c2nonc2CC)=O)CCCCC1c1n[nH]cc1C(=O)NOCC(O)C(C)C 53497,Cn1cc(C(=O)NCCC2CCN(C(c3ncccc3N)=O)C2)c(C(C)(F)F)n1 53498,C1(CC(=O)NC2CN(CCO)CCO2)(NC(C2CCCCC2O)=O)CCCCC1 53499,c1(C(N2CCC(CC(C)NC(C3CC(F)C3)=O)CC2)=O)ccc(Cl)c(C#N)c1 53500,Cc1cccc(O)c1C(N1CC2(CCC2NC(=O)C=Cc2ccccc2)C1)=O 53501,Cc1nc2sc1C(=O)N1CCC(C1)C2.C1(CN(C)C(C2(O)CC2)=O)CC2CCC1C2 53502,C1(NC(c2ccccc2F)=O)CN(C(c2ccc(C3CCOC3)s2)=O)CC1F 53503,C1(NC(C(CC(C)C)O)=O)CC12CCC(NC(C1(N3CCOCC3)CC1)=O)CC2 53504,C(=O)(C1=CSCCO1)NC1C(NC(C(Cn2cccn2)OC)=O)C1 53505,c1(C(=O)NCC2C(C(N(C)Cc3ccn(C)n3)=O)C2(C)C)nccnc1N 53506,CC1CC(N(C(=O)C(F)C2CC(NC(c3c[nH][nH]c3=N)=O)C2)C)CCO1 53507,c1(C(=O)NC2CC(CNC(C(C)OC)=O)C(O)C2)ncc(Cl)cc1F 53508,C12(C(=O)NCC3CCCN(C(C(c4cn(C)nc4)O)=O)C3)CCCC1C2(F)F 53509,C(=O)(C1=NOC2(CCC2)C1)NC(C)CN(CC)CC.CCCC1(CC)C(=O)N1 53510,CC1CCC1CC(C(=O)CCS)=O.C1(CN)CC(OC(c2ccoc2)=O)C1 53511,C(=O)(CC(C(F)F)NC(C1CC1C(F)(F)F)=O)NC(C)(CO)C1CCC1 53512,c1(C(N2C3CC(NC(=O)COCCF)CC2CC3)=O)ccc(F)c2[nH]ccc12 53513,C1(C(=O)N(CCCC2CCC2)CCNC(=O)CCNC(C)=O)(OC)CCC(C)C1 53514,N1(C(=O)CCCc2cc(Cl)sc2Cl)CC2(CCN2C(=O)CCOC2CC2)C1 53515,c1(CC2C(C(=O)OCCCCN(C)C(c3ccccc3)=O)C2)ccccc1F 53516,c1(CCC)onc(C)c1C(=O)N(CCCNC(c1ccc(CC)s1)=O)C1CC1 53517,N1(C(c2c(OCC#C)nccc2)=O)CCCC(NC(=O)CCN2CCCC2)CC1 53518,N1(C(CCCN(C)C(C2CC3OC2C2CC32)=O)=O)CC(C2=NOCC2)C1 53519,C1(C(N(C2CCOCC2)C)=O)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 53520,C1(O)(CC)CCN(C(C2(CNC(c3sccc3OC)=O)CC(C)(C)C2)=O)C1 53521,C1(n2cc(COC)nn2)CCN(C(C23CCCC2CC3)=O)CC1 53522,C(CCNC=O)(Cn1cccn1)NC(=O)CCC1CCC1.C1(CN)CCCN1C1CC1 53523,CC(CC(C)(C)C)C(=O)N1CCC1CNC(c1ccncc1Br)=O 53524,Cc1ccnc(Cl)c1C(=O)NCC1CCN(C(=O)CC2CCCCC2(C)C)CC1 53525,N1(C(CC2C(C)C2)=O)CCC2(CC1)CCN(C(C1CC13CC(C)(C)C3)=O)CC2 53526,c1(C(=O)NCC(CNC(C2(CCC)CCC2)=O)=CC)cc(F)ccc1OC(C)C 53527,c1(C(N2CC3CC(NNc4cnc(CC)s4)C3C2)=O)ccn2nccc2n1 53528,C(CCOC)(C(=O)NC1CCC(C(N)=O)C1)NC(C(C)(C)OCC)=O 53529,C(=O)(C(CCC(C)C)NC(=O)C1=CCC(C)CC1)N1CCC(OC)C1C 53530,CC(C)C(CCN(C(=O)Cc1ccc(-c2nnco2)cc1)C)NC(=O)C(C)O 53531,C1(C(N(CCN(C(c2c(OC)ncc(Cl)c2)=O)C)C(C)C)=O)CCC(=O)CC1(C)C 53532,c1(C(C(=O)NCC2(COC)CCCO2)CO)ccc(F)cc1.N12CCCC1C2=O 53533,Cc1ccc(S(=O)(=O)N2CCCC2CCC(=O)NCC2(F)CCCNC2)cc1Cl 53534,C1(CNC(C(C)Cc2ccncc2)=O)CC2(CC2)CN1C(c1ccc(F)nc1F)=O 53535,CCC(CC)CC(=O)NC1CCN(C(c2ncsc2C(F)(F)F)=O)CC1F 53536,c1(C(=O)NC2CC3CN(C(CSC(C)(C)C)=O)C(C2)C3)cccc2nc(O)[nH]c12 53537,C(N=c1[nH]c2c(c(=NC3CCSC3)[nH]1)CCC2)c1c(N)c(F)ccc1 53538,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CCc2nc[nH]n2)CC1C(F)F 53539,C1(CN(C)CC)CCN(C(c2cnoc2C(C)C)=O)C1 53540,Cc1ccc(C(=O)Nc2csc(C(=O)Nc3nc(Cl)nc(Cl)n3)n2)c(C)c1Br 53541,Cc1ccc(CCNC(=O)C(C)CN(C(=O)C(n2ccnc2C)C)C)cc1 53542,c1(C(N(CC(CC)NC(=O)COC2CCCOC2)C)=O)ncc(C)cn1 53543,c1(-n2ccc(C(=O)NCC(CNC(C3CC(C#N)C3)=O)O)n2)cccc(Cl)c1 53544,N1(C(COC)=O)CCC(NC(c2ccc(C(O)CF)cc2)=O)C(F)C1 53545,c1(C(=O)NC(C)CNC(=O)C(C)CC2CC2)cn(C)[nH]c1=N 53546,c1(C(=O)NC(C)(C)CNC(c2ncccc2Cl)=O)cc2cncn2c(O)n1 53547,c1(C(N2C(C(C)NC(=O)C=CC(=O)N(C)C)CCC2)=O)ccc(S(N)(=O)=O)nc1 53548,CC1(C)OC2(Cc3ccccc3)CCC1(NC(c1ccc(F)c(O)c1)=O)CC2 53549,CC(O)C(C(=O)N1CCC(C)(NC(c2cnn(C3CCOC3)n2)=O)C1)N(C)C 53550,c1(NC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)cnc(C)c(Cl)c1 53551,c1(CC(=O)N(C2CN(C(C34CC(C)C3C4)=O)CC2O)C)cccnc1F 53552,C(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(=O)C#CC1CC1 53553,CS(=O)(=O)c1ccccc1C(N1CCCCC(NC(=O)C2=COCCC2)C1)=O 53554,C1(NC(CC(C(C)OC)NC(=O)Cn2ccccc2=O)=O)CC2(CNC(=O)O2)C1 53555,C1(CNC(c2cn(CCNC(C3CCN(C)C3)=O)nc2)=O)CC2C(C1)C2(F)F 53556,C1(N(CC(N2CCN(C(=O)C(O)C(C)C)CC2)=O)C(C)=O)C2CC3C(C2=O)C13 53557,CN1C(=O)OCC12CN(C(C1(CNC(=O)Cc3ccnc(O)c3)CC1)=O)C2 53558,CC(C)C(C)(O)CNC(=O)CC1(NC(C2CCOC2(C)C)=O)CC1 53559,N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2ccn(C)n2)C1 53560,N1(C(C(C)Cn2ccnc2)=O)CCCC(N2CC=CC2)C1.C(C)(C)(C)NC(=O)O 53561,c1(NC2CN(C(c3c(C)[nH]nc3Cl)=O)CC2C)cc(=O)n(C)cn1 53562,N1(C(=O)C(C)n2ccnn2)CCC2CCN(C(c3cc(C(CC)C)no3)=O)CC12 53563,c1(C(=O)N(C2CCN(c3ncc(Cl)c(O)n3)CC2)CC2CC2)coc2c1COC2 53564,C(=O)(CC(C(F)F)NC(=O)Cc1c(C)n[nH]c1C)NC1C(C)=C1 53565,N1(C(c2cccc(NCC)c2)=O)CCC(C2CC2)(CNC(C2CN(C)C2)=O)C1 53566,CC(C)CCC(=O)NCC(=O)NC1CC(CNC(c2ncn(C)n2)=O)C1 53567,C(=O)(CC(COC)NC(=O)C=CC(C)(C)C)NC1(CSC)CC1 53568,N1(C(=O)CNC(C2(n3nccn3)CC2)=O)CCC(C2CCCC2)C1 53569,C(=O)(C(C)CCN(C)C)NC(CNC(CC(=O)NCC#C)=O)C1CC1 53570,c1(CC)ccc(C(=O)NCC2(O)CC(CNC(=O)Cc3ncc(C)o3)C2)o1 53571,N1(C(c2cncc(C(C)C)c2)=O)CC(C)CCC1CNC(=O)Cc1cnnn1C 53572,C#CC1(C(N2CCC(CC(F)F)C2)=O)CCN(C(=O)C(C)c2ccsc2)CC1 53573,c1(COC)nc(C(=O)NC(C)C(CO)NC(=O)C=CC2CC2)n[nH]1 53574,C1(C(=O)NCC(F)(F)C(F)F)(CC)CCCN(C(c2ccccc2O)=O)C1 53575,N1(C(CC=C=C)=O)CCC(C(=O)NCCC2(C)CCCO2)C1(C)C 53576,CC(CSC(F)(F)F)C(=O)N(CCCCCNC(=O)CC1CNC(=O)C1)C 53577,Cc1c(-c2nnn(-c3ccccc3)n2)cccc1F.C1CC(C(C)C)NC(=O)C1 53578,c1(C(=O)NCC2C(C)CN(C(C3CCCCC3)=O)C2)c(F)ccc(F)c1O 53579,C1(CC)(CC)CC(O)CN1C(=O)C(C1CCN(C(c2cc(F)n(C)n2)=O)C1)F 53580,n1(CC)nnnc1C1C2CCN2Cc2cn(nn2)C2C(COC2)N1.C(C)(C)SC 53581,C1(CNC(C2(CC)CC2(F)F)=O)CN(C(=O)CCc2cccn2C)CCC1(C)C 53582,C1(N(C(C(CC#C)C2CC2)=O)C)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 53583,C1(NC(C(C)=CC)=O)CCN(C(=O)Cc2nonc2C)CC1O 53584,C1(CNC(c2cn(CC)nc2)=O)CC(NC(c2nccnc2N)=O)C(O)C1.C1(C)CC1 53585,C1(C)(NC(C2CCC(C)O2)=O)CCN(C(c2cnn(CCN(C)C)c2)=O)CC1 53586,Cc1nc2cccc(N(C)C)c2[nH]1.C1(c2ccccc2)C(N2CCOCC2)C(=O)N1 53587,CC1CCOC1C(=O)N(C)CCN(C)Cc1cn(C2CCOCC2)nn1 53588,N1(C(c2c(C)oc(Cl)n2)=O)CCCCCC1CNC(=O)CCS(C)(=O)=O 53589,N1(C(c2ccc(C(=O)NC)cc2)=O)CCCCC(CNC(=O)C(C)CSC)C1 53590,c1(CC)nccnc1C(=O)NC(C1(C(=O)N(CC(F)(F)Cl)C)CC1)C 53591,C(=O)(C1=CC2CCCCCC12)N1CCC(C(C)NC(c2ccc(C(C)=O)s2)=O)C1 53592,C(c1ccccc1Cl)=C(C(=O)N(C(CNC(C(CC)(C)OC)=O)C)C)C 53593,C=CCCC1C(=O)N1.C12(CCSC1)C(=O)NC(C)C(=O)N2.OC 53594,C1(N(CCC)C)CCN(C(=O)CCOCCNC(=O)NC(C)C)CC1 53595,Cc1nsc(C(N2CC(F)(C(=O)NCCSC(F)F)C2)=O)c1N 53596,Oc1c(-c2cn(CC3(OCCl)CCSC3)nn2)cc(F)cc1Br 53597,N1(C(C2(F)CCN(C(c3c(C(C)C)c[nH]c3)=O)C2)=O)CC(C)OC(C)(C)C1C 53598,C(=O)(CS(=O)(=O)CC(=O)N1CCCC1CNC(=O)C(=Cc1ccco1)C)OC 53599,c1(CN(CC(N2CCSCC2)=O)C)cc(N)cc(O)c1 53600,c1(C(=O)NCC2(CCNC(C3CC3C(N)=O)=O)CC2)cc2c(cn1)CCCC2 53601,C1(NC(C(=O)NCC)=O)CCC(F)(CNC(=O)CCN2C(=O)CCC2=O)C1 53602,N1(C(=O)CNC(C(C)OCCC#C)=O)CCN(C2CCCC2)CC1.C12CC1NC2=O 53603,Cc1c(NC(C2CCCCN2C(C)C)=O)ccc(Br)c1Cl 53604,C1(NC(CCCCC#C)=O)CCCC2CN(C(=O)CSc3ccc(F)c(F)c3)CC12 53605,n1(C(C(=O)NCCN(CCC)C(C2CSCCS2)=O)C)cnc2ccccc12 53606,Cc1cnn(CC(=O)NCCCCC2(NC(=O)C(C)Oc3cccnc3)CC2)c1 53607,CCC(CC(=O)NCCCOCCCNC(C1OCCC1C)=O)C(F)F 53608,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(C1(C(C)C)CNC(=O)C1)=O)C2 53609,N1(C(C2C(C)=C2)=O)CC2CCCC(C1)N2C(=O)CC(C)c1ccco1 53610,C1(C(=O)NCCC(C)(C)NC(Cc2ccn(C)c2)=O)CCNC(=O)C1 53611,C(=O)(C1=Cc2ccccc2C1)C(C(C)N(CC)CC1COCCC1O)=O 53612,C(=O)(C1=C(Cl)CCCC1)NCc1c(C(=O)NC2(CC#C)CC2)n(C)nn1 53613,N1(C(C(CN(CC)CC)F)=O)CCC2(NC(C3CCN(C)CC3)=O)CCCCC12 53614,C=C(C)C1OCCCC1C(=O)NC1CCN(C(C23CC4CC2C3C4)=O)CC1O 53615,N1(CC(=O)CCNC(=O)Cc2ccc(Br)cc2)CCC(C(F)(F)F)CC1 53616,c1(C(=O)NC2(C)CCN(C(c3ccnn3C3CCCC3)=O)C2)cc[nH]c(=N)c1N 53617,Cc1ccc(C2CC2CNCC2CCN(C(=O)OC3CCCOC3)CC2)c(C)c1 53618,N1(C(CCN2C(C)CCCC2)=O)CC2=C(C1)CN(C(C1CCS(=O)(=O)N1)=O)C2 53619,C12(C(=O)NCC(C(C)C)O)CCC(NC(=O)CC(C)O)(CC1)C2 53620,CC(C)CC(CNC(=O)CCC(=O)C1CC1)C(=O)N1CC(c2ccco2)C1 53621,C(=O)(CC(O)CCNC(=O)CC1CCCC1O)N(CCOC(C)=O)C 53622,Cn1nc(CNC(=O)CC2CCOCC2)c2c1CCN(C(c1sccc1Cl)=O)C2 53623,c1(CC)ccc(C(C)C(=O)N(C2CCCC2)CCNC(=O)CC(C)C2CC2)cc1 53624,C(=O)(C(CC(C)C)SC)NC1(C(=O)NCC)CCN(C(c2sccc2C)=O)C1 53625,C(=O)(C1=CCCCC1C)NC1C(NC(CCc2ncc(C)[nH]2)=O)CCCC1 53626,c1(C(N(CCCNC(=O)Cc2ccnn2C)CC)=O)cnc(Cl)c(F)c1N 53627,c1(C(C)OCC)nnc(N2CCCC2CC(C)(C)NC(=O)C=C(C)C)s1 53628,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(c1cnc(C2CC2)s1)=O 53629,C=CCN(OC)C(=O)CCC1CCCN(C(=O)CC2CC(F)(F)C2)C1 53630,C(C1=NOC2CN(C(c3ccnn3CC)=O)CC12)NC(c1cc(CC)ncn1)=O 53631,Cn1nc(C(F)F)c2cc(C(=O)NC3CC(NC(=O)CCSC(F)(F)F)C3)sc12 53632,c1(NC(C2CC(NCc3ccc(Br)[nH]3)C2)=O)cccc2c1CCO2 53633,C1(C(CNC(CCCC)=O)(C)O)CCCN(C(c2csc(Cl)n2)=O)C1 53634,C1(N(C)C)(C(=O)NC2CCCC(NC(=O)C=Cc3ncc[nH]3)C2)CCCCC1 53635,c1(CC)nc(C)n(C)c1C(N1CC(CCCCNC(C2(C)CCCC2O)=O)C1)=O 53636,Cc1nc(O)nc(O)c1CC(N1CCCC1CNC(=O)C(c1cnn(C)c1)C)=O 53637,C1(C(C)NC(c2cn(CC)nn2)=O)CN(C(=O)Cc2cnc(C(C)C)[nH]2)CCO1 53638,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 53639,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 53640,C12COC(C1)CNC2=O.N1(C(C)=O)CC(C(=O)NCCF)C1 53641,CCCCC(CC)CC(=O)NC(C)CCCNC(=O)C(C)(C)CC 53642,c1(C(N2CCC(N(C(CCCOCCOC)=O)CC3CC3)C2)=O)ccccc1Cl 53643,C1(C(N2C(CCN(C(c3cc(C)oc3C)=O)C)CCCC2)=O)CCCC2(CC2)C1 53644,C1(NC(=O)CC2CCCC2O)C2CCC(C2)C1C(=O)NC1CC(CO)C1 53645,C1(C(C)C)CC(C)CN(C(=O)C(=O)NCC(O)CC2CC2c2ccccc2OC)C1 53646,Cc1cc(Br)ncc1NC(=O)CCC1CCCN1Cc1cnn(C(C)C)c1 53647,N1(c2cc(C)ncn2)CCC(O)C(C(N2CCOC(C(F)(F)F)C2)=O)C1 53648,c1(OC)ncccc1C(=O)NC1CCCC1NC(=O)CC(C1CC1)NC(C)=O 53649,c1(C(=O)NCC2CC(OC)CN2C(c2csc(C3CC3)n2)=O)cc(C)ncc1C 53650,Cc1cc(F)ccc1C(=O)NC1CCCCCC1NC(C1(C)CC(C)(C)C1)=O 53651,C(C)(C)(CC(F)C(=O)N1CCCCC1CC(N)=O)NC(CCC(CC)=O)=O 53652,CC1(C)CC=C(C(=O)NCC(C)(C2CC2)NC(c2ccc(O)nn2)=O)CC1 53653,C1(C(N(CC)CC)=O)CCN(C(c2cc(OC)n(C)n2)=O)CC1C.c12cc(on1)C2 53654,C1(C(=O)NCC(CC)NC(=O)C(C)Cc2ccncc2)CC1C1CC1 53655,N1(C(C2(SC)CCC2)=O)CCCC2(CCN(C(=O)CC(O)C3CC3)CC2)C1 53656,C1(CNC(CSCCOC)=O)CCCCN1C.c1(C(=O)N)cn(C2CCC2)nn1 53657,C1(CNC(N2CC(CC)OC(C)C2)=O)CC2(CO1)CC1(C2)OCCO1 53658,C1(CC(=O)NC)CN(C(=O)CC2(CSC)CC2)CCN1C(=O)C(C)C(C)(F)F 53659,S(=O)(=O)(CC(=O)OC)N(C(C(C)NC(=O)CCCNC(=O)C(C)(C)C)C(C)C)CC 53660,C1(N(C(CNC(CCOC)=O)=O)C)CC2CC1N(C(C1C3COCC13)=O)C2 53661,CN1CC(C(=O)NCC(C)(C)NC(=O)CNC(N)=O)c2ccccc2C1=O 53662,C1(NC(c2n(C)nc(Cl)c2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 53663,N1(C(CSS(C)(=O)=O)=O)CCC2(CC2)CC1C(N1CCCC(CCCO)C1)=O 53664,C1(NC(c2c(F)ccnc2F)=O)CC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 53665,N1(c2nc(OC)nc(OC)n2)CC2CCCC(C1)C2C(N1CCCC(F)C1)=O 53666,C(=O)(C1=C(C)CCCC1(C)C)N(C1CC(NC(=O)C(c2cccc(N)c2)O)C1)C 53667,c1(CC(N2CCN(C(=O)Cc3nc[nH]n3)C(C3CCC3)C2)=O)ccc(F)cc1Cl 53668,Cc1nc(CO)oc1C(=O)NCC1(C)CCN(C(C2(CO)CCCO2)=O)C1 53669,C1(CCOC)CN(C(C2CC(C)(C)C2)=O)CCN1C(c1cc[nH]c1C1CC1)=O 53670,Cc1cc(C(N2CC(C)(C)OCC2CNC(=O)CC(C)C(F)F)=O)cc(N)c1O 53671,C1(NC(C(C)OCC=C)=O)C2CCC1N(C(c1nc(C)n(C)n1)=O)C2 53672,c1(NC(CC(C)NC(c2ccc(OC)c(C)c2)=O)C)ncnc2[nH]ccc12 53673,N1(c2ccnc(Nc3c(C#C)nccc3)n2)CCOCCc2ccc(F)cc21 53674,C(C(=O)NNC(=O)Nc1sc(-c2ccccc2)cc1Br)SC 53675,c1(C(=O)NCC2(C)CCN(C(C3C(C)OCC3)=O)C2)coc2ccc(F)cc12 53676,N1(C(C(CCCC)O)=O)CC2=C(C1)CN(C(c1cc(SC)ccn1)=O)C2 53677,C(C(C)CN=c1cc(C)nc(C2CC2)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 53678,c1(N(C(C=CC(C)N)=O)C)cccc(C(N)=O)c1 53679,C1(NC(CCN(C(c2cc(C)[nH]c2)=O)C(C)C)=O)CCC12CCCC2 53680,CC12COC(C(N3CCC(O)(C(C)CNC(c4ccns4)=O)C3)=O)(C1)C2 53681,c1(C(N2C(C)CN(C(=O)CS(=O)(=O)N(C)C)CC2)=O)ccc([N+](=O)[O-])cc1O 53682,c1(C(CNC(=O)Nc2n(CCC)ccc2)=O)cc(Br)ccc1I 53683,c1(C2CCN(C(=O)Cc3ccc(Cl)cc3)C2)nn(-c2ccccc2)c(=O)s1 53684,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3nnc(S)n3C)=O)(C1)OC2C 53685,N1(C(c2[nH]c(O)nc2C)=O)CC2(C(=O)NCCN(C)CC)CCC1CC2 53686,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(F)C2)ccc(C)c(C)c1O 53687,c1(OC)cc(O)c(C(=O)NCCNC(C2CC2c2cccs2)=O)cc1S(N)(=O)=O 53688,C1(CNC(c2cc(C)on2)=O)CC2COCC2N1C(C1CC(C)(C)CN1C)=O 53689,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1C1CCC1 53690,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 53691,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2cccn2C(C)C)=O)CC1(C)C 53692,C(C(N=[N+]=[N-])C(=O)N1CC(F)(CNC(=O)Cc2c(Cl)cccc2Cl)C1)OCC 53693,c1(C(=O)NCC(C2CCCCC2)NC(C(C)NC(C)C)=O)cccc(N(C)C)n1 53694,C1(NC(C(CC)NC(N)=O)=O)CN(C(c2[nH]c(=N)sc2CC)=O)CC1C 53695,N1(C(c2scc(C)c2)=O)CCOC(C(N2CCC(CN(C)C)C2)=O)C1 53696,C(CCCCCF)NC(=O)C=CC(=O)NOCCCCC1CC1 53697,Cc1cn2c(CC(N3CCCC(N(C)C(C4(C5CC5)CC4)=O)CC3)=O)csc2n1 53698,Cc1nn(CCO)cc1C(N1CCC(N(C(=O)C(O)Cc2ccccc2)C)C1)=O 53699,c1(CC)cc(C(=O)NC(CN(C)C)Cc2ccccc2Br)cc(Cl)c1 53700,N1(C(c2cc(C)cc(C)c2C)=O)CCOC2(CCN(C(C3CCN3C)=O)C2)C1 53701,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)ccc2ncsc2c1 53702,c1(C(N2CCCC(C)C2CCNC(=O)CC#N)=O)cc2cc(Cl)ccc2n1C 53703,c1(C(=O)NCC2(CC(N3C(C(=O)NC)C=CC3)=O)CC2)ccnnc1C 53704,S(=O)(=O)(c1c[nH]c(C(=O)NCC(C)(C(C)C)NC(C2CCCC2OC)=O)c1)NC 53705,C(=O)(CCCCN(C(=O)C(C)C1CCOC1)C)N(CCSC(C)C)CCO 53706,N1(C(C(CCC)C)=O)CCN(C(=O)CCc2ccc(C)o2)CC1C1CC1 53707,N1(C(C(CSC)C)=O)CCC(C)(NC(c2csc(CNc3ccccc3C)n2)=O)C1 53708,N1(C(c2cnc(C)nc2)=O)CCC(NC(=O)Cc2sc(O)nc2O)C(CO)C1 53709,C12(NC(c3ccc(C#C)cc3)=O)CCN(C(=O)CCC(=C)Br)CCC1C2 53710,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3ccccc23)=O)CC1(C)C 53711,CC(C(=O)NCCCCC(CO)NC(=O)CCC(C)(F)F)C(F)(F)C(F)F 53712,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 53713,C1(NC(COCCN(C)C)=O)C2CC(O)C1N(C(=O)Cc1cscn1)C2 53714,c1(C(N2CC(n3cc(-c4ccncc4)nn3)C2)=O)ccc2c(=O)[nH]ccc2n1 53715,c1(NC(C(N2CCC(C#C)C2)C)=O)cc(Br)c(O)c(Br)c1 53716,C1(NC(C(CC(C)C)(F)F)=O)CN(C(C2CC23CCCC3)=O)C2(CCCC2)C1 53717,C1(NC(CN(C(C)C)C)=O)CCC(O)CN(C(=O)C(C)(O)C(C)C)C1 53718,CCCC(CNC(=O)C(N)=O)NC(=O)C(C1(O)CCCC1)CC 53719,C(=O)(C(CNC(=O)CCN1CCC1)NC(=O)C1CC1)N1CC(CCC)C1 53720,N1(C(CSCC(=O)OC)=O)CC2(CCOCC2)CC1CN(C(=O)C(=O)NC1CC1)C 53721,c1(C(CC)NC(=O)C(c2ccsc2)N(C)Cc2n[nH]c(C)n2)ccccc1 53722,C(=O)(C1=CCCCO1)NC1(CCCNC(CN(c2ccccc2)C)=O)CC1 53723,CCCCC(CNC(=O)CN1CCCCC1=O)NC(=O)CCNC(=O)CO 53724,c1(C(C(=O)N(C2CCN(C(=O)C(C)C)C2)CCC)N(C)C)c(F)cccc1F 53725,N1(C(C2C=CCCC2)=O)CCC(O)C(NC(=O)CCc2ccc(Br)cc2)C1 53726,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 53727,c1(CNC(CC2N(C(CCC3C(C)C3)=O)CCC2)=O)ncc(F)cn1 53728,N1(C(c2c(CC)noc2)=O)CCN(C)C(C(=O)NCC2CCCCN2C)C1 53729,O=C1CC2CC(Nc3ccc(N4CCN(C(=O)C(F)(F)F)CC4)cc3)C1C2 53730,C(=O)(C(CCNC(=O)C(c1cccs1)NCCCOC)OC(C)(C)C)OC 53731,c1(C(=O)NC(CN(C(=O)CC2(O)CCCCC2)C)(C)C)cccc(C2CCC2)c1 53732,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 53733,c1(CNC(C2CC(F)(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)ccc(Cl)cc1Cl 53734,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)OCC(C)C)CC1)N1CCCC1=O 53735,N1(C(COC)=O)CCC2(C=C(C(=O)N(C3CC3)CC3CC3)C2)C1 53736,C1(C(=O)OC)CCC(CC(O)C(=O)OCC(C)OCC(F)(F)F)CC1 53737,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 53738,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 53739,N1(C(C(CCOC)(C)C)=O)CC2CCN(C(C3OCCOC34CCC4)=O)CC2C1 53740,C1(=O)CCCC(=O)O1.Cn1cncc1CCC(=O)NCC1CCCN1C(N)=O 53741,c1(CCOC)onc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(F)C(C)C)C1 53742,N1(C(C2CC(C)(F)C2)=O)CCC2(CC1)CC(NC(c1ccc(Br)c(Cl)c1)=O)C2 53743,c1(C(=O)OCCC2CCC(C)O2)ccc(F)c2[nH]ccc12 53744,N1(CCC)CC(NC(=O)C(C2CC2)N(C)C(c2cccc(C)c2)=O)CC1=O 53745,c1(-c2cn(CC(N3C(c4ccc(C)s4)CCC3)=O)nn2)cn2ccccc2n1 53746,C1(NC(COCCCCC)=O)CCN(C(=O)CC(O)C(C)C)CC1O 53747,C(c1cn(C)cn1)=CC(=O)NC(C1CCN(C(=O)C=Cc2ccnn2C)C1)C 53748,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCCc2ccc(O)cc2)=NO1 53749,CCCC(CC(=O)Nc1cc(C)cnc1OCC)NC(C1CN2CCC1C2)=O 53750,CCCCCCC(C(=O)NC1CCn2cc(C(=O)OC)nc2C1)N(C)CCF 53751,C1(CC(=O)NC2CC(C(C)NC(=O)CN3CCCC3C)C2)CC2C=CC1CC2 53752,c1(-c2scc(C(N(C(CNC(CC=CC=C)=O)C)CC)=O)n2)cccc(C)c1 53753,c1(CC)c(C(=O)NC2CN(C(=O)CCc3ccn(C)c3)CC23CC3)cccc1C 53754,C1(CNc2ncc(C(=O)OC)cn2)CCN(C(c2cncc(Cl)n2)=O)C(C)C1 53755,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 53756,c1(C(C)NC(=O)C(=O)NC2CC2OC(C)(C)C)ccc(F)cc1Br 53757,c1(C(=O)NCCNC(C(C)O)=O)ccn(CC(F)(F)F)c(=O)c1 53758,N1(C(CC(=O)OCCC(C)C)=O)CCCN(C(C2CCCCC23CC3)=O)C(C)C1 53759,c1(C(N2CCN(C(c3cncc(C)n3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cn1 53760,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 53761,N1(C(C(C(C)O)NC(=O)Cn2ncccc2=O)=O)CC(C)c2ncccc21 53762,N1(C(C2(C)CC(=O)NC2=O)=O)CC2(CCCC(CNC(=O)CC3CCC3)O2)C1 53763,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CCNC(c2cc(C(F)F)cs2)=O)CC1 53764,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 53765,C1(NC(CCN(CC=C)C(C2CC2Cl)=O)=O)C(O)CC1O 53766,c1(-n2c(COC(c3c(COC(C(C)C)=O)ccs3)=O)nnn2)ccccc1Br 53767,c1(NC(=O)CC2CC(C(=O)NCc3cn[nH]c3)C2)cnncc1Cl 53768,C(=O)(CCCCCCCCN=[N+]=[N-])NCC(=O)NC1CCN(S(C)(=O)=O)CC1 53769,c1(C(=O)NC2CC3C(NC(C4CC(C)OC4)=O)C3C2)ccc(O)cc1[N+](=O)[O-] 53770,CC1(NC(c2cc(Br)cc(Br)c2)=O)CCN(c2ncnc3[nH]ccc23)CC1 53771,C1(NC(COCC(=C)C)=O)CN(C(=O)C(C2CCOC2)NC(C)=O)CCC1(C)C 53772,C1(C(N(C2CC(NC(c3n(C(C)C)ccc3)=O)C2)C)=O)Cc2cc(F)ccc2O1 53773,C(C(=O)O)(C(C)(F)F)SCc1c(CNC)cccc1 53774,N1(C(c2nc(C)sc2)=O)CCN(C(C2C(C)C2C)=O)C2(CCC2)C1 53775,c1(NC(c2cc(CC)on2)=O)ccc(C(=O)OC)cc1[N+](=O)[O-] 53776,C1(C(C)NC(c2ccn(C)n2)=O)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 53777,c1(C(=O)NC(CNC(C(CCC)(C)O)=O)CCOC)cn2cc[nH]c(=O)c2n1 53778,C1(CCC)CC(OC)C(NC(c2nnnn2CCSC)c2ccccc2)C1 53779,N1(C(COCC)=O)CCN(C(=O)CCC(=O)NC23CC(OC)(C2)C3)CCC1C 53780,C#CCC(C(=O)NCCOC(c1cc(-c2ccccn2)on1)=O)OC 53781,c1(SC)cccc(F)c1C(=O)NCC1COCCN1C(=O)CN(C)C(N)=O 53782,C1(C(=O)NC2C(NC(c3cc(=N)[nH]cc3)=O)C2)CCC2(CC1)OCCO2 53783,N1(C(C2(CC)CCOC2)=O)CCN(CCNC(c2ccc(Cl)cc2)=O)CC1 53784,c1(-c2cc(C(N(C)CC3CC4(CCC4)C3)=O)on2)ccccc1C#N 53785,C(=O)(N1OC2CCC1CC2)N1C(C#C)(C(=O)CC2CC(C)(C)CO2)C=CC1 53786,Cc1cc(C(=O)NC(C)C(C)NC(C2CCCN2C=O)=O)ncc1C(F)F 53787,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnc[nH]1 53788,c1(C(CC)C)cc(C(N2CCC(CNC(c3cocn3)=O)C2)=O)on1 53789,C=CCC(C)(O)C(=O)NC1CCCC1C(=O)NOCC(=C)Cl 53790,c1(CCCC(=O)NCC2CC(NC(=O)C(F)n3ccnc3)C2)nc2ccccc2s1 53791,c1(N2CCOCC(CNC(Cc3cccc(OC)n3)=O)C2)cc2nncn2cn1 53792,C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCC12CCC2 53793,CC1(C)CCC(C(=O)NC(C2CCCN2C(=O)CCC2CCCOC2)(C)C)OC1 53794,Cn1nc(CCNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 53795,N1(C(=O)Cc2cccnc2O)CCS(=O)(=O)CC1.N12CC(CO)(C1)C(C)C2=O 53796,C(=O)(C1=CC(O)C(NC(=O)Cc2ccccc2C)C1)NC1(NC(=O)NC)CCC1 53797,C(C(C)C)(C(O)C(=O)NC(C(N1CC=CC1CN(C)C)=O)c1ccoc1)OC 53798,c1(C(c2nnnn2C2CC(F)(F)C2)NC(CC=C)CC)cn(C(C)C)nc1Br 53799,CCCCC(C(=O)NC1CCN(C(C2CC2C(F)F)=O)C1C(C)C)NC(N)=O 53800,C1(CC(=O)NCC2N(C(C(F)OC)=O)CCC2)CCCN(C(C)C)C1 53801,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 53802,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CC)O)=O)C1)CCO 53803,N1(C(=O)CCC2CCC2)C2CCC1CC(CNC(C1(N3CCOC3=O)CC1)=O)C2 53804,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(CCOC)(NC(C=CCC)=O)C1 53805,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 53806,N#CCCCC(=O)NCC(c1ccccc1Br)NC(C1CCCC1CF)=O 53807,c1(OC)c(Cl)ccc2[nH]c(C(N3CCCC(CNC(=O)C4=CCCS4)C3)=O)cc12 53808,C=CC1(CC(=O)N(CCC(C)NC(=O)Cc2c[nH]c(=N)[nH]2)C)CCCCC1 53809,CCC(CO)CN=c1cc(C)[nH]c(=NCc2ncc(Cl)cn2)[nH]1 53810,c1(C(N2CCCC(N(C(C(C=C)(C)C)=O)C)C2)=O)c(C)ccn1C 53811,C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)CCCc2nc(C)no2)CC1(F)F 53812,N1(C(CCc2ccc(C)s2)=O)CCC2(NC(=O)CC(C)(C)C3CC3)CCCCC12 53813,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)C(F)F)CC2)CC1C 53814,CC1CCCCN1C(c1c[nH]nc1CN(C(=O)C1=CCCC1)C1CC1)=O 53815,N1(C(C(F)=CC)=O)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CCC)C1 53816,c12cc(nc(Cl)n1)N2.Cc1ccc(C(N2CCOCC2)C)s1 53817,C(C(C)C(C)C(=O)N1CC(O)CCC1C(=O)NOCCCF)OC 53818,C(=O)(CC(C)CC(C)C)NCCC(C(=O)N(CCCOC)C)(C)C 53819,c1(COC)cc(NC(N2CC(NC(c3cccc(C)c3)=O)C2)=O)ccc1Cl 53820,N1(C(C(=O)NC(C)C)=O)CCC(C)(C)C(CNC(C2(C3CCCCO3)CC2)=O)C1 53821,N1(C(C2(C)CCCC2)=O)CC2(NC(=O)CCC3(C#N)CCC3)CC1C2 53822,C=CCC(C(=O)NCC1(CO)CN(C(c2cc(OC)cc(OC)c2)=O)C1)C(C)C 53823,C1(CN(C(C2CCC(N(C)C)CC2)=O)CC)CCN(C(C2CC(C)C2)=O)CC1 53824,c1(-c2n(C(C)C)nc(-c3cn(C4CCOC4)nn3)n2)n[nH]c2cccnc12 53825,c1(C(=O)OCC)nc(=NC(C)CNC(=O)Cc2cc(O)nc(O)n2)cc[nH]1 53826,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 53827,C1(CCC)CN(C(=O)Cn2cnc(C#N)n2)CC1C(=O)N(C12CC(C1)C2)C 53828,C1(C(=O)NCC(C)(C)CNC(C2COCCO2)=O)CC2(CCC2)CO1 53829,C1(C(=O)NCC2N(C(c3c(OC)ccc(C)n3)=O)CCC2)CCCC1S(C)(=O)=O 53830,CC1COCCN1C(=O)CCCN1CCC1c1cccc(Br)c1 53831,C1(NC(c2ccncc2F)=O)CCOC12CCN(C(c1ccccc1F)=O)CC2 53832,C12(C(=O)NC3CCC(NC(CN(S(CC)(=O)=O)C)=O)C3)C(=O)C3CC1C2C3 53833,C#CC1(C(N2CC(OC)CC(NC(c3cccc(F)c3C)=O)C2)=O)CCOCC1 53834,c1(C(N2CCC(O)C2)=O)nc2ccc(-c3ccc(B(O)O)cc3)cc2[nH]1 53835,c1(C(N2CCCN(C(CS(C)(=O)=O)=O)CC2)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1 53836,c1(C(c2nnnn2C2CCOC2)NCC(C)(C)COC)ccc2c[nH]nc2c1.CC=O 53837,N1(C(c2ccn(CC)n2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1CO 53838,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 53839,N1(C(CC(C)C)=O)CC2CCN(Cc3c(F)cccc3Br)CC2C1 53840,C(=O)(C(O)CCS(C)=O)NCCCCCNC(C(C)Cc1cccc(Cl)c1)=O 53841,c1(OC)ccc(C(=O)NCCOCCCN(C(=O)CC=C(C)C)C)c(F)c1 53842,CC1(C)CCCC(CNS(=O)(=O)CC2(CO)CCOC2)O1 53843,C1(ONC(=O)COCCCC2CC2)CN(C(=O)CC2CCSC2)CC1F 53844,c1(N2CCCCC(C)C2)ccc(S(=O)(=O)NCc2csc(Cl)n2)cn1 53845,c1(C(=O)NC2C(NC(C3N(C)CCC3)=O)CCC2)cnc2c(c1)CNC(=O)N2 53846,c1(C(=O)NCC(CCN(CC=C)C(C2CC23CCC3)=O)=C)scnc1C1CCCO1 53847,c1(C(C)C)ccc(C(=O)NCCC2CCC(NC(=O)CC3(C)CC3(Cl)Cl)C2)o1 53848,C1(CNC(c2cncc(F)c2)C)CC2CCC(C1)N2C(C1CCCCCO1)=O 53849,N1(C(C2(CC(C)C)COC2)=O)CC2CCCC(C1)N(C(c1c[nH]c(=N)o1)=O)C2 53850,c1(CC)cccc(C(=O)NCC(N2CCN(C(c3csc(C)n3)=O)CC2)=O)c1N 53851,O=C(CCC(F)(F)F)NCC(O)CC(=O)N1CC(CO)C1 53852,Cc1nonc1NC(=O)C(C1CC1)N(C(=O)COCC(C)C)C 53853,N1(C(c2cccc(CNC(CSC(C)C)=O)n2)=O)CCNC(=O)C1C 53854,C1(CC(=O)NC2(C(=O)NCCC3CC=CCC3)CSC2)COCC1O 53855,C(=O)(C1=C(Cl)CCCC1)NC(C)CNC(c1ccsc1C(F)(F)F)=O 53856,c1(C(=O)OCC(C)NC(C(C)Sc2ccc(C)cc2)=O)nc2cc(Cl)cnc2[nH]1 53857,C1(CNC(=O)CC2COCCO2)CCCN(C(=O)NCC2CCC2NC2CC2)C1 53858,c1(OC(C)(C)C)ccc(F)c(NC2CCN3CCCC23)c1 53859,C1(C(=O)Nc2cn(CCOC)nc2)CCCOC1C(C)C.n12cc(nn1)C2 53860,C1(C(N(C(CNC(c2ccc(C(C)=O)cc2)=O)C)C)=O)CC12CCS(=O)(=O)CC2 53861,c1(CC)cc(C(=O)N(CCC(=O)NCC=CC2CCC2)CCCO)n[nH]1 53862,C1(CNC(CCN(CCC)C)=O)CCCCC1NC(c1cccc(C(F)F)n1)=O 53863,C#CC1(C)CN(C(=O)C(CCSC)NC(=O)C(C(C)O)NC(N)=O)C1 53864,C1(C(N(C(C)C)CCNC(=O)CCc2ncco2)=O)CNC(=O)CC12CCOC2 53865,c1(C(=O)NCCSc2ccccc2C(F)(F)F)ccc(F)c(F)c1F 53866,Cc1cn2cc(C(N3CCC(F)C(NC(c4ccc(O)cc4F)=O)C3)=O)sc2n1 53867,CCC(C)(C(=O)NCC(CC)(CC)NC(C1CCN(C)C1)=O)C(N)=O 53868,N1(C(=O)OC)CSCC1NC(N1CCC(c2n[nH]cc2N)C1)=O 53869,CCC(C)C(C(=O)N1CC(N(C)C)C1)N(C)C.C12CC1C(=O)NCC2 53870,C1(N(C(c2nc(CC(C)C)sc2)=O)C)C2CN(C(c3coc(N(C)C)n3)=O)CC12 53871,CC1CN(C(=O)CC2(C(F)F)CC2)CC1NC(c1ccncc1N1CCCC1)=O 53872,C#CC(CC)(CC)NC(=O)C=CCNC(=O)CSCCNC(N)=O 53873,n1(CC(CC)O)cc(C(=O)NC2CCC(CCNC(c3cnc(C)s3)=O)C2)nn1 53874,C#Cc1ccnc(C(N2CC3(C2)CN(C(=O)C(F)(F)CC2CCCO2)C3)=O)c1 53875,S(=O)(=O)(c1ccc(C#N)cc1)N(CC(N1CC(C)N(Cc2cccs2)CC1)=O)C 53876,N1(C(c2cncc(OC)c2)=O)CCN(C(=O)C(c2ccncc2C)C)CC(O)C1 53877,c1(C(=O)NC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 53878,C1(NC(C2CCC(F)(F)C2)=O)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 53879,C1(CC)(CC)C(OCc2cccs2)CC1NCc1csc(C(C)(C)C)c1 53880,C1(F)(C(=O)NCC2(NC(CCc3c(OC)cccc3)=O)CC2)CCC(F)(F)CC1 53881,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC(C)C1 53882,C1(c2cn(CC)nn2)(C(=O)N(C2CCC(Cn3cccc3)CC2)C)CCCCO1 53883,N1(C(c2cc(C)c(O)cc2)=O)C(C(N2CCC([N+](=O)[O-])CC2)=O)C2CC(O)C1C2 53884,C(=O)(CC(CNC(c1c[nH]cc1C1CC1)=O)C1CCC1)NC(CN(C)C)CO 53885,c1(OCCCC(=O)OC)ccc(C(C)N(C)CCNC(C2CC2)=O)cc1Br 53886,C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O 53887,C1(CNC(c2ncc(C3CC3)cc2F)=O)CC12CCN(C(c1cocn1)=O)CC2 53888,C(=O)(C1CCCc2ncnn21)N1CCCC(N(C(=O)CCCN=[N+]=[N-])C)C1 53889,c1(CCC(=O)NCC2CCN2C(C2CCCCC2)=O)ccc(F)nc1 53890,c1(NC(CCn2cc(-c3cc(C)ncc3)nn2)=O)coc(S(C)(=O)=O)c1 53891,C1(C(N2CCC(C)(CNC(CC(CC)C)=O)C2)=O)CCCCN(C(C)=O)C1 53892,Cc1cc(-c2ccc(CN3CCC(CNC(=O)CN(C)OC)C3)cc2)cc(C)c1F 53893,CCC(C)CN=C(NC1CC1)N1CCC(c2cccc(Cl)c2OC)C1 53894,N1(C(C(F)=CCC)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(F)C1 53895,c1(S)ccccc1.C1(C(=O)NC(CCNC(CN(CC)CC)=O)C)C=CCCC1 53896,Cc1nn(CN(CCCSc2ccc(F)cc2)C(=O)C=C2CC2)cc1[N+](=O)[O-] 53897,C1(C(=O)O)CC(O)C(O)CC1C(=O)N(C1(C)CCC1)C(CC)C 53898,CCC(CC(C)C)C(=O)N1CC2(CCC2NC(c2cc(C(C)=O)c(C)o2)=O)C1 53899,C(C)(CN=c1[nH]c2c(c(=NCCCN=[N+]=[N-])[nH]1)CSC2)NC(=O)OC 53900,C(=O)(CCCCCO)NCCOC1(CNC(CC2CC(C)C2)=O)CCOCC1 53901,CCC(C)(C(=O)N1CCCC(NC(=O)CN2CC(C)C2)C1CC)C(N)=O 53902,C1(C(N2CCC(NC(c3ccnn3C3CCC3)=O)(CF)C2)=O)CN2CCC1CC2 53903,c1(OCCC)cc(N)ccc1-c1cccc(-c2nccn2CCC)c1 53904,N1(C(=O)C=Cc2cn[nH]c2)CCCC2(CCCCC2NC(=O)CC=CCO)C1 53905,c1(NC(C)=O)cc(Br)ccc1C(=O)NCc1csnc1C.C12CC(C1)C2 53906,c1(C(N2CC(N(C)C(c3cnnc(-c4ccccc4)c3)=O)C2)=O)cc(=O)cc[nH]1 53907,N1(C(C(CCOC)(C)C)=O)CC2(CC(NC(c3nc(C)sc3C)=O)CO2)C1 53908,C1(C(=O)NC(CNC(CCOC(C)C)=O)(C)C2CC2)CCOC(C(C)C)C1 53909,C1(C(=O)NC(CNC(C(CC(=O)OC)C)=O)C)Cc2cccnc2C1 53910,c1(NC(CNC(c2ccc(COC)s2)=O)C2CC2)nc(C)nc2sccc12 53911,N1(C(=O)Cn2ncnn2)CCC(NCC(N2CC3CC3C2)=O)C(O)C1 53912,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 53913,CC(C(=O)N(CCCNC(=O)CCc1ncc(F)cn1)CCO)C(C)(F)F 53914,c1(C(=O)NCCCn2cc(C(C)Sc3nncs3)nn2)cc2sccc2s1 53915,C1(C2CCC2)(C(=O)NC2C(NC(C3(C(F)F)CCCO3)=O)CCC2)CC1 53916,N1(C(C(C)SC)=O)CCCN(C(c2cc(C)n(CCO)n2)=O)C(C)C1 53917,CC(C)C(CCc1ccccc1)C(=O)N1CCC(CNC(c2ccc(Cl)o2)=O)C1 53918,C1(N(C(C2C(C)C2)=O)C)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 53919,O=C(C#CC1CCCC1)N1C(C(=O)NCCc2ncccc2F)CCC12CC2 53920,c12cn(nn1)C1CC2C1.N1(CC(=O)NCC(=O)N2CCC2)CC2CC2C1 53921,c1(C(=O)NC(C2CCCCC2)CNC(C(C=C)(C)O)=O)nccc(C)c1N 53922,C1(CC(=O)NCC2(CNC(C(C)(C)C3CCCCC3)=O)CCC2)CC(=O)NC1=O 53923,N1(C(C23N(C(C(C)N4CCCC4)=O)CCC2C3)=O)CCc2nnnn2CC1 53924,c1(C(N2C(C(C)(C)C)C(NC(C3CC3F)=O)CC2)=O)csc2ccncc12 53925,c1(C(C)C)ccc(OCC(N2CCN(C(=O)CCC#N)C3CC23)=O)cc1[N+](=O)[O-] 53926,c1(CC(=O)NCCCCCCNC(C(COC)O)=O)c[nH]c2ncccc12 53927,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(OC(F)(F)Cl)cc2)=O)C1(C)C 53928,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(O)o2)=O)C(C2CC2)C1 53929,c1(CN(C)C(c2ccoc2)=O)cccc(CNC(=O)CCc2ccn(C)c2)c1 53930,c1(C(C)C)cc(C(=O)NCC(C2CC2)NC(C2(CCF)CCC2)=O)n[nH]1 53931,CCCC(CC)CC(=O)NC1CCN(C(c2ccc(C)cc2)C)C1 53932,C=C1CC(C(=O)N(C2CC(C)C2)C)(CNC(c2cc(Cl)no2)=O)C1 53933,N1(C(C2C(NC(CCCCC#C)=O)CCOC2)=O)CC(O)CCC(C)(C)C1 53934,c1(NCC(CCC)OC)cc(C)c(S(=O)(=O)NC2CCCc3c2cnn3C)cn1 53935,C#Cc1cccc(C(N2Cc3ccnc(Cl)c3C2)C(=O)NCC2CC2)c1C 53936,C1(CNC(=O)CSc2ccccc2)OCC2CCN(C(=O)CC(F)F)CC12 53937,CC(F)(F)C(C)(C)CC(=O)NC(CNC(=O)Cc1ccno1)C(C)(C)C 53938,c1(C(=O)NCC(N2CCN(CC)CC2)(C)C)cc2cc(Cl)ccn2n1 53939,C#CCCC(O)C(=O)NC1COCCN(C(c2ncc(C)cc2C)=O)C1 53940,C(CCCCNC(c1c[nH]c(-c2ccoc2)n1)=O)N(C)C(c1nc(Cl)cs1)=O 53941,N1(C(CCC=C)=O)CC(NC(c2cccc3ncn(C)c23)=O)C(S(C)(=O)=O)C1 53942,C1(C(N(C2CCCCC2)C)=O)CC(O)CN1C(=O)CCc1csnn1 53943,C(C1CCCN1C(=O)CN1CCCCC1)=CC(N1CC(N(C)CC)C1)=O 53944,C(N=c1ccc([N+](=O)[O-])c(C(C)(C)C)[nH]1)C1CCN(C(C(C)CC(F)(F)F)=O)C1 53945,C(c1ccc(F)cc1Cl)=CC(N1CC(C(C)C)N(C(c2ccn(C)n2)=O)CC1)=O 53946,C1(CN(C)C(C2CC2c2ccco2)=O)CC1C1CC1 53947,c1(CNC(C(=O)OCC)Cc2ccccc2)cccc(C(C)(C)C)c1 53948,N1(C(C(C)O)=O)CC(C)(C)OC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 53949,c1(C(N2CC(CNC(=O)C(F)C3CCC3)OCC2)=O)cnc2c(c1)CCOC2 53950,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(CC3CC3)s2)=O)CCC1 53951,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 53952,c1(-c2cncc(C)n2)ccc2[nH]c(C(=O)Nc3cc(C(=O)N(C)C)ccn3)nc2c1 53953,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 53954,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 53955,c1(CC(=O)NCC(C)CNC(C2(CC(F)F)CCCC2)=O)ccc(Cl)c(F)c1 53956,c12ccc(F)c(c1)C(=O)NC1(CCCC1)C(=O)O2.C(C)(CSC)NC(=O)OCC 53957,CCC(CN(C)C)C(=O)NC1CCC(N(C)C(c2ccccc2OC)=O)CC1 53958,N1(C(C2C(c3n(C)cnc3)CC2)=O)CCN(C2COCC2NC(=O)CNC=O)CC1 53959,[N-]=[N+]=NCCCNC(C1(NC(C2N(C(CN3CCCC3)=O)CCC2)=O)CCC1)=O 53960,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1CO)OC 53961,CCCC(C)(O)CC(=O)N1CCCCC(NC(=O)Cc2nc(CC)cs2)C1 53962,N1(C(c2nnn(C)c2N)=O)CC2(CCN(C(C3CCCOC3)=O)C2)C1 53963,CCCCCC=CC(=O)N(CCNC(=O)CN1CC2CC2C1)CCOCCO 53964,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)C2CCCC2)nn1 53965,N1(C(CNC(=O)NC)=O)CCC2C(CCCN2C(=O)C2CCCn3nccc32)C1 53966,n1(CCCNC(=O)NC(c2cocn2)CC)cc(C)cn1 53967,c1(C(N2CC(O)(CNC(C3(COC)CC=CCC3)=O)C2)=O)ccc(O)c(F)c1F 53968,C1(NC(CSCC=C)=O)CCN(C(=O)CN2CCCCCC2=O)CC1F 53969,C1(N(C(=O)COCC2CCC2)CC#C)CCN(C(c2csnn2)=O)CC1 53970,C1(NC(CCCC=C)=O)CCN(C(C2CC3CC3C2)=O)C(c2ccccc2)C1 53971,c1(C(n2c(=O)nc(-c3cccc(CCN(C)C)c3)[nH]2)CO)c(F)cccc1Cl 53972,C(CCCC(=O)NCCC1CN(C(=O)C2=CCOC2)CC1C)N(C(C)C)C 53973,CC1CC2CC2CC1N(CCCNC(=O)CC1CCC(=O)NC1=O)C 53974,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 53975,C(=O)(CCC(=O)NC(C1CCN(C(c2cc(C(C)=O)on2)=O)C1)C)OCC 53976,C(CCCCCCNC(C1(C)CC(F)C1)=O)n1cc(CCOC(C)C(=O)O)nn1 53977,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 53978,c1(CC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cnoc2C)=O)C1 53979,C(CCC(=O)NNC(=S)NCCc1ccc(C)s1)OC 53980,C1(OC)CC1(C)CC(=O)NC1CC1CNC(=O)CN(C1CCCC1)C 53981,c1(N(C(CCC(C)SC)=O)C)ccc(S(=O)(=O)NC(C)CN(C)C)cn1 53982,C1(C(=O)NCC2CC(F)CN2C(=O)C=C2CCCC2)CCN(C2CC2)CC1 53983,N1(C(CSCCOC)=O)CCCCC(C2CN(C(c3cc(C(C)=O)cs3)=O)C2)C1 53984,Cc1n[nH]c2cc(C(=O)NC3CCCC3NC(c3ncccc3F)=O)ncc12 53985,c1(C(N2CC(C(C)Cc3cn(-c4ccc(Cl)nc4)nn3)C2)=O)c(Cl)cncc1Br 53986,CC1CCN(CCOCCC2(c3nn[nH]n3)CC3(CC3)C2)CC1 53987,c1(CC(CO)CN=c2[nH]c3c(s2)COC3)nc2c(c(=NCCC3CC3(Cl)Cl)[nH]1)CCC2 53988,Cc1cc(C(N2CCN(C(=O)CC3CCCCC3(C)C)CC2C)=O)ncc1C#N 53989,C1(C(=O)NC(CC(C)C)c2ccccc2)(CO)CCN(C(=O)OC(C)(C)C)CC1 53990,C1(OC)CN(C(=O)C(O)CNC(C2CC2C(N)=O)=O)CC12CC2 53991,C(=O)(C1NC(C)(C)Cc2ccccc21)Nc1cccc(CCCC(C)(C)C)c1 53992,N1(C(C(CCCNC(CC2CC(C)C2)=O)O)=O)CCc2c(F)cccc21 53993,N1(C(COC)=O)CCC2(CCC(C(=O)NCC3(N4CCOCC4)CCCC3)C2)C1 53994,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 53995,c1(C(N2C3CC(NC(C4C=C(C)CS4)=O)C(C3)C2)=O)cc(F)c(C)cc1Cl 53996,c1(OC)ncccc1CC(N1CC(NC(=O)CCc2nc(O)n[nH]2)C(C)C1)=O 53997,C#CC1(C(=O)OC)CCN(C(c2ccc(OCF)cn2)=O)C1 53998,C1(NC(c2ccc(C(N)=O)s2)=O)CC(NC(C2CCCC(CF)C2)=O)C12CCC2 53999,c1(-c2cn(C(C)CN(C(C(=O)N(C)C)C3CCCC3)C)nn2)c(F)cccc1Cl 54000,n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)n1 54001,c1(C(N2C3CC(CNC(C4C(OCC)C4)=O)C(C3)C2)=O)cn2cc(C)ccc2n1 54002,c1(C(N2C3CN(C(C(C)C(F)(F)F)=O)CC2C3)=O)cc2cc[nH]c(=O)c2s1 54003,CC1CN(C(=O)CCOC2CCC2)CC1CCNC(=O)CC#N 54004,C(C(C(=O)NC1C2CCCCCC12)C(C)(C)C)NC(CN(C1CCC1)C)=O 54005,N1(C(CCC2CNC(=O)N2)=O)CC2CCC(C1)N2C(C1CNC(=O)N1)=O 54006,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54007,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CC(C)O)CC3O)c(C)c2c1 54008,N1(C(CCc2n(C)nc(C)c2)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC(F)C1 54009,C1(C2CN(C(C(C3CC3)OC)=O)C2)CCCN(C(=O)Cn2ncnn2)C1 54010,CC(C)CC(C(=O)NC(CC(C)(C)C)C(=O)NCc1ccc(O)cc1F)C(C)C 54011,C1(C(=O)NCCCN(CC)CC)CC(=O)N(CC)C1.c12ccccc1NC2=O 54012,c1(CC)nc(C(C)NC(C2CC2NC(=O)C(COC)N(C)C)=O)n[nH]1 54013,C1(NC(C2CCN2C(=O)Cc2ccc(O)nc2)=O)CCc2ncnn2C1 54014,CN1CCN(C(C2(C(N)=O)CCC2)=O)CC1C(=O)NCCC(=O)NO 54015,C1(NC(=O)C2CC2)CC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 54016,C1(C(=O)NC(CC(C)NC(=O)OCC)C)CCN(C(=O)CCF)CC1.c1cccs1 54017,c1(C(=O)NCC2(NC(=O)C=Cc3cccc(O)c3)CC2)ccc2cncn2c1 54018,C1(O)(CNC(Cc2c(C)scc2)=O)CCCN(C(C2CCCCCC2(F)F)=O)CC1 54019,O=C(N1CC(O)CCO1)N.C1C2C=CC(C2)C1CO 54020,C(C1=CCCN(C)C1)NC(C(C)NC(C1CSC1)=O)=O 54021,C1(NC(c2nc(CC)oc2)=O)CCN(C(=O)Cc2csc(S)n2)CC12CCC2 54022,N1(C(COCCCCC)=O)CCN(C(C2CCCN2CC(C)C)=O)C(C2CC2)C1 54023,CC1CC(C)N(C(c2nnn3ccccc23)=O)CCN1C(c1c[nH]c(=N)o1)=O 54024,c1(NC2C(NC(C(Br)=C(C)C)=O)CS(=O)(=O)C2)ncnc2c([N+](=O)[O-])cccc12 54025,C1(c2nnnn2CCOC)(NCCOCCC)CCC(C2CC2)C1 54026,c1cccnc1.C(=O)(CN(CC(=O)NCC1(C(N)=O)CC1)C)OCC 54027,C(c1cn(C)nn1)=CC(N1CC(C(C)OC)C1)=O.CC1CC12C(=O)N2c1nccs1 54028,C=C(C)C1CCC(C)=CC1CC(=O)NC1(C)CN(C(c2ccc(Cl)cc2F)=O)C1 54029,C(=O)(C1=CC(c2ccc(F)cc2)=NS(=O)(=O)N1)N(CCN(CC(=O)NC)C)C 54030,C1(O)(CNC(c2scc(C)c2)=O)CCN(Cc2cccc(O)n2)CC1 54031,C=C=CCCC(=O)N(C1CCN(C(c2cc(OC)ns2)=O)C1)CCC 54032,N1(C(=O)NC(C)CCc2ccccc2)CCCC(C2N(CC(=O)NC)CC2(C)C)C1 54033,n1(CC(=O)OC)cc(C(=O)NCCC2CCN(C(=O)C(C)OC(C)(C)C)C2)nn1 54034,Cc1ccc2c(C(=O)NCC(C)CNC(=O)CCc3ccc(F)nc3)coc2c1 54035,c1(C(N2C(C(C)NC(C(C)SC)=O)CCC2)=O)ccc2c(c1)CCC2 54036,Cc1cc(-c2cn(CCCN(C(=O)C=Cc3cn(C)nn3)C)nn2)cnc1C 54037,C(=O)(C(C)(F)C(C)(C)F)N1CC(CC)C(NC(=O)Cc2cn3c(C)csc3n2)CC1 54038,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54039,c1(C(=O)NCC2CCCN2Cc2sccc2Br)cc2ccccc2o1 54040,C(=O)(C(CC1CCOC1)N(CCCCN(C)C)CCOC)NCC=C 54041,C(=O)(CCCCCF)NC1C(N2CCN(C(C3(CC#C)CCC3)=O)CC2)C1 54042,CC(C)CC(C(=O)N1CCOCC1CCO)ONC(c1c[nH]c(=N)o1)=O 54043,C1(C(=O)NCC(CC=C)(F)F)CN(C)CCN1C(c1csc(Cl)c1)=O 54044,N1(C(C2(C)CC2)=O)CCC2OCCN(C(c3ccn4cncc4n3)=O)C2C1 54045,CC1CC(C(N2CCCC2CNC(c2cccc(C3CC3)n2)=O)=O)CC(C)C1 54046,c1(C(=O)OC)c(C)cc(C)nc1NC(C)CC(C)NC(=O)CC(C)CC(C)C 54047,C1(N(C(C(C)SCC=C)=O)C)CN(C(c2ncc(COC)s2)=O)CCC1O 54048,C(c1cncc(F)c1)=C(C)C(=O)N1CC(N(C(=O)CC2CCS(=O)(=O)CC2)C)C1 54049,CC(C)C(C)(CNC(c1cnc(S)n1C)=O)NC(=O)C(c1ccc(Cl)s1)C 54050,c1(CCC(=O)NCC(C)(C2CCC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54051,c1(CNC(=O)CC(O)CC(COCCOCC)C)cnn(C)c1C#N 54052,C(CC(C)C)(C(=O)NC1CC1)ONC(COCC#C)=O 54053,C1(NC(CCOC)=O)CC2(CCN(C(c3cncc(-c4ccoc4)c3)=O)CC2)C1 54054,N1(C(CCN(C(=O)C(CO)OC)CC)=O)CCC(COC)C1C 54055,N1(CC(=O)NC2CC3CC(N)C3C2)CCCC2(CCCO2)CC1 54056,C(CN=C(NCC1CCCO1)NCc1nnnn1C(C)C)NC(=O)OCC 54057,C(C1=CCN(C(c2cncc(OC(F)F)c2)=O)CC1)NC(C(C)(C)NC(C)=O)=O 54058,C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(=O)CN2CCCC2CO)C(CO)C1 54059,C1(CC(=O)NCc2nc(C(C)(C)C)sc2)CC2CC2N1C(c1cnc(S)[nH]1)=O 54060,Cc1nn(C)cc1C1CC1C(=O)NCCCNC(C1CC2CCC1O2)=O 54061,c1(NC(C(c2c(C)n(C)nc2)=O)=O)nn(C)c2c1CCC2.C12CCC1CNC2=O 54062,C(C(C)C)(C(O)C(=O)NCC1CCOC1C(=O)N(C)Cc1ncco1)OC 54063,C1(C)(C(=O)NC(CC)COC(C)(C)C)CC(F)(F)C1 54064,C(CCC(C)C(=O)NC1(CCc2cn(CC(=O)NCO)nn2)CCC1)OC 54065,C1(C)(CCNC(C2N(C(C(C)n3ccnc3)=O)CC2)=O)CCCC1 54066,Cc1ncccc1C(=O)N(CCCN(C)C(C12CC(O)C1C2)=O)C 54067,N1(C(C(COC)O)=O)CC(NC(c2ccc(F)s2)=O)C2CCCCC12 54068,CC1=C(CNC(C2C3CN(C(c4ccno4)=O)CC23)=O)SCCO1 54069,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(C#N)C(Nc2cc(Cl)cc(Cl)c2F)C1 54070,c1(C(N2CCN(C(C(C3CCOCC3)OC)=O)CC2)=O)c(OC)nn(C)c1Br 54071,N1(C(C2C(=C)CC2)=O)CC23CCCC2(C1)CN(C(C1CCC(OCC)C1)=O)C3 54072,C1(OC(C)(C)C)CCN(S(=O)(=O)N2CCS(=N)(=O)CC2)CC1 54073,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54074,C1(C)(C(N(CCCCN(C(=O)C(c2ccccc2)O)C)C)=O)CC(C#N)C1 54075,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC)c(Cl)c1C 54076,C(=O)(CC(F)(F)Cc1ccccc1)Nc1c(OCC(=O)OC(C)C)nccc1 54077,C(=O)(C(C)(C)C(N)=O)NC1CCC(CCNC(c2c(OC(C)C)cncc2)=O)O1 54078,CCC(C)C(C)C(=O)NCCCCNC(c1cnn(-c2cccc(Cl)c2)c1N)=O 54079,N1(C(CSCC)=O)CCC2CN(C(c3ccc(OC)nc3C)=O)CCC2C1 54080,c1(C(=O)NCC2CCCN(C(C(COC)C)=O)C2)cccc(Cl)c1C 54081,c1(C(=O)NCCCN(C(C2CN(C(=O)NC)C2)=O)C2CC2)ccc(C)c(F)n1 54082,CCC(C)(C)CCCC(=O)N1CC(O)(CNC(=O)Cc2ccsc2C)C1 54083,C1(NC(CC2(OC)CCCC2)=O)CCC(C)(CNC(c2nc(C)nn2C)=O)C1 54084,c1(CNC(c2nnnn2C(C)CC)CCOCC)c(C)cc(Br)cc1C 54085,CCC(CNC(=O)CN1CCCS1(=O)=O)(CC)NC(=O)CC1C=CS(=O)(=O)C1 54086,CC(CNC(c1ccccc1O)=O)C(F)C(=O)NCc1c(F)cncc1F 54087,N1(C(C(C)=C2CCC2)=O)CC2CCC(CNC(c3n[nH]c4c3NCCC4)=O)(C2)C1 54088,CS(=O)(=O)CCC(=O)NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C12CC2 54089,n1(COC(=O)CC2CC3(C2)CC32CC2)ncc2[nH]cc(I)c2c1=O 54090,CCCCCC(F)C(=O)NCC(c1ccccc1)NC(C12CC(C)(C1)OC2C)=O 54091,CC1(C)CC(C(=O)NC2COCCC2NC(=O)CC2CC3CCC2C3)CO1 54092,C1(C(=O)NCC2(NC(=O)Cn3cc(Br)cn3)CC2)CCC(=O)N2CCCC12 54093,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54094,c1(C(c2ccsc2)C)nnc(N(C2COCC2(C)C)C)n1CC1CCCC1 54095,N1(C(C2(C)CCN(C(c3cc(C)oc3C)=O)C2)=O)CCCC2C(O)CC12 54096,Cc1[nH]c2ncccc2c1CNC1COCCC1C1CCNCC1 54097,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54098,C1(C(N2CCN(C(C(CC=C)CC)=O)C3C2C3)=O)CS(=O)(=O)CC(=O)N1 54099,c1(C(N2CC(CNC(CC(C)(F)F)=O)OCC2)=O)c(N)c(F)cc(F)c1F 54100,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54101,N1(C(c2ccc(C)nc2)=O)CC(N(C(=O)CCn2cncn2)C)C2(CC2)C1 54102,C1(C)(C(N(CC=C)CCC)=O)CN(C(C2CCC(COC)C2)=O)CC1C 54103,n1(CCC)nnnc1C(c1cnoc1)NCc1cc(C)[nH]n1 54104,CC(CN(C(=O)COCC1CCC1)C1CC1)C(=O)NC(CO)CCC1CC1 54105,C1(C(=O)O)C2CCC(C2)C1NCc1ccc(OC2CCOC2C2CC2)cc1 54106,CCC(CC)CC(=O)NC(C1CCCN1C(c1ccc([N+](=O)[O-])[nH]1)=O)(C)C 54107,CCCC(CC)C(=O)N1CC2CC2(NC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)C1 54108,C1(NC(CCSC)=O)CCN(C(c2ccc(CF)cc2)=O)CC1C 54109,C(=O)(C(C(C)(C)C)NC(N)=O)NCCC(C)N(C(c1ccc(CC)nc1)=O)C 54110,C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NC2C3CCOCC23)CCCC1 54111,C(=O)(C(C)C(=O)NC(C)C(=O)Nc1cncnc1O)OC 54112,C(=O)(C1CNC(=O)c2ccccc21)N1C(CNC(C2(C(C)C)COC2)=O)CCC1 54113,C(=O)(CCCCCS(N)(=O)=O)NCC1(O)CCN(C(c2cc(C)nc(C)n2)=O)C1 54114,C1(CNC(CN(c2nccs2)C)=O)CN(C(c2ccc(F)cn2)=O)C2CCN1C2 54115,c1(C(CNCCN(c2nccc(OCCOC)n2)C)O)cc(C)cc(O)c1 54116,CCCCC(C(=O)NC(C)CN(C)C(c1nc(C)n(C)c1C(F)(F)F)=O)C(C)C 54117,c1(C(N2CC3C(CNC(C(CC)(C)O)=O)(C3)C2)=O)cc2cscc2s1 54118,Cc1c(N)ccc(C(=O)NC(C)CN(C)C(C2CC3CCCCCC23)=O)c1C 54119,C(CCCCCF)NC(C1CC(c2cccs2)C1)=O 54120,c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN(C(C3CCC3C(F)F)=O)CC2)n1 54121,N1(c2nnc(COC)s2)CCC(C)C(C)C1.c12cnc(O)c(c1)NC2=O.OOC 54122,C1(NC(c2c(CNC(=O)CC3(O)CCC3)cc[nH]2)=O)CCCCCC1F 54123,C1(NC(C(C)SCC)=O)CC2CN(C(c3cncc(Br)c3C)=O)CC12 54124,C1(NC(C(C)=C2CCCC2)=O)CC(NC(c2nn(C)nc2Br)=O)C12CCC2 54125,C1(F)(C(=O)NCC2CN(C(C3C=CC=CC=C3)=O)CC2O)CC2(CCC2)C1 54126,CC1CCN(C2CN(C(=O)NC3CCCC(NC4CC4)C3)C2)CC1 54127,C(=O)(C(C)(C)C(=O)N1CCC(F)(C(=O)N(CC(C)OC)CC2CC2)CC1)OC 54128,Cc1cc(C(=O)NC2C3CN(C(C4CN(C)CC4C(F)(F)F)=O)CC23)c(Cl)cc1F 54129,CC1Cc2ccc(C(N3CC(NC(=O)Cc4cccc5nsnc45)C3)=O)cc2C1 54130,c1(C(=O)NCC2CCC(C(=O)Nc3ccc(C)cc3)C2)cc(C#N)cn1C 54131,C1(C(N2CC(C)=C(C)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1C2)=O 54132,N1(C(CNC(CC)=O)=O)CCC=CC1C(=O)NCC1CC(F)(F)CO1 54133,N1(C(C2CCC(N(C)C)C2)=O)CC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 54134,C1(NC(C(C)OCC)=O)(COC)CCN(C(c2c(C)nsc2NC)=O)C1 54135,c1(C(=O)NC(C=CC(=O)NCC(C)CN(C)C)C)cnc[nH]c1=N 54136,N1(C(C)=O)CCC12CCCN(C(c1cc(Cl)ccc1OCc1ccccn1)=O)C2 54137,C(=O)(C1C(F)C(=O)NC(=O)C(CC)COCC1)N1CC(=O)NCC1 54138,c1(CNC(c2c(NC(C(COC)(C)OC)=O)c[nH]n2)=O)cc(Cl)ccc1Cl 54139,CCC(C)C(O)COCCOC(c1csc(NC(=O)OC(C)(C)C)n1)=O 54140,CCCCC(CC)C(=O)N(CCNC(c1cnc(C(F)(F)F)cc1C)=O)CC 54141,c1(C(N(CCCNC(Cn2c(C)cc(C)n2)=O)C)=O)sc2[nH]cnc(=O)c2c1C 54142,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54143,C1(CC#C)(C(=O)NC(CNC(c2cc(OC)ccn2)=O)(CC)CC)CCCOC1 54144,c1(CC)onc(C)c1C(N1C(C(=O)NCCN2CC(C)(O)C2)CC2CC12)=O 54145,C1(CC(=O)NC(C)C(C)NC(c2ccccn2)=O)CCCCC12CC2 54146,Cc1[nH]nc2c1CC(C(N1CCCC(F)(CNC(=O)C(C)(C)C(F)F)C1)=O)CC2 54147,N1(C(CC2(CC)CCC2)=O)CC=C(C(=O)NC(C2CCOC2)(C)C)CC1 54148,c1(C(=O)NCC(O)CCNC(C2(C(=O)O)CC2)=O)cccc2[nH]ccc12 54149,c1(CC)cccc(S(=O)(=O)NC)c1.C12(C)CCC(CC1)C(=O)N2C 54150,N1(C(=O)Cc2cnc[nH]2)CC(C2CCN(C(=O)CC3CCCN(CO)C3)CC2)C1 54151,c1(OC)csc(C(N2CC(O)(CN(C)C(C3CSCN3C)=O)C2)=O)c1 54152,CC#CCCCC(=O)N1CCC(c2ccccc2)(NC(=O)C(C)NC(C)=O)CC1 54153,c1(C(=O)NCC(C(C)C)NC(c2ocnc2C2CC2)=O)ccc2nnn(C)c2n1 54154,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54155,CC1CCc2onc(C(=O)NC3CC4C3CCN4C(c3cn[nH]c3)=O)c2C1 54156,c1(NC(C2CCC(c3nn[nH]n3)CC2)=O)ccc2nc(C3CCCC3)[nH]c2c1 54157,c1(CC(=O)NCCC2CCN(C(CCCc3onc(C)n3)=O)C2)cccc(F)c1 54158,N1(C(C)=O)CCOC(C(=O)NC2CCC(N(C(=O)C=CBr)C)CC2)C1 54159,Cc1nn(C)c2c(N3CCC(CSC(F)(F)F)C3)nc(=NC3CCCOC3)[nH]c12 54160,c1(OC)cncc(C(=O)NC(C2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C)n1 54161,C(=O)(CC(C=C)CCC)NCC1CCCC(NC(CSCC#C)=O)C1 54162,C1(C(=O)Nc2c(C)ccnc2)CN(Cc2cccc(Cl)c2Br)CC(F)(F)C1 54163,c1(OCC(=O)N)ccccc1CN(C1CCN(C(CC)C)CC1)C.OC 54164,c1(C(N2CCCCC2CCO)C(=O)NCC=C)ccccc1Br 54165,N1(C(C(c2ccccn2)C)=O)CCCC(CO)(NC(C2CC3C=CC2O3)=O)C1 54166,c1(C(=O)NCC(CC(C)C)NC(=O)CC2CNC(=O)C2)ccnc(C(F)(F)F)c1N 54167,Cc1[nH]c(C)c(C(=O)NCC(C)(NC(=O)CCC(=O)Nc2nccs2)CF)c1C 54168,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54169,N1(C(C(C)N2CCCC2)=O)CCN(C(c2cn(C(C)(C)CCCO)nn2)C)CC1 54170,C1(NC(c2nc(C)sc2)=O)CCCN(C(=O)COC2CCCC(C)C2)C1C 54171,CCCC(CCC)CC(=O)NC1CC2CC1CC2C(=O)NC1CCN2CCC1C2 54172,N1(C(CCC(=O)OC)=O)CC(SC2CC2CNC(N2CCCC2=O)=O)CC(O)C1 54173,C1(C(=O)NCCN(C(C(CCCC)O)=O)CCC)Cc2nccnc2C1 54174,c1(N(CC(=C)Br)C2CC2)cc(C)c(S(=O)(=O)N2CCOC(c3ccnc(Cl)c3)C2)cn1 54175,C1(CC=C)(C(=O)N(C)CCOCCCNC(=O)C(C)CO)Cc2ccccc2C1 54176,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)Cc1cccc(Cl)c1 54177,N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(O)C1 54178,N1(CCC(N2CCC(CCNC(CC(CC)O)=O)C2)=O)CCSC(C)(C)C1 54179,Cc1cccc(CCC(=O)NCC=CCNC(C2CCCN(C)C2)=O)c1 54180,N1(C(C(c2cn(CC)nc2)=O)=O)CCC(NC(=O)C(N2CCCCC2)C)C(C)C1 54181,N1(C(C23CCOCC2C3)C)CC(C(=O)O)C2(CN(C(=O)OC(C)(C)C)C2)C1 54182,CC(C)C(CNC(C1CNC(=O)N1)=O)C(=O)NC1CCOCC1 54183,c12cccc(c1)NC(=O)NCC(CO)C2.C1(SC)CCC(c2ccccc2)CC1 54184,Cc1cc(C(=O)NCCOC2CCN(C(=O)CC(C)C)C2)c(C)n1CC1CC1 54185,n1(CCC(C)C)ncc2c1CC(NC1CCCC1C(=O)NC(C)C)CC2 54186,c12cc(nc(C(F)(F)F)n1)N2CC1CC(O)CN1C.CC(CN(C)C)N(C)C(C)C 54187,C1(NC(=O)CCCC2CC(NC(CC)=O)C2)COC(CC(C)C)C1 54188,N1(C(c2cc(Br)ncc2N)=O)CC(C)C(OC)C(C)C1 54189,c1(CC)cc(C)ccc1C(=O)NCC1(O)CN(C(=O)CNS(C)(=N)=O)C1 54190,c1(C=O)cccc(F)c1C(=O)O.N1(N2C(C)CCC2)CC(NC(=O)C2CC2)CC(F)C1 54191,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54192,C1(CC#C)(C(=O)NC(C2CC3(CCC3)C2)C)CCN(C(=O)Cc2cccs2)C1 54193,C(CCC)(C(=O)NCC1CC2(CCN2)C1)=CCC 54194,c1(CNC(c2c(SC)csc2)=O)nc(CNC(C2CN(C)C(=O)N2)=O)cc(O)n1 54195,C1(NC(C=C2CCN(C)C2)=O)CCC(N(C(=O)Cn2cnnc2)C)CC1 54196,c1(Nc2scc(-c3ccc(C)cc3)n2)cc(N2CC(F)C2)nc(C)n1 54197,N1(C(C2(C)CC=CC2)=O)CCC(c2cc(CNC(=O)CCF)on2)CC1 54198,c1(N2C(C)CN(CC34COCC3C4)CC2)ncnc2c1ncn2C 54199,C#CCC(C(=O)NCc1nn(C)cc1Cl)NC(=O)CCCCN(C)C 54200,Cc1nc2ccccn2c1C(=O)NCc1nc(CNC(C2(N=[N+]=[N-])CC2)=O)cs1 54201,c1(C(=O)Nc2ccc(NC(CN(CCC)C)=O)c(C)c2)c(C)[nH]c2ccccc12 54202,c1(C(=O)NC2(CC)CCN(C(=O)CC3CC3(Cl)Cl)CC2)cn2ccc(C)cc2n1 54203,N1(C(C2(C)CCC2)=O)CC(NC(C2CCCC2(C)C)=O)C2(CCCC2)C1 54204,c1(C(N2CCC(C(C)NC(c3cnccn3)=O)C2)=O)ccn2ccccc12 54205,C1(C(N2CC(CNC(Cc3nnc(C)s3)=O)C(O)C2)=O)CCC2C(C1)C2(F)F 54206,C12CCCN(C1)C2.c1(NC(=O)Cn2cc(-c3ccncc3Br)nn2)cncc(Cl)c1 54207,CCC(CC)CC(F)C(=O)NC1(C(N2CC3(CCC(=O)N3)C2)=O)CSC1 54208,C(C(C)CC(=O)NC1COCCC1NC(c1snc(Cl)c1Cl)=O)OC 54209,C1(C(=O)NCC2(COC)CN(C(C3CC=CC3)=O)C2)CNC(=O)CC1C 54210,N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(=O)CC(C)(C)O)CC2C1 54211,N1(C(CC(C=C)C)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCC1)C2 54212,c1(CCN2CCC(COCC)(CO)CC2)c[nH]c2cc(F)cc(F)c12 54213,C1(CC)(CNC(C2CN(C(=O)CCCC3CCCC3)CCO2)=O)CCOCC1 54214,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54215,CC1(C)CN(C(=O)NC2CC(n3cncn3)C2)Cc2ccccc21 54216,c1(OC)ccc(CC(C)C(=O)NC(CCC#N)(CO)CO)cc1.C1(=O)CC(=O)N1 54217,C1(C(=O)NCCN(C(C)C)CC)CC(C)CCN1C(c1cnc(C)c(C)c1)=O 54218,Cc1ccc(S(=O)(=O)NC(C)C(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54219,C1(CCOC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)C=Cc1ccc(C)o1 54220,C1(c2nnnn2CCC2CC2)(NCCCCCCOCC)CCC1C1CC1 54221,C12(C(=O)NC3C(C)CN(C(c4cnn[nH]4)=O)C3)CCC(C1)C2(C)C 54222,c1(OC)cc(C(N2CCC(C(=O)NCC3(C#N)CC3)C2C(=O)O)=O)ccn1 54223,C1(CC(=O)NC2CC(CNC(=O)Cc3ccsc3)C2)CCCCC1 54224,C1(CNC(c2cn[nH]c2)=O)COCCN(C(=O)COCCn2cccn2)C1 54225,C12(C(=O)NCC(CNC(=O)CCN(c3cnccn3)C)OC)CCCN(CC1)C2 54226,C1(NC(CCOC)=O)CC2C1CCN2C(c1ccc(C(=O)OC)c(Cl)c1)=O 54227,N1(Cc2ccsc2N(CCCC)C)CCCC(F)(F)CC1.OC 54228,CON=CC(=O)NCCCCCNC(c1nnsc1N)=O 54229,C1(C(N(CCCNC(=O)C(F)n2cccn2)CC)=O)CC1C1CC(F)(F)C1 54230,c12cc(C)cc(c1C)NC2=O.C1(CN(C(C2CC(C=C)C2)=O)O)C2CCC(F)(F)C12 54231,c1(CN2C3CN(C(C4CCC(F)(F)C4)=O)CC2CC3)cn2cccnc2n1 54232,C1(C(=O)NCCCC(C)NC(=O)C(c2ccc(N)cc2)C)(COC)CCCCC1 54233,N1(CC(=C)C)CCC(C(C)C(=O)NCc2cc(C3CCOC3)on2)CC1 54234,CC1(C)CC(=O)NC1CNC(=O)CN(C(c1ccncc1N)=O)C1CC1 54235,c1(C(N(CC(C)N(C(=O)C(C(C)(C)C)C2CCC2)C)C)=O)cc2cccn2cn1 54236,C(C(CO)CC(C)(C)C)NC(Cn1cc(-c2ccc(OC)cn2)nn1)=O 54237,Cc1nc(NCC(c2ccccc2)NC(C2(CO)C=CCC2)=O)cc2nncn12 54238,C1(CNC(=O)CCc2cccs2)CCCN(C(C2CCC(F)(F)C2)=O)CC1 54239,c1(C(N(CC(N2C(CN(C(C)=O)C)CC2)=O)C2CC2)=O)ccc(Br)cn1 54240,c1(C(=O)NCC(CN(C(=O)CC2COC(=O)N2)C)(C)C)cn2ccccc2n1 54241,N1(C(c2ncoc2Br)=O)CC2CCN(C(c3cnn[nH]3)=O)C2C1 54242,Cc1cc[nH]c1C(N1CCC1c1cn(CC2CCCC2=O)nn1)=O 54243,c1(CC)ccc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)cc1N 54244,Cc1nc(CCC(=O)N2CC(C(C)NC(c3sccc3C(C)C)=O)C2)[nH]c1C 54245,S(=O)(=O)(c1cccc(=NCC2CCCC2)[nH]1)NC1C(OC)C2(C1)CCC2 54246,C1(C)(CC)CC(NC(c2c(OC)cccc2C)=O)CN1C(c1cnc(S)nc1)=O 54247,N1(C(c2c(C)n(C)cc2)=O)CCCC(C2CCCN(C(=O)CNS(N)(=O)=O)C2)C1 54248,C12(NC(c3cc4occc4s3)=O)CCCN(C(c3cnccn3)=O)CC1C2 54249,c1(CN)cnc2sccc2c1.c1(C(N2CC(C(=O)O)(C)C2)=O)nccnc1Cl 54250,CC1COCC(CC(=O)NCC2CCN(C(c3cc(=N)[nH]n3C)=O)CC2)O1 54251,c1(COC)cc(C(=O)NCC2(CC(=O)NCC3CCOC3)CC2)no1 54252,C(=O)(C1=C(Cl)CCCC1)NC1C(CO)CCN(C(c2cnc(CC)[nH]2)=O)C1 54253,C1(C2CC2)(C(=O)NCc2cc(C(N(C(C)CC3CC3)C)=O)n[nH]2)CC(=O)C1 54254,c1(NC(C2N(C(CCc3n(C)ncc3)=O)CCCC2)=O)ncc(I)nc1Cl 54255,CS(=O)(=O)CCC(=O)NCCC1(O)CCN(C(=O)CSc2n[nH]c(O)n2)C1 54256,N#CC1(NC(c2ccc(I)o2)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54257,c1(C(=O)NC(C(=O)NCCCCN(CC)CC)C)occ2c1CCC2 54258,Cn1ncc2nc(C(N3CC(C(=O)O)OC(C(F)(F)F)C3)=O)cn12 54259,CC(C)(CCC(=O)N1CC(C)(C(=O)NC2CCCCC2(F)F)CC1(C)C)[N+](=O)[O-] 54260,CC1CCN(C(c2sccc2C2CC2)=O)CC1NC(c1nscc1Br)=O 54261,c1(C(=O)O)cc([N+](=O)[O-])cc(S(=O)(=O)NCc2cc3cc(Br)ccc3[nH]2)c1 54262,c1(SCC(=O)N(C(CNC(=O)C(CO)c2ccccc2)C2CC2)C)ccncc1 54263,C(C(C(=O)NCc1cnc(O)c(F)c1)C(C)C)NC(C1C(C)=CCS1)=O 54264,C(CC1CC1)(C(=O)NCCN1CC=CC1)NC(C1C(C)C1C)=O 54265,C(=O)(C(F)C(C)CC(C)(C)C)NCC1N(C(C2C(OC)CCC2)=O)CC(C)(C)C1 54266,C(CCCC(CO)NC(=O)CC1CSCCO1)NC(CSCCCC)=O 54267,N1(C(C)C(F)(F)F)CC2C(C(=O)NCc3ccc(Cl)cn3)C2C1 54268,N1(C(=O)CC23COC(CF)(C2)C3)CCN(c2ccc(C(C)C)cn2)C(C)C1 54269,c1(CC(=O)NCC(C)NC(=O)CSc2nccn2C)cccc(C(N)=O)n1 54270,C1(C(=O)NC2CN(C(C3CS(=O)(=O)C3)=O)C2)CC2CCCC2N1C(C1CCC1)=O 54271,c12noc(n1)CNC(=O)C(C)N(C)C2=O.C1(CC=C)(CC)CC1 54272,c1(CCC)cc(C(=O)N(CC(C)(C)NC(=O)CCCC2CC2C)C)ccn1 54273,c1(C(=O)NCC(C)CNC(=O)CCS(C)=O)cc(C#N)ccc1N 54274,C(CC(=O)NC12CC(CNC(=O)C(c3cccc(C)c3)F)(C1)C2)(C(F)(F)F)OC 54275,c1(C(=O)NCC=CCNC(c2n(COC)ncc2)=O)cccc([N+](=O)[O-])c1C 54276,C1(C(N(C(C)C(=O)O)CCc2cn(CC3CC3)nn2)=O)CCC(C(O)CO)CC1 54277,C=Cc1cncc(C(N2CCC(NC(C3CCC(C(C)C)CC3)=O)C(F)C2)=O)c1 54278,C=Cc1ccc(C(=O)NCCCNC(=O)Cn2nnc(-c3ccco3)n2)cc1 54279,c1(N2CC(CCNC(=O)Cn3cccc3)(OC)C2)cc(=O)n(C(C)C)c(O)n1 54280,C(COC)(C(=O)OC(C)C)NC(=O)OC1CN(C(C(C)OCOC)=O)C1.C(C)(C)OC 54281,c1(N(C(C2C(C)C2C)=O)Cc2cccc(OC)c2)ccc(S(N)(=O)=O)cc1 54282,c1(OCC)nc(Cl)ccc1C(=O)NC1(C)CN(C(C2CC3(CCC3O)C2)=O)C1 54283,c1(CC(=O)NC2C(NC(C(C)c3cccs3)=O)CC2)cccc(OC2CCC2)c1 54284,C12(C(N(CC(C)NC(C3CN(CCC)C(=O)C3)=O)C)=O)CCOC(C)(C1)C2 54285,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCCn2nc(C)c(C)c2C)C1)NC 54286,c1(C(N2CC3CC3C2)C(=O)NCCSC)cc(Br)no1 54287,N1(C(CN(CC)CC)=O)Cc2ccccc2C(NC(c2ncc[nH]c2=O)=O)C1 54288,n1(COCC)nnc(C(N2CC(CNC(=O)Cc3ccncc3)(OC)C2)=O)c1N 54289,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54290,Cc1ccc(C(N2CCCC2(C)C(=O)NCCC2CCCC3CC23)=O)cc1O 54291,Cc1cccc(C(=O)NCC2CCC(NC(=O)CSc3nncs3)C2)c1 54292,N1(C(CN2C(C)CC2)=O)CCC2(CC1)CCN(C(c1cc(C#N)on1)=O)C2 54293,c1(CNC(CCCCC)C2CC2)ccc(Cl)c(Cl)c1 54294,O=C(C#CC1CC1)NCC1CC(F)CN1C(C1CC1Cc1ccc(Cl)cc1)=O 54295,C1(C)(C(=O)NCCN(C(=O)C(C(C)C)NC(N)=O)CC)CCC(C)=C(C)C1 54296,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2ccco2)=O)CC(O)C1 54297,N1(Cc2ncc(-c3ccc(C)cc3)o2)CCC(F)(F)C(NC(C)=O)C1 54298,C(=O)(C(C)CS(C)=O)NC1(CC=C)CN(C(=O)CCCc2cccs2)C1 54299,N1(C(c2ccc(OC)cc2)=O)CCC(F)C(NC(c2cccnc2N(C)C)=O)C1 54300,C(CC1=CCN(C(C2CCCCN2CC(F)F)=O)CC1)NC(C=C(C)C(F)F)=O 54301,C=C1CCN(C(C2CN(C(=O)Cn3ccc(C)n3)CC2C)=O)CC1 54302,O=C(CCCn1cncn1)NCCC1CCN(C(c2ccco2)=O)C1 54303,c1(CNC(=O)Nc2ccn(C(=O)Cc3ccccc3)n2)cnn(C2CC2)c1Cl 54304,C1(NC(=O)CCc2ccco2)CC2(C1)CC2NC(=O)CCCc1ncco1 54305,C(C(=O)NC(CC(=O)NCCc1ncc(C)o1)C1CC1)(C(C)C)OCC 54306,c1(C(=O)NC(C)CN(C(=O)C(C)N(C)C)C)cc2c(C(F)F)nn(C)c2s1 54307,c1(C(C(=O)NCC(C)CNC(=O)CSC2CCNC2=O)O)ccc([N+](=O)[O-])cc1 54308,C1(C)(N(C2CCCCC2F)C)CCC2(CC1)OCCO2 54309,N1(C(C(CC(F)F)NC(C(CSC)OC)=O)=O)CCC(F)(F)C(F)C1 54310,C1(C(=O)NC(C=C)C2CC2)CC(=C)CCN1C(=O)COCCOCCOC 54311,N1(C(COCCC)=O)CCOCC1CNC(=O)C(F)C(C)C 54312,S(=O)(=O)(c1cccnc1NCC1CCN2CCCC12)N1C(C)CSCCC1 54313,c1(OC)cnc(OC)c(C(=O)NNC(=O)C2CC2(Br)Br)c1 54314,N1(C(C(CC)C#N)=O)CCC2(CC(C=O)C2)C1.N1(C(=O)N(C)C)CC(O)C1 54315,c1(C(=O)NCC(CC(C)C)NC(C(C)(CO)NC(C)=O)=O)cnc2cc[nH]c2c1 54316,C1(NC(CC(c2ccc(C)s2)O)=O)CCn2nnnc2C1 54317,C1(C(N(C2CCN(C(c3c(Cl)cn(CC)n3)=O)C2)CCO)=O)CC12CCCCC2 54318,c1(C(=O)NC(C)(C)CCNC(=O)CC2(O)CCOC2)cc2ccncc2cc1F 54319,CC1(C)CCC(C(N2CCCC(NC(=O)CN3CCCCC(=O)C3=O)C2)=O)CC1 54320,c1(C(N(C(C)C(=O)N(C)C)C2CC2)C)ccc(I)cc1 54321,C1(C(=O)NCC(C2CCCN2C(c2nocc2Cl)=O)(C)C)CN2CCC1CC2 54322,C1(N(CC(=O)OC)CC)CN(c2nccc(OCc3ccccc3)n2)CCC1C 54323,N1(C(CCCOCCOC)=O)CCC2CN(C(c3coc(O)n3)=O)C2C1 54324,C1(CC(F)(F)F)CCCCC1CNc1ncc(C2CCCO2)s1 54325,O=S(=O)(c1ccc(NCC(O)Cn2cccn2)nc1)N1CCc2nocc2C1 54326,C12(C(N)=O)CC(C(=O)NCn3ccc(C(=O)NC4CCN(CCF)C4)c3)(C1)C2 54327,C1(NC(COCC=C)=O)CC2(CCC2)CN1C(=O)Nc1[nH]ncc1C#N 54328,C(=O)(CS(=O)(=O)Nc1ccccc1)N1CCC(CN(C(C=CC=CC)=O)CC)C1 54329,C(=O)(C(C#N)C(C)(C)C)NC(C(NOCC=C(C)C)=O)Cn1cncn1 54330,c1(C(N(C(C)C)CCN(C)C(c2cc(Cl)c[nH]2)=O)=O)ccc2c(c1)N(C)CC2 54331,C1(C)(NC(c2occ(C)c2C)=O)CCC(NC(C2CCN(C3CC3)CC2)=O)CC1 54332,N1(C(C=C(C)C)=O)CC2CCC(NC(c3n[nH]c4ccc(Cl)cc34)=O)CC2C1 54333,N1(Cc2ccc(C(CC)O)o2)CCOCC1C 54334,C1(COC)CC(CNC(c2csc(S)n2)=O)N(C(c2[nH]c(O)nc2C)=O)C1 54335,C1(F)(C(N2C(C(=O)NCCN(OC)C)CCC2)=O)CCCOC1 54336,CC1C(O)CC2CCC1N2C(c1ccnc(CNC(C2C(F)(F)C23CC3)=O)c1)=O 54337,c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC(C)NC(=O)C(C)CC1CC1 54338,c1(C(C)C(N2CC(O)CC2CNC(=O)C=CCO)=O)ccc(Br)cc1Cl 54339,CON(C(=O)CCC1CCCN1C(=O)NC1C(C)(C)C1(F)F)C1CCC1 54340,CCC(CC)(CO)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C)CC1 54341,C(COC)(C(=O)N1CC(O)(CCNC(=O)C(F)(F)c2ncccn2)C1)OC 54342,C1(OC(C)CO)CCN(C(=O)C(Cc2cn[nH]c2)N(C)C)CC1.C1(=O)CC2(CC2)N1 54343,C(C(C)(C)C(=O)NC1CCCC1CC(=O)NOCC=CCl)N(C)C 54344,c1(C(N(C)CC2CCCN2C(=O)CSc2nncn2C)=O)cc(F)nn1C 54345,Cn1ncc(NCc2cccnc2P(C)(C)=O)c(Cl)c1=O 54346,c1(C(C2CN(CC3CCC(O)C3)C2)C2CCC2)ccc(Cl)cc1 54347,c1(C(N(C2CCN(C(=O)C=CC(=O)OC(C)(C)C)C2)CC)=O)cc(=O)n(C)cn1 54348,C1(C(N2C(C)(CC(=O)NC)CC2)=O)CC2(CC(NC(C3CCCC(=O)N3)=O)C2)C1 54349,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54350,N1(C(=O)NCc2ccn(C(C)C)n2)CCN(C2CCCOC2)CC1 54351,N1(C(Cc2c(C)nsc2)=O)CC(NC(c2cc(F)c(Cl)cc2Cl)=O)C(N=[N+]=[N-])C1 54352,N1(CCn2ccn3ncc(C(F)(F)F)c23)CCc2[nH]nc(C(F)F)c2C1 54353,c1(C(C)N(C)C(C2CCN(c3cccc(Br)n3)CC2)=O)ccccc1Cl 54354,c1(CC(=O)NC(C2CCN(CC(O)Cc3ccccc3)C2)C)ccc(F)c(F)c1 54355,c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cnc[nH]2)C)c[nH]c2c(C#N)cccc12 54356,C1(C(=O)OC)(CC)CC(NC2CC2)C1.c1(C(=O)N)ncsc1C.C12(CC1)C(=O)N2C1CC1 54357,C1(NC(=O)C2=CCCC2)CCCCC1OC(=O)COc1cccnc1 54358,c12cc(cc(F)c1)CN1CCN(C(CO)C1)C2=O.c1(C=O)cc(Cl)c(Br)s1.CO 54359,C(C(C)C(F)C(=O)NCCc1cnn[nH]1)NC(c1c(C)nsc1C)=O 54360,C(=O)(C(CC)(CC)CC)N1CC=CC(C(=O)NC(CCC=C)C(=O)OC)C1 54361,N1(C(C(C)c2ccco2)=O)CCCC(C)(N(C(=O)CCc2cccnc2)C2CC2)C1 54362,c1(CC(=O)NCC2CCN(C(COCc3onc(CC)n3)=O)C2)cnccc1C 54363,c1(C(N2CC(C)C(CNC(=O)Cc3csc(Cl)c3)C2)=O)cc(Cl)cc(F)c1N 54364,CC1CCCCC1CC(=O)NCC1(C)CC(C)(C)C1.C12CC(C1)NC2=O 54365,N1(C(C(CCSC)O)=O)CCOCC(C(=O)NCCC(C)COC)C1 54366,C(c1cccc(Cl)c1)=CC(=O)NC(C(C)NC(CN(C(COC)=O)C)=O)C 54367,C1(NC(c2ccc[nH]2)=O)CC(F)(F)CC1NC(C1CC(N2CCCC2)C1)=O 54368,n1(CC(=O)NC2CC(CCNC(C=CC(CC)C)=O)C2)cc(C#N)c(O)nc1=O 54369,c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)COC2)ccc2cccnc2c1N 54370,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54371,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54372,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54373,C1(NC(CC2CN(C(C)=O)C2)=O)CC12CC(NC(c1cccc[n+]1[O-])=O)C2 54374,N1(C(C)Cn2ccnc2)C(=O)NC2(CCC2)C1=O 54375,C1(=O)NNC(=O)C(C)OC23CC1(OC2)C3.c1(C(=O)OCC)cn2ccccc2n1 54376,C1(CCC)CN(C(C2CCC(OC)CC2)=O)CC1NC(C1CC(C)(O)C1)=O 54377,C1(CNC(=O)COCC2CC2)CCNC12CCOCC2 54378,N1(C(C(CSC)C)=O)CCC(C)(CNC(c2c(C)coc2C)=O)C1 54379,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2(O)C(C)(C)OCC2)=O)CCCC1 54380,CC(C)C(O)C(C)C(=O)Nn1cc(CC2CC(c3ccc(F)cc3)C2)nn1 54381,CC1(O)COCCN(C(c2cc(CNC(=O)CCc3ccncn3)no2)=O)C1 54382,N1(C(CCC#CC)=O)CC(NC(C2(OC)CCOCC2)=O)C(C2CC2)C1 54383,Nc1ccc(C(=O)NC2CC2NC(c2cnc(C(F)(F)F)cn2)=O)nc1F 54384,Cc1[nH]nc(Cl)c1NC(=O)N(c1cnn(CCN(C)C)c1C)C 54385,Cc1nc(CCC(=O)NCC2CC2NC(C2(F)CCC2)=O)cs1 54386,C1(CNC(=O)C2=CCCCC2)C(C2CC2)CCN1C(c1cc(Cl)nnc1Cl)=O 54387,c1(C(=O)NCCCNC(=O)OC)ccc(C(=O)NCC(C(C)(C)C)NC)c(C)c1 54388,C(=O)(C(=O)NNc1cc(C)c(Cl)cn1)OC.C1(=O)CC(C)(O)CC2C3CC(CC23)N1 54389,C1(C(C)CO)CCN(C(=O)N(CCC2CCCO2)CCO)C1 54390,C1(C2CC2)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CCN(C(=O)Cn2cnnc2O)C1 54391,N1(C(c2ccc(N)c(C)c2C)=O)CCN(C(=O)CC2CC3CC3C2)CC(C)(C)C1 54392,C(C(CC(=O)N1CC=CC1)NC(=O)C(C)CC#N)OC 54393,N1(C(c2cc(CC)nn2C)=O)CC(N(C(=O)CCCOC(C)(C)C)C)C(C)(C)C1 54394,C1(c2cn(C3CCC(C(N4CC(CO)C4C(C)C)=O)C3)nn2)(OC)CCCC1 54395,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(C1(CCO)CC1)=O)C2 54396,C1(Nc2nc(C)nc(=N)[nH]2)CC2CCC1CN(C(C1(C(C)C)CCC1)=O)C2 54397,c1(C(=O)NC(CC)CNC(=O)CCOC(C)=O)cnoc1-c1cccs1 54398,N1(C(CN(C(C2ON=C(C(C)C)C2)=O)C(C)C)=O)CCCN(C=O)CC1 54399,O=C1NC2(CCO1)CN(C(=O)C(c1ccoc1)NC(C1CCC=CCCC1)=O)C2 54400,C1(C)(C(N(C2(CC)CC2)C)=O)CC(O)CN1C(=O)C(CC1CCC1)OC 54401,CN1CCCC(CNC(C2CC(NC(c3cc(F)n(C)n3)=O)C23CCC3)=O)C1=O 54402,C(=O)(C(C)(F)C(=O)OC)N1CCC(NC(C(CC=CCC)C)=O)CC1 54403,C12CN(CC1C)N2C(c1n[nH]c(C)c1Br)=O.c1(COC2(CSC)CC2)ccccc1 54404,C(=O)(C(CO)C(C)(C)C)NCCC(C)(C)NC(C(c1ccccc1)OC(C)C)=O 54405,c1(NC(C2N(C(C(COCC)C)=O)CCCC2)C)ncc(C)c(SC)n1 54406,Cc1sc(C(=O)NC(CC(C)C)c2nnnn2-c2ccc(Cl)cn2)c(Br)c1C#N 54407,c1(NC(c2ccc(-c3ccccc3)cc2)=O)nc2c(o1)CCC(F)(F)C2 54408,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2C)=O)n1 54409,NS(=O)(=O)c1ccc(-c2c[nH]nc2C(=O)Nc2ccccc2I)cc1 54410,c1(C(=O)Nc2cccc(NC(C)=O)c2O)c(O)ccc2ccccc12 54411,c1(CC)nc(C(=O)NC2CC(CNC(=O)CC#N)C23CCC3)c2ccccn12 54412,c1(C(N2CC(C)N(C(C3(C)CCC(=O)N(C)C3)=O)CC2)=O)cc2nc[nH]c2cn1 54413,N1(C(C(F)OC)=O)CCC(NC(c2ccccc2N2CCCCC2)=O)C(C)C1 54414,C(C(CNC(=O)CCc1cnn(C)n1)CO)NC(C1CN(C(C)=O)C1)=O 54415,N(C1CCCc2c(I)n[nH]c21)C(c1coc(C(F)(F)Br)n1)=O 54416,CC1(C)CCCC(C(=O)NCC2CCCN2C(=O)CC2(C)CCOCC2)C1 54417,c1(OC)cc(-c2csc(C(F)(F)F)c2)ccc1C(N)=O 54418,N1(C(c2nnc(CC(C)C)s2)=O)CCN(C(=O)C2=CC3CCCC23)CCC1C 54419,C12(NC(C3C(=C)C3)=O)CCC(NC(C3CCN(CC(F)F)CC3)=O)(CC1)C2 54420,C(=O)(CCC(=O)c1cccs1)NC(C(C)NC(=O)CN(C1CCC1)C)CO 54421,c1(C(=O)NC2CC(NC(C(C)C(C)O)=O)C2)cc(F)c(Cl)cc1Cl 54422,C1(NC(C(C)OC2CCCCC2)=O)CCCC(CNC(C23CC(C)(C2)C3)=O)C1 54423,c1(C(N2C(CN(C(=O)C(C)(C)C)C)CCC2)=O)cncc(NS(=O)(=O)C2CC2)c1 54424,c1(C(C(=O)N(CC(O)C(=O)N2CC(OCC(N)=O)C2)C)=O)ccc(O)cc1 54425,c1(C(CN(C(C2N(C(=O)OC)CSC2)=O)C)O)ccc2ccccc2c1 54426,N1(C(N(C)C)=O)CCC2(CCN(C(C3(c4ccccc4Br)CC3)=O)C2)C1 54427,c1(C(=O)NC(CNC(COCC=C)=O)C)ncc(C)cc1C 54428,c1(N(CC(C)CNC(=O)CC(C)C2CCCCC2)CCO)ncnc(Cl)c1Br 54429,N1(C(Cn2c(C)ccc2C)=O)CCCC(N(C(=O)C(c2ccccc2)F)C)CC1 54430,N1(CCOCCC(C)C)CCC(NC(C2CC2(C)C)=O)CC(C)(C)C1 54431,C12(C(N3C(CNC(c4c(C)nc(CO)s4)=O)COCC3)=O)CCC(F)(CC1)C2 54432,C1(OC(C)C)C2CC3C1C3C2C(N1CC(CC(=O)N(C)C)C1)=O.C1(C)C(=O)N1 54433,c1(C(=O)NC2C3CN(C(CCc4nc(C)c(C)o4)=O)CC2C3)c[nH]c2nccc-2c1 54434,C1(NC(CC(C)C)=O)COC2(CCN(C(C3CC(n4ccnc4)C3)=O)CC2)C1 54435,C1(C(=O)NC2C(NC(=O)C(c3ccc(O)cc3)=O)CCCC2)CC12CCOCC2 54436,n1(CC)nnnc1C(c1cscc1Br)NCc1nnc(SC)s1 54437,c1(C(=O)NCC2(C)N(C(c3cc(C)c(N)cn3)=O)CCC2)ccc(S(N)(=O)=O)cc1 54438,O(NC(=O)C(C)N(C(=O)CCc1scnc1C)C)C(CC)CC 54439,C1(F)(CNC(CN(C)C(=O)C2CC2)=O)CC(CNC(=O)CC2CCC3CC23)C1 54440,Cc1nc(C(F)(F)F)cc(=NCC(C)N(C(=O)C(c2ncccc2C)(F)F)C)[nH]1 54441,C#CCCCCC(C)C(=O)N1CCC(C(=O)NCCN(C)C2CC2)(CC)C1 54442,S(=O)(=O)(c1ccc(N2CCCCC2)cc1)NCCOCCC#N 54443,C(=O)(CC(O)(c1ccccc1)c1ccccc1)NC(=O)Cn1cnnn1 54444,N1(CC(=O)NCC(CC=C)NC(=O)C(=O)NCC2CC2)C(C)CCC1C 54445,CC1(C)C(NC(C2CCS2(=O)=O)=O)C(C)(C)C1NC(C1C=CC=CC=C1)=O 54446,C1(C(=O)NC(C)(C)CS(C)=O)CN(C(C2CCSCC2)=O)CC12CC2 54447,CC1(C(C(=O)NCc2ccccc2Br)NCC2(C)CC2(F)F)CC(F)(F)C1 54448,Cc1nc(N2CC(NS(=O)(=O)N3CCOCC3)C2)c2cnn(C(C)C)c2n1 54449,C1(NC(C2(CCOCC)CCCC2)=O)CCCN(C(=O)CC(F)(F)CC)C1C 54450,C1(COC)(CNC(C2CCC(C)CC2)=O)CCCN1C(=O)CCOC1CCOC1 54451,c1(C(=O)NC(CC)CN(C)C(c2nscc2Br)=O)cn(CC)nc1C 54452,c1(C(N2CC(CNC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54453,c1(C(N2CCC(CO)C2)C(=O)OC)cccc(Cl)c1F 54454,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)F)C1)NC 54455,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(C1C=CCC1)=O)C2 54456,c1(NC(c2nc(C(N3C4COCC3C4)=O)cs2)=O)cnc(I)cn1 54457,C1(CNC(c2ccc(C3C(C)C3)o2)=O)CCCC(CNC(=O)C(C)(F)F)C1 54458,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54459,c1(C(=O)NCCC2N(C(CCC#CC)=O)CCC2)ccc2c(c1)OCCO2 54460,Cc1nc([N+](=O)[O-])cn1CCC(N1CC(NC(C2(C)CC(C#N)C2)=O)CC1C)=O 54461,c1(C(=O)NC2C(N(C)C(c3ccc(F)c(N)c3)=O)CCC2)cc2c(s1)CCCC2 54462,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 54463,c1(C(=O)NCC(C)C(=O)NCCN2CCCC(CSC)C2)cnc(Cl)c(N)c1 54464,c1(C(N2C(CCC)CN(C(=O)C(C)OCC)CC2)=O)cnc2sccc2c1 54465,C1(CNC(CCC(=O)OC)=O)CC2CCCC2N1C(=O)COCc1cc(C)on1 54466,Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(CN(C)C(c2ccon2)=O)C1)=O 54467,c1(C(=O)NC2CCC3(CN(C(COC(C)=O)=O)C3)O2)cccc2c1CC(=O)N2 54468,c1(C(N2CCC(CN(C)C(C3(C(N)=O)CC3)=O)C2)=O)ccc(O)nn1 54469,C1(=CC(=O)NC(C2(O)CN(C(=O)C=Cc3ccsc3)C2)C)CCSCC1 54470,c1(C(=O)Nc2nc(Cl)c(Br)nc2Cl)c[nH]c2cc(-c3cnn(C4CC4)c3)cnc12 54471,C1(NC(c2cc(CNC(C(CC)=CCC)=O)no2)=O)CC(C)(C)OC1=O 54472,Cc1ncc(Cl)c(C(N2CCC(F)(CNC(c3nn(C)cc3Br)=O)C2)=O)n1 54473,c1(OC)ccccc1OCC(N1CC(O)(C(C)NC(C2CCC(C)O2)=O)C1)=O 54474,C1(C(N2CC(CSc3cccs3)C2)=O)CC(F)(CNC(c2cnn(CF)c2)=O)C1 54475,Cn1cc([N+](=O)[O-])c(C(=O)NC(C)(C)CNC(c2cccc(C3CC3)c2Cl)=O)n1 54476,C1(C(N2CCC(NC(c3ccc(Cl)cc3Cl)=O)C2)=O)CC2(C1)CC1(CCC1)C2 54477,C1(C(N2CC(CN(C(c3c(OC)n[nH]c3)=O)C)OCC2)=O)OCCN(C)C1=O 54478,n1(CC(=O)N(C(C)CNC(c2conc2C)=O)CC)ncc2ncccc12 54479,c1(OC)c(F)cc(C(=O)NC(C)(C)C(C)NC(=O)CC2CC=CCC2)c(N)c1F 54480,c1(C(N2CCC3CN(C(CN(C)C(N)=O)=O)C3C2)=O)coc2c1C(=O)CCC2 54481,c1(C(=O)NC(C2CCN(C(c3cc(C(F)F)on3)=O)C2)C)ccc(O)cc1Cl 54482,C1(NC(C(C=C)(C)O)=O)CN(C(c2ccncc2N2CCCC2)=O)CC(C)(C)C1 54483,c1(C(CNC(C=C(C)CNC(C2CCO2)=O)=O)F)ccccc1 54484,C(C(C)(F)C(C)(C)F)NC(C(Cn1ccnn1)NC(C(C)OCC(C)C)=O)=O 54485,CCC(C(=O)N1CCC(CNC(=O)CC2CCC(O)C2)C1(C)C)C(C)(F)F 54486,C(N=c1[nH]c(N2CCc3sc(Cl)cc3C2)nc2cc[nH]c12)C1(C)CC1(Cl)Cl 54487,C(C1CCCN1C(=O)CC1CC1)=CC(=O)NCC(C)C1CCC1 54488,c1(OC)ccc(C(N2CC(=O)NC(C)C2)C(=O)NCC2CCCO2)cc1C 54489,C1(N(CC(=O)N(C(C)(C)CC)C)C(=O)CN2CC=CC2)CC2CCC1C2 54490,N1(C(C2C(C)CCO2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)C1 54491,Cn1cc(C=CC(N2CCCC2COC)=O)cn1.c1(-c2c[nH]nn2)cccnc1O 54492,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC1CC1 54493,c1(-c2cc(C(=O)NC3CN(C(c4ccn(C)c4)=O)C3)n[nH]2)ccccc1O 54494,C(C1c2ccsc2CCN1C(=O)C(COC)OC)NC(CCCCCCC=C)=O 54495,C1(CC)(CC)CCC(NC2(c3nnnn3C)CCOCC2)CC1 54496,C1(N(C(=O)C(F)CC2CN(C(=O)Cc3cn[nH]c3)C2)CC)CCCN(C(C)=O)C1 54497,Cc1c(NC(=O)C(C)C)cccc1SCC(O)(CO)CO 54498,C(=O)(C(O)CC(C)(C)C)N1C(c2cn(CCC(C(=O)OC)O)nn2)CC1 54499,C1(CC(=O)NCC2(C)CCOCC2)CCN(C(C23CCC2CNC3=O)=O)C1(C)C 54500,C1(C(=O)NC(C2(O)CN(C(C3CCCC(F)(F)C3)=O)C2)C)CCC(C)(C)CC1 54501,c1(C(N2CCC(N(C(=O)C(C)SC)CCC)CC2)=O)cc2sc(C)cc2[nH]1 54502,c1(C(=O)NCC(C(=O)N(CC(C)(C)N(C)C)C)OC)ccc(CO)cn1 54503,C(CC(=O)N1CCC(O)(CO)C1)(C(F)F)NC(c1cncc(CC)c1)=O 54504,Cc1csc(C(N2CSCC2C(=O)NCCOc2ccccc2)=O)c1 54505,N1(C(C2CC(=C)C2)=O)CCC(C(=O)NC2CC(CC(N)=O)C2)(CF)C1 54506,C(=O)(CCCCC(F)(F)F)N(C1CN(C(Cc2cc(CC)c(OC)cc2)=O)C1)C 54507,c1(C(=O)NCC(CN(C(=O)CN2CCCC2)C)O)cc2sc(Cl)cc2s1 54508,c1(C(N2CC=CC(C(=O)NCC(CC)C(C)C)C2)=O)ccc(C)nc1C 54509,c1(C(N2CC(O)(CNC(c3cc(Cl)cc(Cl)n3)=O)C2)=O)cc(Cl)cc(Cl)c1O 54510,c1(OC)ccn2cc(CNC(=O)NC(c3ccnn3C)C(=O)O)nc2c1 54511,c1(CN(C)Cc2ccc(C(C)C)cc2)cc(F)ccc1Cl 54512,CC1(CNC(C2CCCN(C(C3C4CCCCCC34)=O)C2)=O)CCCCC1O 54513,c1(NCC=CC(N2CCN(c3ccccc3)CC2)=O)nnc(O)cc1O 54514,Cc1c(C(N2CC3(CCC3NC(C34CCC(CC3)CC4)=O)C2)=O)cccc1CO 54515,C1(C)(CNC(C(C)n2ccnn2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)C(C)(C)C1 54516,CCC(CC)C(C(=O)N(C(CNC(C1(Cl)CC1)=O)Cc1ccccc1)C)OC 54517,CC(C)(C)CC(=O)N1CCCC(CNC(c2scnc2-c2ccccc2)=O)C1 54518,CCC(CC)(C(=O)NC1CCC(CNC(c2ccc(=O)n(CC)n2)=O)CC1)OC 54519,C1(C(N(CCC(F)(F)F)CC)=O)(CC)CCCN(C(=O)CCC2CCCOC2)C1 54520,C1(OCCCNC(=O)Nc2c(CCC)nco2)CCCCCC1 54521,C1(CC(=O)NC2C=CC(CC(=O)Nc3c(C)coc3)C2)CCCCN1C 54522,CCC(C#N)C(=O)N1CC(F)CC1CNC(=O)COCC(C)C 54523,N1(C(C(c2cccc(O)c2)C)=O)CCC2(C1)CN(C(=O)C(C)C(C)O)CCO2 54524,n1(CC)cc(C(=O)NC2CCC(CCNC(=O)CCc3ccncc3)C2)nn1 54525,N1(C(CC2CCC(C)CC2)=O)CCC2CN(C(c3cnsc3)=O)CC12 54526,Cc1cc(C(=O)NC2CCCCC2NC(=O)CCCn2cncn2)ncc1C#N 54527,N1(C(c2occ(C)c2)=O)CCOCC(C)(CNC(c2cc([N+](=O)[O-])ccn2)=O)C1 54528,CCC(C)(CC)C(=O)NC(C1CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1)C 54529,C1(c2nc(N(C)CCF)nn2C)Cc2cc(N(S(C)(=O)=O)C)ccc2O1 54530,CCC(CCC(=O)NC1CCN(CC)CC1)NC(=O)CC(C)SC 54531,c1(CC)cc(C(=O)N(CCCNC(=O)Cc2cccnc2Br)C)sc1C 54532,C1(NC(C23OCC(COC)(C2)C3)=O)CCCCN(C(=O)C(C)CCN(C)C)C1 54533,N1(C(Cc2ccc(C)nc2)=O)CCC2(CC(NC(=O)CC3(C)CCOCC3)C2)C1 54534,c1(CC)nn(C)c(CN(C=O)Cc2ncsc2Br)c1Cl 54535,N1(C(CNC(C=C(CC)C)=O)C)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54536,C1(NC(C)=O)CC(F)(F)CC1C=O.C(=O)(C1=CCSC1)N1C(C)CCC1 54537,Cc1ccc(C2CC2NC(N2CC(OC)C(n3cncn3)C2)=O)cc1 54538,O(NC(=O)CCCN(C(=O)C(C)CNC(N)=O)C)CCCC 54539,c1(C(=O)NC2(CCCNC(CC(CC)OC)=O)CC2)c(C)cccc1Cl 54540,N1(C(c2cccc(C#C)c2)=O)CCC(NC(=O)C(=O)NCCC(N)=O)C(F)(F)CC1 54541,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54542,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2C(C)C)=O)CC1C 54543,C(N=c1nc2c(cnn2C)c(N(CC(C)(F)F)CCCN(C)C)[nH]1)=CC 54544,N1(C(C2CCC3(CCC3)O2)=O)CC(S(=O)(=O)N2CCC2C(=O)NC2(CO)CC2)C1.C1CC1 54545,c1(C(=O)NCC(=O)NC(CC)CNC(C)=O)ccc2c(c1)CCCN2C(N)=O 54546,N12CCCC(CC1)C(=O)NC(=O)C2C.N1(CCCC)CCC(N2CCOCC2)C1 54547,N1(C(c2nc(CC)[nH]n2)=O)CCC(C2CCCCN2C(c2scnc2Cl)=O)CC1 54548,c1(C(=O)NCCN(C(c2nc(C3CC3)oc2C)=O)CC)cccc(S(N)(=O)=O)c1 54549,Cc1c(C(=O)NCC(O)CN(C(=O)C(C)Oc2ccccc2)CC)cc(O)cc1N 54550,C1(CCC(N2CCC2c2cn(CCOCCO)nn2)=O)CCCC(=O)N1 54551,C12(CC=CC1)N(C(=O)CC1CC1)C2.C=C1CC(C(=O)Nc2ccsc2)C1 54552,C1(C(NOCC(=O)NCCc2cccc(C)n2)=O)CCCCC1(C)C 54553,C1(C(=O)NCCCNC(c2c(CC)onc2C)=O)OCCOC12CCC2 54554,N1(CC(=O)NC2(CN(C(=O)CC3(C)CCCCC3)C)CC2)CCCC(O)C1 54555,c1(C(=O)NC2C3CC(NC(C(CC)(F)F)=O)CC32)cc2ccccn2c1 54556,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(Cc1cnc(C)[nH]1)=O 54557,C(=O)(CCCC(C)NC(c1occc1C1CC1)=O)NC(COC)(C)CO 54558,c1(OCC)cccc2c(NC(=O)NC3CCC(CO)CC3)c([N+](=O)[O-])cnc12 54559,N1(C(C)C(=O)NC(C)(CNC(=O)C(C)(C)CF)C2CC2)Cc2ccccc2C1=O 54560,C1(NC(c2ccc(C)n2C)=O)C(C)(C)CN(C(C2CCNC(=O)C2)=O)CC1(C)C 54561,C(C(C(C)C)NC(c1csc(=N)[nH]1)=O)(c1ccccc1)NC(CNC(=O)OC)=O 54562,C1(NC(C(COC)(C)C)=O)CCN(C(c2cccc(CN(C)C)n2)=O)C(C)C1 54563,C=Cc1cncc(C(=O)NC(CCOC)C(=O)NC(C)COC(F)(F)F)c1 54564,Cc1nscc1C(=O)NC(C)Cn1cc(CNC(=O)OC(C)(C)C)nn1 54565,C1(NC(C(CC)c2ccccc2)=O)CC(C)N(C(C2CCCC2SC)=O)C1 54566,Fc1ccsc1CCCc1nc(-c2cn[nH]c2C(F)(F)F)no1 54567,N1(C(N(CCCCC(=O)O)CC(C)C)=O)CCCC(Cc2ccccc2)C1 54568,c1(NC(c2cccnc2)CC)nc(N2CCN(CCO)C(C)C2)nc2sccc12 54569,c1(C(N2CCN(C(C(C)SCC)=O)C(CCOC)C2)=O)cc2ccsc2c(O)n1 54570,CC(C(=O)N(C1CC(NC(c2ccn(C3CC3(F)F)n2)=O)C1)C)C(F)F 54571,N1(C(c2sccc2CO)=O)CCCC2C1CCCN2C(c1cnn2c1OCCC2)=O 54572,c1(NC)cc(Cl)ccc1C(=O)NCC(c1cc(F)cc(F)c1)NC(=O)C(C)(C)F 54573,C1(CC(=O)NCC(CC)(CC)NC(C2CCC(=O)N(C)C2)=O)NC(=O)CN(C)C1=O 54574,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54575,CCCC(C)(CCC)C(=O)NC1CCCCC1NC(c1cc(C(N)=O)co1)=O 54576,C(C1=CCCN(C)C1)NC(C(N1CC(CNC(c2scc(OC)c2)=O)C1)C)=O 54577,CCC(CC(=O)N1CCC(CCNC(=O)CCn2ccnc2C)C1)C1CCC1 54578,C(=O)(CC1=Cc2ccccc2C1)NCC1CC(C)N(C(=O)Cc2n[nH]c(=N)s2)C1 54579,C(CC(=O)N(CCCN(C(=O)C=CC(=O)N(C)C)C)CCO)OCOC 54580,C1(CNC(c2c(C(=O)OCC)[nH]cc2C)=O)C2CCCCCN12 54581,CC1(C)CC(CNC(c2c[nH]c(Br)c2)=O)N(C(=O)Cc2ccc(F)cc2)C1 54582,C1(C(=O)NCc2n(C)cnn2)CC2(CCC2)CN1C(=O)CCC1OCCO1 54583,C(=O)(C#CC1CCC1)NCC(CC=C)NC(c1cccc(SCCC)c1)=O 54584,C1(OC)CN(C(c2nn(-c3ccc(F)cc3)cc2C)=O)CC1C(F)F 54585,N1(C(CCSCCCC)=O)CCCC1(C)C(=O)NC(CO)CCF 54586,N1(C(c2cc(C(=O)OCC)n[nH]2)C(=O)NC(C)CC)CC(C)CC(C)(C)C1 54587,CCC(C)(C(=O)NC1CCCN(C(=O)C(F)(F)CO)C1)c1nn[nH]n1 54588,Cc1onc(-c2ccccc2)c1C(=O)NCC(n1cnc(C#N)n1)C 54589,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54590,c1(OCC(N2CC(O)(CN(C(c3c(CC)cco3)=O)C)C2)=O)ccc(O)cc1 54591,c1(C(=O)NC(CCC)CNC(=O)C(F)(F)c2ccnn2C)oc(C)nc1CC 54592,c1(C(=O)NC2CC(C)(NC(C3CN4CCN3CC4)=O)C2)cccc([N+](=O)[O-])c1N 54593,C1(CNC(C2CCN(CCCc3cccc(Cl)c3)CC2)=O)CCCCNC1=O 54594,O=S(=O)(c1nc(N2CCOC3(CCCCC3)C2)ccc1Br)NC1(CO)CC1 54595,C1(NC(C(CC)C#N)=O)(CC)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54596,c1(CC(C)NC(=O)CCOCCN(C(=O)CN2CCCC2)C)cn(C)nn1 54597,C1(OC)(OC)CCN(C(CC2CCCCO2)C(=O)NCC2COC2)C1 54598,N1(C(C(C)NC(CC)=O)=O)CC2CC(NC(=O)C(C)Sc3ccncc3)CC1C2 54599,c12cccc(c1)NC(=O)N2.c1(NC(NCC(C)(C)C)=S)ccccc1Cl 54600,C12(NC(C(F)OC)=O)CCC(C1)N(C(c1cccc(Cl)c1C)=O)C2 54601,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CC(=O)C1C 54602,Cn1cc(CCC(=O)NC2CCC(C(N3CC(C(N)=O)C3)=O)C2)nn1 54603,C1(NC(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CC1CCC(C)CC1 54604,c1(C2C(SCC3N(C(CCCN(CCC)CCC)=O)CC3)C2)ccc(C)nc1 54605,c1(NC(N2CC3(C2)CN(c2ncccn2)C3)=O)cc(Br)c2ccccc2n1 54606,C(=O)(C1CN(C)C(=O)c2ccccc21)N1C(CNC(C(CC(C)C)F)=O)CCC1 54607,c1(C(=O)NC2CC(NC(=O)CC3CCC3(F)F)C2)cnccc1CC(=O)OC 54608,C1(C2CCN(C(=O)Cc3ccc(S(C)=O)cc3)C2)(NC(CS(CC)=O)=O)CC1 54609,C1(NC(c2c(C)nn[nH]2)=O)CC2CN(C(=O)C(C)CCF)CC2C1 54610,C(C1=NOC2CN(C(C(=O)Nc3cc(Cl)ccc3Cl)=O)CC12)OC.c1(CC)n[nH]cc1Cl 54611,CN1CCCN(CC(c2cccc(Cl)c2)NC(C2CC3CCC2N3)=O)CC1 54612,C(CNC(=O)CCc1c(C)n[nH]c1C)(C(C)(C)C)NC(C(C)OCCC#C)=O 54613,C12(C(N(CCC)CC3CN(C(=O)CCSC(F)(F)F)C3)=O)CCC(OC)C1C2 54614,C(=O)(CC(O)CNC(=O)CC1(NC(C2(C)CCOC2C)=O)CCC1)OCC 54615,N1(C(CCCC=C)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C(CCC)C1 54616,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2F)c1F 54617,Cc1cc(C(N2CCN(CC(O)COc3ccccc3)CC2)C(C)N)nnc1C 54618,C1(CNC(C2(F)CCC2)=O)CC(C(C)(C)C)CN(Cc2cc(C)on2)C1 54619,c1(CC(N2CC(CNC(C(C)N(C)C)=O)C3(C2)CC3)=O)c(F)cccc1C#N 54620,C1(CC(C)C)CN(C(=O)CC(C)(C)C)CC1NC(=O)CC1C=NN(C)C1=O 54621,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54622,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=C(Cl)CC3)C(CCO)C2)=O)ccc1F 54623,c1(OC)c(Cl)cc(C(=O)N(CC(C)(C)NC(C2CC(C)C2)=O)C)cc1Cl 54624,CCCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)NCc1ncccc1O 54625,c1(C(=O)NC(C(=O)NCC(=O)NCC)COC(C)C)ccc(C)c(C)n1 54626,C(=O)(CCC(N)C(=O)O)N1CCN(Cc2c(OC)cccc2)CC1C 54627,c1(NCc2ccn(CCC)n2)ccc2c(c1)OC(C)C(=O)N2 54628,c1(NC(=O)NCCOc2ccc(SC)cc2)cc(Br)c2c(c1)OCCO2 54629,N1(C(c2cccc(C(=O)NC)c2)=O)CCN(C(c2nc([N+](=O)[O-])n[nH]2)=O)C2CC12 54630,CC1CC(CNC(c2cc(CN(C)C)no2)=O)CN1C(=O)CCn1cncn1 54631,N1(C(CC2CC(=C)C2)=O)C(CNC(c2cc(=O)n(C)cn2)=O)CC2COCC12 54632,C1(C2CN(C(=O)CCc3nc(O)n[nH]3)C2)(NC(C2N(C)CC(O)C2)=O)CC1 54633,C(N=C(NCC1CCCO1)N1CCC2(C1)OCc1ccccc12)c1cc(C)oc1 54634,c1(CNC(c2cccc3[nH]ccc23)=O)cc(F)c(N2CCCCC2)c(F)c1 54635,C1(C(=O)NCC(CCC)O)CC2CCC1N2C(=O)C(C(C)C)NC(C)=O 54636,C1(NC(c2cnn(C3COC3)c2)=O)CC2CCC1N2C(=O)C(O)C1CC1 54637,N1C2CCc3c(cccc32)OCC1.c1(C(C(F)(F)OC)OC)sc2ccccc2c1Cl 54638,CC(O)C(F)(F)C(=O)N1CCC(C(=O)NC(CC2CCCC2)CO)CC1 54639,C1(CCC(=O)NC2C(C(=O)OC)CC2)CCCN1C(=O)CCCNC(C)=O 54640,CCS(=O)(=O)CC(=O)NCC1(NC(C2CCCCN2C)=O)CCOC1 54641,C1(NC(C(N)=O)=O)CCCC2CN(C(c3cccc(-n4cnnc4)c3)=O)CC12 54642,Cn1nccc1C1OCCC1C(=O)NC1CCCC1NC(c1sccc1CO)=O 54643,C(=O)(C(C)CNC(=O)C(Cn1cncn1)N(C1CC=CC1)C)OCC 54644,C1(C(=O)NCC(C)NC(C(=O)NCC)=O)CCC(C)(C)CC1 54645,N(C(=NCCC1CCCN(CC(=O)OC)C1)NCCc1cnccc1Cl)C(C=C)C 54646,C(CN=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)NC(c1nccc(C(C)(C)C)c1)=O 54647,c1(C(=O)NCCCn2cc(CNS(C)(=O)=O)nn2)nc(O)c2ncsc2n1 54648,C1(NC(c2cn(CC(C)C)nn2)=O)CCCCCN(C(=O)CC(C)F)C1 54649,CC1(C(N2CCC(CCNC(=O)Cc3nnc(O)s3)C2)=O)CCCC1 54650,CC1(F)CC(C(=O)NCC(c2ccccc2)NC(=O)CCNC(=O)CO)C1 54651,c1(C(=O)NCC(C)(C)CNC(c2coc3c2CSC3)=O)ccc(S(C)(=O)=O)[nH]1 54652,c1(C(=O)NC2CN(C(=O)COC3CCC3)CC2C(F)F)c(O)cccc1F 54653,C1(C(N2C(CNC(CC(C)n3cccn3)=O)CCCC2)=O)CCCCC1C 54654,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2nccc1-2 54655,C1(NC(=O)NCC2C3CCC(F)(F)C23)C2(CCC2)C12CCC2 54656,CCCCCCCCC(=O)N1CCC(CNC(=O)C(C)NC(c2cccs2)=O)C1 54657,C1(C(=O)NCCN(C(=O)CS(=O)CC)CCC)CC(OC)C(OC)C1 54658,C1(CC(=O)NCC2CC(C(C)C)C2)CCCC1NC(=O)C(c1cccnc1)O 54659,c1(C(=O)NCC(C)CN2CCCC2)cccc(N=[N+]=[N-])c1 54660,c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCC2)=O)cc2c(cn1)COCC2 54661,C(=O)(CCC1CCc2ccccc21)NCCCn1cc(C(C(C)C)O)nn1 54662,N1(C(CN(CCC#C)C)=O)CCCC(C)C1CNC(c1c(Cl)ccnc1OC)=O 54663,C(=O)(CCC(C)(C)NC(C1CCCN1C1CC1)=O)NCc1cn(C)nn1 54664,C(=O)(C(CO)C(F)(F)F)N1CCCC(C(N2C(C)CC(CO)C2)=O)CC1 54665,c1(C(N(C)CC2C(NC(CCCN(C)C)=O)CCC2)=O)cc(O)cc(F)c1 54666,C1(C(=O)Nc2cc3n(n2)CCNC3=O)CCOC2(CCNCC2)C1 54667,Cc1ncc(CNC(C2(NC(=O)CCCn3cncn3)CC2C)=O)o1 54668,N1(C(C2CCC3(CCC3)C2)=O)CCCC2(CCCN2C(=O)CC2CCCOC2)C1 54669,C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CCCN(C(=O)C(F)(F)C2CC2)C1 54670,Cc1cc(N(C2C(c3ccccc3)C2C)C(C2CCC(C)(C)C2)=O)cc(O)c1 54671,C1(CC)Cc2ccccc2CN1Cc1cccc(OC)c1 54672,n1(CC)c(C(=O)NC(C)C(=O)Nc2ccc(OCF)cc2)cnc1O 54673,C(=O)(C1(C)OC(=O)c2ccccc21)NC1Cn2c(C)ncc2CC1 54674,C#CCCCCC(=O)N(C(CC)CC(N1CCCC(CO)C1C)=O)C 54675,C(=O)(C(F)C(CC)CC)NCCCC(CCC)NC(=O)CCCCC#N 54676,c1(CC(=O)NCC(C)(CO)NC(C23CCCC2C3(F)F)=O)cccc(Cl)c1F 54677,c1(C(CNC(=O)C=Cc2ccccc2)NC(C2(C)CSC2)=O)cccc(Cl)c1 54678,Cc1c2n(c(=O)n1C)CC(N=c1cc(C(F)(F)F)c(Br)c[nH]1)CC2 54679,c1(NCc2c(N3CC(C)OCC3)cccc2)cc(OCC(F)F)ccc1F 54680,CCCCC(O)C(=O)N(C1(C(=O)NCC(c2cccnc2)O)CC1)C 54681,c1(C(N2CCC(NC(C(C)OCC=C)=O)C2)=O)ncc(Br)c(SC)n1 54682,C1(CNC(CN(C2CCC2)C)=O)CC(NC(=O)C(C)(C)C#N)CC1O 54683,O=C(CCCn1ccnn1)NC(C(=O)NC(CO)CCF)c1ccoc1 54684,N1(C(c2nc(C)n(C)n2)C(=O)NC2CCC2)CCC2CCN(C)C(=O)C2C1 54685,N(C(=NCC1CCCC12CC2)Nc1ccccc1Cl)CC(=O)NCC(C)(C)C 54686,N1(C(CCC2CCN(C(C(C)=C(C)C)=O)C2)=O)CC23CCC2(COC3)C1 54687,c1(CN(C(c2ncn(C)c2)=O)CCNC2CCC(C)O2)c(C(F)(F)F)ccc(F)c1F 54688,c1(C(C(=O)NCC(C)(CO)NC(C(C)=C2CC2)=O)C)cccc(Cl)c1 54689,N1(C(CCC#C)=O)CCC2(CC2NC(c2cc(Br)ccc2C)=O)C1 54690,N1(C(c2ccc(OC)c(C)c2)=O)CC2(CC(NC(C3CCC(F)(F)C3)=O)CO2)C1 54691,C1(NC(C2(CC#C)CCN(C(=O)CC3(CSC)CC3)C2)=O)CCCCCC1C 54692,N1(C(CCNC(COC)=O)=O)CCC(NC(C23COCC2C3)=O)C2CCC12 54693,Cc1nc2ncc(C(=O)NCCNC(=O)C(C)N3CCCC3)c(=O)n2[nH]1 54694,c1(N2CCC(CCNC(CCNC(=O)C=CCl)=O)CC2)ccn2ccnc2n1 54695,C1(C)(CNC(C(N2CCOC2=O)C)=O)CCN(C(=O)CN2CCC(CO)CC2)C1 54696,c1(C(N2CCC(O)(C(C)NC(COCCCC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 54697,CC(C)(F)C(=O)NCCCCNC(c1cc(C2CCC2)no1)=O 54698,c1(OC)cccc2c1CN(C(=NCCNS(=O)(=O)NC)NCC1CCCCC1)CC2 54699,c1(C(=O)NCCCNC(c2c(C#C)c[nH]n2)=O)cccc2c1ccn2CCOC 54700,c1(C(C)C)cc(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)on1 54701,n1(CC(=O)NC2C3CCN(C(CC4(C)CCCN4)=O)C32)nnc2ccccc2c1=O 54702,c1(NC(C2CCOC2)=O)cccc(CNC(=O)C(F)CC2CCCC2)c1 54703,Cc1nn(C)c(C)c1C(=O)NCCCNC(C1COCCCO1)=O 54704,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 54705,C1(C(=O)NC(c2ncccc2O)C)CC2CCC1N2C(C1CCN1C(C)(C)C)=O 54706,c1(-n2cc(CCNC(CN(CCOC)C)=O)nn2)ccc(N2CCC(O)C2)cc1 54707,CC1C(C(=O)O)CCCN1N(CCO)CCO 54708,Cc1cn(C(C)C)cc1C(N1CC(NC(C2(CF)CC2)=O)C(F)C1)=O 54709,Cc1ccc(Br)nc1CNC1C2CC3C(C2)C13CO 54710,n1(CC)nnnc1C(c1ccc(-c2ccco2)o1)NCCc1cccnn1 54711,c1(CC)ccc(C(=O)NC2CCC2NC(=O)C#CC2(C)CC2)cc1[N+](=O)[O-] 54712,N1(C(CNC(C2CCC2)=O)=O)CCCC(C2CN(C(=O)C3=CCOCC3)C2)C1 54713,N1(C(CC(CC)OC)=O)C(C)CN(C(C2CC3(C2)CC3(F)F)=O)CC1C 54714,N1(CC(=O)NCC23CC(NC(C4N(S(N)(=O)=O)C4)=O)(C2)C3)CCCCS1(=O)=O 54715,N1(C(c2cc(CCC)nn2C)=O)CCC(NC(=O)Nc2ccc(N)cc2)C(C)C1 54716,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 54717,C(=O)(C(C1CN(C(=O)C(C)OC(C)C)C1)ONCC1CN(C2CCCC2)C1)OC 54718,N1(CC(=O)NC2(C)CN(C(C3CCC(=O)O3)=O)C2)CCC(F)(F)C1 54719,c1(C(C(=O)NCC2(CC(=O)N(CCOCCC#C)C)CC2)F)ccccc1 54720,c1(CC2CCCC(C)N2c2cc(N)nc(-c3ccoc3)n2)csc2cccc(Cl)c12 54721,N1(C(c2ncc(OC)nc2)=O)CC2CCCC(NC(=O)CCn3ccnn3)(C2)C1 54722,c1(C(N2CCN(CC=C)C(C)C2)C(=O)NC2CCC2)ccc2c(c1)OCCO2 54723,c1(OCC(=O)N(CCCNC2CN(S(CC)(=O)=O)C2)CCO)ccccc1O 54724,CC(C)C(C(C)NC(c1csc(-c2nc[nH]n2)n1)=O)NC(=O)Cc1ccsc1 54725,N1(C(C(C)Cc2ccco2)=O)CC(C(=O)Nc2cc(F)ccc2I)CC(F)C1 54726,C(=O)(C#CC1CCOC1)NC.C1(OC(C2C(NC)COC2)COC)(OC)CCCC1 54727,C1(C)(NC(C2C(C)CC2)=O)CCN(C(=O)COCC2CCOC2)CC1 54728,N1(C(CC2(C)OCCO2)=O)CC(NC(C2CCS(=O)(=O)C2)=O)CC1CO 54729,N1(C(c2c(CC)nns2)=O)CCC(N(C(=O)C(F)C(C)C)CC2CC2)CC1 54730,Cc1nc2[nH]n(C)c(=O)c2c(C)c1CC(N1CCCC(F)(C(=O)N(C)C)C1)=O 54731,c1(OC)ccc(C(=O)N(C(C)CNC(c2csc3cncn23)=O)C)cc1C(C)C 54732,c1(C(=O)OCC(C(C)C)C(=O)OC(C)(C)C)nc2c(C(F)(F)F)cccc2s1 54733,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 54734,C1(NC(COC(C)(C)C)=O)CC2COCC(C1)N2C(=O)C(O)C1CC1 54735,C(C(=O)NCCCC1CC1)(C(C(C)C)OC)N1CCC(O)(CCCC)CC1 54736,C(=O)(C(CO)C(F)(F)F)N1CCC2(C(C(=O)NCCc3n(C)nnc3)C2)C1 54737,c1(C(C)=O)c[nH]c(C(=O)NC(c2cn(C)nn2)C(=O)N(CCCF)C)c1 54738,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 54739,C(=O)(C(CC(F)F)C1CCC1)NCC(C)NC(c1nc(OC)oc1)=O 54740,C1(NC(C(C)(C)CF)=O)CCN(c2nc3ccccc3s2)CCC1CO 54741,c1(CCOC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 54742,C(CC(C(=O)NCC1(C)CCC1)NC(=O)C=C(C)c1ccco1)OC 54743,C1(C(N(C2CCC2OC)C(=O)NC(C2CC(O)C2)=O)=O)CCCC1F.O 54744,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 54745,C1(C(N2CC(NC(C(C)C(C)(C)C)=O)C(N(C)C)C2)=O)CC2(C1)CC1(CC1)C2 54746,Cc1c(C(N2CCC3CN(C(=O)CC(C)C(C)C)CC23)=O)ccc2cncn12 54747,c1(CCC(=O)NC(C(=O)NC(c2ccn(C)n2)CC)C2CCCC2)cn(CC)nn1 54748,C1(CNC(c2c(C)oc(Cl)n2)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 54749,C1(NC(C(C)=C2CC2)=O)CC(C)CN(C(C23CCC(CC2)C3)=O)C1 54750,c1(CNC(c2ccc(F)c(O)c2)=O)cnn2c1CN(Cc1cnc[nH]1)CC2 54751,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(C)C)=O)C2)=O)ncn1C 54752,c1(C(=O)NC2C(C(N(CC#CC)C)=O)CC2)cnc(CC)nc1 54753,c12ccc(cc1)OC2CC.N1(C(C(C2(COC)CC2)N)=O)CCSC2CC12.OC 54754,C(=O)(C(C)(C)n1cc(Br)cn1)NCCCNC(C(C)n1cncn1)=O 54755,C1(C(F)(F)F)(C(=O)NC2(C)CCN(C(CC(C=C)(C)C)=O)C2)OC2CCC1CC2 54756,N1(C(c2cccc(C)c2)C(=O)NCCCSCC)CCc2cc(C)sc2C1 54757,Cc1ccccc1C(C)C(=O)NCC1CCN1C(=O)CCN1CCC(O)CC1 54758,Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NCC1CCN(C(=O)CCC#N)C12CC2 54759,C=CCC(C)(C)CNC(=O)C(=O)NCC1CCOC1C 54760,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C(C)C)c1Cl 54761,C(c1nnc(C(C)C)o1)=CC(N1CC(NC(c2c(COC)cco2)=O)(CO)C1)=O 54762,Cc1cc(N2CCC3CN(C(=O)C(C(C)C)NS(N)(=O)=O)CC23)ncc1[N+](=O)[O-] 54763,Cc1cc(Cl)cc(Cl)c1OCCNC(=O)C(=O)NCc1ccnc(Br)c1O 54764,C1(C(N2CCC=C(CNC(COC(C)C)=O)C2)=O)CCCCCS1(=O)=O 54765,c12ncc(cc1Cl)S(=O)(=O)N2.CCC(CC)CCCN1CCCC(C(N)=O)CC1 54766,N1(C(C2OCC2(C)C)C(=O)NCC)CCC(C(=O)OC)C12CCC2 54767,c1(CNC2CCCC(NC(c3c(CC)cccc3)=O)C2)cc(Br)cnc1C 54768,N1(C(CCCCC)=O)CC(CNC(C2(c3ccccc3)CCOC2)=O)CC12CCC2 54769,Cc1cc(C(=O)NCCOC2CN(C(=O)CCCC(C)O)C2)c2ncccc2c1 54770,C1(C(=O)NC(C)C(C)(C)C)CCC2(CC2)N1C(c1ccc(Cl)s1)=O 54771,CCC(CC)C(F)C(=O)N1CCCC1CC(=O)N(C1CN(C(C)=O)C1)C 54772,CCCC(C(=O)N1CC(C)(NC(C2CC2c2n[nH]cc2Br)=O)C1)N(C)C 54773,c1(CNC(=O)CC2CCCN2C)cn2c(n1)COCC2.C12(CC=C)CN1C2 54774,c1(N2C3CN(C(C4(C(=O)OCC)CC4)=O)CCC2CC3)nc(Cl)nc2[nH]c(O)nc12 54775,N1(C(CCCNC(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)Cc2cncs2)C1 54776,c1(C(=O)NCCCN(C)C(C2CCC(O)CN2C)=O)ccc2c(c1)OCCN2 54777,C1(CNC(CC=CCC)=O)CC(C(C)C)CCN1C(=O)CCOCC 54778,CN1CC2CCN(C(=O)COC(C3(C4CC(=O)N(C)C4)CCC3)=O)CC2C1 54779,CC1(NC(=O)CSCC2CCC2)CC(NC(=O)Cc2csc(-n3cnnc3)n2)C1 54780,N1(C(CN(C(COC)=O)C)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 54781,N1(C(CC(CNC(=O)CSC(F)F)OC)=O)CC2(CNC(=O)C2)C1 54782,c1(SC)cccc(C(=O)COC(c2nc(C3C4COCC34)cs2)=O)c1 54783,C1(OC)CCCCC1C(N1CCN(CCNC(=O)C(C)(C)C2CCCO2)CC1)=O 54784,CC1CCCC(C(=O)NCC2C3CC2N(C(C2CNC(=O)N2)=O)C3)C1 54785,CCCC(C(O)C(=O)Nc1ccc2c[nH]nc2c1)NC(=O)C(F)C1CCC1 54786,c1(C(=O)Sc2ccc(Cl)cc2)cc(CC(Cc2ccccc2)CO)cc([N+](=O)[O-])c1 54787,Cc1ccc([N+](=O)[O-])cc1N1CCN(C23CC2CCN3)CC1 54788,Cc1cccc2ncc(-c3noc(C4COCC4F)n3)n12 54789,C1(C(=O)NC)CCC(N(C)C)C1.C(F)(C(=O)N1CC(C2C(=O)N2)C1)=CC 54790,c1(C(N(C2CCC(NC(=O)Cn3cnnc3)C2)C)=O)ccnc(Cl)c1N 54791,Nc1ccc(CC(=O)NC(CNC(C2CC2C(F)(F)F)=O)CC(F)(F)F)cc1F 54792,C(=O)(CCC(C)(C)C#N)N1C(C(C)NC(c2cnc(SC)s2)=O)CCCC1 54793,C1(C(=O)NCC(C(C)C)NC(C2CCC(C)(O)CC2)=O)CCCCCCC1 54794,c1(CCC(=O)NCC(C)NC(CCSC)=O)cccc(F)c1.C12CC1C2 54795,C12(CNC(C3(C)CC=CCC3)=O)CCC(CNC(C3CC(F)(F)C3)=O)(CC1)CO2 54796,N1(C(CCN(C)CC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(OC)cc1 54797,C1(C(=O)NCC(C)CNC(=O)C(C)(C(F)F)c2ccccc2)CN2CCN1CC2 54798,CN1CCCC1CCC(=O)NCC1(CF)CCNC1 54799,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 54800,N1(C(C(C)OCC2CC2)=O)CCC(F)(CNC(=O)C(=Cc2cccnc2)F)C1 54801,N1(C(C(C)OCCC=C)=O)CC(NC(c2occ(C)c2C)=O)C(C(F)(F)F)C1 54802,CCCCCOCC(=O)NCC1(N(C(=O)CCc2nncs2)C2CC2)CC1 54803,c1(C2CCC(C(=O)NCCNC(=O)C=Cc3cnc[nH]3)C2)cccc(Br)c1 54804,C1(C(N(CCC#C)CCO)=O)CN(C(C2CCC2)=O)CCO1 54805,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(=O)CCC2CCCC(O)C2)C1 54806,c1(OC)c(C(=O)NC2CC2C(=O)Nc2ccc(Cl)c(C)n2)cc(Cl)cc1Cl 54807,Cc1nncn1CCNC(C1OCCC1CNC(=O)C=CCF)=O 54808,c1(OC)ccc(CN(C(=O)C(=O)Nc2csnc2C2CC2)C)c(C(F)(F)F)c1 54809,C(=O)(CC(=O)NC1(C(=O)NC2CC(=CC)C2)COC1)NCC#C 54810,C1(C(N2CC(CCCCC)C2)=O)N(C(=O)CCCCC(C)C)CCCC1(C)C 54811,CCC(C)(CO)C(=O)NCC(C1CCN(C(=O)CSCC(N)=O)CC1)(C)O 54812,C1(F)(C(=O)NC2(C(=O)NCCC3(CC)CCCC3)CSC2)CCOC1C 54813,N1(C(C=C(C)C(C)C)=O)CCCCC(CNC(C23CCCC2OCC3)=O)C1 54814,C12(CNC(C(CC)OC)=O)CCC(CC1)N2C(=O)C(c1cccs1)SC 54815,CCCC(C)(O)CC(=O)NC1CCCC1(C)NC(C1COCC1(C)C)=O 54816,c1(CC(C(=O)OC)NC(C2OCC3CCCC2C3)=O)c(F)c(F)c(F)c(F)c1F 54817,Nc1c(F)cc(C(N2CC3CC2C3NC(c2csc(C(F)F)c2)=O)=O)c(F)c1F 54818,C#CCCCC(=O)NCC1CSCCN1C(=O)COC(C)(C)CC 54819,CC1C(O)CCCN1C(C1CCC1NC(c1ccc(=O)ncc1)=O)=O 54820,c1(C(N2CCC(NC(C3C(=O)NCC3)=O)C2)=O)cc2cccc(Br)c2s1 54821,c1(N(C2CNCC(C)C2)C(C2CN(C(C)C)C(=O)C2)=O)ccn2ncc(Br)c2n1 54822,C12(N(C)C)CCC(C(=O)Nc3ccc(OC(F)(F)C(F)F)cc3)(C1)OC2 54823,S(=O)(=O)(CC(C)C#N)N1CC(OC)OCC1 54824,c1(C(=O)NCCCN(C(C(CC)OC2CCC2)=O)C2COC2)cccc(OC)c1 54825,N1(C(C2N(C(c3ccc(NC(C)(C)C)nc3)=O)CC2)=O)CCC(C(=O)O)C1(C)C 54826,c1(-c2cn(C(C)CNC(=O)CNC(N)=O)nn2)cccc(-c2cnco2)c1 54827,C1(C(N2CC(CC)(NC(C3CCN4CCCC4C3)=O)C2)=O)CCc2cnnn2C1 54828,CCC(C)(F)C(=O)N1CCCC(NC(=O)NC2CCCC2)C1 54829,N1(C(c2cn(C)nn2)=O)C2CCC1CN(C(C1CCC3CC1C3(C)C)=O)C2 54830,C(=O)(CC(CC)C1CCC1)N(CCCC(=O)NCc1noc(CC)n1)CC=C 54831,O=S(=O)(c1ccc(-n2cc(-c3cccc(F)c3Cl)nn2)cc1)C(F)(F)F 54832,CCCCC(C(=O)N1CC2CC1CN2C(C1(CO)CCC1)=O)N1CCCS1(=O)=O 54833,CCCCCCCCC(=O)NC1CCC(CCC(=O)NC(C)COCCOC)C1 54834,C(=O)(C1=NOC2COCC12)NCC(CNC(c1cn(CCN(C)C)nn1)=O)CO 54835,O=C1Oc2ccc(S(=O)(=O)N3CCC(O)(c4ccccc4Br)C3)cc2CO1 54836,c1(CC2C(C(=O)NC(CCCNC(CCCCC)=O)C)C2)cccc(F)c1F 54837,n1(-c2c(C)cccc2)nc(NC(N2CCCc3[nH]ccc32)=O)c2c1CCCC2 54838,C1(c2cn(C(C)CNC(C3CC4(N)CC3C4)=O)nn2)(N(C)CCO)CCCCC1 54839,CCCC(CNC(=O)CCNC(=O)CO)C(=O)NCCN1CC=C(C)CC1 54840,C1(C(=O)NCC2(O)CN(C(C3CC=CCO3)=O)C2)CC2(CCCCC2)S1(=O)=O 54841,c1(C(=O)NC23CC(CNC(COCC(C)(C)C)=O)(C2)C3)ccc(N)c(Cl)c1O 54842,C1(NC(=O)Cc2csc(O)n2)CCN(C(C2(Nc3ccccc3)CC2)=O)CC1O 54843,C#CC1(C(=O)NCC2CCC(F)(F)C2)CN(C(C2CC(C)CO2)=O)C1 54844,c1(C(=O)OCC)ccc(C(=O)NCC2CCC(NC(=O)CC3CC3(C)C)C2)nn1 54845,c1(C(=O)NC(CNC(c2onc(C)c2C)=O)C2CCC2)cc2c(nc1N)CCC2 54846,N1(C(COC)=O)CC2CCCC(C1)N2C(=O)Cc1ccnnc1O 54847,c1(CN2CCN(CCC(=O)NC3CN(C)C3)CC2)c[nH]c2cccc(F)c12 54848,N1(C(C(C2CCN(C(COCC)=O)C2)F)=O)CCC12CC(CCO)C2 54849,c1(C(C)C(=O)N(CCn2cc(CO)nn2)CCF)ccc([N+](=O)[O-])cc1 54850,CCC(F)(F)C(C)(C)C(=O)N1CCC2=C(CCCC2)C1.C(CCCCCO)n1ccnn1 54851,C(=O)(CCS(C)(=O)=O)NC1C(CNC(c2ccc(CC)[nH]2)=O)CCCC1 54852,c1(C(N(CC(C)NC(C2CCS2(=O)=O)=O)C)=O)ccn2c(C(F)(F)F)nnc2c1 54853,CC1CCN(C(C23CCC(O)(CC2)CC3)=O)C(C)C1NC(=O)Cn1cnnc1O 54854,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 54855,CC(C)CCN=C(NCC1(C2CCCO2)CCCO1)NC(c1cccc(Br)c1)C 54856,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 54857,N1(C(CCCOCC)=O)CC(C)N(C(c2cc3ccncc3[nH]2)=O)CC1C 54858,O=C(C1=CCCCC1)NC1CCCC1C(=O)NC1C=CCC(CO)C1 54859,C1(NC(COCCNC(CCc2cc(C)no2)=O)=O)CNC(=O)C1(C)C 54860,CC(C(=O)N(CCCC(=O)N(C)Cc1ccsc1)C)C(F)F 54861,C1(CNC(C(CN(C)C)NC(=O)N(C)Cc2ccccc2)=O)CCCC1(C)C 54862,N1(C(CCC)C)CCC2(CC1)CC2C(=O)NCc1ccc(N)cc1 54863,c1(C(=O)NCC(CNC(C2(C)CCNC2=O)=O)O)ccc(Cl)nc1N 54864,C1(C(N(C(CCC)C(=O)OC)C)=O)CCCN(c2nncs2)CC1 54865,N1(Cc2nnn(C)n2)CC=C(CNC(C2CCCCN2N=O)=O)CC1 54866,CC1(CCNC(C2C3(CC3)C23CC3)=O)CCN(C(=O)CC2CCCC2)CC1 54867,c1(COC)c(S(=O)(=O)Nc2nc3c(n2C)CCCC3)n[nH]c1C 54868,c1(CCC(=O)NCCSc2c(C)cccc2)nc2ccccc2c(=O)n1C 54869,C(=O)(C(O)C(C)(C)CC)NCCCN(CCCNC(C1C(OC)CC1)=O)C 54870,N1(C(c2c(C)n3c(s2)ncc3)=O)CCN(C(=O)Cc2cn[nH]c2)CC12CCC2 54871,c1(CC)nc(C(N2CCC(CC(C)NC(=O)C(F)C(C)C)CC2)=O)c(N)s1 54872,C(=O)(C(CO)C(C)(C)C)N1CCN(C(c2cc(SC)oc2)=O)CC1CC(F)F 54873,Nc1cc(F)cnc1C(=O)NCC(CC(=O)N1CCC(OCCF)C1)OC 54874,c1(OCCCCNOC(C)(C)C)cccc(CO)c1.C(=O)(C1CC1)CCC 54875,c1(OC)cc(NC(C2CC2NC(c2n[nH]cc2Cl)=O)=O)cc(Cl)n1 54876,c1(CC)onc(C)c1C(N1CC(C(N)=O)(CNC(=O)CN2CCCCC2=O)C1)=O 54877,c1(C(=O)NCC(C)(C2CCC2)NC(C(C)NC(CC)=O)=O)cc([N+](=O)[O-])c(C)s1 54878,Cc1cc(C)c(C(=O)NC2CCNC2C2CC2)cn1 54879,CCCC(CNC(C1CC(C)N(C)C1)=O)C(=O)Nc1ccccc1Cl 54880,Cc1nc(C)n(CC(=O)NCCN(CC(C)O)C(=O)Cc2sc(=N)[nH]c2C)n1 54881,c1(C(N2CC3C(NC(c4c(C(C)C)c[nH]n4)=O)C3C2)=O)cnc2ccncc2c1 54882,N1(C(CCNC(C)=O)=O)CCC(C#N)(c2ccc(C)o2)CC1 54883,c1(C(=O)N(C2CCC3(CC2)CC3)CC(O)Cc2ccccc2)cc2cnccc2o1 54884,CC1(C)CN(C(=O)NC(c2ccccc2[N+](=O)[O-])C#N)c2cc(C(N)=O)ccc2O1 54885,CC(C)CC(C(=O)NC1CCN(C(=O)COc2cncc(Cl)n2)CC1C)C(C)C 54886,N1(C(c2n(CC)cnn2)=O)CC=CC(NC(=O)CN2CCCC2CO)C1 54887,c1(C(N2CC(OC)(CNC(c3ccc(N)cc3O)=O)C2)=O)ccnc2ccsc12 54888,C1(CC)C(NC(c2ccc(=O)n(C)n2)=O)CCCN1C(c1ccn(C)c1C)=O 54889,C1(CCC(=O)N(C2(C)CN(C(c3c[nH]nc3-c3cnn(C)c3)=O)C2)C)CNC(=O)N1 54890,c1(CC(=O)NCCCC(C)NC(C2(F)CCCOC2)=O)cnc2ncccn12 54891,C1(COc2nc(-c3c(C)onc3)n(C3CCOC3)n2)C2CC3CC(C2)CC1C3 54892,C1(F)(CNC(C2(C)CC=CCO2)=O)CC2CCC(C1)N2C(c1cnc[nH]1)=O 54893,CCC(C)CC(=O)C(=O)N1CCCC(C(=O)NC2(CSC)CCC2)C1 54894,C(C1CCOC1)=CC(=O)NCCN(C1CCCCC1)C(C1CC(OC)C1)=O 54895,c1(C(=O)NC2(CNC(C(CC=C)(F)F)=O)CCOC2)ccc2occc2n1 54896,C(c1csc(Br)c1)=CC(=O)NC(C1CN(C(CC(=O)OCC)=O)C1)C 54897,C(=O)(C1=C(C)OCC[SH]1C1CC1)N1CCC(NCC)C1 54898,c1(OC)ccc2ccnc(CN3CCCC3C(=O)Nc3cc(F)cnc3Br)c2c1 54899,C1(C(=O)N(CCCN2CCOCC2)C2CC2)CCN(c2ncncc2F)CC1 54900,N1(C(C2CCC(=O)N2)=O)CCCCC1CN(C(=O)COc1ccccc1F)CO 54901,CC1=C(C(=O)NCC2CN(C(C3CC4C=CC3O4)=O)CC2O)CCCO1 54902,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 54903,c1(C(C)C)c(Cl)cc(NC(C2CC(c3nccn3C)C2)=O)cc1Cl 54904,C1(C)(CNC(CC2CC(OC)C2(C)C)=O)CCN(C(=O)CN2CCN(C)CC2)CC1 54905,N1(C(c2c(C)noc2C)=O)CC2CCCC2(NC(c2cccc3ccnn23)=O)C1 54906,CC(O)(C(=O)NCC(=O)NCCOCCCCCc1ccccc1)c1cccs1 54907,C1(NC(C2C(C)(C)CN(C(C3CCCCO3)=O)C2)=O)CCOC12CCCC2 54908,C1(NC(=O)CSC2OCCC2C(F)(F)F)CCN(C(C2CCCCC2)=O)C12CC2 54909,N1(C(C(CC)C)=O)CC(O)(C2(CNC(C3CCC(N(C)C)C3)=O)CC2)C1 54910,C(=O)(CCCCCF)N1CCC(NC(c2c(C)cc(CC)o2)=O)(COC)C1 54911,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2CCC2)C1 54912,C1(NC(C=CCOC)=O)(CNC(=O)C(C)COC)CCOC1 54913,N1(C(CC=C=C)=O)CCCCC(CNC(C2CCCO2)=O)C1 54914,C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C12CCC2 54915,C=CC1(CC(N2CCN(CCn3cc(CC(O)C4CC4)nn3)CC2)=O)CCCCC1 54916,C12(C(N(CC)Cc3cnc(C)cn3)=O)CCC(NC34CC(F)(C3)C4)(CC1)C2 54917,c1(CCC(N2CC(OCC(=O)NCCCC(C)N(C)C)C2)=O)ccc(Cl)c(F)c1 54918,c1(C(=O)NC(C(=O)NCC2(CC)CCC2)CSCC)cnc(C)[nH]c1=N 54919,C=CCC(C(=O)N(CC(=O)NCC1(C(N)=O)CC1)C)NC(C)=O 54920,C(=O)(CC(CN(C)C)C(F)F)N1CCN(C(Cn2ncc(C#C)c2)=O)C(C)C1 54921,c1(C(=O)NCC=CCC(N2CCCC(COC)C2)=O)cc(C)ccc1O 54922,c1(N2CCC(N(CC)C)CC2)nc(=NC(CCO)C(F)F)[nH]c2ccc(Cl)cc12 54923,C(C1OCCc2ccccc21)n1c(C(C)CC(C)C)nc(C(CC)CC)n1 54924,Cc1nn(C)c(Cl)c1C=CC(N1CC2CC2(NC(C2CC3CCC(C2)O3)=O)C1)=O 54925,c1(C(C(C2CCN(C(=O)C3=COCCC3)CC2)C)=O)cc(Br)cc(F)c1C#N 54926,Cc1nc(Cl)ccc1CC(=O)NC(C)C(C)(C)NC(=O)Cc1ncoc1C 54927,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CCC(CNC(CC(C(F)(F)F)OC)=O)C1 54928,c1(NC(CC2OCCN(C(C(C)OCCOC)=O)C2)=O)ccc(Br)cc1C#N 54929,S(=O)(=O)(C(F)F)N1CC(C(=O)NC2CC(NC(C3CC(N(C)C)C3)=O)C2)C1 54930,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 54931,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NCC(CC)C(C)C 54932,N1(C(CC2N(Cc3ccc(OC)cc3F)CCOC2)=O)C2COCC1CC(F)C2 54933,c1(C(=O)NCCCN(C(C2CC(CCC)OCC2)=O)CC)cn(C)c(=O)nc1O 54934,C1(NC(c2cccc(NC(C)=O)c2)=O)CN(C(=O)C(F)CCC(C)C)CC(F)(F)C1 54935,c1(C(C2CC2)NC(C2(n3cc(C4CC4)nn3)CCOCC2)=O)cccc(F)n1 54936,CCCCC(=O)C(=O)NC(CCCNC(=O)C=CS(C)=O)c1ccccc1 54937,CCC(C(=O)N1CCCC1N(C(=O)C=CI)CC)C(C)C 54938,c1(C(CN(C(c2c(C)sc(CN)n2)=O)C)C(=O)O)ccc(S(C)(=O)=O)cc1 54939,N1(C(C(C2CCCCC2)OC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 54940,c1(C(CNC(=O)CCC2CC2(F)F)(F)F)ccc(Cl)cc1Cl 54941,c1(-c2c(C)nc(Cl)cc2)c(C(=O)NCc2c(C)c(Cl)ccc2)nn2c1CCCC2 54942,CC(C)CC(C)CC(=O)N1CCC(F)(C(=O)N(C)CC2(O)CCOC2)C1 54943,S1(=O)(=O)c2c(C)nn(c2C)CCC2CCCN12.n1(CCCCC)ccccc1=S 54944,C1(COC)CN(C(c2cn(CC(N)=O)nn2)=O)CCN1C(=O)CN1CCOCC1 54945,c1(COC)cncc(C(=O)NC2CCN(C(=O)C(C(C)C)N3CCCC3)CC2)c1 54946,N1(CC(=O)N(CC#C)C)CC2(CC2C(=O)OC(C)(C)C)C1.C1(F)(C=O)CCCN1 54947,C1(C(N2CC(C[Si](C)(C)C)C2)=O)C2CN(C(C3CCC4(CC4)C3)=O)CC12 54948,N1(C(C(C)CF)=O)CCCC(CO)(CNC(=O)C=C(Cl)Cl)C1 54949,C1(NC(C2C(OC)CC2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1(C)C 54950,C(CC1=CCN(c2cc(NC(=O)C3CC3)ncn2)CC1)NCC(N1CCCC1)=O 54951,N1(C(C(C)(C)c2ccccc2)=O)CCC(C)(O)C(O)C1.C12CCCN(C1)C2=O 54952,c1(C(=O)OC)c[nH]ccc1=NCC12CCC(NC(C3CC(=O)N3)=O)(CC1)CO2 54953,N1(C(c2c(C)cc(C)o2)=O)CCC2(COC(CNC(c3cc(C)c(C)o3)=O)C2)C1 54954,CCCCC(O)CC(=O)NC(COC(C)C)CF 54955,CC1CN(C(C2COCCN2C=O)=O)CCCN1C(=O)CS(N)(=O)=O 54956,N1(C(C2(COC)CN(C(C3CC4COCC4C3)=O)C2)=O)CCc2nnnn2CC1 54957,C1(C2CN(C(=O)COC(F)F)C2)(NC(=O)COc2ccc(Br)cn2)CC1 54958,c1(C(=O)NC(CCNC(C(CC2CC2)OC)=O)(C)C)ccc(CO)cn1 54959,C=C(F)CN=c1cc(NCc2cc(Cl)n(C)n2)nc(C(F)(F)F)[nH]1 54960,C(=O)(CC(C)F)N(CCC)CCNC(C1CC(CCO)C1)=O 54961,c1(CC)ccoc1C(=O)NC1CC(NC(C2COCC2OC)=O)C1 54962,C1(F)(CNC(C(CC#C)C)=O)CCC(CNC(=O)CC(O)CN(C)C)CC1 54963,Nc1nc2ncccc2cc1C(=O)NCCCCNC(C1CCC12CCCO2)=O 54964,C1(CNC(c2c(C)onc2CO)=O)CC2CCC(C1)N2C(=O)CC#N 54965,Cc1ccc(C)c(C(=O)NCC2(F)CCC(NC(=O)CCN3CCCC3)C2)c1 54966,c1(CN2CCC(C(C(=O)Nc3nc(C)c(F)cc3)C)CC2)cccc2cccnc12 54967,c1(C(=O)Nc2scc(CC(=O)Nc3ccc(C#N)nc3)n2)ccc(Cl)c([N+](=O)[O-])c1 54968,S(=O)(=O)(c1ccc(N2CCCC(S(C)(=O)=O)CC2)c(Cl)c1)NCCC(=O)NC(C)C 54969,Cc1cc(C(N2CCOC(C(C)NC(c3ccncn3)=O)C2)=O)ncn1 54970,c1(COC(CC)C)cccnc1CNC(=O)Cn1cnc(=N)[nH]1 54971,C1(NC(c2ccc(C(C)C)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 54972,N1(CC(=O)NC2CCC(CC(=O)N(CC)Cc3nnnn3C)C2)CCCNC1=O 54973,Cc1cnc(O)n1-c1cccc(CN2CCC(n3cc(CO)nn3)C2)c1 54974,c1(C(=O)N(CC)CC)ccc(-c2cc(-c3nccn3-c3ccn(C)n3)co2)cc1 54975,CC(CN1CCCC1)N=c1cc[nH]cc1S(=O)(=O)N1CCN2C(=O)COCC2C1 54976,c1(CC)nc(NNC(=O)C2(O)CNC2)c(C#N)s1 54977,C(=O)(C1CCc2nccn21)NC1CN(C(C(CO)NC(C)=O)=O)CC1C 54978,C1(C(=O)NCC(C)N(C)Cc2cccnc2Br)CC2CCC1CC2 54979,c1(C(N(C)CCOCCNC(C2CCCC(C#N)C2)=O)=O)cnc2ccccn12 54980,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 54981,C(=O)(CCCCC(C)C)N1C(C(=O)NCc2ccc(C)s2)CC(C)(C)C1 54982,C(=O)(CC1CCc2ccccc21)N1CC(C)(NC(C2CCC(CN(C)C)O2)=O)C1 54983,C12(NC(C3CCC(C)N3C(=O)COC3CCC3)=O)CC=CC(C1)OC2 54984,N1(C2CCC(NC(C(C)n3cncn3)=O)C2)CCN(C(=O)C2=CCSC2)CC1 54985,Cc1ccc(CC(=O)NCCC(C)NC(=O)CC2CC(C3CC3)C2)cc1Cl 54986,c1(CCC(=O)NCCC2CN(C(=O)CCSc3ccsc3)C2)ncc(F)cn1 54987,c1(-c2ccc(F)c(C)c2C)cnc2cc(C(N3CCCCC3C(N)=O)=O)ccn12 54988,Cc1ccn2cnc(C(=O)NC3CN(C(c4oncc4C)=O)C4(CCC4)C3)c2c1 54989,C1(CNC(C2CC(NC(C(C)n3cncn3)=O)C2)=O)CCOCC1(C)C 54990,C(CCC(=O)NNC(=O)OCC1CCC(=O)NC1)CCN(C)C 54991,C1(N(C(C2CCCN(C(c3c(CC)cno3)=O)C2)=O)C)CCCC(C)C1C 54992,C12(CNC(c3ncn(C)n3)=O)CCC(NC(C3CC4CC4C3)=O)(CO1)C2 54993,C=C=C(C)CC(=O)N(CC(C)O)CCNC(=O)C(CC)NC(=O)OC 54994,C1(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)(C(F)F)CCCCC1 54995,c1(CNC(CN(CCS(C)(=O)=O)C(C#C)C)=O)cc(C(C)C)no1 54996,c1(CNc2c(CC(=O)Nc3ncc(C)c(F)c3)cccc2)ccc(F)c(C)c1Cl 54997,c1(NC(C(C)O)C(=O)O)ccc(S(=O)(=O)NCC2CCCO2)cc1 54998,c1(C(=O)NCC2C(C(=O)NCC(C)OCCO)CCC2)c[nH]c2ccncc12 54999,c1(C(N(CCN(C)C(c2ncoc2-c2cccs2)=O)C)=O)snc2ccccc12 55000,c1(C(=O)NCC2C(NC(C3C(CCC)C3)=O)CC2)ccc(CC)cn1 55001,C1(C(N(C(C)C2CC2)C)=O)C2CC1N(C(=O)C=Cc1ccncc1)C2 55002,CCC1=C(C(=O)NC2CN(C(c3cc(S(C)(=O)=O)co3)=O)CC23CC3)CCCO1 55003,c1(OC)cccc2ccc(NC(=O)CC3CCCN3CC(C)C)nc12 55004,S(=O)(=O)(c1ccc(C(C)=O)cc1)N1CC2(C3(OC)CC(CN)(C3)O2)C1 55005,C(=O)(C(F)C(C)CC(C)(C)C)N(C(=O)C(=O)N=S(C)(C)=O)C1CCCC(C)C1 55006,S(=O)(=O)(c1ccc(N2CCCCC2)c(Br)c1)NCc1ccc(OCOC)c(F)c1 55007,c1(CNC(C2(C#N)CC(C)C2)=O)cnn2c1CN(C(C1CCCC1C)=O)CC2 55008,C=CC1CN(C(=O)CCCC2CC2)CC1NC(=O)C=C1CCC(C)C1 55009,c1(CNC(C)CCc2cc(F)ccc2F)ncnc2cc(Br)ccc12 55010,Cc1nc(NC2(C3CCC3)CC2)cc(=NCCOc2ccncc2)[nH]1 55011,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55012,C=CC1(CNC(=O)CCOC)CCN(C(C2CCOC2C(C)C)=O)CC1 55013,c1(C(N2CC3(C(C(=O)Nc4cc(F)ccc4I)C3)C2)=O)cc2sccc2[nH]1 55014,c1(C(=O)NCC(CN(C)C(c2cc(C(F)F)cs2)=O)(C)C)cccc(F)c1Cl 55015,C(=O)(C(CC)C(F)(F)F)N1C(CC)C(C(=O)N(C(C)COC)C)CCC1 55016,C(=O)(C(C)(C)Cc1cn(CC(=O)NC(C)C)nn1)NCc1ncc(CC)o1 55017,N1(C(C(C)=CO)=O)CCC2CCC12CNC(c1cn(Cc2ccccc2)nn1)=O 55018,N1(C(C)CCO)CCC2(CC1)CC2(C)C(=O)NC1CCOC(CO)C1 55019,c1(SC)c(C(=O)NCC(C)CN(C)C(c2ncccn2)C)cnn1C 55020,c1(COC(c2cc(C3CCC3)no2)=O)coc2ccccc12 55021,c1(C(=O)NCC(CC(C)C)NC(C2(C)CCC(=O)N2)=O)cc2c[nH]cnc-2n1 55022,c1(OC)nc(C(N2CC3(CC(NC(C4CNC(=O)N4)=O)C3)C2)=O)ncc1F 55023,CN1CCC(C)(C(=O)NCC2(C)CCN(C(c3ccccc3)=O)C2)C1 55024,C1(C(=O)NC2(CNC(=O)Cc3nc[nH]n3)CCCCC2)CC2CCC(C1)O2 55025,c1(C(=O)NC23CC(CNC(C(C)(C)O)=O)(C2)C3)cc(O)c2ccccc2c1 55026,C(=O)(CCS(=O)(=O)Cc1ccccn1)NC1CN(C(CC2C(C)CCO2)=O)C1 55027,CN1CCN(C(=O)Cc2csnn2)CC1C(=O)NCCOc1ccon1 55028,N1(C(CC2(OC)CCCCC2)=O)CCC2C(O)C(C)(C)C12.C1(C)C(=O)N1 55029,C(=O)(C#CC1CCCC1)NC(C)CCCCO.C12C(C1(C)C)C(=O)N2 55030,C(=O)(C(C(C)CC1CCC1)N(C)C)NC1CCN(CCOC)CC1 55031,c1(C(N(CC(CNC(C2C(C)OCC2)=O)O)C)=O)ccc(N(C)C)cc1F 55032,c1(C(N(C2CCC(NC(=O)C#CC3CCCO3)CC2)C)=O)cccc2ccnn12 55033,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55034,C#Cc1nc(C(=O)N(CC(N2CCN(C(=O)CCCC)CC2)=O)C(C)C)cs1 55035,N1(C(c2c(N)ncc(C)c2)=O)CCC2(C1)CN(C(=O)C(C)Sc1ccccc1)C2 55036,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(C)(CN(C)C)C1)CC(C)C 55037,CC1(C)C(CNC(=O)Cc2cscn2)CCN1C(=O)CSCC1CCSC1 55038,CCC(CC)C(C(=O)NC1(C(N2CC([N+](=O)[O-])C2)=O)CCCC1)OC 55039,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)c(Cl)c2)=O)C1 55040,Cc1cc(-n2nc(CCN(C)C)nc2Cc2ccc(Br)cc2F)cc(C)c1 55041,C#CC#CC(C)(C)NC(=O)C(C)(CO)NC(C1CC2CCC2C1)=O 55042,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55043,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55044,C(=O)(CC(C)(C)CCC)N(C(C(=O)NC(CCC=C)(C)C)C)CC 55045,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55046,C#CC(CNC(=O)C(CNC(C1(Cl)CC1)=O)CCC)CC(C)(C)C 55047,n1(CC)nc(C(=O)N(C)CCOCCNC(C2CCCOC2)=O)cc1C 55048,C(=O)(C(C(C)C)NCC(C)C)NCCNC(CNC(C1C(OC)CC1)=O)(C)C 55049,c1(C(C)(C)C(=O)OCC(c2ncccc2Br)=O)ccc(C(F)F)cc1 55050,N1(C(C2CCCN(C(C(C)C)CO)CC2)=O)C2CCCC1CN(C)C2 55051,CC(C)CC(N)C(=O)Nc1ccnc(SCC(F)(F)F)c1 55052,C1(C(=O)NCC23CN(C2)C3)CC2(C1)CC(F)C2.C1(C)(C(=O)OC)CC1C(N)=O 55053,Cc1c(N2CCCN(S(C)(=O)=O)CC2)nc(Cl)nc1N1CCN(C2(NC)CC2)CC1 55054,c1(CCNC(c2cc(-c3ccco3)nn2CC(F)(F)F)=O)ccc2cc[nH]c2c1 55055,Cc1nccc(Cl)c1C(=O)NCCN1CCCN(C(=O)CC2CCCC(F)C2)CC1 55056,C12(C(N(C)CCNC(=O)C(c3ccc(O)cc3)=O)=O)CC3CC1C2C3 55057,CC1(CNC(c2cnc(C(F)(F)F)s2)=O)CCCN1C(C1CC2CC2C1)=O 55058,C#CCC(CC#C)C(=O)NC(CNC(=O)Cc1csc2nc(C)cn12)(CC)CC 55059,C1(NC(CC2(CC)CCC2)=O)CC=C(C(=O)NCC2(C3(O)CCC3)CC2)C1 55060,CC#CCCC(=O)N(CCNC(c1cncnc1-c1ccccc1)=O)C1CC1 55061,c1(C(=O)NC2CC3C(NC(c4nccc(C)c4)=O)C3C2)cnc(C)c(C)c1 55062,N1(C(C2(C)CNC(=O)C2)=O)CCC(C2CCN(C(=O)CC=C(Cl)Cl)C2)C1 55063,C1(NC(=O)CCN(C(c2scnc2Cl)=O)CC2CC2)CN2CCC1CC2 55064,N1(C(CCC=CC)=O)CCC(C)(NC(=O)C(C)CC2CCCCC2)C1 55065,n1(CCOC)ccnc(C(=O)NC2(C)CCN(C(=O)CC3CS(=O)(=O)C3)C2)c1=O 55066,C(CCCC(CO)NC(C1(SC2CC2)CC1)=O)NC(C(CC)OCC(F)(F)F)=O 55067,C1(C(=O)NCC(C2N(C(c3n(C)ccc3)=O)CCCC2)F)(CF)CC2(CCC2)C1 55068,c1(NC(C(C(C)C)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55069,N1(C(C2N(C)CCCC2)=O)CCN(C(=O)C(O)Cn2cncn2)CCCC1 55070,S(=O)(=O)(c1cccc(=NC2CCC(C)(N(C)C)CC2)[nH]1)NC(c1cnnn1C)C 55071,c1(N2CCC(N(C(=O)C(O)CCSC)CCC)C2)cc(C)c(C#N)cn1 55072,CC1CC(C(=O)NCC2CC3(CC3)CN2C(c2cc(O)cs2)=O)CCC1C 55073,c1(C(=O)NCCC2CN(C(C(n3c(C)ncc3)C)=O)CC2C)ccc(F)nc1N 55074,C1(NC(C2CCC(C)O2)=O)CCC(CNC(=O)CCF)CC1.C1CCCCC12CC2 55075,CC(CC(=O)c1cccc(F)c1)C(=O)NC(C)CC(C)(O)C1=CCC1 55076,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55077,C(C)(C(=O)NC1CC(NC(c2cc(C)sc2N)=O)C(O)C1)(C(C)C)OC 55078,N1(C(C(C)OCCCC)=O)CC2(CCC(NC(C3C=C(C)CS3)=O)CC2)C1 55079,S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(=O)C=Cc2ccccc2)C2C1C2 55080,n1(CC=C)ncc2c(O)nc(=NNC(=O)c3cc(C)ccc3N)[nH]c12 55081,C(=O)(NN1CCCC1C(=O)NC1CCN(CC(F)F)C1)c1cc(C(N)=O)[nH]c1 55082,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55083,C1(CC(=O)NC2(C)CCN(C(C3(C)C(C(=O)OC)CC3)=O)C2)CCC(C)(C)CC1 55084,C1(NC(C2C(CNC(CCCC3C(C)C3)=O)OCC2)=O)CCOC1(C)C 55085,C1(C(=O)NCC2CC(NC(=O)CCOC3CC(F)(F)C3)C2)CCCCCS1(=O)=O 55086,c1(CC)coc(CC(=O)N(CCNC(=O)C(C)(C)C2(C)CC2(F)F)CC)n1 55087,C1(C(N(CC(C)Br)C)=O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55088,c1(C(=O)NCCCCNC(C#CC(C)(C)C)=O)cc2n(n1)CCCC2=O 55089,C1(NC(COCCOCCOC)=O)CCN(c2ccccc2)C1.C1(=O)C(F)CN1 55090,C12(NC(C(CC#C)O)=O)CCOCC1CN(C(c1cn[nH]c1)=O)C2 55091,CCC(c1ccnc(NCC2CC23CCOC3)c1)=CCO 55092,N1(C(COCC)=O)CCOCC(CNC(c2nc(C)n(C)n2)=O)C1 55093,C=CC1(C(=O)NC(C)CC(C)NC(=O)CCCn2ccnc2C)CCCCC1 55094,N#CC1CN(C(C2(c3ccc(F)cc3)CC2)=O)CCN1C(C1CCOCC1)=O 55095,N1(C(CCC=C(C)C)=O)CCCC2(CCC(NC(=O)CCc3cnn(C)c3)C2)C1 55096,c1(NCC(c2n(C)ncc2)(C)C)nc(NCC23CC(CCO2)C3)nc2sccc12 55097,c1(NCC2CN(C(C3CCCO3)=O)CC23CCC3)c(Cl)cc([N+](=O)[O-])cc1Cl 55098,C(=O)(CCCCCN=[N+]=[N-])N1C(CN(C(C(C)c2ccsc2)=O)C)CCC1 55099,c1(C(=O)NC(C)CC(N)=O)cncc(NC(=O)CP(C)(C)=O)c1 55100,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1ccnn1 55101,n1(CC(N2CC(C(C)NC(c3c(C)n(C)nc3)=O)C2)=O)ncn2nccc2c1=O 55102,N12CC(C3CCCCC3)CC1C2=O.c1(SC)cccc(N)c1 55103,N1(C(CC2CC(=O)OC2)=O)CCC(N(c2nnnn2-c2ccc(F)cc2)CCO)CC1 55104,Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCC1NC(c1csnn1)=O)O2 55105,C(=O)(C#CC1CCOCC1)NC(CCC)CC(=O)NCc1cnccc1OC 55106,N1(C(C2C(C)CC=CC2)=O)CCC(F)CC1C(=O)NCC1(C#N)CC(C)(C)C1 55107,C(=O)(C(C)CC(C)C)NC(CNC(COCCOCCOC)=O)C 55108,CCC(CN(C)C)CC(=O)NCC1CC1NC(=O)CC(C)(C)CC(=O)OC 55109,c1(CSC)cccc(NC(C2C(CNC(c3cccc(C(C)C)n3)=O)CC2)=O)c1 55110,C1(CCC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOC1)=O 55111,c1(OC)ccc(CNC(=O)NNC(C)Cc2cccc(OC)c2)c(F)c1Br 55112,C1(C(=O)NCC(C2CCN(C(C3(O)CCOCC3)=O)CC2)C)CCS(=O)(=O)C1 55113,Cc1cc(C(N2CCC3(NC(=O)C=C4CC4)CC3C2)=O)cc(C)c1O 55114,C1(C(N(CC(C)N(C(=O)CNC(N2CCCC2)=O)C)C)=O)COC(C)CO1 55115,OC1C2CC3C(C2)C13c1nc(-c2ccc(Cl)nc2)nn1-c1ccc(Cl)cc1 55116,c1(C(=O)Nc2cc(C)c(NC(c3ccnnc3C)=O)cc2)ccn2cncc2c1 55117,C(CCC(=O)NC1CC(C)(NC(c2ncsc2Br)=O)C1)OCC=C 55118,O=C(C1=CCOC1)NCC1CC1NC(C1CCCC1(F)F)=O 55119,CCCCCCCCC(F)C(=O)NCCC1(OC)CN(C(c2coc(Cl)n2)=O)C1 55120,c1(N2CC3C(C(=O)NCC4CCOCC4)C3C2)cnccc1[N+](=O)[O-] 55121,C1(CN(C)C(=O)N(C(C)(C)C)C)CC1C1CC1 55122,c1(C(N(C)CC2(O)CCN(C(C3CC4(CCC4)C3)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 55123,c1(C(=O)NCC(CNC(CCCOC)=O)F)cccc2cccnc12 55124,C(=O)(NN1CCCC1C(=O)NC1CC2(CCCCC2)C1)C1CCC(=O)N1 55125,c1(OC)cc(C)c(C(=O)NC2CCCC2CNC(c2c(C)coc2C)=O)cn1 55126,c1(C(=O)NC(CNC(C(CC)Cc2ccccc2)=O)C)ccc(C(C)C)c(F)c1 55127,C12(C)CCCN1C(=O)C(=O)NC2.c1(OC)ccc(CN2CCC(C)CC2)cc1 55128,C1(n2cnnn2)(CC(=O)NC2(C)CN(C(c3cc(C4CC4)no3)=O)C2)CCOCC1 55129,N1(C(C2C(=C)C2)=O)CC(C(=O)OCC)C2(CCC2)C1.c12n[nH]c(c1C)C(=O)N2 55130,c1(CNC(C(CO)NC(C2C(CC)CCC2)=O)=O)ccc(C)cc1O 55131,Cc1nccc(C(=O)NC2CC=CC(C(=O)NCCCC3CCCC3O)C2)c1C 55132,c1(C(N2CCCOCC2)C(=O)NC2COC2)cnc(F)c(F)c1 55133,CC1(Nc2[nH]c(=N)sc2C2CCN(C(=O)OC(C)(C)C)CC2)CC(C2CC2)=NO1 55134,C1(CC)(NC(=O)CN2CCSCC2)CCCN(C(c2ccc(Cl)c(OC)c2)=O)C1 55135,c1(CC(=O)N(CC(C)NC(C)=O)CC)cc2c(OC)cc(OC)cc2[nH]1 55136,CC12CCN(CC1)C(=O)CC1CCOC2C1.C1(C2CCC2)(C(=O)N)CC1 55137,N1(C(C)=O)CCC2(CCC2)C(NC(c2cc3sc(Br)cc3[nH]2)=O)C1 55138,N1(C(C2(Br)CCC2)=O)CCC12CN(c1ncc(Br)c(Oc3ccccc3)n1)C2 55139,CC(C)C(C(=O)NC1CCC(NC(c2ccccc2Cl)=O)C1)Sc1cccnc1 55140,c1(C(=O)NCC2N(C(C(C=C)O)=O)CCN(C)C2)ccc2[nH]ccc2c1F 55141,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55142,c1(CCOC(CC2OCC(C(=O)OCC)C2)=O)ccnnc1S 55143,Cc1cc(C(=O)NCC2(O)CCN(C(=O)C(C)C3=CCCC3)C2)cc2nc[nH]c12 55144,c1(C(N2C(CNC(C3C(C)(C)OC(=O)N3)=O)CCCC2)=O)c(Cl)cccc1[N+](=O)[O-] 55145,N1(C(c2c(CC)occ2)=O)CCc2cc(CN=c3[nH]c(C)c(Br)s3)ccc21 55146,C(=O)(C1=CCCCC1C)N(CCC(=O)N(C)CC1CCCOC1)C(C)C 55147,N1(CCN(C(=O)CC2CC=CCN2C)C)CCN(C(c2ccns2)=O)CC1 55148,C1(NC(c2c(C)nc(O)[nH]2)=O)CCC(C)N(C(c2ccc(C3CC3)c(F)c2)=O)C1 55149,C(=O)(CC(C)n1cccc1)NCCCN(C(C1CC(O)C1)=O)CC 55150,CCCCCC(CC)C(=O)N(CCCCCC(=O)NCCCCSC)C 55151,Cc1cc(Br)c(N)cc1C(=O)NCCN(C(=O)CCCC(F)(F)F)C 55152,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55153,N1(C(c2ccc(OC)nc2)C(=O)Nc2cccc(Cl)c2C)CCC2(CCCO2)C1 55154,c1(C(N2CC(NC(C3(C)CC3(F)F)=O)CC(C)C2)=O)ccc2c(c1)C(=O)C(=O)N2 55155,C1(NC(C(C)NC(=O)NC)=O)CC(C)N(C(c2ccc(C)n2C)=O)C1 55156,c1(C(N2C(CNC(=O)C(O)c3ccco3)CCC2)=O)cnn2cccc(Cl)c12 55157,N1(C(c2cc(C)n(C(C)C)c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55158,c1(C(=O)NCC(CNC(c2ncc(C)cn2)=O)O)c(N)sc2ccccc12 55159,c1(C(N2C3CC(CC(NC(=O)COCC(F)(F)F)C3)C2)=O)ccc2n[nH]cc2c1Cl 55160,c1(NC(CC)C(=O)N(C)CC2(NC(=O)C(N)=O)CC2)cccnc1Cl 55161,C(=O)(C1=CCN(C(c2cnnc(O)c2)=O)C1)NC(C(C)C)CO 55162,N#Cc1ccc(C(=O)NCC#CC(N2CCCCCC2C(N)=O)=O)nc1 55163,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2ccno2)n(C)c1=O 55164,c1(CC(=O)NC2(COC)CCN(C(C3(C)CC(C)(C)C3)=O)C2)ccc(C#N)cc1 55165,C1(C(=O)NCC(C(=O)NC)C)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55166,N1(C(c2c(C)cccc2)=O)CCC(C)C(CNC(=O)C(c2cnccn2)C)C1 55167,CC(C)CC(C)NC(=O)C(C)(CSC)NC(=O)CN1CCNC(=O)C1.C(C)(=O)O 55168,C(=O)(C1=CC2C=CC1C2)N1CC(OC(c2ccc(C)c(C(=O)N(C)CC)c2)=O)C1 55169,N(C(=NCCCn1cccn1)NCCF)CC1CC(OC)(OC)C1 55170,C(=O)(C(CC(C)C)c1ccccc1)NC(CC=C)CNC(=O)CSCC(F)(F)F 55171,c1(C(=O)NCC2(CNC(C3(C)CC4CCC3O4)=O)CC2)ccc(Cl)c([N+](=O)[O-])c1 55172,c1(C(N(C2CCCCN(C(=O)C(C)(C)CF)C2)C)=O)cn2ccc(F)cc2n1 55173,CCCCC(C(=O)N=c1ccn(C(C)CC)[nH]1)NC(=O)Cn1ccnc1C 55174,C1(NC(C(C)SCC)=O)CC1C1CCN(C(C2(C#N)CCN(C)CC2)=O)CC1 55175,Cc1nc(CCC(N2CC3CC3(CNC(=O)CCc3cncnc3)C2)=O)[nH]c1C 55176,C1(CC=C)(C(N(CC(=O)NC)C)=O)CCN(C(=O)CNC(=O)C(C)CC)C1 55177,c1(CN(C(=O)COCC2CCCCC2)C)ccc([N+](=O)[O-])cc1C(F)(F)F 55178,c1(C(=O)NCCCC(C)NC(c2ccc(C)s2)=O)ccnc2c1ncn2C 55179,Cc1ccc(C)n1CC(=O)N(C)CC1CCCN1C(=O)Cc1ccncc1F 55180,Cc1onc(Br)c1C(N1CC(CNC(c2ccc(O)nn2)=O)C(C)C1)=O 55181,c1(C(N(CC(C)N(C)C(C2(n3cccn3)CC2)=O)C)=O)cccc(C(C)(C)C)c1 55182,c1(C(N2CC(CC(=O)N(CCF)CC)OCC2)=O)ccn2ccnc2c1 55183,Cc1cc(C(=O)NCC2CC(NC(=O)Cc3cc(Cl)cs3)C(O)C2)cn(C)c1=O 55184,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CNC(CN(CC(C)(C)C)C)=O)C1 55185,C1(NC(CCSCCC)=O)CC2(CCCN(C(=O)CCC3CCCC(=O)N3)C2)C1 55186,N1(C(CCC2C(C)(C)C2)=O)CCOCC1(C)CO 55187,C(=O)(C(CO)C(C)(C)C)NCCCN(CCC)C(c1ccc(CC(C)C)s1)=O 55188,S(=O)(=O)(C(F)(F)F)N1CC(C(N)=O)(NC(=O)Cn2ccnc2)C1 55189,c1(N2CCN(C)C(c3ccccc3)C2)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55190,c1(C(C)N)ccc(C(=O)NCc2ccc(F)cn2)cc1.C=CC1(C(=O)NC)CCC1 55191,N1(CC(=O)NCCOCC)C2CCC(NC(=O)C=Cc3ccsc3)CC1C2 55192,C1(NC(C2CCCOC2)=O)CCCN(C(c2sccc2OC(F)F)=O)C1 55193,C1(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)OCC2CCCC1C2 55194,C1(CS(=O)(=O)NC(C(=O)OCC)(C)C)CC(C)NC(C)C1.C12CC3C(C3C1)N2 55195,c1(OC)cc(C)cc(C(=O)NC(C)CCCNC(=O)C(O)C(C)C)n1 55196,c1(CCC(=O)NCC2(F)CCC(NC(C(C)(C)C)=O)C2)c(F)cccc1F 55197,CC1(C)CC(NCC2CC2)CC(C)(C)C1.C(=O)(CCCC1CC1)O 55198,Cc1cc(C(=O)N(C(C(=O)N2CC(C(C)(C)C)C2)C2CC2)C)nn1C 55199,Cc1ncc(NC(C2CCC(NCc3cccc(I)c3O)CC2)=O)c(C)c1Br 55200,N1(C(c2c(CSC)cccn2)=O)CCC(CNC(=O)CCCOC(C)C)C(O)C1 55201,C12(C(N3C(CCNC(C4CC5(C4)CC5F)=O)CCC3)=O)CCCCN1CCC2 55202,CC1CC(NC(C2(C)CC2(F)F)=O)CCN1C(c1coc(O)n1)=O 55203,C1(C(=O)NCc2nc(=O)o[nH]2)CN(C(c2cccc3c[nH]nc23)=O)CC12CCC2 55204,N1(C(C2(CCF)CC2)=O)CC2(NC(C3CC3)=O)CCC1C2.c12cccc(c1)C(=O)N2 55205,C(=O)(C1CC=Cc2ccccc21)NC1CC(F)(CNC(C(C)(C)N2CCCC2)=O)C1 55206,C(=O)(CCCC(C)(C)C#N)NCC1N(C)CCN(C(C(C(=O)OC)(C)C)=O)C1 55207,c1(C(=O)NC(CC#C)CO)cc2nccc(OC)c2s1 55208,CCCC(C(F)(F)F)NC(=O)CC1CC1CNC(=O)Cc1ccoc1C 55209,CN1CCN(S(=O)(=O)c2cccnc2N2CC3CCOC3C2)CC2(C)CCCC12 55210,n1(CC(=O)NCC2(OC)CN(C(C3CC=C(C)CC3)=O)C2)c(C)cc(C)nc1=O 55211,N1(C(C2N(C(=O)C(c3ccccc3)F)CC(C)(C)C2)=O)CCC(F)(F)C(F)C1 55212,C(CCC(=O)N1CCCC1C1(C(N2CC(C)(C)C2)=O)CC1)N(C(C)=O)C 55213,C1(C(N2C(Cn3cc(CSCC)nn3)CC2)=O)CC2CSCC(C1)C2 55214,N1(C(C=C(C)C)=O)CC(NC(C2CCOC2c2cccnc2)=O)CCC(O)C1 55215,C(c1ccc(O)c(OCCC)c1)=CC(=O)NCC(CC)Nc1snc(C)c1C#N 55216,C(=O)(CCCc1ccccc1)NC1(CNC(CN(C2CCC2)C)=O)CCC1 55217,CC(CNC(c1cc(CO)ccn1)=O)CC(=O)N(C)CC1CCOC(C)C1 55218,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55219,C1(C)(C(=O)OC)CCN1C(=O)CC1CCCN1C(=O)C=CCF 55220,c1(N(CCC(C)NC(CCCC#CC)=O)C)nc(C(=O)OCC)nc(C)c1OC 55221,C1(C)(NCc2nc(CC)oc2)CCN(c2ccnc(-c3cc(OC)ncn3)n2)C1 55222,C12(C(=O)NC(CN(C(Cc3cc(OC)no3)=O)C(C)C)CO)CC(C)(CO1)C2 55223,c1(CCC(=O)NCC(C)NC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55224,C(C)(C(=O)N(CCC(C)NC(=O)CCc1cncs1)C)(C(F)(F)F)NC(C)=O 55225,N1(C(C(C2CCN(C(c3cc[n+]([O-])cc3)=O)CC2)C)=O)CCC(C)(O)C(O)C1 55226,C1(C(N(C2CCC2O)C)=O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55227,CCC(C)CCC(=O)N(CC(CC)NC(c1cc(OC)ns1)=O)C 55228,c1(CCNC(C(N2CCC(c3ccno3)CC2)C)=O)nc2ncc(Br)cn2n1 55229,c1(C(=O)NCCCCCCNC(c2c(C)nc(C)[nH]2)=O)cccc2oc(C)cc12 55230,c1(C(=O)NCc2nc(CNC(c3n(CC=C)ccn3)=O)sc2)ccc(F)cc1C 55231,c1(C(=O)NC2CN(C(=O)C(O)C(F)(F)F)CC2O)cc2c(F)c(F)ccc2[nH]1 55232,c1(CNC(=O)CCc2cncs2)cc2ccccc2[nH]1 55233,C1(CC(N2CCCC(c3n(C)c(S)nn3)C2)=O)CC2CNCC2C1 55234,C1(NC(C(C(C)OC)NC(c2ccc(O)cc2)=O)=O)CCCCCC1N(C)C 55235,C(N=c1[nH]cnc(NCC2COC(C)(C)CO2)c1C)c1cc(CC)c(F)cc1 55236,C(=O)(C1=NNC(=O)CC1)N1CCCC(F)(CNC(c2c(CCC)onc2C)=O)C1 55237,c1(C(C(=O)NC2C(CNC(=O)C=CSc3ccccc3)C2)=O)ccc(Cl)s1 55238,CCC(O)C(C)C(=O)NC(C)(C)CCC(=O)NC1(c2cc[nH]n2)CC1 55239,c1(CN2C(C)(C(N(CC)Cc3ccccn3)=O)CC2)cccc(C(F)(F)F)c1Cl 55240,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOCC#C 55241,N1(C(Cc2ccc(NC(C(CC(C)C)F)=O)cc2)=O)CCNC(=O)CC1C 55242,CC1(C)CN(C(=O)CN2CCOCC2)CCC1NC(C1CC1)=O.c1(SCO)ccccc1 55243,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55244,CC(C)C(C)(CNC(=O)CC1CC1(C)C)NC(c1ccc(C(F)(F)F)cn1)=O 55245,N1(C(Cc2cccc(SCC)c2)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55246,C1(N(S(=O)(=O)CCc2ccccc2)C(=O)CCc2ccccc2F)CCCCCC1O 55247,N1(C(COC2CN(C(c3c(C(C)C)n[nH]c3)=O)C2)=O)CC(O)C(N=[N+]=[N-])C1 55248,C(CS(=O)(=O)CC(=O)NCC1(C)CN(C(c2ccc(O)cn2)=O)C(C)(C)C1)OC 55249,C(=O)(C(C)(C)C(F)(F)F)NC1CN(C(c2c(C)cn(C)n2)=O)CC1C 55250,C1(C(=O)NCC2OCCC2C(N2CC3(CCOC3)C2)=O)CC2(CCC2=O)C1 55251,O=C(CCCCCNC(c1ncncc1N)=O)Nc1cncc(F)c1 55252,C1(C)(CC)CN(C(c2cccc(OC(C)C#N)c2)C(=O)NCC2CCOC2)CCO1 55253,C(CCF)(C(=O)NC(C)CC1(O)CCC1)NC(Cc1cn(CC)nn1)=O 55254,C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(O)C1)N1C2CC(OC)C2CC1 55255,CC(C)C(F)C(=O)NCc1ccc(C(C)NC(C2CC(C(C)C)C2)=O)cc1 55256,Nc1ccnc(C(N2CC3(CC3)CC2CNC(c2csc(O)n2)=O)=O)c1Cl 55257,c1(C(=O)NCC(CNC(C(CSC)OC)=O)CO)cc(F)cc([N+](=O)[O-])c1 55258,c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cc2n(n1)CC(F)C2 55259,c1(C(C)O)ncc(C(=O)N(CC(C)CNC(c2ccnnc2)=O)C)s1 55260,CC(C)CC(C)(CN1CCOCC1)NC(c1ccc(NC(=O)C2CC2)cc1)=O 55261,C#CCCCC(=O)NCCOCC(N1CCCC1(CC#C)CC)=O 55262,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55263,C12(C(=O)NCC(CC)NC(C3CCCOCC3)=O)CCC(O)(CC1)CC2 55264,CC(C)CC(CNC(=O)CC(C)C(C)C)C(=O)Nn1cnn(C)c1=S 55265,Cn1c(C(N2CC(C(C)(C)O)(CNC(=O)Cc3cccs3)C2)=O)cc2ccsc12 55266,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C12CC2 55267,c1(C(C)=O)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55268,N1(C(C2C(C)CCC2)=O)C2CCC1C(F)C(NC(c1nc(Cl)ccc1C#N)=O)C2 55269,C=CCC(C(=O)N(C)CC1(C(=O)NC)CN(C(C2CC3(CC3)CO2)=O)C1)C(C)C 55270,c1(OC(C(=O)NCCC(C)(C)NC(C(COCC)C)=O)C)cccc(F)c1F 55271,O=C1NCCc2cc(C(N3CCCC(NC(c4cc(Cl)c[nH]4)=O)C3)=O)ccc21 55272,C(N=c1cc(C)[nH]c(=NCCc2ccnn2C)[nH]1)C1CCC=C(C)C1 55273,CC1(CC(=O)NCCCN(CCCNC(=O)CCc2cscn2)C)CCCC1 55274,C1(O)(CC(N2C(CC(C)C)CCC2)=O)CCN(C(C2CCCC2)=O)CC1 55275,CC(C)(C)C(CNC(c1ccc(=N)[nH]c1)=O)C(=O)NC1CC2CCC1O2 55276,CCCC(O)C(=O)NC1CC(F)(CNC(=O)C(C2CCOCC2)O)C1 55277,C(CN(C=O)Cc1ccc(C(F)(F)F)s1)(CC(C)C)OC 55278,c1(CNC(=O)NC(c2cc(C(=O)OC)c(C)cc2)C)cnn2cccc(F)c12 55279,Cc1cc(C(=O)NCC2CC(O)CN2C(C2(C3CCCO3)CCC2)=O)cc(O)n1 55280,C1(NC(=O)CC(O)C2CC2)CC1C1CCCN(C(c2cnc3occc3c2)=O)C1 55281,c1(CCCC(N2CC(O)(C(C)NC(CC(C)O)=O)C2)=O)ccc(S)cc1.C(N)=O 55282,N1(C(C2(N(C)C)CC2(C)C)=O)CCCN(C(C2CS(=O)C2)=O)CC1 55283,N1(C(C2(C)CCOC2)=O)CCN(C(c2cc(CO)on2)=O)C(CCO)C1 55284,CC(c1cccnc1)=CC(=O)NC1(C)CCN(C(=O)CC(O)CN(C)C)CC1 55285,Cc1ccc(OCC(=O)N(C(C)CCNC(=O)CC2CCN(C)C2=O)C)cc1 55286,C1(C(=O)NC(C2CCOC2)CNC(=O)CC2CCSC2)Cc2ccccc2N1 55287,c1(C(=O)NCC(CC=C)NC(=O)C(C)S(C)(=O)=O)coc2cc(F)ccc12 55288,C(=O)(CC1CCOc2ccccc21)N(C)CC1CCN(c2ncccc2C#N)C1 55289,C(N=c1nc(NC2CCCC2)c2ccccc2[nH]1)c1cc(Cl)cc(Cl)c1 55290,c1(N(CCOCCN(C(C(CC(=C)C)NC(C)=O)=O)C)C)cnn2ncccc12 55291,C1(C(=O)NCC23CC(NC(C(C)N(C)C)=O)(C2)C3)COC(=O)N1C 55292,N1(C(C2COCC(C)O2)=O)CC2(CCCC2)C1C(=O)N(C(C)C(C)(C)C)C 55293,c1(OC)ccc(CNC(C23CC2CCN3C(c2[nH]ccc2C2CC2)=O)=O)cn1 55294,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(C(=O)Nc2ccnc(Cl)c2)C1)=O 55295,C1(C(=O)NCCC2(C)CC2)CC2(CCN(C(c3cccs3)=O)CC2)C1 55296,CC(C)(C)C(=O)CCC(=O)NCC1CCCN(C(C2(C)COCCO2)=O)C1 55297,CC1ON=C(C(=O)N(CC(C)O)CCNC(c2cc(-c3ccncc3)no2)=O)C1C 55298,c1(C(N2C(CNC(C3(C)N(C)CCC3)=O)CCC2)=O)cnc(N)c(N)c1 55299,C=CC1(C(=O)N(C(C)CN(C)C(C)=O)C)CCN(C(=O)CC2CC=CCC2)C1 55300,C(c1ccccc1)=CC(=O)NCC1(C(=O)NCC(F)CO)CCCC1 55301,C(=O)(CS(=O)(=O)C1CCCC1)NCCCC(C)NC(c1c(OC)csc1)=O 55302,Cc1nc(=N)[nH]c(=NCC(C)N(C)C(C2CC=CCC2)=O)[nH]1 55303,C(=O)(CC(C)(C)CC(=O)Nn1cc(C(C)OCc2cccc(Cl)c2)nn1)OCC 55304,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55305,c1(C(=O)NC2CC(F)(CNC(CNC(=O)OC)=O)C2)cnc2sccc2c1 55306,C1(OCC#C)CCCN(C(=O)C(C)CNC(C2CCC=CCC2)=O)C1 55307,c1(C(C(=O)NCC=C)N(C2CCC=C2Br)C)ccn(CC)n1 55308,CC(C)CC(C(=O)NCC1C2CN(C(c3cnn(C)c3C#N)=O)CC12)N(C)C 55309,CC1(C)CN(C(c2ncoc2C(F)F)=O)CC(CNC(=O)CCC2(C)CC2)O1 55310,Cc1nc2cc(C(=O)NC3CC(NC(=O)CC4CC(O)C4(C)C)C3)ccc2o1 55311,c1(C(=O)NC(CC#C)C)ccc(C2CCCCN2C(=O)CC2COC(=O)C2)n1C 55312,C(CO)(CCC(C)C)NC(C(CNC(C1CCC(F)(F)C1)=O)OC)=O 55313,CC(O)C(C)(C)C(=O)NCC1(CNC(c2ncccc2OCC(F)F)=O)CC1 55314,C(=O)(C1CCc2c[nH]nc21)N1CC2N(C(C3(CC=C)CC=CC3)=O)C(CC2)C1 55315,C(C(=O)N(CCC(=O)OCc1ccccc1F)OC)N(CCC#N)CC 55316,S(=O)(=O)(c1ccc(Cl)cc1F)N1C(C#N)CN(C(c2scnc2Cl)=O)CC1 55317,c1(-c2cccc(CNCC3OCCN(C(C)=O)CC3)c2)c[nH]c2cc(F)ccc12 55318,C(CCc1ccc(F)cc1)(C(F)(F)F)OC(c1c[nH]c(=N)o1)=O 55319,Nc1cc(F)cnc1C(=O)NC1CCN(C(=O)CSc2ccccc2O)CC1O 55320,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCCC1CCCCC1 55321,C=CC1CN(C(=O)CCOCCNC(C2CC(C)=NO2)=O)CCO1 55322,C(=O)(C(CC(C)(C)C)NC(c1ccc(CF)cc1)=O)N1CCC(C(C)C)CC1 55323,C1(SC)CN(C(=O)Cc2nccn2C)CC1NC(c1ns[nH]c1=O)=O 55324,C(=O)(C1(C)CCn2ccnc21)NC1CC(CNC(c2cc(OCC)ncc2)=O)C1 55325,c1(C(N(CCCCCC)CCNC(=O)CCn2ccc(C)n2)=O)cc(Cl)cn1CC 55326,N1(C(C2(CC=C)CN(C(C3CCCCS3)=O)C2)=O)CCC2(CCC(OC)C2)C1 55327,C1(NC(C(CCC)CC)=O)CN(C(c2cccc(=O)o2)=O)C2(CCOC2)C1 55328,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55329,CC1(C)CC(NC(C2(CF)CCOCC2)=O)CN1C(C1CCCCC1(F)F)=O 55330,C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCCC2)=O)NC1CC(CC(=O)OC)C1 55331,c1(C(N(CCN2CCN(C(C(CCCC)C)=O)CC2)C)=O)cc(F)c(Cl)cc1F 55332,C=CCCCCC(=O)N(CC(C)NC(C1CCN(CCF)CC1)=O)C 55333,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55334,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55335,c1(C(=O)NC2C(NC(C=NOC)=O)COC2)cnc2c(c1)NC(=O)CS2 55336,N1(CC(=O)NCC(C)N(C(C2(OC)CS(=O)(=O)C2)=O)C)CC(=O)N(C)C1=O 55337,C(=O)(CC(C)C(F)(F)F)NCC(C(=O)NCCc1nnc(C)o1)N(C)C 55338,c1(CCC(=O)NC2CC(NC(C(=Cc3ccccn3)C)=O)C2)cc(F)ccc1F 55339,N1(C(C=C(COC)C)=O)CCCOC(CNC(=O)CCN(C)C)C1 55340,C=CCCC(C)(C)C(=O)N1CC(NC(=O)C(C)NS(=O)(=O)CC)C(C#N)C1 55341,C1(C)(Sc2c(NC(C)=O)scc2)CCN(C(c2c[nH]c(=O)cn2)=O)CC1 55342,C(=O)(C(O)C(C)(C)C)N1CCC(C)(CNC(CCc2ccc(C)cc2)=O)C1 55343,c1(NC(C(CC)N(C(=O)CC(C)OC)C)=O)cn(C)nc1OC 55344,c1(C(N2CC(C(=O)Nc3ccc(O)cn3)C2)=O)ccc(F)c2ccccc12 55345,c1(C(=O)NC(C)CCCNC2CC3(CC3)CO2)cc([N+](=O)[O-])cn1C 55346,CC1CC(NC(=O)C(O)CC2CC2)CCN1C(=O)Cn1nccn1 55347,N1(C(C(C(=O)NCC)F)=O)CCN(C(c2cc(OC)nn2C)=O)C(CC(F)F)C1 55348,C(=O)(C1=C(C#N)CCC1)NCCCC(C(=O)NC(c1ccccn1)C)O 55349,C12(CNC(COC3CCN(C(CCC(N)=O)=O)C3)=O)CCCC1OCC2 55350,C1(C(N(C)C)=O)CCC2CCC1N2C(=O)Nc1cccc(-c2ccon2)c1 55351,C(=O)(C(=O)C(C)CC)N(C(=O)CN(CC)CC)CC.C(C(C)N)NC1CC1 55352,C(C)(C)(C(=O)NO)NC(C(c1ccncc1)OCC)=O 55353,N1(C(CC2C(C)(C)C2(C)C)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55354,c1(CC(=O)NC(CC)CN(C(=O)C(C2CC2)OC)C)ccc(OC)cc1F 55355,C(C1=CCC2CC1C2(C)C)(c1n(CCCOC)nnn1)NC1C2CCCCCC12 55356,c1(C(=O)NCC2CCCC(NC(CCCN=[N+]=[N-])=O)C2)ccc2ncnn2c1 55357,S(=O)(=O)(c1ccc(N2CCC(C)C2)cc1Cl)NCc1cccc(OC)c1C 55358,C(=O)(CC(C)C(F)F)N1C(C(N2CC(OCC(=O)NC)C2)=O)CCC1C 55359,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)CC(C)F)CC1F 55360,c1(NCC(C)N(C(C(C(C)C)N(CC)CC)=O)C)ccc(Cl)cc1[N+](=O)[O-] 55361,C(CCC(C)C(=O)NCC1C2CN(C(=O)CSC3CCOC3=O)CC12)OC 55362,C(=O)(C1SCc2cccnc21)N1CC(CNC(COCCC)=O)C(O)C1 55363,c1(OC)ccc(NC(C2CCCN(C(c3sc(Cl)nc3Cl)=O)CC2)=O)c(I)c1 55364,C(CCCCC(=O)Nc1cccc(Cl)c1C)NC(C(C1CCCC1)OC)=O 55365,N12CC(CC(C)C1)C2=O.C#CC1(NC(CCCCC)=O)CC1 55366,c1(OC)ccc(C(=O)NC2CCN(C(c3nc(C)nn3C)=O)CC2C)c(F)n1 55367,C(=O)(C#CC1CCCOC1)NCC1C(C(C)C)CCCN1C(=O)CCC(F)(F)F 55368,C1(CN(C(=O)C(F)F)C)CN(C(=O)CCn2ccnn2)CC1C(F)(F)F 55369,c1(OC)cc(CC(C)N(CC(C)OC2CC2)C)ccc1O 55370,CCCCC(C(=O)N(C)CC1CN(C(C2CCC(=O)N2)=O)CCO1)C(C)C 55371,C(=O)(CCC(N)CC(F)F)N1CC(C)C(C2CCCN2)CC1.C(CCCCCCO)N 55372,CC1OCCC1CC(=O)NCC1CC(NC(c2ccc(Cn3cccn3)s2)=O)C1 55373,Cn1ncc2cc(C(N3CC4CC4(CO)C3)C(=O)N3CCCC3)ccc12 55374,N1(C(c2c(NC)cncc2)=O)CC2CC(C1)C2NC(=O)C=Cc1ccoc1 55375,N1(C(c2ccn(C)c2)=O)C2CCCC1CN(C(C13COCC1C3)=O)CC2 55376,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)C(F)=C(C)C)C(CCO)C1 55377,c1(CC)c(C(=O)NC(C2CCN(C(=O)CSC)C2)(C)C)nnn1C 55378,N1(C(Cc2cc(SC)c(C)cc2)=O)C(CNC(C2CCCO2)=O)CC2CCCC12 55379,C(C(N=[N+]=[N-])C(=O)N1CC(F)(C(N2CC(CC(F)(F)F)C2)=O)C1)OCC 55380,CN1CCN(C(c2cc(Cl)cs2)=O)C(C(N2CCCC2(C)C2CCC2)=O)C1 55381,C1(CCO)C(=O)NC2CC(F)(C2)CNC(=O)CSC1.CC(C)N(C)CCO 55382,c1(OCC2CCN2c2c(-c3ccccc3)ccs2)ccc(Nc2ccccc2)cc1 55383,Cc1ccc(C(=O)NCC2CCCCN2C(c2cncc(CO)c2)=O)c(N)n1 55384,c1(C(=O)NC(C2CCN(c3nccc(OC)n3)CC2)C)cc(F)cc(Br)c1C 55385,CCCC(CCC)=CC(=O)N(CC(O)CN(C)C(C1CC1C1N=C(OC)CO1)=O)C.CC 55386,CC(C)C1=NOC(C(=O)N(CC)CC2(O)CCCN(C(=O)CCC=CC(C)C)C2)C1 55387,Cc1ccnc(O)c1C(=O)NCC(C)NC(=O)Cc1nnc(-c2ccccc2)o1 55388,C(=O)(C1=CC2(CCN(C(=O)C(C3CCCCC3)O)C2)C1)NCc1nc(C)c(C)s1 55389,C1(NC(CCCc2onc(C)n2)=O)CN(C(C23CCCC2C3)=O)CC1CO 55390,c1(C(=O)NCCC(CNC(CCc2cc(C)on2)=O)O)cccc(CC#N)c1 55391,C(CCN=c1[nH]c2c(c(=NCC3(C)COCCO3)[nH]1)SCC2)OC(C)C 55392,c12ccc3cccc(c3n1)[nH]2.C1(C(N)=O)C2CN(C(=O)C3CC3)CC12 55393,CC1(CNC(c2cc(=O)cc[nH]2)=O)CCCN1C(c1nc(Cl)c(Cl)s1)=O 55394,C#Cc1cnc(C(N2CCC2CNC(=O)Cc2cccc(C(C)C)c2)=O)c(C)c1 55395,n1(CC=C)c(-n2nc(C)nc2Nc2ccccc2)nnc1CC(C)(C)C.C(N)=O 55396,c1(N(C)Cc2ccc(CSC)cc2)cccc(F)c1[N+](=O)[O-].C12CCN(C1)C(=O)N2 55397,C1(CC)(CC)CC(NC(=O)C(=O)N(C)C)CN1C(=O)C(C)Oc1cccnc1 55398,c1(CNC(CC2N(C(c3c(CC)n(C)nn3)=O)CCC2C)=O)nn(C)c(=O)n1C 55399,c1(C(=O)NC(C(=O)N(CCO)CC)c2ccco2)cccc(O)c1F 55400,C1(OC)CCN(C(=O)C(C2CCN(C(=O)C(C)C)CC2)(C)C)C1C 55401,C1(C(N2CC(C(=O)NCC3CC(OC)CN3C(C)=O)C2)=O)Cc2nccnc2C1 55402,C(=O)(C(C)CCCOC)NC(C(=O)N(CCC)CCO)CCOC 55403,C1(CNC(COCCCC#C)=O)CC2(CO1)CN(C(=O)C(C)(C)CC=C)C2 55404,C1(C(N(C)CC2CN(C(CC=CC)=O)C2)=O)CCC(C)C1 55405,C12(CNC(CCSC)=O)CCCC1N(C(c1cc(C3CC3)ncn1)=O)CCC2 55406,c1(OCC)ccc(N(C)Cc2ccc(C3(O)CNC3)cc2)cc1 55407,n1(C(COC)C)nc(CCSc2ccccc2)nc1-c1cc(CCC(C)C)on1 55408,C(CCCC(C)NC(C1CC1(C)CC)=O)NC(C1(OCC)CCCC1)=O 55409,C=C1CON(C(=O)CC2CCN(C(=O)COc3ccc(C)cc3)C2)C1 55410,N1(C(c2c(COC)nn[nH]2)=O)CC(NC(=O)CCNC(=O)C2CC2)CC(O)C1 55411,N1(C(=O)NCC(CC(C)C)N)CCc2cc(Cl)ccc2C1 55412,C=CCC(C)C(=O)NC1(C(=O)NCc2cnn(C)c2C(C)C)CC1(C)C 55413,C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CNC(C1CC1CC)=O 55414,N1(C(c2ccoc2)=O)CCN(CCN2CCC(CC)C2)CC1 55415,C1(C(N(CCNC(c2ccn(C(F)F)n2)=O)C2CC2)=O)CC12CC(F)(F)C2 55416,C1(O)(C(C)NC(=O)C=CCn2cccn2)CCN(C(=O)Cn2cccc2)C1 55417,CC(CC(=O)N1CSCC1C(=O)NCC1CCCCCCC1)C(C)(C)C 55418,CC(C)C(CNC(C12CCC(CC1)C2)=O)C(=O)NC1CCCC(O)C1O 55419,CCCC(CCC)=CC(N1CCC(CF)(NC(c2cnn(CCO)c2C)=O)C1)=O 55420,CC(C)CC(CNC(C1(O)CC1)=O)NC(c1ccsc1Cl)=O 55421,C1(OCC(=O)NC2(F)C(CNC(=O)OC(C)(C)C)C2)CCN(C2CC2)CC1 55422,C(=O)(CCCCCO)N1C(C)CC(NC(=O)Cc2ccc(CO)cc2)C1 55423,N#Cc1c[nH]c(C(=O)N(c2cnc(C)[nH]2)CCN)c1.O(C(=N)O)CCO 55424,C1(CNC(CSCCOC)=O)CC2CCC(C1)N2C(=O)C=CC(C)CC 55425,C1(CNC2C(CC(C(F)(F)F)F)C2)CS(=O)(=O)CCO1 55426,c1(C(C(=O)NC2CCCC2)N(CCOC)C)cc(OC)c(F)cc1F 55427,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55428,c1(C(N2C(CN(C(c3c(C)cn(C)c3)=O)C)CCC2)=O)cc2c(C)n[nH]c2cn1 55429,C12(C(=O)NCC(CC)NC(c3cc(C(C)=O)n[nH]3)=O)CC(c3ccccc3)(C1)C2 55430,c1(C(N2C(C(=O)NC(c3cc(C)cs3)CC)CC(C)C2)=O)cc(Br)c(O)cc1O 55431,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CC)=O)C1 55432,c1(C(=O)NCCCNC(C(COC)C)=O)cc(F)cc2cc[nH]c12 55433,c1(C(=O)NCC2(CNC(C3C(C)CCS3)=O)CC2)ccc(F)c(F)c1 55434,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55435,N1(C(C2(CCF)CCC2)=O)CCN(C(=O)C(c2ccccc2F)O)CC1 55436,C(=O)(CC1CCCc2c1cnn2C)OC(c1c(OC)cc(Br)cc1)=O 55437,C1(CNC(=O)C2=CCCCCC2)CN2CCCCC2CN1C(=O)Cc1cnsc1 55438,C1(CC(N2CC(c3ccccc3)(NC(C3CN(C)C3)=O)C2)=O)C=CS(=O)(=O)C1 55439,N1(C(C(C)OCC=C)=O)CCCC(O)(c2cn(-c3ccc(=O)n(C)c3)nn2)CC1 55440,N1(C(c2n(CC)nnc2)=O)CC2CC(C(=O)NCc3ccc(C)cc3F)(C2)C1 55441,N1(C(Cc2nc(COC)sc2)=O)CCC2CN(C(c3cnn(C(C)C)n3)=O)CC12 55442,C1(C(N(CCC(C)NC(C(C)C=Cc2ccccc2)=O)C)=O)COCC(C)(C)O1 55443,N1(C(C)=O)CCCCC1C(=O)NCC=CCNC(c1sc(F)cc1Br)=O 55444,c1(CCOCC=C)ncoc1C(=O)NC1CC(C(=O)N(C)CCOC(N)=O)C1 55445,c1(OC)cc(C(=O)NCCC2CN(C(=O)CSC)CCO2)cc(Cl)c1 55446,C1(NC(CSCC#C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1(C)C 55447,C1(NC(c2cn(CC)nn2)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55448,Cn1cncc(C(=O)NC2(C(=O)NCCC3CC3C3CC3)CC(F)(F)C2)c1=O 55449,Cc1ccc(NCCNC(=O)NC2CCCN(c3ccncn3)C2)c(C)c1 55450,C1(O)(CCNC(=O)C(O)C2CCC2)CN(C(=O)CC2CCOC2=O)C1 55451,C(C(CC(C)C)C(=O)NC(C1CCN(C(c2cnc(C(C)C)nc2)=O)C1)C)OC 55452,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55453,Cc1cnc(CC(N2CCCC(C(N3CCCC(N(C)C)C3)=O)C2)C)cn1 55454,C(=O)(C1=CCCSC1)N(CC(N1CC(F)(CF)C1)=O)CCOC 55455,c1(C(N2CCC(O)(CCNC(C3CC(C#N)C3)=O)C2)=O)cc([N+](=O)[O-])ccc1Cl 55456,c1(C(C)NC(=O)C(C2CCC(C)(C)CC2)N)cc(=O)c2cc(Br)ccc2[nH]1 55457,c1(CNC(C23CC(C(=O)OC)(C2)C3)=O)ccc(O)cc1.c12cn(nn1)CC2.OC 55458,c1(OC(C)C)cncc(C(=O)NCC(C)NC(=O)C(C)(C)c2ccccc2)c1 55459,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CCN(C)C)c2)=O)C1)(C)C 55460,C1(C(N2CCC(CN(C(C(C)SC(C)C)=O)C)C2)=O)COCCN1C=O 55461,C(c1cccnc1)=C(C(N1C(CCNC(C(C=CC)O)=O)CCC1)=O)C 55462,c1(C(=O)NCCC2CCC(NC(CCCOC)=O)C2)nccc(Cl)c1F 55463,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55464,c1(CN(CC(C)C2CC2)C)ccoc1CO 55465,c1(C(=O)NCC2CN(C(=O)C(F)(F)CC3CC3)CC2(F)F)cccc2c1CCO2 55466,N1(C(C(c2ccccc2)C)=O)CCC(C(C)C(=O)N(C)CCN2CC=CC2)CC1 55467,C(=O)(C(C)C1=CCCC1)N1CCCCC(NC(c2cccc(C#C)c2)=O)C1 55468,CC(C)CCN=C(NCC(F)F)NC1C(O)CCN1C.c12ccccc1O2 55469,CCC(C)C(C)NC(C1CN(C(=O)C(Cc2ccccc2)NC2CC2)C1)=O 55470,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55471,c12ccc(nc1)c(=O)[nH]2.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55472,c1(C(=O)S)cc[nH]n1.C(=O)(CC)N1CC(=O)C1.N(C1CC1)(CC)CC.SC 55473,C(CC(C)C(=O)N1CC(OCCNC(c2cnc(N(C)C)s2)=O)C1)OC 55474,c1(CC(=O)NC(C)CN(C)C(C2CC(=O)N(O)C2)=O)ccc(Cl)c(F)c1 55475,c1(C(C(N2CCC(C(=O)NC3(COCC)CC3)CC2)=O)=O)ccc(F)c(C)c1 55476,CCCCCCC(CC)NC(=O)C(C)NC(=O)CNC(=O)C(CC)CC 55477,CC(Cc1ccnn1C)C(=O)N1CCC1N(C(=O)CCC)C(c1ccccc1)(C)C 55478,c1(CNCC(O)CCc2ccccc2)nc2c(s1)CCc1ccccc1-2 55479,c1(C(=O)NCCN(C(c2ccn(CCC)n2)=O)C2CC2)cc(COC)c(C)o1 55480,Cc1ccc2c(c1)CCC2CC(=O)NCC1CN(C(=O)CCCCCF)CC1C 55481,N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 55482,C(CCCCCNC(=O)C(c1ccnn1C)C)NC(C(C)C=C1CCC1)=O 55483,C(CC(F)CN=[N+]=[N-])CNC(C1(NC(C(CC=CC)C)=O)CCSC1)=O 55484,c1(C(N2CCC(C3CCCN3C(c3scnc3C(F)F)=O)C2)=O)[nH]nnc1C1CC1 55485,N1(C(C2C(C)C2C)=O)CCC(CNC(c2cn[nH]c2C(C)(C)C)=O)C1(C)C 55486,CC1CN(C(=O)CC(c2ccccc2F)C2CC2)CC(C)N(C(=O)C(C)(F)F)C1 55487,CCC(C)C(O)C(=O)N1CCCCC1CNC(C1(O)CC1)=O 55488,c1(CCC)cc(C(=O)NC(C)CC(C)NC(c2cn(C)nc2C2CC2)=O)n(C)n1 55489,C#CCCC(C(=O)OC)NC(c1ccc(CNC(C2CCOC2=O)=O)cc1)=O 55490,c1(C(N(CCNC(Cc2c(COC)cccc2)=O)C)=O)ccc(C)nc1N 55491,C1(C(=O)NC2C(CC)N(C(c3nccnc3N)=O)CCC2)CCC2CCC(=O)N12 55492,C1(F)(CNC(=O)CCF)CC2CCC(C1)N2C(=O)C=Cc1nccs1 55493,C(=O)(C(F)C(F)(F)F)N(CC(CNC(c1cccc(C(N)=O)n1)=O)O)C1CC1 55494,C(=O)(C1=NNC(=O)CC1)NCCN(C(=O)C(c1ccc(F)cc1F)C)C(C)C 55495,C=CCC(C(=O)NCCC1(CNC(=O)CN=S(C)(C)=O)CC1)C(C)(C)C 55496,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C2)SCCO1 55497,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55498,[N-]=[N+]=NCC1C(=O)NC2CCN(C2)CCOCC(=O)N1.C1(OC)CCCC1 55499,c1(C(=O)NC2CC(NC(c3cccc(Cl)c3)=O)C2)cnc(OCCO)cn1 55500,N1(C(CC(=C)C)=O)CCC2(CC1)CN(C(C1(C)CCC(=O)NC1=O)=O)C2C(C)C 55501,c1(OC)ccccc1Sc1oncc1C(=O)NCCc1cccs1 55502,c1(CC)cc(C(N2CCC(=CCNC(=O)C(C)N(C)C(C)=O)CC2)=O)c(C)nn1 55503,CCC(CC)C(C)C(=O)NC1CCN(C(=O)Cc2cccc3ccoc23)C1(C)C 55504,C1(C(=O)NC2CC(C#C)C2)COCCN1C(c1cnn(C(C)C)c1)=O 55505,C1(c2nnnn2C)(N(c2ccc(OC)cc2)C(C2CCCC2)=O)CCN(C)CC1 55506,c1(CC)c(NC)cnn1C(CC)CC.C(C(=O)ON)NC(C)C 55507,c1(C(N(C2CN(C(C=CCC)=O)CC2F)C)=O)ccc(=O)n(-c2ccccc2)n1 55508,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55509,N1(C(C2N(C(CCC3CCC(=O)C3)=O)CC(O)C2)=O)CC2CCC2(CO)C1 55510,CC1(C)CCN(C(=O)NC2CCN(C(=O)c3ccc4c(c3)CC4)O2)CC1 55511,c1(C(=O)NCC(=O)NCC(C)NC(CNC(CC)=O)=O)ccc([N+](=O)[O-])cc1Cl 55512,C(C(=O)N1OC2CCC1CC2)C1OCCN(C(=O)CC2CCOCC2)C1 55513,Cn1nc(Br)c2ccc(C(=O)NCC#N)cc12.N12C3CCC(C3)C1C2=O 55514,C(=O)(CC(CC)C(F)F)C(C(CC=CC)N)=O.C(C(C)(C)C(C)(C)C)CN 55515,CC1(C)C2CCC1(C(N1CCN(C(N3CCOCC3)=O)CC1)=O)CC2 55516,N1(C(C(CC)SC)=O)CCCCC(NC(c2cc(CN(C)C)on2)=O)C1 55517,c1(OC)cc(I)ccc1C(N1CCC(C(=O)NC(C2CCC2)C)C(O)C1)=O 55518,N1(C(c2ccc(SCC)cc2)=O)CCC(C)C(NC(C23CCN(CC2)C3)=O)C1 55519,c1(C(=O)NCC2(C)C(C)CN(C(c3ccn(C)c3)=O)C2)nnn2c1CSCC2 55520,N1(C(CCC2CCN(C)CC2)=O)CCOC2(CCN(C(C3CC3C(F)F)=O)C2)C1 55521,N1(C(CCC=C(C)C)=O)CCCC(CCNC(=O)CCSC(F)(F)F)CC1 55522,C=CCC(CNC(=O)CCc1cnco1)C(=O)Nc1ccccc1NC=O 55523,c1(C(C)C(=O)NCC(C2CC2)NC(C23COCC2C3)=O)c(Cl)cccc1Cl 55524,C1(NC(COC(C)(C)CNC(C2CCC(O)CC2)=O)=O)CC2(CCOC2)C1 55525,c1(C(N2C(CNCc3cnccc3Cl)CC(OC)C2)=O)ccc(=O)n(C)n1 55526,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55527,Cc1cc(C(=O)N(C(CNC(=O)CCOc2cccc(F)c2)CO)CC)c(C)n1C 55528,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CC2)=O)ccn2cnnc2c1 55529,Nc1nc(Cl)ccc1C(=O)NCC1CCCN1C(=O)CCOCc1ccccc1 55530,c1(NCCc2cnc(C)[nH]2)nc(N2CCCN(C(C)CO)CC2)nc2sccc12 55531,C(=O)(CCCCC(N)=O)N1C(CN(C(c2c(C)cccc2Cl)=O)C)CCCC1 55532,C(C(CC(F)(F)F)NC(C1(CO)CCOCC1)=O)NC(c1cnc(OCC)nc1)=O 55533,C(C)(CNC(=O)CNC(c1cscn1)=O)(CC(C)C)NC(c1ncc(C)nc1)=O 55534,C1(CCC(=O)NC(CSC)CO)CCCCN1C(c1ccsc1SC)=O 55535,Cc1coc(C)c1C(C1CC1)=O.C12CCC(C1)C(C(=O)NCCCO)N2C 55536,c1(NC(c2c(CNC(C(CC3CCC3)OC)=O)noc2)=O)cnn(C(C)C)c1C 55537,c1(OCC)nc(C(=O)NC(C)C(C)NC(c2ccn(C3CCOCC3)n2)=O)ns1 55538,c1(C(=O)NC2CN(C(CCNC(=O)Cn3cncn3)=O)C2)cccc(F)c1 55539,c1(SCC)cc(Cl)ccc1NC(=O)NC(c1cccc(Cl)c1)C(C)C 55540,N1(C(C(CC)(C)OC)=O)CCC(C2CCN(C(=O)Cc3c(C)noc3C)C2)CC1 55541,c1(C(=O)NCC(C)N(C(=O)CCc2cncn2C)C)ccc(SCC(N)=O)cc1 55542,C12(CNC(C(C)C3CCOC3)=O)CC(CO1)N(C(c1scnc1Cl)=O)C2 55543,C(=O)(CCC(C)C(F)F)N1CCC(C)(NC(c2ccc(C#C)cn2)=O)C1 55544,CC1(C)CN(C(=O)C#CC2CCC2)CCC1NC(c1n[nH]cc1C1CCC1)=O 55545,C#CCCN=C(NCCc1cnccc1O)NCC(O)CC(=C)C 55546,c1(C(=O)NCC(CC)NC(=O)CCOC)ccc(Cl)cc1-c1cccc(C)c1 55547,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55548,Cn1nnc(CNC(=O)CNC(=O)CC(F)(F)F)c1C(=O)NCC1(C)CCSCC1 55549,C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)NCc1ccc(C)s1 55550,C(=O)(C(CO)C(C)(C)C)NCC(CCC)C(=O)NC(c1cccnc1O)C 55551,N1(C(c2cccc(C)c2)=O)CCN(C(c2nccn2C)C2CC23CC3)C(C)C1C 55552,Cc1cc(F)ccc1OCCOC(C1CC2CC1C2)=O 55553,c1(C(=O)NC2C(C)CN(C(=O)CNC=O)C2)cccc(C#CCC2CC2)c1 55554,C12(C(=O)NCC(C)N(C(=O)Cc3cnns3)CC)CCCC1CCC2 55555,c1(-n2cc(C(C)(C)N(C)C)nn2)ccnc(C(=O)NC2CCS(=O)CC2)c1 55556,N1(C(CC(C)N(C)C)=O)CCOCC1CN(C(=O)CN(c1ncccn1)C)C 55557,c1(NCC(C)S(N)(=O)=O)ccc(S(=O)(=O)N2CCC(c3ccc(Cl)s3)C2)cc1Cl 55558,O=C1CN(CC2CCCCC2O)C(=O)N1CC1CCCCC1F 55559,CC(C)C(C(=O)NCC(C(C)C)NC(=O)COc1ccccc1)N(C)C 55560,C1(CCNC(C(C=C)(C)C)=O)CN(C(c2coc(N(C)C)n2)=O)CCCO1 55561,N1(C(C2(CCC)CC2)=O)CC2(CCC2NC(=O)Cn2cnnn2)C1 55562,C1(CC(C)NC(C(Cn2ccc(C)n2)C)=O)CCN(C(=O)C(=O)NC(C)C)CC1 55563,CCC(C)CC(C)C(=O)NC(CNC(c1ccccc1CO)=O)(CC)CC 55564,c1(C(N2CCC(NC(c3c(C)sc(C(F)(F)F)n3)=O)C2)=O)ccnc2ccnn12 55565,N1(C(C2CCCC(C)C2)=O)CCCN(C(=O)C=Cc2ccc(=O)n(C)c2)CCC1 55566,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)C=C2CCC(C)C2)C1 55567,C12(CNC(CSc3nc(C)[nH]n3)=O)CCCC1CN(C(=O)C(F)(F)CC(C)C)C2 55568,C(N=c1ccnc(NC(C2CCCCC2)CC2CC(F)(F)C2)[nH]1)c1c(C)cn(C)c1 55569,C1(C#N)(C(=O)NCCN(C(C2CCCS2)=O)CC)CC1 55570,c12ccc3c(c1)CCCC3C(=O)O2.c1(COC)cn(Cc2cccnc2)nn1 55571,C(N=c1[nH]cnc2[nH]c(C(F)F)nc12)C1CCCN(C(c2ccc(F)s2)=O)C1 55572,C=C=CC(C)C(=O)NCC(N1CC(CNC(=O)C(C2CCC(=O)N2)C)C1)=O 55573,Cc1nn(CC(=O)NC2CC(NC(=O)C(C)CN(C)C)C(O)C2)c(C)c1[N+](=O)[O-] 55574,c1(C(F)(F)F)[nH]c(=NCC2CCCC2c2c(F)cccc2)nc2c1CCC2 55575,c1(C(N2CCCC(CCNC(CC(C)F)=O)C2)=O)ccn2ncccc12 55576,CC(C)(CNC(c1cc(Cl)cs1)=O)CC1CN(C(C2CC2c2ccoc2)=O)C1 55577,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55578,C1(CCNC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(=O)CCSCC(C)C)C(C)C1 55579,c1(CNC(C(=O)Nc2cn(CCOC)nn2)=O)cccnc1O 55580,C1(CC=C)(NC(c2cnn(C)c2OC)=O)CCN(C(=O)CC2CC2C)C1 55581,C(=O)(C1=NN(C)C(=O)CC1)NC1CCCN(C(C2(OC)CC2)=O)C1.N1CCCC1 55582,C(CC(C)(C)C)(C(=O)NCc1cn(C)cn1)OC.C12(CC1)C(=O)N2C 55583,c1(C(N(C)Cc2ccc(C)cc2Br)=O)n[nH]c2cccc(F)c12 55584,C1(NC(c2n(C)c(O)nc2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)CCC1F 55585,Cc1ccc(C=CCNC(N2CCC(C(F)(F)F)(CN(C)C)CC2)=O)cc1 55586,C(CN=c1[nH]c(=NC2CCC(C3CC3)c3ccccc32)[nH]c2c1CSC2)N(CC)CC 55587,C1(CN(CCN(C(CN2CCC(CC)CC2)=O)C)C)COc2ccccc2O1 55588,CN1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC(F)F)C1 55589,CC(C(=O)N1CCC(CNC(c2cnc(Br)c(N)c2)=O)CC1)C(C)(F)F 55590,C(C(=O)NCC(C)N(C(=O)CN1CCC1)C)(C1CC1)SC 55591,C1(C)(C(=O)NC2(C)CN(C(C(c3ccc(F)cc3)(C)F)=O)C2)CC(C2CC2)=NO1 55592,N1(C(C(CC=C)C(=C)C)=O)CCC2(CCC2C(=O)NCc2cc(Cl)ccn2)CC1 55593,C(=O)(CC(O)CC(C)(C)C)NC1CCC(NC(C(C(C)C)n2cncn2)=O)CC1 55594,Cc1c(C(=O)NC(C)C(C)C)ccn1CC1CC1 55595,c1(C(N2C(CNC(CC(C)N(C)C)=O)CC3(CC3)C2)=O)cccc2nccn12 55596,C1(OC)CN(C(c2ccncc2)=O)CC1NC(c1ccc(-n2cccn2)nc1)=O 55597,N1(C(C2CN(C(C(CC)=CCCC)=O)CC2C)=O)CCOC(C2(C)N=N2)C1 55598,N1(CC(=O)NC(CC)CNC(=O)C(F)(F)c2cnnn2C)CCN(C)C(=O)C1 55599,N1(Cc2ccc(S(=O)(=O)NC)s2)CC2(CCN(CC(C)Cl)CC2)CC1C 55600,C=CCC(C)(C)C(=O)NC1CCN(C(c2cc(C(=O)OC)sc2C)=O)C1(C)C 55601,c1(COC(C)C)nc(-c2cc[nH]n2)nn1CC(C)(C)O 55602,C(COC)(C1CCC1)OC.C(=O)(C=CCN(C(C1CC1F)=O)C(C)C)NC 55603,Cc1cn2c(C(N3CCC(C4CC4)(CNC(C4CCOC4)=O)C3)=O)c(C)nc2s1 55604,N1(C(C2CC=C(C)CC2)=O)CCCC(CCNC(=O)C=CC(C)C)CC1 55605,C1(C(=O)NC2CC(C)(C)CN(C(C3CCCCS3)=O)C2)CNC(=O)CC12CCC2 55606,C1(C(C)NC(=O)C(F)Cc2ccccc2)CN(C(c2cnoc2C2CC2)=O)CCO1 55607,C(CC(C(=O)NCCC(F)CN=[N+]=[N-])NC(=O)CCc1cccn1C)OC 55608,Cc1c(C(=O)NCC(C2CCC2)NC(C2CSCCS2)=O)cnn1CCC(C)C 55609,Cc1c(C(=O)NCC2CCN(C(c3cc4c(s3)CCC4)=O)CC2C)sc2cncn12 55610,C1(C(=O)NCC(CC)OC)CN(C(c2ccc(CO)cc2)=O)CC(C)(C)C1 55611,C1(O)(CN(C(c2c(C(C)C)noc2)=O)C)CCN(C(=O)Cn2cnnc2O)C1 55612,c1(C(=O)NCCN(C(C2CC3OC(=O)OC3C2)=O)CC)nn(C)c2c1CCC2 55613,C1(NC(c2occ(C)c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55614,C(=O)(C1=NOC(C)C1C)N(CC(C)NC(C1(C(C)C)CCC1)=O)C 55615,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)c2ncco2)CC(C)(C)C1 55616,C1(NC(=O)COCC2CC2)CCC(NC(=O)Cn2cnccc2=O)CC1 55617,N#Cc1ccc(CN2CCOC(C(=O)Nc3ccc(Br)c(F)c3)C2)cn1 55618,c1(N2CCC(CC(C)NC(c3cc(O)n(C)n3)=O)CC2)nc2ccccc2o1 55619,N1(C(CCC2CNC(=O)N2)=O)CCC(NC(=O)CC2CCOC2)CC1 55620,C1(NC(c2n(CCC)nc(C)c2)=O)C2CCC1N(C(=O)CN1CC3CC3C1)C2 55621,CN1CC(N(C(=O)NCC2(CO)CCCCC2)C2CC2)CCC1=O.C1(C)C(=O)N1 55622,c1(C(=O)NCCC(C)NC(C(C)(C2(C)CC2)OC)=O)ccc([N+](=O)[O-])nc1C 55623,c1(C(=O)NCC(C)N(C)C(C2CCC(C)(C)O2)=O)cccc(O)c1F 55624,C1(CCC)(C(=O)OC)CCN(C(=O)CC2CC2Cc2ccccc2)C1 55625,N1(C(C=CCC)=O)CCC(C)N(C(c2cc3c(s2)CCCN3)=O)CC1 55626,c1(C(=O)NCC2CCN(C(c3cc(C(=O)OC)on3)=O)C2)noc2c1COCC2 55627,C1(C(=O)NC(CCC)CO)CN(C(c2ccsc2)=O)CCC1C 55628,C(=O)(CC(CCC)OC)NC1CCC(C(=O)NCC2(C#C)CCC2)O1 55629,C1(CC#C)(C(=O)NCC2CCN(CC)C2)CCN(C(=O)CC2CCCCC2)C1 55630,C12(CCCCO1)C(=O)N(C)CCn1cc(nn1)C2.C1(C(=O)O)CC(F)(F)C1 55631,C1(CCO)CN(N2CCc3[nH]nc(CO)c3C2)C1 55632,N1(C(C2(C)CC(C)(C)C2)=O)CCN(C(C2C=CCCC2)=O)C(CC(F)(F)F)C1 55633,c1(C(=O)NCc2cn(CCNC(CC=CC=C)=O)nn2)ccccc1C 55634,N1(C(=O)NCC2CC(C(=O)OCC)C2)CCC(C)=C(C)C1 55635,n1(CC)ccc(C(=O)NC2CC3(C2)CC3NC(=O)Cc2ccn(C)n2)c1C 55636,C1(OC(CC2CC(C)NC2)=O)CCC2(CCC2)C1 55637,n1(CC)cnc(C(=O)NC2CCCC2CNC(C23CCC2C3)=O)c1 55638,N(C(=NCc1cnc(C)cn1)NCC1CC1)CC1(CC)CCC1 55639,C12(CNC(c3c(C)ccc(N)c3)=O)CCC(NC(=O)CSS(C)(=O)=O)(CC1)CO2 55640,c1(C(=O)NCC2(CC)CC2)cnc2ccccc2c1N1CCC(C)(CO)CC1 55641,C1(NC(C2CCC3(CC2)N=N3)=O)CS(=O)(=O)C12CCN(C(=O)C(F)=CC1CC1)CC2 55642,CC1(C)C(C(F)(F)F)CCN1C(c1ccccc1C(N)=O)=O 55643,N1(C(C(C)OC(C)(C)C)=O)CCN(CC(=O)NCCCC(O)CO)CC1 55644,N1(C(C(=O)NC(=O)NCC(=O)OC)C(C)C2CCOCC2)CCS(=O)(=O)CC1C1CC1.C.O 55645,CCCCC(C)(F)C(=O)NCc1cc(C(N2CC(C(N)=O)(OC)C2)=O)on1 55646,c1(-c2cc(N(CC)CC)ncc2)c[nH]c2cc(C(=O)N(CCO)CCO)ccc12 55647,C(=O)(C(C)S(N)(=O)=O)N1CCC(NC(c2cc(SCC)ncc2)=O)(CF)C1 55648,c12ccnc(c1)N2.c1(C(=O)NCCNC(C2C(C(N)=O)C2)=O)ncncc1Cl 55649,C1(CN(C(=O)CC2CCCC2)CC)CCCCN1C(C1CSCN1C(C)=O)=O 55650,CCC(CC(=O)NCCCCNC(c1cnc(C2CC2)nc1)=O)C1CC1 55651,N1(C2CCN(C(=O)C=CI)C2)CCN(C(=O)C(C2CCCCC2)O)CC1 55652,c1(NC(C2CN(Cc3cnc[nH]3)C2)=O)ccc(I)c(Br)c1 55653,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 55654,c1(-c2cc(C)nnc2)ccc2[nH]c(C(=O)NC(c3ccc(Br)cc3)C)cc2n1 55655,C1(CNC(C2(OC)CCC2)=O)CCN(C(c2cccc(=O)n2C)=O)C12CC2 55656,C1(O)(C(N(C(C)CNC(=O)C(C2CCOCC2)F)CC)=O)CCC(C)CC1 55657,c1(C(N2C(CC)CN(C(=O)CCC(F)F)CC2)=O)cncc2cnccc12 55658,CCC(C)C(C(=O)NC1CC(CNC(=O)CN(S(=O)(=O)c2cccs2)C)C1)OC 55659,C1(C(N2CCC(CC=C)(NC(c3nsnc3O)=O)C2)=O)C2CCCCCC12 55660,C1(CN)CC2CCC(C1)N2C(c1ccc(F)c(C)n1)=O 55661,c1(CC(N2CCCC2CC(c2ccccc2)O)=O)ccc(C(F)(F)F)nc1 55662,c1(C(N2C(C(=O)NCC(CC)OC)CC(C)C2)=O)c(C)nn(C)c1C 55663,C=C(C)CN=C(NC1CCCCC1)N1CCC(F)(F)C(C)C1 55664,C1(C(=O)NCC2(CCNC(C3C(C=C)C3)=O)CC2)CC(=O)c2cc(Cl)ccc2O1 55665,c1(C(=O)NCC23N(C(C4(C(C)(C)O)CC4)=O)CC(C2)C3)cc2cccc(Cl)c2[nH]1 55666,c1(C(N2CC(NC(COc3c(C(N)=O)cccc3)=O)C2)=O)nccc2n[nH]cc12 55667,C(c1ccc(O)cc1)=CC(=O)NC1(C)CCN(C(C(C)OCC2CC2)=O)C1 55668,C1(CNC(=O)C=CCF)COCC1NC(c1cnc(Br)s1)=O 55669,c1(C(=O)NC2C(N(C(C(CC=CCC)C)=O)C)CCCC2)cc2sccc2n1C 55670,C1(COC)CN(C(=O)CCN(CCCO)C(c2cn[nH]c2)=O)CCO1 55671,C(=O)(CC(O)C(C)C)NCC1(OC)CN(C(c2ccnc(-n3cccn3)c2)=O)C1 55672,c1(N(c2ccc(C)c(C)c2)C)nccc2cc(NC(=O)OC(C)C)ccc12 55673,c1(COC)ccnc(C(=O)NCCC2CCC(NC(=O)CP(C)(C)=O)C2)c1 55674,C(=O)(C(O)(C(F)(F)F)CC1CCC1)NCC1(C)CC1 55675,C1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)CO)CCC(F)(F)CC1 55676,C1(CNC(c2c(C)nc(C)[nH]2)=O)CC(C(C)(C)C)CN(C(=O)CC(C)C2CC2)C1 55677,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3ccnn3)C2C(C)(C)C)CCCCC1 55678,CCC(C(=O)NCC1CCCC1NC(=O)C(C)(C)F)NC(C)=O 55679,C1(C(N2CCC(CNC(C(C(C)C)OC)=O)(OC)C2)=O)CCC(F)(F)CO1 55680,C(=O)(C1=C(C)CCCC1)NC1CCCCN(C(CCCC(=O)NCCC)=O)C1 55681,CCS(=O)(=O)C=CC(=O)NC1(CF)CCN(C(c2ccc3ncnn3c2)=O)C1 55682,C(C(=O)NC(c1cnn(C)c1)C(=O)NCc1cnn(C)c1C)(C(C)C)OCC 55683,CCCCCC(O)C(=O)N1CCCC1C1(NC(C2C(=C(F)F)CCC2)=O)CC1 55684,N1(C(CCC(C)OCC)=O)CCC(C)(C)C(NC(c2cncc(C(N)=O)c2)=O)C1 55685,Cc1nc2cccc(C(N3CCN(C(C4COC(=O)O4)=O)C(C4CC4)C3)=O)c2[nH]1 55686,N1(C(Cc2ccc(SCC)cc2)=O)CCC2CCC(C1)N2C(=O)C(C)NC(N)=O 55687,C1(CN(C(c2ccnc(O)c2)=O)CC)CCCN(C(=O)Cn2ncnn2)C1 55688,c1(CNC(C2CCC(C)(CC)O2)=O)nc2c(s1)CN(C(=O)COC(C)(C)C)CC2 55689,N1(C(C(C(CC)O)C)=O)CC2CN(C(=O)CCn3c(C)cc(O)cc3=O)CCC12 55690,C1(C(=O)NCCN(C(=O)CC2CC(=O)C2)CCC)CCOC(C)(C)C1 55691,N1(C(CC2(COC)CC2)=O)CC(C)CN(C(=O)Cc2c[nH]nc2C)C(C)C1 55692,C1(C(=O)NCC2CC2NC(=O)C(O)CSC)(OC)CCC(C)(C)CC1 55693,C(=O)(N=S(C)(=O)CCO)NC(CC)Cc1ccc(Cl)cc1 55694,c1(CN(C(=O)C(=O)NC2COCCN2C)C(c2ccccn2)C)cccc(Cl)c1 55695,c1(CNC(CCNC(C)=O)=O)occc1C(N1CCCC1C1CCOC1)=O 55696,C(=O)(CC1=CCCOC1)NCC(C)(C1CCC1)NC(CNC(c1cc(C)no1)=O)=O 55697,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 55698,N1(C(C(F)=CC)=O)CC2C(CC(=O)NC(c3ccncn3)C)C2C1 55699,N1(C(CC=CC=C)=O)CCC2CCN(C(c3cc(C(N)=O)co3)=O)C2C1 55700,N12CCN(CC1C)C(=O)CC1(CC1)C2.c12ccc(cc1)C(C)(C)C21CC1.CO 55701,Cc1cc(N)c(C)nc1C(=O)N(CCC(C(C)(C)C)NC(=O)CCc1ccsc1)C 55702,c1(-c2ccc(OCC)cc2F)nc2ccc(C(N3CCC(C(N)=O)C3)=O)cc2s1 55703,NS(=O)(=O)c1cncc(C(=O)NC23CCC2CN(C(C2CCCOCC2)=O)C3)c1 55704,N1(CCC)CC(C(=O)NC(C)C(C)NC(C2CCCN2C=O)=O)CC1=O 55705,N1(C(CCC#C)=O)CCC(C)C1CNC(=O)CCSc1nnnn1C 55706,CON(C)C(=O)C1(N(C(=O)Cc2nccs2)C)CC1 55707,C(C(CC(=O)NC1CN(C)CC1C)NC(=O)CCc1cscn1)OC 55708,C1(NC(=O)CN2C(=O)CCC2=O)CN(C(c2cncnc2)=O)C2(CCOC2)C1 55709,c1(CC)cccc(C(N2CC(OC)C(NC(=O)CCOCCOC)C2)=O)c1 55710,C1(C(N(C)CC2(O)CN(C(=O)CN3CCSCC3)C2)=O)SC2C=CC1CC2 55711,C1(C(=O)NC(CCCNC(C(C)SC)=O)C)OCCOC12CCC2 55712,Cc1coc(C2CC2)c1C(=O)NCCCCNC(C12CCCCC1C2)=O 55713,Cc1cc(C(c2nnnn2CC2CCCO2)Nc2cnoc2)c(Br)cc1F 55714,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 55715,N1(C(=O)NC(c2ccncc2)C)CCC(NS(=O)(=O)NCCC2CC2)CC1 55716,C1(NC(C2C(C(=O)OC)COC2)=O)CC2(CCN(C(C34CCC(CC3)C4)=O)C2)C1 55717,CCC(CCC(=O)N(c1ccccc1CCO)C)NC(C1CC(SC)C1)=O 55718,C1(C(N(C2CN(C)C2)C)=O)CC2CC2N1C(c1ccc(CO)s1)=O 55719,N1(C(c2ncc(CC)s2)=O)CCC(O)(C(C)NC(=O)CSc2cccc(F)c2)C1 55720,N1(C(C2N(C(C)=O)CCCC2)=O)CCN(C)CC1CNC(=O)Cc1coc(C)n1 55721,N1(C(CC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CNC(c1cccc(O)c1)=O)C2 55722,C1(C)(NC(COCCC(C)C)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1 55723,C(CCN(C)C)(C(=O)NC1(C(O)COC)CC1)NC(CC1CC(SC)C1)=O 55724,CC(C)C(C)(O)CNC(=O)C(C1(O)CN(C(c2cc(C3CC3)ccn2)=O)C1)F 55725,CC1CN(C(=O)CCc2ccnc(Cl)c2)CCC1NC(c1c(Cl)csc1Cl)=O 55726,C1(C(=O)OC)CCC(C(N2CCC(CNC(=O)CC=C(C)C)C2)=O)CC1 55727,N1(C(=O)C(Cl)=CCl)CC2CC1CN2C(C1(C(=O)NC2CC2)CC1)=O 55728,N1(C(c2c(CC)nco2)=O)CC(C)OC2(CCN(C(=O)CSCC(C)C)C2)C1 55729,c1(CCC)ccccc1C(=O)NCCOCCCN(C)C(C1COCCC1C)=O 55730,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CC(N3CC(O)C3)C2)=O)CC1 55731,C1(NC(c2cnccn2)=O)COC2(CCN(C(=O)CSCc3cccnc3)C2)C1 55732,C(N1CCC(OCCO)C(C)(C)C1)c1c(SC)cccc1 55733,c1(-c2nnc(N3C(C)(C)CC=CC3)n2CC2CCOC2)ccc2nc[nH]c2c1 55734,CCC(O)C(C)C(=O)NCC12CCC(C(N3CC4CCC4C3)=O)(CC1)C2 55735,C1(O)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCCSC)C)C1 55736,N1(C(c2c(COC)cc[nH]2)=O)CCC2(COCC(CNC(c3cccs3)=O)O2)C1 55737,Cc1ncc2n1CCCC2C(=O)N1CCN(C(=O)C(C)(C)C)CC1C(C)C 55738,N1(C(C(c2ccnn2C)C)=O)CC(NC(=O)Cc2nc[nH]n2)CC12CCCOC2 55739,C1(CCC(=O)NCC(CC)(C)NC(=O)COC(C)C)CCC(O)CC1 55740,N(C(=NCCn1cccn1)N1CCC(n2cncn2)C1)C1CC(OC)C1 55741,c1(NC(=O)NC)cccc(C(=O)NC(C)C(CO)NC(C2(C)CCCC2C)=O)c1 55742,S(=O)(=O)(c1ccc(F)cc1Cl)C(N(c1ccc(S(C)(=O)=O)cc1)C)=O 55743,N1(C(COCC#C)=O)CCC(C)C(CNC(=O)C=CCCC(C)C)C1 55744,C1(CC(=O)N(CCCN(C(CCOCCOC)=O)CCO)CCF)CCCC12CC2 55745,C12=C(Cl)N=CNC1=NCC1CC(CO1)CNC2=O.C1(C(C)C)CC(=O)N1 55746,C1(CC)C(C(=O)NCC2C=CC(NC(=O)Cc3cc[nH]n3)C2)CCN1C 55747,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 55748,N1(C(C(OC)OC)=O)CC(C)(C)OCC1CNC(c1nc(COC2CC2)cs1)=O 55749,C#CCCC(O)C(=O)NC1(COC)CCN(C(c2cccc(Cl)c2O)=O)C1 55750,C1(CNC(C2C(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)CC2(CCC2O)C1 55751,c1(C(N2CCN(C(c3cn(C(C)C)nn3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cc1I 55752,CCCC(C(=O)NC(C)CC(C)NC(c1c(Cl)ccnc1F)=O)C(C)C 55753,CC1=C(CNC(=O)CCn2cc(CCc3ccccc3F)nn2)CCC1 55754,c1(C(=O)NC2C(NC(C(C)=C3CCC3)=O)C2)cc(F)cc(Cl)c1O 55755,C(c1cc(C)cc(C)c1)=CC(N1CCC(NC(c2occ(OC)c(=O)c2)=O)C1)=O 55756,N1(C(C(C2CCCO2)OC)=O)CCCCC1c1cn(Cc2ccc(N)cc2)nn1 55757,CCCCC(CNC(c1ccc(CNC(=O)C(=O)NC2CC2)nc1C)=O)CC 55758,c1(C(C)C(N2CC(O)CC23CCC3)=O)ccc2ccccc2c1Br 55759,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccco2)C1 55760,CC1(C)CC(NC(C2CC3CC2C3)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)C1 55761,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 55762,N1(C(C2(CC#C)CCCO2)=O)CCCC(C)(NC(c2cc(O)nc(O)n2)=O)C1 55763,c1(NC(=O)NCc2cc(Cl)c(Cl)s2)ccc(-c2cnn(CC(O)CO)c2)cn1 55764,CC(CC(C)(C)C)C(=O)N(C)CCOCCNC(C1CCC1c1nncn1C)=O 55765,c1(C(c2nnnn2C(C)(C)C)NC(CCC)CCO)cnc2ncccn12 55766,c1(CNC2C=CC(C(N=c3nc(C)[nH]s3)=O)C2)ccc2c(c1)CCCCN2 55767,N1(C(CCSc2[nH]c(=N)sc2)=O)CC2CC1CCC2NC(C1(NC(N)=O)CC1)=O 55768,Cc1c(Cl)c(C(N2CC(C(=O)NCc3ccc(C#N)s3)CC2C)=O)nn1C 55769,C(=O)(CCCCC(F)F)NCC(c1n(C)cnc1)O 55770,N1(CC(=O)NC(CNC(CC2C(CC)C2)=O)C(C)C)CCNC(=O)C1 55771,c1(C(C)C)ccc2c(c1)C(NC(=O)C(N1CC3(CO)CCCC13)=O)CC2 55772,c1(C(N2CC(F)(C(=O)Nc3cn(CC#C)nc3)C2)=O)cnc(C)cc1C 55773,C(=O)(CCc1ccsc1)N(CCCOCCN(C(=O)CCNC(=O)C=CCl)C)C 55774,Cc1nc(C)c(C(N2CC(CO)(NC(=O)Cc3cc(F)ccc3F)C2)=O)nc1C 55775,CC(C)C(CNC(=O)CCCN(C)Cc1ccccc1)NC(=O)C(O)C1CCC1 55776,Cn1cc(S(N)(=O)=O)cc1C(c1ccccc1)NC(=O)C(=O)NC1CCCC(O)C1 55777,c1(OCC(=O)N(C)CCN(C)C(C2CC3CC2C2CC32)=O)ccccc1C#N 55778,CCCCC(O)C(C)C(=O)NC(c1cnn(C)c1)C(=O)NCC1(O)CC1 55779,c1(C(N(C2CN(C(Cc3cnc(C)o3)=O)CC23CC3)C)=O)ccn2cccc2c1 55780,C12(NC(C(=O)OC)CC3C4CCC(C4)N3C(=O)OC(C)(C)C)CCC(CC1)OC2 55781,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 55782,N1(C(CN(C2CCC3CC23)C(c2n(C)nnn2)=O)=O)CCC2(CCOC2)C(CO)C1 55783,C(N=C(NCC(C)(C)C)NC1CCN(C2CCOCC2)CC1)n1cc(CC)nn1 55784,C1(NC(c2cc(C)cc(C)c2)=O)CC2CC(C1)N(CCOCC(C)C)C2 55785,N1(C(C(N2CCCC2CO)C)=O)CCN(C)C(CNC(C2OCC2(C)C)=O)C1 55786,C1(NC(C(C)(C)c2cncnc2)=O)CC2CN(C(=O)CC3OCCO3)CC2C1 55787,C1(NC(=O)Cc2ccccc2)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 55788,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 55789,c1(C(=O)NC2CN(C(CS(=O)(=O)NCC)=O)CC2O)ccnc2cccnc12 55790,N1(C(COCC(C)C)=O)CC2CCCC2(CNC(C2CC(CN(C)C)C2)=O)C1 55791,O=C(C(F)C(F)(F)F)NCC1CC(NC(=O)C(c2ccccc2F)C2CC2)C(O)C1 55792,C1(C(N(CCCNC(Cc2cn(CC)nn2)=O)C)=O)CCC2(CC1)CC(O)C2 55793,C1(C(C)C)CN2CCCC2CN1C(=O)OCc1nnnn1CCSC(C)(C)C 55794,C(=O)(CCCCC#N)N1C(C(=O)NCC2(C)COCCO2)CC(F)C1 55795,N1(C(c2c(CC)cncc2)=O)CC(C(=O)NNCc2n[nH]c(CC)n2)CC(C)C1 55796,C1(C#N)(C(=O)NC2CCC(N(C(=O)CCS(N)(=O)=O)C)CC2)CC2C=CC1C2 55797,C(C(C(=O)NC(CN(C)C)C(C)C)NC(=O)Cc1ccsc1)OC 55798,c1(C(=O)NC23CCN(C(CCCNC(C)=O)=O)CC2C3)ncc2c(F)cccn12 55799,C=CCCC(C(=O)Nc1csc(COC)c1)NC(=O)CN(c1ncccn1)CC 55800,C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(=O)NCC1(C(C)(C)O)CC1 55801,C1(CN(C(Cc2c(C)nsc2)=O)C)CCCC(NC(c2cc[nH]n2)=O)C1 55802,C1(NC(c2ccc(COC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 55803,C(=O)(CCCCC(=O)OC)NC1C(CNC(CC(CC)CN(C)C)=O)CCC1 55804,C1(C(=O)NC2(C#C)CCOC2)CCC2(CC2)N1C(C1CN2CCN1CC2)=O 55805,c1(OC)ccc(CCC(N2CC=CC2CNC(C2CCCO2)=O)=O)cn1 55806,N1(C(C=CC)=O)CC(C(=O)NC2CC3CCN(S(=O)(=O)N(C)C)C23)CC(C)(C)C1 55807,Cc1cccc(Br)c1CN(C1(C(=O)NC(C)CC(C)O)CC1)C 55808,C=CC(C)(O)C(=O)NC(C1(CNC(c2csc(-c3cocn3)n2)=O)CC1)C 55809,CN1CCOc2cc(C(=O)NC3CCN(Cc4ccsc4)CC3F)ccc21 55810,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 55811,C1(CNC(C2CCN(C(=O)NC)C2)=O)CN(C(c2coc(Br)c2)=O)C(C)(C)C1 55812,C=CCCCCCCCC(C(=O)NC(C)C)N1CCc2ccc(F)cc2C1 55813,Cc1cnnc(O)c1C(N1CCC(O)(C(C)NC(=O)CC2CC3CC3C2)CC1)=O 55814,CC(CN=c1ncc(Cl)c[nH]1)NC(C1C2COCC12)=O 55815,C1(C(N2CCC(C(C(=O)N(C)CC3OCCN(C)C3)F)C2)=O)CC(C)(C)CN1C 55816,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 55817,CCCCC(C)(C(=O)NCCC1CCCCC1O)Nc1ccc(Cl)cc1C 55818,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nnnn2C2CC2)CC1 55819,Cc1ccc2c(CC(=O)NN3CCN(CC(=C4CCC(C)C4)F)CC3)c[nH]c2c1 55820,c1(CNC(=O)Cc2ccnn2C)ccoc1C(=O)NC(C)CC1CCCO1 55821,C(C1=C(C(=O)O)CCCC1)OC(CCC)C(=O)OC 55822,N1(C(c2c(CC)ccs2)=O)Cc2occ(C(=O)NCCN3CCCC3CO)c2C1 55823,N1(C(C2C(C)CCC2)=O)CCC2(CC(NC(c3cccs3)=O)C2)C1 55824,CC1CN(C(c2cn(CCNC(=O)CC3CCCC(=O)N3)nn2)=O)CC(=O)N1 55825,C(CCC(=O)NC1CC1NC(c1occc1Br)=O)N(C)C 55826,C1(NC(c2cc(CC)no2)=O)CC2CC1N(C(=O)C(C)(C)COCCOC)C2 55827,N1(C(C2(CO)CCN(C(c3cc(C)ncc3C)=O)C2)=O)CCCC12CCCOC2 55828,N1(C(CS(C)(=O)=O)=O)CCC(NC(=O)CSCCC#N)CC1C1CC1 55829,c1(C(N2CCC(NCC3CN(c4ncco4)C3)CC2)=O)ccn2ccnc2c1 55830,c1(C(=O)NC(CC)CNC(C2C3CCN(CC3)S2(=O)=O)=O)cc2cccc(C)c2s1 55831,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 55832,N1(c2n(C(COC)C)nc(C3CCC3)n2)C(=O)C2N(CCCC2(C)C)C1=O 55833,C=CCCCCC(=O)N1CCN(C)C(CNC(=O)CNC(=O)CCCCC)C1 55834,Cc1cc2c(cc1C)OC(C(N1CC3(CC(NC(=O)C4=CCCC4C)C3)C1)=O)C2 55835,C(=O)(C(C)C(=O)NCCc1cc(C(N)=O)no1)OC.c12cc(n(C)n1)C(=O)NC2 55836,c1(C(N(CCN(C(CSC(C)C)=O)C(C)C)C)=O)ccc2c(c1)COCCN2 55837,CC1CCC(C(N2CCC(CN(C(=O)C(C)(F)F)C3CC3)CC2)=O)CC1C 55838,N1(C(C2(NC(C3C(C)C3)=O)CCCCC2)=O)C2CCC1CN(C)C2 55839,N1(C(CC2(OC)CN(C(c3cnc(Cl)n3C)=O)C2)=O)CCC(C)(C2CC2)C1 55840,Cc1nc2n(n1)CC(C(=O)NCC1CN(C(c3ncccc3Cl)=O)CC1O)CC2 55841,c1(N)ccccc1Br.c1(CCNC(=O)Nc2cscn2)ccc(C(F)F)cn1 55842,CN1N=CC(CC(=O)NC2CC(NC(=O)CC3(C)CCCCC3)CC2O)C1=O 55843,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CCO)c1)CC)NCC 55844,Cc1ccc(CN2CCN(C(=O)NC3OCCC3(C)C(C)C)CC2)cc1 55845,CC1CCC(c2ccccc2)CN1C(=O)CC1CCN(CC2(S(N)(=O)=O)CC2)C1 55846,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ccnc12 55847,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CCC=CC(C)C)C2)cc1C1CC1 55848,C=C1CC2(C1)CC(C(=O)NCC1CN(C(C3CCN(C)C3)=O)CCO1)C2 55849,C(C(O)CC(=O)NC1CN(C(c2cncc(N(C)C)n2)=O)CC1F)N(C)C 55850,C(=O)(CCS(N)(=O)=O)N1CCC(NC(c2occ(C(C)=O)c2)=O)C1c1ccccc1 55851,C(=O)(CCCCN1CCOCC1)N(C(c1cccnc1)CC)C(C)=O 55852,Cc1ccc(C)c(CN(C)C(=O)NCC2CC(C(C)C)=NO2)c1 55853,c1(OC)cncnc1C(=O)NCC(=O)NC(C1CCCN1Cc1cccs1)C 55854,CC1(C)COC1C(N1CCCC1CCNC(=O)CCC1CCCCC1)=O 55855,Cc1scc(C(=O)NCC(N2CCC(NC(C3CC4C=CC3O4)=O)C2)=O)c1C 55856,N1(C(c2cccc(-c3cn(C)nc3)c2)=O)CCC2CCN(C(=O)C=CCF)C2C1 55857,C1(C(C)(C)NC(CN(C(C)=O)C)=O)CCCN(C(=O)CCc2cncnc2O)C1 55858,c1(CC(=O)N(C(C)CCNC(=O)CC2CCC(=O)N2)C)ccc(C(N)=O)cc1 55859,N(C1CCCc2cc(NC(c3ccc4cccnn34)=O)ccc21)C(COC)=O 55860,CC1CCN(C(=O)C(=O)NCC2CN(C(N)=O)C2)CC1.C12(C)CC1NC2=O 55861,C(=O)(C1=NOC(C)(C)C1)NCCOCCC(N1CCCC(N(C)CC)C1)=O 55862,c1(C(C)C)nnc(S(=O)(=O)NC(C2CCCOC2)C(=O)O)s1 55863,c1(CC)nn(C)c(Cl)c1C(=O)NCC1CCCCC1NC(c1ccncc1F)=O 55864,c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CC(=O)N(C)C)C2)cc(C)c1 55865,C1(CC(=O)NC(CCNC(CC=CCC)=O)(C)C)CCCC(C)(C)C1 55866,c1(OC)cc2cc(c1[N+](=O)[O-])N2.C(=O)(C(C)(C)C(F)F)NCC1CC(F)(CO)C1 55867,C1(CC)(NC(=O)C(c2cccc(C)c2)O)CCN(C(C2COCCC2C)=O)CC1 55868,c1(C(N2CCCC(O)(CNC)C2)=O)[nH]cc2c(=O)n(C)ccc12 55869,N1(C(C=CC(c2ccccc2)NC(C(C2CCC(=O)N2)C)=O)=O)CC2(C=CCO2)C1 55870,CCCCC(N)C(=O)N1CCC(C(N2CCOCC2)=O)C1 55871,N1(C(c2c(CC)non2)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)CCC2C1 55872,C1(NC(C=C=C(C)C)=O)CC12CCN(C(=O)C=C1CCC1)C2 55873,C1(NC(C(c2cc(C)oc2C)C)=O)CCCCN(C(=O)C(F)(F)c2nccs2)C1 55874,C1(NC(c2c(CC(C)C)onc2)=O)(CO)CCN(C(C2(C)C=CCC2)=O)CC1 55875,C1(NC(c2cc(CC)on2)=O)(CO)CCCN(C(C2(C)CCCO2)=O)C1 55876,c1(C(N2CC(C)(NC(CNC(C3N(C)CC(O)C3)=O)=O)C2)=O)ccc(F)cc1F 55877,C(=O)(C(F)(F)CC(C)C)N1CC(CC)N(C(=O)Cc2c(F)cccc2Cl)CC1 55878,c1(C(=O)NC(CC)CN(C)C(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 55879,C1(NC(CCSCC)=O)CCCCC1NC(=O)C(C(C)C)NC(c1cccs1)=O 55880,C1(NC(=O)Cn2nc(O)ccc2=O)CC1C1CCCN(C(=O)CCOC2CC2)C1 55881,C1(C(N2CC(=C(CNC(C(C)(C)OC(C)C)=O)F)C2)=O)CC(C)(C)SC(C)(C)C1 55882,N1(C(C(C)=C(CC)C)=O)CCCCC1CN(C(=O)CCc1cnn(C)n1)C 55883,N1(C(CCCSC)=O)CC(CNC(C23CSCC2C3)=O)C2(CCC2)C1 55884,C(=O)(C1=CCCCC1C)NC(C(C)C)(C)CNC(=O)CC1CCOC1 55885,C(=O)(CS(=O)(=O)c1cccc(F)c1)NCC1N(C(=O)OC(C)(C)C)C2(C1)CCC2 55886,c1(C(=O)NCC2CC(CF)CO2)ccc(C(=O)NCCCNC(C)=O)cc1 55887,C1(OCCN(C(N(C(C)=O)C)=O)C)CC1C(F)(F)F 55888,c1(N(C)C)ccc(C(N2CCC(CNC(C3CCCSS3)=O)C2)=O)cc1F 55889,Cc1nnc2n1CC(C(=O)OC1CCC1)CC2 55890,O=C(N=S1(=O)CCNC2CNCC12)NC1CCCC1C1CC1 55891,c1(C(N2CC3C(CNC(CN(S(CC)(=O)=O)C)=O)(C3)C2)=O)nccc(Cl)c1C 55892,C(=O)(CCCCNC(=O)NC1CCC1C(F)F)N(CCOCC)C 55893,N1(C(n2ccc(OC)c2)=O)CCC(CC(=O)NC)C12CC2.N1CC(OCC)C1=O 55894,N1(C(c2ccsc2Cl)=O)CCOCC1CCNC(C12CCC(C1)C2)=O 55895,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCC)=O)C 55896,c1(OC)noc(C(N2CCCC2C(C)NC(c2cnc(Cl)n2C)=O)=O)c1Br 55897,c1(C(=O)NCC(C(C)C)NC(=O)Cc2ccc(C(N)=O)cc2)cc([N+](=O)[O-])n[nH]1 55898,C1(C(=O)NC(C(C)(C)SC)=O)CCN(C(=O)C2(CO)CC3(CC3)C2)O1 55899,C(CC(=O)NCc1ncn(C2CC2)n1)(CC)NC(C1(CSC)CC1)=O 55900,C1(CNC(COCC)=O)CC(C(F)(F)F)CCN1C(C1CC12CC(C(=O)OC)C2)=O 55901,c1(CN=C(NCN2C(C)CSCCC2)NC2CC2)c(Br)ccc(Cl)c1F 55902,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 55903,C(=O)(C(C)CN1CCOCC1)N1CC(CC(C)NC(c2noc(C(F)F)n2)=O)C1 55904,Cc1c(C(=O)Nc2nnc(C3CC3)s2)cccc1CO 55905,C1(NC(C2CC3(CCC3OC)C2)=O)CCN(C(C2C=CCS2)=O)C12CC2 55906,c1(OC)ncc(C=CC(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)cn1 55907,c1(CCC)ccc2c(N)c(C(N3CC(C(=O)OC)C3)=O)sc2n1 55908,c1(C(N2CCN(C3CCCC3)C(C)C2)C(=O)NCC)cc(N(C)C)cc(Br)c1 55909,C(=O)(CC=C(Cl)Cl)NCC1CCCO1.C12(C(=O)OC(C)(C)C)CC1CNCC2 55910,N1(CCN(C(CCC)C)CC)CC(C)OC(C)C1 55911,n1(CC)cc(CN(C)C(C2CC(NC(=O)C(C)CO)C2)=O)nn1 55912,CC1CC(C(N2CCN(C(=O)CSc3nc[nH]n3)C(C3CCCC3)C2)=O)CC(=O)N1 55913,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)F)C2)=O)CC1C 55914,N1(C(CC(C)CF)=O)C2CCC1CC(N(C(=O)C(N1CCCC(C)C1)=O)C)C2 55915,CC(CCCCNC(=O)CCn1cccnc1=O)NC(=O)C(O)CNC(N)=O 55916,C(=O)(C(C)(C)CO)NCC(C1CCCC1)NC(C(C)CN(c1ccccc1)C)=O 55917,C1(NC(C2(CNC(c3n(C(C)C)ccn3)=O)CCC2)=O)CCCC(C)CC1 55918,c1(C(C(=O)NC2CC2)N(CCC)CC2CC2)cnc(C(C)C)s1 55919,CC1CCCc2nc(C(=O)NCC(F)CNC(c3n[nH]cc3[N+](=O)[O-])=O)cn21 55920,CC1CC(NC(=O)CC=CCNC(=O)CCCC(F)c2ccccc2)CCN1C 55921,C=C(C)CC(C)C(=O)NC(C)(C)CN(C(=O)C(Cl)=CCl)CC 55922,C(=O)(CC(C(F)(F)F)c1ccccc1)NC(CCOC)CNC(=O)CSC1CC1 55923,CCCC(CC(C)C)C(=O)NC(C)CNC(=O)C(C)(C)Oc1ccccc1OC 55924,CC1CN(C(=O)CC2SC(=N)NC2=O)CCC1NCC1CCC2(CC1)N=N2 55925,Cc1cc(=O)oc(C)c1C(=O)OCCc1ccc(F)c(F)c1 55926,C1(C(=O)NC2C(C)CN(Cc3cccc(CO)n3)CC2)C2Cc3ccccc3C12 55927,C(=O)(CC(C)CC(=O)NC1CN(C(c2ccc(C3CCC3)cc2)=O)CC1C)OC 55928,c1(C(=O)NC(C)(C)CCCNC(=O)COC2CCC2)ccc(OC(F)F)nc1Cl 55929,C(=O)(C1=C(C#N)CCC1)N1CC(C(C)(C)O)(CNC(c2cc(CC)nnc2C)=O)C1 55930,c1(OC)c(CC(=O)NC2CCC(C(N3CCOC(O)C3)=O)CC2)cccc1Br 55931,c1(CC)cscc1NC(=O)C(C)(C1CC1)N(C)C(C1CCOCC1)=O 55932,C=CCCCCCCCC(C(=O)NC1CCCNC1)C1CCCC1 55933,CC(CCC(=O)N(C(C)C(=O)NC(C)(C)C)C)N(C)C 55934,CC(C)CCCCC(=O)NC1C=CCN(C(c2ccn(C(C)(C)C)c2)=O)C1 55935,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 55936,N1(C(CCOC)=O)C(C(=O)NCC2CCC(C)(C)CC2)CCC12CC2 55937,CCC(CNC(=O)CSC(F)(F)F)(CC)NC(=O)CSC1CCCCO1 55938,C1(CCCCC(N2CC(C)(CC)C(F)(F)C2)=O)CNCCC12CCOCC2 55939,C1(O)(CNC(CC2C(C)CC2)=O)CCN(C(C2(C(F)F)CC2)=O)C1 55940,N1(C(Cc2n(C)nnc2)=O)CC(NC(=O)Cn2cc(CO)nn2)C2CCCC2C1 55941,c1(CC)nc(C(=O)NC2CC(CNC(=O)C(c3ccccc3)O)C2)c(C)o1 55942,N1(C(c2ccc(Cl)cc2)=O)CC2COCC2(C(N2CCCCC2C(F)F)=O)C1 55943,c1(OC)cc(Br)c(C)cc1NC(C1CCN1Cc1cc(F)c(Br)cc1Cl)=O 55944,N1(C(C(C)SC)=O)CC(O)(C2CCN(C(c3cc4c(s3)COCC4)=O)CC2)C1 55945,CCC(CC(C)C)C(=O)NCCNC(=O)C(c1ccccc1)OC(C)C 55946,c1(N(C)OCC)nnc(SC)n1CCOc1ccccc1 55947,CCCCN=C(NCc1ccc(OC)cc1F)NC(c1ccsc1C)C 55948,N1(C(C2=NOC(C)C2)=O)Cc2ccccc2C(CNC(c2ncc(F)cn2)=O)C1 55949,N1(C(c2c(=N)cc[nH]c2)=O)CCC2CCN(C(=O)CN3C(=O)CNC3=O)CC12 55950,CC(C)CC(C(=O)N1CCC(O)(CN)CC1)NC(=O)C(c1ccccc1)F 55951,C1(CNC(c2ccc(SC(CC)C)cc2)=O)CC2(CCN(C(C)=O)CC2)C1 55952,C1(n2cc(C3(C(C)=O)CC3)nn2)CCCN(C(=O)SC2CCS(=O)(=O)C2)C1 55953,C(C(=O)NC1CCCCC1NC(=O)CC(C)O)(C(C)C)(C(C)C)NC(C)=O 55954,N1(C(c2cnn(CC(F)(F)F)c2)C(=O)NC)CCC(C)CC1C(F)(F)F 55955,CCC(C)(CO)C(=O)NCC(C1CCN(C(c2ccc(F)o2)=O)CC1)(C)O 55956,C1(CNC(=O)Cc2ccc(C3CC3)nc2)CC2CCC1N2C(=O)CC1CCOC1 55957,CC(C)CCC(C(=O)NCc1cccc(Cl)c1)NC(C1CC(OC(C)C)C1)=O 55958,c1(OC)cc(NC(=O)CC2CN(Cc3ccccc3C(C)C)CCO2)cc(O)c1 55959,c1(C(=O)NCC2CC(CNC(C(C)NC(CC)=O)=O)C2)ccc(Cl)cc1 55960,c1(NC(C)=O)ccc(F)cc1C(N1CC2CCC1C2NC(=O)CC1CCCC1)=O 55961,C1(CNC(c2nnc(N3CCCC(CO)C3)s2)=O)C(C2CC2)CCN1CC=C 55962,C1(C(=O)Nc2ccc(COC)cc2)CCOCCN1C(c1cnn[nH]1)=O 55963,c1(C(C(=O)CCCC(N)=O)=O)cc(C)cc(N2CCOCC2C)n1.CCO 55964,C(=O)(C(CC(F)F)NC(=O)CCCCOC(C)=O)N1CC(CC)OCC1 55965,N1(C(C=NOC)=O)CCC(CO)C(NC(c2nnc(C)cc2O)=O)C1 55966,CCCCC(O)C(C)C(=O)NCC1(C)CCN(C(c2nsc(OCC)n2)=O)CC1 55967,c1(C(CNC(=O)CCCC2CC2)NC(c2c(CCC)nco2)=O)ccccc1F 55968,c1(COCC)ccc(C2(CC3(NC(c4cc(O)n[nH]4)=O)CCC3)CC2)cc1 55969,c1(CC)ccc(C(=O)N(C(C)CNC(=O)C#CC2CC2)C)cc1OC 55970,N1(C(C(CCC)N(C)C)=O)CCN(C(=O)CS(=O)(=O)CC)C2COCC12 55971,c1(N2CCC(O)(N(c3cccc(Br)c3)CC)CC2)cc(-n2cccn2)n2nccc2n1 55972,C1(C(N(CCCNC(C2(OC)CCC2)=O)CCO)=O)OCC2COCCC12 55973,C1(C(N2CCC(CCC)C2)=O)CN(C(=O)CCNC(C)=O)C(C)(C)C1 55974,c1(OC)cc(C2(C(=O)NCC3(NC4CCCC4O)CCOC3)CC2)ccc1C 55975,c1(CN(CC(CO)S(C)(=O)=O)CC)nc(C)n(C)c1C.c1(C2C(=O)N2)ccccc1 55976,N1(C(CCCC#C)=O)CCC(NC(=O)CC2CCCN(C(C)C)C2)C1(C)C 55977,CCC(C)(C)C(C(=O)NCC1(OC)CCN(C(c2csc(C#N)c2)=O)CC1)OC 55978,C1(CNC(CC(C)N2CCCC2=O)=O)CCN(C(C2CCC(=O)N2)=O)C(C)C1 55979,c1(C(C)C)ccc(F)cc1C(N1CC(NC(C2(S(N)(=O)=O)CC2)=O)C1)=O 55980,C1(C(N(C(c2ncccc2C(F)(F)F)C)C)=O)CCc2ccncc2C1 55981,N1(C(C2=C(C)OCC2)=O)CC2(CCC(NC(c3ccncc3F)=O)C2)C1 55982,c1(SCC(=O)N(CC)CC)ccc(OCC)cc1.C1(C)C(C)N1 55983,N1(C(C(N2CCCC(O)C2Cc2cccs2)=O)=O)CC2(C1)OCC1CC21 55984,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSC2COC2)C)=O)c1 55985,N(C1CCNc2ncccc21)C(CCn1cc(C(=O)OCC)nc1)=O 55986,c1(C(=O)NC(C)C(C(C)C)N(C)C)ccc(N2CC(C(C)=O)CC2=O)cc1 55987,C1(NC(N2CCN(C(c3ccccc3)c3ccccc3)CC2)=O)CC2(CSC2)C1 55988,N1(C(C)C)CCCC(C(=O)N(CC(C)CNC(=O)CCC(N)=O)C)C1 55989,C1(C(=O)NC2(CC)CC2)C2CC1N(C(c1cnc(CC3CC3)s1)=O)C2 55990,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 55991,C1(O)(CC)CCN(C(=O)C(C)(C)NC(C2(CSC)CCC2)=O)CC1 55992,C1(CC)(NC(=O)COc2cccc(C)c2C)CCN(C(c2sccc2C)=O)CC1 55993,CCC(CC(=O)NCC1C2CN(C(=O)CC3CC4(CCO3)CC4)CC12)C(C)C 55994,c1(C(=O)NCC2(c3cccc(C4OCCO4)c3)CCC2)cncc2n[nH]cc12 55995,C1(NC(c2cc3c(s2)CCCC3)=O)CC(C2CCN(C(C3CCCC3)=O)C2)C1 55996,C1(OCC(=O)NCCCN(CCCNC(C2CC2CSC)=O)C)CCC(F)(F)CC1 55997,C(C)(C)(CN=c1[nH]nc(C#N)s1)C1CCN(Cc2oc3ccc(C)cc3c2)CC1 55998,C12(NC(=O)COC3CC3)CCCC1(C(F)(F)F)C2 55999,Cn1cc(CC(O)CNCCNC(=O)OC(C)(C)C)nn1 56000,c1(OC(CNC(=O)C(C)(C)c2ccns2)C)ccccc1F.CC1CN1C1CC1 56001,CC1CC(NC(=O)C(C)(C)CN(C)C(C2CCOC(C)C2)=O)CC(C)O1 56002,N1(C(C=CC=CC)=O)CC(NC(=O)Cc2cccc(OC(F)(F)F)c2)CC(O)C1 56003,N12CC3NCC3(C1)C2=O.Cn1nc(C(F)F)cc1N1CCCC1 56004,C(=O)(C(F)(F)C(F)(F)F)NCC(CN(C(C1CCCN(C(=O)NCC)C1)=O)CC)O 56005,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56006,C(CN=c1[nH]c(=NC(C)c2cc(Cl)ccc2F)c2[nH]ccc2[nH]1)NC(=O)OC 56007,c1(OC(C)C)cc(NC(C2CCC(C)(C)CO2)=O)cc(C#N)c1 56008,c1(C(=O)NCC(c2cccc(Cl)c2)O)cc(Cl)c([N+](=O)[O-])s1 56009,n1(CC)cc(C2CC(C(=O)NC(C)CN(C(=O)CC3CC3N)CC)C2)cn1.C(C)(=O)OC 56010,N1(C(CCc2cc(C)no2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56011,c1(OCC)ccc(C(=O)NC2CC2C(=O)NCc2ccc(Cl)c(Cl)c2)c(OC)c1 56012,c1(C(N2CC(C(=O)Nc3nccs3)C2)=O)cc(Cl)cc(Cl)c1O 56013,C=CCC(C(=O)NC1CC1NC(=O)CN=c1[nH]c(C)cs1)C(C)(C)C 56014,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(CNC(CCc1c(C)cccc1)=O)(C)C 56015,C1(C#CC(=O)N2CC(O)CC2NC(=O)CCc2cnn[nH]2)(CC)CC1 56016,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56017,N1(C(COCCC)=O)CC(NC(c2cnc(OC(F)(F)F)cn2)=O)CC2(CC2)C1 56018,c1(C(=O)Nc2ccc(F)c(F)c2F)n[nH]c2c1CN(Cc1cnc(C3CC3)s1)CC2 56019,C1(C(NOC(C)C)=O)CCC(NC(=O)CSCC#N)CC1 56020,Cc1cncc(C(=O)NCCC(C)CCNC(=O)C(F)CC2CCC2)c1 56021,CC1=C(Br)CN(C(=O)NC(c2cccnc2)C(F)F)CC1 56022,c1(CC(=O)NC2CCC(CNC(C(F)=CC)=O)C2)cccc(C)c1Cl 56023,c1(OC)cc(Cl)c(CN2CCN(C(C3CCCN3C)=O)CC2C(C)C)c(Cl)c1 56024,c1(C(=O)NC2(C)CCN(CC(=O)NS(C)(=O)=O)C2)ccc(F)c(F)c1F 56025,c1(SC)cc(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CCCC34CC4)C2)c(C)o1 56026,c1(C(=O)NCC(C)(CO)NC(CCC(C)C#N)=O)ccc2cc(O)ccc2n1 56027,C1(C(=O)NCC(C)CNC(c2ccc(O)nn2)=O)CCCCCS1(=O)=O 56028,Cc1cc(NC(=O)COCCNC(C2CC3(C2)CC32CC2)=O)c(F)cc1F 56029,CON1CCC(C(=O)NCC2CCN(C(C3(CCS(N)(=O)=O)CC3)=O)C2(C)C)CC1 56030,C1(=O)CS(=O)(=O)CC(=O)C(NC(COC(C)=O)=O)CCN1 56031,CC1CC(C(=O)NCC2CCN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56032,C1(C(=O)NCCC(O)C(=O)NC)(CC)CCCN(C(=O)Cc2cccc(F)c2)C1 56033,N1(C(c2cc(C)nc(C(C)C)n2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 56034,C1(C)(NC(c2cncc(C(C)C)c2)=O)CCN(Cc2cccc(O)c2Cl)CC1 56035,N1(C(CCCC=C)=O)CCCC(C2CCN(C(c3cncc(C)c3)=O)CC2)CC1 56036,C(C(C)(C)CN(C)C(C1CCCN1C(=O)CCc1nncs1)=O)N(C)C 56037,Cc1cnc(C(=O)NC(CC(F)F)C(=O)N(C)CC2(O)CN(C)C2)cc1C 56038,C1(NC(C(C)OCCOC)=O)CCN(C(=O)CCF)CCC1CO 56039,c1(C(=O)NC(C)C(CO)NC(=O)C=Cc2ccccn2)cc(Cl)ccn1 56040,N1(C(C2NCCN(Cc3ncn(C)c3)C2)=O)CCC2(C1)NC(=O)NC2=O 56041,N1(C(c2c(CC)n[nH]c2)=O)CCN(C(=O)C(COC)OC)CC1CC 56042,Cc1cncc(C)c1C(=O)NC1CCC(C)(CNC(=O)Cn2cc(C(C)O)nn2)C1 56043,CC1CC(N(C(=O)C(c2ccccc2)NC(=O)CCc2cccs2)C)CCO1 56044,C1(NC(CCC#CC)=O)CCN(C(=O)Cc2c(C)cnn2C)CC1C 56045,C1(O)(CCCC)CN(C(=O)COc2ccon2)C1.C12CC(C1)C(=O)N2C 56046,C1(OC)CCC(C(N2CC(NC(c3cnn(CCC(C)C)c3)=O)C(O)C2)=O)CC1 56047,c1(OC)cc(CN(CCCNC(c2csc([N+](=O)[O-])c2)=O)C2CC2)c(OC)cc1C 56048,CCC(C)(CO)C(=O)N1CC2(CCN2C)C1 56049,CCCCCC(F)C(=O)NC1CC=C(C(=O)NC2(C)CCC(O)CC2)C1 56050,C1(NC(CCC=CC(C)C)=O)C(C)CCN(C(=O)CC(Cl)Cl)C1C 56051,c1(C(=O)OC)ccsc1-c1cn(C(C)CNC(=O)C(C)(C)N2CCOCC2)nn1 56052,CC1CN(C(=O)CCC2CCCN2C(C2CC23CCCCC3)=O)Cc2c[nH]nc21 56053,C(CC(C)C(=O)N(C(C)C(=O)N(C1CC(C)(C)C1)C)C1CC1)=CCC 56054,CC(O)CC(C)(C)CNC(C1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F)=O 56055,c1(C(=O)NC(CC)CN(C)C(c2coc(Cl)c2)=O)ncc2[nH]ncc2n1 56056,Cc1ncccc1NC(=O)C(C)CNC(=O)C(O)C1CCC1 56057,C(C(=O)NCSc1ccccc1)(C(C(C)C)OC)N1CC(C#CC)C1 56058,N1(C(CC(=O)OCC)=O)CCC(C(=O)NC2CCC(O)C(F)C2)C(C)C1 56059,C=CCCC(c1ccccc1)NC(=O)NCc1ccn(C(F)(F)F)c1 56060,c1(C(=O)NCC2N(C(c3c(SC)cccc3)=O)CCC2)ccc2nc[nH]c2c1F 56061,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CCC)on2)=O)C12CC2 56062,c1(C(N(C)CC2CCCN(C(COC(CC)CC)=O)C2)=O)cc(C)ccc1N 56063,c1(N2CCC(NC(C3N(C(C)C)C(=O)CC3)=O)C(F)C2)ncc(C#N)cc1Br 56064,C(CCCCC(=O)NC1CC(CC(=O)NCC(=C2CCCCC2)F)C1)SC 56065,c1(OC)cccc(CN(C(=O)C(F)(F)CNC2C(C#N)C2(C)C)C)c1 56066,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56067,CC1CC2CCN1SCC(=O)N2.c1(Cc2nncs2)nnc(-c2ccccc2)o1 56068,c1(SCC(N2C(C3CCN(C(COC)=O)C3)CCC2)=O)ccc2c(c1)OCCO2 56069,C1(C)(C(=O)NC(CNC(c2ccc(SCC)nc2)=O)(C)COC)CC2C=CC1C2 56070,Cc1ccnc(CNC(=O)CC2CN(C(c3cc[nH]c(=N)n3)=O)CC2C)n1 56071,C=CC(C)(C)C(=O)N1CCC(CCCCCNC(=O)Cc2cc(C)n(C)n2)CC1 56072,c1(CO)cccc(-c2cc(C(=O)NC(C(=O)NC)C(C)C)ccn2)n1 56073,C1(CCNC(CCCNC(=O)OC)=O)CCCCN(C(=O)CSC(C)C)C1 56074,C1(F)(C(=O)OCC)CN(C(=O)CC(c2cccc(F)c2)O)CC12COC2 56075,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(OC)C1 56076,c1(C(N(CC(C)NC(C(CCCOC)C)=O)C)=O)cccc2c1OC(C)(C)CC2 56077,Cc1csc2c(C(N3CCCCC3C3CC3)C(=O)NCc3ccco3)cccc12 56078,C1(C(=O)NC(CN(C(c2c(C)nc(C(F)(F)F)o2)=O)C)C)CCCCC12CC2 56079,c1(CN2CCCC(N(C(c3nc(C)c(C)s3)=O)CC)C2)nc(C)ccc1F 56080,C(=O)(C(F)CC(C)C)N(C)CC1(O)CCN(C(C)=O)C1 56081,C12(C)CCN(C1)C(=O)CC2.C1(C2CC2OCC(=O)N(C)C2CC2)CC(C)(C)C1 56082,c1(C(=O)NC(CNC(c2cc(C(=O)OCC)ncc2)=O)CO)ccc(=O)n(C)n1 56083,N1(C(C2C(CC)N(C(C3CCC(C)(C)C3)=O)CC2)=O)CC2(CCC1CO)CC2 56084,C(N=c1[nH]c(=NCC(=O)N=c2cc[nH]cc2)[nH]c2c1CSC2)C1OCC(C)(C)OC1 56085,Cc1cc(N(C)C)c(CSc2cccc(Cl)c2Cl)cc1Cl 56086,N(C(=NCc1nnnn1C)NCCCCOCC1CCOCC1)C(C=C)C 56087,C=C(CNC(=O)Cc1ccsc1)CCNC(C1CCN1C(C)=O)=O 56088,C=C(C)C(C)(C)C(=O)NCC1CCC(F)(CNC(=O)COCP(C)(C)=O)CC1 56089,c1(OC)cc(C(=O)NCC=CCNC(C2CC(C(N)=O)C2)=O)cc2c1OCCO2 56090,c1(C(=O)NCC(C)CNC(=O)CC(C)N(C)C)cc2cc(Cl)c(Cl)cc2[nH]1 56091,C1(NC(CC2(OC)CCCC2)=O)CCN(C(=O)CC(C)N(C)C)CC(O)C1 56092,c1(C(N2CC(NC(C(C)CC(N)=O)=O)(CO)C2)=O)cc(F)c(F)cc1O 56093,N1(CC(N2CCC(OCCC)C2)=O)CCCC(NC(c2ccon2)=O)C1 56094,c1(C(=O)NCc2n(C)ccc2)cc2sccc2cn1.C12(C)CCC(CC1)C(=O)N2 56095,c1(N(C(c2ccco2)=O)CC)ccccc1C 56096,C(=O)(CCCCCC(C)(C)C)N1C(CNC(=O)C=Cc2nccs2)CC(COC)C1 56097,Cc1cnsc1C(=O)NC1CCC(NC(=O)Cc2nc(-c3ccccc3)cs2)C1 56098,N1(C(C(CCC)C(=O)N(C(C)C(=O)OC)CC#C)=O)CC(S(C)(=O)=O)C1 56099,c1(C(N2CC=CC(NC(C(C=C=C)C)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 56100,N1(C(c2cncc(C3CC3)c2)C(=O)NC(C(=O)OC)C)CCC(O)C2CCCCC12 56101,C1(CC)CN(C(C2C(CNC(=O)Cc3cc[nH]n3)CCC2)=O)CCC1CO 56102,CCCC(C(=O)N(C)CCOCCNC(=O)C(c1ccccc1)F)N(C(N)=O)CC 56103,c1(NC(C2CCCCN2C(=O)CN2CC(F)C(F)C2)=O)cnnc(Cl)c1 56104,C1(NC(CN(C)Cc2nnc(C)n2C)=O)CC2CCC1(NC(=O)C(C)O)C2 56105,N12CC3CC(C1)CN(C3)C(=O)CC(CN(C)C)CC2=O.C#CC1CNCCN1C 56106,Cc1ccccc1N=c1[nH]c(SC2CCN(C(=O)OC(C)(C)C)C(C)(C)C2)cs1 56107,c1(NCC2(CNC(CCCC(=C)C)=O)CC23CCC3)nc(C)c(C)c(C)c1C#N 56108,Cc1nc2sccn2c1C(=O)NC(C1CCCN1C(C1COCCO1)=O)(C)C 56109,CC1(C(=O)NCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2)C1 56110,c1(C(=O)NCC(C)CNC(=O)CC23COC(CN(C)C)(C2)C3)ccc(P(C)(C)=O)o1 56111,c1(C(=O)NCC2(O)CC2)nc(C2=CCC(O)CC2)c2ccccn12 56112,c1(C(N(C2CCCN(C(=O)C(F)=CCCF)C2)CC)=O)cnc(C2CC2)nc1O 56113,CCN=c1ccc(C(=O)NCCCNC(=O)CSc2nncs2)c[nH]1 56114,c1(CCC)nccn1CC(=O)N(CCNC(C1CC(n2cnnc2)C1)=O)C1CC1 56115,C12(CC)CCN(C1)C(=O)C(CO)OC(=O)CCNC2=O.C(C)(C)C 56116,N1(C(c2c(CC)nccn2)=O)CCN(C(=O)C(C)CCOC)C(c2cn[nH]c2)C1 56117,C1(C(=O)NCCC(C)NC(c2c(C)onc2CO)=O)CCCCN1S(N)(=O)=O 56118,C1(NC(c2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2CCCO2)C1 56119,c1(C(=O)NC(CNC(CCNC(C)=O)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56120,c1(OCC(=O)NC(CNC(c2cnc(NC(C)=O)o2)=O)C)ccc(F)cn1 56121,CCC(C)C(O)C(C)C(=O)NCC1(NC(=O)C(C)N(C)C)CCCC1 56122,CC1C(NC(=O)C=Cc2nccs2)CCCN1C(=O)CC(C)c1ccccc1 56123,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56124,c1(OCC)c(Cl)ccc(C(=O)NC(C)C(N)=O)c1N.c12cc(ccn1)NC2=O 56125,C1(C(N2C(c3c(C)ccs3)CCC2)=O)CC(F)(F)CCO1 56126,N1(C(C2([Si](C)(C)C)CC2)=O)CCC(C(=O)NC2CCCSC2)=C(F)C1 56127,C(CCN=c1[nH]c(=NC(C)C2CCCCC23CC3)[nH]c2c1CSC2)OC(C)C 56128,C(C(C(=O)NCC(N1CC(C)(C)C1)=O)OC)C1CN(C(C2C(CC)C2)=O)C1 56129,N1(C(CN2CC(C)C2)=O)CC(O)CC1CNC(=O)C(CO)c1ccccc1 56130,c1(OC)ccc(C(=O)NCC(C)N(C)C(c2nnn(C)n2)=O)cc1C1CC1 56131,C1(NC(c2c(C)scn2)=O)CCC(O)CN(C(=O)COC2CCC2)C1 56132,N1(C(C2(NC(c3cc(CN(C)C)on3)=O)CC(O)C2)=O)CCC(C)(O)C1 56133,N1(C(Cc2sc(C)c(C(C)C)n2)=O)C(C)CC2CN(C(C3OC(C)CC3C)=O)CC12 56134,Cc1ccc2oc(N(C3CCCN(C(C4CC45CCOC5)=O)C3)C)nc2c1 56135,CCC(CC)(CC)C(=O)N1CC(CNC(c2nn(C)cc2N)=O)C1 56136,N1(C(C2(CNC(Cn3ncc(CC)c3)=O)CCC2)=O)CCN(C)C(SC)C1 56137,C(=O)(CCCN=c1nccc[nH]1)N1C2CC(NC(C(C=C)(C)CC)=O)(C2)C1 56138,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cc2s1)C1C(C)OCC1 56139,C1(NC(c2c(CC)ncs2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56140,C1(F)(CNC(C2CCC(=C)CC2)=O)CCCN(C(=O)CCc2nc(=N)[nH][nH]2)CC1 56141,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2NC(=O)OC2C)=O)CC12CCCC2 56142,c1(NCC2N(C(c3ccc(CC(C)C)nc3)C(=O)NC)CCC2)ccc(F)cc1 56143,C1(C(N(CC(CC)N2CCCC2)C)=O)CCCCN1C(C1CC(F)CN1C)=O 56144,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56145,c1(C(N2CC(C)C(NC(C3(CC(F)F)CCC3)=O)C2)=O)cnc2c(Cl)cccn12 56146,N1(C(CC2C(C)(C)CCO2)=O)CCCCC(CNC(C2CCS(=O)(=O)CC2)=O)C1 56147,c1(C(N(C2CCN(C(C3(C(F)(F)F)CC(=C)C3)=O)C2)CC)=O)c[nH]cc(Cl)c1=O 56148,N1(C(c2ccccc2OC(F)(F)F)=O)CCC2CCN(Cc3ccccc3)C2C1 56149,CCS(=O)(=O)CC(=O)N(C)CCn1cc(-c2ccc(Cl)c(F)c2)nn1 56150,c1(C(N2CC3(C(C(=O)NCCCSC)C3)C2)=O)ccc(Br)c(F)c1F 56151,C1(CNC(c2c(CC)c[nH]c2)=O)(Oc2ncccn2)CCCCC1 56152,c1(C(=O)NC2C(NC(c3cn[nH]c3)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56153,Cc1c(C(N2CC(CNC(=O)C(C)(C)C)CC2C)=O)cc(Br)cc1N 56154,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(CC)(C)CNC(c1cccnn1)=O 56155,n1(C(C(=O)OC)C)nnnc1C(C1CCOCC1)(CC)NCc1ccc(O)o1 56156,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56157,c1(C(=O)NC(C(C)NC(Cc2c(C)nn(C)c2)=O)C(C)C)cc2ccccc2s1 56158,CCCC(C(=O)NCCc1ccc(C)nc1)NC(c1cnn(C)c1OC)=O 56159,c1(N2CC=C(CNC(C3C(C4C(C)C4)C3)=O)CC2)nc(Cl)nc2c1ncn2C 56160,C#CC1CN(C(c2ncc(F)cc2F)=O)CCN1C(C1OC2CCC1C2)=O 56161,c1(-c2cn(C(CNC(C=C(CC)CC)=O)C)nn2)c(F)cccc1F 56162,C1(NC(c2nc(C)oc2C)=O)CC2(NC(=O)C(C)c3nc[nH]n3)COC1C2 56163,Cc1cc(=NCCCC(C)(C)NC(c2ccccc2S(C)(=O)=O)=O)[nH]c(C(C)C)n1 56164,C1(N(C(=O)CC(CC(C)(C)C)C2CC2)C)CCN(C(=O)C(C#N)C2CC2)CC1 56165,C1(C(N2CCCC(CC)CC2)=O)CC2C=CC1N(C(=O)Cc1ccns1)C2 56166,C(=O)(C(F)C1=CCCCC1)NCCN(C(C1(c2ccccc2)CC=CC1)=O)CC 56167,c1(C(N(CCCCN(C(C(Br)=C(C)C)=O)C)C)=O)cc2ncccc2o1 56168,N1(C(c2ccnc(C)n2)=O)CC2CCCCN2CC1CNC(c1cnc(Cl)s1)=O 56169,N1(C(C)=O)CC2CCC1C1CN(C(c3c(F)cc(F)cc3F)=O)CC21 56170,C1(CC)COCCC1NCCNC(=O)OC(C)(C)C.c1(C=O)csc(CO)n1 56171,c1(NC2CCC(NC(C(C)OC(c3ccccc3)C)=O)CC2)ncccc1C#N 56172,Oc1cc(Br)ccc1CNCC1COC2(CCC2)C1 56173,C(=O)(C(C)C(C)CC)N1CC(CCCCNc2ccc(OCC#C)cc2)C1 56174,c1(C(N2CCCC(COC)C2)C(=O)NCCSC)ccc(-c2cccs2)cc1Cl 56175,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2CCCN2N=O)=O)CC1C1CCC1 56176,CCC(c1ccc(C)cc1)=CC(=O)NC(CNC(c1n[nH]cc1OC)=O)CO 56177,c1(C(N2CC3(CN(C(C4CC(C(C)C)OCC4)=O)C3)C2)=O)ccc2c(c1)OCC2 56178,N1(C(c2ccc(C(C)C)cc2F)=O)CC2(CCN(C(C3CCC34CCC4)=O)C2)C1 56179,C(=O)(CCC(=O)N(C(C)(C)CC(=O)NC)C)NC.C12(OC)CC(C1)C(=O)NO2 56180,CC1(CNC(C2CC(=O)N2)=O)CCCN1C(C1(c2cccc(F)c2)CCCC1)=O 56181,C1(SC)CN(C(=O)CCc2c(C)noc2C)CC1NC(=O)CN1CCCC1=O 56182,c12ccccc1-n1nc(CCn3cncn3)nc1-2.CCSC 56183,c1(C(=O)NCC(CO)NC(C=CS(C)=O)=O)sncc1Br 56184,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C(C)C)=O)C1 56185,C1(C(=O)NC2CCCC2NC(C2(CO)COC2)=O)CC12CC(F)(F)C2 56186,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(C2CCC2)C2CCC2)C1)C(C)C 56187,N1(C(C(F)=CC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56188,C12(NC(=O)Cc3ccno3)CC1CN(C(C1CCCOC1c1cc[nH]n1)=O)C2 56189,C1(CNC(C(C)(C)OCC)=O)COCCN1C(C1CC(OC(F)(F)F)C1)=O 56190,c1(NCC2(C=C)CCCCC2)cc(Cl)c(OC)cc1SC 56191,C1(C(=O)NC(CCC)c2nn[nH]n2)N(C(c2c[nH]c(=NC)o2)=O)CCCC1(C)C 56192,N1(C(C2N(C)CCOC2)=O)CC2(C(=O)OCCNC(=O)OC(C)(C)C)CC1CCO2 56193,Cc1nc(CO)oc1C(=O)NC(C)CNC(C1CCC1C(c1ccccc1)=O)=O 56194,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56195,C(c1cccc(Br)c1)=CC(=O)N(CCCC#C)CCC 56196,C(=O)(C(=O)N=c1ccn(C2CC2)[nH]1)N1C(c2n(C)cnc2)CCC1 56197,C(CNC(=O)C=CC(F)F)(CC(=O)NCC1COC(C)(C)C1)OC 56198,C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2c(C)ccoc2=N)=O)CCC1(F)F 56199,c1(C(=O)NCC2(O)CN(C(C3CC(OC)C3)=O)C2)nn(-c2cnn(C)c2)nc1C 56200,c1(OC)cc(CNC(C2(C)CCCN2C(=O)C(C(C)O)NC(C)=O)=O)cnc1C 56201,N1(N2CCC(C(C)C=O)C2)CC2(CO)CCC1CC2.c1(C=O)cn(C)c(O)n1 56202,c1(SCC(c2ccc(OC)cc2)O)ccc(C)nc1O 56203,N1(C(CCCCCN(C)CCOC)=O)CC2CC(N=c3[nH]nc(OCC)s3)CC1C2 56204,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CC=C(Cl)Cl)CCC2C1 56205,CC1NC(=O)CCC1C(=O)NCC1(C)CCN(C(=O)Cc2ccnc(O)c2)C1 56206,c1(CC(=O)NCC2=CCN(CCOCC3CC3)CC2)cccc2cc[nH]c12 56207,C1(CCOC)CCN(C(=NCC2SCCS2)NCC(C)(C)n2cccn2)CC1 56208,N1(C(CCc2cc(OC)no2)=O)CC(NC(=O)C=C2CCC2)C2(CC2)C1 56209,c1(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C(O)C2)=O)ncc2[nH]ncc2n1 56210,N1(C(C(C)=C(C)C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56211,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56212,N1(C(c2c(C)cno2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(CC2CC2)C1 56213,CC1CCC(Cl)=C(C(=O)Nc2nc(-c3cccnc3)cs2)C1 56214,C(=O)(C1CCCc2nncn21)NCC1C(C)CCN(C(C2C(C(=C)C)OCC2)=O)C1 56215,N1(C(c2c(CC)oc(C)c2)=O)CCC(C(=O)NCCC(C)(C)COC)C(C)(C)C1 56216,c1(-n2cc(CCN(C(CN3CCN(CC)CC3)=O)C)nn2)ccc(F)c(C)c1 56217,N1(C(Cc2cc(C)no2)=O)CCC2(CC2)CC1C(=O)NCC1CCOCC1(C)C 56218,CC(C)C(O)CC(=O)N1CCCC1CNC(c1ccc(NCCN(C)C)cc1)=O 56219,C1(C(C)C)N(C(=O)CCOCCNC(=O)C(C2CCOCC2)C)CC12CCCC2 56220,C1(CC(N2C(COC)CCC2)=O)(NC(=O)Cn2nccn2)CCCCC1 56221,c1(NCCC(=O)NC2CC(C)CN(C(=O)C(F)(F)F)C2)ccccc1[N+](=O)[O-] 56222,C(c1cnc[nH]1)=CC(=O)NCC(C1CCOCC1)NC(c1ncoc1C1CC1)=O 56223,c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)ccc2cccnc2c1 56224,c1(NC(C)=O)cccc(C2CC2)c1F.N1(CC)CCC2(C1)c1nnnn1N2CC 56225,CN1CCN(C(c2ccccn2)=O)CC1CNC(c1ncccc1F)=O 56226,O=C1NCc2cc(C(=O)NC3CCCCC3Nc3ncncc3Br)ccc21 56227,C1(NC(C2OCCN(CC)C2)=O)(CC)CCN(C(C2(C(N)=O)CC2)=O)CC1 56228,C1(NC(CC)=O)CN(C(c2occc(=O)c2Br)=O)C2(CCOC2)C1 56229,C1(OC)CCC(CC(N2CCC(CC(=O)OCCC(C)CCO)CC2)=O)CC1 56230,N1(C(C(C)OCOC)=O)CC2CCC(C1)C(NC(c1cccc(OC(C)C)c1)=O)C2 56231,N1(C(c2nccc(CNC(CC3(OC)CCC3)=O)c2)=O)CC(C)CC1(C)C 56232,C1(C2CCN(Cc3nc(C4CCCC4)no3)C2)(NC(CC=C=C)=O)CC1 56233,CC1(C)CN(C(C2CCCCC2O)=O)CCC1NC(C1CC12CCSCC2)=O 56234,C(=O)(C(F)CC(C)C)NCC(CC)NC(=O)Cc1ccc(OC)cc1OC 56235,N1(c2nccc(OCC)n2)CCC(C)C(NC(C2CCCC2C)=O)C1C 56236,Cc1ccc(C2=CCC(C)(C)CC2)c2nc(C(=O)NCCc3ccnn3C)cn12 56237,c1(C(=O)NCCNC(CSCCN(CC)CC)=O)ccc(O)c(F)c1 56238,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56239,C(=O)(CCCOCC(F)(F)F)N1CC(CC(C)NC(C=C(C)CF)=O)C1 56240,C(=O)(C(C)(COC)OC)NCC(CNC(C(C=C)C)=O)OC 56241,N1(C(COC)=O)CCCC2C1CCCN2C(=O)CN1CCS(=O)CC1 56242,C(CCCCC(=O)N1CCN(C)C(C(=O)NCC(C)N2CCC2)C1)SC 56243,c1(C(=O)OC)ccc(C)cc1SC1CCCN(C(C2(c3ccon3)CC2)=O)C1 56244,N1(C(c2n[nH]c3c2CCC3)=O)CCC2CN(C(C3(CC(F)F)CC3)=O)CCC2C1 56245,C#Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)C=CC2CCCC2)ccc1C 56246,C(CCCOC)(C(=O)NCCCN(C)C(C)C)NC(c1c(CC)cno1)=O 56247,c1(C(=O)NCC(=O)NC(C2CN(C(c3cccnc3)=O)C2)C)ccc(F)cc1 56248,c1(C(N2CCC(C(C)(C)NC(C(C)O)=O)CC2)=O)cc2occc2s1 56249,c1(CN(CCNC(C(N)=O)=O)C(C2CC2C(F)F)=O)ccc(F)c(F)c1 56250,c1(CC)nnsc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 56251,C(=O)(C(C)(O)CC(F)F)NCC(CN(C(CCn1c(C)nc(C)n1)=O)C)(C)C 56252,c1(NC(=O)CCN2CC(F)(c3cn(C4CCOCC4)nn3)C2)ccc(F)cc1F 56253,O(NC(=O)CNC(=O)CCN(CC(C)(C)C)CC)CC 56254,CC(C)(C)C#CC(=O)NCCC1CN(C(C2(C)CCCO2)=O)CCO1 56255,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)cc1 56256,N1(CC(=O)NC(C2CC2CNC(=O)C(F)(F)C2(O)CCC2)C)CCCCC1 56257,C(=O)(C(O)CC(F)(F)F)NCC1(CC)CCCN(C(=O)C(C)(C)C(F)(F)F)C1 56258,C1(NC(c2cscn2)=O)C2CCCC1CC(NC(C1CCC=CCCC1)=O)C2 56259,c1(NC(C2(CNC(C)=O)CSC2)=O)cnc(C)c(C)c1C 56260,C=CCCCCC(=O)OCc1csc(C(C)N)n1 56261,C12(CCC(F)(F)CC1)C(=O)N2.N1(C(=O)OC(C)(C)C)CC2CC1C2CC1CC1(F)F 56262,C(=O)(N=c1[nH]c(=NC2CCCC(F)(F)C2)[nH]c2ccc(Cl)cc12)NC(C)(C)CO 56263,N1(C(c2c(C)cccn2)=O)CCc2sccc2C1CNC(=O)C(C1CC1)N(C)C 56264,N1(c2snc(C)n2)CC2(C)CN(OC)CC2(C)C1.C1(C=O)Cc2nnc(C)n2C1 56265,CC1CC(C(=O)NC2CCCN(C(C3(n4ccnn4)CC3)=O)C2)CC(=O)N1 56266,C1(N=c2cnc3cc(F)c(F)cc3[nH]2)(CC)CCN(Cc2ccc(Cl)s2)C1 56267,C1(C(=O)NC2CCCN(Cc3cnc(C4CC4)o3)C2)(CC)CCC(F)(F)CC1 56268,C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(c2occc2F)=O)CC1 56269,S(=O)(=O)(c1cccc(NC(=O)C(Cl)(Cl)Cl)c1)N(C)C.N12C3CCC1CC(C3)C2=O 56270,c1(OC)ccc2c(c1)CCC2C(=O)NC1CC(CO)N(C(=O)CN=S(C)(C)=O)C1 56271,C1(COC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)Cc2cccc(C#N)c2)C1 56272,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56273,Cc1nc(C(N2CC(NC(c3cn(C)c(=O)n3C)=O)C2)=O)c(C)n1C1CC1 56274,C(=O)(NN1CCCC1C(=O)NCCCN(C)C)c1c(C)ncs1 56275,CC(C)CC(C(=O)NCCn1ccnn1)ONC(=O)CC1CCOCC1 56276,C(=O)(C(O)CC(C)C)N1C(CCNC(c2c(OC)noc2C)=O)CSCC1 56277,c1(CC(=O)NCC(CC)NC(c2n[nH]cc2OC)=O)cnc(C(F)(F)F)nc1 56278,N1(C(CCOCC)=O)CC2(CCC(NC(=O)C(=O)NCC(F)F)CC2)C1 56279,c1(OC)ccc(C(CNC(=O)NCCN2CCCCC2=O)NC2CC2)cc1 56280,c1(NC)c(C(N2CCN(C)C(=O)C2)=O)sc2nccnc12 56281,C1(NC(c2nc(C(C)=O)sc2)=O)CCN(C(c2cnsc2)=O)CC1C 56282,C1(C2(O)CCOCC2)(C(=O)NC2CC3CC(NC(C(C)=C(CC)C)=O)C2C3)CC1 56283,C=CCC(CC(=O)N(C)C)NC(C)=O.c1(C(=O)NCCOCCN)ccc(OC)cc1 56284,N1(C(CCC(=O)NCc2ccncc2)=O)CCC2C(CCN2CC)C1 56285,C1(C(=O)NCC(O)C(=O)NC2CC(O)(CO)C2)CCC(O)CC1 56286,CN1CCN(C(C2(CO)COC2)=O)CC1CNC(=O)CSCc1ccncc1 56287,C(=O)(CCCCCC#N)N1C(C(=O)NC(CCCC)Cc2ccc(F)cc2)CC1 56288,C(=O)(C(CC(N)=O)NC(=O)CCn1cncn1)N(C(CC(C)C)C)C 56289,C1(C(=O)Nc2cccc(CCC)c2)CCC(C)(CC)C1(C)C 56290,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)=O)C1)OC 56291,c1(CC(=O)Nc2ccc(CNC(CC(C)(C)O)=O)o2)ccc2c(c1)CC2 56292,c1(C(=O)NC2CC(O)(CNC(c3coc(Cl)c3)=O)C2)cnc2[nH]nnc2c1 56293,CC1(CC(N2CCC(OCC3CC3)C2)=O)CN(C(=O)CCc2ccco2)C1 56294,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56295,c1(CC(=O)NCC(N(C(=O)CCn2cncn2)C)C2CC2)cccc(C(F)F)c1 56296,N1(CC(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56297,c1(Nc2[nH]nc(C(C)(C)C)c2C#N)ccc2ncc(-c3cccc(F)c3F)n2c1 56298,C1(NC(C(C)Cc2ccccc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56299,c1(CC(=O)NC(CN(C)C(C2(Cl)CC2(C)C)=O)(CO)CO)ccc2ccoc2c1 56300,C(=O)(C1=CCC(F)(F)CC1)N1CCC(C(C)NC(c2ccc3[nH]ccc3n2)=O)C1 56301,c12ncccc1o[nH]2.n1(C(C)(C)C)nccc1-c1cn(C)nn1.c1(C)cccnc1 56302,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56303,c1(CN(C(=O)CC2(c3ccccc3)COC2)CC=C)cccc(F)c1F 56304,c1(C(N(CCOCCCOC)C)=O)ccc(NC(C2N(CC)CC2)=O)c(F)c1 56305,N1(C(c2c(C(C)C)cnn2C)=O)CCC(C)C(NC(=O)C=CCO)C1 56306,CN1CCC(Nc2cc(NCc3nc(Cl)cs3)ncn2)CC1=O 56307,c1(C(N2CC(c3cn(-c4ccc(Cl)c(F)c4)nn3)C2)=O)ccc(C(F)F)c(F)c1 56308,c1(C(N2C3CC(NC(c4c(CC)onc4)=O)C2CC3)=O)c(C)ccc2n[nH]cc12 56309,C(CCC(C(=O)N1CCC(=O)NCC1)NC(C1CC1Cl)=O)OC 56310,N1(C(C2C(=C)C2C(=O)OC)=O)CC2CC1C1CC21.C1CCC(=O)N1C 56311,C1(C(N(CC(CN(C(=O)CC23COC(CF)(C2)C3)C)O)C)=O)CC2OC1C1CC21 56312,S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC2C(C(N3CC(F)C(F)C3)=O)C(CC2)C1 56313,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(c2ccc(N)cc2)=O)C(C)C1 56314,N1(CCN(C(=O)Cc2ccccc2CO)C)CCN(C(=O)CC2(C)CCCO2)CC1 56315,c1(C(=O)OCCC)nc(OC(C)(C)C)cc(N2CC(NC(C)=O)C3(CC3)C2)n1 56316,c1(C(=O)NC2C3CCN(C(CSCCC)=O)C32)cc2ccc(OCC)cc2[nH]1 56317,C1(C(=O)NC2CCC(NC(=O)Cc3ccsn3)CC2)CN2CCN1CC2 56318,c1(CC(=O)N(C(C)CNC(=O)C(O)c2ccco2)C)ccccc1C1CC1 56319,CC1CN(C(C2CC(C)(C)CO2)=O)CC1Cn1cc(CN2CCC2CO)nn1 56320,C1(C(=O)NCCC(C)CO)(OC)CCN(C(=O)C(O)C(C)C)C1 56321,N12CCC(C1(C)C)c1c(cco1)CNC2=O.C1(C(=O)OCC)COCCN1CC 56322,C(=O)(CCC(=O)C1CC1)N1CC(O)(C(C(=O)NCC=CCCC)C)C1 56323,N1(C(=O)CCCF)CCC(C2CCN(C(c3ccc(=O)n(CCO)c3)=O)CC2)CC1 56324,C1(CC(CC)C)CC(C(N2CCN(C(=O)CC=C(C)C)CC2)=O)CCO1 56325,c1(C(=O)NCC(n2cc(-c3cc(=O)cc[nH]3)nn2)C)cn(C)nc1-c1ccccn1 56326,C1(NC(c2ccc(CCC)[nH]2)=O)CC2CC(NC(C3(c4ccon4)CC3)=O)C2C1 56327,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(c1ccc(C(F)F)o1)=O 56328,C1(CC=C)CCCN(C(C2(N(C(=O)CCCC3CC3)C)CC2)=O)C1 56329,N1(C(c2c(COC)ncs2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56330,CCC(CC(F)(F)F)C(=O)N(CCCN(C)C(C12CC(F)C1C2)=O)C 56331,Cc1cc(C)c(S(=O)(=O)NC(c2ccc3ccc(CO)cc3c2)=O)cc1C#N 56332,C=CC(C)CC(=O)NCC(c1ccccc1)NC(c1sc(Br)cc1F)=O 56333,CCCC(O)CC(=O)N1CC(NC(=O)CC2=CCCC2)C(C)(C)C1 56334,c1(NCc2cccc(OCC)c2O)ccc(Br)c2c1CNCC2 56335,c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C)cccc2nc(N(C)C)oc12 56336,c1(OC)ccc(OCC(N2CC(NC(=O)CSCC(N)=O)CC2CO)=O)cc1 56337,C(=O)(CC(C(F)(F)F)OC)N1C(C(C)NC(=O)C(F)(F)C(F)F)CCC1 56338,c1(N2CCN(CC)CC2)nc(C(F)F)nc(=N)[nH]1.C1(=O)CC(=O)N2CCC(C2)CN1 56339,C(=O)(C#CC1CCOC1)NC(CC(=C)Cl)C(=O)NC(CCO)C(C)C 56340,C(C(C)C(F)C(=O)NCCC(F)(F)CO)NC(c1c(C)csn1)=O 56341,C1(NC(CCC(=C)Cl)=O)CCCN(C(=O)C=CC(c2cnn(C)c2)=O)CC1 56342,CC(=O)C(C)(C)CC(=O)NCCOCCCN(C)C(c1cc(C(N)=O)c[nH]1)=O 56343,C(=O)(C1=CCSC1)NCC(CNC(c1scc(C(C)=O)c1)=O)F 56344,c1(C(=O)NC2CC(NC(C3CCCC34CC4)=O)C2)cc2ccc(Cl)c(F)c2o1 56345,C(=O)(C(CC(F)F)N(C)C(C1CCOC1C(C)C)=O)NCCC#C 56346,C1(NC(c2ccccc2)=O)CCSCC1.C12CC1C(=O)NC2C 56347,C(=O)(C(C)(C)CC(C)C)N(CCCNC(C=CC(CC)=CC)=O)C1CC1 56348,Cc1ncc(C(=O)NC(C)C(C)(C)NC(=O)COC(C)C)c(=N)[nH]1 56349,C(=O)(CCC(F)(F)C(F)(F)F)N(CCC)CCNC(C1(C)CCOC1)=O 56350,C1(NC(C2N(C(CC)=O)CSC2)=O)CC2CC1N(C(c1cc[n+]([O-])cc1)=O)C2 56351,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56352,c1(NC(CC)=O)ccc(C(=O)NCCCN(C(=O)C(C)CSC)CCO)cn1 56353,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1ccc(N(C)C)cn1)=O)C2 56354,C1(C(N(CCSC)C)=O)CCOC(C)C1.C1CC(=O)NCC(=O)N1 56355,N1(C(C(C(C)C)NC(=O)OC)=O)CCC2CC(NC(=O)C(Cl)=CCl)CCC2C1 56356,c1(OC)ccc2c(c1)CCC2N(C)C(C1CCS(=O)(=O)N1)=O 56357,Cc1cc(C(=O)NC2COCCC2NC(=O)CCC(F)F)ccn1 56358,C1(C(=O)NC(C)CC(C)C)(OC)CCN(C(=O)CCSC2(C#N)CCCC2)C1 56359,c1(C(=O)NC(CC)CN(C)C(c2oc(C)nc2C(C)C)=O)cc(OC)cnc1F 56360,CC1CCCC(C(=O)NCCOC2CCN(C(=O)CCC3CCCC3)C2)C1 56361,CCC(CC)CC(=O)Nc1cccc(CNC(=O)C(C)(C)C(C)C)c1 56362,Cc1cccc(CC(=O)NC2C(CNC(C3(C)CC3(C)C)=O)C2(C)C)c1F 56363,c1(C(=O)NCC(CNC(CCc2cncc(C)c2)=O)O)ccc2c(c1)CCC2=O 56364,C1(C(N2CCCC(CNC(=O)Cc3cc(Cl)no3)C2)=O)COc2ccccc2C1 56365,C(c1ccc(Cl)cc1Cl)=CC(N1C2CN(Cc3c(OC)ccc(Cl)c3)C(C2)C1)=O 56366,N1(C(C(C)OCC2CC2)=O)CCCC(N(C)C(c2ccc(Cl)c(F)c2)=O)CC1 56367,c1(NC(=O)CCc2ccc(-c3nn[nH]n3)cc2)ccc(F)cc1O 56368,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1C 56369,C1(C)(NC(C(C)Cc2cccnc2)=O)CCN(CC(C)O)C1 56370,CC1(C)CC(C(N2CCCC(O)(CNC(c3ccsc3Cl)=O)C2)=O)CC(C)(C)S1 56371,C1(C(=O)OC)CC12CCC(NC(c1sc(C)cc1C)=O)CC2 56372,c1(CC(=O)NC2(CCNC(Cc3cc(C)n(C)n3)=O)CC2)ccc(Cl)c(Cl)c1 56373,C12(CNC(=O)COC3CC3)CCC(CC1NC(=O)C(C1CCOCC1)O)C2 56374,c1(OC)cc(F)cc(F)c1S(=O)(=O)NC(C)(C)Cc1cc(F)cc(F)c1 56375,c1(-c2ccc(C(C)C)cc2)cccc2c(C(=O)Nc3ncc(Br)s3)[nH]nc12 56376,N1(C(CNC(C(=C)C)=O)=O)CCC12CCN(C(=O)Nc1cc(C)nc(O)c1)CC2 56377,C1(C(=O)Nc2cccnc2)CC12CN(C(C13CC(c4ccccc4)(C1)C3)=O)C2 56378,c1(C(=O)OC)cc(C(=O)Nc2cn(-c3ccccc3)cn2)cn1C.N12CC(C1)C2 56379,c1(CC(N2C(CN(C(CC(CC)(F)F)=O)C)CCCC2)=O)nnc2n1CCOC2 56380,c1(C(N(C(CN(C(C2(F)CC(C(=O)OCC)C2)=O)C)C)C)=O)csc2nccn12 56381,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56382,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56383,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(C1CC1CC(C)C)=O)OC 56384,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(Cc2ccc(CC)cc2)=O)CC1C 56385,N1(C(=O)CC2CC3(COC3)C2)CCCC(N2CCC(CCO)CC2)C1=O 56386,C1(N(C(=O)C=CC2CC2)CCC)(CNC(=O)CSC)CCC1 56387,N1(C(c2cn(CCC)nn2)=O)CC(C)(C)OCC1CNC(c1cnoc1C)=O 56388,C(C(C)(O)CC(=O)NC1CCCCC1C(=O)N(C(C)CCO)C)OC 56389,Cc1ccc(C(C)C(N2CCCC2(C)C(=O)Nc2cncnc2Cl)=O)cc1 56390,c1(N(C(C(C2CC(=C)C2)=O)=O)CC)cccc(-n2cncn2)n1 56391,C(=O)(C1c2c[nH]nc2CN1C(c1ccc(CC)nc1)=O)N1C(C=C)CC1 56392,S(=O)(=O)(c1ccccc1N)N(c1ccc(NCCCc2ccccc2)cc1)C 56393,CC(O)(CNC(C1CC12CC(NC(c1coc(C3CC3)n1)=O)C2)=O)C(F)(F)F 56394,c1(CC(=O)N(C)CCNC(c2cnn(CCO)c2)=O)ccc2nc[nH]c2c1 56395,C1(NC(c2cccc3ncsc23)=O)CN(C(c2cnco2)=O)CC12COC2 56396,c1(C(=O)NC(CN(C(C2CCCCC23CC3)=O)CC)C)ccc(S(N)(=O)=O)s1 56397,N1(C(C)=O)CCC(C)(NC(c2cc(N3CCCC3)cnn2)=O)CC1 56398,O=C(CCC(=O)c1cncs1)NC1CCCCC1NC(C1CCCC(CF)C1)=O 56399,c1(C(N(C(CNC(C2C(C)CCO2)=O)C2CC2)C)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56400,C1(O)(CC(=O)N(C)CC2CCC(NC(=O)C(C3CCCCC3)O)C2)CCCCC1 56401,C(C(=O)N1CCN(C)CC1)(C(C)C)N(CC(C)C)C(C1(C(N)=O)CC1)=O 56402,C1(NC(c2c(C)coc2C(C)C)=O)C2CCC1N(C(=O)CC1COCCO1)C2 56403,n1(CC)nnnc1C(c1ncoc1C)NCCCOCCc1ccccc1 56404,C(C(=O)NCC1(CN(C(C(CC)c2ccccc2)=O)C)CC1)(C(C)C)NC(C)=O 56405,Cn1nccc1C=CC(=O)N(CCNC(c1ccsc1C#N)=O)CC1CCCC1 56406,N1(C(c2scc(OC)c2)=O)CC(O)CC1(C)C(=O)NCc1ncccc1C 56407,N1(C(C2(CCCC)CCC2)=O)CC2(CC(NC(C3(O)CCC3)=O)c3nccn32)C1 56408,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56409,c1(CC)c(C(C)=O)[nH]c(C)c1C(C)=O.N12CCOC(C1)C2=O.C1CCC(=O)N1C 56410,C(=O)(C(F)C(C)CNC(C1(C(N)=O)CCC1)=O)N1CC(CC)OCC1 56411,CC1CCOC1C(N1CC(C(N)=O)(CNC(c2nc(Cl)cs2)=O)C1)=O 56412,N1(C(C(C)(C)C)=O)CC2(C=C(C(=O)N3CCOC4C(O)CCC34)CO2)C1 56413,Cn1ccc(C(=O)NCC(C2CCCO2)O)c1CC(=O)Nc1n[nH]c(C2CC2)n1 56414,CCCC(C)CC(=O)NCCN(C(c1cc(C)nc(C)n1)=O)CC1CC1 56415,N1(C(CC(C)OC)=O)C2CCC(C2)C1CC(N1CC2(C=CCO2)C1)=O 56416,N1(C(=O)CCc2nc[nH]n2)CCCC2C(CCCN2C(c2cc(F)c[nH]2)=O)C1 56417,C1(NC(C(C2CCOCC2)C)=O)CC(C)(NC(=O)CNC(=O)CN(C)C)C1 56418,C(=O)(C#CC1(C)CCCO1)N1C(CN(C)C(c2cn(C)nc2C(F)F)=O)CCC1 56419,c1(NC(c2ccccc2)CN2C(C(C)O)C2)cccc(Cl)c1O 56420,C(CCN=c1[nH]c(=N)[nH]c2c1C(O)CCC2)OCCCC 56421,c1(C(=O)NC2CN(C(c3ccc(C)o3)=O)C2)sc2cncn2c1C 56422,N1(C(=O)Cn2cc(COC3CC3C(F)(F)F)nn2)CC2(C3CCC3)CCC1CC2 56423,C1(NC(C(C)(CO)NC(C(C)OCC=C)=O)=O)CN(C)CC1(F)F 56424,C(C(C)(F)C(C)C)NC(C1C(CNC(c2cc(C(C)C)[nH]n2)=O)OCC1)=O 56425,n1(CC(C)(C)CO)nc(-c2ccc(Cl)s2)nc1-c1ccc(C(F)(F)F)s1 56426,C1(CNC(C2CCC(O)(c3ccccc3)C2)C)CC(C)CC(C)(C)C1 56427,N1(C(c2sc(C)cc2C)C(=O)NCCC(=O)OCC)CCC(C#N)CC12CC2 56428,C1(CC(N2C(CN(C(=O)Cn3cc(Br)cn3)C)CCC2)=O)COCC(C)(C)O1 56429,c1(CC)cc(CC(N2CC(F)(CNC(C3CC(F)(F)C3)=O)C2)=O)n(C)n1 56430,C1(CNC(C=CCN(C)CC)=O)CN(C(c2cn(C(C)(C)C)nn2)=O)CC1C 56431,c1(C(=O)NCCOCCNC(c2sccc2C2CC2)=O)nn[nH]c1Cl 56432,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56433,C1(CNC(c2n(C)cnn2)=O)COCCN(C(C2CCCOCC2)=O)C1 56434,Nc1cc(C(N2CCC(OCCNC(c3cccc[n+]3[O-])=O)C2)=O)cc(F)c1 56435,N1(C(c2[nH]cc(CC(C)C)c2)=O)CCC(NC(=O)C2=C(Cl)CCC2)CC1C1CC1 56436,C(=O)(CCCCCNC(=O)C(=O)C(C)(C)C)N1CC(CCN(C)C)C1 56437,C(CNC(C1CC1C1CC1)=O)(C(C)(C)C)NC(c1n(CC)ncc1)=O 56438,C(c1ccccc1F)=CC(=O)NCC(C1CCCCC1)NC(C12CCCC1CC2)=O 56439,N1(C(C(CCC)OC)=O)CCC2(CC(C(=O)NCCC(C)C(F)F)C2)C1 56440,c1(CCC(N2CC(NC(C(CC)N(C)C)=O)C(F)C2)=O)cnc2ccccn12 56441,Cc1cc(Br)c(O)cc1C(=O)NC12CC(C(N)=O)(C1)C2 56442,C1(NC(CC(CC)C2CC2)=O)CCSC12CN(C(=O)CN1CC3C=CC1C3)C2 56443,CC1OC2CCC1(NC(=O)NCc1coc(C3CCOCC3)n1)C2 56444,c1(C(=O)NCC(C)(C2CC2)NC(C2(C)CC=CCO2)=O)nnn2c1CCC2 56445,c1(C(=O)NC(CCNC(c2ccc(C(=O)OC)[nH]2)=O)(C)C)cc2cc[nH]c2cn1 56446,C1(C(=O)NC(C2CN(C(c3c(SC)n(C)nc3)=O)C2)C)CCC(N=[N+]=[N-])C1 56447,N1(C(C2C(C)C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56448,c1(CN2CC3C(C(=O)Nc4ccnc(O)c4Br)(C3)C2)cc(Br)c(O)cc1O 56449,C(=O)(C1CCc2nccn21)NCC1(C)CCN(C(COCC(=O)NC)=O)CC1 56450,C(=O)(C1=NOC(NC(=O)CC2(C=C)CCC2)C1)NC1C(C#C)CCC1 56451,c1(C(=O)NCC2CN(C(c3c(N(C)C)cncc3)=O)C2)ccc2nc(O)cn2c1 56452,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56453,C1(CC#N)CCCN(c2ccnc(NC(c3cccnc3)CC3CC3)n2)C1 56454,CCN(Cc1cn(CCC(C)C)nn1)N1CCCCC12CCS(=O)(=O)CC2 56455,N1(C(C2(F)CCN(C(C(CCC=C)(F)F)=O)CC2)=O)CC2C=CCN(C)C2C1 56456,c1(C(=O)NC2COCCN(C(C3C4CCCCC34)=O)C2)c[nH]c2ccc(Cl)cc12 56457,Cc1cn(C)cc1C(N1C(C(N2CCOC(CN=[N+]=[N-])C2)=O)CCC1C1CC1)=O 56458,C(CCCCNC(C12CC1C2)=O)NC(C1(C(=O)NCC=C)CC1)=O 56459,c1(C(N2C(C=CC(=O)N(CC(C)(O)C3CC3)C)CCC2)=O)cccc2ccnn12 56460,c1(CCC(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)C)cccc(C(F)(F)F)c1 56461,N1(C(c2c(C)nc(C(C)OC)s2)=O)CCCN(C(C2(NC(C)C)CC2)=O)CC1C 56462,c1(C(=O)NCC2N(C(c3cn(C4CC4)nn3)=O)CC2)c(F)cccc1F 56463,c1(N(CC(N2CC(OC)N(C)CC2)=O)CC(=O)N(C)C)ccc(C#N)cc1F 56464,C1(C(=O)NCCC2CCN(C(c3ncoc3C3CC3)=O)C2)CC(=O)NC(=O)C1 56465,Cc1cc(C(=O)Nc2cnc(F)cc2N(C)C)nc2ccccc12.N12CCC1C2=O 56466,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(c2cc(-c3ccoc3)[nH]n2)=O)C1 56467,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CC(NC(=O)C(Cl)=CCl)C2)c1F 56468,c1(C(N(C2CCN(C(=O)C(C)N3CCCC3)C2)CC)=O)ccc(=O)oc1 56469,C#Cc1cccc(CC(=O)NC2CN(C(=O)C(C3CCC3)OC)CC2O)c1 56470,CC(C)CC(C)(CNC(C1CN(c2cnn[nH]2)C1)=O)NC(c1cc(=O)n(C)cn1)=O 56471,c1(C(=O)NCC(CNC(=O)CCCF)F)ccc2ncncc2c1 56472,CCC(C(=O)N1CCC(CC(=O)NCC(C)(O)Cn2cccn2)C1)C(C)(C)CC 56473,c1(OCC)cccc(C(N2CC(NC(c3cnc(O)n3C)=O)CC(O)C2)=O)c1N 56474,C1(CNC(C(C2CCCOC2)OC)=O)CC2(CCC2)CN1C(c1c[nH]nc1F)=O 56475,c1(CNC(c2cn(C)c(=O)cc2)=O)cc2n(n1)CCN(C(=O)C1=COCCC1)C2 56476,N1(C(CNC(=O)NC)=O)CCCCC1C1CCCN1c1snc(Cl)c1C#N 56477,N(C(=NCCNC(C1CCCS1(=O)=O)=O)NC1CCC1)CCS(=O)(=O)N(C)C 56478,C(=O)(C(=O)CCC(C)(C)C)N(CC(C)NC(CCC(=O)NC)=O)C 56479,C1(C(N(CC(CN(C(c2n(CC#C)cnn2)=O)C)O)C)=O)CCC2(CCC2)C1 56480,C#Cc1cccc(C(=O)NC2CC(CNC(C34CSCC3C4)=O)C2(C)C)c1F 56481,c1(COCC(=O)N(CCCNC(c2oncc2C(F)(F)F)=O)C)cccc(F)c1 56482,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56483,C1(CC(=O)NCC2CC2)CCC(C#N)C1.C12(CC1)C(C)NC2=O 56484,c1(C(=O)NCC2(F)CC(CNC(COCCC(C)C)=O)C2)ccc(F)c(N)c1F 56485,CCCC(C(=O)N1CCC(C(N2CCC2C(=O)N(C)C)=O)CC1)C(C)C 56486,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56487,N1(C(c2c(OC)c(F)ccc2)=O)C2CCC1CN(C(=O)Cc1cccnc1)C2 56488,c1(C(=O)NC2CC(C(C)NC(C3CNC(=O)N3)=O)C2)c(F)cccc1[N+](=O)[O-] 56489,c1(C(N2CCC(C)(CNC(=O)CCC3CCOC3)C2)=O)ccc(F)cc1Cl 56490,c1(C(N2CCC(NC(C(C)OCC#C)=O)C(F)C2)=O)csc2cccnc12 56491,C1(C(C)C#N)CCN(C(=O)C(C)N(C(c2ccccc2)=O)C2CC2)CC1 56492,CCC(CC)CC(C(=O)Nc1ccccc1)N1CCCC(C)C1C 56493,C1(F)(C=O)CCN(OC(=O)C(Cl)=CCl)CC1.c1(S)ccccc1.C12(CC1)CC2 56494,C1(NC(c2n(C)nc(C3CC3)c2)=O)CC2CN(c3cnc(C#N)cn3)CC12 56495,N1(CCC(=O)N(CCC(C)NC(=O)CC2COCCO2)C)CCc2ccccc21 56496,c1(CC(=O)NC(COC)NC(=O)C(C)(C)SC)cccc(O)c1 56497,Cc1nc(=NCCC2CCCCC2NC(=O)Cc2cnccc2C)s[nH]1 56498,C1(CNC(C(C)OC)=O)CCC(NC(C2CCOC2)=O)CC1 56499,C1(NC(C2CC(F)CN2C(=O)Cn2ncnn2)=O)CCn2ncnc2C1 56500,C#CCC(CC(F)F)C(=O)NC(CNC(=O)CSCc1ncc[nH]1)CC(C)C 56501,Cc1cccc(NC(=O)C(Cc2cnc[nH]2)NC(=O)CC2CCC2)n1 56502,N1(C(c2c(N)ccc(OCCCC)c2)=O)CCC2(CCN(C(=O)C(C)CF)C2)C1 56503,C(=O)(CC(C)(C)N(C)C(C1COCCC1C)=O)N(CC(=O)OCC)CC 56504,c1(CC(N2CCC(NC(C3(CC)CCCOC3)=O)CC2)=O)cnn2ccccc12 56505,Cc1nn(C2CCC2)cc1NC(=O)C(C(C)C)NC(=O)CNS(N)(=O)=O 56506,Cc1ccnc(C(=O)NCCC(C)NC(=O)CC2CCC2(F)F)c1N 56507,c1(C(=O)NCC2N(C(CCC=CCC=C)=O)CC(C)(C)C2)ccn2c1CSCC2 56508,Cc1cncc(C(=O)NCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC2)c1 56509,S(=O)(=O)(c1cccc2nsnc12)N1C2CCN(C(c3ncn(C)c3)=O)C2CCC1 56510,N1(C(C2N(C(CCC)=O)CCCC2)=O)CCN(C(c2ccnc(NC)n2)=O)C(C)C1 56511,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C3CC3)=O)C2C1)OC 56512,C=C1COCCN(C(C2CN(C(=O)C(C)C(F)F)CCO2)=O)C1 56513,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56514,N1(C(CCOCCC)=O)CCN(C)CC1CNC(=O)COCc1nccn1C 56515,c1(OC)ccc(F)c(N)c1C(N1CC(CCCCNC(C2C=CCCC2)=O)C1)=O 56516,N1(CC(N2C3C(C(=O)NC(C)COCC4CC4)C(C3)C2)=O)OC(C)(C)CC1=O 56517,C(=O)(C(CC(C)C)N(C(=O)C(C#N)C(C)C)C)NC(c1cc(C)no1)C 56518,C(CCNC(c1cc[n+]([O-])cc1)=O)(C(=O)NCCCSCCO)OC 56519,CCCCCCCCC=CC(N1CCCCC1)=O.c1(NC=O)ccc(C)cc1 56520,S(=O)(=O)(c1ccc(NC)c(F)c1)N1CC(COC)OCC1.N1CCOCC1 56521,CCCCCC(O)CNC(=O)CC(CNC(c1cn(CCO)nn1)=O)C1CCC1 56522,C1(NC(C(N2CC(OCC)C(CO)C2)=O)=O)CN(C)C(C)(C)C1 56523,N1(C(CCSC)=O)CCC(O)C(NC(=O)Cc2csc(-c3ccccc3)n2)C1 56524,N1(C(c2ccccc2F)=O)CCC2CCCC12C(=O)NCC1CCC2(CC2)C1 56525,C1(CC)CN(C(C2CCOC2CNC(c2cccnn2)=O)=O)CCCO1 56526,c1(C(N2C(COC)CN(C(=O)C(C)(O)C3CCC3)CC2)=O)cc2ccccn2c1 56527,C1(C(=O)NCC(=O)NCCCC(F)Cl)(CC)CCOC1 56528,C1(c2c(C)n(C)nc2)C(C(=O)N(C)Cc2cnco2)CC(=O)N1C 56529,C(C)(C(C)(C)NC(C1CC(F)(CO)C1)=O)NC(C(=C(C)C1CC1)F)=O 56530,c1(NC(c2sccc2OC(F)F)=O)cccc(Br)c1.N12CC(C1)C(C)NC(=O)C2 56531,c1(C(=O)NC2CCN(C)C2)ccnc2[nH]c(C(N)=O)nc12.C12CN(C1)C(=O)CO2 56532,c1(CC(N2CC(O)(CNC(CCCOCCC)=O)C2)=O)cccc(CC)c1 56533,C(=O)(C(CC)C(C)C)NC(C(=O)N(CCOC)CC1CC1)CCSC 56534,C(=O)(C1=NOC(C)C1C)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)OC 56535,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCC2(C)N=N2)CCC12CCC2 56536,N1(C(c2ccc(OC)s2)=O)C2CCC1C1CC1(NC(c1cnc(O)s1)=O)C2 56537,N1(C(CCC)=O)CCC(C(=O)N(C(CNC(=O)OC(C)(C)C)C)C(C)C)CC1C 56538,C(C(C)(CO)NC(=O)CNc1c(NS(=O)(=O)CCC)scc1)NC(CCC)=O 56539,C1(C(=O)NC2(CCC)CCNC2=O)CN(C(c2ccc(C(C)=O)[nH]2)=O)C2(CCC2)C1 56540,c1(C(N2CCC(c3cncn3C)CC2)C(=O)NC(CC)C)ccc(Cl)c(C)c1Cl 56541,N1(C(c2n(CC)ccn2)=O)CCC(NC(C2(C)CCCS2)=O)C(CO)C1 56542,C12(CNC(c3nc(COC)sc3)=O)CCCC1N(C(C1CCOC1C)=O)CCC2 56543,C(CC1=CCN(c2ncc(NC(CCC(C)OC)=O)cn2)CC1)OC 56544,c1(OC)cc(C(=O)N(C)C)ncc1-c1ccc(F)c(CN2CCS(=O)(=O)CC2)c1 56545,C(=O)(CC(O)CC(C)C)N1CC(O)CC(NC(C=CCC)=O)C1 56546,c1(NC(C2CC3(CC3)C23CCC3)=O)cncc([N+](=O)[O-])c1 56547,C(=O)(C1CCCc2c1ncn2C)NC1CC(C)(NC(CC=C(C)C)=O)C1 56548,c1(C(=O)NC(C(=O)NC(CN(C)C)CCO)CN(C)C)cnc[nH]c1=N 56549,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2(CC1)CC(CNC(c1cocn1)=O)C2 56550,CCCCC(O)C(=O)N1CC(F)CC1CC(=O)NC1CCN(CCF)C1 56551,N1(C(C=CC)=O)CCC2(CC1)CC(CNC(C1CC(=O)N(CCC)C1)=O)C2 56552,c1(C(N2CC(N(C(=O)Cc3ccsn3)C)C2)=O)cc(C2CCOCC2)on1 56553,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NCc2cc(C)[nH]n2)C1 56554,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(=O)CC1CCOCC1 56555,C1(C(C)=O)CCC2CCN(C(c3cnn(C)n3)=O)C12.Cc1cnc(C(=O)N)cc1C 56556,C1(N(C(CCC(=O)N(C)C)=O)C)CCCN(C(c2ccc(O)cc2)=O)CC1 56557,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56558,Cc1c(NC(=O)CC(C(F)F)C2CCC2)cccc1F 56559,N(C1CCc2cc(Cl)ccc21)CC(=O)OCCOc1ccc(OC)cc1 56560,N1(C(Cn2c(=N)scc2)=O)CCC(C(=O)OC(=O)CC2(n3ccnc3)CC2)(CF)C1 56561,CCCC(C)(CCC)C(=O)NC(C)C(C)C(=O)N1CCC(SC)C1 56562,N1(CCc2cc(CC)no2)CC(CO)CC(F)(F)C1.N12CCCC(CC1)C2=O 56563,c1(N2CC(C#N)OCC2)ccc(Br)c(S(=O)(=O)NCC=CBr)n1 56564,c1(OC)ccc(CC2CC2(Cl)Cl)cc1.n12cc(nn1)COCC(=O)N(C)CCC2 56565,CC1CC(NC(=O)COc2cccc(NC(N)=O)c2)CN1C(C1CC(F)C1)=O 56566,Cc1c(CCC(=O)NCC2(C(=O)OC)CC2)cnn1C.C12CN(C1)C(C)C(=O)N2 56567,c1(C(=O)NCC2CC(NC(C(CCC)C#N)=O)C2)[nH]c2cc(Cl)ccc2c1C 56568,CCCC(C(O)C(=O)Nc1cc(C)c(C)cc1C)NC(=O)CC1NC(=O)NC1=O 56569,C(=O)(C(C(C)C(C(=O)OC)CCC=O)N1CCOC(C)CC1)OCC 56570,c1(C(=O)OC)cc(F)cnc1NC(C1CC1C(=O)Nc1ccc(C#N)cc1)=O 56571,S1(=O)(=O)c2cccnc2N1CC(C)C.c1(C(CCO)CC(=C)C)cccc(Br)c1.OC 56572,C(=O)(CC(O)CNC(c1csc(F)c1)=O)NCC(C(C)O)C 56573,C(C(N=c1[nH]c2c(c(=NCC=CC3CC3)[nH]1)CSC2)c1ccc(Br)cc1)OC 56574,N(C(=NCCC1COC(C)(C)C1)NC)CC1CC1.c1(OC)ccc(C(=O)N)cc1 56575,CC1CCCN(C(c2cncc(NC(=O)CN(C)C(N)=O)c2)=O)C1CCO 56576,C1(C(N(CC(=O)NC(CCC)C2CCC2)CCC)=O)CCN(C)C(=O)C1 56577,N#Cc1ccc(O)c(C(=O)NCC23CC(CO2)N(C(=O)CCNC(=O)CO)C3)c1 56578,C(=O)(CC(C)(F)F)NCC(COC)NC(c1ccnc(N(C)C)c1)=O 56579,C=CCCC(F)(F)C(=O)N1CCN(CC2CCN(C(=O)CN(C)CC)CC2)CC1 56580,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(c2ccc(OC)cc2)=O)C12CCC2 56581,C(CN=c1[nH]c(NC2CCCc3n[nH]cc32)nc2c1CCCC2)(C(C)(C)C)OCC 56582,Fc1ccc(Cl)c(F)c1CNc1ccc(C2CCCCC2)cn1 56583,c1(OC)ccsc1C(N1CCC(C(=O)N(CC(C)N(C)C)C)C1)=O 56584,C(=O)(CC(C)(C)C)NC1CC(C(C(=O)NC(c2cnccn2)C)F)C1 56585,N1(C(c2cc(CC)ncn2)=O)CC2CCN(C(=O)C(F)C(F)(F)F)C(C2)C1 56586,C1(NC(Cc2c(C)cc(Br)cc2)=O)COCCN(C(=O)CC(F)F)C1 56587,c1(OC)ccc(C(=O)NCC(C2CC2)NC(C2(C)SCCCS2)=O)cc1N 56588,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56589,c1(C(=O)NC2C(NC(C(C=C)C)=O)CC2)nnc2ccccc2c1O 56590,C1(C(=O)NCCCN(C(=O)C(=O)NCC2CC2)CC)CCCN(S(=O)(=O)CC)C1 56591,N1(C(C(CC)N(CC)CC)=O)CC2=C(C1)CN(C(c1cc3n(c1)CCCC3)=O)C2 56592,C(=O)(C(CCCOC)NC(=O)CC(O)c1ccccc1)NCC1(CCC)CCC1 56593,C1(C(N2CCNCC2C)=O)(NC)CCSCC1 56594,C1(NC(C2(NC(CC(C)O)=O)CC(O)C2)=O)CCN(C)C1=O 56595,Cc1c(CN2CCCCC(NC(c3ccn(C(C)(C)C)n3)=O)C2)ccc(F)c1F 56596,CC(C)C(F)(CNC(C1(CCO)CC1)=O)C(=O)Nc1cn(C)nc1C1CC1 56597,C=CC1(C(=O)NC(C)CN(C(C2C=C(C)CS2)=O)CC)CCOCC1 56598,c1(N(CC(F)(F)F)C(=O)NC2CC(SC)C2)ccc2c(c1)OCCO2 56599,N1(C(C(C)OCCCC)=O)CC(C(=O)NCC(N2CCCCC2)C)OC(C)C1 56600,C1(CC)C(C(=O)NC2(CCO)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56601,N1(C(C2CN(C(C3C(C(C)C)CCO3)=O)CC2(F)F)=O)CC2(C(N)=O)CCC1CC2 56602,c1(C(=O)NCCCC(C)NC(C2C3COCC23)=O)cc2c[nH]cnc-2n1 56603,CCC(C)(C)C(=O)N1CCC(C(C)CNC(=O)Cc2csnc2C)CC1 56604,N#Cc1cc(Cl)cnc1N1CCCC(NC(C2CC(O)C2)=O)CC1 56605,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(c2scnc2C(C)C)=O)CCC1F 56606,Cc1cc(CNC(c2conc2CNC(=O)C(O)C(C)(C)C)=O)cnc1F 56607,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(=O)CSC(F)F 56608,CCC(C)(C)C(C)CC(=O)NC(C1CCCN1C(C1CC1C(C)(C)C)=O)C 56609,C(Cc1cnc[nH]1)(C(=O)NCC1CC1c1ccsc1C)NC(C(=O)NC(C)C)=O 56610,c1(S)nc(C(=O)NCCN(CC(C)O)C(=O)COC)cs1.C1(SCOC)CCOC1 56611,C=CCC(C)C(=O)NC1CCN(C(c2ccc(-c3ccc(F)cc3)s2)=O)CC1 56612,C(=O)(C(C)CCCC(C)C)N1C(C(N2CCC(SC)C2)=O)CC(F)CC1 56613,c1(NC(C2CC(NC(Cc3ccc(C)cc3Br)=O)C2)=O)ccc(C#N)c(Cl)c1C 56614,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56615,C1(C(=O)NCC(C2(O)CN(C(C(C)=C(C)C)=O)C2)(C)C)CC=CCC1C 56616,N1(C(CC(CC)SC)=O)CCC(C)CC1CNC(c1cnoc1-c1ccco1)=O 56617,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 56618,N1(C(CC(=O)NCC#C)=O)CCC(C)(C)C1C(N1CCC1(C)CCO)=O 56619,c1(NC(C(C(C)C)NC(C=CC)=O)=O)cnc(Cl)nc1C 56620,C1(OC)CN(C(=O)CC2CCOCC2)C(C)(CNC(=O)Cn2cnnc2O)C1 56621,C(C(C1CCCCC1)NCc1ccc(S(C)(=O)=O)s1)(C(C)C)NC(=O)C(N)=O 56622,C=CCC(C)(CC)C(=O)NC1CN(C(=O)CCC2CCCC(=O)N2)CC2(CC2)C1 56623,N#Cc1ccc(CCNCc2nnco2)cc1 56624,C(=O)(C(CC(C)C)C(N)=O)NCCC1CCN(C(C(F)=CCC)=O)C1 56625,n1(CC)cc(C(=O)NCC23CC(CN2C(=O)CSC)C3)c(C(C)C)n1 56626,c1(C(C(=O)NC)C)cn(CCCOCCNC(c2cnn(CCOC)c2)=O)nn1 56627,c1(CC)[nH]ccc1C(=O)NC(CC1CC1)C(=O)NCC1CC1(F)F 56628,c1(C(N(CCC)C)=O)ncnc2sccc12.c1(NC(C=C(C)C)=O)cc(C)on1 56629,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 56630,n1(CC#C)ccnc1NC(=O)N(C1CC(F)(F)C1)C(c1ccccc1)CC 56631,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 56632,c1(C(N2CCN(C(c3c(C(C)=O)cncc3)=O)CC2)=O)cnc(N(C)C)c(Cl)c1 56633,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 56634,N1(C(=O)Cc2cscn2)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 56635,c1(N2C(C3CCN(C(c4ccns4)=O)C3)CCC2)nc(Cl)nc2[nH]ccc12 56636,C1(CC(=O)N(c2ccccc2)C)C(=O)NCCN1Cc1ccncn1 56637,C1(OCC)(CNC(=O)CCc2cnoc2)CCN(C(=O)C(C)n2cccc2)C1 56638,N(C(=NCc1coc(C)n1)N1CCC(C(C)(C)O)C1)C(COC)C 56639,Cc1nc(N2CSCC2C(=O)Nc2cnc(I)cn2)c2cc[nH]c2n1 56640,C12(NC(C=CCN(CC)CC)=O)CC(C(=O)NCCc3cccnc3)(C1)C2 56641,C1(CNC(c2nnnn2C2CCC2)C2(c3ccoc3)CC2)CC2(CCC2O)C1 56642,N1(C(CSCC(N)=O)=O)CCC(CCCNC(c2cccc(CCO)c2)=O)CC1 56643,c1(C(N2CC(C(N)=O)(CNC(C3(N(C)C)CC3)=O)C2)=O)cc2ccccc2s1 56644,Cc1cc(C(=O)NC(C2CCCCC2)CNC(=O)CCNC(=O)CO)ccn1 56645,c1(OCC)ccc(NS(=O)(=O)CC2CCC2)cc1Cl.N12CC3CC3(C1)C2=O 56646,N1(C(C2=C(C)CC2)=O)CCn2nnc(C(N3CCC(C(C)O)C3)=O)c2C1 56647,CC1COCCN1CCNC(=O)CNC(C1CC12CC(O)C2)=O 56648,CP(C)(=O)C(O)C(=O)N1CCC(CCCCNC(C2CCCC(=O)O2)=O)CC1 56649,NS(=O)(=O)CCCC(=O)N1CCN(C(=O)CCCN2CCCCC2)C2CC12 56650,c1(OC)cc2ccc1OCC(=O)NC2C.c1(Nn2cncn2)ccc(C)cc1Cl 56651,c1(OC)c(F)cc(C(=O)NC2CCC2NC(=O)CC2CC(C)(C)CO2)c(N)c1F 56652,N1(CC(C)NC(=O)CN(C)C2CC2)CCN(C(C2CCCSC2)=O)CC1 56653,CC12CCCC1N(C(=O)CCC1C3CN(C(=O)Oc4ccccc4)CC13)CCC2 56654,c1(OC)c(CNC(=O)NCC2C3CCC23)nc(O)nc1O 56655,C1=CC2CC1CC2CNCCn1cccn1 56656,C1(C(N2C(CN(C)C(c3ccc[n+]([O-])c3)=O)CCC2)=O)OC2CCC1CC2 56657,C(=O)(C(F)(F)C(F)F)N1CCC(CCNC(C(C)n2cccn2)=O)CC1 56658,c1(C(N2CC(C(C)NC(C(C)NC(CC)(C)C)=O)C2)=O)cc(F)cnc1OC 56659,C#CCC(CCCO)NC(c1cc(CCNC(=O)CC2CNC(=O)O2)on1)=O 56660,N1(c2nc(SC)nc(Cl)c2N(C)C)CCOc2ccccc2C1 56661,c1(SCC(=O)NC2CCN(C(C3CCCC3O)=O)C2)n[nH]c(O)n1 56662,C(=O)(CCCN1CCCCC1)N(C1CC(CNC(=O)CNC(N)=O)C1)C 56663,C1(C(=O)NCC(CNC(C2(N3CCCC3)CCC2)=O)OC)CC(C)CC(C)(C)C1 56664,c1(NC(N2CCC(CC3CC3)C2)=O)ccc(C(F)(F)F)cc1O 56665,CCCC(CC(C)C)C(=O)NC1CCC(NC(=O)C(c2cccnc2)N(C)C)CC1 56666,c1(-n2cc(C(N(CCCCC)CCCC)=O)nn2)ccc(F)cc1C 56667,CN1CCN(C(=O)CCCC2CCCC2)C(CNC(c2nscc2N)=O)C1 56668,C=CCC(CNC(=O)CCC(=O)N(C(C)CC)C)C(=O)N(C(C)CC)C 56669,c1(C(=O)NC(CC)CNC(c2cccnc2)=O)nn(C)c(Cl)c1I 56670,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 56671,Cn1cc(Cl)c(CNC2CC(C(=O)Nc3cnccc3CO)C2)n1 56672,C1(CC(=O)NCC(C)NC(=O)CC(c2cccc(F)c2)O)CCCCCC1 56673,CC(C)C1=NOC(C(=O)NCCOCCNC(=O)Cn2cc(Br)cn2)C1 56674,Cc1cc(NC(=O)NC(Cc2ccc(Br)cc2)CC(=O)O)c(C)s1 56675,CC1CCC=C1C(=O)N1CCCC(N(C(=O)Cn2ccc([N+](=O)[O-])n2)C)C1 56676,c1(CNC(C2C(C(C)C)CCO2)=O)cnn(C)c1C(=O)NC(C(C)C)C1CC1 56677,C1(C(=O)OC2(COC)CC2)CC12CCN(C(=O)OC(C)(C)C)CC2 56678,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)nc1)=O 56679,c1(CC(N2CC3N(C(Cc4n(C)ccn4)=O)C3C2)=O)noc2ccccc12 56680,CC1(C)CCC(C(=O)NC(N2CCCC(C(F)F)C2)c2ccccn2)C1 56681,C(=O)(CCCCCCC)N1CCN(C2C(NC(C(C=C)O)=O)CCC2)CC1 56682,C(C)(C)(C(C)CC(=O)N1CC(Oc2cnc(S)nc2)C1)NC(COCCC)=O 56683,C1(CS(=O)(=O)NC(C)Cc2cccnc2Cl)CCC2(CCCC2)O1 56684,CC(O)CCCNC(=O)CC1CCCC1NC(=O)Cc1ccsn1 56685,c1(C(=O)OC(CC)C)cn(C)c(=O)cc1OC 56686,N1(C(CC(CC)C)=O)CCCC2(CCN(C(C)C(=O)NCC(C)C)C2)C1 56687,c1(-c2cn(C(C)CC)nn2)cccc(N2CCCC2CCc2ccccc2)n1 56688,c1(CC(=O)NC(CNC(C2(C(C)C)CC2)=O)CO)ccc2c(c1)CCCS2 56689,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(C(C)C)C2)=O)CC)C1 56690,c1(C(N2CCN(c3cccc(C4CC4)c3)CC2)C(=O)NC)ccc(F)c(OC)c1 56691,C1(CNC(COCC=C)=O)C(C)CCN1C(c1ccsc1-n1cnnn1)=O 56692,c1(C(N2CC(=C(CNC(C3CC(SC)C3)=O)F)C2)=O)ccnc2ccc(F)nc12 56693,N(C1CN(C(=O)CC2CCCO2)Cc2ccccc21)C(CS(=O)(=O)NCC)=O 56694,c1(C(N2CCC(NC(c3ccoc3Cl)=O)C2)=O)ccc2occc2n1 56695,c1(NC(CC(=O)NC)=O)cccc(C(N2CCC(CN(C)CCC(C)C)C2)=O)c1 56696,Cc1cc(CNc2ccc(Sc3cccnc3F)cc2)ccc1N1CCOCC1 56697,C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 56698,C1(=O)C(C)C(C)CN1.c1(C(N(CCC)CCO)=O)ccc(OCC2CC2)nc1 56699,C(=O)(C(O)C(C)(C)CC)N1CCC(NC(N(c2cc(O)ncn2)CCC)=O)CC1 56700,C1(CC=C)N(c2ncnc(NCCC(O)C(C)C)c2C)CCCC1(C)C 56701,Cn1ncc2nc(Cl)nc(N3CCC(NC(=O)CCC(N)=O)C34CCC4)c12 56702,C1(NC(c2ncn(CCNC(C3C(C(C)C)CCC3)=O)c2)=O)CCC(O)C(O)C1 56703,C(=O)(C(C)C(C)(C)C)NCC1N(C(CCCc2c(C)ccs2)=O)CCCC1 56704,c1(C(c2n(CCCSC)nnn2)NCC(C)(C)C(F)(F)F)cccc2c1CCO2 56705,CC1CCN(C(c2cnc(N)c(O)c2)=O)CCN1C(=O)Cn1c(C2CC2)nnc1O 56706,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(C3)C2)=O)cc(Cl)ccc1N 56707,C(=O)(CC1=CCCCC1)N1C(C(N2CCSCC2)=O)CCC(C)C1 56708,C1(C(=O)NC2C(C)CCN(C(c3cccs3)=O)C2)CCC2CCCCC2C1 56709,N1(C(C2(NC(C3CC(CC)(CC)C3)=O)CC(CO)C2)=O)CC2CCCCC12C 56710,c1(-c2c(C(=O)NC(C(C)NC(CCCC)=O)C)[nH]cc2)ccc(Cl)cc1 56711,N1(C(C(CO)NC(C(CC)CN(C)C)=O)=O)CCC2(CCOC2)CC1 56712,C(=O)(CCCCCSC)N(C(C(=O)NC1C(C#C)CCC1)C)CC 56713,c1(C(N2C3CC(NC(CC=C=C)=O)(C3)C2)=O)cc(C(C)C)cc(Br)c1 56714,C#CCC(CO)NC(c1n[nH]cc1CNC(c1c[nH]cc1C(C)C)=O)=O 56715,C1(CN(C(C2C(CC)C2)=O)CC)CCCN1C(=O)C(n1nccc1C)C 56716,N1(C(CSC(C)C)=O)CCC(NC(C2(C)CC(O)CN2C)=O)C(F)C1 56717,C1(C(=O)NCC2(SCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 56718,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(=O)C(C)SC)C(C)C1)OC 56719,C(=O)(C#CC(C)(C)CNC(c1cnn(C2CC2)c1)=O)NC(CCC(=O)OC)C 56720,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 56721,c1(C(N(C(=O)CNC2CCN(C(CCSCC)=O)C2)C)=O)ccc(Cl)cc1 56722,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2C=CCOC2)=O)o1 56723,C1(NC(C2CCC(CCC)CC2)=O)CN(C(=O)C(F)Cl)CCC1(F)F 56724,C1(C(=O)NC2CN(C(CCC(=O)OC)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 56725,C(=O)(CC(C)C(=O)N1CCC(CNC(c2cnc(S)nc2)=O)C(C)C1)OC 56726,C1(CN(C(CC2(N(C)C)CC2)=O)C)OCCCC1(C)C.C1(C2CC2)C(=O)N1 56727,N1(C(C2N(C(C)C)CCC2)=O)CCCCC1CNC(=O)CC(O)CN(C)C 56728,Cc1ccc(S(=O)(=O)N(C2CN(C(c3c(C(F)F)cccc3F)=O)C2)C)cc1C 56729,CCC(O)C(C)(C)C(=O)NCC(C)CNC(c1csc(-c2ccc(Cl)cc2)n1)=O 56730,C(=O)(C(CCCOC)NC(C1CC(=O)NC(=O)N1)=O)N1C(C)(COC)CC1 56731,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 56732,N1(C(COC)=O)CCN(C(c2c(C(=O)OC)cnn2C)=O)CC1C1CC1.C1CO1 56733,c1cc(Cl)ccc1OC(F)(F)F.C1(C(=O)Cc2ccccc2)COCCN1C=O 56734,C1(NC(C2CCN(C(C(C)OCCC=C)=O)C2)=O)CCC(N(C)C)CC1 56735,C1(O)(COC(c2ccc(C(N)=O)o2)=O)CC2CCC(C2)C1 56736,N1(c2nc(NC(C3(C(=O)N(C)C)CC3)=O)cc(C)n2)CCCC2(CC1)CNC(=O)C2 56737,N#Cc1cc(S(=O)(=O)N2Cc3ccccc3C2)ccc1NCc1ncncc1Cl 56738,C1(C)(NC(C2C(C)C2)=O)CCN(C(c2ncccc2CO)=O)CC1 56739,C1(C(N(C2CC(NC(N)=O)C2)C)=O)CN(C(=O)CCCn2ccnc2)CC12CC2 56740,CC1OCCN(C(C2CC(=O)NC2(C)C)=O)C1C(=O)NC1CSC1 56741,N1(C(C(C)N2CCC2)=O)CC2CC1CN2C(C1CC(C)(C)CN1C)=O.C1(O)CCCC1 56742,C1(CC(=O)NC(CC=C)CNC(=O)CCc2cnco2)CCCC(C)(C)CC1 56743,C1(NC(C2C(=C)C2)=O)CCC2(CC1)CC2NC(c1ccc2nn[nH]c2c1O)=O 56744,Cc1cccc(C)c1Sc1nc(CC(F)(F)F)ns1.N12CCC(C1)N(C)CC2=O 56745,N1(C(C(C(CC)C)OC)=O)CCN(C(=O)CCCN(C)C)C2(CCC2)C1 56746,N1(C(CCCOCC)=O)CCCCC1.c1(CCC(=O)NC(C)C)ccc(Cl)cc1 56747,N1(C(C(C)C#N)=O)CCOCC1CC(=O)N(C)CC1(O)CN(C)C1 56748,C1(C2N(C(CCCC)=O)CCC2)CCCN(C(=O)CCOCC)C1 56749,C1(C)(CCCC(=O)NC(c2ccc(OC(C)=O)cc2)CC)NC(=O)NC1=O 56750,C12(CNC(c3sccc3Cl)=O)CN(C(c3ccc(O)cc3F)=O)CC1CCO2 56751,c1(C(C(=O)NC2CC(CNC(C3(CC(C)O)CCC3)=O)C2)C)ccccc1 56752,n1(CC(=O)NC2CCCN(C(C3N(CC)CCC3)=O)C2C)ncc2cccnc12 56753,C(c1cccc(C2OCCO2)c1)=CC(N1CCNCC1C1CCCCC1)=O 56754,N1(CC)CCN(c2cc(Cl)ncn2)CC1.C1(NC(=O)OC)CCN(C(C)=O)C1 56755,N1(C(CCCC(=C)C)=O)CCC2(CCCC2NC(c2[nH]nc3ncccc23)=O)C1 56756,CCCC(CN=c1ccc(S(=O)(=O)N2CCCC(O)C2)c[nH]1)OC 56757,c12ncc(cn1)[nH]c2=O.C1(CC)(NC(=O)COC(C)C)CC(F)(F)C1 56758,CC(C)C(CNC(=O)CCC1CCCCO1)NC(=O)CCCN(C)C 56759,C1(C(NOCC(CC)C)=O)CCCN1C(=O)CCOCCCOC 56760,c1(OC)cccnc1-c1cn(C2(C(=O)NCC3CC=CCC3)CCOC2)nn1 56761,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCN(C(C2CC23CCSCC3)=O)CCC1 56762,O=C1CCOC(C(N2CCCC2c2cn(CC3COCCO3)nn2)=O)C1 56763,C1(CNC(CCN(C(c2ccc(CC#N)cc2)=O)CC)=O)CCCN(CC)C1 56764,C1(C(=O)OC)CNCCCN1C(C1CSCCN1c1ncccn1)=O 56765,N1(C(C2(CCC=C)CN(C(=O)C(O)C(C)C)C2)=O)CC(C)(C)C1COC 56766,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 56767,CC1(CNC(=O)CCC2C(=O)NN=C2C)CCCN1C(c1cccnc1O)=O 56768,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-c2nc[nH]n2)sc1C(C)C 56769,CC(C)C#CC(=O)NCCCCNC(=O)CC(C)NC(c1ccco1)=O 56770,c1(CC(C2CC=CCC2)NC(=O)NC(C)(CCl)c2ccco2)nncn1C 56771,C1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 56772,c1(N2CCCC(CNC(C3(OC)CCCC3)C)C2)ccc(C#N)cc1[N+](=O)[O-] 56773,Cc1ncc(Br)c(N2CC(C)(CC(N3CC(O)C(F)C3)=O)C2)n1 56774,C(=O)(CCS(=O)(=O)C1CCCCC1)N1CCC(NC(c2ccc(C)cc2C)=O)C1 56775,Cc1nscc1C(N1CC=CC1CNC(=O)C(c1ccccc1)N1CCCC1)=O 56776,C1(OC)CN(C(=O)CC2(C)CCOCC2)CC1NC(C1(NC(C)C)CCOCC1)=O 56777,c1(C(=O)NCCNC(CSC2C(C)CCC2)=O)cccc(CCO)c1 56778,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 56779,C(=O)(CC(C)CC(=O)N1CC(=O)CC1C(N1CCOC(C2(C)CC2)C1)=O)OC 56780,C1(C(=O)NCCC(COC)(C)C)CCC(C)(C)N(C(=O)Cc2ccsn2)C1 56781,c1(CC(=O)NC(CCCC)CNC(C2CC(C)(O)C2)=O)cnc2ccccc2c1 56782,C1(CC)(NC(C2C(C)C2C)=O)CCCN(C(c2ncc(OC)cn2)=O)C1 56783,CC1=C(C(=O)NC(CNC(=O)CCCC2(C)CCC(=O)N2)CC(F)(F)F)CCO1 56784,Cc1nnc(O)c(C(=O)NCCCCN(C(=O)Cc2cn3ccsc3n2)C)c1C 56785,CC1(C)CC(CNC(=O)CNC(=O)C(C)(C)C)N(C(=O)CC2SC(=N)NC2=O)C1 56786,c1(CC(=O)NC(CC(C)C)C(=O)OC(C)(C)C)c[nH]c2ccccc12 56787,CC1CCN(C(=O)Cc2cccc(F)c2O)CCN1C(C1CC2(CCO1)CC2)=O 56788,c1(C(N2CCC3C(NC(c4cc(=O)cc(Cl)[nH]4)=O)C32)=O)c(F)cccc1F 56789,C(=O)(CC(C)(C)C#N)NC1CCN(C(C)C(=O)NCCN2CCCCC2)CC1 56790,N1(C(C2(CCNC(C3C(C)CCO3)=O)CC2)=O)CCC(C)(CCO)CC1 56791,CC(c1ccccc1)=CC(N1CC(C)(OCC(=O)NCC2CC(C)CO2)C1)=O 56792,N1(C(C(C)(C)c2ccccn2)=O)CCC2C(C1)CN2C(c1c[nH]c(C(N)=O)c1)=O 56793,c1(C(N2C(CNC(C(C)SCCCC)=O)CC2)=O)ccccc1O 56794,CC(C)C(C(C)NC(=O)Cn1cnccc1=O)NC(=O)CCn1cnccc1=O 56795,CN1CCN(C(=O)CC2(C#N)CCCCC2)CC1CNC(c1cnc[nH]1)=O 56796,CC1CCC(O)(c2nnc(NC(=O)NCc3ccc(C(C)(C)C)nc3)o2)C1 56797,C(=O)(C(C)(C)C(=O)NCC(C)(O)CNC(C1CC2CC2C1)=O)NC 56798,c1(N2CC(NC(c3csc(Cl)n3)=O)CC(C)C2)ncc2[nH]ccc2n1 56799,N1(C(C2CN(C(=O)NC)C2)=O)CC2C(CNC(C3CCOC(C)C3)=O)C2C1 56800,c1(C(N2CC3(CCC(CNC)O3)C2)=O)[nH]c2cc(OC)ccc2c1C 56801,c1([SH](C(C)(C)COC)CC(=O)NCC(C=C)O)nnnn1CCCCCC 56802,Cc1[nH]c2ccccc2c1C(=O)NCC1CC(F)CN1C(c1ccns1)=O 56803,C1(C)(C(N2C(C)CN(C(C3CC4(CC4)C3)=O)CCC2)=O)CCc2ccccc2C1 56804,C(=O)(C1CCCn2cncc21)Oc1c(OC)cccc1 56805,Cc1ccc(C(=O)NC2CCN(Cc3ncccc3O)C(C)C2)cc1C(C)(C)C 56806,CC(C(=O)NNC(=S)N1CC2CCN(C)CC2C1)c1cccc(OCC(F)(F)F)c1 56807,Cc1cc2[nH]c(C(N3CC(O)(CNC(=O)CCc4ccc(O)nc4)C3)=O)cc2o1 56808,c1(C(=O)NCC2C(NC(C(C=C)(C)CC)=O)CCCC2)cc2c(F)cccc2[nH]1 56809,C(CCCCNC(c1cnn(CCF)c1)=O)N(C(=O)Cc1cncnc1)C 56810,C1(NC(=O)CC2(O)CCCCC2)CCN(c2cc(C(F)(F)F)ncn2)CC1O 56811,c1(NC(c2cc(C)ns2)=O)ccc(CNC(=O)COC2CCCOC2)cc1 56812,CCCC(CC)CC(=O)NC12CCC(CC1NC(=O)COCCCOC)C2 56813,c1(CNC(CC(CCC)O)=O)cccc2c1CN(C(c1cn(CCC)nn1)=O)C2 56814,c1(CCCC(=O)N(CCN(C(CC=C(C)C)=O)C)C)ccccc1Br 56815,Cc1nn(C)c(Br)c1C(N1CCCC(c2cc[nH]n2)C1)=O 56816,C(=O)(C#CC1CC1)N(C1(C(=O)NCC2C(OCC)CC2)CC1)CC1CC1 56817,C1(C(=O)NCCc2cccc(C)n2)C2CCC(C2)N1C(c1c[nH]ccc1=O)=O 56818,c1(C(C)C)cc(C(=O)NCC(C(C)C)NC(c2ccnnc2O)=O)cc(O)n1 56819,C1(NC(=O)COC2CC(F)(F)C2)CCN(C(c2csc(O)n2)=O)CCC1CO 56820,N1(C(C(C)OCC)=O)CCC(NC(=O)CNC(C2CCOCC2)=O)C12CC2 56821,O=C(C1=CC2(CCOCC2)C1)NC(c1ccc(Cl)c(F)c1)CO 56822,C(N=c1ccnc(NCC#CC2CC2)[nH]1)CC(C)C.C1CC1 56823,C1(C)(C(N(CC(C)SC)C)=O)CCCN1C(c1sccc1CO)=O 56824,n1(CC)ncc(C(=O)OCC2CC2c2cocn2)c1C 56825,CC(C)CCCC(C)NC(C1CC2(C1)CN(C(=O)Cc1noc(C(C)C)n1)C2)=O 56826,C1(C(=O)NCCCCNC(c2ccnn2-c2ccncc2)=O)(CC)CC1(F)F 56827,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 56828,CCCCCCCCC(C)NC(C1CSCCN1Cc1ccc(C2CC2)o1)=O 56829,C=C(C)CC(C(=O)N1CCC2(CC2NC(c2cccnn2)=O)C1)OC 56830,C(CS(=O)(=O)CC(=O)NC1CC2CC1N(C(C1CCc3nc[nH]c3C1)=O)C2)OC 56831,c1(N(CCC(=O)N(C)CCN(C(=O)CSC2CCC2)C)C(C)=O)ccccc1F 56832,c1(C(=O)NC2(N(C(C=CC=CCC)=O)C3CC3)CCCC2)ccc(F)cc1 56833,C1(CC(=O)NCC(CNC(c2c(C(=O)OC)csc2)=O)CO)CC=CCN1C 56834,CCC(C(=O)N1CCC(CC)(NC(=O)CCc2ccccc2Cl)CC1)C(C)C 56835,c1(NC(=O)NC(C(CC)C)c2ccccc2)ccnc(Br)c1 56836,N1(C(C(C)OCc2ccccc2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 56837,CCC(CCCO)NCc1cccc(OCC(F)(F)F)c1 56838,CCC(CC)(CO)C(=O)NCC1CCC2(CN(C(c3sc(F)cc3C)=O)C2)O1 56839,Cc1cc(C(C)C(=O)NCC2CCN(C(=O)C(C)(C)CF)C2)c(C)o1.C1C(=O)N1 56840,c1(C(N2CC(C)C(NC(=O)COCC3CCCO3)C2)=O)cnc2ccccn12 56841,c1(C(=O)NC(C(C)(C)NC(C(C)NC(C)=O)=O)C)c[nH]c2ccc(F)cc2c1=O 56842,C1(N(C(c2cn(CCCC)nn2)=O)C)CCCN(C(C2CCCOCC2)=O)CC1 56843,C(=O)(CC1=NNC(=O)C1)NCC1C(CNC(c2ccnc(C)c2O)=O)C1(F)F 56844,C1(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 56845,N1(CC(=O)NCCOCCCN(C)C(C2C3CC(=O)CC23)=O)C(=O)CCCC1=O 56846,C(=O)(C(C)S(C)(=O)=O)Nc1cccc(CNC(C2OCC(C)C2)=O)c1 56847,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CNC(C2CCCCC2)=O)CC(O)C1 56848,N1(C(C(CCC)O)=O)CCC(C)CC1CNC(c1ccc(SCC)cc1)=O 56849,N1(C(C(C)SC(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 56850,N1(C(C(COC)O)=O)CCC12CN(C(=O)CC1(C)CCOCC1)C2 56851,c1(OC)c(Cl)cc(C(=O)NC(C)CN(C(=O)CC23CC(CCO2)C3)C)cc1Cl 56852,CS(=O)(=O)CCC(=O)NCC(C1CCOC1)NC(c1cocn1)=O 56853,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 56854,n1(CCC(=O)NCC2N(C(C(C)C(C)(C)C)=O)CCCC2)cnc2ccccc12 56855,CCC(C)CCC(=O)NC(Cn1cncn1)C(=O)NC1CC(C#N)C1 56856,c1(NC(C(N2CCN(CC(=O)OC)CC2)=O)=O)[nH]c2c(c1C)CN(C(C)=O)CC2 56857,c1cccc(C(=O)O)n1.N1(C(C2CCN(OC)C2)=O)CCC(CC(=O)NC)CC1 56858,C12(C(N3CC(NC(C(CC)n4cccn4)=O)C3)=O)CC(CN1Cc1ccccc1)C2 56859,C(=O)(CC(C)(C)CN(C)C)N1CC(OCC)C(NC(=O)CSc2nnc(S)s2)C1 56860,N1(C(c2c(C)noc2C)=O)CCC(C(=O)NC2CCCSC2)CC1(C)C 56861,n1(CC(=O)NC(C)CCNC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 56862,Cc1cc(CNC(=O)NCCCC2CCC2)nc(C)c1 56863,Cc1n[nH]c(C)c1OCC(=O)NCC1(F)CCC(NC(c2cc(Cl)n(C)n2)=O)C1 56864,CCCCC(O)C(C)C(=O)NC(C)C(=O)NCc1ncc[nH]c1=O 56865,C1(CNC(C(CC)n2cncn2)=O)CN(C(C2CC(n3cnnc3)C2)=O)CCO1 56866,n1(C(C(=O)N(C(CNC(c2c(CC)n[nH]c2)=O)C)C)C)cnc(C#N)n1 56867,C(=O)(C(C#N)CCc1ccccc1)N(c1c(C)cccc1)CCO.C(CCN)S 56868,CC1CC=C(C(=O)N2CC(NC(C3(CF)CC3)=O)CC2(CO)CCC#N)CC1 56869,C1(C(=O)NC2CC3(CCC3)C2)CCC2(CN(C(c3cncs3)=O)C2)O1 56870,Cc1[nH]nc2c1CC(C(N1CC(C(N)=O)(CNC(C3COC(=O)N3)=O)C1)=O)CC2 56871,N1(C(=O)OC(C)(C)C)CC2(CC(=O)NCC2O)C1.C1(N(CC)CC)CCC1 56872,Cn1nc(C(=O)NC2CC(OCC(=O)NCC3CC3)C2)cc1C#N 56873,c1(C(=O)NCCOCCCNC(C2(C)CCCS2)=O)cn2cccc(F)c2n1 56874,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1nccc(CO)n1)=O)CC2 56875,c1(C(=O)NCCCN(C(CC2(COC)CC2)=O)C)cc(C#N)ccc1C 56876,Cc1ccc(N(Cc2ccccc2N2CCOCC2)CC2CCOC2)c(C)c1 56877,N1(C(C2(C(C)C)COC2)=O)CCC(NC(=O)CN2CCN(C)CC2)C(C)(C)C1 56878,c1(OCC(=O)OCc2ccccc2)cnn(C)c1CCO.C1(O)CCNCC1 56879,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 56880,O=C(N=c1[nH]c(Br)cnc1Cl)c1csc(C(=O)Nc2nc3ccc(Cl)cc3[nH]2)n1 56881,CN1CCC(CO)(CNC(C23CC2CCN3C(=O)C(O)C2CCCC2)=O)C1 56882,C1(C)(COC)CCCN(C(C2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)=O)C1 56883,N1(C(C2C(CC)OCCC2)=O)CC2(C1)CN(C(=O)CCSc1ccccc1)C2 56884,Cc1cccc2c1OCC2C(=O)NCCOC(C)(C)CNC(C1CC1C(C)(C)C)=O 56885,C1(C(=O)NC(c2cn(CC(=O)NC(C)C)nn2)C(C)C)(CO)CCOCC1.C(C)C 56886,C12(C(=O)NCC(CC)SC)C3C4C5C3C1C5C24.c1(CCC)ccccc1C(=O)NC 56887,Cc1cc(C(=O)N(C(CNC(=O)CC2COCCO2)C2CC2)C)cc(C)c1F 56888,CCC(CC)CC(F)C(=O)N1CCCC1CC(=O)NC12CC(C(=O)NC)(C1)C2 56889,c1(COC)nc(N2CCC(NC(=O)Cn3cncc3C)C(F)C2)cc(C)n1 56890,N1(C(c2[nH]cc(CC)c2)=O)CC(C)N(C(c2nc(N)sc2C)=O)CC1C 56891,C1(CNC(c2cccc(C3CCOC3)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 56892,Cc1cc(C)c(NC(C2CC2C(C)NC(c2cc(C)c(N)cn2)=O)=O)cc1O 56893,CCC(C)C(=O)C(=O)NCc1cc(C(N2CCCCC2C(N)=O)=O)no1 56894,C(=O)(CCCC(=O)N1CCOCC1C(=O)NC1CCCCC12CC2)OCC 56895,c1(C(N(C(C)CC(=O)N(C2(CO)CC2)C)C)=O)cc(F)ccc1F 56896,C(CCC(CO)NC(=O)C(C)c1ccsc1)NC(Cc1cc(C(C2CC2)C)no1)=O 56897,c1(C(N(CCNC(c2nc(OC)c(F)cn2)=O)C(C)C)=O)c(Cl)oc2ccccc12 56898,C(=O)(C#CC(C)(C)C)NC(CC)CN(C(=O)C(c1ccc(C)cc1)OC)C 56899,c1(C(=O)NC(C(C)NC(=O)C=CC2CC2)CO)cc([N+](=O)[O-])n[nH]1 56900,C1(OC)CN(C(=O)N=C(C)C2CC2)CC12CC2 56901,CC(C)C(F)C(=O)NCC(C1CCN(c2nccnc2F)CC1)(C)C 56902,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 56903,c1(CNC(C(F)=CC)=O)csc(CNC(c2ccnn2CC#N)=O)n1 56904,c1(CNC(COCC)=O)cccc(CC2CC2C(N2CC(CO)C(C)C2)=O)c1 56905,C1(C(N2CCCC(NC(CCC(=O)NC)=O)(CO)C2)=O)OC(C)(C)OC1(C)C 56906,CCC(C)CC(C)C(=O)N1CCCC(NC(C2(CO)CCOCC2)=O)C1C 56907,CC(C)C(C(=O)N1CCC(CO)C1)C(C)NC(c1nnsc1N)=O 56908,N1(C(c2cn(CC(=O)OCC)nn2)=O)CCCN(C(C2CCS(=O)(=O)C2)=O)CC1 56909,c1(CN(C(C(CSCC)NC(C2CSC2)=O)=O)C)ccccc1O 56910,Cc1n[nH]c(C)c1CCC(=O)NC1CC1CNC(c1c(C2CCC2)cnn1C)=O 56911,CC1(C)COC(C(=O)NCC2(CNC(=O)Cc3ccns3)CC2)C1.C1CO1 56912,C1(NC(COCCCC(C)C)=O)CCCN(C(c2ncccc2F)=O)C1C 56913,c1(NC(=O)OC(C)C)ccc(NCCC(C)NC(C2(C(N)=O)CC2)=O)cc1F 56914,c1(C(N2CCCC(C(C)NC(CC=C=C)=O)C2)=O)c(OC)cccc1Cl 56915,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 56916,c1(CC2CCN(CC=CCNC(=O)Cn3ccnc3)C2)ccccc1Br 56917,C1(NC(Cc2c(SC)cccc2)=O)CC2(CCCCN2C(=O)CCn2cnnn2)C1 56918,N1(C(C=CC)=O)CCCC(O)(CNC(c2cnc(CN3CCOCC3)s2)=O)C1 56919,c1(CC)cn2c(n1)CC(C(=O)NCC1CC(NC(=O)CC3CCOCC3)C1)CC2 56920,C(C(=O)N1CCCO1)SCCNC(c1cc(Cl)ccc1C(F)(F)F)=O 56921,c1(CC)oc2ccccc2c1CC(=O)NCC(C)N(C)C(c1ccnc(O)c1)=O 56922,C12(C(N3CC(C)C(NC(c4ccnc(O)c4)=O)C3)=O)CCCC1CCC2 56923,N1(C(c2ccc(C)cc2)=O)CC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)CC2C(=O)O 56924,N(C1CN(C(=O)C(c2ccc(Br)cc2)F)Cc2ccccc21)C(=O)CO 56925,N1(C(CC2CC(C)C2)=O)CCC(NC(c2ccccc2CN2CSCC2=O)=O)CC1 56926,C1(n2cc(CNC(C)COCc3ccccc3)nn2)(C(=O)OC)CCOCC1 56927,C(=O)(C(C)C(=O)NC1CCCC(NC(=O)C(Cl)=CCl)C1)OC 56928,c1(C(c2n(C(CC)(C)C)nnn2)NC2(C)CCC2)ccc(F)cc1Br 56929,c1(-c2c(C)nccc2)c(NCc2cccc(Br)c2F)nn2c1CCCC2 56930,C1(C(=O)NCC(CCNC(C(C)=C2CC2)=O)O)CCCCCC1 56931,C1(C(=O)NCC(C)N(C)C(c2csnc2Cl)=O)CCCCC12CCC2 56932,C1(CC(N2CCC(C(C(=O)NC(CC)CSC)C)CC2)=O)COCCOC1 56933,C12(CCSCC1)c1n(nnn1)CCSC(C)C(=O)N2.c1(CSC)ccccc1F 56934,CC1(C(=O)NCC2(NC(=O)Cc3cccc(C(F)F)c3)CCC2)CCCCCC1 56935,N1(C(Cc2ccc(C=O)cc2)=O)CCC2(CCCCO2)CC1 56936,c1(NCc2onc(C(=O)OC)n2)ccc(C(C)(C)OC)cc1 56937,C(C(C)(C(C)C)NC(C1CNC(=O)N1)=O)NC(c1c(CC)scn1)=O 56938,C1(NC(c2c(CC)c[nH]c2)=O)C2CCN(C(c3cc(O)nn3C)=O)C12 56939,c1(NC(CCN(C(=O)CCN(C2COC2)C)C)=O)cncc(CO)c1 56940,C(=O)(C(F)CC(C)(C)NC(=O)C1CC1)NCCC(=O)OC 56941,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)Cl)C1 56942,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 56943,N1(C(C2CCC(c3ccccc3)N2)=O)CCN(C(=O)C2CC2)C(CCO)C1 56944,C(=O)(C(CCNC(C1(O)CCCC1)=O)OC)NC(C#C)CC1CCCC1 56945,C=C(C)C(C)(O)C(=O)NC1CCC(N(C)C(c2ccc(CSCC)[nH]2)=O)CC1 56946,C1(C(=O)NCC(C2CC2)OC)CCCCN1C(=O)CN1CC=CC1 56947,C1(C(N2CCCC(CNC(C(C)C3CCOC3)=O)C2)=O)CCCCC12OCCO2 56948,C1(CC2CC(C(=O)NCC)C2)(OC)CCN(C(=O)C(O)Cc2cnn(C)c2)CC1 56949,C1(OC)CC(C(N2CC(CCO)C2)=O)N(C(=O)Cc2ccns2)C1 56950,c1(C(=O)NCC(CC)NC(C2(C)C=CCCC2)=O)cc2n(n1)CC1(CC1)C2 56951,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(CN(C)C(C2CCC3(CCOC3)O2)=O)C1 56952,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 56953,c1(CC(=C)Br)nnc(N2CCC(C(C)C)CC2)n1CCCc1ccc(OC)cc1 56954,C1(F)(C(N2CCCCC(CNC(C3CN(C)C3)=O)C2)=O)CS(=O)(=O)CC12CCC2 56955,N1(C(c2cc(OC)no2)=O)CCC(C)(C)C(NC(c2cc(C3CCC3)[nH]n2)=O)C1 56956,c1(C(N(CC(N2CC(CO)OC(C)C2)=O)CCOC)=O)ccc2occ(C)c2c1 56957,C=CCCC(O)CN(C(=O)C(C1CCCN(C(=O)Cc2nonc2C)C1)(C)C)C 56958,C(=O)(C1=CCCOCC1)NC(c1nc(-c2c(OC)ccc(C)c2)sc1)C 56959,C1(C(=O)N(CC(C)N(C(=O)CCOCC)CC=C)CC)C2CC(=O)CC12 56960,c1cc(F)ccn1.C123CC1CN(C2)N(S(=O)(=O)Cc1ccccc1)C3=O.CCO 56961,Cc1ccc(O)cc1NC(C1COC(=O)N1)=O.C1(Cc2cccs2)CC(=O)N1 56962,c1(CN(C2CCN(C(CCC=C)=O)CC2)CCO)cccc(C#N)c1 56963,C(=O)(C1CCc2c[nH]nc21)N1CCC(CNC(C2N(C=O)CCOC2)=O)C1 56964,CCC(C)(CNC(C)=O)NC(=O)COc1cnn(COC2CCCCO2)c1 56965,c1(C(N(C2CCN(C(=O)CC(C)(C)C)C2)CC)=O)cccc2ncnc(O)c12 56966,CC1(C)CN(C(=O)CNC(C2SCCS2)=O)CCO1.C(N)(=O)NC 56967,C1(O)(C(C)NC(=O)Cc2cnns2)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)C1 56968,C1(S(C)(=O)=O)(C(N(CC(CC)NC(C2CCN(C)C2C)=O)C)=O)CCC1 56969,C1(C(=O)NCCC(C)O)CCC2CCC1N2C(c1cnn2c1CCC2)=O 56970,Cc1ccc(C(C(=O)NC2CCOCC2)N(C)Cc2cocc2Br)cc1O 56971,C(=O)(CCC=CC)NCC(CNC(C1(CCCC)CCC1)=O)OC 56972,c1(OCCC)ccccc1C(=O)N(C)CCNC(C1CCCN1CC(C)C)=O 56973,N1(C(c2ccc(Cl)c(Cl)c2)=O)CCC2(CC1)CN(C(c1ccc[nH]1)=O)C2 56974,c1(C(=O)NCC(C)CNC(=O)CC2CC23CC3)c[nH]c(C(N)=O)c1 56975,C1(N(C(C2CC2(C)C(C)C)=O)CC)CCCN(C(=O)CC2CCSCC2)CC1 56976,C1(N(C(C(C)OCC)=O)C)CCC(NC(c2ccc(=O)oc2)=O)CC1 56977,C(CS(=O)(=O)CCO)NCc1cnc(C(F)F)s1 56978,C1(CN(C(=O)COC2CCN(C)CC2)C)CCCN(C(C2CCC(CO)CC2)=O)C1 56979,c1(C(c2nnnn2C2CCC2)NCC(CF)F)cccc(Br)c1 56980,C(=O)(CCCCCCNC(=O)C(=O)N)N(CCC(F)(F)F)C.CN 56981,CCC(CC)C(C(=O)NC1CC2(C1)CN(C(c1cnc(OC)cc1Cl)=O)C2)OC 56982,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CNC(C3CC3C)=O)CC2)C1 56983,N1(C(C2CCC(CC)O2)=O)Cc2[nH]nc(C(N3Cc4c[nH]nc4C3)=O)c2C1 56984,C(=O)(C(O)C(C)(C)C)NC(c1n(C)ncc1)C(N1CCC(COC)CC1)=O 56985,C1(C(N2C(C3(CNC(C4C(C)=CCS4)=O)CC3)CCC2)=O)CC(=O)N(O)C1 56986,N1(C(Cc2ccc(C(=O)NC)s2)=O)CCCN(Cn2c(Cl)cccc2=O)CC1C 56987,C(c1cn[nH]c1)=C(C)C(=O)NCCCN(C(C1CCC(F)C1)=O)CC1CCCC1 56988,C(CCC(=O)N1CC(OCC(=O)NCC2CC2[N+](=O)[O-])C1)SC 56989,c1(NC(C2(CNC(COC(CC)(C)C)=O)CCC2)=O)cc[nH]c(=N)c1 56990,C1(CNC)CCCCN1C(=O)C(=O)NC1C2CCC=CC12 56991,N1(C(C(CSCC)NC(=O)C=C(CC)CC)=O)CCCN(C)CC1CC 56992,Cc1c(F)ccc(NCC2(O)CCN(Cc3c(C(F)F)nn(C)c3Cl)C2)c1F 56993,CC1CN(C(c2cnc(O)c(F)c2)=O)CC2(CCN(C(C34CC3C4)=O)C2)O1 56994,C1(CC(=O)NC2C(CC)N(C(C3CNC(=O)C3)=O)CC2)CCC2(CC1)OCCO2 56995,CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C(N1CCC2(CC1)CC2CO)=O 56996,c12cc(n[nH]1)C(=O)N1CC(C1)OCCOC2.C(C(F)(F)F)OC1(CC)CC1 56997,c1(C(C(=O)NCC2(C)CN(C(c3cc(F)ccn3)=O)C2)O)ccc(F)cc1 56998,N1(C(C(C)(C)NC(=O)OC)=O)CC=C(C(=O)NCCC2CCCN2C)C1 56999,CC1CC2(CC(C(=O)NCC34CC3CN(C(=O)COc3ccccc3)C4)C2)C1 57000,C=C(F)C1(CC(N2CCCCC2CCN(C)C(c2nc(C)c(C)s2)=O)=O)CCC1 57001,CC(C)C(C(=O)N1CC(O)(CNC(=O)CCN2CCNC(=O)C2)C1)NC(=O)C1CC1 57002,Cc1cnc(Cl)c(NC(C2CCC(NC(=O)Cc3cnc(C)s3)CC2)=O)c1 57003,c1(NC(C2C(NCc3ncc(C)c(Br)c3)CCCC2)=O)ccc2oncc2c1 57004,C(=O)(CC1=CCN(C(c2ccsc2C#N)=O)CC1)NCC1C(OC)CC1 57005,C1(CNC(CN(C2CC2)CC)=O)CN(C(=O)CCc2ncc[nH]2)C2CC12 57006,C(=O)(CC1=CCCCC1)NC(CN(C)C(C1CC(C)(C)CN1C)=O)(C)C 57007,c1(NC(c2ccc(C)o2)=O)cccc(Cn2cc(-c3cc[nH]n3)nn2)c1 57008,C(C(C)C(F)C(=O)N(C)CC1CC(F)(F)C1)NC(Cn1nnc(C)n1)=O 57009,CCCCC(CNC(C1CCN(C(=O)CCCOC(C)=O)C1C(C)C)=O)CC 57010,Cc1cccc(C(N2CC(O)(C(C)(C)CNC(=O)C(O)C3CCC3)C2)=O)c1F 57011,N1(C(C(C(C)(C)C)SC)=O)CCC2(CC1)CC2NC(C1Cc2nnc(C)n2C1)=O 57012,N1(C(C(c2ccnn2C)NC(=O)CC(=O)NCC)=O)CCNC(=O)C1 57013,C1(C(=O)NCC[Si](C)(C)C)(CC)CCCN(C(c2cn(C)ccc2=O)=O)C1 57014,CCCCC(C(=O)NCC(C1CC1)N(C)C)NC(=O)CCNC(=O)CO 57015,c1(CC(=O)NCC2N(C(CSCC#C)=O)CCN(C)C2)cccc2c1OCCO2 57016,c1(OC)cncnc1NCCCOC(=O)CC(C)NC1CC1 57017,C=CCC(CC)C(=O)NCCC1(NC(=O)Cc2csc(-c3ccoc3)n2)CC1 57018,C1(NC(Cc2cc(C)sc2)=O)CC(C)CN(C(=O)CCN2CCCC2)C1 57019,C(CC(O)CNC(C1CCC1n1ccnc1)=O)NC(c1cn(C2CCC2)nn1)=O 57020,Cc1scc(C(=O)NC2CC3C(NC(=O)CCc4nccn4C)C3C2)c1C 57021,N#CC1CCC(CC(=O)N(CCNC(c2nocc2C2CC2)=O)C2CC2)C1 57022,C1(C(=O)NC(c2scc(C)n2)C)CC12CCN(C(=O)Cn1cccnc1=O)C2 57023,C(c1cn(C)c(=O)n1C)=CC(N1CCC(C(C)NC(C2CC(C)(C)C2)=O)CC1)=O 57024,c1(CCNC(=O)NCC2(c3ccc(Cl)cc3)CCCC2)cccc(F)c1O 57025,C(N=c1[nH]c(=NC(C)CF)[nH]c2c1SCC2)C1(SC)CC1 57026,c1(C(=O)Nc2nnc(C3CC3)s2)cc2ncccn2n1 57027,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C)(C)C(C)(C)C 57028,N1(C(C2C(=C)CC2)=O)CC2CCN(C(c3cccc(Cl)c3Br)=O)CC12 57029,CC(CN(C)C)CCC(=O)N1CCC(O)(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C1 57030,Cc1nc2sccn2c1C(=O)NC1CN(C(C2C3(CC3)C23CC3)=O)CC1O 57031,c1(C(=O)NCC(CC)NC(=O)CC2NC(=O)CNC2=O)cc2c(C)ccc(F)c2o1 57032,C(=O)(C(C)S(N)(=O)=O)NCC(CN(C(C(=O)NC(CC(C)C)(C)C)=O)C)(C)C 57033,O=C1CNc2cc(C(N3CCCC(NC(C4CCCOC4)=O)CC3)=O)cnc2N1 57034,C1(NC(=O)C(CO)c2ccccc2)CCCCCN(C(c2nccc(Cl)c2F)=O)C1 57035,C1(C(=O)NC(C)(C)COCCNC(=O)CCc2ccc(F)cc2)CCC=CCCC1 57036,CC(C)(C)C(O)CC(=O)N1CCC2(CC1)CC2NC(=O)OC(C)(C)C 57037,c1(C(CN2CCC(SC)C2)NC(c2cn(C)cn2)=O)cccc(C(F)(F)F)c1 57038,C(=O)(C1CNC(=O)c2ccccc21)N1CCC(O)(CNC(C2CN(C)C2)=O)CC1 57039,c1(C(N2CC(CNC(=O)Cc3cnccc3Cl)C2)=O)cc2n(n1)CCC2 57040,c1(CCC)occc1C(=O)N(C(c1ccccc1)C(N1CC(N(C)C2CC2)C1)=O)C 57041,N1(C(CCSCCC)=O)CC2(CCC(NC(c3coc(C(C)(C)C)n3)=O)CC2)C1 57042,N1(C(=O)Cc2cnsc2)CCC2(CCN(C(=O)Cc3nncn3C)C2)C1.c1cc(F)co1 57043,c1(C(N2C(C)CCC(NC(c3ccc(C)nn3)=O)C2)=O)ccc2[nH]c(=N)sc2c1 57044,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57045,Cc1cc(C(=O)N(CC(C)N(C(=O)C=CC2(C)COC2)C)C)ns1 57046,C1(OC)CCC12CC(C(=O)NC1CCCC1CNC(=O)CCc1ccnn1C)C2 57047,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1C(C)NC(C1(C)CCNC1=O)=O 57048,c1(CC(=O)NCCOCC(=O)NCC(CO)OC)cncnc1O 57049,N1(C(CCCNC(=O)OCC(C)C)=O)CC(NC(=O)CC2CCCCO2)C(C)C1 57050,c1(CCNC(c2cc(C(=O)OC)oc2)=O)cn(C)nc1C.C12CC1CC(=O)NC2 57051,Cc1cc(OC(=O)Cc2ccn(-c3ccc(Br)cc3)n2)c(C)nc1C 57052,N1(C(C2COCCN(C(c3ccn(CCC)n3)=O)C2)=O)CCCN(C)C(=O)C1 57053,C1(NC(COCc2ncc(C)o2)=O)CN(C(C2CCC(=O)N2)=O)CCC1F 57054,C=CC1(CNC(=O)CCN(C(=O)CCc2ccoc2)CCO)CCOCC1 57055,Cc1cc(OCC(N2CCCC(C(=O)NCCCO)C2)=O)cc(C)c1 57056,CC#CCC(C(=O)NCCC12CC(CO1)C2)NC(=O)CC(C)OC 57057,c1(CC(N2CCC(C)C(NC(c3ccncc3)=O)C2)=O)ccc2cccnc2c1 57058,N1(C(CCOC)=O)CCCC2(NC(=O)Cn3cc(-c4cccnc4)nn3)CC12 57059,C1(NC(=O)N)CCN(C(CC(C)Oc2ccccn2)=O)C(COC(C)(C)C)C1 57060,c1(C(N)=O)c(F)cc(NCc2ccc(-c3cncnc3)cc2)cc1F 57061,c1(C(N(C)CCC2CCCCO2)=O)coc2c1CN(C(=O)C=CC1CC1)C2 57062,N1(C(C2CCC(C(N)=O)O2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57063,C(=O)(CCCC(C)(C)C)N1CC2(CC(CC(=O)N)C2)C1.CCCS(=O)CC 57064,C1(C)(C(=O)NC(C(C)O)CO)CCCN(C(=O)CCC2CC2C)C1 57065,c1(C(N(CCC)CCN(C)C)=O)ccnc(CNC(=O)C(C)C2CCOC2)c1 57066,C1(C(=O)NC2C(CN(C)C)C2)C2CCC(C2)N1C(C1CC2COCC2C1)=O 57067,c1(C(=O)OC)cncc(C(N2CCC2CNC(C2COC(C(F)(F)F)C2)=O)=O)n1 57068,c1(CC)sc(=N)[nH]c1C(=O)NCCN(C)C(c1cncc(C(F)F)c1)=O 57069,CC12CN(C(=O)CN3CCC3)CC1(C)CN(C(=O)CCc1ccsc1)C2 57070,c1(CNC(C2N(Cc3c(C)n[nH]c3C)C3C(C2)C3)=O)cccc2nsnc12 57071,C1(CNC(COCCCC(C)C)=O)CCN(C(=O)C(c2cncn2C)O)C12CCC2 57072,CC(C(=O)NC1CN(C(=O)COc2cnn(C)c2)CC1(C)C)C(C)(F)F 57073,C=C1CC2(C1)CC(C(=O)N(C1CCN(C(=O)CC3(C)OCCO3)CC1C)C)C2 57074,C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cc([N+](=O)[O-])n[nH]1)=O 57075,c1(NC(C2CCN2Cc2cc(O)ncc2Br)=O)ncnc2occc12 57076,CCC(CC(=O)NC(C)CCCNC(=O)Cn1cnnn1)C1CCC1 57077,c1(N2CC(NC(C(CCC)C)=O)(CSC)C2)ccc([N+](=O)[O-])cc1N(C)C 57078,N1(C(c2c(C)occ2)=O)CCCC(C2(NC(c3ncc[nH]c3=O)=O)CC2)C1 57079,CCCCCCC(=O)NC(C1CCN(C(C2CC2(Cl)C(=O)OC)=O)CC1)C 57080,C1(NC(c2c(C(C)C)cccc2)=O)COC2(CCN(C(c3cnon3)=O)CC2)C1 57081,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57082,C1(N(C)CCO)COc2ccc(CNC(=O)OC(C#N)CCC#N)cc2C1 57083,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C(c2snc(C)c2Br)=O)C(CO)C1 57084,C(=O)(C(C)(CC)CO)N(CCN(C(c1ccc(SC(F)(F)F)cc1)=O)CC)CC 57085,c1(C(N(CCCCCNC(c2n(CC)ncn2)=O)C(C)C)=O)occ2c1CCC2 57086,N1(C(c2c(C)nn[nH]2)=O)C2CCC1CN(C(C1CCOC(C(F)(F)F)C1)=O)C2 57087,C1(C(C)C)N(C(=O)CC2(NC(=O)CC3CCOC3=O)CC2)CC1(C)C 57088,N1(C(CC(C(C)C)NC(=O)Cn2cnnc2)=O)CCN(C)CC(C)C1 57089,CN(C)NC(=O)CCC(=O)NC(C(=O)Nc1ccccc1C1CC1)C1CCCO1 57090,C(=O)(C(C(C)(C)C)OC(C)(C)C)NC(C(=O)NC1CC(C(C)N)C1)=O 57091,C1(C(N(CC(C)O)CCNC(c2cnn[nH]2)=O)=O)CCOC(C)C1 57092,C1(C(NOC)=O)CCN(CCC(C)N)CC(C)(C)C1.N1CCCC1=O 57093,c1(C(c2nnnn2C2CCC2)NCc2snc(C)c2Cl)cccc(F)c1Br 57094,N1(C(c2nc(-c3cn(C)nc3)oc2)=O)CC(NC(=O)CCSCC#N)CC1CO 57095,N1(C(CCc2cnc(C)o2)=O)CCCC(CNC(C2CC2(F)F)=O)CC1 57096,c1(CC(=O)N(C2CC(CNC(=O)Cc3ccns3)C2)C)ccc(Cl)cc1 57097,C(=O)(C1Cc2c(Cl)cccc21)N.N1(CC2(CS(C)(=O)=O)CC2)C2CCC1CCC2 57098,C(=O)(CC(CN(C)C)C(F)F)N(CC(C)NC(=O)CCCCN1CCOCC1)C 57099,CC1CCC(NC(C2CNC(=O)C2)=O)C1 57100,N1(C(c2cc(CNC(CCC(CC)=O)=O)oc2)=O)CCCC(C2CCC2)C1 57101,c1(C(=O)NC(C2CCOC2)CNC(=O)CCC2OCCO2)c(F)cc(F)cc1F 57102,C1(n2cc(CCN(C(=O)CCOC3CCOC3)C)nn2)(CC)CCOCC1 57103,C(CCCCCNC(=O)CC1CCCN1CC)NC(C=CCC)=O 57104,Cn1[nH]c(C(=O)NCC2CCN(C(=O)COCC3(F)CC3)CC2)nc1=O 57105,Nc1ncccc1-c1cscc1C1CCS(=O)(=O)C1.N12CCC(CC1)C1CC1C2=O 57106,c1(C(=O)NCC(CCC)NC(c2cnc([N+](=O)[O-])n2C)=O)cc(F)cc(Cl)c1N 57107,C(=O)(CC(C)(C)c1ccccc1)NCC(Cn1cc(CCCOCC)nn1)(F)F 57108,C1(F)(CNC(C(CC)(C)OC)=O)CCCN(C(=O)C(C)(C)Cc2cnn[nH]2)C1 57109,C1(C(=O)NCC2C(NC(c3nnn(CC)c3C)=O)CCCC2)CC2CCC(C1)C2 57110,c1(-c2cccc(C(OC)OC)c2)cccc2nc(C(=O)NCC3CC3)ccc12 57111,Cc1cnn(C)c1CC(=O)N(CCOCC(=O)NC(C)(CO)CCF)C1CC1 57112,C1(C(=O)NCC(=O)NCCOC(c2n[nH]cc2[N+](=O)[O-])=O)CC(=O)NC(=O)C1 57113,C(c1ccc(O)cc1)=CC(=O)NCC1(F)CCN(C(C2CC(F)(F)C2(F)F)=O)C1 57114,n1(CCC(=O)N(CC(CNC(C2ON=C(CC)C2)=O)(C)C)C)cc(S(N)(=O)=O)cn1 57115,C1(S(=O)(=O)NC(N2CCC(NCC(C3CCCCC3)O)CC2)=O)(CC=C)CC1 57116,n1(C(C)CN(C)C(c2sccc2-n2cnnn2)=O)cc(CCS(C)(=O)=O)nn1 57117,c1(NC2C(C)CN(C(C3(C)CCC(=O)N3)=O)C2)ccc2nnnn2n1 57118,C1(c2n(CC)nnn2)CCCN(C)CC1.C1(NCC2CC2)CCC2(CC1)CC2 57119,c1(CN(C(C)=O)C)cn(C2CCN(C(=O)CC3CN(C(C)=O)C3)C2)nn1 57120,N1(C(C(N2CCC3(OCC(OC)C3)CC2)=O)=O)CCc2ccc(Cl)cc2C1C 57121,C(=O)(CC1=NN(CC(F)(F)F)CC1)NC(C1CCN(C(=O)C(F)C(C)(C)O)C1)C 57122,C1(C(=O)NCCCCN(C(c2cn(C3COC3)nn2)=O)CCO)CC12CCSCC2 57123,N1(C(C(C(C)C)C2CCC2)=O)CCCCC(C(=O)NOCCC(C)O)C1 57124,C(CCCC(=O)N(C1CCC1(C)C)C)N(C(C(C)N(C(C)=O)C)=O)C 57125,O(NC(=O)C(CNC(=O)CC(F)(F)C(F)(F)F)CC(C)C)CC(CC)C 57126,N1(C(C2CCC(=O)N2)=O)CCN(C(=O)CC2COCCOC2)CC1 57127,c1(C(N)=O)cncc(CCC(=O)NCCN2CC3CCC2C3)c1 57128,C=CCC(CNC(c1ccc(CC(C)C)s1)=O)NC(c1csc(C(F)F)n1)=O 57129,c1(C(=O)NCC2(F)CCC(NC(CS(CC)(=O)=O)=O)C2)cn2cc(C)ccc2n1 57130,N1(C(C2CC=CC(NC(Cc3c(C)con3)=O)C2)=O)CCN(C)C(=O)C1CCO 57131,c1(C(=O)NC2C(NC(CC(=C)C)=O)CCC2)cn2cc(Br)cc(C)c2n1 57132,C(N=c1nc[nH]cc1C#N)C1CC(NC(c2ccc(C)nc2)=O)C1 57133,C1(C(=O)NC(C(C)C)CN)CCCN(Cc2ccc(C(C)C)cc2)C1 57134,CS(=O)(=O)c1cc(C(N2CC(NC(c3cnccc3Cl)=O)C3CC23)=O)cc(N)c1 57135,N1(C(CCN(C(C2CCC(=O)CC2)=O)C2CC2)=O)CC2(CCC2)CC1CO 57136,c1(OCCNC(c2cnsn2)C)ccccc1F 57137,c1(COC(C)CN(CC(O)CO)CCC#N)ccccc1 57138,CC1CC2(CO1)CN(C(=O)CC(C1CC1)NC(C1CCCN1C1CC1)=O)C2 57139,C=CCC(CNC(C1CC1(C)C(F)(F)F)=O)NC(=O)C=CC(C)(C)C 57140,N1(Cc2ncc(C)nc2)CCCN(C(C2(F)CCN(Cc3ccccc3)C2)=O)CC1 57141,N1(C(c2n(CC)ccc2)=O)CC2C(NC(c3ccn(C4CC4)n3)=O)C1C2 57142,c1(C(=O)Nc2cc(F)cc(Cl)c2)n[nH]c2cc(C3=CCOCC3)ccc12 57143,c1(C(Cc2ccccc2)NC(=O)NCC(CC)O)ccc(C(C)C)cc1 57144,CCCCCC(CCCCC)C(=O)N(C1CCN(C(=O)C(O)CC2CCCC2)C1)C 57145,c1(CC2CCC2)cc(NC(=O)CCCC2C(OC)C2)cc(N)c1.C12(CC1)C(=O)NC2 57146,C(=O)(CC1=CCOCC1)N1C(C(=O)NCC(c2ccccc2)F)CC(F)CC1 57147,CC1(C)CCCN(C(=O)CCC2CCCCCC2)C1CNC(c1n[nH]cc1F)=O 57148,c1(OC)ccc(C(=O)NCC2(C)CCOC2)c(C)c1OC 57149,C1(CC(N2CCC(N(CCCOC)CCO)CC2)=O)CCn2cncc2C1 57150,N1(C(Cc2nc(C)c(C)o2)=O)Cc2n[nH]cc2C1C(=O)NCC1CCCC(O)C1 57151,CN1CCN2CC1C(N(C1(C)CCCC1)C)C2=O.c1(CC2CCC2)ccccc1 57152,C1(NC(c2c(C(=O)OC)cn(C)n2)=O)CC2CCC1N2C(=O)C(C)NC(C)=O 57153,N1(C(c2ccc(C(=O)OC)o2)=O)CC2CCC2(CCNC(=O)C=C(C)C)C1 57154,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57155,c1(COC(CC(C)CCc2ccccc2)=O)cc(F)c(Cl)cc1[N+](=O)[O-] 57156,CC1CCCCC1Oc1ccc(NC(=O)N(C)C)cc1 57157,Nc1ccc(CN2CCN(Cc3cn(CC4CCCC4)nn3)CC2)cc1O 57158,C1(NC(c2c(C)ncs2)=O)CN(C(=O)CC2CCNC(=O)C2)C2(CCCCC2)C1 57159,S(=O)(=O)(c1ccc2c(c1)N(C(C1CCOC1c1ccccc1)=O)CCC2)NCC 57160,c1(C(=O)NC(C)CNC(C2CCCCCCC2)=O)cccc(S(=O)(=O)C(F)F)c1 57161,N1(CCOc2ccc(OC)cc2)C2CCC1C(CNC(c1cccc(Br)c1)=O)C2 57162,c1(CC(=O)NCC(F)CNC(c2cc(F)n[nH]2)=O)nccc2ccccc12 57163,CC(C)C(C(=O)NCC1(CNC(c2ccccc2)=O)CC12CCC2)N(C)C 57164,C(=O)(C1OCCc2c(O)cccc21)NC(CC)CNC(C12CC3CC1C2C3O)=O 57165,C1(C#CC(=O)NCc2ccc(C(=O)NC(C)CCOC)nc2)(CC)COC1 57166,c1(C(=O)NC(c2c(C(NOCCOC)=O)noc2)C)cccnc1F 57167,c1(C(=O)NC2(C)CCN(C(CC(CC)(C)C)=O)C2)cc2cccnc2nc1O 57168,C(CN=C(NCc1cnc(OC(F)F)cc1C)N1CC=C(F)C1)SC 57169,Cc1[nH]c(C(C)(C)C)cc1C(=O)NCC(C1CCC1)NC(=O)CCC1CC1(F)F 57170,c1(C(CNC(C(C)CF)=O)NC(C2(C(N)=O)CC2)=O)cccc(Cl)c1Cl 57171,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(Cl)Cl)C(CO)C2)=O)C1C 57172,COn1cnc(C)c1C(=O)NCC1COCCN(C(=O)CC=C(C)C)C1 57173,c1(C(=O)NCC(C)CNC(c2ccc(CO)cn2)=O)cc2cccnc2nc1N 57174,N1(COC)CCCCC1C(=O)NC1CC(C)N(C(c2ccccc2OC)=O)C1 57175,C(=O)(CC(C)CC(=O)OC)NCC(CC)(C)NC(=O)CN(C)CCO 57176,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57177,CC(F)(F)C(C)(C)CC(=O)NCC1CCCCC1NC(=O)C1CC(O)CCO1 57178,NS(=O)(=O)CCCNC(C1CCCCN1C(=O)CCc1nc[nH]n1)=O 57179,C(CS(=O)(=O)CC(=O)N(C)C(C1CCCCN1C(C)=O)C1(C)CCCC1)OC 57180,c1(C(=O)NC2CCC3(CN(Cc4c(C)nn(C)c4)C3)O2)cc2cnccc2nc1C 57181,C1(CNC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)COCCOCCO)C12CC2 57182,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)N(C)C)CCC2(CCC2)O1 57183,c1(CC(=O)NC2C3CN(C(C(C)(C)CO)=O)CC2C3)csc2c(F)cccc12 57184,N1(C(C2(CC)CN(C(=O)CC3CC=CCC3)C2)=O)CCC(C)(O)CC1 57185,O=C1CCC(C(=O)NCCC2(NC(=O)Cc3c[nH]nc3O)CC2)CN1 57186,N1(C(Cc2c(C)nsc2)=O)CC2CC2(CNC(=O)C(C)n2ccnn2)C1 57187,c1(C(=O)NC(CNC(CNC(CC)=O)=O)C2CCC2)ccn2c(C)cnc2c1 57188,C1(CN(C(c2c(C)con2)=O)C)CN(C(C2CC2F)=O)CCO1 57189,N1(C(C(C=C)(C)C)=O)CCC(NC(c2oc(C)nc2C)=O)C(F)(F)CC1 57190,N1(C(c2nc(C(N)=O)sc2)=O)CCC2CCN(C(C3C=CCC3)=O)CC2C1 57191,N1(C(C(CC)OC)=O)CCOCC(NC(C2CN(CC)C(=O)N2)=O)C1 57192,CC1(C)CCCN(C(c2cccc(C(F)F)c2)=O)C1CNC(=O)C1=CSCCO1 57193,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57194,C1(C(=O)NC2(COC)CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)CCCCCN1C 57195,Cc1cc2[nH]nc(CNC(=O)NCc3ccc(C#N)s3)c2o1 57196,C(C(C)(O)CC(=O)NCCCCN(C)C(c1c[nH]nc1C(=O)O)=O)OC 57197,Cc1cc(=O)c(C(N2CCC(C(=O)NCC3CC34CCC4)C23CC3)=O)c[nH]1 57198,c1(-c2c(OCC)c(F)ccc2)cccc2sc(C(N3CC(F)(F)CC3C)=O)cc12 57199,C(=O)(C(CNC(c1n[nH]c(C)c1O)=O)C(C)(C)C)NC(c1cnccn1)CC 57200,C1(C(=O)NCC)(NC2CN(C(c3cn(C(F)F)cn3)=O)CC2F)CCOCC1 57201,n1(CC#C)c(C)cc(C(=O)NCC2(CCNC(=O)C(C)(F)C(=O)OC)CC2)c1C 57202,CC1CCN(CC(=O)NCC2CCN(C(c3cc(CN(C)C)on3)=O)C2)C1 57203,Cc1c(Br)ccc(N2CCN(C3CCN(C(C4C=CCC4)=O)C3)CC2)c1[N+](=O)[O-] 57204,Cn1nc(C(N2CC(NC(c3cscn3)=O)CC(O)C2)=O)c(Cl)c1C(F)(F)F 57205,C12(CNC(C(N3CCOCC3)C)=O)CC(CNC(=O)CCc3cn[nH]c3)(CO1)C2 57206,CCC(C)CCCC(=O)NC1CC(CC(=O)OCCC(CC2CC2)CO)C1 57207,Cc1csc(C(C(=O)NCc2nc(C(C)(C)O)n[nH]2)NC(=O)OC(C)(C)C)c1Cl 57208,CCC(CNC(=O)NC1(F)CS(=O)(=O)C1)C(C)C 57209,c1(OC(N2C(COC(=O)Cn3ccnc3)CCCC2)=O)ccc(Br)c(F)c1F 57210,C(CC(=O)N(CC(=O)N(CCCC1CC1)C)C1CC1)SCC 57211,N1(C(CN(C(=O)OCC)C)=O)CCC2CC12C(=O)NC(C)Cn1cccn1 57212,C1(NC(C(C)O)=O)CN(C(=O)Cc2csc(Cl)n2)CC1c1cnn(C)c1 57213,c1(CC)nn(C)c(Cl)c1C(=O)NC(CCNC(C1CC12CCOC2)=O)CC(C)C 57214,N1(CC(N2CC3C(CNC(C45CC(C(=O)OC)(C4)C5)=O)(C3)C2)=O)CCS(=O)(=O)CC1 57215,C1(C(=O)NC(CNC(C=C(C)CN2CCOCC2)=O)C2CCC2)CCCN1C(C)C 57216,C1(CNC(Cc2ccn(C)n2)=O)C2CN(C(C3(CO)CC(F)(F)C3)=O)CC12 57217,C(C)(CO)(C(=O)NC(c1ccc(CNC(=O)C2=COCC2)cc1)C)OC 57218,CC1=CCC=CC1N(CC(N1CCN(C)CC1)=O)C.N12CCC1(C)C2=O 57219,C1(CNC(c2ccc(Br)cc2)=O)CCCCN(C(C2OCC2F)=O)C1 57220,C1(CC)CN(C(=O)OC(C)(C)C)CCC1C(=O)O.c12cnc(c(F)c1)[nH]2 57221,N1(C(CSCC)=O)CC2CCCN(C(c3cc4c(C)nn(C)c4nc3C)=O)C2C1 57222,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(c2cncn2C(C)C)=O)C1)CC 57223,N1(C(C(CC)CCOC)=O)CC2CC3CC2C1C3NC(C1COCCC1(F)F)=O 57224,c1(CNC2C(C(N(CC)Cc3ccsc3)=O)C2)ccnc(F)c1Cl 57225,C1(NC(c2cc(CNC(CCc3ccn(C)c3)=O)on2)=O)C2CCCOC12 57226,C1(C(N2CC(C)C(NC(C3(O)CCOC3)=O)C2)=O)CCC(C)(F)CC1 57227,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(Cl)cn1C)=O 57228,Cc1cnsc1C(c1nnnn1C1CCOCC1)NCCC1CC1(F)F 57229,Cc1nc(C)c(C(C)NC(=O)C(C2CC2)N(C(=O)CCC(C)N(C)C)C)[nH]1 57230,c1(CN2CC(CNC(c3n(CC)ccc3)=O)OCC2)ccn2ccnc2c1 57231,CC1(C)CN(c2ccc(-n3cc(Br)cn3)nn2)CC2(CCOC2)O1 57232,c1(C(N2CCC(C)(NC(C3C(C)CCCC3)=O)C2)=O)cnc2n1CCS2 57233,c1(C(N(C2CCN(C(=O)CSC)C2)CCC)=O)ccc(C(OC)OC)nc1O 57234,c1(C(C(N2CC(c3cn(CC(CC)O)nn3)(N(C)C)C2)=O)O)ccc(F)cc1C 57235,C#CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cnn(C)c2F)=O)C1 57236,C(=O)(C(C=Cc1cccs1)NCCCCCn1cc(CO)nn1)OC 57237,N1(C(c2c(C)con2)=O)CCCC(N(C)C(c2ccn(CCC(F)(F)F)n2)=O)C1 57238,N1(C(COCC(c2ccccc2)=O)=O)CCCC(CNC(C2(O)CCOC2)=O)C1 57239,C(=O)(CCCCCNC(c1ccoc1)=O)N(C)CC1CCCCS1 57240,N1(C(C2CN2C)=O)CC2(CC(NC(=O)C(CCC)OC)CO2)C1.OC.OC 57241,c1(N2CCC(C(=O)OC)(COC)C2)ncc(S(C)(=O)=O)cc1Cl 57242,c1(C(=O)NC(CCNC(C(CC)CCOC)=O)C)cc(O)cc(F)c1F 57243,CC1=C(C(=O)NC2CC(Nc3ncc4ccnc-4[nH]3)C23CCC3)CCS1(=O)=O 57244,C1(N(C(C2C(CC)CCO2)=O)C)CCN(C(=O)CCCc2ncco2)CC1C 57245,c1(CC)ccc(Cl)c(-c2cnc(CC(CC)CC)cc2)c1 57246,c1(C(=O)NC(C2CCN(C(C(COC)(F)F)=O)C2)C)ccc2nnn(C)c2c1 57247,C(=O)(C(C)CC(=O)NCC(C(C)C)NC(C1CSCN1C(C)=O)=O)OC 57248,C1(C(=O)NC(CC)(C)CNC(C2CCC(=O)N2)=O)CC(c2ccccc2F)=NO1 57249,O=C1CCCC(C(=O)NCCCCC(=O)NC(CO)CCF)CC1 57250,N1(C(C=CC(C)C)=O)CCC(CO)C(NC(=O)C(C)S(N)(=O)=O)C1 57251,CC1(CNC(C2CC(=C3CC3)C2)=O)COCCN(C(=O)C2=NNC(=O)CC2)C1 57252,Cc1cncn1CC(N1CC(CC(C)NC(C2CCN(C3COC3)C2)=O)C1)=O 57253,C1(N(C(=O)COCC(C)(C)C)C)CCN(C(C2COC(=O)O2)=O)C1 57254,N1(C(C2(c3cccc(Cl)c3)CCC2)=O)CCN(C(=O)C2CC2)CC(O)C1 57255,C1(C(=O)OC)CCC2CCC1N2C(=O)CCOCCNC(c1noc2c1CCC2)=O 57256,C1(NC(c2nc(C(C)(C)C)oc2)=O)CC2CCCC(C1)N2C(=O)C(F)CC1CC1 57257,C1(C(=O)Nc2ccc(CCN)cc2)CC2(C1)CC(C#N)C2 57258,c1(OC)ccccc1CC(=O)Nc1cn(CCC2CCCN2)nc1C 57259,C1(NC(c2c(CC)cns2)=O)CCCN(C(C2CCCN2S(C)(=O)=O)=O)C1C 57260,N1(C(CN(S(N(C)C)(=O)=O)C)=O)CCC(C)(C)C(Nc2nccc(C(C)(C)C)n2)C1 57261,N1(C(C(C)N2CCCC2)=O)CCC(CC(=O)NCC2CC(=O)C2)CC1 57262,c1(C(C2(COC)COC2)NC2(NC(C)=O)CC2)nnnn1-c1ccon1 57263,C1(CC(=O)NCC(C=C)O)(CNC(c2cn(CCC)nn2)=O)CCCC1 57264,C1(NCCOc2c(C)cccc2)CCCN(C(C)C(N)=O)CC1 57265,C1(C(N2CC3CC(NC(CC4C(C)(C)C4)=O)CC3C2)=O)CNc2ccccc2O1 57266,Cc1cc(C(F)(F)C(N2CC3CC3C2CNC(=O)CC2CC2)=O)ccc1Br 57267,C(=O)(CC(C)CC(=O)N1CCCC(NC(=O)C(N2CCN(C)CC2)C)C1C)OC 57268,C(C)(CNC(c1cc(Cl)c[nH]1)=O)(CNC(=O)C(c1cccnc1)OC)OC 57269,N1(C(c2n(CC)nnc2)=O)CCC(C(=O)NCC(C)(O)CN(C)C)CC(C)(C)C1 57270,c1(C(=O)NC2(C(N)=O)CN(C(C3CCCS(=O)(=O)C3)=O)C2)ccn2ncnc2c1 57271,n1(CC(=O)NCC(C(C)(C)C)NC(CSC(C)C)=O)ncc(=O)c2ccccc12 57272,N1(C(C2N(C(c3cccc(C)n3)=O)CC=CC2)=O)CCc2ccc(C#N)cc21 57273,C1(CC)CCN(C(C2C3CN(C)CC23)=O)C1CNC(c1csc(=N)[nH]1)=O 57274,C1(NC(C2(C)CCCCO2)=O)CCC2(CCN(C(=O)C3=CCCSC3)C2)C1 57275,CCC(C)(C)CC(=O)N1CCC(CNC(=O)Cc2cc(C(C)C)nn2C)C(C)C1 57276,C1(NC(CCc2cn(C)nc2)=O)COCCN(C(=O)CCC2CC2(C)C)C1 57277,c1(C(=O)NC(C)(CNC(=O)C(F)F)CO)cc2c(Br)cncc2s1 57278,C(=O)(C(C)(C)SC(C)C)N1CC(CCNC(CCN(C(C)=O)C)=O)C1 57279,Cc1cc(CC(=O)NCCN(C(C)=O)CCn2cncn2)cc(F)c1 57280,C(CCN(C)C(C1CCC(C)(COC)O1)=O)(C(C)C)NC(c1c(CC)ncs1)=O 57281,C1(COC)(NC(=O)C(n2nccc2C)C)CCN(C(=O)CSS(C)(=O)=O)CC1 57282,C1(CCNC(c2ccco2)=O)(OC)CN(C(=O)CN(C)C(C2CCCCC2)=O)C1 57283,c1(NC2CCCN(C(c3ncncc3Cl)=O)C2)ccnc2ncnn12 57284,N1(C(CC2C(C)(C)CC2)=O)CC(CO)C2(C1)CN(C(=O)C=CBr)C2 57285,N1(C(c2sc(C)c(O)n2)=O)C2CCC1CC(F)(CNC(c1ccco1)=O)C2 57286,N1(Cc2ccc(C)c(C)c2)C2CCC1CC(NC(c1ccc(I)cc1)=O)C2 57287,C12(C(=O)NC3CCN(C(c4ccc(N(C)C)cc4)=O)CC3)CCCCC1C2(F)F 57288,CCCCC(C)CCC(=O)N1CCC(COC)(NC(c2ccn(C)c(=O)c2)=O)C1 57289,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57290,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57291,c1(OCCCC(=O)NC(CCNC(C(C)C2CC2)=O)(C)C)cc(F)cc(F)c1 57292,c1(CC(=O)OCC)ccc(NCC=Cc2ccsc2)cc1 57293,N1(NC(c2cc(C)no2)=O)CC2(CC(N(C)C)CO2)C1.C12CC1NC2=O 57294,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57295,N1(C(C(c2cn(C)nc2)=O)=O)CCN(C(C2CCCOCC2)=O)C(C2CC2)C1.CO 57296,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57297,C1(NC(c2c(-c3n(C)ccc(=O)c3)cncc2F)=O)Cc2ccc(C#N)cc2C1 57298,c1(CCC(=O)NCC(CO)C2CC2)ccnc(Br)c1 57299,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57300,C=CCC(C)(C)CC(=O)NC(CCN(C)C(C1(C(N)=O)CC1)=O)C(C)(C)C 57301,c1(C(=O)NC(CC)CNC(=O)C(CC2CC2)OC)cnncc1OCC 57302,N1(C(COCCCCC)=O)CC(COC)CC1(C)CNC(c1c[nH]nc1OC)=O 57303,N1(C(C(C(C)O)N(C)C)=O)CCC2(CC1)CC(NC(c1cncn1C)=O)CCO2 57304,c1(C(N2CCOCC2C(C)C)C(=O)NCCCSC)c(C)nn(C)c1C 57305,c1(OC(F)(F)F)cccc(CN2CCN(Cc3cc(C4CC4)no3)CC2)c1 57306,C(=O)(C(F)(F)C(F)F)NCC(N1CCN(C(C(C)=CC2CC2)=O)CC1)C(F)F 57307,c1(C(N(CC(CC)NC(c2cnsc2)=O)C)=O)cc(C)c(C#N)cn1 57308,c12cncc(c1)C2=O.C1(NC)(NC(=O)CC(C=C(C)Cl)=O)CC(OC)C1.C1CC1 57309,C(C1CCCc2ccccc21)NC(CC1N(CC2C(C)CCC2)CCC1)=O 57310,Cc1cnc(F)c(C(=O)NC2CC(F)CN(C(=O)CC(=O)OCCC(C)C)C2)c1 57311,C(=O)(CCCC(C)(F)F)N1C(CNC(C2CCC(SCC)CC2)=O)C(C)CC1 57312,C1(C)(CNC(C2CC(c3ccc(CC(=O)OC(C)(C)C)o3)C2)=O)CC2CC2C1 57313,CC(C)C(C)C(C)CC(=O)N1CCOC(CNC(=O)C(C(C)C)NC=O)C1 57314,N1(C(c2cn(CCNC(C3CCC(=O)C3)=O)nc2)=O)CCCCC1CC(O)CO 57315,c1(C(=O)NC(C)CN(C)C(C2CCC(N(C)C)CC2)=O)ccc(F)cc1F 57316,C#CCCC(O)C(=O)N(C1CCN(C(C2(CC)CC2)=O)C1)C 57317,C=CCC(F)(F)C(=O)NCC1CCN(C(C)=O)C1.C12CCC(C)(C1)NC2=O 57318,c1(N2CCC(CNC(C(C)SC)=O)C23CC3)nc(C)nc2scnc12 57319,C1(C(N(C2CCN(C(=O)C(CO)NC(N)=O)CC2)CC)=O)CC(=O)N(C(C)C)C1 57320,n1(C(C)C(=O)NC(C)CC(C)NC(C2CC(=O)N2)=O)cnc2ccccc12 57321,C(N=c1[nH]c2c(c(=NCc3c(C(N)=O)ccc(Cl)c3Cl)[nH]1)CCCC2)C1N(C)CC1 57322,C1(NC(C=C2CCC(C)C2)=O)C2CC3CN(C(c4ccc(N)cc4)=O)C1C3C2 57323,C1(C(C)NC(=O)CSC2CC2)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 57324,C(=O)(C(CCN(C)C)NC(=O)C(C)C#N)NC1C(C)CC1 57325,N1(C(C(CC)CC)=O)CC2OCCN(C(C3(C)CCCOC3)=O)C2C1 57326,c1(CC)c(C(=O)NCCCNC2CC(C)(C)CN2C(=O)C(C)OC)cccc1C 57327,C(COC)(C(=O)NC(C#N)CCNC(=O)Cc1ccco1)NC(=O)OC(C)(C)C 57328,CS(=O)CCC(O)C(=O)NCCCNC(=O)Cc1cccc(CC(F)(F)F)c1 57329,Cc1ccc(C2CCCC(NC(C3C4CN(C(SC(F)(F)F)=O)CC34)=O)C2)cc1 57330,N1(C(c2ncc(CC)s2)C(=O)NCCC2CC2)CCCOCC1C 57331,Cc1cc(NS(C)(=O)=O)nc(=NCCOc2csnn2)[nH]1 57332,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57333,CC(C)(CNC(N1CCOC(CCO)C1)=O)C(N)=O 57334,N1(C(CC2CCC(CNC(C(C)Cn3cccn3)=O)CC2)=O)CC2CC(C)C2C1 57335,Cn1nccc1CC(=O)NCCC1CC(NC(=O)CO)C1 57336,N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)CCC=C1CCSCC1)C2 57337,C1(C(CNC2(C(=O)OCC)CC2)C)CCN(C(=O)C(F)(F)C2CCC2)CC1 57338,C1(c2nnnn2C2COC2)(Sc2c(C)cccc2Br)CCOC2(CCOCC2)C1 57339,S(=O)(=O)(c1ccc(NCc2ccc(Cl)o2)cc1Cl)NC1CC(C)N(C)CC1 57340,N1(C(C2CCCOC2)=O)CCCC(C2CCCN(CC=C3CCCCC3)C2)C1 57341,C1(CN(C(=O)CCN(CCO)CCO)C)CN(C(=O)C=Cc2cccnc2)CCO1 57342,N1(C(CC(COC)NC(CC(C=C)(C)C)=O)=O)CCC(O)C(C)(O)C1 57343,CC1CN(C(c2cscc2C(F)F)=O)CCN1C(=O)CCSc1nnnn1C 57344,CC(C)C(C(=O)N(CC(O)CN(C)C(C1CCN(C)C1)=O)C)NC(N)=O 57345,c1(N2CCCC(C)(C)CC2)nc(N2CCCOCC2)c2ncsc2n1 57346,C1(CNC(CCC(=C)Cl)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57347,C1(C2(O)CN(C(c3ccc(CO)cn3)=O)C2)(CNC(=O)CC23CC(C2)C3)CC1 57348,N1(C(C2ON=C(C(C)C)C2)=O)CC2CCC(NC(=O)C(C)C)CC2C1 57349,C12(C(=O)OC3CCC(c4n(C)ccn4)CC3)CCC(=O)N1CC1(CC1)C2 57350,c1(OC)ccc(Br)cc1C.n1(C(N(C)C(C)C2CC2)=O)cc(C(C)(C)O)nn1 57351,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57352,C1(c2ccc(OC)o2)CS(=O)(=O)CCN1C(=O)C(c1ccc(I)cc1)C 57353,N1(CC(=O)N(CCCCN(C(C(C)Cn2ccnc2)=O)C)C)CCCCCC1=O 57354,c1(CC)cc(C(N2CCC(O)(C(C)NC(=O)CNS(=O)(=O)N(C)C)C2)=O)c(C)o1 57355,Cc1c(Cl)c(C(N2CC3CC3(NC(=O)CC3CC(F)C3)C2)=O)nn1C 57356,N1(CCC(=O)NC2(CC(C)NC(=O)CCCF)CC2)CCOC1=O 57357,C123CC(CCO1)(C2)NC(=O)C(=O)N3.c1(NC(=O)OC(C)(C)C)cnccc1OC 57358,c1(C(=O)NCC2(F)CN(c3cc(CO)ncn3)C2)cccc2nccn12 57359,S(=O)(=O)(c1ccc(-c2cccc(CF)c2)cc1)NC1CCC(=O)NC1 57360,O=C(CC1NC(=O)c2ccccc21)NCC1CCN(C(c2coc(O)n2)=O)C1 57361,c1(NC)cncc(C(=O)NC2CCC(CCC(=O)NCCc3ccoc3)C2)c1 57362,CCCC(C)CC(=O)NCC12C(NC(=O)CC3CCOC3=O)C3CC1C2C3 57363,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57364,N1(C(C(C(CC)C)O)=O)CCC2CN(C(=O)CNS(=O)(=O)NC)CCC2C1 57365,c1(CNCc2ccc(-n3c(C)cc(C)n3)cc2)nc2ccccc2[nH]1 57366,C1(C(N(C(C)C)Cc2cscc2Br)=O)CCc2ccccc2C1 57367,c1(CCCOCC)nc(CCCCl)n(-c2ccc(OC3CCOC3)cc2)n1 57368,CCCC(CCC)=CC(=O)NCCN(CCOC)C(C1CC(=C)C1)=O 57369,C1(CNCC(O)CNC(=O)C(F)(F)F)CCCCC1OC.CC1C(=O)OCCO1 57370,C1(C(=O)NC2CCCC(NC(c3c(C)cccc3C)=O)C2)CCC12CCOCC2 57371,N1(C(Cn2cc(OCC(=O)Nc3cccnc3)nn2)=O)CCc2ccncc2C1 57372,N1(C(c2csc3nccn23)=O)CCC2(CCCN2C(c2cc(O)cs2)=O)C1 57373,C1(NC(C(C)C#N)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)CC(O)C1 57374,c1(CCC(c2n(CCCOC)nnn2)NC2CC2(C)C)ccccc1Br 57375,c1(C(=O)NC2C(C(=O)OC)C2)ccnc(C)c1.c12cn(nn1)C1CN(C1)C2=O 57376,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57377,CN1CC2CC2(SCc2c(C(=O)Nc3ccc(F)cc3F)cccc2)S1(=O)=O 57378,C(=O)(C(C)(F)C(C)(C)F)N1CCN(CCNC(C(C)=CC)=O)CC1 57379,C(CCCCCCC(=O)NCC(C)(C)C1CCCO1)NC(C)=O 57380,Cc1ccnc(C(F)(F)C(=O)NCC2CCCN(C(C3CCCN(C)C3)=O)C2)c1 57381,N1(C(C=CC)=O)CCC(OCCNC(=O)CCCc2nccs2)C1 57382,N1(C(CNC(C2(c3ccno3)CC2)=O)=O)CC2(CCC2)CC1CNC(C1(F)CC1)=O 57383,CCCC(C)CCCC(=O)NC1(CCOC)CCN(C(C2(CC(C)C)CC2)=O)C1 57384,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(=O)Cc1ccnc(C)c1 57385,N1(C(C2(Cl)CCCC2)=O)CCCC1CCc1cn(CC23CC(CO2)C3)nn1 57386,C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)NC1CCN(C(CC=CC)=O)C12CCC2 57387,CC1CN(C(C2CN(C(C3CN(CC(F)(F)F)C3)=O)CC2C)=O)CC(C)O1 57388,c1(C(=O)NC2C(C)CN(C(=O)C3=CCC3)CC2)cnn2c1CC(C)CC2 57389,C12(C(N3CC(NC(=O)COc4nc(O)nc(O)n4)C3)=O)CCCCC1OCC2 57390,c1(C(=O)NC2C(CNC(C(C(C)(C)C)SC)=O)COC2)cc([N+](=O)[O-])ccc1C 57391,c1(C(N(C2CN(C(=O)Cc3ccoc3)CC2O)C)=O)cnc2ccccc2c1 57392,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1CC(F)F 57393,N#Cc1cc(-c2cc(C(=O)Nc3ccc4c(c3)CCO4)ccn2)ccc1O 57394,C1(NC(CCSCC)=O)COC2CN(C(C3CC3c3cccnc3OC)=O)CC12 57395,Cc1ccc2c(=NCC(=O)N=c3cc[nH]cc3)[nH]c(N3CCN(C)CC3)nc2c1 57396,n1(CCC)cc(C(=O)NC(C2CCN(C(c3cc(C)cn3C)=O)C2)(C)C)c(C)n1 57397,C(=O)(CC1=CCOCC1)NCC1(C)CCN(C(C(C)n2ccnc2)=O)CC1 57398,N1(C(C2C(C)CC2C(=O)OC2CC2)=O)CCC(C2CCN(C(=O)CN(C)C)C2)CC1 57399,C1(NC(c2ccc(F)cc2)=O)CC2CN(C(c3ccc(F)c(Br)c3)=O)CC12 57400,C1(NC)CCN(C(=O)C(C)(C)O)CC1.N12CC3C(C3C1)C2=O 57401,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccc(C)n1)N1CC(C#C)C(OC)C1 57402,Cc1cccc2cc(C(=O)NCC3CN(C(C4NC(=O)OC4C)=O)CC3O)oc12 57403,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57404,c1(C2N(CC(=O)NC3CC(C)(NC(CC4(C)CC4)=O)C3)CC2)ccccc1 57405,CC1(C)CC(C)(CNC(C2(CF)CCC2)=O)CN1C(=O)CCCC1CCCCC1 57406,c1(C(=O)NCC(C(=O)NCc2cc(CC)on2)N(C)C)cncc(C)n1 57407,CCC(C)C(C(=O)N1CCC=CC1C(=O)NCCOCC(C)(C)O)OC 57408,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCC(NC(C3CN4CCN3CC4)=O)C2C1 57409,CC(CS(C)=O)C(=O)N1CCN(C(=O)CN(C)C(c2ccc(Cl)cn2)=O)CC1 57410,C1(CN(C(C(C)CN(C)C)=O)C)CCCN(C(C2CCC(=O)N2)=O)C1 57411,CC1CCc2ncc(-c3nc(CCCO)nn3-c3cccc4ccccc34)n2C1 57412,CC(C)(CNC(c1ccc(-c2cnco2)cn1)=O)CC(F)F 57413,C(=O)(C1=CCCCO1)N1CCC(CN(C(C(C)Sc2ccc(Cl)cc2)=O)C)C1 57414,C1(NC(C2(CCN(C)C)CC2)=O)CCC(NC(=O)CN2CCOCC2)C1 57415,C1(C=O)CCOCCN1N1C(COC)CCC1.C(=O)CCc1cncs1 57416,N1(C(CC2(C)CCCCC2)=O)CC(NC(=O)C(N)=O)C(C2CC2)C1 57417,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57418,c1(C(=O)OCC)cc(C(=O)NC(CNC(c2c(Cl)cnn2C)=O)CO)c(C)s1 57419,C(=O)(CCCC(=O)NCc1csc(C(N2CCC(CCO)C2)=O)c1)OCC 57420,CC(C)CC(C(=O)N1CCC(OCC(=O)N(C)C)C1)Nc1nccnc1Cl 57421,C(C(C)(C)C(C)C)N1C(=O)CO1.C1C(=O)N(CC(C)C)C(CC)N1CC 57422,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(C(c2ccc(F)c(F)c2)C)CC1F 57423,c1(CC(=O)NC2(CNC(c3c(Cl)cn(C)n3)=O)CCCCC2)ccccc1C#N 57424,C1(OC)CCCC1C(=O)NC(C)CCNC(c1cn(C)cn1)=O 57425,C(C(CO)CC(C)C)NC(C1(C(C)NC(C(C)=C2CC2)=O)CCC1)=O 57426,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1CC 57427,c1(OC)ncnc(C(N2CCCC2CCNC(C2CC2Cl)=O)=O)c1F 57428,C1(NC(CCn2c(C)ncc2)=O)CCCC(CN(C)C(c2nn(C)cc2Cl)=O)C1 57429,C(=O)(C1CCCc2cc(C#N)ccc21)NCCCNC(C(CCOC(C)(C)C)F)=O 57430,C=CC(C)CN=C(NCC1(SC)CC1)NC1CCOc2ccccc21 57431,Cc1nc(N2CCCC23CCN(c2ccncn2)C3)c2cc(Br)ccc2n1 57432,N1(C(=O)Nc2n(COC)ncc2)CC2CN(C(=O)COC(F)(F)F)C2C1 57433,C(CCC(O)CO)N(C)C(C1(CNC(=O)CC(F)(F)F)CCCCO1)=O 57434,C1(NC(C(C)OCC(C)C)=O)CN(C(c2cn(C3CCCCC3)nn2)=O)CC1C 57435,c1(SCC(=O)NC2CN(C(C34CC(C)(C3)C4)=O)CC23CC3)ccccc1[N+](=O)[O-] 57436,c1(OC)cc(F)c(F)cc1CN1CCC(C(=O)Nc2cccc(C#N)n2)C(O)C1 57437,C1(OC)CN(C)C(C)(C(=O)NCCCNC(c2ccoc2C2CC2)=O)C1 57438,C#CCC(CCOC)NC(C1COCCC1NC(=O)CC(C)OC)=O 57439,CC1OCCN(C(=O)CC(Cl)Cl)C1C(=O)NCC=Cc1ccccc1 57440,C1(C(=O)NCCN(CCCCCC)C(c2conc2C2CC2)=O)CCS(=O)(=O)C1 57441,c1(SCC(=O)NCCC(C)NC(c2sncc2Br)=O)ccccn1 57442,N1(C(C(c2cn(CC)nc2)(F)F)=O)CCCOC(CNC(c2sccc2Cl)=O)C1 57443,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57444,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57445,c1(NC(=O)Cc2csc(C(F)F)n2)cncnc1SCCCC1CCCC1O 57446,C1(C2CCCC2)(C(N2CC3(CC(NC(C4CCOC4C4CC4)=O)C3)C2)=O)CCC1 57447,CC1(C)CC1(c1cn(C2C=CCCC2)nn1)NC(=O)CCNC(C1CCCC1)=O 57448,c1(N2C3CN(C(C4(SCC)CCCCO4)=O)C(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57449,c1(NC(C)=O)ccc(C=CC(N2CCOCC2CNC(=O)CC(C)CF)=O)cc1 57450,N1(C(c2c(CC)occ2)=O)CCC(C)C(NC(c2cc3c([nH]2)CCCC3)=O)C1C 57451,c1(C(N2CC(NC(C=Cc3nc(C)c(C)[nH]3)=O)(CO)C2)=O)nccc2occc12 57452,N#Cc1cncc(OCCNC(C2CCCCC2c2nc(S)n[nH]2)=O)c1 57453,Cc1cc(C)c(NC(C2CC3CC3N2Cc2cnc(C3CC3)s2)=O)cn1 57454,C1(C(N(C)CC2COCCN2C(C2CC=CCC2)=O)=O)CC2(CCOCC2)CO1 57455,C12(C(N(CCCn3cc(C(COC)C)nn3)C)=O)CC3CC(C1)CC(C)(C3)C2 57456,c1(CCC)ccc(N)c(C(=O)NC2CC3CC(NC(C4CC(O)C4)=O)C2C3)c1 57457,N1(CC(C)(C)O)CCCC(C(=O)OC2CCCCC2)C1 57458,N1(C(c2c(C)nc(CC3CC3)s2)=O)CC(C)CCC1CNC(=O)COC(C)C 57459,N1(C(C(C)O)=O)CCC(CNC(=O)CNC(=O)Cc2ccsc2)C12CCC2 57460,C#CCC(O)C(=O)N(CCCCNC(c1cnn(-c2cccc(F)c2)c1C)=O)C 57461,S(=O)(=O)(c1ccc2c(c1)NC(=O)CCS2)NCC1(C)CC1Br 57462,N1(C(c2c(C)nns2)=O)CC2C(CC(=O)NCc3ccc(CN(C)C)o3)C2C1 57463,C1(=O)C(C(C)(C)C)CO1.N1(C(C)=O)CCCCC1CNC(c1cnc(S)[nH]1)=O 57464,c1(C(N2CCS(=O)(=O)CC2)C(=O)NC2CC2)noc2c(Cl)cccc12 57465,N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CC1(C(N1CC(CC(F)F)C1)=O)C2 57466,c1(C(=O)NC(CC)CNC(C2(C)CCCCCCC2)=O)ccc(S(N)(=O)=O)c(C)c1 57467,CC1ON=C(C(=O)N2CCCCC(NC(C3CCC3)=O)C2)C1C 57468,c1(C(N2CCCC(NC(C(C=C=C)C)=O)C2)=O)cccc2c1CC(C)(C)C2 57469,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57470,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(N)ccc3O)=O)CC12 57471,C(=O)(C(C)C(C)C)NCC(c1ccccc1F)NC(C1(C(C)(C)OC)CC1)=O 57472,C(=O)(C1CC=Cc2ccccc21)NC1(C)CCN(C(=O)CC2CCC3CC23)CC1 57473,C(C)(C)(CN=c1nc(C(F)(F)F)[nH]s1)NC(c1nn(C)c(C2CC2)c1)=O 57474,N1(C(c2c(CC)onc2C(F)(F)F)=O)CCC(NC(=O)C=NOC)C(F)C1 57475,C(=O)(C(F)=CC1CC1)NCCCCN(CCCNC(C1CCO1)=O)C.CCO 57476,c1(C(N2C(CN(C(C=C(CCC)C)=O)C)CCC2)=O)cnc(C)cn1 57477,c12ccc(cc1)NC2c1n(CC(=C)C)nnn1.C(C(C)C=C)OC(F)F 57478,c1(C(=O)NC(CNC(CC(C)OC)=O)C(C)C)cc2cc(Cl)sc2[nH]1 57479,C(CCC(C)(C)C(=O)NC1CC(C)OC(C)C1)NC(c1cc(COC)no1)=O 57480,c1(CNC(c2ccc(N3CC4CCC3C4)cc2)=O)ccc(C(F)(F)F)c(I)c1 57481,C1(C(N(CCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C)C)=O)CN2CCC1CC2 57482,C(=O)(C(COCC)CC(C)C)NCCN(C(C(CC)NC(N)=O)=O)CCCN(C)C 57483,CC1CC(NC(c2cc3n(n2)CCC3)=O)CCN1C(C1CN(C)CC(C)O1)=O 57484,c1(OCC)ccccc1OCCNCC1COCC1(C)C 57485,N1(C(C(C)OCCCn2cc(Br)cn2)=O)CCCC1CNC(N)=O 57486,C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cc(C3CC3)no2)=O)CC1(C)C 57487,C12(NC(c3ccc(=O)n(CCF)n3)=O)CCCC1N(c1ncc(Br)cn1)CCC2 57488,c1(NC(=O)Nc2cccc(Oc3cc(C)cc(F)c3)c2)cc(Br)cc(C)c1C 57489,CC(C)CCCOCC(N1CCC(C(C)NC(C2CCNC2=O)=O)C1)=O 57490,c1(C(C(=O)NC(CC)(C)C)N(CC(F)F)CCN(C)C)ccc(-c2cnn(C)c2)o1 57491,N1(C(C2(CC)CCCCC2)=O)CCCCC(CNC(c2nccc(Cl)c2C)=O)C1 57492,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57493,C(CN=C(NCC1CCC(F)(F)CC1)NC(C)COC)C1(c2c(C)cccc2)CC1 57494,CC1(C)CC(C(F)F)=NON1C(=O)C1CN(CCCO)C1 57495,C1(CNC(c2onc(CC)n2)=O)CCCC(NC(c2ncccn2)=O)C1 57496,CCC(CC)C(C)C(=O)NCc1ccc(C(=O)NCc2nn(C)c(=O)o2)o1 57497,C1(CN(C)C(c2n[nH]cc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC2(CCC2)O1 57498,c12cc(no1)C(=O)N2.C1(OC(C)=O)CN(C(=O)C(C2CCCC2)SC2CC2)C1 57499,N#CC1(C(=O)NC2(CCCNC(C3CC(F)(CO)C3)=O)CC2)CCC1 57500,c1(NC(C(c2cc(C(C)C#N)[nH]n2)N(CCCF)C)=O)ccc2c(c1)CCC2 57501,C1(NC(C(CO)OC)=O)CN(C(c2ocnc2C2CC2)=O)C2CCCC12 57502,c1(C(N(CC(C)NC(C(C(=C)C)(C)C)=O)C)=O)ccc2c(c1)NCCC2 57503,CCCCC(CC)CCC(=O)NCCN(C(=O)CC(C)c1ccco1)CCC 57504,N1(C(C2C(C(C)C)OCC2)=O)CC2CC3CC2C1C3.C1(=O)C(O)C2CN1C2 57505,C(=O)(CC(C)C(=O)NCC(C)CC(=O)N(C)Cc1cncn1C)OC 57506,C(C(C)C(=O)NCC(C)CNC(=O)CCC1CCCCC1)OC(C)=O 57507,c1(OC)c[nH]c(C(=O)NC2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)cc1=O 57508,Cc1[nH]c(=NC(C)c2ncc(Br)cn2)sc1C#N 57509,c1(C(C(C)C)NC(=O)N(C)C(C2CCC2)C)ccccc1F 57510,CC(CO)(C(F)F)NC(=O)CC1(NC(=O)C(N)=O)CC1 57511,C1(C(=O)NC(C(C)NC(=O)CCC2(C)CC2)CO)OCCN(C)C1=O 57512,c1(C(N2CCC(O)(C(C)CNC(C3(F)CC3)=O)C2)=O)ccnc2c1ncn2C 57513,C1(C(=O)NC(=O)COCC=CC(=O)N(CCOCC(C)(C)C)C)(CC)COC1 57514,N1(C(C)=O)CCN(C(=O)C(C)(C)CN(C(=O)COc2cnn(C)c2C)C)CC1 57515,Cc1ccc2[nH]c(=NCC3CC4(CC(NC(=O)CC5CCC6CC56)C4)C3)sc2n1 57516,C(CC(O)CO)N(C(=O)CN1CC(O)(NC(=O)CCOC2CCCC2)C1)C 57517,CCC(N=c1cccc(S(=O)(=O)NC(C)(C)C2CC2)[nH]1)c1cc(C)ccc1F 57518,C(=O)(C(C(C)C)C1CCCC1)N1C(C=C)CC1 57519,CC12CC1CCN2c1cc(SC(F)(F)F)ncn1 57520,N1(C(C(C=C)(F)F)=O)CCC2(CNC(c3c(F)cc(F)cc3F)=O)CCCCC12 57521,n1(CCCC(=O)NCC2(COC)CN(C(C3(C4CC4)CC3)=O)C2)nc(C)cc1C 57522,CCC(C)(CNC(=O)C(OC)OC)C(=O)NCC(=O)NC(N)=O 57523,C(c1ccc(O)cc1)=CC(=O)NCCC1CCC(NC(C(C2CCC2)OC)=O)C1 57524,c1(C(=O)NCCCCN(C(C=Cc2ncc(C)[nH]2)=O)C)cnc2ccccc2c1 57525,c1(N2CCC(N3C(NC(C)=O)CCC3)C2)ccc(C)c(C)c1 57526,C#CC1(C(=O)NCCn2nc(C)cc2C)CCN(C(c2sccc2C#N)=O)C1 57527,N1(C(CC(C)n2cccn2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57528,c1(CC(=O)NC23CCCC(NC(=O)Cn4nccn4)(C2)C3)csc2ccccc12 57529,C1(CCNC(=O)C=Cc2ccccc2)CN(C(=O)CSCc2cn[nH]c2)CCO1 57530,N1(C(C(c2cn(CC)nc2)=O)=O)CCCCC(NC(c2ccc(N)c(F)c2)=O)C1 57531,N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)CCc2nc[nH]n2)CC(C)C1 57532,CC(C(C)(C)O)N(C)C(=O)Nc1nc(Cn2cc(Br)cn2)cs1 57533,C1(OCC(C)C)CCN(C(=O)COC(=O)NC2CCCCC2)C1 57534,C(=O)(C(C)(C)CC(F)(F)F)N1C(CN(C)C(c2cc(O)cc(F)c2)=O)CCC1 57535,c1(CNC(=O)CC2CC2)ccnc(-n2cc(C3OCCO3)nn2)c1 57536,N1(CC)CCCCC1C(=O)NC1CC(CC(=O)NCC2CC(=O)N(CC)C2)C1 57537,c1(C(N(C)CC2CCCN(C(C(C)SC(C)C)=O)C2)=O)cc(F)c(F)cc1O 57538,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cc(Cl)no2)=O)CC1c1ccncc1 57539,N1(C(CCCc2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)Cc2cnsc2)CC1 57540,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57541,CC1CN(CCNC(=O)NC(c2ccc(Nc3ccccc3)cc2)C)CCO1 57542,C(=O)(CN=c1cc[nH]cc1)NC1CN(C(c2c(C)n(C)nc2C(F)(F)F)=O)CC1C 57543,C1(CCNC(CCC=C)=O)CCCN(C(c2cn(CC3CCCO3)nn2)=O)C1 57544,c1(OC)cc2nc[nH]c2cc1C(=O)NCC1CCN(C(=O)CC2CC3(CC3)C2)C1 57545,c1(CCCCC)cccc(C#N)c1.N1(C(C)=O)CCC(C2OCCO2)CC1 57546,c1(C(=O)NC2(C)CCCN(c3cc(C)ncn3)C2)cc(Cl)nc(Cl)c1F 57547,CC1(C(=O)NC2CCCC(NC(c3cccc(C(F)(F)F)c3)=O)C2)CCCCO1 57548,Cc1nc(N2CCC3CCCC23CNC(=O)Cc2cn(C)nc2C)ncc1[N+](=O)[O-] 57549,Cc1nc(=O)n(C2CCN(C(=O)CCNC(c3ccc(F)cc3)=O)CC2)[nH]1 57550,C1(C(=O)NCC(=O)N(C2CCN(Cc3cnn(C)c3)CC2)C)C2CC3C(C2=O)C13 57551,C1(CC)(CNC(C(c2ccccc2C)C)=O)CCN(C(c2sc(F)cc2C)=O)C1 57552,C1(C(=O)NCCC(C)(C)NC(c2cc(C3CCOCC3)no2)=O)C(C#N)C1(C)C 57553,C=C=CCCC(=O)NC(Cn1cccn1)C(N1CCCCC1CN(C)C)=O 57554,c1(COC)ccc(C(=O)NC(C(=O)NC2CCC2C(=O)OC2CC2)c2ccoc2)s1 57555,n1(CNC(C2CC(CNC(C3(CC)CC3)=O)C2)=O)ccc(C(F)(F)F)n1 57556,c1(CC)cc(C(=O)NCCCN(C(=O)C(C)NC=O)CC)c(C)nn1 57557,C(=O)(CCCCC(F)F)NC(C)CN(C)C(c1ccc(Cl)cc1Cl)=O 57558,c1(N(CCCC)C)ncc(C)cc1S(=O)(=O)N1CCC(C2CCCO2)CC1 57559,c1(C(N(CCCC(C)C)C)=O)coc2c1CN(C(c1cc3n(n1)CCO3)=O)C2 57560,c1(C(=O)NC2CCC(CCNC(c3c(C)ncs3)=O)C2)cc(F)cnc1O 57561,N1(C(C2(NC(c3nccc(C)c3N)=O)CCCC2)=O)CCCC2CCCCC12 57562,Cc1cc(C(=O)NCC2CC2CNC(c2ccsc2)=O)c(C)s1 57563,C1(CNC(C2CCC(=O)O2)=O)CC(C(=O)N2CCCCC2)=NO1 57564,c1(CC(N2C(C(=O)N)C(C)C2)=O)cccnc1O.C12CC1CC2C.CC 57565,n1(CC)nnnc1C(C(C)C1CCC1)NC1CCC(C(=O)NC2CC2)C1 57566,c1(CC)onc(C(=O)NC2CCOCC2C(N2CCCC2CC2CCC2)=O)c1C 57567,CCC(C)(C(=O)Nc1ccccc1CN(C(=O)C(C(=O)OC)OC)C)C(N)=O 57568,c1(C(N(C(C)CNC(C23CCCC2(C(N)=O)C3)=O)C)=O)cccc(Br)c1F 57569,Cc1nc(-c2ncc[nH]2)sc1C(=O)NCCNC(=O)Cc1ccccc1Br 57570,C(=O)(CC1=CCCC1)NC1CCN(C(C)C(=O)N(CC2CCCO2)CC2CC2)C1 57571,N1(C(C2(CC=C)CCN(C(=O)C(CC)C(C)C)CC2)=O)C(CC)C2CC(O)C1C2 57572,N1(C(=O)OC(C)(C)C)CCCC(NC(C2CCC(=O)N(C3CC3)C2)=O)CC1 57573,Cc1cnsc1C(=O)NC1CC(NC(c2cn(-c3ncccn3)cn2)=O)C1 57574,N1(C(C)C)CC2CCC1C1CN(C(=O)CCC(=O)N(C)CC3CCC4CC34)CC21 57575,CP(C)(=O)CCC(=O)N1CCCCC1C1(NC(c2[nH]ncc2C#N)=O)CC1 57576,C1(C(N2CCCC(C)(CC)C2)=O)CC(C)(C)CN1C(=O)C(O)C1CCC1 57577,C(=O)(C1CC(=O)c2ccccc21)NCC1CN(C(c2ccc(C)[nH]2)=O)C(C)CC1 57578,c1(C(=O)NCCCCNC(c2ccc(OC)cc2O)=O)cc([N+](=O)[O-])cc(C)n1 57579,Cc1[nH]nc2ncc(C(N3CCN(C(=O)C(CO)NC(N)=O)C(C)C3)=O)cc12 57580,c1(NCC2C(CF)C2)nc(N2CCn3nncc3C2)c2c(n1)CCC2 57581,N1(C(CC=C=C)=O)CC(C)CN(C(C2CC(C(F)(F)F)C2)=O)C(C)C1 57582,c1(C(=O)NC(C)CCCCNC(c2cccc(CO)n2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 57583,C1(SC)CCC(CCC(=O)N(CCO)CCO)C1.C1CC(=O)N1OC(F)F 57584,c1(C(N2CCC(NC(CSC(C)C)=O)C(F)C2)=O)ccc(Cl)c2ccccc12 57585,CC1C(N(C(=O)CCC2CCC(NC(c3cc(C#N)cs3)=O)C2)C)CCCC1C 57586,c1(N2CCC(CC(N3CC(S(C)=O)C3)=O)CC2)cc2ccccc2s1 57587,Cc1ccc(C(=O)NCCCCC2CN(C(=O)CCC(F)F)C2)c(C)n1 57588,c1(C(=O)NCCN(C(C=C(CCC)C)=O)CC)cnc(CO)nc1C 57589,N1(C(C(CCC)NC(=O)Cn2nc(C)cc2C)=O)CCC2(CCOC2=O)C1 57590,c1(OCCOc2c3c(ccc2)C(NCC(=O)ON)CC3)ccc2c(c1)S(=O)(=O)NC2 57591,c1(CNC(=O)CC2CCCN2Cc2c(C)[nH]nc2O)cnc(C(=O)O)nc1C 57592,N(C1CCc2c(C(F)(F)F)cccc21)CC(C(C)(C)F)(C)F 57593,N1(C(C(CC)CCOC)=O)CC2CCC1CN2C(=O)CN1CCCCC1C 57594,C=CC1(CC(N2CCC(CC)(CO)C2)=O)CN(C(c2ccncc2OC)=O)C1 57595,C(CS(C)=O)(C(C)(C)C)NC(c1n(CCSC)nnn1)(C)CCC1CC1(Cl)Cl 57596,C1(C2CCN(C(c3cc(C(=O)C4CC4)no3)=O)C2)(NC(c2c(CC)cc[nH]2)=O)CC1 57597,C1(CNC(C(=O)N(c2ccc(OC)c(OC)c2)C2CC2)=O)CCCC2(CCC2)C1O 57598,c1(C(N2CCOCC(CNC(C3CC3F)=O)C2)=O)cc2c(nc1O)CCCC2 57599,C(=O)(C(CC)N(C)N1Cc2ccc(OCc3ccccc3)cc2C1)NCCC(C)CO 57600,C1(CC(=O)NCC=CC(=O)NCC2(OC)CCOC2)CCCCC1O 57601,C1(NC(C2(NC(C)C)CC2)=O)CCC(CNC(C2(F)CCOC2)=O)CC1 57602,Clc1cccc2c1CCC(NCc1csc(C(F)F)n1)C2 57603,N1(C(C(CNC(c2n[nH]c(C)c2Cl)=O)C)=O)CCC2(CCCC2)CC1 57604,c1(C(=O)NCC2(F)CC(NC(=O)CC3CC34CC4)C2)nn2cccnc2c1Cl 57605,c1(C(N(CCCN(C(C(C)CC(N)=O)=O)C)C)=O)ccc(Cl)c(O)c1N 57606,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(C(C)(C)C)c2ccccc2)CC1C 57607,c1(NCC(=O)N(C(c2cn(CCCC(=O)O)nn2)C)C)cc(F)c(F)c(F)c1 57608,c1(C(=O)Nc2c(OC)cc(SC)cn2)cnn2ncccc12 57609,C12(NC(CCCC(C)C)=O)CCCC1N(C(c1ncccc1S(C)(=O)=O)=O)CC2 57610,c1(NC(CN(CC#C)C(c2c(SC)cn(C)n2)=O)=O)cccc2c1OCO2 57611,C(C(CNC(c1cn(CCC)nc1C)=O)C(F)(F)F)NC(C(C=C)(C)C)=O 57612,c1(OCCC(=O)COC(C2(CN(C)C)CC2)=O)ccccc1F.C12CCCC1C2 57613,N1(C(C2C(C=C(C)C)C2(C)C)=O)CCCC(C2(NC(c3csnn3)=O)CC2)C1 57614,c1(C(N(C(C)CNC(=O)C=CCN2CCC2)CC)=O)cccc2nc[nH]c12 57615,N1(C(C(C)CNC(N)=O)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(F)F)C3 57616,C#CCC(O)C(=O)N1CCCC(OCc2cn(-c3nc(C)c(Cl)s3)nn2)C1 57617,N1(C(C(C)(C)NC(=O)C(CO)NC(N)=O)=O)C2CSCC1C2 57618,n1(CC)c(O)nc2cc(NC(=O)C(=O)NS(=O)(=O)CCCN(C)C)ccc12 57619,C1(NC(CC2C(C)OCC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 57620,N1(C(c2ccc(C(C)F)cc2)=O)CC=C(CNC(C2CC23CCCCC3)=O)CC1 57621,c1(OC)ncc(F)cc1C(=O)N(C1CCCCN(C(C2CC(C)=NO2)=O)C1)C 57622,C(C)(C(C(=O)NCC=CC(C)(C)C)NC(c1cc(CO)n(C)n1)=O)OC 57623,c1(C(N(CCC(N2CCOC(CCF)C2)=O)C)=O)cncc(CO)c1 57624,C1(C(=O)NCC(C)NC(C2CC(O)C2)=O)CCCC1O 57625,C1(C(C(=O)NCCC2CC2)N(C)CC2(CC(C)C)CC2)CC(C)CC(C)C1 57626,N1CC2(C1)CN(n1c(-c3cncc(Cl)c3)nc(CC(=O)OC(C)(C)C)n1)C2.C1CC1 57627,C(C(CC(F)(F)F)NC(C1CCC(C)(C)O1)=O)NC(COC1(C)CCOCC1)=O 57628,c1(OCCC)ccc(C(=O)NCC2CC(NC(C3(n4nccn4)CC3)=O)C2)cc1N 57629,CC1(CNC(C2CCCC(F)(F)C2)=O)CCN(C(c2sccc2Cl)=O)CC1 57630,c1(C(=O)NCCN(C(c2n(CC)ncc2)=O)CC2CC2)cnnc(Cl)c1 57631,N1(C(C2CC(C)CN2Cc2ccc(Cl)c(F)c2)=O)CCN(C)C(C)(C)C1 57632,CC1(C)C(NC(c2cscn2)=O)CC1CNC(c1nncs1)=O 57633,Cc1cnccc1C(CC(=O)N(C1CCCC1)C)NC(c1cccnc1)C1CCC1 57634,N1(C(C(CCC)N(C)C)=O)CC2CCC1CN2C(=O)C(O)CC(C)C 57635,N1(C(c2c(Cl)cc(C)s2)=O)CC2(CCC(CNC(C3(C)CC(C)(C)C3)=O)O2)C1 57636,c1(CC)nn[nH]c1C(=O)NCC(C)(C)CNC(c1ncn(CC)n1)=O 57637,c1(C(N2C(C(=O)O)CC3CCCCC32)=O)cc2cc(Cl)ccc2cn1 57638,CCCCCCCC(F)C(=O)OC(c1ccc(C(F)(F)C(F)(F)F)cc1)=O 57639,N1(CCOC)CC(C(=O)NCCOCCNC(=O)C(n2ccnc2C)C)CC1=O 57640,C1(NC(c2c(C)n[nH]c2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 57641,n1(CC(=O)N(CC(=O)NCCCCNC(=O)CCC)C)cnc2ccccc12 57642,N1(C(COCC=C)=O)CC(NC(C2(SC)CC2)=O)C2(CCC2)C1 57643,c1(CC)cncc(C(N2CC=CC(C(=O)NCC3CCC=CO3)C2)=O)c1 57644,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2ccccc2)C(C)C)n1 57645,C(=O)(C(O)C(F)(F)F)N(CCC(=O)NC(C#C)CCC)C(C)C 57646,CC1(C)COCCC1CNC(C12CC(NC(c3sccc3CO)=O)(C1)C2)=O 57647,c1(C(N(C)CC)=O)csc2c1CCN(Cc1ccc(N(C)C)cc1C)C2 57648,c12cccc(c1)NC(CC)CNC2=O.C1(C(=O)NC)CCN(C(=O)C2CC2)CC1 57649,C1(NC(Cc2ccc(OC)cc2)=O)(CO)CCN(C(C2CCCC(C)C2)=O)CC1 57650,N1(CC2CC3CC2C2CC32)CCc2nnc(NCc3ccccc3)cc2C1 57651,C#CCCCCC(=O)N(C)CC1CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)C)C1 57652,N1(C(C(CCC)CC2CCCC2)=O)CCC(C2(NC(c3ccc(C)s3)=O)CC2)C1 57653,c1(C(C)CC(=O)NC(C2CCN(C(C3(F)CC=CC3)=O)C2)C)ccc(F)c(F)c1 57654,C(=O)(C(CNC(N)=O)C(C)C)N(C(CN(C(CCCN(C(C)=O)C)=O)C)C)C 57655,c1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)ccc2snnc2c1 57656,CC1CCCCC1(CNC(c1c[nH]nc1[N+](=O)[O-])=O)NC(c1cc([N+](=O)[O-])c[nH]1)=O 57657,n1(CC(=O)NCC(C)N(C(C(CC)(C)C(N)=O)=O)C)ncc2ccccc2c1=O 57658,CC1CC(CC(N2CC(CCNC(=O)CCOC3CCC3)C2)=O)CCS1 57659,C1(F)(CCNC(=O)C=CBr)CN(C(c2csc(CCOCCOC)n2)=O)C1 57660,C1(n2cc(C(N3CCCC3)(C)C)nn2)CCCN(C(C2CC23CCCC3)=O)C1 57661,c1(C(=O)NCCCNC(CCCC(CC)C)=O)ccc2c(c1)OCCN2 57662,c1(OCCOC)cccnc1C(=O)NC1CC(C)N(C(=O)C=C(C)C(F)F)C1 57663,N#Cc1cc(C(=O)Nc2nnn(SCC3CC3)c2-c2ccccc2)on1 57664,c1(C(=O)OC)ccc(F)c(COC(=O)CCC(=O)c2cccc(Cl)c2)n1 57665,C(CN=c1[nH]cncc1I)(N(C(c1ccc(C#C)cc1)=O)C)C1CC1 57666,N1(CC(C)(C)C)CCC(C(=O)NCC(C2CCCC2)N)CC1 57667,CCCS(=O)(=O)c1ccc(C(=O)NCC(C)NC(c2csc(C3CC3)n2)=O)cc1 57668,O=C(C1COc2ccccc21)NC1C2CC1CN(C(=O)Cc1cnoc1)C2 57669,N1(C(C(C=C)(C)CC)=O)CCC2CCC(C1)N2C(c1cnc(O)c(F)c1)=O 57670,C=C1CC(C(N2CCCCC2c2ccccc2F)=O)N(C(c2ccncc2)=O)C1 57671,COn1cnc(C)c1C(N1CC(CNC(=O)Cc2ncc(Cl)s2)C(C)C1)=O 57672,C=CC1(CC(=O)NCc2[nH]nnc2CC)CN(C(C2(COC)CC2)=O)C1 57673,C1(C2CN(C(c3ccc(C)s3)=O)C2)(NC(C(C2CCCCC2)NC(C)=O)=O)CC1 57674,C(=O)(C1=CCC(C)(C)CC1)NCC(CC)(C)NC(C1CC1(COC)COC)=O 57675,c1(C(C23C(CCN(C(=O)Nc4nc(Cl)cs4)C2)C3)=O)cc2ccccc2[nH]1 57676,c1(NCC2CC(OCCOC)(OC)C2)c(Cl)nc(C)nc1C 57677,c1(C(=O)NCC2(O)CCN(C(C3CCCCO3)=O)C2)cc(Br)cnc1S 57678,C1(NC(CC2(OC)CCC2)=O)CC2CC(NC(=O)CCSC)C1C2 57679,C(=O)(C(C(C)(C)C)OC)NC1N(C(c2c(CC)nn(C)c2)=O)CCC1C(C)C 57680,C1(C#CC(=O)NC(CCF)C(N2CCCC(O)C2C)=O)(CC)COC1 57681,C1(NC(c2nc(CC)[nH]n2)=O)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 57682,n1(CC(=O)NCC2N(C(c3ccnc(C)c3C)=O)CC=C2)nc([N+](=O)[O-])cc1C 57683,C1(C(N2CC(C)(CCO)C2)=O)(NC(=O)COCCF)CCOCC1 57684,C1(NC(c2nnnn2CCc2cccc(F)c2)(C)C2CC2)CC(=O)N(C(C)(C)C)C1 57685,c1(C(N2CC(SC)C(NC(=O)CC3CC3CC(C)C)C2)=O)c(F)ccc(C)c1F 57686,c1(OC(C)C)cccc(C(=O)NC2COCCC2NC(=O)CC2(CO)CC2)c1F 57687,c1(C(=O)OC)cc(N2CCN(C(=O)C=Cc3ccccc3)CC2)ccc1F 57688,c1(CCCC)nc(C(=O)NCC2CC(CCNC(=O)C(C)COC)C2)cs1 57689,N1(C(C(C)N(C)CC)=O)CCC(CNC(=O)CCn2nc(C)nc2C)(COC)C1 57690,Cc1c(C(=O)N(O)Cc2nc(-c3cccs3)no2)cccc1F 57691,C1(CNC(C2CC(C)OC2)=O)CCCCN(C(c2ccnc(Cl)c2F)=O)C1 57692,C12(CNC(C3CCC(C)O3)=O)CCC(CC1)N2C(=O)C(c1ccc(F)cc1)(C)C 57693,N1(C(c2ccc(-c3c(C)nn(CC(C)C)c3C)cc2)=O)CC2CCCOC2C1 57694,c1(C(=O)NC2C(C)CN(C(c3cnc[nH]3)=O)C2)cnc2c(c1)OCCN2 57695,Cc1ncc(CN(C(=O)CC2CC(NC(=O)CC3CC4(CCC4)C3)C2(C)C)C)n1C 57696,N1(C(c2c(OC)cncc2)=O)CCN(C(c2cc(CC3CC3)on2)=O)C(CO)C1 57697,c1(-n2c(C3CCC4CC34)nc(-c3ccc(C(F)F)cc3)n2)cccc2ccccc12 57698,C1(NC(c2c(C)nsc2)=O)CC2CC1N(C(=O)CCc1ccnn1C)C2 57699,c1(C(N2CC(NC(c3cccc(O)n3)=O)C2)=O)ccc2nc[nH]c2c1F 57700,N1(C(COCC(=O)NC)=O)CCC2(CCC(CNC(C3(Br)CC3)=O)O2)CC1 57701,c1(N(C(CC)CO)C)ccc(S(=O)(=O)N2CCC(C)(N(C)C)CC2)cc1Br 57702,C1(OC)Cc2ccccc2C1N1CCN(CC(=O)Oc2ccc([N+](=O)[O-])cn2)C1 57703,Cc1ccccc1CC(=O)NCCCNC(C1CCC1(OC(C)C)OC)=O 57704,C1(NC(C)=O)CCN(C(c2cccc(OCC(F)F)c2)=O)CC1F 57705,Cc1cc(C#N)nc(NCC23CCCC2NCC3)n1 57706,Cn1ncc2ncc(C(N3CCC4(CC4NC(=O)Cn4cnnc4)C3)=O)cc12 57707,CCS(=O)(=O)CCn1nc(-c2ccc(OC(C)(C)C)cc2)nc1CCOC 57708,C(C(C)C(F)C(=O)N(C)CCc1cccs1)NC(C(C)=C(C)C)=O 57709,Cc1onc(CO)c1C(=O)NCC1C(CNC(C2CCOC(C)C2)=O)C1(F)F 57710,C1(C(=O)NC2C(C(=O)NC)CCC2)CCN(C(C2(C)C(C)(C)C2(C)C)=O)CC1O 57711,C1(CCCC)CN(C(C2CC23CCSCC3)=O)CCN1C(=O)C(C#N)C(C)C 57712,C1(C(=O)NCc2cn(CCO)nn2)CC2CC1N(C(=O)C(N1CCOCC1)=O)C2 57713,c1(NC(C2(C)N(C(c3n(C)ncc3)=O)CCC2)=O)ccc(F)cc1I 57714,C(=O)(CC(C)C(F)(F)F)NC(C(=O)NC(CC=C)CC=C)COC 57715,CN1CCCCC1C(=O)NC(C(=O)NCC(C)(C)F)C1CC1 57716,N1(C(CC(CC)OC)=O)CCCC(C)(NC(c2oc(C)cc2C)=O)C1 57717,C#CCCC(O)C(=O)NCC1(CCNC(=O)C(C)Cc2ccccc2Cl)CC1 57718,S(=O)(=O)(c1c(C)nn(C)c1C)NC1C(O)CCN(Cc2c(C)cccn2)C1 57719,C1(CCNC(CCSCCCC)=O)CCN(C(C2(OC)CCOC2)=O)CC1(F)F 57720,N1(C(C)=O)CC2(C1)CN(C(c1cnc(C)n1C)=O)C2.C1(C)C(=O)N1.C(C)C 57721,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 57722,C1(CNC(c2cc(C)c(F)cn2)=O)CN(C(=O)COCC2CCCC2)CCC1C 57723,c1(CN2CCCC(C(N(CCCC)CCOC)=O)CC2)nc2ccccc2n1C 57724,c1(C(=O)NCC(C)N(C(=O)C(C)(C)C#N)C)nn(C)c(Cl)c1Cl 57725,c1(CSc2c(N3CCN(CC)CC3)cccc2)ccc([N+](=O)[O-])o1.C1CN1 57726,C1(C)(NC(C(N2CCC(C)C2)=O)=O)CCCC1NC(c1ccc(N(C)C)cc1)=O 57727,Cc1c(C(N2CCC(c3ccccc3F)C2C(C)C)=O)sc2ccc(F)cc12 57728,Cc1cc(C(=O)NC(CNC(=O)Cc2cnoc2)C(C)C)cnc1O 57729,CCCC(CNC(c1ccc(OC)o1)=O)C(=O)NC1CC12CCC2 57730,c1(OC)nsc(OC)c1C(=O)N(C1CCC(NC(c2ncccc2N)=O)C1)C 57731,C1(CC)CN(C(=O)CNC(c2ccc(Cl)cc2)=O)CCN1C(=O)C#CC(C)(C)C 57732,c1(C(=O)NCC2CCN(C(C(CC)F)=O)CC2C)cc2c(C)nn(C)c2nc1C 57733,C1(C(=O)NCC2N(C(c3nc(C)[nH]n3)=O)CC(O)C2)CCC([N+](=O)[O-])CC1 57734,N1(C(C(N2C(CC)CCC2)=O)=O)CCC(N(C)C(c2ncc(F)cn2)=O)CC1 57735,C(c1ccc(Cl)cc1)=CC(=O)NC(C)CCNC(=O)CCNC(N)=O 57736,C1(NC(CCc2cc(OC)c(F)cc2)=O)CCC(O)CN(C(C2CCC2)=O)C1 57737,c1(CCN(N2CCCC2)C)ccc(F)cc1F.c1(C)ccccc1 57738,CCC(C)CC(C(=O)N1CCC(N2CCCC2)C1)NC(c1n[nH]cc1C)=O 57739,C1(NC(c2ccoc2)=O)CN(C(c2cccc(OCC(F)F)c2)=O)CC1O 57740,C12(C(=O)NCCC3CN(C(c4cnc(CC)[nH]4)=O)C3)CCCN1CC(O)C2 57741,N1(C(CN(C2CCC2)C)=O)CC2CN(C(c3ccnc(Cl)c3O)=O)CCC12 57742,C1(NC(CN(C(C(C)C)=O)C)=O)CCN(C(C2CC3CCC2O3)=O)CC(C)(C)C1 57743,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 57744,Cn1c(C(=O)NC2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)nnc1S 57745,c1(CCC(=O)NCC(CC=C)NC(=O)CC(C)OC)cc(C)cc(C)c1 57746,N1(C(C=C)=O)CC2(C1)C(NC(c1cc3sc(C)cc3s1)=O)CCS2(=O)=O 57747,c1(CCC(=O)NCC2CN(C(=O)CN3CCCCC3)CC2O)ccc(F)c(F)c1 57748,C(=O)(CC(N=c1[nH]c(=N)[nH]c(=NCC2CC(F)C2)[nH]1)c1cccc(Cl)n1)NC 57749,C1(C(N(CC(CNC(Cc2c(C)nn(C)c2C)=O)C)C)=O)CC2(C)CCC1(C)O2 57750,C(=O)(C(CC)(CC)CC)NC1C(CC)CN(C(=O)Cn2ncn(C)c2=O)CC1 57751,c1(NC(C2N(Cc3cccc(C#C)c3)C3C(C2)C3)=O)ccc(S(=O)(=O)C2CC2)nc1 57752,C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(c2cc(Cl)c[nH]2)=O)CC1 57753,Cc1cc(C(=O)NCC2(CNC(=O)C(F)CC3CCOC3)CCC2)nc(C)c1 57754,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(c3scnc3C)=O)C12 57755,c1(OC)ccnc(C(=O)N(C(C)(C(=O)NCC(O)CN(C)C)NC(N)=O)C)c1 57756,C12(CNC(Cc3cnn(C)n3)=O)CC3CC(CC(NC(=O)C=CBr)(C3)C1)C2 57757,CC(CNC(=O)CN1CCCC1=O)C(F)C(=O)N(C)CC1(CO)CC1 57758,c1(NC)cccc(C(=O)NCCC(C)(C)NC(=O)CCNC(C)=O)n1 57759,N1(C(CN2C(=O)CCCC2)=O)CC2OCCN(C(C3CC4(CCC4)CO3)=O)C2C1 57760,c1(C(N2CC(NC(c3ccc(SC)cc3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 57761,C=C1CCN(C(c2cn(C)cc2C)=O)C(C(=O)NC(C)CSC)C1 57762,C1(CCNC(=O)CC2CCCCC2(F)F)CC(N=c2[nH]ncs2)CCN1 57763,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)NS(CCCC(=O)OC)(=O)=O 57764,c1(OCC)cc(F)ccc1N(C(c1nnnn1CC(F)F)c1cncs1)CC 57765,c1(OC)ccc2c(NC(=O)NCC(C)(C3CCCC3)NC3CC3)c[nH]c2c1 57766,CC#CCCCC(=O)N1CCC1C(N1CC(OC)C1(C)C)=O 57767,Cc1cc(C)c(C(=O)N(C2CCC(CNC(=O)C=Cc3cn(C)nn3)CC2)C)o1 57768,CN1CC(c2nn[nH]n2)(NCC(C2=NOCC2)SC)CCC1=O.C(CO)O 57769,c1(C(=O)NC(C(C)NC(CCC2CC(OC)C2)=O)CO)cccnc1C(F)(F)F 57770,C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCN(C(=O)CC2(O)CCC2)C1 57771,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 57772,c1(C(=O)NC(C)C(c2ccccc2)NC(=O)COCCF)ccc(N)cc1O 57773,c1(N(CCCN(C(=O)C2=CCSC2)C)C)ncnc2c1nnn2C1CCCC1 57774,c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC(F)C3)C2)cc2c(s1)CCOC2 57775,N1(C(CCc2nc(C)sc2)=O)CCCOC(CCNC(C2CCCN(C)C2)=O)C1 57776,O=S(=O)(c1ccc(=NCc2cc(F)ccc2F)[nH]c1)NCC12CCCC1OCC2 57777,c1(CC)noc(C)c1C(=O)NCc1csc(C(=O)NC2CCC2(C)C)c1 57778,N1(C(C(F)OC)=O)CC2(C1)CN(C(c1cc(CO)ccn1)=O)CC2CO 57779,C(=O)(C1=CCCS1)NCCCOCCN(C(=O)CCc1cccc(OC(F)F)n1)C 57780,c1(OC)sccc1C(=O)NCc1c[nH]nc1C(=O)NC1(C(C)(F)F)CC1 57781,c1(NCC2C(C)(C)CN(CC3CCC=CCCC3)C2)ccc(C#N)c(C(F)(F)F)n1 57782,CC12CCC(C(=O)NCC3CC3NC(=O)CCCN3CCCC3)(CC1)CO2 57783,c1(C(=O)OCc2cc(F)ccc2Br)cc(F)c2c(c1)CCC2 57784,c1(C(N2CCC(NC(C(CC)n3cncn3)=O)C2CC)=O)ccn2nccc2c1 57785,C12CC3COCC3N1C2.c1(OC)ccnc(C2(NC(=O)OC(C)(C)C)CC2)c1 57786,c1(CC)[nH]c(C(N2CCC2CNC(c2cccc(CSC)c2)=O)=O)nc1Cl 57787,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 57788,C1(C(=O)NC2(c3ccccc3)CC(C)C2)CC(=O)N(Cc2ccccc2)C1 57789,C(c1ccc(F)c2ccccc12)=CC(N1CC(NC(CC2C(C)C2)=O)C1)=O 57790,c1(C(=O)OC)c(C)ccc(NC(=O)NCC2CC2CO)c1C 57791,Cc1ccc(C(C)NC(C2CN(C(=O)C(C)CSC(F)(F)F)C2)=O)cc1F 57792,C(=O)(C1CCCc2nccn21)N1CC(F)(CNC(c2ncc(OC)cn2)=O)C1 57793,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 57794,c1(CC(=O)NC2C(CNC(C(CC)NC(C)=O)=O)C2)cc(OC)cc(OC)c1 57795,CC1CC(C(=O)NCCCN(C2(CC(C)(C)C)CC2)C)C(=O)O1 57796,CCCC(C(=O)N1CC(NC(=O)Cn2ccnc2C(C)C)C(C)C1)OC 57797,C1(N(C2CC23CCOS(=N)(=O)CC3)C)CC2CCC(C1)N2C(=O)OC(C)(C)C 57798,C(=O)(CS(C)(=O)=O)NCC(C)N(C(=O)CCC(=O)C1CC1)C 57799,c1(NC(C2CCN(Cc3cnsn3)CC2F)=O)cc(C(F)(F)F)cc(Br)c1 57800,C1(CNC(c2ccncc2F)c2n(CCC)nnn2)OCCOC1(C)C 57801,N1(C(CCC#CC)=O)CCCC12CCN(C(=O)CCOC(C)(C)C)CC2 57802,N#Cc1cc(Cl)c(C(=O)NCCCNC(c2c[nH]nc2F)=O)s1 57803,c1(C(=O)NCC(C)NC(c2n(CC)c(O)nc2)=O)noc2ncccc12 57804,c1(-n2nc(C)c(CC(C)NS(=O)(=O)CC#N)c2C)cccc2ccccc12 57805,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 57806,N1(C(C2C(C)(C)C2)=O)CCC(C2CCC2)(CNC(=O)CC23CCCC2C3)CC1 57807,N1(C(C2CCN(C(=O)C3(F)C(C)C3)O2)=O)CCCCC(C(=O)N(C)C)C1 57808,C(=O)(CCCCCCCC(=O)N1CCC(N(C(=O)C(F)CC2CC2)C)CC1)OC 57809,c1(CN(C2CN(C(C(C)=C3CC3)=O)C2)C)cccc(F)c1 57810,c1(C(N2CC3C(C(N(CCCC)CCO)=O)(C3)C2)=O)c(OC)ccc(Cl)c1F 57811,CC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)Cc1n[nH]c(=N)s1 57812,c1(OC(C)C)ccc(F)c(C(N2CCC(O)C2C(=O)NC2CC(O)C2)=O)c1 57813,N1(c2cccc(C)c2)N=C(C(=O)N(C)CCNC(c2ccn(C)c2)=O)CCC1=O 57814,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 57815,C1(NC(CCC)CN(C)C)CCCCN1CCc1csc(C(=O)O)n1 57816,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(N(C(c2coc(C3CC3)n2)=O)CC)CC1 57817,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 57818,C12(CNC(c3c(SC)cccn3)=O)CCC(CC1)N2C(=O)C(c1ccccc1)O 57819,CN1CCOCC1C(=O)NCC(C(N1CCOCC1CC1CC1)=O)C1CCC1 57820,C1(NC(C2(C)CS(=O)(=O)C2)=O)CC2CCC(C1)N2C(C1COC2(CCC2)C1)=O 57821,N(C(=NCC1CC(F)(F)C1O)NC(C)C)Cc1ccc(C)o1 57822,C1(C(N)=O)CCCN1C(C1COC(CNC2CC2)C1)=O.C12(CCC1)C(=O)NC2 57823,C1(C(=O)NCC2CC(NC(c3c(C)cc(C4CC4)o3)=O)C2)COCCC1(F)F 57824,C(=O)(CC1=CCOCC1)NCCC(C(C)C)NC(=O)C(N1CCCCC1=O)C 57825,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CC(CC(N)=O)C1 57826,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 57827,C12(NC(COCCC#C)=O)CCCC1N(C(c1[nH]nnc1C)=O)CCC2 57828,c1(NC(N2CCC(C)C2C)=O)ccc2c(ccn2C)c1.C(C)(C)(C)OC(=O)O 57829,c1(NC(=O)NC2CCN(c3ccc(F)cc3F)C2)ncc2c(I)cnc-2[nH]1 57830,C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2C(=O)CSc1cc(F)ccc1F 57831,c1(C(=O)NC(CC)CN(C(=O)C(=O)NC)C)cccc(C(C)(C)C)n1 57832,c1(C(=O)NC(CNC(CCCCSC)=O)C)ccc2c(c1)N(C)C(=O)CO2 57833,C1(C2(O)CN(C(C3CN(C)C(=O)N3)=O)C2)(CNC(c2ccc(C)cn2)=O)CC1 57834,C=CC(C)C(C)C(=O)N1CC(C(C)NC(c2c(C)ccnc2Cl)=O)C1 57835,N1(C(CCNS(C)(=O)=O)=O)CCN(Cc2ccsc2)C(C2CC2)C1 57836,c1(N2CCC(C(C)C(=O)NC3CCN(C)CC3)CC2)ccn2ncc(C#N)c2n1 57837,C1(CN2C(=O)CN(C(=O)OC)C2=O)C2CCC3(CNCC13)O2.c12ccccc1C2 57838,c1(OC(C)C)cccc(C(=O)NCC=CCNC(C2CC23CCOC3)=O)n1 57839,CC1CCCCN1C(C1(NC(c2cnn(C)n2)=O)CC1C)=O 57840,C1(CN(C(=O)COc2cccc(Br)c2)C)CCCN(C(=O)C=CC(F)(F)F)C1 57841,C1(CNC(C2C(C)(C)C2CO)=O)CCN(C(=O)Cn2nnc(C3CC3)n2)CC1 57842,N1(C(C2(OCC)CCOC2)=O)C2CCC1CC(CNC(=O)C(C)(C)C)C2 57843,C12(C(=O)NC3CCC(CCNC(C(CCCC)C)=O)C3)CC3CC(CC(C3)C1)C2 57844,CC1(C)C(NC(=O)CCC(=O)c2ccc(Cl)cc2)CCN1C(=O)C1=CCOCC1 57845,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1CCC(=O)O1)=O 57846,CCC(CNC(C1CCNC1=O)=O)(CC)C(=O)N(C1CC(C)C1)C 57847,C(=O)(C(CO)C(C)(C)C)N(C(CNC(C(C)=CC=C)=O)C(=O)NC)CC 57848,c1(C(=O)NC2CCN(C(CCCSC)=O)C(C)C2)ccc2c(c1)CC(=O)NC2 57849,C1(NC(CCSCCC)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC(O)C1 57850,C1(CC)CC(CC(=O)N(C(C(=O)NC2(C)CSC2)C2CC2)C2CC2)C1 57851,n1(CCC(N)=O)cc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)nn1 57852,C1(F)(C(N2CC3(CCN3C(=O)C(F)(F)c3ccccc3)C2)=O)CCCC=C1F 57853,CC(C)CCC(C(=O)NCc1cnn(C2CC2)c1)NC(=O)C(C)NC(N)=O 57854,C(=O)(C(C)(C)S(C)(=O)=O)NCCC(C)N(C)C(c1coc(N(C)C)n1)=O 57855,CS(=O)C1CN(C(=O)CN(C(=O)CCc2ccccn2)CCOC)C1 57856,c1(SCC(=O)N(C)CC2CCN(C(c3c(C)c[nH]n3)=O)CC2)cccc(Cl)c1Cl 57857,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CC(=O)NC(C)SC1CC1 57858,CC12CCOC(C(=O)NC3CCN(C(c4scnc4C4CC4)=O)CC3O)(C1)C2 57859,CCC(CC(=O)NC1CC(NC(=O)C=Cc2ccc(F)cc2F)C1)CC(F)(F)F 57860,N1(CC)CCC(C(=O)NCC(CNC(=O)Cc2nonc2C)OC)CC1 57861,c1(NC(CSCC(=O)OCC(C)(C)O)=O)cccn2cncc12 57862,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCCn3cccn3)CCC2C)C1 57863,C(=O)(CCCCC(C)(C)C)N1CC2CCC(NC(c3cc(C)c(F)cc3)=O)C2C1 57864,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 57865,N1(C(Cc2nc(C)sc2)=O)CCC(C)(C)C1C(N1CCC(O)C(C)C1)=O 57866,CC(CS(C)(=O)=O)C(=O)OC(=O)NC1CC1.C12CN(C1)C2=O 57867,c1(CC(=O)NC2CN(C(C3C(C)C3)=O)CC23CCC3)cnc2n1CCCC2C 57868,N1(C(CCC2CCC(C)O2)=O)CCC(NC(=O)OC(C)(C)C)C(C2CC2)C1 57869,Cc1cccc2c(C(=O)NCC3CCCN(C(C4CC(C)CO4)=O)CC3)cnn12 57870,C=C=CC(C)C(=O)N1CC2C(CNC(=O)CCc3ccccc3Cl)C2C1 57871,C1(O)(CNC(CCCC#CC)=O)CCCN(C(=O)CCC(=O)N2CCOCC2)CC1 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57906,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 57907,c1(N2CCC(CCO)C2)nnc(CCC#N)[nH]1.c1ccc(-c2n[nH]cc2CN)cc1 57908,C1(Cn2c(-c3ccc(-n4cncn4)cc3)nc(C(CC)C)n2)CCS(=O)(=O)CC1 57909,N1(C(CNC(C=CC(C)NC(COCCSC)=O)=O)=O)CCOC(C)C1 57910,N1(C(CC(C)c2ccco2)=O)CC(NC(c2cc3ccsc3s2)=O)CCC1C 57911,Cc1nc(CN=C(NCCC(C)O)N(C)C)cn(C)c1=O 57912,c1(C(C(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)O)ccccc1Cl 57913,Cc1[nH]nc2cc(C(=O)NCC3COC(C)(C)CN3C(=O)COC3CC3)ccc12 57914,N1(C(C2OCC(=O)C2)=O)CCCOC(CNc2nccc(CO)n2)C1 57915,C1(NC(CC2(C)OCCO2)=O)C2CN(C(C3CCCN(C(N)=O)C3)=O)CC12 57916,CC(C)C(O)C(C)C(=O)N(CCCN(C)C)CCNC(=O)CC(C)CN(C)C 57917,C=CCC(CNC(c1ccc(O)nc1)=O)C(=O)N(CC(C1CC1)OC)C 57918,c1(CC(N2CCC(CCNC(Cn3ccc(C)n3)=O)C2)=O)ccc(C#N)cc1 57919,c1(C(=O)NCC(CC)(C)NC(c2c[nH]nc2OC)=O)cc(C)cc(Cl)c1 57920,C1(NC(C2(C#N)C(C)(C)C2)=O)CCC12CCN(C(C13CC(OC(C)=O)(C1)C3)=O)CC2 57921,CC1=NS(=O)(=O)NC(C)=C1CC(=O)N1CCC(N(C)C(C2CC2C)=O)C1 57922,C1(C2C(C)C2)CCCN(NC(CCC2N(C(C3(C4(C)CC4)CC3)=O)CCC2)=O)C1 57923,c1(C(=O)NC(CNC(C(CC)O)=O)C2CCC2)cc(C)cc([N+](=O)[O-])c1 57924,c1(CNC(C2C(=C)C2C(=O)OC)=O)cc[nH]c1NC(C1CC(CC(C)(C)C)C1)=O 57925,N1(C(CN(C(C)C)C)=O)CCC(NC(=O)C(=O)NC(C)C)C1 57926,CCCCCS(=O)(=O)CC(=O)NCC1CN(C)CCN1C(=O)CC1CCC(=O)C1 57927,c1(-c2cn(C(C)C(N3CCC(c4ccncc4Cl)C3)=O)nn2)ccc(CO)cc1 57928,C1(CC)CN(C(=O)CCCN(C)C)CCC1C(=O)NC(C)C(CO)SC 57929,N1(c2n(CCC=C)c(C3CCCN(C)C3)nn2)CC(CO)OC2(CCC2)C1 57930,c1(CCC(=O)NC(C2CN(C(C3CCCCO3)=O)C2)C)cccnc1Cl 57931,C1(NC(c2nc(CCC)oc2)=O)CCCCN(CC2CCCC2)C1 57932,c1(C(=O)NC(C(C)NC(=O)CCNC(=O)NC2CCOCC2)CO)cccnc1O 57933,Cc1ccc(O)c(C(=O)NCC2(CNC(C3(C)CC4(CCC4)C3)=O)CCCC2)c1 57934,C12(C(=O)NCCCCSC)CC(C)(CN1C(=O)C(C1CCCCC1)O)C2 57935,N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cnn3c2OCC3)=O)CC1 57936,C1(C(N2C(C)CC(NC(C3C(OC)CCC3)=O)C2)=O)Cc2cccnc2C1 57937,C(=O)(CC(O)C(C)C)NCCN(C(C(CC)(C)OC)=O)Cc1ccccc1 57938,N1(C(C2N3CC(C)N(CC3)C2)=O)CCC(C2CN(C(C3(C)CC3F)=O)C2)CC1 57939,c1(CCC(N2CCC(CNC(=O)Cc3cnccc3Cl)C2)=O)ccc(O)c(O)c1 57940,CC1CCC(NC(c2ccccc2Cl)=O)CN1C(=O)CS(C)(=O)=O 57941,C(=O)(C(F)C(C)(C)O)NC(C1(O)CN(C(C2ON=C(CC)C2)=O)C1)C 57942,[N-]=[N+]=Nc1ccccc1NC(=O)C(O)CNC(C1CC2CCC1O2)=O 57943,c1(C(C)C)ncoc1C(N1CC(C(C)NC(=O)C(C)N(C2CCCCC2)C)C1)=O 57944,Cc1cccc(Cl)c1CCC(=O)N(C1CC1)Cc1nc(Br)n(C)n1 57945,Cn1nc(O)cc1NC(=O)CC1CCN1C(c1nccn1-c1ccccc1)=O 57946,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 57947,c1(C(N2CC3C(NC(CCNS(C)(=O)=O)=O)(C3)C2)=O)cc(=O)n2nccc2[nH]1 57948,N1(C(C(C)O)=O)CCN(C(CC2CCOC2)C(=O)NC(C2CCCCC2)C)CC1 57949,c1(C(=O)NCC2C(NC(c3c(CC)con3)=O)CCC2)ccc(F)c(Br)c1 57950,C1(NC(c2ccc(OC)s2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 57951,C1(CC(=O)NC2C(C)N(C(=O)C=Cc3cnc[nH]3)CCC2)CC2(CCC2)CCO1 57952,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(CCC(C)OC)=O)CC1 57953,c1(C(N2CCCN(C(C(CC(C)C)OC)=O)C(C)C2)=O)cccc2cnccc12 57954,CC1CCN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)C(c1ccccc1F)F 57955,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCc1nc(C)co1)C2 57956,CC1(C)CC(CNC(C2CC(CF)C2)=O)CN(C(c2nn[nH]c2Cl)=O)C1 57957,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 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57976,c1(OC)nc(C(=O)OCC(=O)N(CCCC2CCCCC2)C)sc1C 57977,C12(NC(CN(C)C)=O)CCCC1N(C(C1Nc3ccccc3C1(C)C)=O)CCC2 57978,CCC(CC(C)C)C(=O)NCC1CCN(C(C2CCSCC2)=O)C(C)C1 57979,c1(OC)ccc(C(F)(F)F)c(C(=O)NCC2CC(CNC(=O)CC(C)F)C2)c1 57980,C1(C(=O)OC)CC12CN(C(C13CC1CCN3C(c1cc(C)sc1C)=O)=O)C2 57981,C12(C(=O)N(CC3N(C(C4(C#C)CC4)=O)CCCC3)CC)CCCCN1CCC2 57982,C1(CC(C)C)C(=O)O1.Cc1ccc(-c2noc(CCO)n2)cc1 57983,c1(CCCC)ocnc1C(=O)NCCCCCNC(=O)C(CC1CCCC1)OC 57984,Cn1ccc(=NC(=O)CCOCCNC(C23CCCCC(F)(C2)C3)=O)[nH]1 57985,C1(C(N2CC(CC)(CO)C2)=O)CN(C(=O)C=Cc2ccc[nH]2)CC(C)(C)C1 57986,C1(CC(=O)OCC)CCCCC1C(=O)NC1CN(C(C2CC=CCC2)=O)C1 57987,n1(C(COC)C)nc(-c2ccccc2)nc1CC(C)CC(C)C 57988,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(c2ccnn2C(C)(C)C)=O)CC1 57989,c1(C(N2CCCC(C(=O)Nc3ncc(F)cc3O)CC2)=O)cc(Cl)cc(Cl)c1Cl 57990,c1(C(C)C)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 57991,C1(C(=O)N(C(CCC(C)(CO)N)=O)CCC)CCC(F)(F)C1.N1(CC(C)=CC)CCOCC1.OC 57992,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccnc12 57993,C1(C(=O)NC2(CNC(C(F)=C(C)C)=O)CCCC2)CCn2cnnc2C1 57994,N1(C(c2c(F)ccc(NC(c3n(C)ccc(=O)c3)=O)c2)=O)CCC2(CNC(=O)N2)C1 57995,N1(C(CSCC=C)=O)CCC2(CCC(C(=O)Nc3ccc(C)nc3NC)O2)CC1 57996,C1(C)(CNC(C2(F)CN(C(c3c(C)scn3)=O)C2)=O)CCCC1O 57997,Cc1ccc(Cl)cc1NNC(=O)NCC1Cc2cc(Br)ccc2O1 57998,c12cnc3cc(ccn13)[nH]c2=O.c1(NC(C(C)(C)c2ccno2)=O)ncc(C#N)s1 57999,C(CCCC(CO)NC(c1ccc(C)nn1)=O)NC(Cc1cccc(OC)n1)=O 58000,c1(C(N(CC(=O)Nc2cc(C)ncc2)C)=O)cc(Br)c(N)c(Br)c1 58001,c1(C(=O)NCCC2CC(NC(c3cccc(C)c3C)=O)C2)ccc2nc[nH]c2n1 58002,N1(C(CCC=C)=O)CCC2(CC(NC(=O)COC3CCCC3)CO2)C1 58003,C(c1ccc2c(c1)OCCO2)=CC(=O)N(C)CC1N(c2ncc(C)cn2)CCC1 58004,C(CC(C(C)(C)C)NC(C1CN(C)CCN1C)=O)N(C(=O)CSS(C)(=O)=O)C 58005,C1(CCNC(c2ccc(CO)cn2)=O)CN(C(C23CCC2COC3)=O)CCCO1 58006,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)CCCC(=O)O 58007,C(=O)(CCC(CF)CF)NC(C)C=CC(=O)N(C1CCOC1)CCF 58008,CC(CC(F)(F)F)C(=O)N1CCCCC(c2cn(CCOCCOCCO)nn2)C1 58009,c1(NCC2(CCC#C)CC2)c(Cc2ccc(OC)cc2)cccc1F 58010,CC(C)CC(O)C(=O)N1CCC(NC(C23CC(C2)C(C)(C)O3)=O)C1 58011,c1(NC(Cc2nccc(-c3cc(C)nnc3)c2)=O)csc2nccnc12 58012,N1(C(=O)CCC2CCCOC2)CCC2C(CCCN2C(c2ncoc2Br)=O)C1 58013,C12(CCNC(C=C3CCC(C)C3)=O)CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 58014,c1(N(CC(C)(C)OC)C)nc(NC2CCCCCC2F)c2ccc(C)cc2n1 58015,c1(C(N(CCC)C(C)C)=O)cnc2cc(-c3ccc(C(C)=O)nc3)ccn12 58016,Cc1cc(C(=O)NCC2CC(NC(=O)CS(C)(=O)=O)C2)c2ccc(F)cc2n1 58017,C1(NCCC(=O)NC(CC(=O)OCC)=O)CCN(C2CC2n2cnnn2)CC1 58018,CC1CN(C(c2cc(N)ccn2)=O)CC1NC(C1CCCO1)=O 58019,N1(C(C(CC)(C)CO)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 58020,N1(C(COC)=O)CCC(F)(F)C(CNC(c2cnccc2C(C)(C)C)=O)C1 58021,N1(C(CC(=O)NCC#C)=O)CCC(F)(C(N2CCCC(C(N)=O)CC2)=O)CC1 58022,C(C(=O)N1CCCCO1)(c1cn(C)nn1)NC(COCCCOC)=O.C(C)(=O)O 58023,c1(C(=O)NCCNC(C(C)C(C)C2CCCCC2)=O)ccc2c(ccn2C)c1 58024,N#Cc1ccc([SH2]C2CC2)cn1.c1(C(=O)N(CCSCC(=O)N)C2CC2)cnccn1 58025,Cc1c(C(=O)NC(CO)CCCNC(=O)CCc2ccccn2)cccc1Cl 58026,C(C(=O)Nn1cnn(C)c1=S)NC(CNC(c1c(CC)ccs1)=O)=O 58027,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58028,N1(C(c2c(COC)cco2)=O)CCC(C)C1CNC(=O)C(C)NC(N)=O 58029,C1(C)(C(C)O)CCOCC1.c12conc1CNC(=O)COCCNC2=O 58030,c1(C(=O)NCC2CC2CNC(=O)C2CC2)cc(F)cc(F)c1Br 58031,C1(NC(c2c(CC)nns2)=O)CC(CNC(=O)Cc2c[nH]nc2C)C12CCC2 58032,C1(C(N2CC(C)(c3n(C(C)C)ccc3)OCC2)=O)CCCCN(C)C1=O 58033,N1(C(C(C=CC)O)=O)CCCCC(C(=O)N(C(C)C(C)SC)C)C1 58034,N1(C(Cc2nc(C(=O)OC)sc2)=O)CCC(C)C(NC(=O)C2=COCCC2)C1 58035,Cc1cc(C(=O)NC(C)CNC(C2(Cl)CC2(C)C)=O)cc2nn[nH]c12 58036,CCC(C(F)(F)F)NCC1CC(CC#N)(C(C)C)C1 58037,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)NC(=O)CC1NC(=O)NC1=O 58038,CC(C)C(C)(CNC(c1nsnc1O)=O)NC(C1C=CCC1)=O 58039,c1(C(=O)NCC2CCC(CNC(C3(C)CC3(F)Cl)=O)CC2)cnc2[nH]ncc2c1 58040,CC(C)(C)C#CC(=O)N1CC(C(N)=O)(CNC(=O)CSCc2cscn2)C1 58041,c12ccc3cccnc3c1C(=O)O2.C1(COC)CCC2(CCOCC2)C1 58042,N1(C(CN(CC)CC)=O)CC(C(=O)NC(COC)C2CC2)C(C)(C)C1 58043,c1(CCN2CCC(N3CC(C)C=C(C)C3)CC2)ccccc1[N+](=O)[O-] 58044,c1(NC(C2CN(c3ncncc3C#N)CCS2)C)nc(S(C)(=O)=O)ncc1C 58045,Cn1cnnc1C(C)(C)C(=O)NCC1CCCN1C(=O)CC1CCCCO1 58046,CC1OC(C)C(C(=O)NCC2(C)CCCN2C(c2ccc(C(N)=O)[nH]2)=O)C1C 58047,C1(NC(C(c2n(C)cnc2)O)=O)CCN(C(=O)CCN2CCCC2=O)CC1 58048,N1(C(C(CC)OC)=O)CC2(CCC2NC(c2cc(COC)cn2C)=O)C1 58049,CC(O)CCCNC(=O)CCNC(C1(C(C)(F)F)CC1)=O 58050,CC(C)(O)C(F)(F)C(=O)N1CC(C(N)=O)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58051,C1(CCNC(C(C)CF)=O)CCCN(C(C2CC(F)(CF)C2)=O)C1 58052,c1(OC)cc(C(=O)NC2CN(C(=O)COC(C)C)C2)cc(Cl)c1 58053,C1(NC(CCC(C)(C)F)=O)CC2CN(C(=O)CCc3ccoc3)CCN2C1=O 58054,N1(C(=O)NC2CCC3CNCC3O2)CCC2(CCOc3ccccc32)CC1 58055,c1(C(=O)NCCCC(c2ccccc2)NC(c2ccoc2)=O)ccc(Cl)nc1O 58056,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(C)Cn2ccnc2)C1 58057,c1(OC)ccc(C(N2CC(CNC(=O)C(C)N(C)C(C)=O)C2)=O)cc1S(C)(=O)=O 58058,CN1CCN(C(C2CN(C)CCO2)=O)CC1CNC(=O)CCc1ccc(Cl)nc1 58059,NS(=O)(=O)c1nc(Cl)ccc1NC(C1CN(Cc2ccc(O)cn2)CCO1)=O 58060,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CCNC(C1CC1(C)C)=O 58061,CC#CCCCC(=O)NCC1(C)CCCN(C(=O)Cc2ccccc2Br)C1 58062,O=C1Cc2ccc(NC(c3c(F)cccc3Cl)CC(=O)O)cc2N1 58063,S(=O)(=O)(c1cccc(SCC2CC2)c1)N1C(C(C)C)CCC1C 58064,N1(c2cc(C(C)(C)C)ncn2)CCCC(CO)(NC(=O)C=Cc2cccnc2)C1 58065,C1(CNC(C(C)(N(C(=O)C(F)=CC2CC2)C)C2CC2)=O)CCOC(C)(C)C1 58066,c1(C(N(C(C)C(=O)N2CCC(N(C)C)C2)CC)=O)n[nH]c(C)c1C 58067,N1(C(CN(CCOC)C)=O)CCCC1CN(C(C12CC(CO1)C2)=O)C1CC1 58068,N1(C(CSCCOC)=O)CC2C3CCC(C2C1)N(C(=O)CC1CCC(C)(C)O1)C3 58069,CON1CCC(C(N2CC(NC(=O)CC3CCN(C)C3)CC(F)C2)=O)CC1 58070,C12(C(=O)NCC(CO)N(C)C)CCC(CN(C(=O)Cc3cc[nH]n3)C1)C2 58071,c1(NC(CC2CN(C(C3C(NC(=O)OC(C)(C)C)CC3)=O)C2)=O)ccc(Cl)cc1 58072,N1(C(CC)C)CCCC(C(=O)NC(C(=O)O)C(O)c2ccccc2)C1 58073,c1(OC)cc(C(=O)NCC2CCCN2C(C2(C)CCSCC2)=O)c2c(c1)CCC2 58074,c1(C(=O)NCC2(F)CCN(C(=O)Cc3cnsc3)CC2)coc2cccc(F)c12 58075,N1(C(C2(OCC)CN(C(=O)C3=NNC(=O)C3)C2)=O)CC(C)CC(C)C1 58076,C(=O)(C(CN(C)C)CC)N(CCC(=O)N(C)CC1CCC1O)CC#C 58077,c1(OCC)cncc(C(=O)NC2(CN(C)C(c3cc(C#N)c[nH]3)=O)CC2)c1 58078,C(C)(CCC(=O)NC1CCC1CNC(C1(CN(C)C)CC1)=O)OC 58079,C(=O)(CC(COC)COC)N1C(C(=O)NC(CCCCC)C2CC2)CCC1 58080,n1(CCC)ncc(C(=O)NCC(C2CC2)N(C)C(c2sccc2SC)=O)c1C 58081,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(c2cc(Cl)on2)=O)C1 58082,CC(C)(CF)C(=O)NC1CCCCC1NC(=O)COCC1CCC1 58083,N1(C(C(C2CCC2)NC(=O)C(O)C(F)(F)F)=O)CCC2(CCCO2)C1 58084,c1(C(=O)NC2(C)CC(CNC(C3N(C)C(=O)OC3)=O)C2)cccc2sccc12 58085,N1(C(C2CCC(N(C)C)C2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58086,N1(C(C2(C)CSC2)=O)CC(CC(=O)N(CCO)CCO)C2(CC2)C1 58087,C1(C(N(C2CCOC2)CC#C)=O)CC(O)C(O)CC1CNC(=O)C(CC)C(F)(F)F 58088,N1(C(c2ccc(OC)cc2)=O)CC2CCN(C(C3NC(=O)C4CCC34)=O)C(C2)C1 58089,c1(C(=O)NC2C(C)CN(C(C3(C)CCC3)=O)CC2)cnc2[nH]ccc2n1 58090,N1(C(Cc2nc(C)c(C)s2)=O)C2CCC1C1CC1(NC(C1CC=CCC1)=O)C2 58091,C1(CCC)CN(C(=O)CSC(F)F)CCN1Cc1c(C(=O)OC(C)=O)scc1 58092,C1(C(N2CCC(O)(CCNC(C3CC3(F)F)=O)C2)=O)CC(C2CC2)=NO1 58093,C=CC(CCC)CC(=O)N1CC=C(C(=O)NC2(CO)CC3CCCC23)CC1 58094,C1(C(=O)NCCC(C)N(C(=O)Cc2ccsn2)C)(N(C)C)CC(F)(F)C1 58095,C(=O)(C#CC1CCOCC1)N1CCCC(CC(=O)NCCC(=O)NO)CC1 58096,Cc1cc(C(=O)C(C2CC3(CCCO3)C2)=O)c(N)c(F)c1.C(CNC1(C)CC1)(CO)N 58097,Cc1cnc(C(=O)NC2CCC(CCNC(c3cccc(N(C)C)n3)=O)C2)cn1 58098,c1(OCC(=O)NC2(C3N(C(C=CCCC)=O)CCC3)CC2)cccn2ncnc12 58099,C1(C(=O)NC(C#C)(C)C2CCC2)CC(NC(=O)CC2CCCOCC2)CCO1 58100,C(=O)(C(C(C)C)C(C)C)N1C(C(=O)Nc2cncc(C)c2)CCC1C 58101,c1(C(N2CCCC(N(C)C)C2)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 58102,c1(C(N(C2CCN(C(C(C=C)c3ccccc3)=O)C2)C)=O)cc(OC)ncc1Cl 58103,N1(C(C(CC)CC(C)C)=O)CCC2(CCN(C(=O)CCc3cnc[nH]3)CC2)C1 58104,CN=c1nc(N2CCOCC(C3CCC3)C2)[nH]c(=NC2CCCCCCC2)[nH]1 58105,c1(N2CCC(CNC(=O)Nc3sccc3Br)C2)c(F)cccc1[N+](=O)[O-] 58106,C1(C(=O)N(C(C2CCCC2)CC)C(C)=O)CC2CCC1N2C(=O)Cn1nnc(C)n1 58107,c1(C(=O)NC(C)CN(C)C(c2ncc(F)cc2F)=O)cc(F)cc(Br)c1F 58108,c1(OC)ccc(F)cc1CNC(=O)CC1(C)CN(c2ncc(C)c(SC)n2)C1 58109,C(=O)(CCS(=O)(=O)CC(C)C)NCC(C)(CC)NC(C=CCOCCOC)=O 58110,C1(CN(C(C(OC)OC)=O)C)CCN(C(C2(Br)CC2)=O)C1 58111,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58112,C1(NC(c2ccns2)=O)CC2CC(C1)N(C(=O)CCOCC1CCCO1)C2 58113,C1(CNC(C2CC(CC)OCC2)=O)CC(C(F)(F)F)CCN1C(=O)C=NOC 58114,Cc1cc(O)ccc1NC(c1ccnc(C2(N)CCC2)n1)=O 58115,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C1)=O 58116,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58117,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58118,C=CCCC(C(=O)N(CC(=O)NC)CC)NC(c1ccc(C)cn1)=O 58119,N1(CC(CNC2C(C(=O)NCc3cc(C)sc3)C2)F)CCN(C)CC1 58120,c1(C(=O)NCC2(O)CN(C(c3nc(CC)sc3Cl)=O)C2)cc(C)ccc1N 58121,C1(C(N(C2CN(C(C3CCN(C)CC3)=O)C2)C)=O)CCc2nn[nH]c2C1 58122,c1(CN(CCOC)CCN(C)C)cn(CCC(=O)OC)nn1.CC(C)C 58123,c1(CC)c(C(N2CCC(N3CCCCC3)(CC)C2)=O)cnn1C(CC)CC 58124,C1(N(C)C(c2cc(=O)n(C)cn2)=O)CCCN(CCN2C(=O)CNC2=O)CC1 58125,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58126,c1(C(N2CCC(N(C(C=CCC)=O)CCOC)C2)=O)cncc2c[nH]nc12 58127,N1(C(c2c(C)csn2)=O)CCCCC1C(=O)NCC1CC=CC(O)C1 58128,N1(c2c(C#N)cncc2)CCC2(CC1)OCCC2NC(=O)C(=O)NCC(F)F 58129,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58130,c1(C(N2C(C(=O)NCCC(C)O)CC(O)C2)=O)c(F)cncc1Br 58131,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCCc2ccccn2)C(CO)C1 58132,c1(CC(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)ccccc1Cl 58133,n1(CC(N2CC(F)(CNC(c3c(OC)nn(C)c3)=O)C2)=O)cc(C)c(O)nc1=O 58134,c1(C(=O)NC(CC)CN(C(=O)CCNC(=O)CO)CC)n[nH]c2c1CCSC2 58135,c1(C(=O)NC(C(=O)NCC(c2ccncc2)C)C)cccc(CO)n1 58136,C1(c2nc(C)[nH]n2)CCN(C(=O)NC2CN(c3ncc(Br)cn3)C2)CC1 58137,C1(OCCC)CCC(CC(=O)NC2CCCN(C(=O)C(C)CSC)C2)CC1 58138,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58139,N1(C(c2c(NC)nccc2)=O)CCCOC(CNC(C23CC(C)C2C3)=O)C1 58140,N(C(=NCCCNC(=O)Nc1ccccc1)NC1CCC12CCC2)CCNC 58141,C1(NC(c2ccc(C(N)=O)cn2)=O)(CF)CCN(C(C2C=CCC2)=O)C1 58142,c1(C(N(C2CCN(C(C3(CF)CCN(C(C)=O)C3)=O)C2)C)=O)sc(C)c(C)c1C 58143,N1(CC#N)CCN(C(c2ccc(CC(N3CC(N(C)C)C(O)C3)=O)cc2)=O)CC1 58144,C1(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cncnc2)COCCC1(F)F 58145,N1(C(C=CC(CC)=CC)=O)CCCCC1C(C)(C)NC(c1ccnn1CCC)=O 58146,c1(CC(=O)NCCn2ncc(CNC(C3C(C)(C(F)F)C3)=O)c2)cccc(O)c1 58147,n1(CC)ncc(Cl)c1C(=O)NCC(C)CNC(=O)CCc1cc(C)[nH]n1 58148,C1(N(CC#C)C(c2ccoc2Br)=O)CCN(C(C2CCCCN2C(C)=O)=O)CC1 58149,C1(C(=O)NCC(C)CNC(c2cc(O)nc(Cl)c2)=O)CCC2(CCC2)O1 58150,C(C(F)(F)C(F)(F)F)N1CCC(C(N2C3(CC(N)=O)CCC2CC3)=O)CC1 58151,N1(C(=O)NC(CCC)Cc2ccccc2)CCC(C)(CCN(C)C)C1 58152,C1(N(C(=O)C(C)NS(C)(=O)=O)C)CCCN(C(c2c[nH]nc2C(C)(F)F)=O)C1 58153,n1(CC(=O)NCC(O)CNC(c2cccc(C3CC3)n2)=O)ccc([N+](=O)[O-])n1 58154,c1(C(=O)NC2C(CNC(CC(C)C)=O)CC2)ccc(N(C)C)cc1 58155,Cc1ccnc(C(=O)NC(c2ccccc2F)CNC(=O)CCOC(C)(C)C)n1 58156,c1(C(C)N(C(=O)CC2CCC(C)C2)C2CC2)nocc1NC(=O)CC1CCC1 58157,C=CCN(CC=C)NCCCC(=C)Cl.C1(C2C(=O)N2)CCOC1 58158,CC(C)(C#Cc1cn(C2CCC(CO)CC2)nn1)NC(C1(CNS(C)(=O)=O)CC1)=O 58159,C#CCCC(O)C(=O)NCCC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 58160,Cc1nc(N2C3CCCC2CC(NC(=O)C2=C(Cl)CC2)C3)c2ccsc2n1 58161,C#CC1(C(N2CC=C(C(=O)NCCCOCC=C)C2)=O)CCCCC1 58162,C1(C(CNC(C(C)OCC=C)=O)(C)C)CCCCN1C(=O)CN(C1CC1)CC 58163,c1(CC(C)C(=O)NCCN(C(=O)CSC2CC2)CC2CCCO2)ccccc1F 58164,c1(CN(CCC)C(=O)OCC2CCCO2)cc(C)cc(Br)c1.C1(=O)CO1.O 58165,CC(CC(=O)N1CCC2(CC(C(N3CCS(=O)(=O)CC3)=O)C2)C1)C(C)(C)C 58166,CCCN=C(NCc1ccccc1)NCCCS(C)(=O)=O.C12(CCCC1)OC2 58167,CC(C)C(CN(C1C2CC1N(C(=O)OC(C)(C)C)C2)C)C(=O)NC1CCCCC1 58168,C(CN=c1nc(N2CCC(NC(N(CC)CC)=O)C2)c2c([nH]1)COC2)OC 58169,c1(C(N2C(CNC(c3c(CC)nc(C)nc3)=O)CC2)=O)ccc(C#N)c(O)c1 58170,C(=O)(CCC(C)(C)NC(=O)C1=C(C)CCC1)NC(C(C(=O)OC)C)C 58171,C(=O)(C(C)CN(C(=O)C(C1CCOCC1)O)C)NC(COC)CO 58172,C(=O)(C(C)CC(F)F)NC(CC)(CNC(=O)CCOCCCOC)CC 58173,c1(C(=O)NC(C)CCNC(=O)C#CC(=O)N(C)C)cc(C(C)=O)oc1C 58174,c1(CNC(C(Cc2cn[nH]c2)NC(C2CCCSC2)=O)=O)c(F)cccc1Cl 58175,C1(CNC(C)=O)CC(C)CN(C(N2CCC(N3CCOCC3)CC2)=O)C1 58176,N1(C(C(C(C)OC)N(C)C)=O)CC2CCC2(CC(=O)NCC(n2ccnn2)C)C1 58177,c1(C2C(C(=O)NC3CC(C)(NC(CC(C)SC)=O)C3)CCO2)cn(C)nc1C 58178,C1(C(=O)OC)(CC)CCN(C(=O)CCNC(=O)C=Cc2ccnn2C)CC1 58179,c1(NCc2cc(C)cc(O)c2)nccc2ccc(-c3cnn4cccnc34)cc12 58180,N1(C(CCNC(=O)Cc2cnn(C)c2)=O)CCC2(C)CCCC12.C1(OC)CC1 58181,C=CC1(CC(=O)NCC2CC3C=CC2C3)CN(C(c2cncc(CN)c2)=O)C1 58182,C=CCC(CNC(=O)CC1CCCOC1)C(=O)NCc1cc(C)nc(C)n1 58183,C1(C(C(=O)N(CC(=O)OC)CC)F)CCN(C(c2[nH]ccc2CC)=O)C1 58184,C(=O)(C(F)(F)CCc1ccccc1)NCC1CN(C(C2(COC)CC2)=O)C1 58185,C=CC1(C(=O)Nc2cnc3c(c2)CCC3)CCN(C(=O)C(N)CC2CC2)CC1 58186,Cc1cc(OCC(=O)NC2CCC2NC(c2coc3c2COC3)=O)cc(C)c1Cl 58187,C#Cc1ccc(OCC(=O)NCCCC)cc1.c1(C(=O)NCC(C)SC)conc1 58188,c1(C(=O)NCC2CCN(C(c3cc(OC)n[nH]3)=O)C2)[nH]cnc1C#N 58189,C(=O)(C(C)CNC(=O)Cc1ncccn1)NC(C#C)(C)C1CCC1 58190,n1(CC)ncc(Cl)c1C(=O)NCC1CCCC1NC(C1(O)CC(F)(F)C1)=O 58191,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)cc(C)n1 58192,C1(NC(C(COC)Cc2ccccc2)=O)CC2CCC(C1)N2C(=O)C1=CCCS1 58193,N1(C(=O)Cc2ccon2)CCc2nc[nH]c2C12CCN(C(C1CCCCS1)=O)C2 58194,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58195,c1(C(N2CCC3(NC(c4cscn4)=O)C(C2)C3)=O)n[nH]c2c1CCCC2 58196,CC1CC1(CO)CNC(=O)C=CC(C)NC(=O)CNc1ccsc1 58197,CC1CN(C(C2CN(C(C3CC3C(F)(F)F)=O)CCN2C)=O)CC(=O)N1 58198,c1(N(C)C)ccc(CC(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCC2)cc1 58199,C123COCC1CN(C2)CCON3.C1(c2n(CCC)nnn2)(N(C)C)CCN(C)C1 58200,c1(C(N(C2CCN(Cc3ccc(F)cc3Cl)C2)C)=O)cn2ccnc2cn1 58201,N1(C(CCCCCNC(=O)CSc2cccs2)=O)CCCC(O)(C2CC2)C1 58202,c1(C(=O)NC2C(C)(C)C(CNC(=O)CN3CC4CCC3C4)C2)cc2sccc2s1 58203,C1(CC=C)(C(=O)NC2(CC)CC(F)(F)C2)CCCN1C(=O)C(C)C=C 58204,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)CC(F)(F)F)C1C1CC1 58205,C(C)(CNC(C1CC(=O)N(c2nccs2)C1)=O)(C(C)C)NC(C1C(=C)C1)=O 58206,C(=O)(C(C)(C)CS(C)(=O)=O)NCC1CCN(C(CCNC(=O)NC)=O)CC1C 58207,CC1(C)OCC2CC12NC(C1(NC(c2ccnn2CCF)=O)CC(F)(F)C1)=O 58208,C1(C(=O)O)(CC)CCN(C(=O)CCCc2ccccc2F)CC1 58209,CC(C)(CCNC(C1CCCS1)=O)NC(=O)COCCN(C)C 58210,c1(NC)ccc(C(=O)NC(C)CCNC(=O)C(=O)NC2CCCC2)c(Br)c1 58211,c1(COCC)ccc(C(=O)NCCC2CC(NC(=O)COC(C)(C)C)C2)[nH]1 58212,Cc1ccc(O)c(C)c1CNC(=O)COC1CN(C(=O)C=Cc2cocn2)C1 58213,c1(C(=O)NCC(C)(C)NC(C2C(CC)CN(C)C2)=O)ccc2c(c1)OC(C)(C)C2 58214,N1(C(Cc2c(C(=O)OC)c(C)sc2)=O)CC2CS(=O)(=O)CC2(C#N)C1 58215,CNS(=O)(=O)NCC(=O)N(C1CN(C(=O)Cn2nnc(C3CC3)n2)C1)C 58216,C12(NC(Cc3scc(C)c3)=O)CCC(CC1NC(c1c[nH]nc1C(C)(F)F)=O)C2 58217,C1(NC(c2ccoc2)=O)CCN(C(c2cccc(OCC(F)F)c2)=O)CC(O)C1 58218,N1(C(CCCC(C)O)=O)CC(NC(c2cnnn2C)=O)C2CCCCC12 58219,C(=O)(C(C)(C(F)(F)F)c1ccccc1)N1CCCN(C(C(CC)(C)F)=O)CC1 58220,CC1(C)C2CCC1(C(N1CC(=C(F)CNC(C3CCS3(=O)=O)=O)C1)=O)CC2 58221,CC(C(=O)NCC1CCN(C(C2CCCC2F)=O)C1)C(C)(F)F 58222,CCCCS(=O)(=O)NCC(=O)NCC(O)CCNC1CCCN1S(C)(=O)=O 58223,C1(NC(COC)=O)CC2CCC1(NC(=O)CCc1ccc(C)cc1)C2 58224,c1(C(=O)NC(C(=O)NCC2CC(N(C)C)C2)CO)ncc(Br)cc1F 58225,c1(C(=O)Nc2cncc(Cl)n2)ccc(=O)n2c1CNCC2 58226,C1(C)(CC)CN(C(=O)C(Cn2cncn2)NC(=O)CCC2CC(OC)C2)CCO1 58227,C=C(Cl)CC(C(=O)N1CC(OC)CC(O)C1)NC(C1C2CCC(F)C12)=O 58228,N1(C(CCC2CC(C)C2)=O)CCN(C(c2cc(Br)cnc2O)=O)CC2(CC2)C1 58229,C(=O)(C1=CCN(C(c2cn(C)c(=O)cn2)=O)C1)NCC1(C(=O)OCC)CC1 58230,N1(C(COCCOC)=O)CCCC2CN(C(=O)C(CC(F)F)OC)CCC12 58231,c1(C(C(=O)N(C(C)CNC(=O)CCC2(C)CC2)CC)O)ccc(Cl)cc1 58232,C1(F)(CNC(C2CCC(CN(C)C)C2)=O)CCC(CNC(C2CC2C#N)=O)CC1 58233,N1(C(c2cnc(C)[nH]2)=O)CC2OCCN(C(=O)CC3CC4CC4C3)C2C1 58234,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58235,c1(OCC)ccc(C(=O)N(C(C)CCNC(c2cscc2CC)=O)C)cc1C 58236,Cc1nc2cc(C(=O)NCC(C)N(C)C(C3CCCCN3N=O)=O)c(F)cc2[nH]1 58237,N1(C(COCC)=O)CC2CCC2(CNC(c2ccc(N3CCC(C)C3)cc2)=O)C1 58238,C=C(C)CCCC(=O)Nc1nc(Cl)ccc1NCCNC(C1CCC1)=O 58239,Cc1ccc(C(=O)NCC2(O)CCCN(C(c3nnc(O)nc3O)=O)C2)c(N)n1 58240,N1(C(CN(C(=O)CN2CCNC2=O)CC#C)=O)CCCC2(CCCO2)C1 58241,C1(C(N(C(C)(C)C)CC)=O)CCC(CS(=O)(=O)NC(c2cnco2)C)O1 58242,C(CCC(C)(C)C(=O)N1CCC(O)(C=C)C1)n1cc(N(C(C(C=C)CC)=O)C)nn1 58243,C1(C(=O)NCC(C(C)(C)C)NC(=O)C(C)O)(OC)CCCCCCC1 58244,c1(C(=O)NC2CC3(C(NC(c4occ(C)c4)=O)C3)C2)ccc2c(c1)C(=O)CCC2 58245,CCC(C)(CNC(C1CCCCC1O)=O)C(=O)NC(c1ccccc1)C 58246,N1(C(CC(CC)O)=O)C(C(=O)NC2CCCCNC2=O)CCC12CC2 58247,C1(NC(C(CC)OCC)=O)CCCN(Cc2ccnc(Cl)c2F)C1C 58248,C=CC1CN(C(C2CC(C(F)F)(OC)C2)=O)CC1NC(C1CCCCCCC1)=O 58249,CC1(C)C=C(C(=O)NC2CCC(NC(C3(F)CCCOC3)=O)C2)C1 58250,C1(C(=O)NC(CC)C(O)c2ccccc2)CCc2cnn(CCC(C)C)c2C1 58251,C(C)(c1cnn(C)c1)=CC(=O)NCC(CNC(CN(C(=O)OC(C)(C)C)CC)=O)F 58252,C1(CNC(c2cn(C(C)C)nn2)=O)CN(C(C2(C(=O)N(C)C)CC2)=O)CCC1C 58253,C#CC1(C)CCC(CNC(=O)C(CNC(C2COC(=O)N2)=O)C(C)C)CC1 58254,N1(C(CC#C)=O)CCC2C(CCN2C(C2COc3ccccc3O2)=O)C1 58255,C1(C(N(C2CCN(C(c3cccc(F)n3)=O)CC2)C)=O)C2CCCOC12 58256,C=C=CC(C)C(=O)NC1CC(c2ccccc2)(CNC(=O)CN(C)C2CC2)C1 58257,C12(NC(C(CSC)O)=O)CC(C1)N(C(=O)C(c1cccc(C(F)(F)F)c1)O)C2 58258,C(=O)(C1Cc2ccc(F)cc21)OC.C12(N)CC(C1)CN2 58259,C=CC(C)(O)C(=O)N(CC(=O)NCC(O)C(C)(C)C)CC(C)C 58260,N1(C(C2CC(C)(CC)C2)=O)CCCCCC(NC(c2ccc(F)cn2)=O)C1 58261,c1(C(=O)NC2CCC(N(C(C(CC)CC)=O)C)C2)ccc2c(c1)C(=O)NC2=O 58262,c1(CNC(C(c2ccc(F)c(F)c2)C)=O)nc2c(s1)CN(C(=O)CC(C)(F)F)CC2 58263,Cc1nccn1CCNC(c1nnnn1C1(C)CC1)C1C=CCC1 58264,CC(C)CC(CNC(c1cc(CO)[nH]n1)=O)C(=O)NC1CC(CO)C1 58265,c1(C(N2CC(CC(C)NC(c3cnc(O)nc3O)=O)C2)=O)ccc2snnc2c1 58266,N1(C(C(C)CN)=O)CCCC2(C(=O)NCc3ccccc3)CC2C1 58267,FCCCN=C(NCc1ccc2ccoc2c1)NCC1(C2CC2)CCCO1 58268,C(=O)(C(C)C(C)NC(=O)CC1CN(C(c2cncn2C)=O)CC1C)OC 58269,C1(C(=O)NC(CC=C)CC=C)CC(NC(=O)Cc2cccnc2C)C12CCC2 58270,c1(C(=O)NCC(CNC(c2c(C)coc2)=O)C)ccc2nc(O)nc(O)c2c1 58271,c1(C(N(CCOCCCNC(C2CC2COC)=O)C)=O)ncncc1Cl 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58307,c1(C(CC)Nc2csc(-c3ccccc3OCCN(C)C)n2)ccnc(F)c1 58308,c1(OCC)ncccc1C(=O)NC1(CCCNC(C2CC(=O)NC2=O)=O)CC1 58309,C1(NC(C(C)(CO)OC)=O)CCN(C(C2CSCC(=O)N2)=O)CC1O 58310,N1(C(C2C(NCc3c(C(=O)O)cccc3)CCCC2)=O)CC2CCCCC2C1 58311,C1(CNC(C(F)OC)=O)(OC)CCN(C(=O)C(C)CSc2ccccc2)C1 58312,C(C1CN(C(=O)Cc2cnc(C)s2)CC1C(=O)NC1CC1c1ccsc1)=CC 58313,c1(SCC(=O)NCC(CN(C)C(c2noc(C(C)(C)C)n2)=O)O)ccc(Cl)cc1 58314,N(C1=C(C#N)CCC1)CCNC(=O)C(N1CCC(N2C(C)CCC2)CC1)=O 58315,c1(N(C(=O)NC(c2cc(F)ccc2N)C)C)ccc(S(C)(=O)=O)o1 58316,C1(N(C)C)CCN(C(c2c(CNC(=O)C=Cc3cccnc3)cnn2C)=O)CC1 58317,CCCCC(F)C(=O)NCc1cc(C(=O)NCc2cc(C)[nH]n2)co1 58318,S(=O)(=O)(c1ccc(NC2CCOC3(CCCC3)C2)c(F)c1)NC(CC(C)C)C 58319,CC1CC2(CC(C(=O)NCC3(NC(=O)COCC4CCOC4)CCOC3)C2)C1 58320,C1(NC(c2cc(C)sc2C)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 58321,C1(NC(C2CN3CCC2C3)=O)COCCN(C(C2(CC3CCC3)CC2)=O)C1 58322,CC1(C)CCCC(O)(C(N2CCC2CNC(=O)CC2CC2(C)C)=O)CC1 58323,CC1(C)C(CC(=O)NCCN(C(=O)CSc2ccco2)C2CC2)CC1O 58324,CC1(C)COC(C(=O)NC2CCCC(CNC(c3cc(Cl)ccc3Cl)=O)C2)CO1 58325,C1(C(=O)NCCCC(=O)NC(c2ccc(O)cc2)C)C2C=CC(C2)C1N 58326,C1(C(N=c2ccn(C)[nH]2)=O)CCCC12CCN(C(=O)Cc1cc(F)c(Br)cc1F)C2 58327,Cc1[nH]ccc1C=CC(=O)NC(C1CC1C(=O)N(C)Cc1nncn1C)C 58328,C(CCNC(=O)CCc1cc(C)no1)(C(C)C)NC(COC(CC)(C)C)=O 58329,C(=O)(CC(CCC)OC)N(CCNC(=O)Cc1cc(C2CCOCC2)no1)C1CC1 58330,C(=O)(C(C)CC(F)(F)F)N(CCN(C(=O)Cc1ccn(C)c1)CC)CC 58331,C(CCC(O)C(=O)NCc1ncco1)NC(c1cc(CC)nn1C)=O 58332,C(=O)(CCCC(=O)N1CC(N(C)C(C2CCC(C)O2)=O)C(O)C1)N(CC)CC 58333,CN1CC(C)(C)CC1C(=O)NC1CC=C(C(=O)NCCCCF)C1 58334,c1(OC)cc(OC)cc(CS(=O)(=O)N(C(c2cnc(C)n2C)=O)CC2CCC2)c1 58335,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CN3CCC2CC3)=O)C(O)C1 58336,N1(C(Cn2ncc(C#C)c2)=O)CCC2(CCCN2C(c2ncoc2C2CC2)=O)C1 58337,C1(O)(C(N2CC(C)(C)OCC2CNC(c2c[nH]c(=N)s2)=O)=O)CN2CCC1CC2 58338,c1(C(=O)NCC(C)NC(=O)CC2CC2C(F)(F)F)c(O)nnc2c1CCC2 58339,c1(OC)cc(NC(C)(CNC(=O)CN2CCSCC2)CO)cc(I)c1OC 58340,C1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)C2)CCC(C(F)(F)F)CC1 58341,c1(C(c2n(CC(=C)C)nnn2)NCCc2ncc(C(C)(C)C)s2)cc(Cl)ccn1 58342,C1(NC(=O)NCc2onc(C(C)OCC)n2)CC(=O)N(C2CCC(=O)NC2)C1 58343,CCCC(C#N)C(=O)NC(C(=O)NOCC(=O)OC)c1ccoc1 58344,c1(C(=O)NC(C(C)C)CNC(c2cc(CF)on2)=O)nc(Cl)ccc1F 58345,CC1CC=C(C(=O)NCC#CC(=O)NCCn2cnnn2)CC1 58346,C(=O)(C(CC(C)C)C(C)C)N(C(CC)CNC(c1nnn2c1C(=O)NCC2)=O)C 58347,C1(N(C(C2CCN(CC)CC2)=O)C2CC2)CN(C(C)=O)C(C)(C(=O)O)C1 58348,C#Cc1ccc(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CC2(C)C)cc1F 58349,C1(F)(C(=O)NCCN(C)C(c2cncc(-n3cncn3)n2)=O)CCOCC1 58350,Cc1ccc(C(=O)NCCCCCCNC(C2CC2Cl)=O)c(O)c1 58351,N1(C(C2C(CCOC)C2)=O)CC2(CNC(c3cnccn3)=O)CC1(COC)C2 58352,C1(CNC(C=C(COC)C)=O)C(C)CCN1C(C1(C)CC2(CC2)C1)=O 58353,C1(C(N)=O)CN(C(=O)CC2(CNC(=O)CN3CC4CC4C3)CC2)C2(CCC2)C1 58354,Cc1cccc2c1CC(C)(C(=O)NCC1COCCN1CC1(NC(N)=O)CC1)C2 58355,N1(CC)CCCC1CC(=O)N(CC(C)(C)CNC(=O)C=Cc1ncc[nH]1)C 58356,C(=O)(CCC(=O)N1CC(c2ocnc2C(=O)NCC2COCCO2)C1)NC 58357,c12coc(cc1=O)C(=O)N2.C1(C)(COC)CCCN1C(=O)C(=O)NCC1CC1 58358,C1(OC)CCCCC1C(N1CC(C(N)=O)(CNC(c2cc(C)sc2C)=O)C1)=O 58359,C1(NC(C23C(CN(C(C(CC)n4cncn4)=O)C2)C3)=O)CC2(CCCO2)C1 58360,C1(O)(CCNC(c2c(C)nsc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1 58361,C(=O)(CCCCCC(C)O)N1CCN(C(COCCCOCC)=O)CC1CO 58362,c1(N(C)C)ccc(C(=O)NC2CCN(C(C3CC3(F)F)=O)C2C2CC2)c(O)c1 58363,C1(CC(=O)NCC2CC(NC(c3cc(C)[nH]n3)=O)C2)CCC2(CCOCC2)CO1 58364,C1(C(N2C(CCNC(c3ccc(NC)cc3)=O)CCC2)=O)CC2(C1)CC21CC1 58365,N1(C(CCSC)=O)CCN(C(C2CCC(=O)N2CCC(F)(F)F)=O)CC1C(C)C 58366,C12(C(N(C3CCCCCC3)CCNC(=O)CCc3ccco3)=O)CCC(CO1)C2 58367,N1(C(c2nc(C)on2)C)CCC2(CCN(C(C3CCOC3)=O)CC2)C1 58368,c1(CNC(C2(CN(C)C)CC2)=O)ccc(CNC(=O)CC2(O)CCCC2)cc1F 58369,C1(C(=O)OC(C)(C)C)CC(OC)C12CCOCC2.c1(OC)ccc2cc1-2 58370,C1(c2nccc(Cl)n2)(C(=O)NCCC(C)O)CCCC1 58371,N1(C(C(C)(C)CO)=O)CC2CCN(C(c3conc3C3CCCC3)=O)CCC2C1 58372,C1(C(N(C2CCN(C(=O)C(CC3CC3)OC)C2)CC)=O)CCOC(C)C1 58373,c1(C(=O)NC2C(CNC(C(C)NC(N)=O)=O)CCC2)ccc(N)cc1 58374,c1(C(=O)OC(C)(C)C)nc(C(=O)NCC(C2CCCC2)NC(C2CCCO2)=O)cs1 58375,c1(OC)ccc(C2(C(N3CC4CC4(CNC(c4ccccc4)=O)C3)=O)CC2)cc1 58376,CC1(CNC(C2CC2C#N)=O)CCN(Cc2cccnc2Cl)CC1 58377,C#Cc1ccccc1CNC1C2CC1N(c1nccc(OC)n1)C2 58378,c1(N(C)CC)nc(CN(C(CC)C(=O)Nc2ccccc2F)CC)nc(=N)[nH]1 58379,c1(N(CC(F)F)C)ccn2ncc(S(=O)(=O)NC3CCc4c(nnn4C)C3)c2n1 58380,N1(C(CC(CCC)O)=O)CCC2CCCCC2CC1 58381,C1(=CCNC(C(C)OCc2ccccn2)=O)CCN(C(c2cnco2)=O)CC1 58382,C12(CNC(c3ccn(CCNC(C(CCC)F)=O)c3)=O)CCCN(CC1)C2 58383,Cc1nn(C2CC2)cc1C(C=O)NCCCF.c1(CC2CCC2)nc(C2CC2)cs1 58384,CC1CC(NC(=O)C(=O)NCC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58385,CC(C)C(C(F)(F)F)NC(C1COCC1NC(C1CCCCO1)=O)=O 58386,N1(C(CC23CC(NC(COC(C)=O)=O)(C2)C3)=O)CCC(CO)C1(C)C 58387,c1(CC(=O)NC2C(SC)CN(C(=O)C3=CC(C)(C)C3)C2)cc(Cl)c2c(c1)CCO2 58388,N1(CC(=O)NCCN2CCC(C)C2)CCN(C(=O)Nc2ccccc2)CC1=O 58389,N1(C(C(c2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58390,C1(F)(C(N(CCOCC#C)C)=O)CCN(C(C23CCN(CC2)CC3)=O)CC1 58391,N(C1CCCc2occc21)C(CC1(C=C)CN(C(C2(COC)CCCC2)=O)C1)=O 58392,C1(N(C(Cc2c(C)non2)=O)CCO)CCCN(C(=O)C(F)CC2CC2)C1 58393,c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)c(C)ccc2ncccc12 58394,Cc1nnc(CCCC(=O)N(CC(O)CNC(c2ccc(CO)cn2)=O)C)n1C 58395,Cc1nc(CC(=O)NC(CO)CCCNC(c2cccnc2N)=O)n[nH]1 58396,C(=O)(CC(C)C(=O)NC1COCC1CNC(c1cnn[nH]1)=O)OC 58397,CN1CCC(n2cc(C(=O)NCC3COC(CNc4nccs4)C3)cn2)CC1 58398,N1(C(C2CCCN(C(C)=O)C2)=O)CC2(CC(NC(c3cc(F)cnc3O)=O)C2)C1 58399,C(=O)(CC(C)(C)C(C)(F)F)N(C)CC1(NC(C2N(CC)CCC2)=O)CC1 58400,c1(CC(=O)NCCN(C(C=Cc2scc(C)n2)=O)C2CC2)ccc2ncnn2c1 58401,c1(C(N2CCC(NC(C(CC)N(C)C)=O)C2C)=O)cnn2cc(OC)ccc12 58402,N1(C(c2nc(CC)sc2)=O)CC(N(C(=O)CN=S(C)(C)=O)C)C2(CC2)C1 58403,c1(C(=O)N)cnc(N(C)C)nc1.N1(CC(=O)NC)CC=CC1.C1(=O)CC2(CC2)N1 58404,C(=O)(C#CC1CCC1)NCC(CC)C(=O)N1CCOC(c2nn[nH]n2)C1 58405,C1(CNC(Cc2cc(C)[nH]n2)=O)CCN(c2nnc(CC3CC3)s2)CC1 58406,c1(C(N(CC(O)CN(C)C(C2CCC2)=O)C)=O)ccc2nn[nH]c2c1 58407,CC(CC(C)NC(=O)CC(C)c1cnn(C)c1)NC(c1n[nH]cc1Cl)=O 58408,N1(C(c2ccc(C=C)cc2)C(=O)NCCC#N)c2ccccc2C(C)C1C 58409,C(CNC(c1ccc(F)cc1)=O)(CC(=O)NC1CCCOC1)OC 58410,C12CCCCCN(C1)C2=O.c1(NC(C=CCOCCOC)=O)ccccn1 58411,N1(C(CCCCCN(C)C)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58412,c1(OC)nc(-c2ccco2)ccc1C(=O)Nc1cnnn1C 58413,C1(C(=O)NCCCOCC#C)CCC2CCC1N2C(c1cccc(=O)n1C)=O 58414,C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2(C(F)F)CC2)=O)CCO1 58415,c1(N(CC(=O)NC2(COCC)CCOC2)CC)ccc(Cl)cc1 58416,c1(C(N2C(C(=O)Nc3ccc(C)cc3)CSC2)=O)ccc(C)c(Cl)c1 58417,C(=O)(C(CNC(C1CC(N2CCCC2)C1)=O)Cc1ccc(O)cc1)OCC 58418,N1(C(C2(C)CC(C)(C)C2)=O)CCC(C2CC2)(NC(=O)C(Cl)=CCl)C1 58419,c1(C(C)(C)C)cc(C(=O)OCCCNC(=O)Cn2cnnc2)ccc1F 58420,N1(C(C(=C(C)C2CC2)F)=O)CCC(CNC(C2CCC(C)O2)=O)C1(C)C 58421,CN1CC(NC(c2cnn(CCNC(=O)CC3CNC(=O)O3)c2)=O)CC1=O 58422,N1(CC2CN(CCC)C(=O)C2)CC2(C1)CN(C(=O)C(OC)OC)CC2CO 58423,CSC1=C(C(=O)NCC2CCC(NC(C3CCC(C(C)C)CC3)=O)C2)CCCC1 58424,Cc1cc(C(=O)N(CC(C)CNC(=O)C(=O)N(C)C)C)ccc1C1CC1 58425,C1(C(=O)NCCc2n[nH]cc2C(=O)NC(C)C(C)SC2CC2)(CC)CCOC1 58426,C(=O)(C(COC)(CC)CC)NCC(CC=C)NC(=O)C=C1CN2CCC1CC2 58427,N1(C(CC2CCC(C)CC2)=O)CC2(CCC2NC(=O)C=Cc2cn(C)cn2)C1 58428,Cc1cccc(O)c1C(N1CC(NC(=O)C(c2cncnc2)C)C(C)(C)C1)=O 58429,S1(=O)(=O)c2ccc(c(Br)c2)NC2CCCN1C2.C(CC(C)(C)F)N 58430,C(CC(=O)NC1CC1)OCCN(C(=O)C(C1CC1)NC(N)=O)C 58431,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58432,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)COC(C)C)C2)CC1 58433,C1(NC(=O)C(F)CC2CCC2)C2CC1N(C(C1(N3CCOCC3)CCOC1)=O)C2 58434,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2(F)Cl)=O)C1 58435,C1(C(=O)NCC(CCNC(=O)CNC(N)=O)OC)C(C#N)C1(C)C 58436,Cc1c(NCCCN2CCN(C)CC2)ncnc1N1CCCC2(CC2)C1 58437,c1(OC)cccc(CC(N2CCCC(NC(c3scnc3C3CC3)=O)C2)=O)c1F 58438,c1(OC)nscc1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 58439,C1(NC(C(C)OCCOC)=O)(COC)CCN(C(c2cnc(C)s2)=O)CC1 58440,N1(C(CNC(=O)C(C)Cc2cnn(C)c2)=O)CCCC1CN(C)C.CO 58441,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58442,Cc1ncccc1CC(=O)NC(CNC(C1(C(=O)N(C)C)CC1)=O)CC(C)C 58443,C1(CN(C(C)=O)CC)CCN(C(c2c[nH]cc2-c2csc(C)n2)=O)CC1 58444,C(=O)(C(F)n1ccnc1)NCCCN(C(C1CCSC1)=O)CC 58445,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58446,CCC(CC(=O)NC12CC(C(=O)NC3CC(OC)C3)(C1)C2)CC(C)C 58447,c1(C(N(CC(CC)NC(=O)CC(C)C2CC2)C)=O)cc(O)ccc1OC(F)F 58448,Cc1cnc(NC2CCN(C(=O)Cn3ccc(O)nc3=O)CC2C)nc1C 58449,C1(CNC(C(COc2ccccc2)OC)=O)(CO)CCN(C(=O)CC(C)C)C1 58450,C#CCC(C)(C)C(=O)NCC1(C(N2CCCCC(SC)C2)=O)CC1 58451,C1(OCC(=O)NCc2ncc(CO)o2)CC2(C1)CC2C(=O)NC1CCOC1 58452,Cc1c(F)ccc(Cl)c1C(=O)NCCN(C(=O)CC1=CCCC1)C(C)C 58453,Cc1csc(CCCC(=O)NCC)n1.C1(C)(N)CCOC1.C12CC(C1)NC2=O 58454,C1(C(N2CC(C(=O)OC)CC(C)C2)=O)(NC(CCC#C)=O)CCC(C)(C)C1 58455,C1(C(=O)NC2C(C)C2)CCOCCN1C(=O)CNC=O 58456,N1(C(CN(C)C(N)=O)=O)CCC(CN(C)C(C2CC(O)(C(F)(F)F)C2)=O)C1 58457,c1(C(N2C(CNC(C(C=C)(F)F)=O)CCCC2)=O)cccc(Br)c1F 58458,N12CCC(C(c3ccccc3)C1)N(C1CC1)CCC2.Clc1nccs1 58459,C(=O)(C1=CCCOC1)N1CCC(CCOC)(NC(=O)CC2CCCN2C)C1 58460,c12cnc(nc1)[nH]c2=O.c1(C2CC2)ccc(C2CC2)o1.C12(CC1)C(=O)N(C)C2 58461,C(CNC(C1CCC(N(C)C)CC1)=O)(CC(F)(F)F)NC(C(c1ccccn1)C)=O 58462,CCC(C)C(O)C(=O)NC1(C(C)NC(=O)CCC(=O)NCCC)CCOCC1 58463,CCCC(C)(C)CC(=O)NCC(C)CC(=O)NCCc1cc(C)no1 58464,C12(CCNC(CCCC#N)=O)CCC1CN(C(=O)CCc1cnc(O)[nH]1)C2 58465,c1(NC(=O)C=CC(=O)OCC)ccc(C(N2CCC(CCC=C)C2)=O)cn1 58466,c1(CCOC)nc(=NCC2(CNC(=O)C3=CCCO3)CCCC2)s[nH]1 58467,c1(CC(N2CC(NC(c3cc(C)sc3)=O)C3C2C3)=O)cc(F)cc(F)c1 58468,c1(NCC2C(C)CCN(C(C3CCCS3)=O)C2)cccc(F)c1[N+](=O)[O-] 58469,CC(N=c1[nH]c(N2CC3CCC(CC3)C2)nc(=N)[nH]1)c1ccc(O)nc1 58470,C1(NC(C(CC)C)=O)CN(C(=O)C(C)(C)CC)CC12CCOCC2 58471,C1(N(C(C2CC2CCN(C)C)=O)CC)CCCN(C(=O)Cc2cnc(C)o2)C1 58472,c1(C(c2nnnn2C2(C)CC2)CC(CSC)OC)ccc2ccccc2c1Br 58473,CC(CC1=CCCCC1)(c1nnnn1C1CCC1)N(CCCF)C(N)=O 58474,CC1(C)CN(C(=O)C(N2CCC3(C2)OCCO3)=O)Cc2cc(Br)cnc21 58475,C1(C(=O)NCCOC)CCC2CCC1N2CC(=O)NCC(c1cccc(Cl)c1)=O 58476,C1(CNC(C(c2ccccc2)OC)=O)CN(C(c2cnc(O)cc2C)=O)C(C)(C)C1 58477,C1(NC(c2cn(CC=C)nc2)=O)CCCC(NC(c2c[nH]nc2Br)=O)CC1 58478,C(C(C(=O)NCC(C)OCCO)C(C)C)NC(C1(C#C)CCCC1)=O 58479,C1(CNC(C(C)Oc2ccc(O)nc2)=O)CN(C(=O)COCCCF)C(C)(C)C1 58480,c1(-n2cc(C3N(C(C(C)OCC)=O)CCC3)nn2)c(F)cccc1Cl 58481,Cc1nc[nH]c1CC(=O)NCCOCCCNC(=O)CC1CS(=O)(=O)C1 58482,c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nn2)c(C)noc1C 58483,C1(C)(C(N2C(CCNC(C3N(C)CCCC3)=O)CCCC2)=O)CCC2CC2C1 58484,N1(CC(N2CC(=O)N(CCc3ccccc3)C2)=O)C(=O)c2cccnc2C1=O 58485,C1(NC(c2cn(CCN(C)C)nn2)=O)CC(CNC(C2C=CCCC2)=O)C(O)C1 58486,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)COCC2)=O)cnn2c1OCCC2 58487,C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(CCC#C)=O 58488,C1(C(N(C(CC)COC)C)=O)CC2CCC(C1)N2C(c1csc(Br)c1)=O 58489,C1(n2cc(CN(C(Cc3c(C)c(Cl)ccc3)=O)O)nn2)CCC2(CCCOC2)O1 58490,C1(O)(CN(C(C(C)c2cc[nH]n2)=O)C)CCN(C(=O)CCn2ncn(C)c2=O)C1 58491,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58492,Cc1ccnc(C)c1C(=O)NCC12CC1CN(C(C1CCOC1)=O)C2 58493,N1(Cc2cc(OC)c(Br)cc2)CCC(F)(F)C(C(=O)N=c2cc(C)[nH][nH]2)C1 58494,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1C(F)F)C(F)(F)C(F)F 58495,Cc1cn2cccc(C(=O)NCCC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58496,c1(C(N2CC(NC(C(C)C3CCC3)=O)C(C)CC2)=O)ccc2scnc2c1 58497,C1(NC(C=COCC)=O)CN(C(=O)CC(C)OC)CC2(CC2)C1 58498,CC(CC(C)(F)F)C(=O)NC(C)(C)CCNC(c1ncc[nH]c1=O)=O 58499,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CC(=O)NCc2c(C)con2)C1(C)C 58500,CC1(C)CCC2(CC1)OCC(COC1CCc3nc(CN)cn3C1)O2 58501,N1(C(c2nc(C)on2)=O)CCC(C2CCN(C(=O)C(C3CCOCC3)F)CC2)CC1 58502,c1(C(N2CCN(C(c3cc(CC(C)C)[nH]n3)=O)C3C2C3)=O)cc2ncccn2n1 58503,c1(CC)cscc1CC1N(C(=O)Cn2ccc(C(F)(F)F)n2)CC1 58504,CCC(C)CC(C(=O)N(CC(C)(C)COC)C)NC(=O)C1=C(Cl)CCOC1 58505,N1(C(Cc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CCOC(C)C)CC1 58506,C12(C(N3CC(NC(COCCOC)=O)C3)=O)CC(c3ccccc3)(C1)C2F 58507,C1(C2CCN(C(=O)C=CC(F)(F)F)CC2)(NC(CC2CCN(C)C2=O)=O)CCC1 58508,C1(SC)CN(C(=O)C(C)OC2CCOCC2)CC1NC(c1ccoc1Cl)=O 58509,N1(C(CNC=O)=O)CCCC1C1(NC(c2sccc2NN2CCC2)=O)CC1 58510,C1(C(=O)NC(CCC(=O)NCC(=C)F)C)CC(=O)C12CCC2 58511,C1(NC(c2cccc(C)c2)=O)CC(NC(c2nn(C)cc2CO)=O)C12CCC2 58512,C1(N(C(=O)CSCC(c2cn(CC(=O)O)nn2)C)CC)CCCCC1 58513,N1(C(C(Cc2cnc[nH]2)OC)=O)CC(NC(=O)CCF)C(c2ccccc2)C1 58514,c1(-c2cn(CCCC(=O)NC(COC)C(C)C)nn2)cc(Br)c(C)o1 58515,CC1(F)CN(C(c2ccoc2Br)=O)CCN(C(c2cnccc2Cl)=O)C1 58516,CCC(C)C(CC(=O)N1CCN(C=O)CC1)NC(c1ccncc1OC)=O 58517,C1(C(=O)NOCC2CC3CCC3C2)CSCCN1C(=O)Cc1ccco1 58518,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)C(C)NC(c2ccoc2)=O)CC1C 58519,N1(C(c2cccc(C#C)c2C)=O)CCC2C(CCN2C(c2cnccn2)=O)C1 58520,c1(SC)cccc(C(=O)NC2CCC(CNC(C3(C)C=CCC3)=O)C2)c1Cl 58521,CC1(NC(c2nccnc2Cl)=O)CCN(Cc2ccccc2)CC1 58522,CC1CC(c2cn(-c3ccncc3)nn2)CCN1C(=O)C(C)(C)Nc1ccccn1 58523,C(=O)(CCC(C)CN(C)C)NC(CC(C)NC(c1sc(C(=O)OC)c(N)c1)=O)C 58524,CC1CN(C(c2cccc(C3(F)CCN(C(=O)OC(C)(C)C)C3)c2)=O)CC(=O)N1 58525,CC1(C)CC(CNC(c2cnn(CC3CC3)c2)=O)CN1C(C1CCCC(=O)O1)=O 58526,c1(OC)cnnc(C(N2CC(CNC(=O)CC(c3ccccc3F)O)C2)=O)c1 58527,C1(C(=O)NCCOCC#C)(CSC)CCCN1C(=O)CC1(O)CCCCC1 58528,c1(NC(C2(F)CCN(Cc3nc(C)sc3)C2)=O)cncc(Br)c1C 58529,c1(C(N(CCN(C(c2ccc(C#C)o2)=O)C)C)=O)ccc(C(F)(F)F)cc1O 58530,Cn1c(C(N2CC=CC(NC(=O)C(O)CN3CCOCC3)C2)=O)nnc1S 58531,N1(C(c2c(C)cc[nH]2)=O)CC(NC(c2cnn(C)c(=O)c2)=O)C(C2CC2)C1 58532,C1(NC(c2ccc(CNC(CCC#CC)=O)cn2)=O)CCCC(O)C1O 58533,C12(CNC(C(C)=CC)=O)COCCN1C(=O)CN(C(c1cc3n(n1)CCC3)=O)C2 58534,N1(C(c2ccn(CC)n2)=O)CCC(NC(c2cn(C)cc2C)=O)CC1C1CC1 58535,c1(N2C(C(=O)Nc3ccc(C#N)cc3F)CC3CC32)ncnc2ccc(Br)cc12 58536,Cc1oc(C)c(C(=O)N(C(C)CNC(=O)CNC(c2nc(C3CC3)no2)=O)C)c1C 58537,C(=O)(C#CC1CCCCO1)N(C1CCC(NC(c2sc(C)c(C)c2C)=O)CC1)C 58538,c1(-c2c(C(=O)OCC(=O)NC3CC(C)OC3=O)cccn2)ccn2ccccc12 58539,S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCN(C(=O)CCn3cncn3)C2CCC1 58540,CCC(F)(F)CC(=O)NCC1CN(C(c2coc(CC3CC3)n2)=O)CCCO1 58541,c1(C(=O)NCC(c2ccc(F)cc2)NC(CCCC)=O)c(F)cc(C)cc1Cl 58542,CC(CC(=O)NCC(CNC(=O)C=Cc1ccoc1)CO)c1cnn(C)c1 58543,c1(OC)nccc(C(N2CCN(C(=O)C(C)CC3CCCC3)C(CF)C2)=O)c1N 58544,N1(C(C(CC(=C)C)OC)=O)CCCC(O)(CNC(=O)C(C)OCC)CC1 58545,c1(C(N2CCN(C(C3(CC=C)CC3)=O)CC2C2CC2)=O)ccc2c(c1)CCC=C2 58546,C12CCCC(C1)C(=O)N2.Cc1nc[nH]c1CC(=O)NC1(C)CN(C(C)C)C1 58547,c1(C2C(C(=O)NC(CC(C)NC(c3n(CC)nnc3)=O)C)C2)cccc(C#N)c1 58548,C(Cc1ccoc1)(C(=O)N(C1CC1)Cc1nncs1)NC(C=CC(C)(C)C)=O 58549,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58550,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)c1ccco1)NCC(CC)NC(=O)NC 58551,Cc1cc(C(=O)NCC(C)(C)NC(=O)CCc2cnn(C)n2)cn1C(C)C 58552,C1(NC(c2scc(C(N(C(C)C)C)=O)c2)=O)CC(F)(F)C1(C)C 58553,CCC(CN(C)C)CC(=O)N(CCCC(=O)NCC1(C)CC1(F)F)C 58554,c1(CCNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58555,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58556,N1(C(C(C)Sc2ccncc2)=O)CCC(CO)(NC(=O)COCCCF)C1 58557,C(=O)(C(C)(CO)NC(=O)C=CC1CCCCC1)N1CC(F)(C(N)=O)C1 58558,C1(CNC(C(Cn2cccn2)NC(C(C=CC)O)=O)=O)CCCC12CC2 58559,C(=O)(C(O)CC(=O)OC(C)(C)C)NC(CN(C(CN(C)C)=O)CCC#N)C 58560,N1(C(C2(CO)CC(F)(F)C2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58561,c1(CCn2c3nc(n2)C3)cc(F)cc(Cl)c1.n1(COC(C)(C)C)ccnc1 58562,C=CCC(CC(F)F)NC(=O)C(COC)NC(=O)C(c1cccn1C)=O 58563,C1(N(C(C2C(C(C)NC(=O)Cn3ccnn3)C2)=O)C)CCCCCC1O 58564,N1(C(c2n(C)nc(O)c2)=O)CCS(=O)(=O)C(CCNC(=O)C(F)C2CCCC2)C1 58565,CCC(CC)(CCNC(c1nnc(CO)s1)=O)NC(=O)Cc1ccc(Cl)cc1F 58566,CCCCC(CNC(=O)CC(C)F)NC(c1cnc(-c2cccs2)o1)=O 58567,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CC=C)=O)C2CCCCCC12 58568,N(C1CCCOc2ccc(SC)cc21)C(=O)Nc1ccc(OC)c(F)c1 58569,CCCC(C)(C)CC(=O)N1CC2CC1(C(N1CCCC(C)CC1)=O)C2 58570,N1(C(CCN(C(C2(CC#C)CCCO2)=O)C2CC2)=O)CCSC(C)(C)C1 58571,C1(OC)CCC12CC(C(=O)NC1CC1NC(c1c(C)noc1C)=O)C2 58572,c1(OCCC(=O)N(C2(O)CCN(C(C3(SCC)CC3)=O)C2)C)ccc(C)c(C)c1 58573,c1(C(=O)OC)cc(CNC(c2cccc(C(C)C)c2)=O)c(C)o1 58574,C1(Nc2cc(NC(c3cnncc3Cl)C)ncn2)CCCCCCC1 58575,c1(NC(CNC2CCC(CCC(=O)NC)CC2)=O)ccc(OC)nc1OC 58576,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58577,C1(C(N2CCC(C(C)(C)NC(C3CC4CC3C4)=O)CC2)=O)CN(CP(C)(C)=O)C1 58578,C#Cc1ccc(C(N2CC3(CCN(C(=O)C(CCC)OCC)C3)C2)=O)cc1C 58579,C(CCC(c1ccccc1)C1CC1)OC.C1(C)CCN1 58580,c1(C(=O)NCCCCC(C)NC(CCC(C)OCC)=O)cnn2ccncc12 58581,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58582,C1(CNC(c2c[nH]c(=O)cn2)=O)CCCCN(C(C2CC3CC3C2)=O)C1 58583,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2ccc(F)o2)=O)C1 58584,C1(C(N2CCOCC(O)C2)=O)(C(=O)NCCSCC(F)(F)F)CC2CCC1CC2 58585,CC(=O)CC(C)(C)CC(=O)NCC(C)N(C(=O)C#CC1CCCOC1)C 58586,CON(Cc1ccccc1)C(=O)C(F)(CNC(C1(c2ccno2)CC1)=O)C(C)C 58587,Cc1ccc(C(=O)NCC2CCC(NC(c3cnns3)=O)C2)cc1C 58588,N1(C(C(CCC)C)=O)CC(C)(C)OCC1CNC(C1CC(S(C)(=O)=O)C1)=O 58589,C1(C2CC2)(C(N(C(CNC(C(C=C)O)=O)Cc2ccccc2)C)=O)CCC1 58590,c1(OC)cccc2ccc(C(N3CCN(C(=O)C(O)P(C)(C)=O)C(C)C3)=O)nc12 58591,Oc1c(CSc2ccc(F)cn2)cc(Br)c2ccccc12 58592,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCCN(C(c3cnc(O)c(C)c3)=O)C2)C1 58593,C1(CN(CCCNC(C2CC2c2cncn2C)=O)CC)CC1C1CCC1 58594,C=CCN=C(NCc1nccc(C(F)(F)F)n1)NCC1CC1C 58595,c1(C(=O)NCCOC2CCN(C(C3CC(C)N(C)C3)=O)C2)c(F)cc(F)cc1Cl 58596,c1(SCCC)c(C)[nH]c(C(=O)NC2CC(NC(=O)C(C)C3CCCC3)C2)c1C 58597,N#CC1(CC(=O)NC2(CNC(c3ccn(C(F)(F)F)n3)=O)CC2)CCCCC1 58598,Cc1cc(NC(=O)C(CN(C)C)NC(=O)CC2CSCCO2)cs1 58599,C1(NC(c2nc(OC(C)C)oc2)=O)CCN(CC2CCCCO2)CC1O 58600,c1(COC(C(c2cn(CC)nc2)(F)F)=O)nc(O)c2ccc(Cl)cc2n1 58601,Cc1noc(C)c1-c1nc(NC(N2C(c3cccs3)CCC2C)=O)co1 58602,C(CCC(=O)NCCOC1CCN(C(=O)C(C)(C)C2CC2)C1)OCC=C 58603,C(C(CSC)CC(=O)N1CCOC(C)(C)C1)NC(C1N(CC)CC1)=O 58604,N1(C(=O)CCC2OCCO2)CC(C2CC2)(C(=O)NCc2ccc(F)cc2)C1 58605,C(=O)(C(CC(C)CCC)N(CC)CC1(C)CC1)NCCCCCC 58606,N1(C(C(=O)CSCc2ccccc2O)=O)CC(F)CC1CO 58607,CC(C(=O)NCC1CC1NC(=O)Cc1c(F)cccc1Br)C1=CCCC1 58608,CCC(CC)CCNC(C1(C(C)NC(c2cc(C)[nH]n2)=O)CC1)=O 58609,c1(C(N2CCN(C(=O)N(c3ccns3)C)CC2)C)cccc(O)c1 58610,C1(C(=O)NCC2CCN(Cc3ccc(I)cc3)C2)CCC2(CCC2)O1 58611,C(C(F)(C(=O)N(c1cccnc1)CC1CC1)C(C)C)NC(C1(CC(C)C)CC1)=O 58612,CC(C)C(C(=O)N1CCC(CF)(NC(=O)C(=O)NC)C1)c1cccc(Cl)c1 58613,c1(CCC(=O)NC(C2CCCN2C(c2ccccc2)=O)C)cn(C)cn1 58614,Cc1cccc(C(=O)NC2CCCCC2N(C)C(C2OCCCO2)=O)c1 58615,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 58616,C1(C(=O)OC)CCC(NC(C2CN(C(c3ncccc3SC)=O)C2)=O)CC1 58617,N1(C(C(CC)NC(C)=O)=O)CC2(CCN(CC(=O)N=CC(C)(C)C)CC2)CC1C 58618,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ccc(O)c(C)c2)=O)CC1C 58619,CN(NC(=O)C(F)c1cscn1)n1nnn1-c1ccccc1 58620,c1(C(N2CC(C)C(F)(F)C2)C)ccc(F)c(F)c1.C12(C(F)(F)F)CC(C1)C(=O)N2 58621,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)cn12 58622,c1(NC(C)=O)ccc(NC(C2CCCN(C(C)C)C2)=O)cc1C 58623,C1(OC)CC2CCC(C1)N2C(=O)CC(CC)NC(=O)C(C)OCC(C)C 58624,C1(C(=O)NC(CC=C)C(=O)NCC2CCCC(=O)N2)CC2(C1)CC21CC1 58625,c1(C(=O)NCCN(C(=O)CC(C)C2CCCCC2)CC)nc(O)[nH]c(=O)n1 58626,CCCCCC(O)C(=O)N1CCC2C(NC(=O)CSCCc3ccccc3)C2C1 58627,c1(CC(=O)NCC(=O)NCC2N(C(C(CC#C)C)=O)CCC2)cccc(F)c1F 58628,n1(CCC)cccc1C(=O)NCC(C)(CO)NC(=O)CC(C)n1cccn1 58629,C1(NC(C2N(C)CC(O)C2)=O)C2CC3C(C2)C13C(N1CC(F)CC1C)=O 58630,C1(CNC(C2(CC)CCOC2)=O)CCCCN(C(=O)CSCc2ccncc2)CC1 58631,c1(CC)ccc(F)c(C(=O)NC2CCC2NC(C2CCOC2C(C)C)=O)c1 58632,C12CC3CN(CCN3C1)C(=O)NC2.c1(C(=O)OCC)c[nH]c(CC)c1COC 58633,CCCCCC(=O)NCC(CC)N(C(=O)C(C1CCCOC1)OC)C 58634,Cc1nc(NC(C)CCC2CCCC2)cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]1 58635,C1(NC(C(CC)C2CCOCC2)=O)(NC(=O)CN2CCCNC2=O)CCCCC1 58636,C1(CNC(C(F)=CCC)=O)CCCC1NC(=O)COCC1(F)CC1 58637,CC1CN(C(=O)CCC(C)(F)F)CCC1NC(c1ncccc1F)=O 58638,C1(C(N2CCOC(c3ccco3)C2)=O)CCCCN1C(c1ccc(Cl)cc1)=O 58639,CC(C)C(CNC(=O)CC(O)CN(C)C)C(=O)NCCCN(C)C 58640,CC1CC(CNC(=O)CCC2CC2)CCN1C(=O)C(C)(C)C#N 58641,C1(C(=O)OCCOC(C)(C)C)CN(CCN(C)C)CCCO1 58642,CCC(CCC1CCC1)N=c1[nH]c(=NCC(C)n2cncn2)c2ncccc2[nH]1 58643,c1(CC(=O)NCC(=C2CN(C(=O)CCc3ccsc3)C2)F)cc(Cl)ccc1Cl 58644,c1(CN2CC(NC(C(C)OCC=C)=O)C(C)C2)cccc([N+](=O)[O-])c1 58645,NC(=O)CC(c1cn(C2CC2)nn1)NC(=O)NC1CCCN1c1ccccc1 58646,N1(C(C(C)(C)CF)=O)CC(CNC(c2ccncn2)=O)C(F)(F)C1 58647,Cc1cccc(CNC(C23CCC(NC(C4CCC(CO)O4)=O)(CC2)C3)=O)c1C 58648,c1(C(N(C(c2cn(CCCC(=O)O)nn2)C)CC)=O)ccoc1-c1ccccc1 58649,N1(C(CCCCN(C)C(C2CCOC2)=O)=O)CCC2(CC1)CC2CO 58650,CC1CCCN(C(=O)C(O)Cc2cn(C3CCN(C)CC3)nn2)C1CO 58651,CC#CCC(C(=O)O)NC(=O)C(C)(C)C1CCO1 58652,c1(C(C)NC(N2C(C=C)CCC2)=O)ccc(C#N)cc1F 58653,CC1CCC(C(=O)NCC2(NC(=O)CCCNC(=O)C(C)(C)C)CCC2)C1 58654,C1(C(N(C2CCN(Cc3ccnn3C)C2)C)=O)CC(=O)N(c2ccccc2)C1 58655,Cc1cnc2c(C(=O)N(CCC(C)NC(=O)C(CO)N(C)C)C)cnn2c1 58656,C(C(F)(C(=O)NCC(C)C=O)C(C)C)OC.C12CCC3(CC13)C(=O)N2 58657,C1(CNC(CC2N(CC)CCOC2)=O)CC(NC(=O)C(=O)NC(C)C)C12CCC2 58658,CCCC(C)(C)C(=O)NC(C)CNC(c1nc(C)oc1Oc1ccc(Cl)c(C)c1)=O 58659,N1(C(c2nc(CC)sc2)=O)CCCC(O)(CNC(c2ccnc(Cl)c2OC)=O)C1 58660,n1(CC)ncnc1C(=O)NCCOCCNC(=O)C(CC1CC1)OC 58661,c1(C(=O)NCCN(CCCCCC)C(=O)CCc2cn(C)nn2)scnc1C#N 58662,O=C(C1=COCCC1)NC1CCN(C(c2cnn(CCO)c2)=O)C(C2CC2)C1 58663,c1(C(=O)NCCC(C(C)C)NC(=O)C(C)(O)C(F)(F)F)csc2c1CCOC2 58664,C12(NC(C3C(=C)C3)=O)CCCC1CN(C(c1cc(-c3csc(C)n3)c[nH]1)=O)C2 58665,c1(C(N2CCC(CC(N3CCCC(=C)C3)=O)C2(C)C)=O)cc2ccccc2o1 58666,Cn1nc(C(=O)NCC2CC2NC(c2cccnc2C(F)F)=O)cc1Cl 58667,c1(C(=O)NCCN(C(c2cc(C)cc(Cl)c2)=O)CC)ccc2nccnc2n1 58668,N1(C(c2nc(CC(C)C)sc2)=O)CCC(n2cc(CNC(=O)CO)nn2)CC1 58669,C1(NC(=O)CC2CC(O)C23CCC3)CC2CN(C(c3cc(F)cc(F)c3)=O)CC12 58670,N1(C(CCS(C)=O)=O)CC2CC(C)CC(C1)N2C(=O)CCc1ccc(Cl)s1 58671,C1(NC(C(C)c2ccco2)=O)(CNC(=O)C=Cc2ccc[nH]2)CCCCC1C 58672,c1(C(=O)NC2CCC(N(C(C(C)NC(CC)=O)=O)C)CC2)cc([N+](=O)[O-])ccn1 58673,CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCCc2cccc(Cl)c2)[nH]1 58674,c1(C(=O)NCC2(OC)CN(C(C(CC=CC)CC)=O)C2)cc(C)cc(C)c1O 58675,c1(C(=O)NCC(CC)(C)NC(C2CCCC(F)C2)=O)c(OC)cccc1O 58676,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C(C)(C)C)c(C)cc(C)nc1O 58677,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 58678,c1(NC(c2ccccn2)CC)ccc(S(=O)(=O)NC2COCC2O)cc1Br 58679,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CNC(C1C(OC)CC1)=O)(C)O 58680,C12(C(=O)NC(C3CN(C(=O)CN(C)S(N)(=O)=O)C3)C)CC(C(F)F)(C1)C2 58681,CCC(CC)C(C)C(=O)N1CCC(CNC(=O)CCOCC2CCCO2)(CC)C1 58682,C(CCN(C(=O)CN1CCCOC1=O)C)(C(C)(C)C)NC(CCCNC(C)=O)=O 58683,C1(C(=O)NC(CCCC)C)CC2CCC1N2C(c1ccn(CC)n1)=O 58684,C1(C(N(C)CC2CCS(=O)(=O)C2)=O)CC2(CCC2=O)C1 58685,C(=O)(CCCC=O)NC(CCCCNC(CSCCCC)=O)C.c1(C)ccccc1 58686,Cc1ncc(C(N2C(C(=O)N(CCCCN(C)C)C)CCC23CC3)=O)c(C)n1 58687,C1(CN2CCC(C(N3CCC(c4ncc(C)cn4)CC3)=O)CC2)CC2CCC1CC2 58688,C(=O)(C1=CCN(C(C2CCCN(C3CC3)C2)=O)C1)N1CCC(=C)CC1 58689,Cc1ncsc1C=CC(N1CCC(CNC(C2CCC(=O)N2)=O)CC1)=O 58690,c1(C(N2CC(N(C(CC3ON=C(C)C3)=O)C)C(O)C2)=O)cn2ccncc2n1 58691,C(C)(CCC(=O)NC1CCN(C(=O)C(F)(F)c2cnn(C)c2)C1)SC 58692,C(=O)(CCCCN(C)C)N(C)CCOCCNC(c1ccc(F)o1)=O 58693,C1(C(N(CCCCC(C)C)C)=O)CCN(C(C2CCN(C)C2C)=O)CC1C 58694,CCC(CNC(C1CN(C(C)=O)CCO1)=O)(CC)C(=O)NCC(O)COC 58695,C1(COC)(N(C(=O)CCN2CCCCC2)C2CCC2)CCN(C(C2CCOC2)=O)C1 58696,C1(C2CCCCC2)(NC(c2ccc(C)cc2Cl)c2n(CC=C)nnn2)CC1 58697,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCC1CC1)C2 58698,CCC(C)C(C)C(=O)NCCC1CCCN(Cc2c(C)nn(C)c2C)C1 58699,c1(C(=O)NCCCNC(c2ccc(COC)[nH]2)=O)cc(N)c(O)c(F)c1 58700,N1(C(C2CCN(C(CC)=O)C2)=O)CC2(CCC2NC(=O)CCc2ccc(Cl)s2)C1 58701,C1(C(=O)NCCNC(CC)=O)CCN(C(C2(F)CCCCC2)=O)CC1C 58702,C(c1cccc(F)c1F)=CC(=O)NCC1CCCC(NC(c2c(C)scc2)=O)C1 58703,c1(C(N2CCC(N(C(=O)C(F)C3CCC3)CCC)CC2)=O)ccc(=O)n(CC)n1 58704,CCS(=O)(=O)c1ccc(CC(=O)NC2CC3(C2)CN(C(C2CC2OC)=O)C3)cc1 58705,c1(C(n2ccnc2COC)C(=O)NCCCC(=O)OC)c(C)cccc1Br.C1(C)CC1 58706,C1(C)(NC(C(n2cc(Br)cn2)C)=O)CCCN(C(C2(O)COC2)=O)C1 58707,c1(NC2CCC(C#C)C2)ccc2c(c1)CCC(=O)N2 58708,C(=O)(C(C)CS(=O)(=O)c1ccc(F)cc1)NC1CN(C(C(C)C)=O)C2C1C2 58709,C1(C)(C(N2CCC(CN(C)C(c3ccon3)=O)C2)=O)CCCN1C 58710,CC(C)CC(O)CNC(=O)C(C1(O)CCC1)NC(C1CCOC1(C)C)=O 58711,n1(CC(=O)N(C)CC2CCN(C(CSCC#C)=O)C2)c(O)nc2ccccc12 58712,CC(CC(F)(F)F)C(=O)NC(CCF)C(=O)NCC1CCC(=O)O1 58713,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)CSc2nc[nH]n2)cccc(Cl)c1 58714,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC(NC(=O)CC3CCOC3)C2C1 58715,C1(OCC(=O)N(CCCNC(=O)COC2CCSC2)C)CCCOC1 58716,C12(C(=O)NC(C)C(=O)N(C)C)CC(CCO1)N(C(=O)C(C)SCCF)C2 58717,C1(C(=O)NC2(C)CN(C(c3cncc(C(F)(F)F)n3)=O)C2)CCC2CC1C2(C)C 58718,C1(CN2C(C)C2=O)(CO)CC12CCN(C(=O)CC1CC(=O)C1)CC2.C#CCOC 58719,Cc1nc(CC(N2CCSCC2C(=O)O)=O)ccc1Br 58720,N1(C(C2C(=C)CC2)=O)CCC2(CCC2CNC(=O)C2=CCOCC2)CC1 58721,C=CCC(C(=O)NC1CCCCN(C(=O)C(C)(C)C(=O)OCC)CC1)C(C)C 58722,c1(C(N2CCC(CN(C(c3n(C=C)ncc3)=O)C)C2)=O)ccc2ncn(C)c2n1 58723,CC1CCCc2cc(C(=O)NCCCN(C)C(C3CCC4(CCC4)OC3)=O)nn21 58724,N1(C(C(C)CN(C)C)=O)Cc2nccn2CC(NC(c2cnccc2Cl)=O)C1 58725,N1(C(c2ccc(C)cc2C)C(=O)NCCCOC)CC(C)OC2CCCCC12 58726,Cc1n[nH]c(C)c1C(=O)N(CCCN(C)C(c1coc(-c2cccs2)n1)=O)C 58727,C1(CC(C)NC(C=CCOC)=O)CCN(C(C2COCC2(C)C)=O)CC1 58728,c1(CC(N2CC(NC(c3cn(C)c(O)n3)=O)C(F)C2)=O)coc2ccc(F)cc12 58729,c1(C(N(C)CC2CN(C(c3csnn3)=O)C2)=O)cc([N+](=O)[O-])ncc1Br 58730,c1(OC)ccc(Cl)c(CN2CCCC(C(=O)Nc3ncc(F)cc3Br)C2)c1 58731,c1(C(=O)NC2CCN(C(C3(C#N)CC4CC4C3)=O)CC2)ccnc2ccccc12 58732,C1(C(=O)NCC2CCCN2C(C2CC23CC3)=O)CC12CCOC2 58733,C1(N(CCC(=O)NCCCCNC(=O)C2CC2)C)C2CC3C(C2)C13 58734,C(C(C)(CCO)NC(c1cn(CCNC(C2C=CCC2)=O)cn1)=O)OC 58735,CCCCCC=CCC(=O)NCCCNC(c1[nH]ccc1CC1CC(C)C1)=O 58736,N1(C(C(C(C)NC(C(=O)NCC)=O)C)=O)CC2CCC(C1)O2 58737,N1(CC(N2C(CC(=O)NCc3ccncc3Cl)CC(F)C2)=O)CCS(=O)(=O)CC1 58738,N1(C(CCOC(C)=O)=O)CC=CC1C(=O)N(C)CCN1CCCCC1 58739,N1(C(c2ccccc2)CN(CCC(C)O)C)C(=O)C=CC1=O 58740,N1(C(c2c(C)noc2)=O)CC2(CCC(CNC(C3CC4CCC(C3)C4O)=O)O2)C1 58741,C1(C)(C(N(CCCO)C)=O)CC12CCN(CCC1CC3CCC1O3)CC2 58742,CC1CN(C(c2cc(O)cs2)=O)CC(C)CN1C(=O)CC1CCN(C)C1=O 58743,CCCC(CCC)CC(=O)NCC(O)CNC(c1sccc1CC)=O 58744,c1(CN(C(C2(OCC)CC(N3CC4C(COC)C4C3)C2)=O)C)cc(Cl)c(Cl)n1C 58745,CN1CCC(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 58746,c1(OC)cc(F)c(C(=O)NCc2oc(CO)nc2C)c(F)c1 58747,CC1(CNC(=O)C=CC(=O)N(C)C)CCCN(C(=O)CCN2CCCC2)C1 58748,C(N=c1[nH]c(=NC2CCN(COCC3CC3)C2)c2sccc2[nH]1)c1c(C)nns1 58749,O=C(C#CCNC(C1CCC(=O)O1)=O)NCC1CCOC1 58750,S(=O)(=O)(c1ccc(=NCCn2ccc(Br)n2)[nH]c1)NCC(C1CCOCC1)(C)C 58751,C(=O)(C1CCc2cccnc21)Nc1cccc(NC(=O)C2=COCCO2)c1 58752,c1(CN(C(C(CC)Sc2ccccc2)=O)CC2CCCCC2)cn(C)cc1C 58753,c1(CNC(c2ccc(NC)s2)=O)ccc(C(N2CC(CN(C)C)C2)=O)cc1 58754,C1(NC(c2cc3ccsc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 58755,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CC(CCNC(C(C(C=C)C)C)=O)C1 58756,c1(C(=O)NC2CC(NC(=O)COc3ccc(F)cc3)C2)ccc(Br)c(Cl)n1 58757,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CCNC(c2ccc(C#C)o2)=O)C1 58758,C1(CNC(C#CC(C)(C)C)=O)C2CCC1CN(C(=O)CCN1CCCCC1=O)C2 58759,C1(C(=O)NCC(C)CNC(c2cc(CO)[nH]n2)=O)CCN(C)C(=O)C1 58760,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 58761,c1(C(c2ccc(Oc3nnnn3C3COC3)nc2)NC2C(C)(C)C2)ncc(Cl)cc1Cl 58762,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 58763,O=C1CC(NCc2ccc(-c3cc[nH]n3)cc2)CCN1 58764,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)C(C3(O)CCCC3)F)C2)c1Cl 58765,C#Cc1cnc(N2CC3C(C(=O)NCc4nc(C(C)(F)F)cs4)C3C2)nc1 58766,c1(CC(=O)NCC(CN(C)C(c2cn(CCO)nn2)=O)O)csc(C2CCCC2)n1 58767,c1(N2CCC(NC(C(C3CC3)OCC)=O)(CF)C2)ncc(Cl)c(O)n1 58768,N1(C(CSC)=O)CCC2(NC(c3cncc(C4CC4)c3)=O)CC2C1 58769,C1(CNC(c2c(C)nn(CCO)c2)=O)C(C)CCCN1C(C12CC1C2)=O 58770,c1(C(=O)NC2CCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)nccc(Cl)c1O 58771,C1(NC(c2cc(C)sn2)=O)Cc2ccccc2N(C(c2oncc2C)=O)C1 58772,c1(C(C)=O)ccc(C(N2CCCC(NC(C3CCC4(CCC4)O3)=O)C2)=O)c(F)c1 58773,N#CC1CCN(C(C2(NC(c3conc3C3CC3)=O)CCOCC2)=O)C1 58774,n1(C(C)C)nnnc1C(c1cncs1)NC(c1noc(C(F)(F)F)n1)C 58775,C1(C#N)(C(N(CCNC(CCSCCCC)=O)C)=O)CC2CCC1C2 58776,C1(CC(=O)OC)CN(C(=O)Cc2cnn(C(C)(C)C)c2)CC12CC2 58777,C1(N(C(c2cccc(OCC)c2)C(=O)NCC)C2CC2)CCS(=O)(=O)C1 58778,N1(C(C=CCC)=O)CCN(C(=O)CC(C)(C)c2ccccc2)C(c2nccn2C)C1 58779,CC1(C)CCCC(C(=O)NC(C2CCCN2C(=O)CN=S(C)(C)=O)(C)C)O1 58780,N1(C(c2ccn(C(C)C)n2)=O)CC(C)CN(C(=O)CS(=O)(=O)C(C)(C)C)C(C)C1 58781,c1(CNC(C(COC)(F)F)=O)nnc2n1CCN(C(=O)CC(C)(C)C(C)(F)F)C2 58782,C1(NC(CC(=O)OCC)=O)CC(NC(c2cnc(COC)nc2C)=O)C12CCC2 58783,N#CC1(C(=O)NCC2CC(NC(=O)CCF)C2)CCCO1 58784,C1(NC(C(C2(OC)CCCC2)(F)F)=O)CS(=O)(=O)C2CN(C(=O)C(F)OC)CC12 58785,C#CC1(OCC(=O)NCCC(C)(C)CNC(=O)CC2CC23CC3)COC1 58786,c1(CC(N2C(Cn3cc(CCN(C)CC)nn3)C=CC2)=O)cc(F)ncc1Cl 58787,C1(NC(c2c(C)[nH]cc2)=O)CCCCC1N(C(=O)Cc1ccc(Cl)s1)C 58788,c1(NCC)ncc(C(=O)N(CC(C)NC(=O)CC2(C)CCS(=O)(=O)N2)C)cc1Cl 58789,n1(COC)nccc1C(=O)NCC1CC(NC(=O)CNC(N)=O)C1 58790,C12(OC(=O)OC(C)(C)C)CC(COC3(OCCN(C)C)CC3)(CO1)C2 58791,S(=O)(=O)(c1ccc(NC2CCCC3CCCCC23)c(C#N)c1)N(C)CCF 58792,c1(CC)oc(N2CCOC(CC(=O)OC(C)(C)C)C2)nc1Br 58793,N1(Cc2c(OC)nsc2)CCN(CC(=O)Nc2ccc(C)o2)CC1 58794,n1(CCC(=O)NCC2(C(=O)NCC(F)(F)F)CCOC2)cnc2ccccc12 58795,c1(NC(Cc2c(C)nccc2)=O)cc(Br)c(F)cc1C#N 58796,C(C(CC(C)C)C(=O)N)NC(CCCCOC)=O.C1(C(N)=O)CCC(O)CC1 58797,C(=O)(C(O)CNC(=O)Cn1cc(C)cn1)NCC(CC)N1CCCC1 58798,N12CCC(C)C(C1)NC(=O)C1(CCSC1)C2=O.c1(OC)ccc(SC(F)F)cn1 58799,CCCCCCC(C)C(=O)N1C2CCC1(CNC(=O)C(=O)NCC(F)F)CC2 58800,c1(-n2c(-c3ccn(C4CC4)n3)nc(C(C)SC)n2)ccc(Cl)c(Br)c1.C1CC1 58801,N1(C(CC2C(C)C2)=O)CC2CC2(NC(c2ccc(OCC3CC3)nc2)=O)C1 58802,C(C(CC1CC1)C(=O)NC1CCC(O)C1)NC(C1CCCN1C1CC1)=O 58803,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 58804,C12(C(=O)NCCOC)CCC(n3c(-c4cc(C)ccn4)nnc3C)(CC1)C2 58805,CCS(=O)CC(=O)NCC(C)CN(C(=O)CC(C)(C)SC)C 58806,CC1CN(C(=O)Cc2ccnn2C2CCCCC2)CC1NC(C1CCNC1=O)=O 58807,c1(OC(C)C)cc(-c2ccc(NC(C3COCCO3)=O)nn2)cc(C#N)c1 58808,C(CC1C(=O)N1)SC.C1(C(=O)NCC2CC2)CC(OC)C1.C(CCO)S 58809,S(=O)(=O)(C1CCC2(CCC2)CC1)NC12C(NC(=O)OC(C)(C)C)C3CC1C2C3 58810,c1(C(=O)NCC(C)NC(=O)CN2CCc3sccc3C2)nnn2c1CCCC2 58811,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)CC)[nH]1)C1CCCC(C)C1 58812,S(=O)(=O)(CCC(F)(F)F)N1CC(C(=O)Nc2cnc(Cl)c(F)c2)C(O)CC1 58813,N1(c2cccc3ccc(OC)nc32)Cc2ccccc2OC2(CCOC2)C1 58814,c1(C(=O)NCC(CNC(CC(C=C)C)=O)F)cc(C)ccc1OCC 58815,c1(CCC)cc(C(=O)NC23CCN(C2)C3)c(C)o1.c1(C(=O)OC)c(C)coc1C 58816,c1(C(=O)NCC2CCCCCN2C(c2cscc2Cl)=O)ccc2cnoc2c1 58817,C(=O)(C(CC(C)C)ONC(=O)C1(CCOC)CC1)NC(CCCC=C)C 58818,C(=O)(CCCS(C)(=O)=O)NC1CCCC(NC(CCCCOC)=O)C1 58819,c1(C(N2C(C)CCC(NC(COCCCC#C)=O)C2)=O)ccc(C)c(C)c1O 58820,c1(C(=O)NC2(CC=C)CN(C(=O)CC3CSC3)C2)cc2ccc(C)cc2[nH]1 58821,C(C(C(=O)NCC(C)(C)CO)NC(=O)CC1CCOC1)OCC 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58839,c1(C(=O)NC(c2ccccc2F)CNC(CC)=O)c(C)nn(CC#N)c1C 58840,C(=O)(C1=NOCC1)NC(c1ccccc1)CNC(C(Cc1ccccc1)OC)=O 58841,C(c1ccc(Cl)c(F)c1)=CC(N1CCC(NC(C(CSC)(C)C)=O)C(C)C1)=O 58842,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 58843,Cc1cc(C(N2CC(NC(c3cnc(C)n3C)=O)C(C)C2)=O)c2c(C)noc2n1 58844,C1(CNC(CCC=C)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CC1OC 58845,Cn1c(O)nc2cc(C(N3CCC(CCNC(=O)CCCC#N)C3)=O)ccc12 58846,Cc1ccc(C)n1CC(N1CCCCC1CC(=O)NOCCO)=O 58847,C1(C)(CC)CCC(C(=O)NNC(=O)c2cnoc2)O1 58848,c1(N2CCC(C)(F)C2)nc(=NCCNC(C2CCC2)=O)[nH]c2c1COCC2 58849,c1(C(=O)NC2C(NC(CN(C(=O)OC)C)=O)C2)cc2n(n1)CCO2 58850,C(=O)(C(c1ccccc1)=C(C)C)NC1CC2(N(C(C(COC)OC)=O)C2)C1 58851,c1(CNc2snc(-c3ccc(C)o3)n2)ccc(F)cc1C#N 58852,C1(C(=O)OC)CC(C)N1C(=O)C(=O)C1(CC(=O)Oc2ncn(C)n2)CC1 58853,CC(CC(N)=O)C(=O)NC1CCCC1NC(c1cc(N(C)C)ccn1)=O 58854,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 58855,c1(CN2C(CC#C)CCCC2)c(C)cccc1C.C12CCCCN1C2=O 58856,N12CCN(CC1)C(=O)C1(CC1)C2.C(CCC(=O)NCC1CC(C(C)(C)C)C1)SC 58857,C(=O)(C(F)C(C)(C)O)NC(CN(C(=O)Cn1ncnn1)C)(C)C 58858,c1(CC)nccnc1C(=O)NCC(C)(C)CNC(c1cc(Cl)cnn1)=O 58859,S(=O)(=O)(c1ccccc1C1CC(F)(F)C2CCCN12)NC1CC(C)CC(CO)C1 58860,c1(C(N2CC(CN(C)C(c3cnco3)=O)C3(C2)CC3)=O)ccc2c(n1)CCCC2 58861,c1(C(N2CCC(C(=O)Nc3c(C(C)=O)cccn3)CC2)=O)c(C)cc(Br)cc1C 58862,c1(C(C(C)C)C(=O)N(C2CCCCC2N(C)C)C)ccc(Br)cc1F 58863,c1(C(N2CC(NC(c3ccco3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 58864,c1(CCCCN(C(C)C)C(C2CCS2(=O)=O)=O)cn(CCCC(=O)O)nn1 58865,C(=O)(CC1OCCc2ccccc21)NC1CC(N(C(C=CC(CC)C)=O)CC)C1 58866,c1(C(=O)NCC2N(C(C(C)O)=O)CC2)cc2cccc(Br)c2o1 58867,C(C#Cc1ncccn1)N1CCC(NC(C(c2cccnc2)C)=O)C1 58868,C(CCC1CCC1)(C(=O)NC(c1nccn1C)CC)NC(CC=CC)=O 58869,CCC(C)CC(C(=O)OC)NC(=NCC12CC(C)(C1)OC21CCC1)NC(C)C 58870,C=C(C)CC(C(=O)N1CCC(CCCC)C1)NC(=O)C(C1CCOCC1)F 58871,c1(CC(=O)N(CCN(C(=O)CN2CCCC2CO)CC)CC)nonc1C 58872,N1(C(C2CN(CC(F)(F)F)C2)=O)CCCC(CC(=O)Nc2cc(C)no2)C1 58873,C1(NC(C(=O)NCC2CC2)=O)CCCCN(C(c2sccc2C2CC2)=O)C1 58874,C1(NC(c2cn(CCC)nc2)c2nnnn2C(C)C(=O)OC)CCC(=O)N(C)C1 58875,C(=O)(C1=NN(C)C(=O)CC1)N1CC(CCCCNC(c2c(C)nns2)=O)C1 58876,N1(C(c2n(C)ccn2)=O)CCC(NC(c2cc(CCO)on2)=O)C(CO)C1 58877,c12n[nH]c3c1CN(C3)CC(=O)N2.C1(C(=O)OC)CCN2CCOCC12 58878,N1(C(c2coc(COC)n2)C(=O)NCCC)CCCN(C(C)CC)CC1 58879,c1(C(=O)NCC(=O)NCCCNC(c2c(CC)noc2C)=O)ccc(C)cc1O 58880,N1(C(CCNC(=O)OC)=O)CCC2(C1)CN(C(C1CC(CC(C)C)C1)=O)CCO2 58881,N1(C(C2N(C(CCN=[N+]=[N-])=O)CCCC2)=O)CC(C2CCCOC2)C1 58882,Cc1oc(C(C)(C)C)cc1C(N1CC(O)(CN(C)C(C2CCC(C)(C)C2)=O)C1)=O 58883,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C12CC(C1)C2)=O 58884,C12(CC(=O)N(C3CCN(CC)C3)CCC)CCC1CN(C(C1CC(F)(F)C1)=O)C2 58885,Cc1ccc(C(=O)C2CC2)c(O)c1.c12cccc(n1)C(=O)NC2.C1(C2CC2)CN1 58886,Cc1nc(C(=O)NC2CC(CCNC(=O)C(O)CC(C)C)C2)cc(O)n1 58887,N1(C(c2c(C)nc[nH]2)=O)CCC2(CCCN(C(C3CCC4CC34)=O)C2)C1 58888,N1(C(CN(C(=O)COCC2CC2)CC#C)=O)CCSCC1C(=O)NC 58889,N1(C(CC2CC(=C)C2)=O)CC(CNC(c2[nH]nnc2C(=O)OC)=O)C2(CC2)C1 58890,c1(C(N(CC(C)O)CC)=O)cn(CCNC(C2OCCO2)=O)nn1 58891,C(C(C)(C)C(=O)NCCCCC1CC1C)NC(Cc1cn(CC)nn1)=O 58892,C(C)(CCC(C)(C)C)NC(c1nn(C)cc1OC)c1n(CCCSC)nnn1 58893,C1(C(=O)OC)CCC2(CC2)N(CC2CCC3(CCC3)O2)C1 58894,N1(C(c2c(C)nns2)=O)CC(C)C(NC(c2cncn(C)c2=O)=O)C(C)C1 58895,CC1=C(C(=O)NCC(F)(F)F)C(c2cnc(C)nc2CO)NC(=O)N1C 58896,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1 58897,c1(N(C(=O)C=Cc2ccc(C)cc2)C(C)C)cc(Br)c(N2CCOCC2)c(Br)c1 58898,C=C1Cn2c(C(=O)NCC3CN(C(C4(C(=O)NC)CC4)=O)CCN3C)nnc2S1 58899,C(=O)(C1=CC2C=CC(C1)C2)NCc1ccc(C)cc1C.C=CCCC1C(=O)N1 58900,Cc1nc(C(C)(C)C)c(C(=O)NCC2(NC(=O)CC3(O)CCCOC3)CCC2)s1 58901,C1(COC)(NC(C2CC3C(C2)C3(C)C)=O)CCCN(C(C2CN(C)C2)=O)C1 58902,c1(SC)ncc(C(=O)NCC2CCCN2C(c2cnn(-c3ccccn3)c2)=O)s1 58903,N1(C(c2c(OCC)nccc2)=O)CCC2CN(Cc3ccc4nn[nH]c4c3)CC12 58904,c1(C(=O)NCC2(F)CC(NC(C(C)OCCCC)=O)C2)ccc(C)c(S(C)(=O)=O)c1 58905,N1(C(CC(C)N(C)C)=O)CCCCC1C(=O)NCC1COCCO1 58906,C1(CNC(CC)=O)CN(C(=O)Cn2cnc(C(F)(F)F)n2)CCC1(C)C 58907,C1(NC(=O)CNC(C2CC(F)(F)C2)=O)C2CCN(C(=O)C(F)(F)F)CCC12 58908,C=C(Cl)CCCN=c1[nH]c(=NC(C)c2ccnc(C)n2)[nH]c2c1COCC2 58909,c1(N(C)C(C2(CNC(=O)CC3CCOCC3)CC2)=O)ccc(Cl)cc1N 58910,N1(C(c2n(CC)nnc2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 58911,N(C(=NCC1CCN(C)C1=O)NC1(C)CCC1)CC1(OC)CCCOC1.C(C)(C)S 58912,C1(NC(CC2CCC(=O)NC2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 58913,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(C)CC(N)=O 58914,N1(C(c2cc(C)nn2C)=O)CCC2(CO)CN(C(=O)CCc3cn[nH]c3)CC2C1 58915,C1(C(=O)NCC(C)N(C(c2cc(C)c(C)nn2)=O)CC)CCc2ncsc2C1 58916,c1(C(N2CCC(F)(F)CC2)=O)cnc2c(-c3ccc4[nH]ccc4n3)cccc2c1 58917,C1(=CC(=O)NCC(CC)NC(c2ccc(C(=O)C3CC3)[nH]2)=O)CC2CCC(C1)N2C 58918,C1(NC(c2nc(C)[nH]n2)=O)CC2CCC1CN(C(=O)C(C)CSC(F)(F)F)C2 58919,C(CCCCCNC(=O)Cc1ccccc1Cl)N(C(=O)C(c1ccccc1)O)C 58920,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(F)(Cl)c1ccccc1)C2 58921,c1(OC)cc(-c2ccc(F)cn2)c(OC)cc1CN(C1CC1(C)C)C 58922,C1(NC(C2C(C(=O)OC)CC2)=O)(CNC(=O)Cc2nc(C3CC3)cs2)CC1(C)C 58923,C#Cc1cn(C)nc1C(N1CCC(CNC(=O)Cn2cccnc2=O)C(OC)C1)=O 58924,C(=O)(C1=CCCOCC1)N1C(C)CC(CNc2nc(C(=O)OC)c(Cl)cn2)C1 58925,CC1CCN(C(c2ccnn2CC(F)F)=O)CC1NC(c1cn(C)c(=O)n1C)=O 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58944,Cc1nc(C(=O)NCCCN(C(C2CNC(=O)N2)=O)C2CC2)cc(O)n1 58945,c1(CC(=O)N(C(C)C(=O)NC(C)Cn2cccc2)C)cccc([N+](=O)[O-])c1 58946,c1(C(=O)NC(C(=O)NCC2CC(F)(CNC(=O)OC)C2)C)cc2sc(F)cc2[nH]1 58947,Cc1nn(C)c(C(=O)NC2CS(=O)(=O)CC2NC(c2ccc(Cl)s2)=O)c1Cl 58948,c1(C(=O)NCC2C(F)(F)CCN(C(CC#N)=O)C2)ccc2cccnc2c1 58949,N1(C(CC(C)C2CC2)=O)CCCC(NC(c2ccc(N)c(N)n2)=O)CC1 58950,c1(-c2cnc(NC(Cc3cccc(OC)c3Cl)=O)c(C)c2)cnc(C#N)c(F)c1 58951,C1(N(C(c2cn(CC(N)=O)nn2)C)C)CCC(O)(c2ccccc2)CC1 58952,C(CC(=O)N1CC2(CC(O)C2)C1)(C(F)(F)F)NC(C(C)SCC)=O 58953,C1(NC(c2n(C(CC)(C)C)nnn2)Cc2cnc(C)o2)CCC(C2CC2)C1.C(=O)OC 58954,C12(NC(=O)Nc3cn(C=C)nc3)CCC(C(=O)NC)(CC1)CC2 58955,N12CC(C)(C)C1C2=O.n1(OCC)ccnc1-c1cn(C2CCC(CC)C2)nn1 58956,C12(CNC(C=CC)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C(C)CSC)C1)O2 58957,C(=O)(C=C1SCC(=O)N1C)N(C)CCC1CCCCN1C(C1(CC2CC2)CC1)=O 58958,C1(C(=O)NCc2ncoc2CCNC(C2CS(=O)(=O)C2)=O)(COC)CCCCC1 58959,C12(C(=O)NCCOCCCSC)CCC(CN(C(=O)CCCNC(C)=O)C1)C2 58960,CC1CCc2c(C(N3CC(C)(C)CC3CNC(=O)CC3CC34CC4)=O)csc2C1 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58978,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CO)C2)=O)C1 58979,C1(CC(N2CCN(C(CNC3C(C(N)=O)CCC3)=O)CC2)=O)CCCC(C#N)C1 58980,O(P(C)(=O)CNC(C1CC(F)CN1C(=O)CC1CCCOCC1)=O)CC 58981,CCCCCCCCOCC(=O)N(c1cc(N)nc(Cl)c1)CC(=O)OC 58982,N1(C(c2c(SC)cccc2)=O)CCCN(CCNC(c2cnoc2C(C)C)=O)CC1 58983,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 58984,C1(NC(COCC(=C)C)=O)CN(C(c2nncn2C2CC2)=O)CC1C(F)F 58985,N1(C(C(=O)NCCOC)C2COC2)CCCC2(CCCOC2)C1 58986,c1(C(=O)NC(CNC(C(CC)(CC)OC)=O)CCOC)cnc2[nH]nnc2c1 58987,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 58988,C1(C(=O)Nc2cn(CC)nc2)CSCCN1C(c1cnc(C)[nH]1)=O 58989,C(=O)(C(C(C)(C)C)NC(=O)NC(C)(C)C)N1CCC(NC(c2c(C)cno2)=O)C1 58990,CCC(C(=O)NC1CC1)C(=O)NC1CC2(C1)CN(C(c1ccc(OC)cn1)=O)C2 58991,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 58992,c1(C(=O)NC2CCC(N(C)C(c3ccns3)=O)C2)ccn2ccnc2c1 58993,C1(CN(C(C2CC(C(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 58994,C(N=c1cc(CC2CCCCO2)nc[nH]1)C1(NC(C(CC)OC)=O)CCCCC1C 58995,C1(C(=O)NC2C(NC(c3cnc(C4CC4)s3)=O)CCCC2)CS(=O)(=O)CCO1 58996,N1(C(C=CC)=O)CC(O)CC1C(N1CCCC1C1(N(C)C)CC1)=O 58997,c1(CC)ccccc1C(CNC(C12CCC1C2)=O)NC(C1CCCCO1)=O 58998,N1(C(c2cnc(CC)o2)=O)CCC(CC)C1CNC(c1ccsn1)=O 58999,C1(Br)(C(=O)NC(C)CN(C(=O)CCN(C)C(c2ccco2)=O)C)CC1(F)F 59000,N1(C(c2nn(C)c(Cl)c2)=O)CC2CC(C1)C(CO)C2NC(c1cccc(F)c1)=O 59001,N1(C(=O)NCCCC)CCC(C)(NCC(C(C)C)N2CCCC2)CC1=O 59002,c1(C(CC)CN(C(C)C(=O)O)CCc2nc[nH]n2)ccccc1 59003,CCCC(C)C(=O)NC1(C)CN(C(C2COCCN2CC(F)(F)F)=O)C1 59004,CC1(NC(C2CCCN(C(=O)C3CC3)C2)=O)CCN(C(=O)C(C)(C)CF)C1 59005,N1(C(C(CC)F)=O)CCC(N(C)C(c2ccn(C3CCC3)n2)=O)C2(CC2)C1 59006,CC(C)CC(O)C(=O)NC1COCCN(C(=O)C(C)(C)C2CCCCC2)C1 59007,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CN1C(c1nc[nH]c2nccc1-2)=O 59008,C(CC(C)CCNC(c1cc(C(N)=O)no1)=O)NC(CCCOCC)=O 59009,c1(C(=O)NC2CN(Cc3c(O)ccc(F)c3F)CC2F)cc(F)cc2nc[nH]c12 59010,C(=O)(C(CCOCCO)NC(=O)C(F)C(C)C)NCC(=O)NCCOC 59011,CC1(CNC(C2CCOC2CNC(=O)COC2CCC2)=O)CC=CCC1 59012,c1(C(=O)NCC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(Cl)nn(C)c1C 59013,C1(NC(C2C(=C)C2)=O)CCN(C(c2cnn(C3CCCCC3)c2C)=O)CC1 59014,C(=O)(C(C)CC(F)F)NCCCCC1CN(C(C(c2cccc(C)c2)F)=O)C1 59015,c1(C(=O)NCC2C(NC(=O)CC34CCCC3C4)C2)cccc([N+](=O)[O-])c1Cl 59016,C(=O)(C#CC(C)(C)CNC(C12CSCC1C2)=O)NCCC(=O)OC(C)(C)C 59017,C(=O)(C(C)(C)CC#N)N1CCC(N(C(=O)CC2C=NN(C)C2=O)CCC)C1 59018,N1(Cc2c(C(N(C)C)=O)ccc(C(F)(F)F)c2)CCOC2(CCS(=N)(=O)CC2)C1 59019,C1(CC(=O)N(CCCCCCNC(=O)CSCC(N)=O)C)CCCNC1=O 59020,n1(CC(=O)NC2CC(CNC(=O)C(O)C3CC3)C2)cc(Br)cn1 59021,c1(OC)cc(OC)[nH]c(=NCc2ccc(CNc3cnccn3)cc2)n1 59022,Cc1nc(C2CCOC2)sc1C(=O)NCC1CCN(C(=O)CCC2(C)N=N2)C1 59023,C1(C(=O)Nc2cccc(OC(F)F)c2)(OC)CCN(C2CC3C=CCC23)CC1.OC(F)F 59024,n1(CC2C(C)OCC2)nc(-c2ccnn2C)nc1Cc1csnn1 59025,C1(NC(=O)NCc2nc(C(C)C)on2)CCCC(O)CC1 59026,C12C3CC4C(C3)C14C(=O)N2.n1(CC)nccc1C=CC=O.N1(CC)CCCC1 59027,C1(C(=O)NC(CC)(C)C)CCCN(C2CCc3ccccc32)C1 59028,CC1(CO)CCCN1C(c1ccnc(CNC(=O)CC2COCCO2)c1)=O 59029,C1(N(CC#C)C(C2CC(SC)C2)=O)CCN(C(c2cnn(CCC)c2)=O)CC1 59030,C1(N2CCOC(c3ncc[nH]3)C2)CCCCC(F)(F)C1.CC 59031,C(=O)(CCCCN=[N+]=[N-])N(C1CCC(NC(=O)C#CC2CC2)CC1)C 59032,C1(c2ncc(C(=O)OCCCSCC)s2)CCN(C(C)=O)CC1 59033,C(=O)(C(C)C(C)COC)NCC#CC(=O)NCCC#C 59034,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59035,c1(NC(C2CC(NC(c3cn(CCOC)nc3)=O)CC2O)=O)cc(C)cc(Cl)n1 59036,C(c1cc[nH]n1)=CC(=O)NC(C1CCCN1C(=O)C(O)CC1CCCCC1)(C)C 59037,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)N)C1.C(C(C)CC)N(C)C 59038,N12CCN(CC1)CC(C)NC1CC(C1)CC2=O.C(=O)(C(C)CC=CCC)CC=C 59039,C1(C(=O)NCC(C)NC(c2sc(C)c(Br)n2)=O)CNC(=O)C(C)(C)C1 59040,c1(NC(=O)NC(c2ccnn2C)CC)cn(CC2CC2)nn1 59041,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)Cn3ccnn3)C2C1 59042,C1(NC(CC2C(C)CCO2)=O)CCN(C(C2COC(=O)N2)=O)C12CCCC2 59043,c1(-c2cn(C)nc2)cccc(C(=O)NCC2(O)CN(C(=O)CC3CC3)C2)c1 59044,C(C)(CNC(=O)C(COC)CC)(C(C)C)NC(CC=CC)=O 59045,c1(N2CCCC(CNC(CS(=O)(=O)NC)=O)C2)ccc2ncnn2n1 59046,c1(NC(C2C3(CC(OCC)C3)C2)=O)cccc2oc(C)nc12 59047,CC1(C)CCN(C(C23CC2COC3(C)C)=O)CC1CNC(=O)C(O)CC1CCCC1 59048,C1(C(=O)NC(C(C)C)CO)(CO)CCN(C(c2ccc(C(F)F)o2)=O)C1 59049,c1(C(=O)OCC)ncc(N2CCC(CNC(=O)CC(C)(O)C3CC3)C2)nc1C 59050,C(=O)(C1=CCCN(C(=O)CC2(C)CC2)C1)NC(C)CN1CCC1 59051,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CCC2CC3)C1 59052,CCCCC(C)C(=O)NCCOC1CN(C(c2ccn(C)c(=N)c2)=O)C1 59053,CCCCC(C(=O)NC1CCC(C(N)=O)CC1)NC(=O)CC1CCOC(C)(C)C1 59054,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59055,C1(N(C(C(C)CNC(C23CC(CO)(C2)OC3C)=O)=O)C)CCC(CO)CC1 59056,N1(C(CC=C)=O)CC2CC(NC(=O)C(C)C=Cc3ccccc3)C2C1 59057,c1(C(=O)NC(C)(C)CCNC(N)=O)ccnc(-c2nn[nH]n2)c1 59058,c1(C(=O)NCC2(O)CN(C(C3CC(C)(O)C3)=O)C2)coc2c(F)c(Cl)ccc12 59059,Cc1c(C(N2C3CCC(C3)C2C(=O)N2CC(O)CO2)=O)cccc1Cl 59060,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59061,C1(CC)CN(Cc2ccc(OC(C)(C)C)c(Cl)c2)CCN1S(=O)(=O)CC(F)(F)F 59062,c1(C(N2CCN(C(C3CC3F)=O)CC2c2cn[nH]c2)=O)cc(Cl)ncc1C(F)F 59063,Cc1ncn(C)c1C(=O)NCC(C)(CO)NC(C1CC(F)(CO)C1)=O 59064,n12nccc1[nH]c(=O)[nH]2.c1(C(OC)SCCc2ccn(C3CC3)n2)ccccc1 59065,C1(NC(=O)CCc2ccccn2)CCN(C(c2coc(O)n2)=O)C12CCCC2 59066,c1(OC)cnc(C(N2CCC(N(C(=O)C(c3ccc(F)cc3)F)C)C2)=O)c(F)c1 59067,c1(NC(c2nccc(Cl)c2Cl)c2n(C(C)C)nnn2)cnc2c(Br)c[nH]c2c1 59068,N1(C(C2N(C)CCC2)=O)CCC(NC(c2coc(O)n2)=O)C2(CCC2)C1 59069,C1(C(N(CC(=O)N(CCCF)CC)CC)=O)C2CC(=O)CC12 59070,c1(OC)cc(NC(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)ccc1O 59071,C(=O)(C(CCC(C)C)Nc1nonc1C)NC(C1CN(C(C)=O)C1)=O 59072,C(CNC1CCC1)(CO)(CO)N(C(C(=O)OC(C)(C)C)c1cncs1)C 59073,Cc1cc(C(=O)NC2CCC(C(=O)Nc3ncccc3C(C)O)C2)cc(F)c1 59074,Cc1nc(Cl)[nH]c(=NC2CN(C(C3(C(C)C)CC3)=O)CC23CCC3)c1F 59075,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CCCCC1 59076,N1(C(c2n(C)c(Br)nc2)C(=O)NCC2CCOCC2)CCCN(CCCO)CC1 59077,c1(C(=O)NC2CC(NC(c3sc(C)c(Br)c3)=O)C2)cccc(F)c1N 59078,CN=c1[nH]nc(CC(=O)NCCC2(NC(=O)COC(F)F)CCCC2)s1 59079,N1(C(C2(CCCC)CC2)=O)CCCC(CN(C(=O)C(F)=C(C)C2CC2)CC)C1 59080,C1(NC(c2c(C(C)C)ccs2)=O)CCC(C)(CNC(=O)CCc2csnn2)C1 59081,N1(C(c2cncc(OC)c2)C(=O)OC)CCN(C)CC1C1CC1.N12CC=CC1C2 59082,c1(CC(CNC(C2CN(C(C)=O)C2)=O)CN(C)C(c2cnc[nH]2)=O)ccccc1 59083,c12[nH]c(=NCC3(C)CC3)nc3ncn(c13)NCCOC(CC)CS(=O)(=O)N2.C=CCCCS.CC 59084,c1(CC(=O)N(C(C)CCNC(=O)CCN2CCC2)C)ccc2c(c1)NC(=O)CO2 59085,Cc1cc(CNC(C2CC23CN(C(=O)CC(C)c2ccccc2)C3)=O)ccn1 59086,C1(C(=O)NCCOCCNC(Cc2c(C)ccnc2)=O)C2CCN(CC2)S1(=O)=O 59087,C1(S(=O)(=O)NC(=N)SN2CCCC(CCF)C2)(C(C)C)CC1 59088,CCC(C)(C)C(O)C(=O)NCCC1(OC(C)=O)CN(C(=O)C(F)F)C1 59089,C(C(C)(C)C(=O)NC1C=CCN(C(C2CCCN(C)C2)=O)C1)NC(C)=O 59090,CC1(F)CC(C(=O)NCC(CNC(=O)CSS(C)(=O)=O)CO)C1 59091,N1(C(c2nccc(CC)c2)=O)CC2(CCN(C(=O)C(CO)NC(=O)C(C)C)C2)C1 59092,C1(CC(=O)NC2C(CCC)CN(C(=O)C=C(CC)CC)C2)CC(C)(C)CCO1 59093,c1(CNC(N2CCC(NC(COC)=O)C2)=O)ccc(C(F)(F)F)cc1C 59094,N1(C(c2ccc(Cl)cc2)=O)CCC2C(CCN2C(c2ccoc2)=O)C1 59095,C(=O)(CCCOC1CC(NC(=O)CNC(C2CC2C)=O)C1)OC 59096,C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(c1coc(C2CC2)n1)=O)CC 59097,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59098,c1(NC(C2CCOCC2)(COC)C)ccc(Br)c(Cl)c1.c12nnnn1CCCS2 59099,CC1(C(=O)NC2CCC(NC(C3CN4CCC3CC4)=O)CC2)CCC(O)CC1 59100,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(CO)CC2)C1 59101,c1(C(=O)NC2(C3CCCN3C(=O)C(F)=C3CCCC3)CC2)cc(C(N)=O)c[nH]1 59102,C1(C(N(CCC2CCC3(C(C=C)C3)C(=O)N2)C)=O)CCOC2(CCCCC2)C1 59103,Cc1[nH]nc2cc(NC(C3CC3NC(c3cc(Br)cnc3Br)=O)=O)ccc12 59104,C12(CC(=O)NC(CC=C)CNC(=O)C=Cc3cncs3)CCC(C(F)F)(CO1)C2 59105,C1(C(=O)NCC2(C(C)(C)C)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59106,C1(N(CCC)C(c2cnc(N(C)C)s2)=O)CCN(C(=O)CCOC2COC2)CC1 59107,c1(C(N2CC(O)(C(C)NC(C(CC)(C)C#N)=O)C2)=O)cn2ccc(C)cc2n1 59108,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59109,c1(C(N2C(CNC(C(CC)COC)=O)CC(O)C2)=O)cccc(F)c1C#N 59110,C=CCCCC(C(=O)N(CCCC(=O)NC(C)(C)C)C)c1ccccc1 59111,c1(SC)ccc(CC(=O)NC2CCCC(C(N3CC(N(C)C)C3)=O)C2)cc1 59112,N1(C(=O)Cn2cc(Br)cn2)CC2CN(Cc3ccc(O)cc3Cl)CC12 59113,C1(CC)CN(C(c2cccc(F)c2F)C(=O)NC(C)(C)C)CC(=O)N1 59114,N1(C(CCC2CCC(C)O2)=O)CCC(NC(=O)CCNC(=O)NC2CC2)C(F)C1 59115,CC1(C)CN(C(=O)CCCn2cc(C(=O)O)nn2)C(C)(C)C1O 59116,C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCc2n(CCC)cnc2)CCOCC1 59117,C=CC(C)C(C)C(=O)N1CCCC(CNC(=O)CCc2ccc(OC)cc2)CC1 59118,C1(CC(=O)NC(CCCCC)C2CC2)CNCCS1(=O)=O 59119,C1(C(N(C(C)C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)CC12CC(C)(C)C2 59120,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59121,c1(C(N2CCC(NC(c3ccc(C)cc3Cl)=O)C2)=O)cc(Br)cc2c1OCC2 59122,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59123,Cc1nn(C2CC2)cc1C(N1CC(F)(CNC(=O)C(C2CCCCCC2)O)C1)=O 59124,CCC(C)C(C)C(=O)N1CC=CC(NC(=O)CN2C(=O)CNC2=O)C1 59125,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59126,Cc1cc(C(=O)N(CCNC(=O)C(N2C(C)CCC2C)C)CC2CC2)cc(C)n1 59127,N1(C(CN(CCC)C)=O)CCC2(NC(C3CC3CC)=O)CCCC12 59128,CC1CN2CCN1C(C(N1CC(CNC(=O)CCc3ccc(N)cc3)C1)=O)C2 59129,O=C1NCCn2ncc(C(N3CCC4CN(C(=O)C(F)CC5CCC5)CC34)=O)c21 59130,C1(C(=O)NC2CCC2)(CC)C=CCN1C(=O)CC.C(CO)(CCOC)N 59131,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59132,C1(C(=O)NCC(C)N(C(c2c(OC)nn(C)c2)=O)C)CCc2ccc(F)cc2O1 59133,C1(NC(C(C)OC(F)F)=O)COCC1NC(=O)C(F)(F)OC1CCOCC1 59134,Cc1cc(S(N)(=O)=O)cc(-c2cc(N)c(C#N)c(F)c2)c1C 59135,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CCS1(=O)=O)=O 59136,N1(C(CC2(NC(CN(C(COC)=O)C)=O)CCC2)=O)CC(CO)CC(C)C1 59137,N1(CC(=O)NC(=O)NCC)CCCN(C(C2CCCC(OC)C2)=O)CC1 59138,Cn1nc([N+](=O)[O-])cc1C(=O)NC1CCC(NC(=O)Cc2ccc(F)c(F)c2)C1 59139,c1(C(=O)NCCC(=O)NCc2cnc(CC)o2)cc(SC)oc1C 59140,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC(=O)N(C)C)o1)OC 59141,c1(OC)nccc(N(CC(C)NC(=O)Cc2ccns2)C)n1 59142,c1(C(=O)NC2CCCCCN(C(C(CC)(C)CO)=O)C2)cc(F)c(Cl)c(N)c1Cl 59143,CCC(C)CC(=O)C(=O)NCCc1n[nH]cc1C(N1CCOC(CCF)C1)=O 59144,C1(NC(N(CC(C)C)C)=O)CC2CCC1C(CO)C2 59145,C12(C(=O)NC3C(NC(c4cc(C)n(C(F)F)n4)=O)C3)CCC(C)(C(=O)O1)C2(C)C 59146,C1(CNC(C2(C(O)C(F)(F)F)CC2)=O)CC2(CCC2)CN1Cc1cccc(C)c1 59147,c1(C(N2CCCC(N(C(C(C)=CC)=O)C)C2)=O)ccc2cnnc(O)c2c1 59148,C=CC(C)(C)C(=O)N(C)CC1CCCN1C(C)=O.CC1CCC1N 59149,N1(C(CCCN(C(=O)CCC2CC2(C)C)C)=O)Cc2cccc(O)c2C1 59150,c1(CC(=O)OC)ccc(C(N2CCOCC2CNC(=O)C#CC2CC2)=O)cc1F 59151,C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(CC(CC)C)=O 59152,c1(C(N2CCC(NC(C=C(CC)C)=O)CC2C)=O)c(C)nn2cccnc12 59153,N1(C(c2ccc(-c3ccco3)s2)=O)CCC2CCC(C1)N2c1nnc(C(F)F)s1 59154,c12nc(C)c(s1)C(=O)NC(C)C(C)(C)NC2=O.C(=O)(C(=O)N)NC1CC1.CC 59155,C1(C)(c2cn(CC(=O)OCC)nn2)COCCN1C(C1CC(=O)CO1)=O 59156,N1(C(=O)Cc2ccn(-c3ccccc3)n2)CCC2(CCCN2C(=O)C2CC2)CC1 59157,N1(c2nc(N(C(C)CCCO)C)nc3c2[nH]cc3)CC2CCCCCC2(C#N)C1 59158,c1(C(=O)NC2C(NC(c3cnsn3)=O)C2)ccc(=O)n2c1COCC2 59159,C(=O)(CCS(C)(=O)=O)NC1CC(C)N(C(c2cc(Cl)nnc2Cl)=O)C1 59160,Cc1c(C(N2CCC3(NC(=O)CC4CC4)CCCCC23)=O)sc2cccnc12 59161,Cc1cn2cc(C(N3CCC(C)(C)C3CNC(c3cccc(=O)o3)=O)=O)nc2s1 59162,N1(C(c2ccn(C)n2)=O)Cc2ccc(C(N3CC4CC3CO4)=O)cc2C1 59163,N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(c1ccnc(S)c1)=O 59164,N1(C(CCCC)=O)CC2COCC2(C(N2CCCC(CC#N)C2)=O)C1 59165,C(CCN=C(NCC=C1CCOCC1)NC1CC1)NC(C1(C)CCS(=O)(=O)N1C)=O 59166,N1(C(C(CO)NC(COC(CC)(C)C)=O)=O)CCCN(C2CCC2)CC1 59167,c1(SC)cc(C(=O)NC(C)(C)CN(C)C(c2cccn2C2CC2)=O)c(C)o1 59168,c1(C(N2CCCC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)ccc2nncn2c1 59169,C(=O)(CCCCCF)N1C(C(CNC(c2c(OC)ccnc2)=O)(C)C)CCCC1 59170,N1(CC(c2cccc(OCC(=O)OCC(F)(F)F)c2)=O)CC2CCC(CC2)C1 59171,C1(C(N(CCCCNC(C(c2cnn(C)c2)C)=O)C)=O)CC2(CC2)CO1 59172,c1(C(c2nnnn2Cc2ccco2)Nc2cc(C)oc2)cccc(Cl)n1 59173,C1(c2n(CCC(=O)OCC)nnn2)(NN2CCSCC2C)CCCSC1 59174,c1(C(N(C)CCOC(=O)COc2cc(F)ccc2F)=O)occ2c1CCCC2 59175,N1(C(C2CC(=O)NC(=O)N2)=O)CC2(NC(=O)C3CC3)CCCC2(F)C1 59176,N1(C(C)=O)CCCN(Cc2cccc(F)c2)C(C)C1.C1(N)CCN(CC(F)F)C1 59177,Cc1nc2ncnn2cc1C(=O)NCC#CCNC(=O)CO 59178,c1(NC(C2(C(=O)O)CC2)=O)onc2c1CNCC2 59179,c1(CC(=O)NCC(CNC(c2cccc[n+]2[O-])=O)OC)nnc(S)n1C 59180,c1(C(N2CCCC(CNC(c3cccc(C)c3I)=O)C2)=O)cnc2snnc2c1 59181,c1(C(=O)NC2CCCN(C(C3CCCC(C)(C)C3)=O)CC2)ccc2nnnn2c1 59182,N1(C(C(C)(C)N(C)C)=O)CCC(C)(CCNC(C2CC2C2CC2)=O)C1 59183,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2ccc(SC)s2)=O)C1 59184,CC1CC(=O)NC1C(=O)NC(c1ccnn1C)C(N1CCC(OCC(N)=O)C1)=O 59185,c1(C2C(NC(C(N3CC(CS(N)(=O)=O)C3)=O)=O)CC2)ccc(Br)cc1 59186,c1(N2CCC3(C(C(=O)Nc4cc(N(C)C)cc(F)c4)C3)C2)ncnc2occc12 59187,N#Cc1cccc(C(=O)NC2CC3CC2N(C(=O)CCC2CCCO2)C3)c1F 59188,c12ccccc1O2.c1(NC(C2C(C(=O)NCc3nncs3)C2)=O)ccccn1.CN 59189,c1(C(=O)NC(C=CC(=O)NCC2N(CC)CCC2)C)cc2ccccn2n1 59190,c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCc2ccccn2)ccn1 59191,N1(C(C(CC)(C)CNC(=O)Cc2ccc[nH]2)=O)CCN2CC(C)CC2C1 59192,N1(C(C2C(C)(Br)C2)=O)CCC(NC(c2ccc[nH]2)=O)C(F)C1 59193,CCCCC(C(=O)N1CC(OCC(=O)NC)C(CC(=O)N(C)C)C1)N(C)C 59194,c1(C(N(CC(CC)NC(=O)CCN2CCC(F)C2)CC)=O)cc(CO)oc1C 59195,CC1=NOC(C(C(=O)NCCCOc2ccccc2)N(C)CCc2ccccc2)C1 59196,C(=O)(CCCN=[N+]=[N-])NC1CCC(CCNC(CCNC(=O)NC)=O)C1 59197,Cc1ccc(C)c(C(N2CC(OCCNC(=O)C(N)=O)C2)=O)n1 59198,c1(CC(=O)NCC2CCN(C(C(C(CC)C)O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 59199,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CCC2C(=O)NN=C2C)CC1)CC 59200,C1(C(=O)NCCC(C)N(C)C(C2CCCN2c2cnccn2)=O)CCCC12CC2 59201,c1(C(N2CCC(OC)(CNC(=O)C(C)c3ccco3)C2)=O)ccc(F)c(F)c1N 59202,C(=O)(C#CC1CCCCO1)NC(C)CNC(c1coc(CO)c1)=O 59203,c1(OC)ccc(C(=O)NC2CCCC2SC)cc1.C12CC(C1)CCC2.C1(=O)CN1 59204,CC1(C)CCCC(CNC(=O)C(=O)NC2CCN(C(c3ccccc3)=O)C2)C1 59205,c1(CC(=O)NCC(C)N(C(c2coc(C)c2N)=O)CC)ccc(C)cc1F 59206,C(=O)(C1OCCn2ccnc21)NC1C(NC(C(C)(F)C(F)(F)F)=O)CCC1 59207,C=C(Cl)CN=C(NC1CCC(SC)CC1)NC1CCC1 59208,CC1ON=C(C(=O)N2CCN(C(=O)COC(F)F)CC2C2CC2)C1C 59209,CCCCCCc1ccc(C(=O)NC(C)CN(C(=O)CC2CC23CC3)C)s1 59210,CC1CN(C)CCC1NC(=O)CC1(C)CCN1C(=O)C(F)F 59211,CCC(CC(=O)N1C2CCC1CC(CNC(C1CCOC1)=O)C2)C(C)C 59212,N1(CC)N=C(C(=O)NCC2CC(O)(CNC(c3cnc(SC)s3)=O)C2)CCC1=O 59213,Cc1ccc(C(=O)NCC2C(C)CCN2C(=O)CCc2ccnc(Cl)c2)n1C 59214,c1(C(=O)NC(C(=O)NCCn2c(CC)ncc2)CN(C)C)cc(C)nc(O)c1 59215,c1(OC)c(F)ccc(NC(=O)C(C)NS(C)(=O)=O)c1F 59216,Cc1ccc(O)cc1CNc1ccc(C2CCN(C(=O)CC(C)C)CC2)cn1 59217,Cc1nc2c[nH]nc2cc1C(=O)NCC1C(C)CCCN1C(=O)CCS(N)(=O)=O 59218,C1(NC(c2c(C)scn2)=O)CC=C(C(=O)N=c2cnc(Br)c[nH]2)CC1 59219,c1(C(=O)NCC(CC)N(C(=O)CSCC(F)(F)F)C)occc1CC 59220,C(=O)(C1OCCc2c(C)cccc21)NC(CNC(C(C)=CC1CC1)=O)(C)C1CCC1 59221,C1(CNC(C(C2CCCCC2)OC)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1(C)C 59222,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59223,c1(CC)ccc(CN(C(=O)C(C)(C2CCC2)NC(=O)C(O)C(C)C)C)cc1 59224,Cc1cc(Cl)c(C(N2CCCC2CNC(=O)C(c2cccc(Cl)c2)O)=O)s1 59225,C(C)(C(CC(=O)NCC12CC(CN1C1CC1)C2)NC(=O)C(C)N1CC(C)C1)OC 59226,C1(C)(C(=O)OCC)C=CCN1C(=O)CC1CCCN(C(=O)CSC(C)C)C1 59227,N1(C(C2(N(C)C)CCC2)=O)CCCC2(CCN(C(=O)C(C)(C)C3CCCO3)C2)C1 59228,c1(OC)ncc(-c2noc(-c3ccc(OCC(C)C)cc3F)n2)c(C)n1 59229,c1(CC(N2CC3C(CNC(=O)C=C(Cl)Cl)C3C2)=O)cc2ccccc2o1 59230,C1(CNC(c2c(CC)con2)=O)(COC)CCN(C(C2CC(C)CO2)=O)CC1 59231,CCCC(F)(F)C(=O)N(CC(O)CN(C(=O)C(O)CNC(C)=O)C)C 59232,c1(C(=O)NCCC2CCN(C(COC(C)C)=O)C2)cnccc1NC(C)C 59233,C(CCC(=O)NCC(CO)NC(c1cnc(C2OCCO2)s1)=O)NC(N)=O 59234,CC1CC(CNC(=O)CNC2(C)CCOCC2)CN(C(=O)C(C)OC(C)(C)C)C1 59235,C(=O)(C1=CC2C=CC(C1)C2)NC1CC(C)(NC(c2c(OC)c(F)ccc2)=O)C1 59236,N1(C(C(C)N2CC(C)C2)=O)CCCC2(CNC(c3cccnc3Cl)=O)CCCC12 59237,CCCC(C)CC(=O)N(C(C)C(=O)NOCC1CCC1)C 59238,c1(N2C(C)CCC(NC(C(C#C)(C)C)=O)C2)cc(C(C)C)nc2ncnn12 59239,C=CC1CN(C(C2CN(C(c3cnn(C)c3Cl)=O)CC2OC)=O)CCO1 59240,C(C)(C(C)COC)(c1nnnn1C1COC1)NCc1onc(-c2c(C)scn2)n1 59241,c1(C(=O)NC2C(CNC(C(CC)(C)OC)=O)C2)ccc(OC)nc1F 59242,c1(C(=O)Nc2c(C(=O)NCc3ccc(Cl)s3)n[nH]c2)ccc(Cl)c2[nH]ccc12 59243,C=CC(C)CC(=O)N1CC(CC(=O)NCc2c(C)noc2C)(OCC)C1 59244,N1(CC(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)CCN(C)CC1 59245,c1(C(=O)NCCNC(C2CCCC(F)C2)=O)ccc(-c2cnccn2)cn1 59246,C=CCC(C(=O)NCC1(O)CCN(C(=O)Cc2ccno2)C1)c1ccc(Cl)cc1 59247,c1(C(=O)NC2CC(F)(CNC(C(C)(C)OCC)=O)C2)cc(C)c(CC)o1 59248,c1(C(N2CCC(O)(C(C)NC(c3nccc(OC)c3)=O)C2)=O)nc(C)ccc1O 59249,c1(CN2CCN(C3CN(NC(CCSC)=O)C3)CC2)cccc2c1COC2 59250,Nc1ccc(C(=O)NC2CCCC2NC(c2cnc(O)o2)=O)cc1Cl 59251,N1(C(c2cccc(CCC)c2)=O)CC2(CC(NC(C3(C)CCC(=O)N3)=O)CO2)C1 59252,c1(C(N2C(CC)(CC)CC(NC(=O)C3=NNC(=O)C3)C2)=O)c(C)ccc(C)c1O 59253,N1(C(C2N(C(c3ccc(C(C)=O)[nH]3)=O)CC=CC2)=O)CCOC(C)(C)CC1 59254,c1(C(=O)NCC2N(C(Cc3c(C)noc3Cl)=O)CCC2)cnc2c(c1)OCCN2 59255,Cc1cnc(C(C)NC(=O)C(COC(C)C)NC(=O)CC(=O)NC2CC2)o1 59256,C1(NC(CCNC(CC)=O)=O)C2CC3CN(C(=O)COC(CC)CC)C1C3C2 59257,N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(C1CC1(C)C)=O)C2 59258,N1(C(CCC2(C)CN(C(C3(CC(C)=O)CC3)=O)C2)=O)CC2CC(O)CC1C2 59259,C1(C(N2C(C(=O)NC)CC(O)C2)=O)CN(C(=O)CC2C=CCCC2)CCC1(C)C 59260,O=C1NCc2c1ccnc2C(N1CC(NC(c2cccc(F)c2)=O)CC1CO)=O 59261,C1(C(N2CCC(N(C(=O)CC3(CO)CC3)CC#C)CC2)=O)CCCC(C#N)C1 59262,C(C(C)(C)CC(=O)NC1CN(C)CC1C)NC(C1(CC)CCC1)=O 59263,c1(CC(=O)N(C(C)=O)CCN(C2CCCC2C)C2CCC2)cccc(Br)c1 59264,Cc1cccc(NC(C2CCCN(C(c3c(C)nn(C)c3C)=O)C2)=O)c1O 59265,N1(C(c2cncc(C#C)c2)=O)CCC(NC(=O)C#CC2CC2)C12CCC2 59266,N1(C(c2cccc(OC)n2)=O)CC2CCN(C(c3cccc(O)c3)=O)CC2C1 59267,c1(CC(=O)NC2C(NC(CCC=C)=O)CCC2)nc2ncccn2n1 59268,C1(NC(COC)=O)(NC(=O)CCc2cscn2)CSC1.C1(=O)CN1C 59269,c1(NC(C)=O)cccc(C(N2CCC(C(C(=O)O)Nc3ccnn3C)CC2)=O)n1 59270,Cc1sc2ncc(C(N3C4CCC3(CNC(=O)C(C)O)CC4)=O)c(=O)n2c1C 59271,Cc1cc(C(=O)NC(C2CCN(C(=O)CCOC3CCC3)C2)C)cc2nn[nH]c12 59272,c1(COCC(=O)N(C(CCNC(C(C)=C2CCCC2)=O)C)C(C)C)ncc(C)o1 59273,n1(CC)cc(C(=O)N(C)CCN(C)C(C2CCCCO2)=O)c(I)n1 59274,C=CCC(C)(C)CC(=O)NCc1cncc(CNC(=O)C(N2CCC(C)C2)=O)c1 59275,C1(C(=O)NCC(C)(C)CNC(=O)C(c2ccc(Cl)s2)=O)CC2(CC2)CO1 59276,Cc1ccc(F)c(O)c1C(=O)NC1CC(C)(NC(C2OCCC2(C)C)=O)C1 59277,C1(C(N2CCOCC2)=O)(CSCC(=O)OCc2sccc2Br)CC12CCC2 59278,c1(C(N2CCN(CC=O)CC2)=O)cc(F)cnc1O.N1(CC)CCCC1CNC 59279,c1(C(=O)NCCN(C(C2C(OCC)C2C)=O)C)cn(C)nc1-c1cccc(F)c1 59280,CC(C)C(C(=O)NCCc1ccncn1)NC(c1cccnc1)=O 59281,c1(C(=O)NCC(C)N(C)C(c2ccc(CO)o2)=O)ccc(OCC(N)=O)cc1 59282,c1(C(N2CCN(C(C(C(CC)O)C)=O)C(C(C)C)C2)=O)cccc2sncc12 59283,c1(C(=O)NC2C(NC(C3C(C)CC3)=O)CCC2)cnn(C)c1Cl 59284,C1(C(N(CC(=C)CCOC)C)=O)CCC(n2cccc2)CC1 59285,C(=O)(N=c1nc2ccccn2[nH]1)C1CC(NS(C)(=O)=O)C1 59286,C1(COC)C=CCCN1C(=O)CN(C(=O)C(C)C1CCCC1)C(C)C 59287,c1(NC(C2CC2C(=O)Nc2cc(SC)ncc2)=O)cc(S(C)(=O)=O)ncn1 59288,C1(CC#C)(C(=O)N(CC)CC2CCCCN2C)CCN(C(=O)CC(O)CC)C1 59289,c1(C(=O)NC2C(CNC(=O)CC3CCOC3)C2)c[nH]c2cc(Cl)ccc12 59290,CC1CC(CCNC(=O)C(=O)NC2CC2)CCN1C(c1cnc(C(N)=O)cn1)=O 59291,C1(C)(NC(C(CNC(C)=O)O)=O)CCc2ccccc21 59292,c1(C(=O)NC(C(C)(C)NC(C=CCC)=O)C)cnc2scc(Br)c2c1 59293,c1(OC)cc(-c2noc(-c3cc(C)cc(C)c3)n2)c(N)cc1Cl 59294,c1(C(=O)NCC(C)CN(C(=O)C(N2CCCCC2=O)C)C)cccc(F)c1N 59295,C(CC(=O)N1CC(C)(C)C12CCC2)(CC(C)C)NC(CCC(C)OC)=O 59296,C1(c2cc(NC(C3(c4ccc(Cl)cc4)CCC3)=O)on2)COc2ccccc2C1 59297,N1(C(C(CO)NC(C2C3CC(=O)CC32)=O)=O)CC2(CCNC2=O)C1 59298,c1(C(=O)NC2CC(N(C)C(C3C=CCS3)=O)C2)cnn(Cc2ccco2)c1O 59299,C=CC(C)CC(=O)N(C)CC1CN(C(=O)CCc2cncnc2)C1 59300,C1(C(=O)NCC2(C(C)(C)O)CN(C(COCC(=O)OC)=O)C2)CCc2ccnn2C1 59301,c1(C(=O)OC)cnc(C)cc1N1CCCC1C1(NC(=O)C(C)NC(N)=O)CC1 59302,N1(C(c2cc(CC)nn2C)=O)CCC(N)c2ccc(Cl)cc2C1 59303,c1(C(N(C2C3CN(C(=O)CC4(O)CCC4)CC23)C)=O)cncn(C)c1=O 59304,c1(NC(c2cccc(C)c2NCC)=O)ccc(Cl)c(C(=O)OCCCSCC)c1 59305,Cc1ccc(-n2cc(C3(NC(=O)C4CC4)CCC(C)CC3)nn2)cc1[N+](=O)[O-] 59306,c1(Sc2scc(C)n2)nnc(CNC(=S)SC)n1-c1ccc(CO)cc1 59307,C(CC(=O)NC(C(C)C)C1CC1)(C(F)F)NC(c1cc(OC)ncc1)=O 59308,N1(C(C2(C)CCCN(C(c3ccncc3N)=O)C2)=O)CCCCCCCC1 59309,Cc1nc2ccc(C(N3CC(Cc4cccc(Cl)c4)C3)=O)cc2o1 59310,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)CC1CCCCC1 59311,C(=O)(C(CNC(C1CCOC1C)=O)CC(C)C)Nc1c(F)ccc(OC)c1 59312,C1(CNC(C23CC2C3)=O)CCCCN1C(c1ccc(C(F)F)s1)=O 59313,c1(C(=O)NCCNC(C2C(CNC(Cc3cc(C)no3)=O)C2)=O)c[nH]ccc1=O 59314,CCCC(F)C(=O)NCCC1(NC(=O)CCCC2CC2C)CCC1 59315,CC(C)(C)C(CCc1ccccc1CN1CC=CC(O)C1)NC(=O)C1CC1 59316,CON1CCC(C(=O)NC2CC(F)(CNC(C3CCN3S(C)(=O)=O)=O)C2)CC1 59317,C1(NC(c2nccc(OC)c2O)=O)CCCC12CN(c1nccc(CO)n1)C2 59318,C1(CC#C)(C(=O)NCc2ccccc2F)CCN(C(C2CC2c2ccsc2)=O)C1 59319,C1(c2n(C)ccn2)CCCN1N1CCC(c2ncccn2)CC1 59320,C1(CN(C(=O)CC(C)(C)n2cc(C3(O)CCCCC3)nn2)C)CCC(N=[N+]=[N-])C1 59321,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCS(=O)(=O)CC2)C(CF)C1 59322,C1(OCC)CN(C(C)=O)CC1NC(c1nc(O)n[nH]1)C.c12ccccc1OC2=O 59323,C(CCC(=O)NC(CN(C)C)C(=O)N(C1CCN(C)C1)C)OCCOC 59324,Nc1cccn(CC(N2CCN(C(=O)CCC3CCC(=O)N3)C(CO)C2)=O)c1=O 59325,CCC(C)C(O)C(=O)NC1(CNC(c2cc(-n3cccn3)ccn2)=O)CC1 59326,C(CC(C(C)(C)C)NC(=O)Cn1nnnc1C)N(C(c1c(C)nccc1)=O)C 59327,CCC(CC)(CCNC(=O)C(C)Cc1ccncc1)NC(c1cc(F)n(C)n1)=O 59328,Cc1c(Cl)c(C(N2CCC(C)(NC(=O)CC3CCC4CC34)C2)=O)nn1C 59329,N1(C(C(=O)NC(C(=O)N(C(=O)C2CC2)CC)C)=O)CCCC2(C=CCO2)C1 59330,C12(NC(CSCC(=O)OC)=O)CC1CN(C(=O)C(c1cnn(C)c1)C)C2 59331,C1(CNC(CCOCC#C)=O)(OCC)CN(C(c2sccc2F)=O)C1 59332,CC(C)(C)CC(O)CC(=O)NCCCC1(NC(=O)Cc2nn(C)cc2Cl)CC1 59333,C(=O)(CCCCCF)NC(CC)CC(=O)NCC1(C)CCN(C)C1 59334,c1(C(=O)NC(c2cc(Cl)n[nH]2)C(=O)OC)nc2nccc(C)n2n1 59335,c1(CC(=O)NCC(CC)NC(C2CCCOC2)=O)cnc(COC)s1 59336,c1(NC(=O)N(C2CC2)Cc2cn(CCCO)nn2)nccc(C(F)(F)F)n1 59337,CC(C)CC(C(=O)N1CC2(CCC(CNC(C3OCCOC3C)=O)O2)C1)C(N)=O 59338,c1(-n2c(CCCC)nc(C3CCOCC3)n2)c(C(F)(F)F)cccc1Br 59339,N1(C(C2CN(C(C(C(C)(C)C)SC)=O)CC2C2CC2)=O)CCC2(CCC(O)C2)C1 59340,C1(C(N(CCCNC(C(C(=O)OCC)OC)=O)C2CC2)=O)CN2CCCN1CC2 59341,c1(C(=O)NCC(C)CN(C)C(C2COC(C)CO2)=O)ccc2c(c1)C=CS2(=O)=O 59342,C1(CNC(c2n(C(CC)C)ncc2)=O)CCCN(C(=O)C(C)(C)CC)C1 59343,C1(C)(CNC(c2ccc(CCC)s2)=O)CCC(NC(C2(CF)CC2)=O)CC1 59344,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C(C(=O)NC2CC(C)(C)C(=O)NC2)C1 59345,C(C(N=c1nc2scnc2c(NCC(C)C(F)(F)F)[nH]1)c1ccccc1)SC 59346,n1(C(C)C)cnc2c(NCCCCN(C)C)[nH]c(=NCCC3CCC4CC34)nc12 59347,C(C)(C)(C(=O)NC1CC(NC(C2(F)CCOC2)=O)C1)NC(=O)NCCC 59348,C1(Cl)(C(=O)NCC2(NC(c3nc(CCCC)sc3)=O)CCC2)CC12CCC2 59349,c1(C(=O)NCC(CC)NC(=O)COCC2CCCC2)cc(C(F)F)ncn1 59350,c1(C(N(CCCNC(C=C(C)C(F)F)=O)C2CC2)=O)ccc2nc(S)oc2c1 59351,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59352,c1(C(C(=O)NCCOC)N(CC(C)OC2CC2)C)cc(C)c(C)c([N+](=O)[O-])c1C 59353,[N-]=[N+]=Nc1ccc(C(=O)NCC2CCCN2C(C2CCC3CCCCN23)=O)cc1 59354,C1(C(N2C(CNC(C3CCC(O)CC3)=O)CCCC2)=O)CC2CS(=O)(=O)CC2C1 59355,C1(CNC(c2n(C)ncc2)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59356,C1(CC(=O)NCC=C=C)CN(C(C2(O)CC(CF)C2)=O)CCO1 59357,c1(CCN2C(C(C)N(C)C)CCC2)cn(C(C)CNC(C2CC3CC3C2)=O)nn1 59358,N1(C(C2CN(C)C(=O)N2)=O)CCC(C2CC2)(CNC(C2CN(C(=O)NC)C2)=O)C1 59359,C12(NC(c3cccc(-c4ccccc4)c3)=O)CC(C1)N(C(=O)CCC1CC1)C2 59360,c1(C(=O)NC(C(C)(C)C)CNC(c2cnc(Cl)s2)=O)ccc(C#N)cc1F 59361,N1(C(CC(Cc2ccc(OC)cc2)N)=O)CCC(O)CC1(C)C 59362,O=C(CC(C(F)F)n1cccn1)NC(c1ccnn1CC1CCCO1)=O 59363,C1(NC(=O)Cn2cc(C3CC3)nn2)(CNC(c2c[nH]cc2Br)=O)CCOC1 59364,c1(CSC)ccc(C(=O)NC(C)CCNC(=O)CC2CCCCO2)cc1 59365,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59366,C1(C)(C(N2CCCC(F)(CNC(c3c(CC)nn[nH]3)=O)C2)=O)CC(C(C)(C)C)=NO1 59367,C1(NC(C2(C)C=CCN2)=O)CCCC12CCCC2 59368,N1(C(C(CSCC)NC(c2ccsc2)=O)=O)CCC2(CCC(OC)C2)C1 59369,C1(c2cnc(C)[nH]2)NC(=S)N(C2(C)CC(O)C2)C2=C1C(=O)NCC(C)(C)C2 59370,C1(C)(C(N(CCC)CCNC(=O)COCC2CCCOC2)=O)CCC(C)=C(C)C1 59371,C1(NC(c2cc(C)sc2C)=O)CC(NC(=O)CCOC2CC2)C12CCOCC2 59372,c1(C(=O)NCC(C2CCC2)NC(C2CC=CCC2)=O)ccnc(-c2ccco2)c1 59373,CCC(N=c1[nH]c(=NC(C)c2cncnc2)[nH]c2cccnc12)C(C)C 59374,N1(C(CCN(CC)CC)=O)C2CCC(C2)C1CSc1cc[nH]c1 59375,C#CCC(C)(C)C(=O)N1CCCC(C(N2CCOC3CC23)=O)CC1 59376,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59377,CC1CCN(C(c2cnn(C)n2)=O)C1CNC(=O)CCCN1CCCCC1 59378,C1(NC(C(C)Oc2cccc(Cl)c2)=O)CC(N=c2[nH]ncs2)C12CCC2 59379,Cc1ccc(NC(=O)CCc2cncnc2)cc1C.C12CC3CCC1(C3)NC2=O 59380,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59381,N1(C(C2C(C)N(C(c3ccn(C4CC4)n3)=O)CC2)=O)CCC(O)C12CCC2 59382,C1(C(=O)NCC2C3CN(C(c4nn(CC)c(O)c4)=O)C2C3)CCc2c[nH]nc2C1 59383,C(=O)(CCS(C)(=O)=O)N(CC(=O)N(CC(C)N)C)C.C(N)=O 59384,c1(CC)nccnc1C(=O)NC1C=CC(C(=O)N(C2COCC2OC)CC)C1 59385,c1(-c2cc(C)cc(C)c2)cccc2c1CCN(C(c1ccc(CCF)cc1)=O)C2 59386,C(=O)(CCS(C)(=O)=O)NCC(CNC(CC(COC)C)=O)C 59387,c1(C(N(C2CCN(C(CC(c3c(C)noc3C)C)=O)C2)C)=O)cn2c(n1)CCC2 59388,N1(C(c2ccc(C)o2)=O)CCC(C)CC1C(=O)NCC12CC(CO)(CO1)C2 59389,CC(C)(CC(=O)N1CCN(C(c2ccc(N)c(F)n2)=O)CC1)C(F)F 59390,C1(NCC2(COC)CCOCC2)CCCN(C(C)C(C)(C)C)CC1 59391,c1(C(=O)NC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(F)cccc1Br 59392,C#CCCN=C(NCc1ccc(CC)cn1)NCC1(C)CCCCO1 59393,c1(C(=O)NCCC2CCN(C(c3c(CC)csc3)=O)C2)ncc(N(C)C)cn1 59394,c1(CCC(=O)NC2(CC=C)CCCN(C(=O)C(C)SC)C2)cnc2n1CCCC2 59395,CC(C)C(O)C(=O)NC1CCC(NC(C2(Cc3ccccc3)CCC2)=O)C1 59396,c1(C(N2CCC(NC(C3(NC(C)C)CC3)=O)C2)=O)ccc(Cl)c(C(F)F)c1 59397,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59398,C1(CC(=O)OC)C(NC(=O)CN(C2COCC2O)C)C1(C)C 59399,c1(C(=O)NCC(C)CNC(=O)CNC(N)=O)cc2c(C(F)(F)F)cc(O)nc2o1 59400,c1(C(=O)OC)cnc(NC2CN(C(=O)COC(C)(C)C(F)(F)F)CC2C)c(F)c1 59401,N1(C(c2ccc(C)[nH]2)=O)CC2(C)CN(C(c3ccn(C(C)C)c3C)=O)CC2(C)C1 59402,CCCCCC(O)C(=O)NC1CN(C(=O)COc2ccc(C(C)C)c(C)c2)CC1C 59403,c1(C(=O)NCCCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59404,C12(C(=O)NCC3(NC(CC=C=C)=O)CCCC3)CCCCC1C2(F)F 59405,Cn1cc2cccc(C(=O)NCC3(C)CN(C(=O)CCOC4CC4)CCO3)c2n1 59406,N1(C(c2cc(N)cc(F)c2)=O)CCCC2CN(C(=O)Cn3[nH]cnc3=N)CCC12 59407,n1(CCNC(NC(CCC)C(N)=O)=NCC2CCC2)nc2ccccn2c1=O 59408,C=CCC(C)(C)CC(C(=O)NCCSC)N1CCC(C)(F)C1 59409,Cn1ncc2nc(O)c(C(N3CC(CCCCNC(c4ccc[nH]4)=O)C3)=O)cc12 59410,CCCC(CCCCCC)NC(=O)CC1CNC1 59411,Cc1cc(C(=O)NCC2CC(C(F)(F)F)CN2C(=O)COCCCF)n(C)n1 59412,C(CNC(CNC(C1CCCN1S(C)(=O)=O)=O)=O)(CC(F)(F)F)OC(C)C 59413,c1(CC(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2F)cccc2sccc12 59414,N1(C(C2C(OC)CCOC2)=O)CCC(NC(=O)C(=O)NC2CC2)C2(CCC2)C1 59415,C(=O)(CCC(C)(C)C)Nc1cnc(C)c(C)c1.C12(COCC)CCCN1C2=O 59416,c1(C(C)C)cc(C(=O)N(CCCCCNC(=O)C(=O)NC(C)C)C)n(C)n1 59417,CC(O)C(C)C(=O)NCC1CC(NC(c2ncc(N(C)C)cn2)=O)C1 59418,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59419,c1(C(=O)OC)ccc(=NCCC2CCCN(C(c3snc(Cl)c3Cl)=O)C2)[nH]c1Cl 59420,Cc1cnc2c(cnn2CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)c1 59421,C12(NC(CCCOC)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59422,N#CC1CN(C(C)(C)C)CC1NC(=O)OCCC(=O)Cc1ccccc1Br 59423,C(C(=O)NC(C1CN(C(=O)C(F)=C(C)C2CC2)C1)C)(C1CCC1)OC 59424,C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2onc(CC)c2C)=O)C1 59425,c1(C(N2CC3CC(NC(c4coc(Br)c4)=O)C3C2)=O)ccnc2cc[nH]c12 59426,CN1CCC(O)C(NC(C2CC2CNC(c2cn3c(n2)CCC3)=O)=O)C1 59427,N1(C(c2c(C)nc(CC)s2)=O)CC2CCN(C(C3CCC(C)(C)O3)=O)C2C1 59428,CC1(C)CC(C)(C(=O)NCCCN(C(=O)CC2CC(C)(C)C2)CCO)C1 59429,c1(C(N2CCN(C)CC2CNC(C2CCCSC2)=O)=O)scc2c1CCCC2 59430,c1(C(=O)Nc2cccc(-c3cc(C)c(O)nc3)n2)ccc(C#N)c(F)c1 59431,C(=O)(NNc1ccc2nc[nH]c2c1)C1N(CN2CCC3(NC(=O)OC3)CC2)CCC1 59432,c1(C(N2C3C(NC(C=C(C)C(F)F)=O)CC(C3)C2)=O)cc([N+](=O)[O-])cn1C 59433,c1(C2C(C(C(=O)NC3CC(CCF)C3)OC)C2)ccc(Br)cc1 59434,C(=O)(C(C)(C)C1CCOC1)NCCC(C)N(C(C=C(COC)C)=O)C 59435,CCCCCCCC(F)C(=O)NCCC1CCN(C(=O)C(C)=C2CC2)C1 59436,N1(C(C2CCC(CCCCOC)C2)=O)CCN(C(C2CCCC23CC3)=O)CC1 59437,N1(C(CCc2ccc(C(=O)OC)nc2)=O)CCN(C(=O)C(O)CF)C2COCC12 59438,C1(CNC(C(CC)CC)=O)CCN(C(=O)Cn2c([N+](=O)[O-])cnc2C)CC1(F)F 59439,N1(CCCC(CC)=O)CCNC12CCOCC2 59440,N1(C(CCC2N(C)CCC2)=O)CC2CC1C2NC(c1cc(CN(C)C)on1)=O 59441,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)ccnc(F)c1OCC 59442,C1(NC(C2(F)CCN(C(c3n(CCC)ncc3)=O)C2)=O)CCCC(O)C1O 59443,C1(CN(C)C(C2CC2F)=O)CN(C(=O)CCOC2CC2)CC12CC2 59444,c1(C(N(C2CCN(C(=O)CCCC(N)=O)C2)CC)=O)cccc2ncc(C)cc12 59445,C1(NC(=O)CSC(F)(F)F)CCCC12CN(C(=O)C(F)C1CCCC1)C2 59446,N1(C(=O)C(c2ccccc2)NC(=O)COC(C)(C)C)CCCC(C)(CSC)C1 59447,C1(NC(COCCNC(COCCC)=O)=O)NC(=O)NC1=O 59448,N1(C(C(C)SCC)=O)CC(NC(c2ccnc(-c3ccccn3)n2)=O)C(C)C1 59449,c1(C(=O)NC(C(c2ccccc2)NC(C(CC)(C)OC)=O)C)ccc(Cl)cc1O 59450,C(=O)(C#CC(C)(C)C)NCCCN(C(c1snnc1C1CC1)=O)CC 59451,Cc1ccc(Cl)cc1C(=O)NC(C1CCCC1)CNC(C1COCC(C)O1)=O 59452,N1(C(C(OC)OC)=O)CCCCCC(CNC(c2cncc(OC(F)F)c2)=O)C1 59453,S(=O)(=O)(c1cnc(NCC(c2nccs2)C)c(Cl)c1)N1CCn2c(C)ncc2C1 59454,CCC(C)C(O)C(=O)N1C2CCC1C(CNC(C1(C)CCC1)=O)C2 59455,c1(C(N(C2C3CN(C(=O)CC#N)CC23)C)=O)cc2scc(Br)c2[nH]1 59456,C1(CNC(C2C(C)C2)=O)(CO)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 59457,C(CNC(=O)Cc1cnnn1C)(CC(F)(F)F)NC(C(C)SC)=O 59458,C1(C(=O)NC2C(c3ccn(C)n3)C2)CCCCN(C(C2CCCC23CCC3)=O)C1 59459,c1(OCC(N2C(CNC(c3n(C=C)nnc3)=O)CCC2)=O)ccc(F)cc1O 59460,Cc1nc2cc(C(=O)OC3CC(CNC(=O)CC4COC5CC4C5)C3)[nH]c2s1 59461,c12nc(ncc1F)N2.c1(CSC)ccnc(C(=O)NC2CONC2=O)c1 59462,N1(C(C2N(CC)CC2)=O)CCN(C(c2c(C)cnnc2O)=O)CC1CC(F)(F)F 59463,N1(CC)CC(NC(=O)C(CC2CCCC2)NC(=O)C(C2CCOCC2)=O)C(C)C1 59464,N1(C(C(=O)NCC)=O)CCCC(C)(NC(C2CC23CC(O)C3)=O)C1 59465,CCC(C)C1CC(=O)N1.CC1CC(O)CN1C.C1(C(=O)N)CCCN1C=O 59466,N1(C(Cn2c(C)ccn2)=O)CC2C(CNC(C3CC4CCC3O4)=O)C2C1 59467,N1(C(CC2(C#C)CC2)=O)CC2(CC2)CC1CNC(=O)CN1C(=O)CCCC1=O 59468,C(=O)(CS(=O)(=O)C1CCCC1)NC1CN(C(Cc2nc(C)oc2)=O)C(C)CC1 59469,C(CCCCNC(c1nnnn1C(C)C)(CC)C1CCC1)NC(=O)NC 59470,C(c1ccccc1Cl)=C(C)C(=O)NCCC1CCCN1C(=O)CC1CC1(Cl)Cl 59471,C(c1ccncn1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59472,C1(CC(=O)NCC(CNC(c2cc3n(n2)CCC3)=O)OC)CC(C)(C)OC1=O 59473,C1(c2c(F)cccc2F)CC1N=c1ccnc(NC2CCN(c3ccccc3)C2)[nH]1 59474,c1(-n2c(CC)nc(C3CN(C)CCO3)n2)ccc(C)c(Cl)c1.n12ccnc1C1CC21 59475,c1(N2CCC(C)CC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CCO 59476,c1(C(=O)NCC(C(=O)NCC2C(C(C)C)CCO2)N(C)C)cc(O)nc(C)n1 59477,c1(C(=O)NC2CC(F)(CNC(C3(CC)C=CCC3)=O)C2)[nH]c(O)nc1C 59478,CCCC(C(=O)N1CCOC(C(=O)NCC(O)(CC)CC)C1)OC 59479,N1(C(CCNC(=O)OC)=O)CCC(N(C)C(C2COCCN2C)=O)C1C 59480,C1(C(=O)NCCC(C)(O)COC)(OC)CCN(C(=O)CCC2CCCCC2)C1 59481,c1(-n2cc(C3(NC(c4cccnc4)=O)CC3)nn2)ccc(Cl)cn1 59482,N#Cc1cc(C(N2CCC(=CC(=O)Nc3ccc(F)c(F)c3Cl)CC2)=O)ccc1F 59483,C1(NC(CCN(C(CC=C=C)=O)CCCO)=O)CCOC1C=C 59484,N1(C(=O)NCc2nccnc2Br)CCC2CCC12c1cccs1 59485,N1(C(c2c(C)cc[nH]2)C)CCCC(C(=O)N(c2ccc(F)cc2)C(C)CO)CC1 59486,C1(C)(C(=O)NCCCCC(=O)OC)CCCN(Cc2cccc(O)n2)C1 59487,C(=O)(C(F)C(C)CNC(c1cccc2c1CC2)=O)NCc1cc(C)n(C)n1 59488,C(=O)(CC1C(=O)Nc2ccccc21)N1CC(C)C(CNC(=O)COCC(F)F)C1 59489,C(CCN=C(NCC(=O)NC(C)C)NC1CCOC(C(C)C)C1)OC 59490,C(=O)(C1CNc2ccccc21)NCC1CN(C(CC2C(C)(C)CCCO2)=O)C1 59491,C12(NC(=O)CCn3ccnn3)CC(C1)N(C(C1CC3C=CC1C3)=O)C2 59492,c1(C(=O)NC(C2CC(NC(C3(Cl)CC3(F)F)=O)C2)C)cc(-c2cnn(C)c2)[nH]n1 59493,CC1CN2CCN1CC2C(=O)NCC(C1CC1)NC(c1c[nH]c(Br)c1)=O 59494,c1(C(C(=O)O)NCC2=CCCCCC2)cc(Cl)cc(Cl)c1F 59495,Cn1cc(C(=O)NCC2CCCC2NC(c2ccccc2Cl)=O)nc1O 59496,c1(C(=O)NCC(CN(C(=O)C(CC)OC)CCC)O)ccnn1C1CCC1 59497,C1(C(N2CCC(CCF)CC2)=O)C2CC(O)C(C2)N1C(=O)C(O)CC(F)(F)F 59498,CC1CCc2nc(C(N3CCC(NC(c4ccc(N(C)C)cc4Cl)=O)C3)=O)cn2C1 59499,C1(O)(C(N(C(CCNC(c2ncn(CC)n2)=O)C)C)=O)CCC(C)CC1 59500,c1(C(=O)Nc2ccc(O)c(F)c2)ccc(F)cc1Cl 59501,c1(CC(=O)N(C(C)CNC(c2cscn2)=O)CC)conc1C 59502,N1(CC)CCN(Cc2ccc(O)c(OC)c2N)CC1=O.c12ncccc1NC2=O 59503,C(=O)(CC(C(F)(F)F)NC(=O)C(C)OCC(C)C)NC1(CC)CC=CCC1 59504,N1(C(C2CCC(CC)O2)=O)CC=CC(NC(c2csc(CO)n2)=O)C1 59505,c1(C(=O)NC2CC(CCNC(c3ccnnc3O)=O)C2)cccc2[nH]nc(O)c12 59506,C#Cc1cncc(NC(C2CCN(C(c3n[nH]c(C)c3Cl)=O)CC2O)=O)c1 59507,C(=O)(CCC(C)(F)F)NCCCCC(C)NC(C(C)C)=O 59508,c1(OCC(=O)OCC)ccccc1F.c1(C(N2CCC2)=O)conc1C1CCC1 59509,C(=O)(CC(C)OCCO)OCCCNC(=O)COC(CC)CC 59510,c1(C(C(N)=O)=O)ccccc1C(=O)NCC1C2CC1N(C(C1CC3CCC3C1)=O)C2 59511,c1(C(C(=O)NCCOCC)N(CCc2ccco2)CC)ccc(I)cc1 59512,C1(NC(c2ccn3cnnc3c2)=O)CC12CCN(C(=O)CCC(F)(F)F)CC2 59513,c1(N(CC)CC2CCN(C(=O)C(C)Oc3ccccc3Cl)CC2)ccccc1F 59514,C12(C(=O)NCc3nnn(C4CC4)c3-c3ccc(C)cc3)CC=CCN1CCC2 59515,c1(NCCCOCC)ncc(S(=O)(=O)N2CCS(=O)(=O)CC2C)cc1Cl 59516,Cc1cccc(Cl)c1C(N1CCC(OCCNC(=O)Cc2ccsc2)CC1)=O 59517,C(=O)(CC(C)CC(=O)OC)N1CCCC(CC(=O)NCC(C)NC)C1 59518,c1(C(N(c2c(C)nn(C)c2C)Cc2ccccc2)=O)ccc2c(c1)sc(=O)n2C 59519,CC(C)CC(C)(CN=c1[nH]c(Cl)ncc1Br)NC(c1cn2c(n1)CC(C)CC2)=O 59520,C1(C(C(=O)NC2(c3ccccc3Cl)CC2)O)CCC2(CCOCC2)CO1 59521,c1(CN2CCCC(C)(C(=O)NCC3(F)CCC3)C2)cc(F)c(Cl)cc1O 59522,Cn1cnc2c(N3CCOCC(NC(c4ccc(Br)c(O)c4Br)=O)C3)ncnc12 59523,C1(NC(C)=O)CCC(C(=O)NCCC2CCCN(C(=O)CC3CCCO3)C2)CC1 59524,C1(N(C(=O)CC2(NC(c3cc(F)n[nH]3)=O)CCCC2)CC)CCCN(C(C)=O)C1 59525,C1(CN(C(=O)C=Cc2ccoc2)C)CCCN(C(C2CCC(=O)N2C2CC2)=O)C1 59526,c12ccn(n1)CC(=O)N(C)C(C)CNC2=O.c1(C(=O)NC(N)=O)ccco1 59527,S(=O)(=O)(CC(=O)NCC1CN(C(c2conc2C2CC2)=O)CC1C(F)(F)F)NCC 59528,C1(C)(CNC(C(C)COc2ccccc2)=O)CN(C(=O)C(=O)N(C)C)CCO1 59529,C1(C(F)(F)F)(C(=O)OCC)CCCN1C(=O)COc1ccccc1C 59530,CCCC(CCC)C(=O)N1CCCN(C(c2cnc(O)s2)=O)C(C)C1 59531,C1(C(N2CC(C(=O)NC(CSC)(C)C)C2)=O)CCC(C)CN1C(=O)OC(C)(C)C 59532,S(=O)(=O)(C1CCC(C)C1)NC1(SCCCCC(=O)OC)CC1 59533,N1(C(c2onc(CC)n2)=O)CCC(CNC(c2ccnn2CC#N)=O)C(O)C1 59534,N1(C(C(C)CF)=O)CC2(C1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 59535,C1(C(N(C(C2CCC2)C)CC)=O)CC12CCN(C(c1ccsn1)=O)C2 59536,C1(c2n(CCCCCNCC(C)C)nnn2)(OC)CC2CC1CC2O 59537,c1(CC(=O)NC2C(NC(CCC(c3ccc(C)cc3)=O)=O)C2)cc(F)ccc1Cl 59538,C(CNC(c1cnn(CC2CCOCC2)c1)=O)(C(C)C(C)C)NC(CCC)=O 59539,N1(C(c2c(CC)n[nH]c2)=O)CCCC(N(CCO)C(c2ccoc2C)=O)C1 59540,N1(C(C2CC(Cl)(Cl)C2)=O)CC2CN(C(C3CC(CF)C3)=O)CC2C1 59541,c1(C(=O)NCC2C(CNC(=O)Cc3cc(F)cc(Br)c3)C2)ccc2occc2c1 59542,C12(C(C(C)C)NC(c3nc(-c4cnccn4)no3)=O)CC3CC(CC(C3)C1)C2 59543,c1(NC(C2CC(F)CN2C(c2cnc[nH]2)=O)=O)nc(Cl)cc(Cl)n1 59544,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59545,N1(C(C(c2ccn(C)c2)C)=O)CCCC1c1ccon1.N1CCCC1 59546,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59547,C1(C(N2CC(NC(c3c(C)oc(-c4ccco4)n3)=O)C2)=O)CCn2ccnc2C1 59548,c1(-c2cn(C(CCCC)C)nc2)ccc(N=c2ncnc3[nH][nH]c(C)c2-3)s1 59549,C1(CNn2cc(CCC=C)nn2)CC2(CC2)CN1C(=O)CC1(C(F)(F)F)CC1 59550,C1(C(=O)NC2CC(F)CN(C(=O)C(F)=CCCF)C2)CC2C=CC1C21CC1 59551,C(=O)(C(F)(F)c1cncs1)N(CCN(C(=O)Cc1ccc(Cl)s1)C)C 59552,N1(C(c2ccc(C)cc2)CF)C(=O)CN(C)C1=O.O(CO)CC 59553,Cc1nc(NC2CC2C(=O)Nc2cccc(I)c2Cl)nc2ccccc12 59554,C1(O)(C(N(C2CCC2)C(=O)NCCNC(c2nc(Cl)cs2)=O)=O)CCCCC1 59555,C#CCCN=C(NCCc1ccccc1C#N)NCc1ccn(CC(F)F)n1 59556,CC1C(C)N(C(c2cnccn2)=O)CCN1C(c1ccc(C#N)cc1O)=O 59557,N1(C(CC2(CN(C)C)CCOCC2)=O)CC(NC(=O)CS(C)(=O)=O)CC12CCC2 59558,C(CC(C(=O)N1CCCCC1CC(N1CCC(F)C1)=O)OC)OC 59559,c1(C(=O)NC2CC3CCC(C2)N3c2nccc(CO)n2)nc2ccccn2c1F 59560,c1(C(C)C(=O)N(C)CC2CCCN(C(c3ccnnc3)=O)C2)ccc(F)c(F)c1 59561,N1(C(CC2CC(OC)C2)=O)CC(C(=O)Nc2cc(C)cnc2O)CC(C)C1 59562,C(=O)(C1=CCCCO1)N1C(C(=O)NCC2CCCN(C)C2)CC1 59563,c1(C(N2C3CC4(NC(c5cncs5)=O)C(C2CC3)C4)=O)ccc2c(n1)CCCN2 59564,C(C1C(C(=O)NCC2CCC2NC(=O)CC(F)F)C1(C)C)=C(C)C 59565,CC1(C)CNC(=O)C1NC(=O)CN(C(c1ccc(F)cn1)=O)C1CC1 59566,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59567,C1(C(=O)NC(CNC(C(C)=C(C)C)=O)(C)C(C)C)C2COC(C)(C)OCC12 59568,c1(C(N(CC(Cc2ccccc2)NC(CC2(OC)CC2)=O)C)=O)cc[n+]([O-])cc1 59569,C1(O)(CNC(C2CC(SC)C2)=O)CCCN(C(=O)C(N2CCCCC2)C)CC1 59570,C1(NC(CC2CN(C(CCOCC#C)=O)C(C)C2)=O)CN(C)C(C)(C)C1 59571,Cc1ccc(C)c(CCCC(=O)NCC#CCNC(=O)CNC(=O)C2CC2)c1 59572,c1(C(C)NCc2ccc(F)c(C(=O)N(C)C)c2)ccc2nc(O)[nH]c2c1 59573,c1(CC(=O)NC2CCC(CCNC(C3(CNC(N)=O)CC3)=O)C2)ccc(Cl)cc1 59574,C(C(=O)NC(CC)C(=O)N(c1cn(C(C)C)nn1)C)(C(C)C)SC 59575,C(=O)(C(C)(C)C)N(CC(C)(C)OCCNC(CN(C)C)=O)C1CC1 59576,c1(C(=O)NCC2(O)CCN(C(C(C)SC)=O)C2)coc2ccc(OC)cc12 59577,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59578,C12(C(N3CC(CCCC)C3)=O)CCCC1CCN2C(c1cncc(C)c1)=O 59579,CC1(C)CCCN(C(c2cscn2)=O)C1CNC(=O)CSCc1ccccc1 59580,C1(C(=O)NCCCOC2CC(NC(=O)C3CC3)C2)CCCC(F)C1 59581,C=C(C)CCC(=O)NC(CN(C(=O)C(C)(c1cccnc1)OC)C)(CO)CO 59582,CC1(C)Cc2cc(-c3noc(CC4CCCCC(C)(C)C4)n3)sc2C1 59583,N1(C(CCOC(C)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 59584,C1(F)(C(=O)NC(C)CCCNC(=O)Cn2cc(C3CC3)cn2)CCCN(C)C1 59585,C1C(O)CC(=O)NC(=O)C1.c1(CC)cccc(F)c1.CCC(C)C(=O)N 59586,c1(C(=O)NCC2N(C(c3cncc(C=C)c3)=O)CCC2)ccc2c(c1)CCO2 59587,C1(OC)(CNC(C2(OC)CC2)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 59588,N1(C(C(C)OCC2CCCO2)=O)CC2CC2(c2cn(CC3COCCO3)nn2)C1 59589,c1(C(=O)NCCC(=C)CNC(=O)CCOCC)ccc(O)c(N)n1 59590,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3cc(Cl)ncc3Cl)C2)cc1Br 59591,C1(NC(C2(COC)COC2)=O)C(C)(C)CN(C(=O)CC(=O)NC2CC2)CC1(C)C 59592,C(=O)(C1c2ccc(O)cc2CCN1CC(=O)NCC(F)(F)Cl)OC 59593,C1(CCNC(C(C=C)O)=O)CCN(C(=O)Cc2ccnc(C(N)=O)c2)C(C)C1 59594,N1(C(C(C)=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 59595,N1(C(C2(OC)CC(C)(C)C2)=O)CCCC(F)(C(N2CCNC(=O)C2C)=O)C1 59596,Cc1c(F)ccc(C(N2CCN(C(=O)CCC(N)=O)CC(O)C2)=O)c1C#N 59597,c1(C(N2CCC(C)(NC(c3cnc(C)[nH]3)=O)C2)=O)cc(F)c(F)c(Cl)c1F 59598,c1(C(N2CC(CCNC(CC(=O)NC)=O)OCC2)=O)cc2cccc(O)c2[nH]1 59599,Cc1cc(F)ccc1-n1ccnc1C(=O)NCC1(C(=O)O)CCCOC1 59600,CC1=C(C(=O)NCCN2CCC(NC(=O)CC3CCOC3=O)C2)CCO1 59601,c1(NC(c2scc(C(=O)Nc3cccc(CC)n3)n2)=O)c[nH]c2cc(OC)ccc12 59602,CC1(C(=O)NCCC(N)=O)CCN(Cc2ccncc2Cl)C1 59603,C1(C(N(C2CCN(C(c3cnc(C(C)OCC)s3)=O)C2)C)=O)COCCOC1 59604,N1(C(CC)=O)CC2=C(C1)CN(C(c1cnc(CC)[nH]1)=O)C2 59605,C(=O)(C(F)(F)C(F)F)NCC(CNC(CCC=CC)=O)(C)C 59606,C(C(CNC(=O)CNc1ccccc1)CO)NC(C1(NS(N)(=O)=O)CCCC1)=O 59607,N1(C(c2cnn(CCNC(C3(CO)COC3)=O)n2)=O)CCC(CO)C(F)(F)CC1 59608,c1(C(N2C3CN(C(CCCC(C)=O)=O)CC2C3)=O)nc2cccnc2s1 59609,Cc1sc(Br)c(C(=O)NC2CC(F)CN(C(=O)C=CCO)C2)c1C 59610,CC1CN(C(=O)C(C2CCCO2)C2CC2)CC(C)CN1C(=O)CCC(C)(C)C#N 59611,Cc1cccc2cc(C(=O)NCCNC(=O)C(C)Cc3ccc(C#N)cc3)nn12 59612,C1(C)(C(=O)NCCN(C(c2cn(CC)nc2)=O)C)CC(C(F)(F)F)=NO1 59613,N1(C(C(C)n2cncn2)=O)CCCC(NC(c2cc3ccsc3[nH]2)=O)CC1 59614,Cc1ccc(NC(N2CCN(c3nccc(SC(F)F)n3)CC2)=O)c(C)c1C 59615,Cc1c(C(=O)NC(C)CN(C)C(C2(O)CCSCC2)=O)sc2[nH]cnc(=O)c12 59616,N1(C(c2c(C)coc2C)=O)CCC(NC(c2cnn(C)c2C(F)(F)F)=O)C(F)C1 59617,c1(CC(=O)NCC(CCOC)NC(C2(O)CC(CF)C2)=O)cccc(Cl)c1F 59618,c1(CC(=O)N(CC(CC)NC(=O)CCOC)CC)cc(=O)n(-c2ccccn2)[nH]1 59619,C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)CCC[SH]=CC2CC2)CC1n1cccn1 59620,N1(C(CSC)=O)C(CNC(c2c[nH]nc2C2CCOCC2)=O)CC2CCCC12 59621,CCC(C(=O)NCC1(C2(O)CN(C(=O)CC3(O)CCCC3)C2)CC1)C(C)(F)F 59622,n12ccc(n1)-n1cc(nn1)CC2C.C(C(=O)O)OC(F)F 59623,c1(C(N(CCO)Cc2ccc(CC)cc2)=O)ccc(O)c(C)c1C 59624,O=C1NC(CSc2ccc(C(=O)Nn3cncn3)cc2)C(=O)N1c1ccon1 59625,C=C1CCCN(C(=O)CCN(CC(N)C(C)C)CCOC)C1 59626,N1(C(C(CC=C)(F)F)=O)CC2(CC(NC(c3c[nH]c(=NC)o3)=O)c3nccn32)C1 59627,CCC(C)(COC)C(=O)NCCC1(NC(=O)C(N)=O)CC1 59628,C1(F)(CNC(c2cc(C(F)F)no2)=O)CCCN(C(c2ccccc2Br)=O)C1 59629,N1(C(C(C)N(C(C(C)OCCOC)=O)C)=O)CC(F)(COC)C1 59630,Cc1cc(CCN2CCCCC2c2ccc(C(F)(F)F)cc2)c(C)s1 59631,N(C(=NCCc1ccc(F)cc1C)NN1CCN(C(=O)NC2CC2)CC1)C(C)C 59632,C(CCC(C)C(=O)NC1CC(CN(C)C(C2CCC(=O)N(C(C)C)C2)=O)C1)OC 59633,N1(C(c2c(C)cc(CC)o2)=O)C2CCC1C(CNC(=O)CC1CCC(=O)N1C)C2 59634,c1(CCCC(=O)NCC2CN(C(C3C(=C)C3)=O)C2)cc(F)ccc1F 59635,O=C(CCc1ccccc1F)NNC(=O)C(F)(F)c1c(Cl)cccc1Cl 59636,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)C2CCCC1CN(C(=O)C=C1CCC1)C2 59637,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 59638,c1(NC(C2CC(NC)C2)C)cc(Br)ccc1S(=O)(=O)N1CCSC(C)(C)C1 59639,c1(C(N2CC3C(C2)N3C(=O)Cn2nc(O)ccc2=O)=O)ncc(Br)cc1Cl 59640,O=CN1CCCC1C(N1CCC(CCNC(=O)CCc2cnc(O)[nH]2)C1)=O 59641,c1(C(=O)O)nc2c(F)cccc2s1.c12ccc(cc1)-n1nc(C3CC3)nc1C2C.C 59642,Cc1ccc2ncnc(NC3CN(C(c4ncccc4C)=O)CC3C)c2c1 59643,c1(C(N2CCCC(N(C(=O)Cc3n[nH]c(=N)s3)C)CC2)=O)cnc2[nH]cncc1-2 59644,C1(NC(CC2C(C)C2)=O)(CNC(=O)CCCOC(C)=O)CCCC1 59645,N1(C(c2nc(COCC)oc2)=O)C2CCC(C(=O)Nc3csnc3C)C1CC2 59646,C(=O)(C(O)CC(F)(F)F)N1C(C(N(C2CCCCC2)CC)=O)C(CC)CC1 59647,c1(CN=c2c3ccc(OCC)cc3nc[nH]2)cccc2c1CCN(C(C)=O)C2 59648,Cc1nc(-c2ccccn2)sc1C(=O)NCCC1CN(C(C2(C)COC2)=O)C1 59649,c1(CCCC(=O)NCC(c2n(C)ncc2)CCO)ccc2c(c1)C=CCCC2 59650,CN1CCN(C(C2CCN2C(=O)Nc2ncccc2F)=O)C(c2ccccc2)C1 59651,C12(NC(C(C)Oc3cccnc3)=O)CCC(CC1CNC(=O)COCCF)C2 59652,c1(CNC(C(F)OC)=O)ccccc1CNC(=O)Cn1ccnc1C 59653,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 59654,c1(CN2CCC(C(C(=O)NCCCC(OC)OC)C)CC2)c(C)ccc(C)c1O 59655,C(CNC(C1CC1c1ccn(C)n1)=O)(CC(C)C)NC(c1nc(OCC)sn1)=O 59656,CC(C(=O)Nc1ccc(NC(=O)NC2(CC(C)(C)C)CCC2)cn1)S(N)(=O)=O 59657,c1(C(=O)NC2CC(CCNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 59658,C(=O)(CCC(C)(C)NC(C12CC1CN(C(c1snc(C)c1N)=O)C2)=O)OC 59659,C1(CC=CCNC(C(=O)Nc2ccc(C)cc2)=O)COC2(COC2)C1 59660,C1(N(C)C(C2CCC3CCCCN23)=O)CC2CCC(C1)N2c1nnc(CO)s1 59661,CC1CN(C(c2ncc(Cl)cc2F)=O)CC(C)C1NC(c1cnc[nH]1)=O 59662,N1(C(=O)COCC2CC2)CC2CCC1(CO)C2 59663,N1(C(CS(=O)(=O)NC)=O)CCC2CCN(C(=O)CN3CCN(CC)CC3)CC2C1 59664,CC1(C)OCCN(C(=O)CCc2ccco2)C1c1nc(-c2ccncc2Cl)no1 59665,Cc1cc(=NCc2nnc(CCO)s2)[nH]c(NC2CCCC2C)n1 59666,Cc1nc(C(=O)NCC(CNC(=O)C(C)C(F)(F)F)CO)ccc1[N+](=O)[O-] 59667,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 59668,c1(CC(=O)NC2(C3N(C(Cc4nc(C)sc4)=O)CCC3)CC2)cc(F)cc(F)c1 59669,c1(C(=O)NCC(C)NC(C23CCC2C3)=O)ccccc1C(F)F 59670,C12(CC(N3CC(COC)(CNC(C4CCCC(C)C4)=O)C3)=O)CCC(CC1)CC2 59671,c1(C(N(CC(CNC(C(C)=C2CCC2)=O)O)C)=O)cnc2nc(C)ccc2c1O 59672,c1(NC(C(C2CC2c2ccco2)N(C)CCC2CC2)=O)cncn1C 59673,C1(C(=O)NCC2CC(NC(c3cc(OC)ns3)=O)C2)C(C)(C)C1(F)F 59674,CN1CC2CC1CN2C(C1CSCCN1C(=O)C(C)(C)c1ccccc1)=O 59675,C1(CC(=O)N(CC(C)C#N)CCOC)CC2(CCC2)CO1 59676,C1(C(N2CC(OC)C2)=O)(CSC)CN(C(=O)CC2C(CC3CC3)C2(F)F)C1 59677,C12(CC(=O)N(c3cccc(C)c3)CC)CCC1CN(C(c1sc(F)cc1C)=O)C2 59678,C(=O)(C1(C)CCn2ccnc21)NCCN(C(CCCCC=C)=O)CCC 59679,C(=O)(CC(C)C(F)(F)F)NC1(C(N2CC(CC)C(O)C2)=O)CC(CO)C1 59680,C(CCF)(C(=O)NCCCOC(F)(F)F)NC(=O)C=C1CCOCC1 59681,C1(F)(CNC(c2ccon2)=O)COCCN(C(c2ccc(Cl)s2)=O)C1 59682,N1(C(C(C)CC(F)F)=O)CC2(CCCC2NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 59683,c1(C(C)C)scnc1C(=O)N(CC(O)CN(C)C(c1nccn1C)=O)C 59684,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCCN1C(C)C)=O 59685,c1(C(=O)NCC(C2CCC2)NC(C(C)OC(C)=O)=O)ccc(OC)cc1F 59686,n1(CC(=O)OCC2CC2)cc(OCOC)nn1 59687,Cc1ccc(C(N2CC(F)CC2C(N2CCN(C3COC3)CC2)=O)=O)nc1C 59688,c1(CC(=O)NCCC2(CNC(C(C)S(N)(=O)=O)=O)CC2)cccc2c1OCC2 59689,C(=O)(C1=C(F)CN(C(=O)CC(O)C(C)C)CC1)NCC(COC)O 59690,c1(C(=O)NCCC(=C)CNC(=O)C(O)C2CCCC2)cc(OC)c(OC)cc1N 59691,S(=O)(=O)(c1cnn(C2CCCCO2)c1)NCC(=O)OCC1CC1 59692,N1(S(Cc2cccc(C)c2)(=O)=O)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 59693,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 59694,c1(C(=O)NCC(CNC(C(N2CCOC2=O)C)=O)F)nc(O)nc(O)c1F 59695,c1(C(C)C)nccc(=NCC2(NC(c3csc(O)n3)=O)CCCC2)[nH]1 59696,N1(C(C2(F)CCN(Cc3cncc(N(C)C)c3)C2)=O)CCc2ccc(O)cc2C1 59697,C(=O)(C(CCF)NC(C1CC(C)=NO1)=O)NC(COC(C)=O)CO 59698,N1(C(c2ccc(CC)cc2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 59699,CC1(C)CCCC1(C)NC(c1cnc(CNC(C2COC3COC23)=O)nc1)=O 59700,c1(C(N2C(CC(=O)NC(C#N)C(N)=O)CCC2)=O)nc[nH]c1[N+](=O)[O-] 59701,c1(Nc2scc(-c3ccc(CO)o3)n2)cc(Cl)cc(Cl)n1 59702,c1(C(CC)O)nc(CCn2ccnc2)n(-c2cccnc2)n1 59703,C1(C(N2CC(NC(CC3(CCN(C)C)CCCC3)=O)C2)=O)(NC(C)=O)CCCSC1 59704,c1(N2CCCC(CC)(CO)C2)nc(=NC)nc(NC2COCC2C2CC2)[nH]1 59705,N1(C(c2[nH]cc(C#N)c2)=O)CCC2CCN(C(c3nncs3)=O)C2C1 59706,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCC(NC(c2ccc(COC)[nH]2)=O)CC1 59707,C(C)(C(N=c1nc(C2CCCCC2)[nH]s1)C(C)C)NC(C(CC)OC)=O 59708,c1(OC)cc(C(=O)NC2CCC(NC(c3ccn(C)c3)=O)CC2)c2c(c1)CCO2 59709,c1(C(N2C(CNC(C3C(COC)C3)=O)C=CC2)=O)cncc(Cl)c1C 59710,N1(C(CC(C)NC(=O)COc2ccccn2)=O)CC2(C1)OC1(C)CC2(N(C)C)C1 59711,C1(NC(C2C(OCC)C2)=O)CCC(C)N(c2ncc(Br)c(C(=O)NC)n2)C1 59712,N1(C(C2(CC)CCCO2)=O)CCC(C)(C)CC1C(=O)N(CC(C)C(C)(C)C)C 59713,C=CCCCCCCN(C(=O)C(C)CNC(c1ncn2c1CCC2)=O)C 59714,C(=O)(C(CC)CCCCC)N1CCC(C(=O)NC(C#C)CC2CCCC2)C1C 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59876,c1(C(N(CCNC(C(C2CCOC2)SC)=O)C2CC2)=O)ccc(C2CC2)nc1O 59877,C1(NC(C2(N(C(C(C)Cn3ccnc3)=O)C)CC2)=O)CC2(C1)CC2(F)F 59878,CCCCCCC(F)C(=O)NCCC1(O)CN(C(=O)CC(C)(O)C2CC2)C1 59879,CC(CO)C(C)N=c1nc(N2CCN(CCCC#N)CC2)c2c([nH]1)COC2 59880,CC1(F)CC2(CN(C(=O)C(CNC(=O)CC3CCSC3)C(C)(C)C)C2)C1 59881,C1(C(N(C(CC)C(=O)OC(C)CSc2ccccc2)C)=O)CC2COCC2C1 59882,C1(CNC(C(=O)NCC(C)SCC)=O)CC2(CCNC2)CO1 59883,N1(C(C2CCC(COC)C2)=O)CCC(CNC(c2cc(C)sc2C)=O)C12CC2 59884,Cc1cc(NCC2CCN(S(C)(=O)=O)CC2)nc(C)c1C#N 59885,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(c1c[nH]c(=N)s1)=O)C2 59886,C1(N(C(=O)C(C)SC)CC)CCCN(C(c2n[nH]c(CC)c2C)=O)C1 59887,c1(C(=O)NCCN2CCCC(N)CC2)c(F)ccc(I)c1Cl 59888,C(CCCOC)(C(=O)NCC(C)(C)C(C)(C)C)NC(C(C1CC1)OCC)=O 59889,CCCC(C)(C)CNC(=O)CC1CC1CNC(=O)CCc1ccc[nH]1 59890,C(CCCNC(C1(C2CCCC2)CCC1)=O)NC(=O)Cc1ccon1 59891,c1(C(=O)NC2CC(C)N(C(c3n[nH]c4c3CSCC4)=O)C2)ccc(S(C)=O)cc1 59892,c1(CNC(=O)NC(c2ccccc2)C#C)c(OC)cc(OC)cc1Br 59893,c1(CNC(C(N2C(C)C(C)(C)CC2)=O)=O)n[nH]c2cc(Br)ccc12 59894,n1(CC)cc(C(=O)NCCCNC(c2cc(Cl)ccc2OC(F)F)=O)ccc1=O 59895,CC1(C)CC(C(=O)NCC(C)(O)CNC(C2CCS(=O)CC2)=O)CNC1=O 59896,S(=O)(=O)(c1cn(-c2ccccc2)nc1C1CNC1)NC(CCOCCOC)C 59897,N#CCN=c1nc(N2CCC(N3CCC(C(N)=O)C3)CC2)c2ncn(CC)c2[nH]1 59898,C#CCC(C)C(=O)NCCC1CCN(C(c2n[nH]c(C)c2O)=O)C1 59899,c1(C(N2CC3C(CNC(c4c(C)n[nH]c4)=O)(C3)C2)=O)cnc2snc(C)c2c1 59900,N1(C(C2CCC(C(N)=O)O2)=O)CCCCC1CCNC(=O)CCOCC1(F)CC1 59901,N1(C(C2(CC(F)F)CCC2)=O)CCCC2CN(C(C3CCSCC3)=O)CC12 59902,c1(OC)ccnc(O)c1C(N1CCC(C(=O)NC2(c3ccc(F)cc3)CC2)C1)=O 59903,N1(C(C2(COC(C)C)CC2)=O)CC2CCC(C1)N2C(C1Cc2nncn2C1)=O 59904,c1(CCC(=O)N(C(C)C(=O)N(CCCCOCC)C)CCC)nccn1C 59905,O=C1CC2OCCC2(C(N2CCC3CCN(C(=O)CNC=O)C3C2)=O)CN1 59906,c1(CC(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)ccc(Br)c(C)c1 59907,CC1CCN(C(=O)CCN2CCCCCC2)C1CNC(=O)Cn1cccnc1=O 59908,c1(OC)noc(C)c1NC(=O)C(c1ccccc1)NC(=O)CC1CCCC12CC2 59909,N1(C(C)=O)CCC2(CCN(C(=O)Cc3ccco3)CC2)C1.C1CC1 59910,C(=O)(C1CCCn2cncc21)N(C)CC1(CNC(C(CCCC)F)=O)CC1 59911,C1(C)(C(=O)NC(C2CCCN2C(=O)C(C)(C)C(F)F)C)CC(C(C)C)=NO1 59912,C1(C)CCCC(=O)N1.C1(NC(CC=CCCCCC)=O)CCOC1(C)C 59913,N1(C(C)C(=O)OCCOc2ccc(Cl)cc2)Cc2ccccc2C1=O 59914,CN1CCC(C(N2CCC(CNC(c3cnc(O)n3C)=O)C2)=O)S1(=O)=O 59915,CC1(C)COC(CC(N2CCCCC2C2(NC(=O)CNC(N)=O)CC2)=O)C1 59916,N1(C(c2cn(CCNC(C(CC=C)C(C)C)=O)nn2)=O)CCC2(CNC(=O)C2)C1 59917,C1(NC(C2N(C(c3cccc(C)n3)=O)C3(CC2)CC3)=O)CCc2ncnn2C1 59918,C1(CNC(CC2CC(C(=O)OC)C2)=O)C2CN(C(=O)CC3OCCC3C)CC12 59919,C12(C(=O)NC3C(NC(c4c(N)cccn4)=O)CC3)CC(CO)(C1)OC21CCC1 59920,c12cc(n(C)c1C)C1(n3cc-2nn3)CC1.C(CCNC(=O)C1CC1)SC 59921,C(=O)(C(CO)C(C)(C)C)N1CCCC(CNC(C(C(C)C)OC)=O)CC1 59922,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)N(C1CCC1(C)C)C 59923,C1(NC(c2n(CC)ncc2Cl)=O)CN(C(c2c(Br)nnn2C)=O)CC12CC2 59924,N1(C(CC2(OC)CCCC2)=O)CCC(C2(NC(=O)CCC(C)SC)CC2)CC1 59925,N1(CCC(=O)OCC)CCN(C(=O)CCc2nnc(C(C)C)o2)CC1=O 59926,N1(C(C2OCCN(C(COC(CC)CC)=O)C2)=O)CCOC(C2CC2)(C2CC2)C1 59927,C(=O)(C(CNC(=O)C(C1CC1)C1CC1)C(C)C)NCc1oc(C)c(CO)c1 59928,c1(C(N2CC(C)(C)C(NC(=O)C(O)CF)CC2)=O)c(F)ccc2occc12 59929,N1(C(c2cc(OCC)c(Cl)cc2)=O)CC2CC(C)N(C(C3CCC4CC34)=O)C2C1 59930,C(C(CNC(=O)CSc1nc[nH]n1)C(F)(F)F)NC(C=CC1C(C)C1(Cl)Cl)=O 59931,C1(NC(c2cncc(Br)c2)=O)CC2(C1)CC(C(=O)NCc1cnco1)C2 59932,c1(C(N(CCCNC(=O)CC2CCC(=O)NC2=O)CC)=O)cc(C)cc(C)c1C 59933,N1(C(C2(CNC(C(CCC)C(C)C)=O)CCCO2)=O)CCc2nnnn2CC1 59934,C1(C(=O)NC2CCC(N(C(CC(COC)C)=O)C)CC2)Cc2ccccc2S1 59935,c1(OC)cc(Cl)c(C(=O)NC(C)CCCNC(=O)CCCCCN(C)C)cc1Cl 59936,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC(NC(c1cc(SC(F)(F)F)c[nH]1)=O)C2 59937,C(C(COC)CC(=O)N1CCC(CC(=O)NC(C)CS(C)=O)C1)OC 59938,c1(C(=O)NC(C(C)(C)NC(CCNC(=O)OCC)=O)C)cc(C#N)ccc1N 59939,c1(NC(C2CC(F)CN(C(c3sccc3I)=O)C2)=O)cnc2ccc(F)cn12 59940,CCC(C(=O)OC)C(=O)N1CC(CO)(CNC(c2csnc2OC)=O)C1 59941,c1(CC)ccc(C(=O)NC(C)C(C)(C)NC(=O)COCC2CCCC2)[nH]1 59942,c1(C(=O)Nc2ccc(C)nc2)cc2c(nc1N)CCC2 59943,C1(CC(=O)NC(C)CCNC(=O)CCn2ccnn2)C2CC3CC(C2)CC1C3 59944,C1(CNC(c2scc(C)c2Cl)=O)CN(C)CCN1C(=O)C(C)OCCN(C)C 59945,N1(C(COC2(C#C)COC2)=O)CC2CC1CN2C(=O)C(C1CCS(=O)(=O)CC1)(C)C 59946,C(C)(C(=O)NCCN(C(=O)CN(C)C(C)C)C1CC1)NC(=O)OC 59947,C1(OC)C2CC3CC1CC(C(=O)NC1(C)CN(C(=O)C(O)C4CC4)C1)(C3)C2 59948,c1(C(N2CCC(C(C)NC(=O)C3=CCOC3)C2)=O)cnc(O)c(F)c1 59949,C#CC1(C(N2CCN(C(C)C)CC2CCO)=O)CCCCC1.C1(=O)C(C)CN1 59950,C1(N(C(=O)C(O)CC2CC2)C)CCN(C(=O)C(C)(C)c2ccccn2)CC1 59951,c1(OC)cnnc(C(=O)NC(c2ccccc2)C=Cc2ccccc2)c1 59952,c1(C(=O)NCC2(NC(CCC)=O)CC2)cn(CC(F)(F)F)nc1C 59953,C1(CCCN2C(c3ccc(C)o3)CCCC2)NC(=O)CN(C)C1=O 59954,N1(C(CCN(C(C)=O)C)=O)Cc2[nH]nc(C(=O)NCc3cocn3)c2C1 59955,N1(C(C(C=C)(C)C)=O)CCC2(CC1)OCCC2NC(C1CCN(CCF)CC1)=O 59956,N1(C(CCOCCN(C(=O)Cn2ncccc2=O)C)=O)CC2OC(=O)N(C)C2C1 59957,N1(C(C(C)Cc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 59958,N1(C(CC2CN(C(c3cc(C(C)C)[nH]n3)=O)C(C)C2)=O)CCC(C)(C2CC2)C1 59959,CCC(C)CCC(=O)NCC12CC(CO1)N(C(=O)CCC1(C)CC1(F)F)C2 59960,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 59961,Cc1cc(Cl)cc(C(=O)NCC2CN(C(c3ncc(Cl)cc3Cl)=O)C2)c1N 59962,C(=O)(C(C)CS(C)(=O)=O)NCCC1CCN(C(C2C(CC(C)C)C2)=O)C1 59963,c1(C(N2CCCC(NC(CCC#CC)=O)C2)=O)ccc(C#N)c(C)n1 59964,C(C)(C(O)C(=O)NC1CCC1CNC(=O)C(C)(C)Oc1ccccc1)SC 59965,c1(CCCCn2cc(-c3cccc(OC)c3OC)nn2)cc(Cl)c(Br)cc1F 59966,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccnn2CC(C)C)=O)CC1 59967,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(c1cocn1)=O 59968,C1(C(=O)NCC(CNC(c2c(CC)scc2)=O)(C)C)CCC(N(C)C)CC1 59969,C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C)C(C)NC(c1cnc2[nH]ncc2c1)=O 59970,c1(OCCC)cccc(C(=O)OC(c2cnsn2)C)c1 59971,C1(C(=O)NC(c2ccnn2C)C(=O)N(C)CC2(CC(C)C)CC2)CCCN1C=O 59972,c1(C(=O)NC(C(C)NC(c2csc(CO)n2)=O)C)ccccc1Br 59973,C(CCCN(C(C1C(C(=O)OCC)C1)=O)CC)NC(=O)C=CC(C)(C)C 59974,C(=O)(CC(C)(C)CC(F)F)NC1CC2N(C(C3N(C)C(=O)CC3)=O)C(CC2)C1 59975,N1(C(c2cn(CCOC)nc2)=O)CC(C)(C)OC2(CCOC2)C1 59976,C1(C(=O)OC)CN(C(=O)OC(C)(C)C)CCO1.CCC(C(=O)N)N1CCCC1 59977,c1(C(C)NC(CC)COc2cccnn2)cc(C(F)(F)F)ccc1Cl 59978,Cc1ncc(C(=O)NCC2CCCC2NC(C2C3CNC(=O)C23)=O)cc1C#N 59979,C1(N(C(C(CC#C)C2CC2)=O)C2CCN(C(=O)CCC(C)(C)F)C2)CC2(CCCO2)C1 59980,C(=O)CC(C(F)(F)F)P(C)(C)=O.C(=O)(C(C)(C)C1CCCN1Cc1ccccc1)OC 59981,N1(C(CS(=O)(=O)NC)=O)CC2CCCC(NC(=O)C(O)C3CCCC3)C2C1 59982,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 59983,CS(=O)(=O)c1cccc(-c2nc(NCCS(=O)(=O)N3CCOCC3)cs2)c1 59984,C1(CNC(C(F)OC)=O)C2CC2CN1C(c1cncc(Cl)c1)=O 59985,c1(OC)ccc(O)c(NC(=O)CCC2CCCN2C(=O)CCCC(=O)N(C)C)c1 59986,C1(CC)C(C(=O)NCCN(C)CCOC)CCN1C(=O)CCc1cccnc1C 59987,c1(OC)cc(F)c(Br)cc1C(=O)NCC=Cc1cc(Cc2ccccc2)ns1 59988,Cc1c(C(N2CC(O)(SCC(N3CC(C(N)=O)C3)=O)C2)=O)ccn1C 59989,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2occc2Cl)=O)C(C2CC2)C1 59990,CC1CCN(CCC(=O)NC2CC2C2CCCN2C(=O)CSCC(F)(F)F)CC1 59991,C1(C)(C(N2CCC(COCC)C2)=O)CCCN1C(=O)C(C)C(C)C 59992,C=CCN=C(NCC(=C)Cl)NCc1csc(CC)n1.C1CO1 59993,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(=O)CC1CCC(C)C1 59994,C(=O)(C1=C(C2CC2)N(CC(F)F)C(=S)NC1c1cn2ccsc2n1)OC 59995,c1(C(N(CCNC(C(C(CC)O)C)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 59996,c1(C(N2CC(CNC(c3cncc(C)c3)=O)C(C)(C)C2)=O)cccc2occc12 59997,N1(C(C2C(C)(CC)C2)=O)CC2CCC(NC(=O)Cc3cncnc3O)CC2C1 59998,C=CC1(CC(=O)N(C2CCC(O)CC2)C)CN(C(C2CC2CC(C)C)=O)C1 59999,C(N=c1nc2sccc2c(NCCF)[nH]1)C1C(c2ccn(C)n2)CC1 60000,Nc1c(C(=O)NCCC2CN(C(c3cc(Cl)ns3)=O)C2)nc(O)nc1O 60001,C1(C(=O)NCC(C)N(C)C(C2NC(=O)CC2C)=O)CCC(c2ccccc2)CC1 60002,Cc1c(C=CC(N2CCC(C)C(NC(=O)CS(=O)(=O)N3CCCC3)C2)=O)cnn1C 60003,c1(CCC(C(=O)OC)NC(CC)C2CCC2)ccc(Cl)c(F)c1 60004,c1(CC)[nH]nc(C(=O)NC2CCCCCC2NC(=O)CC(C)C)c1[N+](=O)[O-] 60005,C1CCN(C)OCC(NC)COCC(C2CC(C)CC(=O)N2)C(=O)N1 60006,CN1CCN(C(c2cnc[nH]2)=O)CC1C(=O)NC(C)(C)CF 60007,c1(CCC(=O)NC(C(C)NC(c2cnoc2C2CC2)=O)CO)ccc(CO)cc1 60008,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60009,C1(C)(C(=O)NCCC(COC)OC)CC(O)CN1C(C1CC(=O)N(C)C1)=O 60010,CCC(Cc1ccccc1)CC(=O)NCC1(O)CCN(C(=O)C(O)CSC)CC1 60011,C1(C(N(C2CN(C(=O)CN3CCSCC3)C2)C)=O)SCCCS1 60012,C(=O)(CC(C)(C)C(=O)NC1CCC(CCC(=O)N(CC(C)O)CC(C)O)C1)OC 60013,c1(OC)cccc(NC(C2CN(Cc3ccc(I)cc3)CC2F)=O)c1C 60014,c1(C(N(CC(=O)NC2CCOC2)CC2CC2)=O)coc(C(=O)O)c1 60015,N1(C(C2OCC3CCCCC23)=O)CCC2(CCN(C(c3cncc(O)c3)=O)C2)C1 60016,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1cn(CC(N)=O)nn1)=O)F 60017,c1(C(=O)NCCN(CCO)CC)ccc(C(=O)NC)cc1 60018,C1(C(=O)NC2CN(C(c3cncc(C)c3)=O)CC2O)CCC2(CCC2)CC1 60019,C1(NC(C2CN(C)CC2O)=O)CC2(CCN(c3ccc([N+](=O)[O-])c(O)n3)CC2)C1 60020,C=CCCCC(C)N(C)C(C1(N(C(=O)C=CCOC)C)CC1)=O 60021,C(C(C)(C)CNC(=O)CC(C)N(C)C(C)=O)N(C(C(c1ccccc1)OC)=O)C 60022,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60023,C12(NC(Cc3cc(=N)[nH]cc3)=O)CCCC1CN(C(c1c(O)cc(Cl)cc1F)=O)C2 60024,c1(CC(=O)NC2(CCCC(=O)N(CC(CCC)C)C)CC2)ccc(F)cc1 60025,N12CC(CC(O)C1)C2=O.n1(CONC(c2ccc(CCC)[nH]2)=O)nc(C)cc1C 60026,c1(C(N(CC(C)N(C(=O)CC(C)C(F)F)C)C)=O)ccc2c(c1)CCC2 60027,N1(C(C2N(OC)CCC2)=O)CCC2(CC1)OCCC2NC(C1CCCN1N=O)=O 60028,c1(NC(c2scc(CNC(C3CCCCC(=O)N3)=O)c2)=O)cccc2c1CCO2 60029,c1(C(=O)NCCCC(C)NC(CC2(C=C)CCCCC2)=O)coc(S(N)(=O)=O)c1 60030,C12CCCCCCN1C(=O)C1CCN1C2=O.C12OCCC1NC2=O.CC.OC 60031,c1(C(=O)NCC(C(C)C)NC(CCCC(=C)C)=O)nn(C)c2c1CSCC2 60032,c1(CNC(C2CC(F)CN(C(c3ccc(I)c(Cl)c3)=O)C2)=O)cccc(F)c1Cl 60033,C(C(=O)NCCNC(C1(F)CC1)=O)(C(C)C)OC 60034,CC(C)CCC(=O)NC1CCC(N(C(=O)COCc2nc(C3CC3)no2)C)C1 60035,CC1(CNC(=O)CCC(N)=O)CCN(C(=O)C(c2ccccc2)O)C1 60036,c1(C(N2CCCC(NC(C(C)OCCC=C)=O)C2CC)=O)cnc2n1CCCC2 60037,c1(CC(=O)N(CCCNC(=O)CS(=O)(=O)N(C)C)C)ccc2nc[nH]c2c1 60038,N1(C(c2cc(C)ncc2)=O)CC(C)CCC1CNC(=O)Cc1ccccc1Cl 60039,C(=O)(CS(C)(=O)=O)NCC1CC(CN(C)C(c2ccon2)=O)C1 60040,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60041,CN1N=C(CC(=O)NC2CC(CNC(=O)C=C3CCC(C)(C)CC3)C2)CC1=O 60042,c1(CC)ccc(C(=O)C(=O)N(CC(O)CNC(C2(c3ccno3)CC2)=O)C)s1 60043,C1(C(=O)NCCCN(C(=O)CCOCC(F)(F)C(F)(F)F)C)CC2(CCC2O)C1 60044,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2C2CCCC2)=O)C1C 60045,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60046,C1(NC(C(CCC)CNC(=O)CCCNC(N)=O)=O)C2CCCCCCC12 60047,Nc1cnc(C(=O)NCC(c2ccccc2)SC2CCC2)cn1.C12CC1NC2=O 60048,c1(NC(C2C(NC(C(CO)N(C)C)=O)C3CCC2C3)=O)ccc2nn[nH]c2c1 60049,c1(C(N2CC(OCCNC(c3cc(CCC)n(C)n3)=O)C2)=O)cnc(N)c(Cl)c1 60050,C(C1C(C(=O)NCCOC2(C(N3CC(OC)C3)=O)CSC2)C1(C)C)=C(C)C 60051,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60052,C(=O)(CCN(C(=O)COCCS)C)NCCSC.C1CC1 60053,N12CC(CC1(C)C)C2C.c1(-n2cc(CCN(C)C)nn2)cccc(C(C)(C)C)c1 60054,C(=O)(CC(C(F)(F)F)n1ccnc1)NCCC(C)NC(c1ncc(F)cc1F)=O 60055,C=CCC(CNC(c1ccnn1CC)=O)C(=O)N1CC(CCC)C1C(C)C 60056,c1(CC)ncc(C(N2C(CNC(c3cccn3CC)=O)CC3CC23)=O)c(C)n1 60057,Cc1cn2cc(C(=O)NC3CC4(NC(=O)C(O)C(F)(F)F)COC3C4)ccc2n1 60058,c1(CCNC(=NC)NCC2CC(OC(C)(C)C)C2)nccnc1C 60059,c1(C(N(CCNC(C(C)N2CCC2)=O)CCN(C)C)=O)cnn2ccncc12 60060,C(c1ccsc1)=CC(=O)NCC1CC(=C2CC2)C1.C1=CCNC1=O 60061,CC=C=CCCN=c1nc(SCCCC(C)O)c2ncccc2[nH]1 60062,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc2c(N(C)C)cccc2s1 60063,c1(CNC(c2c(C)nc(-c3nn[nH]n3)s2)=O)nc2ccsc2s1 60064,N1(C(CN(C(C)C)C)=O)CCCC(O)(NC(=O)COC2CCCC2)CC1 60065,c1(NC(C2C(C(=O)Nc3cnc(OC)nc3C)C2)=O)ccc2ccccc2c1O 60066,c1(C(=O)NC2CN(C(C3(CO)CC3(F)F)=O)C2)nc(OCC(F)(F)F)ccc1Cl 60067,CCCC(C)CCNC(C1(C(C)NC(=O)C(O)CCN(C)C)CC1)=O 60068,c1(C(=O)NC(CCCNC(Cc2cc(C)on2)=O)(C)C)cc(O)nc(O)c1 60069,N#CC1(C(=O)NCc2ccoc2)CCC1.C12CC(C1)C(=O)N(C1CC1)CC2 60070,c1(Nc2c(Br)cnc(C(C)C)n2)ccc(S(N)(=O)=O)c(F)c1 60071,CS(=O)(=O)CCCNC(=O)CC1(NC(c2cc(N3CCCC3)ccn2)=O)CCC1 60072,N1(C(c2cc(C)sc2C)=O)CC(F)(F)CC1C(=O)NC1(C)CCCC1(C)C 60073,C1(CC(=O)NCC(C)(C2CC2)NC(C(C)C2(O)CCC2)=O)CCC=CCC1 60074,c1(N(C)CC2CCC2)nc(=NC2COCC2C2CC2)[nH]c2c1CSC2 60075,c1(C(N(CCNC(=O)Cn2cc(Cl)c(O)nc2=O)CC)=O)cn2nccc2nc1C 60076,N1(C(C2(CSCC)CC2)=O)CCC2(CC1)C(N(C(=O)CCS(C)=O)C)CS2(=O)=O 60077,C1(CCNC(CC(C)C)=O)CC2CCC(C1)N2C(c1ccc(C(C)O)cc1)=O 60078,c1(Cn2ncc(SC(N3CCC(CCC)C3)=O)c2)cn2nc(C)sc2n1 60079,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)Cc2c(C)n[nH]c2C)C(CO)CC1 60080,S(=O)(=O)(c1ccc(Br)cc1C(=O)O)NCCCc1cc(C)c(F)c(C)c1 60081,CC(C)(C)C(=O)C(=O)NCC1CCC(CC(=O)NCCCCCCF)CC1 60082,C1(NC(C2CCOC2)=O)CCC2CN(C(=O)C(O)C(F)(F)F)CC12 60083,C1(COC(C2(C)CC(F)C2)=O)CCCN(CC(=O)NCc2ccccc2)C1 60084,c1(CCC(=O)NC2(C(=O)Nc3ccc(C)cc3O)CC2)ccc2ccn(C)c2c1 60085,C1(CC(N2CC(OC)(CO)C2)=O)CNC2(CC2)CO1 60086,c1(COC)ncc(C(N2CCC(C(C)NC(=O)CC3CC=CCC3)C2)=O)s1 60087,N1(C(C(C)O)=O)CCc2[nH]nc(C(=O)NC(C3CC3)C3CC3)c2C1 60088,S(=O)(=O)(c1csc(Cl)c1)Nc1cccc(-c2onc(CN(C)C)n2)c1 60089,C(=O)(CCC(C)C)NCC(CCOC)NC(C1(CCF)CC1)=O 60090,CC(C)C(CCC(=O)N1CC2CC(C1)C2(C)C)NC(=O)CCCC(=O)N(C)C 60091,C(CS(=O)(=O)CC(=O)N1CCC1CNC(=O)CCCC(C)(C)C#N)OC 60092,CC1(N2CCCCC2)CCN(C(=NCCF)NCC2=CCCNC2)C1 60093,N1(C(c2ccc(OCC=C)cc2)=O)CCN(C(C2CC(O)C2)=O)CC1C 60094,C12(C(=O)NCC3(C(C)(C)O)CC3)CCC(CC1)N(C(c1ccn3ccccc13)=O)C2 60095,C(CC(=O)NC1CC(NC(=O)C(=O)C2CC2)C1)OCC.C(C)(C)(C)O 60096,CC(C(=O)NC1CC(OCCO)C1)n1cccc1.C12CC1C(=O)N2C1CC1 60097,N1(C(C2OCCC(NC(c3c(C)con3)=O)C2)=O)CCc2c(C#N)cccc21 60098,C1([SH2]CCSC(C)C)CCC(C)(C)CC1 60099,c1(CC)cc(C(N2CCC(NC(=O)CCc3nc(O)n[nH]3)CC2C)=O)cc(C)c1 60100,C1(CN(C(=O)CN2CCCCCC2)C)CCCN(C(c2ccoc2C(F)(F)F)=O)C1 60101,N1(C(C(C)N(C(c2cc[nH]n2)=O)C2CC2)=O)CC2(C1)CC(C)(C)C2 60102,c1(C(=O)NC(C2COCCN2C(=O)C(c2ccccc2Cl)C)C)cccc(F)c1Cl 60103,n1(CC)ncc(NC(=O)NC2CC(F)(COC)C2)c1CC 60104,CC1CC(NC(C2CC(C)(NC(c3cn4ccnc4s3)=O)C2)=O)CC(C)(C)C1 60105,N1(C(C2C(NC(C(Cc3ccccc3)OC)=O)C2)=O)CCOC(CN(C)C)C1 60106,C(=O)(NN1CCN(Cc2ccc(Cl)cc2)CC1)c1c(C)n[nH]c1C 60107,N12CCC(C(F)C1)C(=O)N(C)C1(CC1)C2=O.c1(CC(C)C)cnn(C2CC2)c1C 60108,c1(OC)csc(C(=O)N(C(CC)C(=O)N2CC(N3CCOCC3)C2)C)c1 60109,c1(C(=O)NC(C2CCCN(C(Cc3c(C)nsc3)=O)C2)C)cc[nH]c2nccc1-2 60110,C1(C(C2CCCC2)NC(CNC(c2c(C)nc[nH]2)=O)C2CC2)CCCC(=O)N1C 60111,c1(C(=O)NCC2CC(NC(c3cccc(OC)c3)=O)C2)ccc2c[nH]nc2n1 60112,N1(C2CN(C(C3C(NC(c4ccns4)=O)COC3)=O)C2)CCCOCC1 60113,C(=O)(C#CC(C)C)NCC(CCOC)NC(=O)C(c1cccc(F)c1)C(C)C 60114,c1(C(N(C)CC2N(C(CC(C(C)C)O)=O)CCC2)=O)ccn2ccnc2c1 60115,N1(C(COCC#C)=O)CC2C(NC(=O)C=CC(=O)N(C)OCCCC=O)C2C1 60116,c1(N(C(c2cn(C)nn2)C(=O)NCC=CCNC(N)=O)C)ccccc1F 60117,c1(C(=O)NCC(C(C)C)NC(=O)CC2CCOCC2)c(C)oc2ncnc(O)c12 60118,C1(N2C(SCCCNC(C3=C(C)CCCC3)=O)CCC2)C2CC3CC(C2)CC1C3 60119,c1(C(=O)NCC(C)NC(=O)CC2CCC(=O)NC2)cc(Cl)nn1C 60120,C(=O)(C1CC(=O)N(C)c2ccccc21)NCCCCCNC(CC(C(C)C)O)=O 60121,c1(C(=O)N(c2cncn2C(C)C)CCNC(C(CC)OC)=O)cccc(C)c1 60122,c1(C(N(CCCCCC)CCNC(=O)C(C)c2cccs2)=O)ncc(N)cc1Cl 60123,c1(CNC(C(C(C)C)NC(C(CSC)O)=O)=O)cc(F)ccc1F 60124,C1(CNC(C2CCC(C)(C)C2)=O)CC(F)(F)CN1C(C1C2(CC2)C12CC2)=O 60125,C(=O)(C(C(C)CC)NC(=O)C(CC1CC1)OC)N(CC(CCC)C)C 60126,C(=O)(C(CC(C)C)NC(=O)C(C1CCCC(C)C1)N(CC(F)(F)Br)C)OC 60127,C1(C(=O)NCC23CC(CO2)C3)C2CCCC2CN1C(=O)CCCN1CCCC1 60128,Cc1cc(=O)c(NC(C2CCN(C(=O)C(=O)NC3CC3)C23CC3)=O)c(C)[nH]1 60129,c1(C(=O)OC)cccc(C#CCNC2CCC2c2cc(Cl)sc2Cl)c1 60130,C1(CNC(=O)OC(C)(C)C)CCN(c2cccc(CN(C)C)n2)C(C)(C)C1 60131,C1(C(=O)NCC(CNC(c2cc3[nH]ccc3s2)=O)O)Cc2cccnc2C1 60132,CCC(CNC(c1conc1C(C)NC(C1CCSC1)=O)=O)CC(C)C 60133,C1(C(N2C(CN(C(=O)CN(c3ccncc3)C)C)CCC2)=O)CN2CCN1C(C)C2 60134,CCCC(C(=O)N1CCC(CC(=O)NC)C1)NC(=O)COCC(=O)OC 60135,CC(=O)CCCC(=O)NCC12CC(CN1C1CC1)C2.c1(C)cc(C)c(C=O)o1 60136,c1(C(N(CC(=O)OC)CCO)=O)ccc(F)c(-c2c[nH]c(=NC)s2)c1 60137,N1(C(c2cccc(CSC)c2)C(=O)NCC)CCCC(C(=O)OC)C1 60138,c1(C(=O)NC2CCC(NC(c3nccc(OC)c3)=O)CC2)noc2c1CCCC2 60139,c1(SC)cccnc1C(=O)NC1CCCC1NC(C1C=CCCC1)=O 60140,c1(CO)c[nH]c2cccc(F)c12.c1(COC)nc(C2c3nnnn3CCN2)cs1 60141,c1(OCCOC)cc(Br)ccc1NC1COCCC1C(F)F 60142,N1(C(c2cc(C)nnc2)=O)CCOc2c(C(=O)N(C)C)cccc21 60143,S(=O)(=O)(c1ccc(F)cc1F)N(C1CC2CC1CN2)C(c1cc(C(C)C)no1)=O 60144,c1(CC)noc(CC(=O)NC(C)CCN(C)C(C2(C)CCCS2)=O)n1 60145,c1(C(=O)NC2CCC(CNC(CCc3nc(C)sc3)=O)C2)ncnc2sccc12 60146,C1(SC)CCC(NC(=O)CO)C1.C12(CC1)C(=O)NC2 60147,CCC(C)C(C)(O)CNC(C1CCCC1CNC(c1cncc(O)c1)=O)=O 60148,CC(C)C(CCCC(=O)N1CC(O)CC12CCC2)NC(C1CC(=O)C12CCC2)=O 60149,N1(C(CC(C)(C)N(C(C(=O)N(C)C)=O)C)=O)CCC2(CC=CCO2)C1 60150,c1(C(N(CC(C)(C)NC(C2=CCCCC2C)=O)C)=O)cnc2ncnn2n1 60151,C(CN=c1c(C#N)c[nH]c2ccc(C)cc12)N(C(C1(CC#C)CC=CCC1)=O)C 60152,C(N=c1[nH]nc(CC(=O)NC2CC2c2ccccc2)s1)C1CC(C2CC(=O)NC2)C1 60153,c1(C(N2CC(C)(NC(C(CC)CSC)=O)C2)=O)ccc2c(c1)CCN(C)C2.CC#N 60154,c1(C(N2C(C)CC(NC(c3ccc(NC)cc3)=O)C2)=O)ccc(P(C)(C)=O)s1 60155,C1(CC)CN(Cc2nncnc2O)CCN1C(=O)Cc1ccccc1C(=O)O 60156,C1(NC(CSCCCC)=O)CC2CN(C(=O)Cn3nnc(C)c3N)CC2C1 60157,c1(OC(C)C)ccc(NC(=O)NCC(Cc2ccccc2)N(C)C)cc1 60158,CCCC(C)(C)CC(=O)NC(CCC)C(=O)N1CCC1C(N)=O 60159,C1(CC)(CNC(C2(NC(c3cc(OC)no3)=O)CC(O)C2)=O)CCOC1 60160,c1(CC)cc(C)nc(N2CCCC2CN(C)C(C2(C3CC3)CCCO2)=O)n1 60161,CC1(C(=O)NCC2C(CO)CCN2C(=O)CN2CCSCC2)CCCCC1 60162,C(=O)(C(C)(CO)NC(=O)CN1CCNC1=O)N(C)Cc1ccoc1 60163,C1(NC(=O)NC)CC(C)(C)CN1C(=O)CCn1cc(-c2cnc(C)n2C)nn1 60164,C(C(C)(C)CNC(c1ncoc1C(C)(C)C)=O)N(C)C(c1coc(O)n1)=O 60165,CC1C2CCCCC2CN1C(=O)C(CC1CC1)NC(C1CCC(=O)O1)=O 60166,c1(CSCCC(=O)NCCC2CCN(C(CC(=O)NCC)=O)C2)ccc(F)cc1 60167,N1(C(Cc2ccc(C#C)cc2)=O)CCC2C(CCCN2C(c2cn(C)nn2)=O)C1 60168,C=CC1(C(=O)N(C)Cc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60169,CC1(C#CC(=O)NC2CC3CCC2N3C(=O)CCC2CCCCC2)CC1 60170,C1(C(=O)NC2CCN(C(C)=O)CC2)CCC2(CN(C(=O)C(O)C(C)C)C2)O1 60171,C1(NC(Cc2c(C)non2)=O)CN(C(C23CC2COC3(C)C)=O)C2(CCC2)C1 60172,c1(C(=O)NC(C2CCCN(C(=O)C(C)(C)C(=O)N(C)C)C2)C)nccc(Cl)c1C 60173,CCC(C)CC(C)C(=O)NC(Cn1cncn1)C(=O)Nc1cc(CO)cc(C)c1 60174,CC(CC(=O)NCCCOC1CC1)NC(C1SCCS1)=O 60175,C=CCC(CC(=O)N1CCC(NC(=O)C(C)OCC2CC2)CC1)OC 60176,C1(N(C(=O)CC2COCCO2)CCF)CCCN(C(C2CC(=C(F)F)C2)=O)C1 60177,CC(CC(=O)NC(C1CCOCC1)C(N1CC=CC(O)C1)=O)C(F)(F)F 60178,C(CCCCC(=O)NCC1CC(OC)CN1C(c1cn(C)nc1COC)=O)OC 60179,c1(C(N2C(CNC(=O)CCc3ccncn3)CCC2)=O)nc(Cl)ccc1Cl 60180,C1(C(=O)NCCCCCCNC(=O)C(O)c2ccsc2)C2CC3C(C2=O)C13 60181,CC1(C)CCCN(C(C2CCO2)=O)C1C(=O)NC1(n2cnnn2)CC1 60182,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60183,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60184,CC#CCCCC(C)NCCCSc1conc1C 60185,c1(OC)ccc(F)c(C(=O)NCCC(C)NC(C2CC(=O)N(OC)C2)=O)c1N 60186,C(C(C)C(C)C(=O)N1CCCC1CCNC(=O)CCN(C)C(C)=O)OC.C(C)(C)(C)O 60187,CC1CC(C(=O)NOC(=O)C(C)NC=O)CCO1 60188,Cn1cc(C(C(=O)NCCC2(CO)CC2)NC(C2(Cl)CCC2)=O)cn1 60189,C1(NC(C2CCC(C)C2)=O)CCOC12CCN(C(=O)COC(=O)CO)CC2 60190,C1(C(=O)NC2(CC=C)CCCCC2)CC(C)CN(C(=O)Cc2ccc(O)cn2)C1 60191,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60192,C1(C(=O)NCCC2CCN(C(C(c3n(C)ccn3)(F)F)=O)C2)CCC(F)(F)CC1 60193,N1(C(c2cn(CCC=C)nn2)=O)CCN(CC(C)NC(c2n[nH]cc2Cl)=O)CC1 60194,CCC(C)(CN(C(=O)CN1CC2CC2C1)CC)C(=O)N1OC2CCC1CC2 60195,C#CC1CCN(C(=O)CC2COCCN2C(=O)C(C)OCC=C)CC1 60196,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2CO)CCC(O)CC1 60197,c1(C(=O)NCC2CCCCN2C(=O)C2=NOCC2)n[nH]c2cc(Br)ccc12 60198,c1(C(=O)NC2CC3CN(c4ncc(C#N)nc4)CC32)nnn2c1COCC2 60199,C12(NC(CC(COC)NC(=O)Cn3nc(C)nc3C)=O)CCC(C1)OC2C 60200,C1(NC(CNC(CC)=O)=O)(CO)CCN(C(C2CC2C(C)(C)C)=O)CC1 60201,C=Cc1cccc(CN2CCCC(C(N3CCCC3c3ccccc3)=O)C2)c1 60202,C1(NC(CCC#C)=O)CN(C(c2cc(C)cc(Br)c2OC)=O)CC1N=[N+]=[N-] 60203,c1(C(=O)NCC2N(S(CC(=O)OCC)(=O)=O)CCOC2)ccc(OC)c(Br)c1 60204,CCCCC(O)C(C)C(=O)N1CCC(C(=O)NCCc2nncn2C)(OC)C1 60205,c1(C(=O)NCCN(C)C(C2CC2C(C)(F)F)=O)cnc(C2CC2)nc1 60206,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCCn1cncn1 60207,c1(C(N(C)CC2N(C(c3c(C)[nH]cc3)=O)CCC2)=O)cccc(=S)n1O 60208,c1(OC)ccccc1C(N1CCCC(CCNC(=O)CC(O)CN(C)C)C1)=O 60209,Nc1cccnc1S(=O)(=O)NCC1CCC2(CC2)C1 60210,c1(C(N2CC3C(NC(C(C(C)(C)C)OC)=O)C3C2)=O)cccc2cc(F)ccc12 60211,c1(C(N2CC(C)C(NC(=O)CN3CC4CC4C3)C2)=O)cc(N)c(Br)c(F)c1 60212,N1(C(C2C(SC)CCC2)=O)CC2CCC(CNC(C3CCCN(C)C3)=O)(C2)C1 60213,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2)=O 60214,C1(N(C)C(c2ncc(Cl)cc2F)=O)CC2CCC(C1)N2C(=O)C(=O)N=S(C)(C)=O 60215,CN1CCNC(=O)C12CCCN(C(c1cnc3ccc(Cl)nn13)=O)C2 60216,C1(C(=O)NCC2(CO)CCCC2)CC2(CCC2)CN1C(c1ccnc(O)c1F)=O 60217,C(c1ccc(C)cc1)=C(C(N1CCC(CCNC(C(CCC)OC)=O)C1)=O)C 60218,C1(NC(=O)CC2CC3C=CC2C3)CC2CC1N(C(C1CCCCC1)=O)C2 60219,c1(C(N2C(C(N3CCCC(CCC)C3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60220,C1(OC)CCC2(C(=O)N(CCCCC(=O)N(C)Cc3cnco3)C)CC12 60221,Cc1cc(Br)cnc1CNC(N1CCC(C(F)(F)F)C1)=O.C(CCF)N 60222,C(CN=c1nc2c(cnn2C)c(NCC2CCN(C)C2=O)[nH]1)N(CC)CC 60223,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2[nH]1 60224,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60225,C(CCC(O)C(=O)NC1CCN(C)C1(C)C)NC(C(CCC)NC(C)=O)=O 60226,N1(C(c2c(C)cc(C)[nH]2)=O)CCC2(NC(=O)Cc3ccncc3C)CCCCC12 60227,N1(C(C(C)(C)OC)=O)CC2CCN(C(c3sccc3F)=O)CC2C1 60228,Cc1cnc(C)c(C(N2CC3(NC(c4ccc(F)cc4F)=O)CC2C3)=O)c1 60229,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60230,N1(C(C)=O)CCCC(C(=O)NC(C)(CNC(C2(C)CCOCC2)=O)C(C)C)C1 60231,c1(SC)cc(C)c(C(=O)NCc2nc(CNC(=O)CC3(C)CC3(F)Cl)cs2)s1 60232,C(=O)(C(C)C(C)(C)C)N(C1(CC(=O)NC(C#C)C(C)OC)CC1)C 60233,c1(CCNC(N(C)CC2(O)CCOC2)=O)ncc(C(C)(C)O)cn1 60234,c1(OC)cnc(Cl)nc1N1CCCC(C(C)NC(c2cnn(C)c2C2CC2)=O)C1 60235,C1(NC(=O)Cc2cc[nH]n2)COC2CN(C(=O)C(C3CCOCC3)F)CC12 60236,c1(-c2cc(CCN(C)C)on2)nc(C2CCCCC2)nn1CCS(C)(=O)=O 60237,c1(OC)ccc(CCCN(C(=O)CC2CCCC2)C)cc1.n1(C=O)cc(C)nn1 60238,Cc1ncnc(C)c1C(=O)NCCCN(C(=O)C1=NOC(C(C)(C)C)C1)C 60239,C1(C(=O)NCC(C)(C)OCCNC(C2CCCOCC2)=O)(OC)CCS(=O)(=O)C1 60240,c1(-c2nc(-c3[nH]cc(C)n3)nn2C(C)C)cc(N(C)C)nc(Cl)c1 60241,N12CCC(C1C(C)C)C(=O)NC1(CC1)CC2=O.C(COC)OC 60242,N1(C(C2CC(OC)C2)=O)CC2OCCN(C(c3cc4c(cc3N)CCC4)=O)C2C1 60243,N1(C(c2csc(Cl)n2)=O)CCCC2C1CCCN2C(c1cc(=O)cc(Cl)[nH]1)=O 60244,C1(C(=O)Nc2c(Cl)nc(N(C)C)n2C)CCC2(CCN(C(C)(C)C)C2)O1 60245,C(C(C(=O)NC1CC(C)(NC(=O)C=Cc2ccc[nH]2)C1)OS(C)(=O)=O)OC 60246,c1(OC)cncc(C(=O)NCC2CCC2NC(C2CC2CCOC)=O)c1C 60247,C1(NC(=O)CN2CC3CC3C2)CC2CN(C(=O)CNC(=O)CO)CC12 60248,c1(NC)ccc(C(=O)NC2CCCCC2NC(=O)C=CC2(C)COC2)nc1 60249,C(CC)(CC)(CCO)NC(CCC1(C)CN(C(c2n(CC#C)ccc2)=O)C1)=O 60250,c1(C(N2C(C)CCC(NC(CN(C(C)=O)C)=O)C2)=O)c[nH]c2c(C#N)cccc12 60251,C12(NC(C(Cc3c(C)n[nH]c3C)C)=O)CCCC(CN(C(=O)C#CC3CC3)C1)C2 60252,CCC(C)(F)C(=O)N1CC(CCCCNC(=O)CCSc2ccccc2NC)C1 60253,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC2CCN(C)C2=O)C1 60254,C12C3CCCC3N1C(=O)C2.O=C1CCC(NC(=O)CCCn2cccn2)CN1 60255,c1(-c2cccc(CC)c2)ncc(F)c(NC(Cc2cc(OC)cc(Br)c2)=O)n1 60256,Cc1ccc2[nH]c(C)c(CN=c3cc(NC)nc[nH]3)c2c1.c1(S)ccccc1 60257,N1(C(c2ccc(CCC)s2)=O)CCC(C)(CNC(=O)CC2COCC2O)C1 60258,CCC(C)C(O)C(C)C(=O)N1CCC(C(N2CCC3(CCSC3)C2)=O)(C(C)C)C1 60259,C1(NC(CCOCCSC)=O)CN(C(c2snc(C)c2N)=O)CC1O 60260,C1(C(N2CC(COC)(NC(C3CCCCO3)=O)C2)=O)CCC(=O)N(C2CC2)C1 60261,C1(NC(C(C=C)CC)=O)CN(C(=O)CNC(=O)CCC)CC1C1CC1 60262,Cc1c(C(=O)NCC2CCCCC2NC(=O)OC(C)(C)C)cccc1O 60263,c1(CC(=O)NCCn2cc(NC(=O)CC3C=CCC3)cn2)cncnc1 60264,N1(C(c2nnc(C)s2)=O)CCN(C(C2Cc3cscc3C2)=O)C(C)C1 60265,N1(C(c2cccc(C)c2)=O)CC2CC(NC(=O)CCN(C)C(C)=O)C2C1 60266,N1(C(C(C)O)=O)CCC2CN(C(c3ccncc3N)=O)CC12 60267,c1(NC(CN(C(=O)C(=O)N(C)C)CC)C)ccc(C(=O)OC)cc1[N+](=O)[O-] 60268,C(C(COC)CC(=O)NCC(C1CCOC1)NC(c1sc(C)nc1C)=O)OC 60269,C=CCC(C)(C)CNC(=O)CC1CCCC1NC(=O)C(c1cccnc1)O 60270,N1(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC(NC(C2C3CC4C(C3)C24)=O)C2(CCCC2)C1 60271,C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(F)(CNC(C23CC(C)C2C3)=O)C1 60272,N1(C(CC2CC(C)(O)C2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60273,N1(C(c2scc(OC)c2)=O)CCCC1C=CC(=O)NCC1(O)CCOC1C 60274,c1(C(=O)NC(C(C)NC(C2=C(C)CCC2)=O)C(C)C)ccc2nc(O)[nH]c2n1 60275,c1(C(=O)NCCC2COCCN2C(=O)COCC2CC2)nccc2n[nH]cc12 60276,c1(CC(N2CC(F)(CNC(C3(COC)CCCO3)=O)C2)=O)cc(C)ccc1OC 60277,N1(C(C(c2cccc(F)c2)C)=O)CC2(C1)CN(C(c1csc(Cl)c1)=O)CC2CO 60278,C1(NC(C(C)NC(=O)NC)=O)CCC(O)CN(C(c2cn(C)c(O)n2)=O)C1 60279,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2ccc(N)cc2NC)=O)CC(C)(C)C1 60280,Cc1nc(O)c(C(=O)NC2CCC(NC(c3ccsn3)=O)CC2)nc1C 60281,N1(C(C2C(C(C)O)C2)=O)CCOC(CCNC(=O)COCP(C)(C)=O)C1 60282,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60283,C1(O)(C(C)NC(C(c2cncnc2)C)=O)CCN(C(c2nnn(C)c2N)=O)CC1 60284,c1(C(N2C(CCCNC(CSC)=O)CCC2)=O)ccc(F)cc1N 60285,CN1CC=C(CC(=O)NCC(C2CC2)N(C)C(C23CCCC2OCC3)=O)CC1 60286,c1(C(N(C2CC2)CC2CCN(C(C=CC(=O)OCC)=O)C2)=O)cn2c(n1)SCC2 60287,N1(SCNC(C(C)C)Cc2ccc(Cl)cc2)CCCCC1C#N 60288,C12CCCN(CC1)C2=O.C1(N(C)C)(CNC(C2C(=C)C2)=O)CCCC1 60289,C(N=c1nc(C)[nH]s1)C1CC(NC(C(CC)F)=O)C1 60290,N1(C(c2ccc(Cl)cc2)=O)CCC(C(=O)NCC2(SC3(O)CC3)CC2)C12CC2 60291,c1(C(N2CCC(CCN(C(CCC(=C)Br)=O)C)CC2)=O)ccc(C)c(CO)c1 60292,c1(C(C)OCCC(c2nnnn2C2(C)CC2)NCCC(C)C)ccccc1F 60293,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)N(C(c2ccc(F)cn2)=O)CC1C 60294,C1(C(=O)N(CCN(C(C(C)N(C(C)=O)C)=O)C(C)C)C(C)C)CC(S(C)(=O)=O)C1 60295,C1(OC)(CNC(=O)C=CC2CCOC2)CN(C(=O)CCOCCN(C)C)C1 60296,c1(CC)c(C(N2CCCC(NC(=O)CN(C)C(C)=O)C2)=O)oc2ccccc12 60297,c1(C(=O)NCC2(O)CCCN(C(C3C(C=C)OCC3)=O)C2)cc2ccccn2c1 60298,c1(CC)[nH]nc(C(=O)N(C)CC2CCCCN2C(=O)CCC2OCCO2)c1C 60299,C(CN=c1[nH]c(N2CCN(C)C(C3CC3)C2)nc2c1CSC2)N1C(C)CCCC1 60300,C1(CC)CN(C(c2cc(C)c(C)s2)=O)CC1C(=O)NC(c1cccs1)C 60301,CC(CC(F)F)C(=O)N1CC(C(N)=O)(CNC(=O)CC2CC2c2ccccc2)C1 60302,N1(C(C(C)(C2CC2)OC)=O)C(CNC(c2ccoc2Cl)=O)CC2COCC12 60303,CON1CCC(CC(=O)NC(C(C)NC(=O)CCNC(=O)C=CCl)C(C)C)CC1 60304,Cc1ccnc(O)c1C(N1CCN(C2CN(C(c3c[nH]c(=N)s3)=O)C2)CC1)=O 60305,C1(NC(C(=O)NC(c2ccc(N(C)C)cc2)C)CO)CNc2ccccc2C1 60306,n1(C(C)C(=O)NC2CCSC23CN(C(=O)Cc2ccsc2)C3)cnc2ccccc12 60307,C1(CNC(CCSCC)=O)CC2CCC(C1)N2C(=O)CCOC1CCCCC1 60308,C1(CNC(CC=C=C)=O)CN(C(c2cnc(C)[nH]c2=N)=O)C2(CCC2)C1 60309,Cc1nn(CC(N2CCC(NC(C3C=CCCC3)=O)C(C)C2)=O)c2ncccc12 60310,c1(C(=O)NCCNC(C2CCC(=O)NC2)=O)coc2c(F)c(Cl)ccc12 60311,c1(NC(=O)NC2CN(C(CCC3(C)CCC(=O)N3)=O)C2)ccc(F)c2cccnc12 60312,c1(CNC(c2ccc(CO)s2)=O)cnn2c1CN(c1ncnn3cccc13)CC2 60313,C1(CN(CCOC)C(=O)Nc2ncsc2-c2ccccn2)CCCCO1 60314,n1(CCC(=O)NC(CC)CN(C)C(C2CC2C(N)=O)=O)ncc2c1CCCC2 60315,N1(C(C(C)NC(COC)=O)=O)CCN(C)CC1CNC(c1scnc1C)=O 60316,Cc1ccc(F)cc1C(=O)NCCCOCCNC(C12CCCC(C1)OC2)=O 60317,C1(C(=O)NCC2CCN(C)C2)CCN(C(C2C3CN(C)CC23)=O)C12CC2 60318,C(=O)(C(C#N)C(C)(C)C)N(CC(N1CCS(=O)C(C)C1)=O)CC 60319,CS(=O)CCC(=O)NC.C1(CC)CCN(C(C2CN(C(N)=O)C2)=O)C1 60320,N1(C(CC(C)(C)OC)=O)CCC2CCCC12CNC(C1(C)CC(C)C1)=O 60321,C1(CN(C(c2c(COC)noc2)=O)C)CC(F)CN1C(C1CC2CC2C1)=O 60322,Cc1cnc(C)c(C(=O)NC2(C)CCN(C(=O)CC3CCC(=O)NC3)C2)c1 60323,c1(C(=O)NC(CN(C(C(CCC)(C)C)=O)C)C)cn2cc(C)sc2n1 60324,CC1=C(C(=O)NC2CCC(CNC(C3(c4ccc(F)cc4)CC3)=O)CC2)CCO1 60325,N1(C(c2c(C)ccnc2O)=O)CC2OCC(NC(c3coc(Cl)n3)=O)C2C1 60326,CCC(COC)C(=O)NC(c1cnn(C)c1)C(=O)N(C)Cc1cccc(C)n1 60327,C(=O)(CC(CC1CC1)NC(=O)C(C1CCCC1)OC)NC(CCC)c1nn[nH]n1 60328,N1(C(C2CC23CCOC3)C(=O)NCC)CC(N(C)CC)Cc2cc(OC)ccc21 60329,c1(C(N2CCCC(C(C)NC(C3CCC4CC34)=O)C2)=O)cc(Cl)cc2c1CCC2 60330,N1(C(C(=O)NCCCSC)Cc2cnc(C(F)(F)F)s2)CCC(C)(CS(C)(=O)=O)C1 60331,c1(C(=O)NC2C(C)CN(C(=O)C#CC3CC3)C2)cc(=NS(C)(=O)=O)cc[nH]1 60332,Cc1nc(C2CCC2)ccc1-c1nc(C2CC2)nn1CC(C)C 60333,N1(C(=O)COCC2CCOCC2)CCCCC(C(=O)Nc2cncnc2O)C1 60334,N1(C(C2C(C)C2C)=O)CCC(C)C1CNC(C1CN(S(C)(=O)=O)C1)=O 60335,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)O)=O)cc([N+](=O)[O-])n[nH]1 60336,C1(NC(c2sccc2Cl)=O)CCN(C(=O)CN2CC3(CC3)CO2)C12CCCC2 60337,N1(C(C=CC)=O)CC(NC(c2cc(F)cc3nccnc23)=O)C2CCCCC12 60338,C12(CNC(CN(C)C(N)=O)=O)CCCC1CN(C(C13CCC(CC1)CC3)=O)C2 60339,N1(C(c2cc(C)c(C)[nH]2)=O)CCC(CNC(c2coc(Br)c2)=O)C12CCC2 60340,C1(C(N(C2CCCN(C(=O)CCOC3COC3)CC2)C)=O)CCN(C)C(=O)C1 60341,C1(C(=O)NCC2N(C(c3cncc(OC)n3)=O)CC=C2)(OC)CCCC(C)(C)CC1 60342,C1(c2cn(C)nc2)CN(C(=O)C(C)(F)F)CC1NC(=O)CN1CCSCC1 60343,N1(C(C(C)C2CCC2)=O)CCC(F)(CNC(=O)COCCCF)C1 60344,c1(CN(CC)N)c(Cl)ccc(F)c1O 60345,CCC(C(=O)NC(C1CN(C(=O)CC2COC(C)(C)C2)CCO1)C)C(C)C 60346,C1(S(C)(=O)=O)(C(=O)NCCC2(O)CCN(C(C(=O)NC(C)C)=O)C2)CCOCC1 60347,c1(SCC(=O)NCCN(C(=O)CCc2nc[nH]n2)C)ccc(F)cc1 60348,C12(C(=O)NC(CCC)CNC(=O)COCC(=O)OC)CC(CO)(CCO1)C2 60349,C1(C)(NC(CCN(C(C2C(C)C2C)=O)CC2CC2)=O)CS(=O)(=O)C1 60350,N1(C(C(CC(=O)NCC)C)=O)CC(NC(c2cn(C)nc2OC)=O)C2(CCC2)C1 60351,O=C(C1=CS(=O)CCC1)NC(CNC(c1ncncc1Cl)=O)CC(F)(F)F 60352,C1(COC)(NC(c2ccc(Cl)cn2)=O)CCN(C(C2CCCC(F)C2)=O)CC1 60353,n1(CC)cnc2c(NCC(C(C)(C)C)NC3CC3)[nH]c(=NC3CC3CCF)nc12 60354,C1(C2(O)CCCOC2)(CNCc2cc(C)c(F)c(C)c2)CC1 60355,C(=O)(C(C(C)C)n1ccnc1)NC1CCC(N(C(COCC(=C)C)=O)C)C1 60356,CC1(C)CC(NC(c2cc(=O)cc[nH]2)=O)CN1C(C1CC12CCSCC2)=O 60357,CC1CCSC1C(N1CC(CNC(c2cnn(C3CCCC3)c2)=O)C1)=O 60358,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60359,C1(C(=O)NCC(C)N(C)C(c2coc(N(C)C)n2)=O)COC2COCC2O1 60360,N1(C(C=CC(=O)N(C)C)=O)CCC(CC(=O)NCC2CCSC2)C1C 60361,N1(C(c2n(CC#C)ccc2)=O)CC(F)(F)CC1CNC(=O)C(COC)OCC 60362,C1(N(CCC)C)CCN(C(=O)C(C)NC(c2ccnc(OC)c2)=O)CC1 60363,c1(CC2(C(N(CCC)CCNC(C3CCSC3)=O)=O)CC2)ccccc1F 60364,N1(C(C(c2cccs2)NC(Cc2c(C)nccc2)=O)=O)CC(=O)N2CCCC2C1 60365,C1(CNC(c2cc(C(=O)OC)on2)=O)CN(C(c2ccn(C(F)F)n2)=O)CCO1 60366,c1(N2CC(SC)(CNC(=O)NCCSc3ccccc3)C2)cc(C)nc(C)n1 60367,N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)C=CC2CCOC2)CC1 60368,n1(CC(F)F)nnnc1C(c1ccccn1)NCC(C)(C)SC 60369,CC(CCCNC(=O)CCc1ccncn1)NC(C1CC(O)C1)=O 60370,c1(N(CC(N2CC(CNC(=O)OC(C)(C)C)C2)=O)C)ccc(C#N)cc1F 60371,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(C)c2)[nH]c2c1CSC2 60372,C1(C(=O)NC23C(CN(C(C(C4CCC4)OCC)=O)C2)C3)CCOC(=O)CC1 60373,O=S1CCC(NC(C2=CCSC2)c2nnnn2CC(F)F)C1 60374,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60375,C12CCCCN1C2.c1(OC)ocnc1C(N1CCCC1C(N)=O)=O 60376,Cc1ccc(C=CC(N2CCC(NC(=O)COc3cccc(Cl)c3C)C2)=O)cn1 60377,N1(C(C2CCC(C)O2)=O)CCCC2(NC(c3ccc(Cl)nc3Cl)=O)CC2C1 60378,Cc1ccc(OCCCC(=O)N(C)CCNC(=O)C(C)N2CCC2)cc1 60379,c1(C(=O)NC2CN(C(CCC(=O)NCC)=O)C2)c[nH]c2c(CC)cccc12.C(C)C 60380,c1(C(N2CC(CCNC(C=NOC)=O)C2)=O)ccc(C(N)=O)cc1 60381,CC1(C)CC(NC(C2SC3C=CC2CC3)=O)CN1C(=O)CCCNS(C)(=O)=O 60382,N1(CC(N2CC(C3N(C(CC(C)OC)=O)CCC3)(O)C2)=O)C(=O)CN(C)C1=O 60383,CCCCCCN(C(=O)C(n1ccc(C)n1)C)CCN(C(C1CCCC1C)=O)CC 60384,Cc1cc(N(C2(c3nnnn3C)COC2)Cc2ccc(S(C)(=O)=O)s2)cc(C)c1F 60385,c1(C(N2CCC([N+](C(=O)CC(C)F)([O-])C(=C3CC3)C)C2)=O)sc(Cl)c(Cl)c1C 60386,C1(C(=O)NC(CCNC(C(c2ccc(C)cc2)=O)=O)C)CC12CCSCC2 60387,c1(C(=O)NC2CC3CC(NC(=O)C=Cc4ccsc4)C3C2)c[nH]c2ccc(Cl)cc12 60388,c1(C(N2CCCC(CCNC(CC3OCC(C)(C)C3)=O)C2)=O)cc(Cl)ccc1Cl 60389,c1(C(N2CC(CNC(C=CC)=O)C2)=O)cnn(CC2CCCC2)c1 60390,C(CCC(=O)NC1CCC(N(C)C(c2sccc2C)=O)C1)N(C(C)=O)C 60391,C(=O)(C#CC1(C)CC1)N(C1CCC(C(=O)Nc2cn(C)nc2C2CC2)C1)C 60392,CCCCCC(C)CC(=O)OC.C(=O)(C(C)(C)n1cc(Cn2cc(C)cn2)nn1)NCC 60393,Cc1cc(C(C)NC(N2CCCCC2CCSc2ccccn2)=O)sc1C 60394,c1(C2(C)CN2c2cn[nH]c2)ccc(Br)cn1.C1(CN(C)C)CCCO1 60395,c1(CCCC(=O)NC2C(OC)CN(C(c3cnoc3C)=O)C2)ccc(F)c(F)c1 60396,c1(CNC(C2(C)N(C(CCCCOCCC=C)=O)C2)=O)ccc2ncccc2c1 60397,c1(CNC(c2n(CC#C)ccc2)=O)ccc(CNC(=O)CNC(=O)C(C)C)cc1F 60398,CC1=C(C)CC(C(=O)N(C2(CC(N3CCCC(C)C3CO)=O)CC2)C)CC1 60399,C1(C(=O)NC(CN(C(=O)C(C)n2cnnn2)CC)C)CCC(=O)N1C 60400,CCC(F)(F)CC(=O)NCc1c[nH]nc1C(=O)NCC1CC2CC2C1 60401,C1(NC(CSCC)=O)CC2CN(C(c3cc4cc(C)sc4[nH]3)=O)CC2C1 60402,N1(C(C2CC(C)N(C)C2)=O)CCC(NC(c2ccncc2)=O)C(O)C1 60403,CC1(C)C(C(N2CC3C=CC2CC3)=O)CCN1C(=O)CN1CCOCC1 60404,C1(CC)CN(C(c2cnc(Cl)cc2I)=O)CCN1Cc1ccnc(OC)c1 60405,c1(C(=O)NC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)C)cc2nc[nH]c2cc1F 60406,CC1(C(=O)NC2CN(C(C3C4CC5C(C4=O)C35)=O)CC23CC3)CC2CCC1CC2 60407,N1(C(C2C(C(=O)Nc3c(OC)nc(Br)cc3)CCC2)=O)CCc2ncncc2C1 60408,c1(-c2ccc(NC(C)=O)s2)cccc(NCC2C=CS(=O)(=O)C2)c1 60409,c1(OC)cc(CCC(N2CC(O)(CCNC(C3(Cl)CC3)=O)C2)=O)ccc1F 60410,N1(C(=O)Cc2cc(F)ccc2Cl)CCN(C(=O)C2=CS(=O)CCC2)C2(CC2)C1 60411,c1(OC)cc(C(N2CCN(C(=O)CC34CC(C3)C4)C3CC23)=O)c(O)c(Br)c1 60412,CN1CCC(C)(C(=O)N(C)CC2CCN(C(C3(CO)CCC3)=O)C2)CC1 60413,N1(CCN(C(=O)OC)CC)CCC(C)C(NC(=O)C(c2cnn(C)c2)C)C1C 60414,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CCOC2(C1)CN(C(=O)C(O)C1CC1)C2 60415,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1CC(C(=O)CCN1CCCC1)=O 60416,C(N=c1[nH]c2c(c(=NC3CN(C(C)(C)C)C3)[nH]1)COCC2)C1(N(C)C)CCCC1 60417,C1(C(C)CO)CCCCN1C(c1coc(CNC(c2ccc(C(F)F)o2)=O)c1)=O 60418,C1(NC(C(C)Cc2ccccn2)=O)CC2CC1N(C(=O)Cc1csnn1)C2 60419,N1(C(c2c(C(CC)C)cccc2)=O)CC2CCCCC2(C#N)C1 60420,CCCC(C(O)C(=O)NC1CCN(C2CC2)C1)NC(C1(n2cccc2)CC1)=O 60421,c1(C(=O)NC)ccc(S(C)(=O)=NC(=O)c2cc(C)n(C(C)C)n2)cc1 60422,C(C1c2ccccc2CN1C(C1C2CCC(F)C12)=O)NC(COCCC#C)=O 60423,N(C1CCCn2ncnc21)C(C(C)N(C(=O)CC(C)C(F)(F)F)CCC)=O 60424,Cc1nc(C(=O)NC2CC(NC(C3CCCN3C3CCCCC3)=O)C2)cc(O)n1 60425,C=CCCCC(C(=O)NC1(C)CC2(CC2)C1)NC(=O)C(F)C(C)C 60426,C1(NC(CC2C(C)C2)=O)CCCC12CN(c1nc(Cl)ncc1Cl)C2 60427,C1(C)(C(=O)NCCc2cc(C(N(CCC)CC)=O)no2)C=CCCC1 60428,N1(C(C(=O)NCC)=O)CCC2(CCN(C(c3cccnc3OCC)=O)C2)C1 60429,c1(C(=O)Nc2ncc(Br)cc2I)cc2c(s1)CCN(C(c1cc(Cl)ccn1)=O)C2 60430,CON1CCC(CC(=O)NCCOCCN(C)C(C2(C)CCCS2(=O)=O)=O)CC1 60431,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)CSCc1cccs1 60432,C1(CC(C)NC(c2ccc(N)cn2)=O)CCN(C(=O)Cc2cncs2)CC1 60433,CC(C)(C)C(=O)C(=O)N1CCCOC(CNC(=O)CC2CCNC2=O)C1 60434,c1(C(N2CC3(Cn4cc([N+](=O)[O-])cn4)CCC2CC3)=O)cnn2c1CCCC2 60435,c12ccccc1NC2=O.C(=O)(C(C)CNC(=O)C=CCOC)OCC 60436,c1(OC)cccc(C(N2CCC2C(=O)Nc2c[nH]nc2C)=O)c1OC(F)F 60437,N1(C(CC=C=C)=O)CCCCC1C(=O)NCC1CCCC(F)C1 60438,N1(C(Cc2nnc(C)o2)=O)CCCN(CCNC(C2CNC(=O)N2)=O)CC1 60439,CCCCC(O)C(=O)N(C1CCCCN(C(=O)CC2(n3cccn3)CC2)C1)CSC 60440,C1(C(=O)NCC(CC)NC(=O)C(C)NC(=O)NC)CCC(F)(F)C1O 60441,C1(C(N)=O)(CNC(C2C=CCC2)=O)CN(C(=O)Cc2csc(-c3ccoc3)n2)C1 60442,c1(C(N2CC(O)(C(C)NC(CN(CCC#C)C)=O)C2)=O)ccc(C(=O)CC)cc1 60443,CC1CN(C(C2CC(C)(F)C2)=O)CCC1NC(c1cc(N(C)C)cs1)=O 60444,C=CCC(C(=O)N1CCC(N(C(=O)CCC2CCOCC2)CC)CC1)C(C)C 60445,c1(CC)ccc(C(=O)NC2CN(C(=O)CC3CC(=O)NC3=O)CC2(C)C)c(O)c1 60446,N1(CC(=O)NC2CCN(C(=O)NC(c3cc(O)n(C)n3)C)C2)Cc2ccccc2C1 60447,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(NC(C2CCC(F)(F)C2)=O)C1 60448,N1(CC)CC2CCC(NC(c3ccc(CNC(C)=O)o3)=O)CC2C1.C(C)CC 60449,N1(C(CC2CN(C(C)=O)C2)=O)CC2CC(NC(=O)CC3CCC3)CC(C2)C1 60450,Cc1nn(-c2ccc(Cl)cc2)c(C)c1C(=O)NNC(=O)c1c(O)noc1C 60451,C1(CNC(c2cncc(C3CC3)c2)=O)CCCCN1C(c1cnnc(O)c1)=O 60452,c1(C(=O)NC2CCC(CNC(CCCSC)=O)C2)ncc(C)cc1F 60453,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(c1ccccc1F)=O 60454,C1(C(F)(F)F)(C(=O)OC)CCCN(CC(O)C(C)c2ccccc2)C1 60455,c1(CN=C(NC(C)C)NCc2cnsc2)cn2cc(F)ccc2n1 60456,C(=O)(CCCS(N)(=O)=O)NC(C1CN(C(C(CCCOC)C)=O)C1)C 60457,N1(C(C(C)=C2CCC2)=O)CCC2C1CCCN2C(=O)C(C)SC(F)(F)F 60458,C(=O)(CC1OCCc2ccccc21)N1CCC(OC)CC1 60459,C1(CC(=O)NCCCC(C)NC(c2cnc(N(C)C)o2)=O)SC(=N)NC1=O 60460,c1(C(=O)NC2C(NC(C(C)OCC)=O)C2)ccc2cccc([N+](=O)[O-])c2n1 60461,c1(OCC)ccc2ccccc2c1-c1cncc(C(=O)Nc2cccc(F)c2O)n1 60462,CC(C(O)CC(=O)NCC(C)(C)CNC(=O)CSc1cccs1)N(C)C 60463,c1(C(=O)NCC2CN(C(COCC)=O)C3C2C3)cnn2c1NCCC2C(F)(F)F 60464,N1(C(c2cc(C)[nH]n2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)(C)C#N)C1 60465,C1(NC(c2cccc(C(C)C)n2)=O)CCCCN(C(=O)C(=O)Nc2ncc[nH]2)C1 60466,N1(C(C2(C#N)C(C)C2)=O)CC(CNC(=O)C=CC2CC2)C(C)(C)C1 60467,N12CCC(C(C)C1)NC(=O)C1(CC1)Nc1ccccc1CC2=O.CC(C)=C1CC1 60468,c1(C(=O)OC)cnccc1C(=O)NC1CC1CNC(C1CCC(C)C1)=O 60469,C(C(COC)CC(=O)NC(CNC(=O)C(C)=CC1CC1)C(C)(C)C)OC 60470,CC1CCCc2cc(C(=O)NC3(CNC(=O)CC(=O)NC4CC4)CCOC3)nn21 60471,CC1(C2CCN(C(=O)CC3CCN(C(c4c[nH]c(C(N)=O)c4)=O)CC3)C2)CC1 60472,c1(NN2CC(CC)N(C)CC2)nc2cccnc2c(=NCC2CC23CCC3)[nH]1 60473,S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)N1C(C=O)CC(C)C1.C1(CCC(C)C)CCCN1 60474,c1(C(=O)NCC2OCC(C)N(C(=O)CCOC3CC3)C2)cnc(S(C)(=O)=O)s1 60475,c1(NC(CN(C2CCS(=O)(=O)C2)C)=O)nc(=O)n(C)[nH]1 60476,C12(NC(CSCC)=O)CCC(CC1)N(c1nc(COC)cc(C)n1)C2.C1CN1 60477,C1(C(N(C2CCCN(C(c3n[nH]c(C)c3O)=O)C2)CCO)=O)Cc2ccccc2O1 60478,C1(NC(CC(COC)NC(C2N(CCC)CCC2)=O)=O)CC2CC1CC21CC1 60479,c1(C(=O)NC2CCN(C(c3c(SC)csc3)=O)CC2C)cnn2c1CC(F)(F)C2 60480,c1(C(N(CCC(=O)NC(C2CCOCC2)CC)C2CC2)=O)ccc(C)cc1O 60481,C(N=c1ncc(I)c[nH]1)C1CC(C)N(C(=O)CCNC(=O)Nc2ccccc2)C1 60482,C(=O)(CC(C)C(C)C)NCC1(CNC(C2N(C(C)C)CCC2)=O)CCC1 60483,N1(C(CC2N(C(CCCC3C(C)C3)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60484,c1(C(=O)NCC(CC2CN(C(C(C)c3ncco3)=O)C2)(C)C)cccc(=O)n1C 60485,C(CCCC(=O)NCC(C)(O)CNC(=O)CCNC(=O)OC(C)(C)C)OC 60486,C1(NC(=O)NCc2nnc(CC)o2)(CSC)CCCCCCC1 60487,N1(C(CN(C(C(CCCC#C)C)=O)C2CCC2)=O)CCC2CCCC2CC1 60488,C1(CCC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1CC=CC1)=O 60489,C=C(C)CC1C(=O)N1.C1(C(=O)NC2C(COC(C)=O)C2C)CCCSC1C 60490,c1(CN2C(C(N3CCCC(C)(O)C3)=O)CC2)n[nH]c2ccc(F)cc12 60491,CCC(CCC(=O)N1CCCCC1CN(C(=O)CN1CC(C)(OC)C1)C)OC 60492,N1(C(c2ccn(CCNC(CC=C)=O)c2)=O)CCN(C)C(=O)C1CSC 60493,CC1CN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1NC(C1CCC(=O)N1)=O 60494,c1(CC)ccc([N+](=O)[O-])cc1C(N1CC(O)(C(C)NC(C2CC2CC)=O)C1)=O 60495,Cc1cc(C(N2CC3CC(CNC(=O)C=CCF)C3C2)=O)ccc1C#N 60496,C(CC1CCC1)(C(=O)NC(CC1CCC1)C(=O)NC(C)C(F)F)OC 60497,c1(C(N2CC3C(NC(c4cc(CC)no4)=O)C3C2)=O)cnc2ccoc2c1 60498,c1(C(C)C)nc2n(n1)CC(C(=O)NCC1(CF)CC1(F)F)CC2 60499,c1(CC)cc(C(N2CC(O)(CCNC(c3cn(CCO)nc3C)=O)C2)=O)ccn1 60500,CC1CCN(C(=S)SC(CC(C)C)C(=O)OC(=O)NC(C)(C)C)CC1 60501,CC(C)C(O)C(C(=O)O)NC(=O)Nc1cc([N+](=O)[O-])c[nH]1 60502,c1(CC)n[nH]c(=NC2CCN(C(c3cnn(C4CCCC4)c3C)=O)C(C)C2)s1 60503,N1(C(COC(=O)OCC)=O)CCN(c2ccnc(OCC(C)CS(C)=O)n2)CC1 60504,C=CCCCC(C(=O)NCCc1cc(Br)c(F)cc1F)N(C)C1CC1 60505,c1(C(=O)NCCC2(CNC(c3cn(CC)nn3)=O)CC2)ccccc1SC(C)C 60506,C1(C(=O)NCC2CC(C(=O)NCCC(O)C3CC3)C2)CCCN1C=O 60507,Cn1nnc(=NC(=O)C2(c3ccccc3C3CCOC3)CC2)[nH]1 60508,C1(C(N2CCC(N(C(c3cnc(O)n3CC)=O)CC)C2)=O)CCCCC1(C)C 60509,C1C2c3ccsc3CCN2C(=O)CN(C)C(=O)N1.C(=O)(C(C)SC)OC 60510,Cc1cc(CS(N2CCCCC2C2(O)CC2)(=O)=O)ccc1Br 60511,S(=O)(=O)(c1cc(C)cnc1NCC(O)C1CC1)NCCC=C=CC 60512,C(=O)(C(=O)CCC(C)C)N1CCC(OCC(=O)N(CCO)CC)C1 60513,C#Cc1ccnc(C(=O)NC2(C)CC(CNC(=O)CC(CN(C)C)CC)C2)c1 60514,Cc1cc(C(N2CC=CC2C(N2CC(C(=O)NC3CC3)C2)=O)=O)oc1C 60515,c1(OC)cccc(-c2cn(C3CCC(C(=O)NCC4CCC(=O)N4)C3)nn2)c1F 60516,c1(C(=O)NC2CC(NC(C(C)Cc3ccccc3Cl)=O)C2)cc2ccccc2[nH]1 60517,C=CC1(C(=O)NC(C2CCCCC2)CC)CCN(C(=O)CN2CCCC2C)CC1 60518,c1(C(N(C(CNC(c2cc(C(C)=O)on2)=O)C)C)=O)cnc2c(c1)CCOC2 60519,c1(C(C)C)cnn(C)c1CNC(N1CC(NS(N)(=O)=O)C(C)C1)=O 60520,c1(OC)c(C)csc1C(=O)NCC(C)CN(C(=O)COCCc1ccncc1)C 60521,c1(SC)cnc2[nH]cc(CC(=O)OC3CCN(C4CC(F)(F)CO4)CC3)c2c1 60522,c1(C(=O)NC(C)Cc2ccc(CNC(C3CC3Cl)=O)cc2)ccc(N)cc1F 60523,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60524,Cc1ccc(O)c(NC(c2nnnn2-c2ccccc2)CC2CCC2)c1 60525,CC1CN(C(=O)CNC(N)=O)CC1NC(c1cncc(C(C)(F)F)c1)=O 60526,CC(c1ccsc1)=CC(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 60527,C(c1cccnc1)=CC(=O)NCC1CCC(NC(=O)Cc2cc[nH]n2)C1 60528,c1(C(=O)NC2(CCNC(=O)CCn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60529,Cc1cc(C(=O)NCCC(C)NC(c2[nH]nnc2C)=O)cc(C)c1Cl 60530,C1(CNC(c2n(CC)nc(C)c2)=O)CC(F)(F)CN1C(=O)CC(C)SC 60531,C1(CNC(C(CC=C)N(C)C)=O)COCCN(C(c2ccncc2COC)=O)C1 60532,C1(CN(C)C(C2CCCN2C)=O)CCCN1C(C1(C2CCCO2)CC1)=O 60533,C1(C(=O)N(c2ccns2)C(=O)C2CC2)(CC(C2CCC2)C)CCCC1 60534,c1(C(=O)NC(C(=O)NC(C)C2CC2)C(C)(C)O)ccc2c(c1)CN(C)CC2 60535,c1(C(=O)NCC2(CN(C)C(C3CNC(=O)N3)=O)CC2)cnccc1C(F)F 60536,C#Cc1ccc(C(=O)OC)cc1.C1=CCN(CC(=O)N(C)C)C1=O 60537,c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)CC2)=O)ncnc2c(C)csc12 60538,Cc1ccc(C2CC2C(N2CCCC(NC(c3cnccc3Cl)=O)C2)=O)cc1 60539,c1(C(=O)NCC2N(C(=O)CN3CCC3)CC=C2)cccc(-n2cccn2)n1 60540,C1(C(N(C(C)C)C)=O)CC2(CCN1C(C1CCOCC1)=O)CC2 60541,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)con2)=O)C1)CCO 60542,C1(C(=O)NCCOC2CCN(C(C(C)=CC3CC3)=O)C2)CCN(CC)CC1 60543,C1(C(=O)NCCOCCN(C(C(C(C)C)O)=O)C)CN2CCN1C(C)C2 60544,C(N=c1cccc(S(=O)(=O)N(c2ccc(C)cc2)C)[nH]1)C1C(C(N)=O)CCC1 60545,N1(C(COc2cccc(C)c2F)=O)CCC2(CNC(=O)CC3CC3)CCCCC12 60546,Cc1nc(Cl)[nH]c(=NCC2C3CN(C(c4cc(Cl)sc4Cl)=O)CC23)c1F 60547,C(=O)(C(O)C(CCC)N(C(=O)C(C#N)C(C)C)C1CC1)NCC#C 60548,C12(CNC(C(CC=C)(F)F)=O)CCC(CNC(=O)CS(=O)(=O)NCC)(CC1)CO2 60549,c1(C(N2CCC(NCCNC(c3nccc(C=C)n3)=O)C2)=O)cccn2ccnc12 60550,CC(C(=O)N(C1(C(=O)NC2CC(O)C(F)C2)CC1)C)C(F)(F)F 60551,N1(C(COCC(C)(C)C)=O)CC(n2nc(-c3ccccc3)oc2=O)C(O)C1 60552,C1(NCC(CC)(CC)NC(=O)Cc2cnc[nH]2)CS(=O)(=O)CC12CCC2 60553,C12(C(N(C(C)CNC(c3ccnn3C)=O)CC)=O)CC3CC(CC(C3)O1)C2 60554,N1(C(Cc2c(C)ccnc2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60555,[N-]=[N+]=NC1CC2(C(N3CC(F)(CNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60556,N1(C(=O)CO)CCC(CN2CCN(C(c3cnoc3CC3CC3)=O)CC2)CC1 60557,C(=O)(C(C)(C)CC(C)C)NC1(CNC(C(C)SC)=O)CC1 60558,C=Cc1ccc(C(=O)N(C(CC)C(N2CC3CCC3(CO)C2)=O)C)cc1 60559,C(=O)(C1CCCn2cnnc21)NC1C2CN(C(CNC(C(C)(C)C)=O)=O)CC21 60560,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60561,Cc1nc(CC(N2CCC(CNC(=O)CCC3CSCCS3)C2)=O)cs1 60562,c1(OCC)ccc(S(=O)(=O)N(C)C)cc1C(=O)NC1CC(S(C)(=O)=O)C1 60563,Cc1cnc(C)c(NC(C2CC(F)CN(Cc3ccc(Cl)c(C(F)(F)F)c3)C2)=O)n1 60564,C1(C(N2CCCC(CC=C)C2)=O)CCN(C(c2cnc(C3CC3)o2)=O)C1(C)C 60565,N1(C(c2cc(CC)no2)=O)CC(NC(=O)Cc2cccnc2C)CC(C)(C)C1 60566,c1(OC)ccc(C(=O)NCCN(C(c2cnoc2C)=O)C(C)C)nc1Br 60567,C1(CNC(C2C(CC(C)(C)C)C2)=O)CC2(C1)CC2F 60568,C=CC(C)(O)C(=O)N(C)CC1CN(C(=O)C(c2cccc(Cl)c2)OC)CCO1 60569,N1(C(Cc2c(C)occ2)=O)CC2CCN(C(=O)CSc3ccccn3)CC12 60570,CN1CCC(NC(C23CC(CO)(CN2C(c2cncn2C)=O)C3)=O)C1(C)C 60571,CN1CCCC(CCC(N2CC=CC(NC(=O)Cn3ncnn3)C2)=O)C1 60572,c1(C(=O)NC(C)C(C2CCCCC2)NC(C2CCCOC2)=O)cnccc1N(C)C 60573,c1(C(N(C)CCN(C(=O)C(O)CC(N)=O)C)=O)cc2sc(Cl)cc2[nH]1 60574,C1(C2N(C(C3CC4(CC4)C3)=O)CCC2)CCCN(C(C23CC(F)(C2)C3)=O)C1 60575,N1(C(CCOCC(C)C)=O)CC(NC(c2cccc[n+]2[O-])=O)C2(CCC2)C1 60576,CCCCS(=O)(=O)NC(C)C(=O)NCC12CC(CN1C(=O)C(=O)N(C)C)C2 60577,c1(CN(C(C)CNS(=O)(=O)Cc2ccccc2CC)C(C)=O)cnc(Cl)cc1Cl 60578,c1(C(N(CC(C)NC(c2ccnnc2S)=O)CC)=O)cc(Br)cnc1OC 60579,N1(C(C2CN(S(C)(=O)=O)C2)=O)CC2CS(=O)(=O)CC2(NC(C2CCCCO2)=O)C1 60580,C12CC(CO1)C(=O)N2.N1(CCNC(C(C)NC(=O)OC)=O)CCCCC1 60581,c1(N2C(C)CCN(C(=O)CCC(=O)OC(C)(C)C)CC2)ncnc2ccccc12 60582,CCC(C(=O)NC1CC(CN(C(=O)C(C)N(C)C)C)C1)C(C)(C)CC 60583,C(CC(C(=O)N1CCC1(C(=O)N(C)C1CC1)CC)NC(=O)C(F)C(C)C)=CC 60584,O=C(C1=CCCO1)NCCOCCNC(=O)C(F)(F)Cc1ccccc1 60585,CC1CCC(N)CC1.c1(C=O)cn(C)nc1OC(C)(C)C.N1(C)CCN1C 60586,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1CC(C)(C)C1 60587,Cc1nc2ccccn2c1C(N1CCC2(CCC2)C(NC(=O)CC(C)C)C1)=O 60588,N1(C(CC(C)Sc2ccccc2)=O)CC2(CNC(=O)COCCF)CCC1CC2 60589,C(=O)(C(=O)N=S(C)(C)=O)NCCC1CN(C(=O)C=Cc2ccsc2)CC(C)O1 60590,c1(OCC)cc(Br)c(C(=O)N(C2CC3(CNC3)C2)C(C#N)C(N)=O)cc1OC 60591,C1(NC(=O)CC2CCC3CC23)CCCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 60592,c1(NC(=O)NCC2(C(=O)OC)CCCO2)ccc(Br)c(CO)c1C 60593,N1(C(=O)CCCF)CCCC2C1CCCN2C(=O)CSCC(F)(F)F 60594,C1(CS(=O)(=O)NCCCC2CCC2)CCS(=O)(=O)C1 60595,CCC(CC(=O)NC1CN(C(c2ccnc(OC(F)(F)F)c2)=O)C1)C(F)F 60596,N1(C(C2C(C)C2C)=O)CC(C(F)(F)F)C(CNC(=O)Cn2cc(CO)nn2)C1 60597,c1(CC(=O)NCCC(=O)NCC(CNC(C(COC)C)=O)(C)O)cccc(F)c1 60598,CCCCCC(O)CC(=O)N(C)C(c1ccc(N(C)C)nc1)=O 60599,N1(C(C(=Cc2cccs2)C)=O)CC2CC(NC(=O)Cc3cnn(C)n3)CC(C2)C1 60600,C(C(=O)NNC(=O)C(F)(F)F)c1c(OC)c(C)cc(C)c1 60601,Cc1nc(C)n(CCC(=O)NC2COCCC2NC(=O)CC(=O)N(C)C)n1 60602,N#Cc1ccc(CN2CCOCC2Cc2nn[nH]n2)cc1 60603,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 60604,c1(OC)cncc(C(N2CC3CC2CN3C(c2ccnc(C)c2Cl)=O)=O)c1C 60605,N1(C(c2sccc2F)=O)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 60606,Cc1cc(CC(=O)NCC(C)(C)CNC(c2nccn2C)=O)nn1C 60607,C(=O)(C(F)CC(C)(C)NC(c1ccccc1)=O)N1C(C)(CC)CC1 60608,C(CC(C)(C)NC(c1cnoc1-c1cnn(C)c1)=O)N(C(=O)C=CC(F)(F)F)C 60609,C1(C(N(C)CC2CN(C(=O)C(C)(F)F)CCO2)=O)CCCC(F)(F)CC1 60610,C1(NC(=O)COCCCF)CN(C(c2cnc3ncccn23)=O)C2(CCCC2)C1 60611,C(=O)(C(C)(C)C)NC(C)C(=O)NCC1(C(=O)NCc2ccsc2)CCCO1 60612,Cn1cnc2ccc(NC(c3ccc(-c4cnc(F)c(F)c4)cn3)=O)cc12 60613,c1(OC)ccc(Br)cc1C(N1CCN(C(C2(C3CC3)CC2)=O)C(C(F)(F)F)C1)=O 60614,n1(CCOC)c(SC(c2nnc(C)o2)C)nnc1-c1ccccc1 60615,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)Cn2cc(Cl)cn2)CC1O 60616,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)C)cc(C(C)C)cc(F)c1 60617,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)C=CC2CCCC2)C1 60618,c1(C(=O)NC2C(CNC(c3cn(C(C)C)nc3)=O)CC2)cccc2c1CCCC2 60619,N1(C(=O)OCc2ccccc2)CCN(CC(c2ccccc2)F)CC1 60620,C(=O)(C(C)(CC)OC)N(CCC)CCNC(=O)C(F)CC1CC1 60621,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 60622,C1(C(N2CCC(NC(C3C(C(C)C)CCO3)=O)C2)=O)CC2CC1CC2(F)F 60623,c1(OC(C)C)ccccc1CC(N1CC(N(C)C(c2cscn2)=O)C(F)C1)=O 60624,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cscn2)C1 60625,C(=O)(CC(C)C(F)F)NC1C(OC)CN(C(Cc2cccc(SC)c2)=O)C1 60626,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)CC2)=O)ccc(F)cc1C 60627,N1(SC)CCC(NC(=O)C(CC2CCCC2)NC(=O)CCC(C)OCCO)CC1 60628,C(=O)(C(O)C(F)(F)F)NCC1CC(NC(C(C)Sc2ccccc2)=O)C1 60629,CCC(CC(=O)NCc1cc[nH]c1C(=O)N(CCC(=O)OC)C)SC 60630,C1(C(N2CCC(COC)C2)=O)CCN(C(c2cscn2)=O)CC1 60631,N1(C(CNC(=O)NC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 60632,Cc1cc(CCC(=O)OC2CCCC(C(C)C)C2)ccc1F 60633,c1(OC)cc(C(=O)NC(C)(C)CN(C(=O)CCC2CCOCC2)CC)cc(C)c1 60634,c1(CC)c(C(=O)NC(C)CCCNC(c2conc2C2CCC2)=O)cccc1C 60635,C1(OC)CC(SC)CC1C(N1CCC1c1cn(CC(C)=CCO)nn1)=O 60636,C(CC(C)C)(C(=O)OCC1CCC=CO1)ONC(COC)=O 60637,CC(C)CCC(=O)NCCCN1CCN(C(C2CCOC2=O)=O)CC1 60638,CC1(CNC(=O)CCC2CCCC(=O)N2)CCC(NC(c2cnn[nH]2)=O)CC1 60639,c1(CC(=O)NCC=CC(=O)NC(C(C)C)C2(CO)CCC2)csc(Br)n1 60640,C1(CC#N)CN(C(C2CSCCS2)=O)CCN1C(c1cc[n+]([O-])cc1)=O 60641,C1(CNC(C(=O)N(C)C)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 60642,c1(OC(C(=O)NCC(CC)Cn2cc(CCC(C)(C)O)nn2)C)cccc(C)c1 60643,C1(CNC(C(C)OCC)=O)CC(C)N(C(c2cc(C(F)F)no2)=O)C1 60644,c1(OC)csc(C(=O)NC2CCC(NC(=O)CCCOC(C)(C)C)C2)c1 60645,C12(NC(CC(=C=C)C)=O)CCCCC1N(C(c1ccn3nccc3c1)=O)CC2 60646,N#Cc1sc(=NCC2CCN(C(c3cc(Cl)no3)=O)C2)[nH]c1Cl 60647,C1(NC(c2ccsn2)=O)CC2(CCN(C(c3ccc4ncoc4c3)=O)C2)C1 60648,c1(C(=O)NCC2C(CNC(=O)CC3CCC3)C2)cc(C2CC2)ncn1 60649,C(=O)(C(CCC)CCCO)N1CCOCC(NC(CCOCC#C)=O)C1 60650,c1(N2CCCC(NC(C(=O)N(CCSC)CC)=O)CC2)ccccc1[N+](=O)[O-] 60651,CC(C)C(O)C(=O)N(CCCNC(=O)CCN1CCCCCC1)C 60652,c1(C(N2CCC(CNC(C(CCC)F)=O)C2(C)C)=O)nccc2cccnc12 60653,Cc1cc(NC(c2ccc(CNC(c3c[nH]c(C#N)c3)=O)cc2)=O)c(O)cc1F 60654,C1(C(N2CCC(CCO)C2)=O)(CC)CCCN1C(=O)CC1CCCN(C)C1 60655,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(c3cnn[nH]3)=O)C2)=O)cc1 60656,Cn1cnc(C(F)(F)F)cc1=O.c12cccc(c1)SC(=O)NCC21CCC1 60657,N1(C(=O)NC2(c3ccc(C)o3)CC2)CCn2c(C)nnc2C1C 60658,C=CCC(C(=O)N(C)CCN(C(=O)CCC1CC=CC1)C)C1CC1 60659,C(=O)(CCC(C)C(=O)N1CCC(NC(=O)CCC2CCC2)C1(C)C)OCC 60660,c1(C(=O)NCC2(OC)CCN(C(=O)C=CC3CCCO3)C2)cc(C)c(C)cn1 60661,C(=O)(CCCCC(C)C)NCC(CC(=O)N(C1CCCO1)CC#C)C1CCC1 60662,N1(CC(=O)NCCCC)CCCC(N(C(c2cnn(C)c2CC)=O)CC)CC1 60663,N1(C(C2CN(C(CN(C(=O)OC)C)=O)CC2(F)F)=O)CCC2(CCOC2)CC1 60664,C(N=c1[nH]c(=NCC(C)(C)C(C)(F)F)c2[nH]ccc2[nH]1)C1C(C)(C)CCC1 60665,C(C1CCN(C(C23CCCC2CCC3)=O)CC1)=CC(=O)NC(CC#C)CC 60666,c1(N(C)Cc2nnc(C)o2)ccc(C(N2CCC(NC(=O)C=CS(C)=O)C2)=O)cc1 60667,N1(C(C(CC(CC)C)OC)=O)CC2CCCN(C(C3CC3(C)C)=O)C2C1 60668,C1(NC(N(CC(O)C(=O)OC(C)(C)C)C)=O)CCCCCCC1 60669,C1(NC(C2CN(CC)C(=O)C2)=O)CCC12CN(C(c1ccn(CCF)n1)=O)C2 60670,CC1(C)C(CNC(=O)Cn2ncnn2)CCN1C(=O)COc1ccsn1 60671,C12(NC(Cc3cnc(C)o3)=O)CCN(C(c3ccns3)=O)CC1C2 60672,c1(C(C)C)cc(C(=O)NC(=O)N(C)CCN(C)C(C2CC23CCC3)C)n(C)n1 60673,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 60674,c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(c3coc(C4CCC4)n3)=O)CC12 60675,Cc1nn(CC(F)F)c(C)c1NC(N1CCC(O)(C(F)(F)F)C1)=O 60676,CC1CN(C(=O)CNC(=O)Cc2ccccc2)CCN1C(=O)C(C)n1ccnc1 60677,c1(NC(CC(CC)NC(=O)C(C)(COC)CC)=O)ccc2nccn2c1 60678,C1(NC(C(CC#C)(C)NC(c2c[nH]c(=NC)o2)=O)=O)CC2CC1CC21CC1 60679,C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2ccnc(Cl)c2I)=O)CC1C#N 60680,N1(C(C2NC(=O)OC2C)=O)CCCCC1COCCOc1ccc(OCC)cc1 60681,N1(CC(N)=O)CCN(C(=O)C(C2C3CCC(F)C23)C2CC=CCC2)CC1 60682,C(=O)(CS(=O)(=O)C(C)C)NCCC(C(C)C)NC(C1CCCOC1)=O 60683,CC1CC(C)N(C(c2cccc3oncc23)=O)CCN1C(c1ccco1)=O 60684,N1(C(C(C=C)O)=O)CCN(C(c2c(COC)nn(C)c2Cl)=O)CC1CO 60685,C1(NC(C2CCC(C)O2)=O)CCC2CN(C(=O)C(c3ccccc3)C)CCC2C1 60686,c1(-n2ncc(C(=O)NCC3(C(N)=O)CN(C(=O)CO)C3)n2)cccc(Br)c1 60687,N1(C2CCC(NC(COCCCCC)=O)C2)CCN(C(=O)C(Cl)=CCl)CC1 60688,CC(C)CCN=C(NCCS(=O)(=O)NC(C)(C)C)NC1CCC(NC(C)(C)C)C1 60689,C1(N)CCN(C(c2cc(C3CCC3)no2)=O)CC12CCC2.C(CC(=O)C(=O)CO)N 60690,N1(C(C(C)OCCCC)=O)CC(NC(=O)Cc2cnn(C)c2CC)CC12CCC2 60691,C(=O)(C(C)S(C)(=O)=O)NCCC(=O)N(CC(C)O)CC(F)F 60692,N(C1CCCc2cc(C#N)ccc21)OCc1cc(C(=O)OCC)no1 60693,C(C(C)C(F)C(=O)NC(C)C(C)n1cccn1)NC(CC1(CC(=O)OC)CC1)=O 60694,C(C)(C)(C(C)CC(=O)NCCCNC(=O)C(C)C)NC(c1c(CC)nn(C)c1)=O 60695,Cc1onc(C(F)(F)F)c1C(=O)NC1CCC1CNC(C1(O)CCSC1)=O 60696,Cc1nc(-c2ccc(F)cc2)nc(NC(C2CCC(NC(=O)C(C)CN)C2)=O)c1C 60697,CCC(C)(C)C(C)CNc1c(OC(C)C(=O)OC)cccc1Br 60698,C1(CC)C(C(=O)N(CCS(C)(=O)=O)C)CCN1C(=O)CN(C1CC1)CC 60699,CC(CCN=c1[nH]c(=NCc2csc(N(C)C)n2)c2[nH]ccc2[nH]1)CC(C)(C)C 60700,CCCC(C)(O)CC(=O)N(C1CCC(CNC(=O)Cn2cnnn2)CC1)C 60701,C1(Cl)(C(=O)NCCNC(c2cnc(C(F)F)s2)=O)CC12CCOCC2 60702,C12(C(=O)NCC3(O)CC(NC(=O)CNC(C4CCC4)=O)C3)CCCCC1C2(F)F 60703,Cc1nc(N(C(CNC(=O)Cc2ccnnc2O)(CO)CO)C)c2cc[nH]c2n1 60704,c1(C(=O)NCC(C)CN(C)C(c2cnn(CC(F)F)c2)=O)cc(CO)c[nH]1 60705,c1(C(=O)NCC2=CCN(C(CN3CCC(C)C3)=O)CC2)ccc2c(c1)N(C)CC2 60706,C1(C(=O)N(CC(O)C(=O)OC)C)(NC(c2c(CCC)n[nH]c2)=O)CCCCC1 60707,C(=O)(N=c1[nH][nH]c2c1CN(C(=O)OC(C)(C)C)C2)NCc1ccc(COC)o1 60708,CCC(C)C(C(=O)N1CCCC1(CO)CO)N(C)C(C1CC1C#N)=O 60709,C1(C(=O)NCCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 60710,C1(NC(Cc2c(C)ccs2)=O)CCCC(CNC(=O)CC#N)CC1 60711,N1(C(CCn2c(C)ccc2C)=O)CCN(C(=O)C(C)Cc2cnco2)C(CF)C1 60712,c1(C(N(C)CCOCCCNC(=O)C(O)C2CCCC2)=O)cc(P(C)(C)=O)cs1 60713,c1(CC(=O)NCC2CC(NC(c3snc(O)c3Cl)=O)C2)c[nH]c2ccc(F)cc12 60714,c1(C(=O)NCC2OCCN(C(CC(CCC)O)=O)C2)ccc(N)cc1[N+](=O)[O-] 60715,C1(OC)CCC(C)(C(N2CC(CNC(c3cccc(F)c3Cl)=O)C(O)C2)=O)CC1 60716,CC(C)C(C)C(=O)N(CC(C)NC(c1ccnc(-c2ccco2)c1)=O)C 60717,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 60718,n1(CCC)cc(Cl)c(C(=O)NC2CCC(C)(CNC(C3CN(C(C)=O)C3)=O)C2)n1 60719,C1(C(=O)NC(CCCNC(C(C)SC)=O)C)CCC(C)(C)O1 60720,Cc1ccccc1C=CC(=O)Nc1ccc(C(N2CC3(CC3CO)C2)=O)[nH]1 60721,c1(C(=O)NC2CC(NC(C3(C)CCCCO3)=O)C2)cc2sc(Cl)cc2s1 60722,N1(C(CC2C(CC)C2)=O)CC(N(C(=O)C(c2ccccc2)OC)C)C(O)C1 60723,C(c1cc[nH]n1)=CC(=O)NC1CCCC1CNC(=O)COC1CCCC1 60724,Cc1cccc2c1CC(C(N1CCC(NC(c3csc(Cl)c3Cl)=O)C(F)C1)=O)N2 60725,CC(O)(C(=O)N1CC(CNC(=O)CN2C(=O)CCCC2=O)C2(CCC2)C1)C(F)(F)F 60726,C#CCC(C(=O)NC(C1CCOCC1)CC)NC(=O)C(C1CCC1)OCC 60727,C1(CC)CCN(C(c2cscc2Cl)=O)C1C(=O)NC1(CC(C)C)CC1 60728,c1(CC(=O)NCC2(CN(C(c3c(C)cccn3)=O)C)CC2)ccc2c(c1)CCC2 60729,CC1CC(NC(=O)COc2cccc(F)c2)CN(C(C2CC3CCC(C2)C3)=O)C1 60730,C(=O)(C(CCC)C(C)C)N1CC(NC(CCC=CC)=O)C2(C1)CC2 60731,N1(C(C(C(C)(C)C)OC)=O)CC2(CC(NC(=O)CSCc3ccccc3)CO2)C1 60732,C(C)(CNC(c1cn(-c2ccn(C)n2)cn1)=O)(CO)NC(C=C(C)C)=O 60733,c1(OC)cccc(C(C)CC(=O)N(C)CC2(NC(=O)Cc3ccnn3C)CC2)c1 60734,CCCC(C)(CC)C(=O)NCC=CCNC(c1ccc(CSCCCOC)o1)=O 60735,CC1(C)CN(C(C2(C)CC2Br)=O)CC(CNC(c2scnc2C2CC2)=O)O1 60736,Cc1c(C(=O)NCC2(NC(=O)C(C(C)C)NC(N)=O)CCOCC2)cnn1C 60737,C(CC(=O)N1CCC(C)(CO)C1)(C(C)(C)C)NC(Cc1ccc(C#C)cc1)=O 60738,N1(C(COCCOC)=O)CCOC(CC(N2CCCCC2C(N)=O)=O)C1 60739,Cc1cc2c(C(=O)N(C(C)CCNC(C3CCNC(=O)C3)=O)C)cccc2o1 60740,c1(C(N(CCC(=O)N2CCC2)CCCO)=O)cc2occc2[nH]1 60741,c1(C(=O)NC2(C)CC(NC(C(C)(C)NC(C)=O)=O)C2)cc(C)nc2cc(C)nn12 60742,C1(CNC(C2(C#C)CN(C(=O)Cc3ncoc3C)C2)=O)CCC2(CC2)CO1 60743,c1(C(N2CCC(NC(C3C(C)C3(F)F)=O)C2)=O)cnc2cc(C(F)(F)F)ccn12 60744,C(=O)(C1=C(C)OCCC1)NCCN(CCC)CCOC(CC)CC 60745,c1(C(=O)NCC(C)CN(C)C(C2CCCN2C)=O)cn2ccc(F)cc2n1 60746,C#Cc1cncc(C(=O)NCC(O)CNC(c2cnc(C(F)(F)F)c(C)c2)=O)c1 60747,Cc1cc(C(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)C2CC2)[nH]c1C 60748,C1(CC(N2CC(O)(C(C(=O)NCC(C=C)C)F)C2)=O)CC2(CCC2)C1 60749,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 60750,c1(C(N(CC)CC2CCN(C(=O)C(F)C(C)(C)O)CC2)=O)ncsc1S(N)(=O)=O 60751,CCS(=O)CC(=O)NCCOC1CN(C(C2CCCC(C3CC3)O2)=O)C1 60752,C(C)(CCC(=O)N1CC(CCCCNC(c2cnc[nH]2)=O)C1)OC 60753,C=C(Cl)CCC(=O)N1CCC(C(N2CC(OC)C2)=O)(OCC(C)C)C1 60754,N1(C(Cc2cc(C)no2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 60755,Cn1cc2c(n1)CC(C(N1CC(O)CC1CNC(c1nn[nH]c1Cl)=O)=O)CC2 60756,Cc1ccc([N+](=O)[O-])cc1CN1CCNCC1C(=O)Nc1c(O)cccc1Cl 60757,c1(C(N2C(C(N3CCC(F)C3)=O)CC3CC32)=O)c(F)cc(F)cc1Br 60758,C(C)(CCC(=O)NC(CCC1CC1)C(=O)NCc1ncccc1F)OCC 60759,CC1(C)CC(NC(=O)CC2CC3(C2)CN(C(=O)CC2(C)CC2)C3)C(=O)O1 60760,c1(CC)ccc(C(N2CCCC(C(N3CC4CCC3C4)=O)C2)=O)cc1CC 60761,c1(C(C)=O)oc2ccccc2c1NC(c1csc2ccc(Cl)cc12)=O 60762,N1(C(CN2CCC(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 60763,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 60764,c1(-c2cccc(C(=O)Nc3ncc(C(=O)OC)cn3)c2)nc2cc(C)ccc2o1 60765,CCC(CC)C(C(=O)N1CC2(C)CC1(C(N1CCCCC1CC(C)C)=O)C2)OC 60766,C=CC(C)(CC)C(=O)NCC1=CCN(C(C2CNC(=O)N2)=O)CC1 60767,CCCCC(C(=O)N(C)CC1(O)CCCN(C(c2cccn2CC)=O)C1)N(C)C 60768,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 60769,CC1(C)C(c2cn(CCc3cccnc3)nn2)CCN1C(=O)COc1ccc[nH]1 60770,C=CCC(C(=O)NC(CO)CCCCNC(=O)CN(C)C(=O)OC)C(C)C 60771,CC(C)(C(=O)N1CCC(C)(CCNC(=O)CCCCN(C)C)CC1)C(N)=O 60772,c1(COCC(N2CC(CC(C)NC(c3cnc(S)[nH]3)=O)C2)=O)ccccc1 60773,C1(CCC(=O)NCC2(C)CCCO2)CCCCN(C(c2cccc(F)c2F)=O)C1 60774,CC1CN(C(C2(C)COC2)=O)CCC1CNC(=O)CC1(C)CCCCC1 60775,C(=O)(C1=C(Cl)CCC1)NCCCCCN(C)C(C1CCN(CCO)C(=O)C1)=O 60776,N1(C(C2CC(N(C(C(Cc3ccccc3)OC)=O)C)C2)=O)CCN(C)CC1 60777,C(=O)(C(CC(N)=O)NC(=O)CCCCCSC)NCc1cc(C)sn1 60778,c1(C(N(C2CCCN(C(=O)CCc3ncc[nH]3)C2)C)=O)cnc2c(Cl)cccn12 60779,S(=O)(=O)(CCC(=O)NC1CCN(C)CC1C)N(C(c1ccc(C)cc1)C)C 60780,c1(C(=O)NCC2N(C(COCC)=O)CCC2C)ccc2c(c1)N(C)CCO2 60781,N1(C(Cc2nc(C)sc2C)=O)CCCC2(CCN(Cc3ncc(F)cn3)CC2)C1 60782,c1(C(N2CCC(NC(C3(C)CCCNC3=O)=O)C2)=O)cccc2c1OCCCO2 60783,N1(C(CC=CC=C)=O)CCCC2CN(C(=O)C=CC(C)(C)C)CCC12 60784,Cc1nc2ccccc2c(C(=O)NCC2CCCN2C(=O)CC2(O)CCC2)c1O 60785,N1(C(=O)Nc2c(CCC#N)c3n(n2)cccc3)CCC2(CC1)CC(O)(CO)C2 60786,CCC(CC(=O)NC1CC(SC)C1)N(C(=O)C(C)CSC)C 60787,Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCCCN(C(=O)C(C)CF)C 60788,Cc1cc(OC(c2ccc(OC(=O)NC3(C)CCC3)cc2)=O)ccc1[N+](=O)[O-] 60789,C(C)(CCC(=O)NCCCC)N(CCCC)C=O.C1CCCN1.[SH](C)(=O)=O 60790,CCCCC(C)CCC(=O)N(CCC(=O)N(CCCC)C(C)C)CC(=O)OC 60791,C1(CCC(=O)NC(CNC(C2(COC)CCOC2)=O)(C)CC)C(=O)ON=C1C 60792,c1(CC(=O)NC2CN(C(CN(C(COC)=O)C)=O)C(C)C2)cc(F)ccc1Br 60793,C(=O)(CCCCCn1cc(C(C2CC2)C2CC2)nn1)N1CC2C(C(=O)OC)(C2)C1 60794,C(=O)(C1=CCCCC1C)NCCCOC1CCN(C(CCCN(C(C)=O)C)=O)C1 60795,C1(COC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCC(F)(CC1)C2)=O 60796,CC(C)CC(CNC(=O)CCc1ccc(F)nc1)NC(=O)CC(C)N(C)C 60797,N1(C(c2ccc(OC)cc2)=O)CCCC2(NC(C3CN4CCC3CC4)=O)CC2C1 60798,Cc1nc(C(C)(C)C)sc1C(=O)NC1CC(C)(NC(C2CCC(C)(C)C2)=O)C1 60799,C1(CNC(C(CC)SC)=O)CC2(CC2)CN1C(c1ccc(Cl)c(OC)c1)=O 60800,C1(NC(C2CC(NC(=O)C=Cc3cocn3)C2)=O)(CN(C)C)CCCCC1 60801,C12(NC(c3nccc(C)c3F)=O)CCCC1N(C(C1CC13CCCCC3)=O)CC2 60802,C1(NC(CCCOCC=C)=O)CCCCN(C(=O)Cn2cc(C)ccc2=O)CC1 60803,CCCCC(C(=O)NCC1(CO)CCCO1)NC(=O)C1=CC2C=CC1C2 60804,c1(OC)ccc(C(N2CC(CNC(C3CC3F)=O)(CO)C2)=O)nc1Cl 60805,Cc1ncc(Cl)cc1C(=O)NCCN(C(=O)C(C)(C)c1cnco1)CCCN(C)C 60806,N12CCCC(C)(C1)C2=O.Cc1cccc(-n2ncc(-c3nn[nH]n3)c2C)c1 60807,N1(C(c2c(NC)nccc2)=O)CC(CNC(=O)CC(C)(C)SC)CC(C)(C)C1 60808,Cc1ccnnc1C(N1CCC(Cn2cc(-c3csc(C)n3)nn2)C1)=O 60809,C(CCF)(C(=O)N1CCCC(C(c2cn(CCCCF)nn2)N(C)C)C1)N(C)C 60810,C(=O)(CC(C(F)(F)F)NC(=O)CC1CCC(=O)C1)NCc1cccc(C)n1 60811,CCC(C)CCC(=O)NC1(CCNC(=O)C(c2ccccc2F)C)CCC1 60812,N1(C(C(C2(C)CC2)NC(CC2CCN(C)CC2)=O)=O)CC2(CCC(=O)N2)C1 60813,c1(C(C2(COC)CN(C(C=CC)=O)C2)=O)cc(-c2ccccn2)ccc1Cl 60814,c1(C(=O)NCC2(NC(C(C)NS(C)(=O)=O)=O)CC2)ccc(C2CCC2)nc1 60815,C12(NC(c3nnn(C)c3N)=O)CCCC(NC(=O)CNC(N)=O)(C1)C2 60816,C1(NC(C(C)=CC2CC2)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 60817,N1(C(c2c(C)nc(Cl)cc2)=O)CCOC2(CCN(C(=O)COc3ccon3)C2)C1 60818,CC(C)C1=CCC(NC(C2CCN(C(=O)CC3(O)CCC3)C23CC3)=O)CC1 60819,CCCCC(=O)CNC(C1CC(OC)CN1C(c1occc1C(C)C)=O)=O 60820,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 60821,C(=O)(C(N)CCCCC#N)N(N1CCCC(CC)CC1)CC 60822,C1(C(=O)NCC23C(CN(C(c4cc(SC)on4)=O)C2)C3)CCc2nnnn2C1 60823,Cc1noc(C)c1N(C(=O)N(C(C)C)C)C.c1(-c2ccccc2)cn(C)cn1 60824,Cc1conc1CC(N1CCCC1Cn1cc(C2CCCN2C2CCC2)nn1)=O 60825,C1(C(=O)NCC2CC(SC)C2)CCN(C(c2cc(Cl)ns2)=O)CC1C 60826,C1(NCCc2c(OCC)ccc(Br)c2)CCC2(CCCCC2)CC1 60827,C1(C(N2CC3C(NC(C4N(C)CCC4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 60828,c12cc(c(CC)cc1CC)C(=O)O2.C=C1COCC1N(C)C 60829,c1(NS(CCC)(=O)=O)cccc(C(=O)N(C)CCN(C(=O)CCSCC(N)=O)C)c1 60830,CC1(C)CCN(C(C2(NC(=O)C(O)C3CCC3)CC(O)C2)=O)C1 60831,c1(C(C)OC(=O)NCCC2N(C(N3CCC(C)C3)=O)CCC2)c(F)cccc1F 60832,c1(C(N2CC3C(NC(COCC=C)=O)C(C3)C2)=O)cnc2cc(C)nn2c1 60833,C(C(C(=O)NCCCC(N)=O)NC(c1cocc1C(N)=O)=O)OCC 60834,C1(NC(C2CN(C(=O)NC)C2)=O)C=CCC(C(=O)NCCN2CCOCC2)C1 60835,N1(C(C(=O)NCC(C)F)=O)CCOC(N(C)CCN(C(=O)OC(C)(C)C)CC)C1 60836,C=CC1(C(=O)N(C)Cc2ccoc2)CCN(C(c2ccncc2O)=O)C1 60837,C(=O)(C(CCC1CCC1)N(C(C)C(C1CC1)Sc1ccccc1)CC)NC(CC)C 60838,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 60839,c1(C(=O)NCC(C)NC(c2nocc2C(C)(C)C)=O)cccc(Cl)n1 60840,c1(CC)nc(C)n(C)c1C(=O)NC1C2CCN(C(c3csnn3)=O)C12 60841,C(=O)(CCC(=O)C1CC1)NC1C(NC(C=C)=O)CCC1 60842,c1(CNc2nccc(-c3cn(C)c(=O)cc3)c2)c[nH]c2cccc(Br)c12 60843,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC1 60844,c1(CC)cc(Cl)ccc1C(=O)NC(CN(C)C(C1CCOC1CC)=O)(CO)CO 60845,Cc1cc(C(N2CC(C3(NC(=O)CC4(C)OCCO4)CC3)C2)=O)cnc1C(F)F 60846,C1(C#N)(C(=O)NC(C)CN(C(=O)C(F)(F)c2cscn2)C)CCCC(=O)C1 60847,N1(C(c2c(C)nccc2)=O)CCN(C(=O)C(CO)NC(=O)C(C)C)CC(C)(C)C1 60848,C1(O)(CN(C(C2C(OC)CCC2)=O)C)CCCN(C(c2ccncc2Cl)=O)C1 60849,C#CC1(C(N2CCC3CC23)=O)CN(C(=O)C(c2cnn(C)c2)=O)C1 60850,c1(NC(=O)NC(CC)C(=O)Nc2ncc(C(F)(F)F)s2)cccc(CC#N)c1 60851,C1(CC)(OC(=O)CCc2cnc(O)[nH]2)CCN(C(=O)OC(C)(C)C)C1 60852,C1(NC(c2c(CC)onc2C2CC2)=O)COC2(C1)CN(C(=O)C1=COCC1)C2 60853,C(=O)(CC(C)P(C)(C)=O)N1CC(CCNC(c2cc(OC)c(C)cc2)=O)OCC1 60854,c1(C(=O)NC2CCC(CCNC(CC(C)(C)N(C)C)=O)C2)ccc2c[nH]nc2c1 60855,CC1CC2(CCO1)CCN(C(C1CCOC1CNC(=O)CC1CCCC1)=O)C2 60856,C1(C(=O)NCC(C)(C)N2CCCC2)CCN(C(C2CC(=O)C23CCC3)=O)C12CCC2 60857,N1(C(C2CNCC(C)O2)C(N2C3CCC2CN(C)C3)=O)CC(=O)N2CCCC2C1 60858,CCC(CC)CCCC(=O)NCCCN(CCCNC(c1cncc(C)c1)=O)C 60859,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)(CC)CC)CC1 60860,c1(C(N(CCNC(C)=O)C)=O)nccc(-n2ccc(C)n2)n1 60861,C1(CN(C(c2c(C)scc2)=O)C)CCCCN1C(=O)C(c1ccncc1)C 60862,C1(C(N(CCC)CCNC(C2CCN(CC)C2)=O)=O)CCc2nn[nH]c2C1 60863,c1(C(N2CCC(N(C(CC=CCC)=O)C)C2)=O)cc(Cl)c(C)cn1 60864,c1(C(=O)NCC2(O)CCN(C(CC=CC=C)=O)C2)cc(F)cc2cc[nH]c12 60865,N1(C(COC(CC)C)=O)CC2CC(NC(=O)C(c3ccnn3C)O)CC(C2)C1 60866,CC(C)C(C(=O)N(C1CC2CCC1O2)C)NC(=O)CN1CC=CCC1 60867,c1(C(N2CC(NC(C3C(C)CCC3)=O)CC2(C)C)=O)cc(S(=O)(=O)N(C)C)c[nH]1 60868,C1(CN(C(=O)CCOC2CCC2)C)CN(C(c2c[nH]c(C#N)c2)=O)CCO1 60869,C(c1ccccc1)=C(C)C(=O)NCC(=CBr)CSc1nncs1 60870,C(CN=c1nc(C2CC2)[nH]s1)N(C(C(CC)OC1CCCC1)=O)C 60871,C1(C(=O)NC(CN(CC)CC)C)CCCC(NC(=O)C(C)(C)O)C1 60872,c1(C(N2CCC(NC(CNC(COC)=O)=O)C2C(C)C)=O)cc(O)cc(N)c1Cl 60873,C(=O)(C(C)(C)C(F)c1ccccc1)NC1CC(NC(Cc2cn(C)[nH]c2=N)=O)C1 60874,c1(NC(C2C(C)CN(C(=O)C(F)=CC3CC3)C2)=O)cnc(O)n(C2CC2)c1=O 60875,c1(C(N(CC(=O)OC)Cc2cn(CCCO)nn2)=O)cc(Br)cc2nc(O)[nH]c12 60876,CCC(O)CCNC(=O)CCOC1CN(C(=O)C=CC(=O)N(C)C)C1 60877,c1(NC(C(C)NC(C)=O)=O)ccc(C(=O)NC(C)C(CO)NC(=O)CC2CC2)cc1 60878,CC(C)(C)CC(O)C(=O)NCCC(O)C(=O)NCCC1CCOC1 60879,c1(C(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CC2)cc(OC)c(OC)cc1F 60880,C1(C(N(c2cccc(Cl)c2)C)=O)CC(O)CN1C(=O)CN1CCOCC1=O 60881,C1(NC(Cc2c(CC)con2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 60882,c1(OC)ccc(F)c(F)c1C(N1CC(C)CC1C(N1CCC(C(N)=S)CC1)=O)=O 60883,Cc1ccc(C(F)F)c(C(N2CC(O)(C(C)NC(c3conc3C)=O)C2)=O)c1 60884,N1(C(C)=O)CCC2(CCN(C(=O)N(c3ccsc3)C3(CC(F)F)CC3)CC2)C(C)C1 60885,N1(C(C(C)N=[N+]=[N-])=O)Cc2[nH]nc(C(=O)N(C3CCN(C(C)C)C3)C)c2C1 60886,CCC(C)(CNC(=NC)NCc1cc(C)[nH]n1)Cc1ccccc1 60887,CC(C)(CN=C(NC1CCOCC1)NCC1(F)CCCC1)OC1CCC1 60888,C(CC(C(=O)N(CCCN(C)C1CC1)C)NC(N)=O)SC 60889,C1(C(N(CCCNC(=O)Cc2cncn2C2CC2)CC)=O)NC(=O)OC1(C)C 60890,c1(CCC(=O)NC2CCC(CNC(CSCC)=O)C2)n[nH]c2c1CCCC2 60891,N1(C(Cc2cccc(C)c2)=O)CC2OCCN(C(=O)C3=CCCCCC3)C2C1 60892,C(=O)C(CC(C)C)ONC(C1CCCOC1C)=O.C1(=O)CN1CC.CCO 60893,c1(C(=O)NCC(C)N(C)C(c2c[nH]cc2-c2cnn(C)c2)=O)ccc(N)c(O)c1 60894,N1(C(=O)CC2OCCCO2)CC2CCC1CN2C(c1ccc(CO)c(Cl)c1)=O 60895,N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NOCc2ccc(F)cc2)C(O)C1 60896,N1(C(C(c2ccccc2)C2(C)CC2)=O)CC(CNC(=O)CCC=CBr)C(O)C1 60897,N1(C(c2nc(C)cs2)C(=O)NC(C(=O)OC)C)c2ccccc2CC1C 60898,c1(CC)ccc(CNC(C2C(CC(=O)NCC3CC3CC)C2(F)F)=O)cc1 60899,c1(C(N(CCNC(=O)CCc2cc(C)no2)CC)=O)c(F)cccc1[N+](=O)[O-] 60900,CCCCCCC(C)(c1nn[nH]n1)NC.c1(SCCCCNC(=O)OC)ccc(Cl)s1 60901,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 60902,C(C(C)(C)CCNC(=O)CCc1ccsc1)NC(C(C)OCC(C)C)=O 60903,CC12COCC1CN(C(c1conc1CNC(=O)CC1CCOC1=O)=O)C2 60904,c1(C(=O)NCC(C(=O)OCC)(C)CC)cc(S(N)(=O)=O)cc(C(F)(F)F)c1C 60905,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2c(C)c(N)cnc2)=O)C)C1 60906,n1(CC)cnc2c(N3CCOCC3)[nH]c(=NCC3CC(F)(F)CO3)nc12 60907,C1(C(=O)NC(CCOC)CNC(c2cnns2)=O)CC2(C1)NC(=O)NC2=O 60908,c1(OC)cccc(-n2nc(-c3ccco3)nc2C(=O)OC)c1 60909,C1(NC(C=CCN(C(C2CN(C(C)C)C2)=O)C)=O)(CO)CC2CCCC12 60910,C1(F)(CNC(C(C2CCCC2)OC)=O)CC(CNC(=O)COCC(F)F)C1 60911,C(C)(CCN=c1[nH]c(=NCCSCC)[nH]c2c1CCC2)CC 60912,N1(C(c2ccc(O)cc2F)=O)CCC2C(CCN2C(c2nocc2Cl)=O)C1 60913,C1(C)(CNC(C(CC)(C)C)=O)CN(C(C2CC3CCCCC3O2)=O)C(C)(C)C1 60914,N1(C(c2cc(C)c(C)[nH]2)=O)CCC(C)(C)C1C(=O)NC1CCCC1(F)F 60915,N1(C(C(C)OC)=O)CC=C(CNC(=O)C(c2ncccc2Cl)(F)F)CC1 60916,c1(CC(=O)NCCC2CCC(NC(=O)C=CCN3CCC3)C2)cnccc1Cl 60917,N1(C(CCc2ccc(C)o2)=O)CCC(CNC(c2cnc(C(N)=O)s2)=O)C(C)C1 60918,Cc1cccc(C(=O)NCC2(CNC(=O)CCc3cnccn3)CC2)c1Cl 60919,c1(CC(=O)NCC2C(NC(c3c(C)n[nH]c3)=O)C2)c(F)cccc1Br 60920,C(=O)(CCCC(F)(F)C(F)(F)F)N1CC2C(CNC(c3cc(O)ncn3)=O)C2C1 60921,N1(CCN(C(CC2C(C)CCC2)=O)C(C)C)CCN(C(=O)C(C)(C)N(C)C)CC1 60922,c1(C(=O)NCCCN(C(=O)OC(C)C)C)cccc(Br)c1 60923,C(=O)(CC(C(F)(F)F)OC)NC1(CC=C)CCN(C(=O)C(C2CCCC2)OC)C1 60924,c1(C(C)C)ccc(NC(=O)NC2(C(=O)N(C)C)CC2)c(C#N)c1 60925,N(C1CCc2cc(CNC(=O)Cc3cncs3)ccc21)C(Cc1cnc(C)[nH]1)=O 60926,c1(C(=O)NC(C=CC(=O)N(CCOC)CC)(C)C)sccc1OC 60927,C1(C(=O)OCC)CC(OC)CN(c2nnc(-c3cnccn3)n2CC(C)C)C1 60928,N1(C(c2nccc(OC)c2)=O)CCC(NC(=O)C(N2CCCCCC2)C)C(C)(C)C1 60929,N1(C(Cc2ccn(CC)n2)=O)CCN(C(C2C=CCC2)=O)CC1CC(F)(F)F 60930,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 60931,N1(C(CCCC(=C)C)=O)C2CCC1C(C)C(NC(C1CC(=O)N1)=O)C2 60932,CC(C)C(C)(C)COC(=O)CCC1CC1 60933,C1(N(C(=O)NC(c2nnc(C)n2C)c2cnccn2)CC)CC2CCC1C2 60934,c1(C(=O)NC2CCOCC2C(=O)NCCc2cc[nH]n2)c[nH]c2cccnc12 60935,c1(C(=O)NC2C(NC(c3ccc(C(F)F)cc3)=O)C2)cccc([N+](=O)[O-])c1 60936,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1SCCS1 60937,Cc1cc(=NC(=O)C2CCC2C2OCCCO2)[nH]n1C(C)C(=O)N(C)C 60938,C1(C(=O)NCC(C)(C)O)CCOCC1NC(=O)C(Cl)Cl 60939,CC(C)CC(C)C(=O)N(C1CCCN(C(=O)COC2CCCCC2)C1)CCF 60940,C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CCc2cscn2)C12CCC2 60941,n1(C(C(=O)NCCN(C(C2(Cl)CC2(F)F)=O)CC)C)cc(C)cn1 60942,c1(OCC(=O)NC(C2CN(C(=O)CCCOC)CCO2)CC)cc(C)ccc1C 60943,c1(-c2c(NC(=O)NCCC(C)NCC)cccc2)ccccc1[N+](=O)[O-] 60944,C1(C(=O)NCCC2CCCN2C(=O)Cn2ccnn2)CCC2CC2CC1 60945,c1(NC(CCC)CNC(=O)Cn2ccnn2)cc(C(C)(C)C)ncn1 60946,C(CO)(C(=O)N1CC(C)(NC(=O)Cc2csc(O)n2)C1)NC(=O)OC(C)(C)C 60947,CCC(CCC(=O)Nc1ccc(N(C)C)nc1)NC(=O)C(F)C(C)C 60948,C1(C(=O)NCCCCCN(C)C(C23CC2CCC3(F)F)=O)(OC)CCC(C)CC1 60949,c1(C(=O)NCC2C3CN(C(c4cc(OC)n[nH]4)=O)CC32)n[nH]c2c1CN(C)CC2 60950,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 60951,C1(NC(C=CC)=O)CC2CCC1N(C(c1cnn(CC(F)F)n1)=O)C2 60952,CC(C)C(CC(=O)NC1(C)CCN(C(c2cc(C#N)c[nH]2)=O)C1)c1ccccc1 60953,c1(C(=O)NCCCNC(C2N3CC(C)N(CC3)C2)=O)ccc2c(c1)C(=O)NCC2 60954,C1(CC(=O)NCc2cnc(CC)s2)CN(C(C2(F)CCC2)=O)CC(C)O1 60955,C1(C(=O)NCC(O)Cn2cccn2)(CNC(COC(C)(C)C)=O)CCOC1 60956,C1(CCNC(C(CO)OC)=O)CCN(C(C2C3COCC23)=O)CC1(F)F 60957,CC1CC(CC(=O)OCCN2CCN(CC(F)(F)F)CC2)CCS1 60958,C1(C(=O)NCCC(=O)N(C2C(C)OCC2)C)CC2(CC(=O)C2)C1 60959,C(C(C)(C)C(=O)NC1CCC(CNC(c2cc(Br)oc2C)=O)C1)OC 60960,N1(C(c2cc(CC)nnc2C)=O)CCC2CN(C(=O)CC3CCCN3C)CCC12 60961,Cc1cc(NC(C2(C)CN(C(=O)CCc3ccccn3)C2)=O)cnc1F 60962,c1(CNC(C2CCCC2NCc2cccc(O)c2)=O)cccc(F)c1F 60963,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 60964,C(=O)(C1CN(c2nnc(-c3ccco3)o2)c2c(C)cccc21)OC 60965,N(C(=NCC1CC1(F)F)NCC1(OC)CCC1)CCNC(C1CCCO1)=O 60966,C1(CNC(c2ncc(OC)nc2)=O)(CNC(=O)CCC(=O)N(C)C)CCCCC1C 60967,C1(OC)CC(NC(=O)C(=O)Nc2cccs2)C(OCCN)C1.c1(O)cccnc1C.CC 60968,N1(C(c2nncc(OC)c2)=O)CC(O)CCC1C(=O)NCC1(Cl)CC1(F)F 60969,CN1CCC(O)C(NC(=O)CN(C(C2C3CCC(F)C23)=O)C2CC2)C1 60970,Cc1cnc(C(N2CC3CC2C3C(=O)N(C(C)CC(N)=O)C)=O)nc1 60971,N1(C(C(F)=C(C)C)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CC1CC1 60972,c1(CC(=O)NC(CC)(C)CN(C(c2coc(C3CC3)n2)=O)CC)ccnc(Cl)c1 60973,C(=O)(C1=C(Cl)CCC(C)C1)NCCC(=C)CNC(c1[nH]nnc1C)=O 60974,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 60975,c1(OC)ccc(-c2ccc(F)c(CO)c2)cc1C(N1CCC(OC(C)=O)CC1)=O 60976,C(C(CNC(c1cnccn1)=O)C(F)(F)F)NC(C1(C)CCOCC1)=O 60977,CC(C)CC(CNC(=O)C(C)C(F)(F)F)C(=O)Nc1ccc2nc[nH]c2c1 60978,CCC(C)(C(=O)NCC1(F)CC(NC(=O)C(c2cnn(C)c2)O)C1)C(F)F 60979,c1(SCCCC2CC2)nnc[nH]1.C1(CC(=O)NC)(C(=O)OC)CCC1.C1(=O)CN1 60980,N1(C(Cc2c(C)cccn2)=O)CC(C(=O)NOCC(C)O)CCC1(C)C 60981,C(=O)(CC1=Cc2ccccc2C1)N1CC(OCC)C(CNC(C2CC2C)=O)C1 60982,C=CCC(CNC(=O)C(c1ccnn1C)C)C(=O)N(CC)OCC=CCl 60983,C#Cc1ccc(C(N2CC(C3(NC(=O)C(F)CC4CCC4)CC3)C2)=O)cn1 60984,N1(C(C2=C(C)OCCS2)=O)CC(NC(=O)C(C)c2cncs2)CC2(CCC2)C1 60985,Cc1cn2cc(C(=O)N(C3CCN(C(=O)CC(C)C(C)C)C3)CC3CC3)nc2s1 60986,N1(C(C(C2CCC2)NC(=O)CCc2cnccn2)=O)CC2CCC(CO)(C2)C1 60987,N1(C(C(CCC)C)=O)CCC(COC)(NC(=O)CC(C(F)F)N(C)C)CC1 60988,N1(C(C=CC=CC)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 60989,C#Cc1nc(C(N2CCN(CCN(C)C(C3CCCC(OC)C3)=O)CC2)=O)cs1 60990,C(=O)(C1=CCC(C)(C)CC1)N(CC(N1CCC(c2nc[nH]n2)C1)=O)CCOC 60991,C1(NC(C(C(C)C)C#N)=O)CN(C(=O)CC2CC3CCC2C3)CC2(CCC2)C1 60992,c1(CNC(c2ccc(F)cc2)C(CC)C)ncc(OC)cn1 60993,C(C)(C(O)C(=O)NC1CCC1CNC(=O)OCC)SC.C(C)(C)C 60994,C(CCCCCC1(NC(CNC(C)=O)=O)CCC1)NC(=O)CC1CC=CC1 60995,C(=O)(C(Cc1ccccc1)NC(C)COc1ccccc1)OC 60996,C1(CNC(c2c(COC)cco2)=O)CC2CCC1N2C(=O)COc1ccon1 60997,N1(C(c2cn(C)nn2)=O)CCN(C2CCCC2NC(=O)CN2CC3CC3C2)CC1 60998,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cnnn2)CC1 60999,c1(CN2CCC(O)(C(=O)Nc3nc4c(s3)CCC4)C2)cnc2ccccc2c1 61000,CC(C)CC(O)C(=O)NC(C)CN(C(=O)Cc1ccc(Cl)c(F)c1)C1CC1 61001,C1(C(=O)Nc2ccccc2C(F)F)CC2CC2N1CCOc1ccnnc1 61002,N1(C(C(CO)NC(=O)C2CC2)=O)CCCCC1C.O=CC=C1CCC1 61003,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(CC1CCC1)OC)C2 61004,C1(n2cc(CNC(C)=O)nn2)CCCN(C(c2csc(C(F)(F)F)c2)=O)C1 61005,c1(C(=O)NCC2CN(C(c3c(Cl)nc(OC)s3)=O)CC2C)cc2ncccn2n1 61006,Cc1ccc(C(N2CCCC(NC(C3CC3)=O)C2)C(=O)NCCCF)c(F)c1C 61007,c1(C(N2CCC(NC(c3c(C)cccn3)=O)(CO)C2)=O)ccc(N=[N+]=[N-])cc1 61008,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3F)=O)cccc2[nH]1 61009,C(CN=c1[nH]c(=NCCc2nccn2C)[nH]c2c1COC2)N1CCN(CC)CC1 61010,CCC(C)(C)C(=O)N1CCC(C(=O)NCCN=[N+]=[N-])O1 61011,C#CCCC(O)CCN(C(C(O)CCOC)c1ccccc1)C 61012,CC(C)C(C(=O)N(CCNS(N)(=O)=O)C1CC1)n1cc(CCC2CCCN2C)nn1 61013,Cc1ccc(C(N2CCCC(C(N3CC(=O)NC(=O)C3)=O)C2C)=O)cc1C 61014,C1(C(N(C(C)C)CCN(C(=O)Cn2cccn2)C)=O)CC2CCC1NC2=O 61015,Cc1nc(CO)ncc1C(=O)NCCN1CCN(C(=O)COc2cccnc2)CC1 61016,CCC(C)(C(=O)NC1CC(C(=O)NCCO)C1)C(F)F.c1(SC)cccnc1 61017,CC(C)CC(F)(F)C(=O)N1CCOC(CN(C(=O)C(C)Sc2ccccc2)C)C1 61018,n1(CCCC)nnnc1C(CC)(C1CCC1)NCc1nnc(C)o1 61019,c1(C(N2CCC(N(C(=O)C(F)(F)CNC)CC)C2)=O)cccc2c1NC(=O)CC2 61020,C1(NCCC2CC(OCC)C2)CCS(=O)C1 61021,c1(C(=O)NC(C(C)(C)NC(C(COCC)C)=O)C)cc(C)n(C(F)F)n1 61022,Cc1c(C(=O)NCC(C2CCC2)NC(=O)C=C2CCC(C)C2)ncn1C 61023,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)CCCN1C(=O)CCC1=O)NC 61024,C1(C(N(CCCCCCC)C)=O)CC2(CCN1C(=O)C(CC1CC1)OC)CC2 61025,c12ncncc1C(=O)NCC(C)N2C.c1(CCOC)cc(Cl)cs1 61026,Cc1nc(C)c(N)c(C(=O)NCCCCN(C(=O)C(F)(F)c2cncs2)C)n1 61027,C1(C(=O)NCC2N(C)CCCC2)CCN(C(c2ccc(Cl)s2)=O)C(C)(C)C1 61028,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61029,c1(C(N(C2CCN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)C)=O)cc(Cl)c(Cl)cc1N 61030,C12CCCCN1C2=O.N1(C(COCC(=O)NC)=O)CCCC1C(C)(C)OC 61031,C(CCCCCNC(=O)C(O)c1ccco1)NC(=O)CCCn1cncn1 61032,C12(C(N(CC(=O)NCCCC(C)N(CCC)C)C)=O)CCCC(CO1)C2 61033,N1(C(COCCOCC#C)=O)CCC(NC(=O)CC2CCCC(O)C2)CC1 61034,C1(C(N(CC(C)=O)CCNC(C2CCN2C2CCCC2)=O)=O)CCC(=O)N1 61035,c1(C(N2C(CN(C(C3C4CCC34)=O)CC)CCC2)=O)ccc2cccc(F)c2n1 61036,N1(C(c2c(Cl)ccc(NC)c2)CSC)CC2(CCCC(c3ccccc3)O2)C1 61037,CC(C(=O)N1CC(O)CC1CNC(=O)C=CC(N1CCCCC1)=O)C(C)(C)C 61038,c1(C(=O)NCCC(C)CCNC(C2CCCO2)=O)ccc2c(c1)C(=O)NC2 61039,Cc1ncc(C(=O)NCCC2CCN(C(C3(c4cccnc4)CC3)=O)C2)c(C)n1 61040,CCC(CC)CCC(=O)N1CC2CC2(NC(C2(C)C=CCC2)=O)C1 61041,C1(CNC(=O)C(F)=CC2CC2)CC12CCN(C(=O)Cc1cccnc1O)CC2 61042,c1(C(C)C)nc(CN(C)CCC2CCCO2)no1.c12nnnn1C2 61043,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)CSCc2ccccc2)C)CC1 61044,C1(NC(c2c(CC)n[nH]c2)=O)CCN(C(c2ccccc2C2CC2)=O)CC1O 61045,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61046,C(=O)(N1CC(O)C(O)CO1)C1(NC(C(C)C2CCC2)=O)CCCCC1 61047,N1(CCNC(C2ON=C(C)C2)=O)CCN(C(C2(CF)CC2(F)F)=O)CC1 61048,C1(C(=O)NCc2cnc(Cl)s2)CC12CCN(C(=O)CC1CC3(CC3)C1)C2 61049,C1(NC(CC(C)N(C)C)=O)CN(C(=O)CSc2ccco2)CCC1(C)C 61050,N1(C(=O)Nc2c(OC)cc(C(F)(F)F)cc2)CC2(CCCC2)CCC1CO 61051,C(CCC(CC)CC)NC(=NCC=C)NCC(C)COC 61052,N(C(=NCC(F)(F)C(F)F)NCC1CCC1)CC1(OCC)CCCS(=O)(=O)C1 61053,C12CCCN(C1)C2=O.c1(C2C(OC)C2)ccncc1F.C1=CCN(C)C1=O 61054,c1(C(=O)NCC2CCN(C(c3c(OC)scc3)=O)CC2C)cnc2ccoc2c1 61055,N1(CC)CCC(C(=O)NC2CCCC2(C)CNC(C2CC(F)C(=O)N2)=O)CC1 61056,c1(C(N2CC(N(C)C(C3COCCO3)=O)C2)=O)ccccc1OC1CC1 61057,N1(C(Cc2cc(CC)no2)=O)CC2CN(C(=O)C=CC(F)F)CCC12 61058,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61059,c1(C(=O)Nc2ccc(OC)c(CO)c2)c[nH]c2c(C)c(Cl)ccc2c1=O 61060,c1(C(N(C(C)CNC(=O)CSCC(F)(F)F)C)=O)csc(C(F)(F)F)n1 61061,C1(C(N2CCC(NC(c3c(C(C)(C)C)con3)=O)C2)=O)CC2(C1)CC(F)(F)C2 61062,C(c1cnn(C)c1C)=CC(=O)NCCN(CCC)C(c1cc(OC)ccc1Cl)=O 61063,n1(CC(=O)NCC2=CCN(C(=O)CC3C=CCCC3)CC2)nc2n(c1=O)CCCC2 61064,CC1CCCCCN1C(C1(NC(=O)C(F)C(F)(F)F)CC(F)(F)C1)=O 61065,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61066,c1(C(=O)NC(C2CN(C(CCNC(C)=O)=O)C2)C)ccnc(S)c1 61067,C1(CCC)CN(C(c2sccc2SC)=O)CC1NC(=O)COCCOC 61068,CCC(C(=O)NC1(C)CCCN(C(=O)Cc2ccn(C)n2)C1)C(C)(C)CC 61069,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)COCCCF)CC2 61070,Cc1cc(CNC(N2CCC(C)CC2C(=O)O)=O)cnc1C 61071,C(=O)(C(C)(O)CC(C)C)N1C(CCCOC)CN(C(=O)CC2C=CS(=O)(=O)C2)CC1 61072,N1(C(=O)OC(C)(C)C)CCCC(C(C)(O)CNCc2cn[nH]c2)C1 61073,c1(C(N(CCN(C(=O)Cn2cnnc2O)C(C)C)C)=O)ccc(C(F)(F)F)cc1 61074,C1(C2CCOCC2)(C(N2CC(NC(=O)C=CC3CCOCC3)C2)=O)CC1(F)F 61075,n1(CC(=O)N(CCC)CCNC(=O)CC2CCC(F)(F)C2)ccc(C)cc1=O 61076,Cc1nsc(C)c1NC(C1(NC(=O)CC(=O)N(C)C)CC(F)C1)=O 61077,N1(C(C(=O)N(C)C)=O)CCC2C(C1)NC(=O)CN2C(c1ccc(O)nn1)=O 61078,c1(NC(=O)OC)cnc(S)nc1C(N1CCC(NC(C)=O)C(c2nccn2C)C1)=O 61079,C1(CC(=O)N(C2CN(C(C3CCN(C4COC4)C3)=O)CC2F)C)C(=O)N(C)N=C1C 61080,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61081,c1(C(C(=O)NCCOC)N(C)C(c2cncn2C)C)ncoc1C 61082,CC1(CNC(=O)CCOC2CC2)CCC(NC(=O)C=Cc2ccccc2F)CC1 61083,N1(C(c2c(OCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61084,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccccc3)CC2C1 61085,N1(C(c2nccc(C#C)c2)=O)CCN(C(=O)C(F)(F)C(C)O)C2(CC2)C1 61086,N1(C(Cc2c(C)ccs2)=O)CCC(NC(C2CCOC2C)=O)C(F)C1 61087,N1(C(c2ccc(F)c(F)c2)=O)CCC2(CCCN(C(C3CC(O)C3)=O)C2)C1 61088,C(=O)(C1CCCc2nc[nH]c21)N1C(CNC(c2c(C)n(C3CCC3)nc2)=O)CC1 61089,N1(C(C(CC)(F)F)=O)CCC12CN(C(=O)CCC(C)c1ccccc1)C2 61090,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61091,C(=O)(C(O)P(C)(C)=O)NCC(C)CN(C)C(c1cncc2c1CCC2)=O 61092,Cc1c(C(N2CC3CCC3(CC(N3CCCN(C(N)=O)CC3)=O)C2)=O)[nH]ccc1=O 61093,c1(C(=O)NC2CC3(C2)CN(S(=O)(=O)c2cnc[nH]2)C3)ccc2ccccc2c1Br 61094,c1(C(c2n(CCC)nnn2)NC2(C)CC2)c(F)cc(Br)c(F)c1F 61095,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61096,C(=O)(C(F)C(C)(C)O)NC(C)CCNC(=O)CNC(c1ccc(F)cc1)=O 61097,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CC#N)n1)=O 61098,c1(C(N2CCOC(c3ccco3)C2)C(=O)NCCC)ccc2cc(Br)ccc2c1 61099,C(=O)(C1N(C)C1=O)OC.C(=O)(CCOC1CC1)C1(COCCCO)CC1 61100,Cc1cccnc1CCNC(=O)C(Cn1cncn1)NC(=O)C(O)C(C)C 61101,N1(C(CCOCCN(C)C(C23CC(F)(C2)C3)=O)=O)CC2(CCOC2)C1 61102,C(=O)(CCCCC(C)C)N1CCC(C(N(CC#C)CC2CCCO2)=O)(CC=C)C1 61103,C12(C(=O)NCC(C(C)C)NC(=O)COCC3CCCCO3)CCCC(C)(C1)OC2 61104,Cc1cc(=NCCCCC#N)[nH]cc1S(=O)(=O)NC(c1ccc(C)o1)CO 61105,c1(C(c2n(-c3n(C)ncn3)nc(CCCN(C)C)n2)O)ccc2cnn(C)c2c1 61106,c1(C(=O)NCC2C(CC)CCN2C(c2cccn2C(C)C)=O)nc(C)ccc1C 61107,CC1(C)COC(CC(=O)NC2(C[SH](=O)=O)CC(F)(F)C2)CO1 61108,c1(C(C)C)nc(C(=O)NCCN(C(C2CC3CC3C2)=O)CC2CC2)cs1 61109,N1(C(C(C)SCC)=O)CCC(NC(CN(CCCOC)C(C)C)=O)C(F)C1 61110,N1(C(C=C(CC)C)=O)CCc2nc(CNC(C3(C)CC(C)OC(C)C3)=O)sc2C1 61111,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCNC(Cc1c(C)nsc1)=O)CC1CC1 61112,N1(C(C(CCC)OCC)=O)CCC(C2CC2)C1C(=O)NC1CCCC1COC 61113,C1(CN(CCc2cccc(-c3nn[nH]n3)c2)CC)CC2CCC1O2 61114,C1(NC(c2cc3sccc3[nH]2)=O)CC2CN(C(c3ccc(Cl)o3)=O)CCN2C1=O 61115,C1(CNC(CC2ON=C(CC)C2)=O)COC(C)(C)CN1C(c1cc(C)sn1)=O 61116,N12CCC(C)(CC1)C2=O.N1(CC(=O)NC(c2nc(C)sc2)C)CCN(C)CC1 61117,N1(C(=O)CCc2ccccc2)CCOCC1CNC(C12CC(O)C1C2)=O 61118,C1(C(=O)NCCC2(CNC(c3nsnc3O)=O)CC2)(CC)CCCC1 61119,c1(C(N2CC(NC(CCC=C(C)C)=O)C(C)(C)C2)=O)ccc2c(c1)S(=O)(=O)NC2 61120,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61121,c1(C(C)NC(=O)CCn2cc(-c3cccc(C(=O)O)c3)nn2)cccc([N+](=O)[O-])c1 61122,C12(NC(c3cccc4[nH]ncc34)=O)CCC(CC1)N(C(=O)CCCN1CCCC1)C2 61123,C1(CN(C)C(C2CC(=O)N2)=O)CCCN1C(c1csc(C2CCCO2)n1)=O 61124,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2CCOC2)=O)C1 61125,CC(C)(C)C(O)C(=O)N1CC2CC1C2C(=O)NCc1cnn[nH]1 61126,C(=O)(C1=CCCC1C)NCC1(C(=O)NCc2cn(CC)nn2)CCCO1 61127,c1(CN(C(C(CC)OC)=O)C)cc(Cl)cc(Cl)c1F 61128,C1(=O)CCCCNC(=O)C(=O)NC(CCO)C2=CC=CCC12.CC(C)N 61129,N1(C(CC2(OC)CN(C(c3nocc3Cl)=O)C2)=O)CCCN(C=O)CC1 61130,Cc1cc(F)c(N)cc1C(=O)NC(C)CCNC(=O)CC1CCCC1(F)F 61131,N1(C(C(CC#C)NC(=O)CN(C)C2CC2)=O)CCC(C2CC2)C1 61132,c1(OC)cccc(F)c1CNC(C1CCN1C(c1ccc(Br)s1)=O)=O 61133,c1(OCC)ccccc1CSc1nnc(SCC)s1 61134,N(C1c2ccccc2OCC1CO)C(C(=O)Nc1cccc(OCC(N)=O)c1)=O 61135,C#CCCCC(=O)NCCCC(CO)NC(c1ccncn1)=O 61136,N1(C(c2cc(C)c(C)nc2C)=O)CC2CCN(C(=O)C3=CCCC3C)CC2C1 61137,N1(C(c2c(C)ccnc2O)=O)CC2(CCCC2)C1C(N1CCN(C)CC1CCO)=O 61138,C(N=c1nc(N(C)C)c2[nH]ccc2[nH]1)N1C2CCN(C(C3CCC3)C)CC1CC2 61139,C1(CNC(c2c(C)n[nH]c2)=O)CC2(CC2)CN1C(=O)C(C)CN1CCOCC1 61140,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(CC1CCCCC1)OC 61141,C1(N(C(C(C)=CC)=O)C)CS(=O)(=O)C12CCN(C(C1(CC)CCCO1)=O)CC2 61142,C12(C(=O)NCC#CCNC(C(C(C)C)N3CCCC3=O)=O)COCC1C2(F)F 61143,c1(C(=O)Oc2c(OC)ccc(C#N)c2)cccc2c1CCC2NC(=O)OC(C)(C)C 61144,c1(C(C(C(C(=O)NCCC(CN)OC)OC)=O)=O)cc2oc(C)cc2[nH]1 61145,C1(NC(c2coc3c2CSC3)=O)CC2(CCN(C(c3ccncc3)=O)C2)C1 61146,c1(C(N(C)CCNC(c2ccnc3ncnn23)=O)=O)cc2c(=O)cc[nH]c2s1 61147,n1(CC(N2CCC(CN(C)C(C3CCC4CC34)=O)C2)=O)cc(Br)c(O)nc1=O 61148,C1(c2n(CCCSCC)nnn2)(NCc2nn(CC)cc2C)CC2CCCC12 61149,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C)C(C1(C)COCCO1)=O)O 61150,C(=O)(CCCCC(N)=O)N1C(N(C(=O)CNCCOC2CCCC2)C)CCC1 61151,N1(C(C(C)(C)N(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C(O)C1 61152,N1(C(C(C)O)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C(C(F)F)C1 61153,CC(C)CC(F)C(=O)NCCC1(O)CCN(C(c2cc(CCCO)on2)=O)C1 61154,C1(C(C)NC(CSC(C)C)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 61155,C(C)(CNC(=O)C(c1ccc(C)cn1)=O)(CC(C)C)NC(C(C)OCC=C)=O 61156,Cc1c(C(=O)NC2CCN(C(=O)Cc3cccs3)C23CC3)cnc2c(O)nnn12 61157,c1(C(=O)NC2C(=O)N(c3ccccc3)CC2)ncc(Br)cc1OC(F)F 61158,C(C(C)(C)CNC(=O)CCc1cnco1)NC(CC=CC=C)=O 61159,C1(N(C(CC2C(C)C2)=O)C)CCN(C(c2sc(N(C)C)nc2Cl)=O)CC1 61160,C=CCC(CNC(=O)CCCF)C(=O)N(C)CCn1cccn1 61161,Cc1cc(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)c2c(C)noc2n1 61162,N1(C(CC(C)C2CC2)=O)CCCCC1CCC(C)(C)NC(=O)CC1(O)CCCC1 61163,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1cnc[nH]1)C2 61164,c1(C(N2CC3CN(C(C4(F)CCOCC4)=O)C3C2)=O)cc(F)c(Cl)c(F)c1 61165,C(CN=C(NCc1ncccc1C)N1CCC(F)(c2ccccc2F)C1)OC 61166,c1(C(=O)NCC(=CC(NOCCOC)=O)C)ccncc1F 61167,C(C(C(=O)N1CCN(C)C(CO)C1)C(C)(C)C)NC(C1(SC)CC1)=O 61168,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61169,c1(C(C)C)cccc(C(=O)N(C2CCC(NC(=O)CC3CC=CC3)C2)C)n1 61170,c1(C(N2CC(CCNC(CCC(=C)Cl)=O)(OC)C2)=O)coc2ccc(Cl)cc12 61171,N1(C(c2nc(C(C)=O)sc2)=O)CC2CN(C(=O)CC(O)c3ccccc3)CC2C1 61172,C(=O)(C(O)CC(F)(F)F)N1CCCCC(CCC(=O)Nc2c(C(C)C)c[nH]c2)C1 61173,C(C1=CCN(C(=O)C(C2CCCCCC2)O)CC1)NC(C1C(C)OCC1)=O 61174,n1(C(CC)CC)nccc1C(=O)N(C)Cc1cc(N(C)C)ns1 61175,n1(CC(=O)NCCN(C(C(C)Oc2ccc(C)cc2)=O)C)c([N+](=O)[O-])cnc1C 61176,C1(CNC(C(CO)OC)=O)CC2(CC2)CN1C(=O)Cc1cccc(C(F)F)c1 61177,C1(C(=O)NC2CC(CNC(c3cnn(CCF)c3)=O)C2)C2CC3C(C2)C13 61178,c1(C(=O)NCC2CCC(NC(C3C(CC)CCCC3)=O)C2)ccc(C)c(C)c1N 61179,c1(CN2C(CC(=O)Nc3ncc(C)cn3)CCC2)ccc(Br)c2nsnc12 61180,c1(NCCCC#C)ccc(NC(C)C(C#N)CCC)cc1C(F)(F)F 61181,c1(C(=O)NCCCNC(C2(CC#C)CCOC2)=O)cc(O)cc(F)c1F 61182,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61183,C1(CC)CN(C(=O)C(F)(F)C2CC2)CCC1NC(=O)CC1COCC1(C)C 61184,Cc1nc2cc(C(=O)NCC34CCCC3CCN4C(c3cocn3)=O)ccc2o1 61185,Cc1c(C(=O)NCC2CN(C(C3CC(F)(F)C3)=O)CC2(C)C)nn2ccccc12 61186,C(=O)(CCCC(C)(C)CC)NC1CN(C(c2c(CC)nc[nH]2)=O)CC1C(F)(F)F 61187,c1(OC)cc(F)c(-c2nc(CNc3cc(Br)c(C)cc3CO)c(C)s2)cc1F 61188,N1(C(CCCCN(C(=O)C(C)(C)CC2CC2)C)=O)CCC(O)C(F)(F)C1 61189,c1(C(=O)NC2(C(=O)NC(C#C)C)CSC2)cc(C)nnc1C 61190,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61191,n1(CCC(N2CC(NC(C(CC=C)(F)F)=O)C(C)C2)=O)cc([N+](=O)[O-])nc1C 61192,Cc1nnccc1C(N1CCOCC1C(=O)NC1(c2cccnc2)CC1)=O 61193,c1(C(=O)OCCC)cc(NC(=O)NC2CCC(=O)NC2)ccc1OC 61194,c1(C(N2CCC(O)(CNC(c3cncc(C)c3Cl)=O)C2)=O)noc2c1CCCC2 61195,N(C(=NCCF)NCc1ccccn1)Cc1c(C)con1.c1(N)cccc(C)c1 61196,C1(C(N2CC(C#N)C2)=O)CC(F)(F)CN1C(c1cccc(O)n1)=O 61197,c1(CN(C)C(c2cc(CO)[nH]n2)=O)cnn2c1CN(C(C1C(C)C1C)=O)CC2 61198,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61199,CC(C)C(C)CC(=O)NC1CCCC(NC(c2ccoc2C2CC2)=O)C1 61200,c1(OC)cccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C3CC23)=O)c1C 61201,C1(NC(=O)C(C2CCCCC2)F)COC2(CCNCC2)C1 61202,c1(OC)ccc2[nH]cc(C(=O)NC3CC3C(=O)Nc3nc(Cl)nc(Cl)n3)c2c1 61203,c1(NC2C(C)CN(C(C3CCC(C)C3)=O)C2)nc(Cl)nc2ccc(Cl)nc12 61204,CON=Cc1ccc(C(=O)N(C2CCC(NC(c3n[nH]c(C)n3)=O)C2)C)cc1 61205,C#CCC(O)C(=O)N(C)CCN(C)C(c1cc(N(C)C)ccn1)=O 61206,N1(C(C(C=C)(F)F)=O)CCC2(CC1)OC1(CO)CC2(NC(c2cncn2C)=O)C1 61207,c1(C2(C(N(CC(CN(C(Cn3ccc(C)n3)=O)C)O)C)=O)CC2)ccccc1Cl 61208,C(=O)(C1CCSc2ccccc21)NCC(C(C)C)NC(C1CCS1(=O)=O)=O 61209,c1(C(N2CC(C(C)NC(Cn3c(C)ccn3)=O)C2)=O)cnnc(Cl)c1 61210,CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCC1NC(=O)CC=CC(C)(C)C 61211,C(C)(C)(CCCN=c1ccn2ccnc2[nH]1)NC(c1ccnc(C)n1)=O 61212,N1(C(C(c2ccccc2)OC)=O)CC(CNC(=O)CC(C)(O)C2CC2)C(C)(C)C1 61213,c1(OC)ccccc1C(=O)NC(CNC(C1(n2cnnn2)CC1)=O)C(C)C 61214,Cc1nnc2c(N3CC(NC(=O)NC(c4ccco4)C)C3)cc(Cl)nn12 61215,C1(CSCC(=O)NC(CNC(C(=C(C)C2CC2)F)=O)CO)CCCCO1 61216,CCC(CCCC(=O)NCCC(C)C)NC(=O)CN1CCCC1C 61217,c1(C(=O)NCC2(NC(CNC=O)=O)CCCC2)cc(Cl)sc1S(N)(=O)=O 61218,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C)CCN1C(C1CCCO1)=O 61219,Cc1oc(CC(C)C)nc1C(=O)NCC(C)CNC(C1CC1(Cl)Cl)=O 61220,c1(CC(=O)NCC2CCC(NC(Cn3cnc(=N)[nH]3)=O)C2)c[nH]c2ccccc12 61221,O(NC(=O)C(CCF)NC(c1ccncc1OC(C)C)=O)C(C=C)C 61222,CC1CN(C(c2ncc(F)cc2F)=O)CCC1NC(c1nn[nH]c1Cl)=O 61223,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61224,Cc1ccc(NC(N2CCCC(C(F)C(=O)O)CC2)=O)c(O)n1 61225,N1(C(=O)C(C)C)C2CCC1CC(C(=O)NC1N(C(CCC)=O)CSC1)C2 61226,C1(CN)CCc2nc[nH]c2C1.C12(N)CNC(=O)C(C1)C2.C1CCNC(=O)N1 61227,Cc1nccnc1C(C(=O)NCCCOCC(=O)OC)N(C1C=CCC1)C 61228,C1(CC(=O)Nc2cn(CCOC)nc2)CCCCC1(F)F.C1C(=O)NCCS1 61229,C1(NC(=O)CCNC(=O)NCC(F)(F)F)CC12CCc1ccccc12 61230,C(=O)(C1=CCC(C)CC1)N1C(CC2c3nnnn3N2)CCC1.N1(CC)CCCC1 61231,CC1CC(NC(c2ccc(CO)o2)=O)CN1C(c1ccccc1Cl)=O 61232,C1(C(=O)NC(C(=O)N(C)C)Cc2ccccc2)CCCN(CCc2ncc[nH]2)C1 61233,c1(C(=O)NC(C)CCCCNC(c2ccc(Cl)cn2)=O)n[nH]cc1[N+](=O)[O-] 61234,CC(COc1ccc(Cl)s1)C(=O)OC1CCCCC1 61235,c1(CCN(C(C=CC(C)NC(=O)C(F)C2CCC2)=O)C)ccccc1 61236,C#Cc1cncc(C(=O)NC2CC(NC(=O)C(C)OC(c3ccccc3)=O)C2)c1 61237,CCC(C)C(CC(=O)NCCC1CC(C2CC2)C1)NC(=O)COCC1CCCC1 61238,c1(C2CCCN(C(C(=O)NCCC3C(C)C3)C3CCSC3)C2)ccccc1C#N 61239,CC(Cc1ccccc1)C(=O)NCC(O)CNC(C1CCN1C)=O 61240,N1(C(C(C)(C2CC2)NC(C)=O)=O)CCC(CCNC(=O)C(C)CC2CCCC2)CC1 61241,c1(N(C)CCc2ccccn2)nc(=N)nc(NCC(c2ccccc2)F)[nH]1 61242,C(CC(C(=O)N1CCCC(OC)C1)NC(=O)CCCSC)OCC.OC 61243,N1(C(C(CCSC)O)=O)CC2CCCC(CNC(C3CC(C)(C)CCO3)=O)C2C1 61244,C1(C(N(CCCC(C)C)C)=O)CC(NC(=O)CCC2CCOC2)CCO1 61245,C1(C(N2C(C)(COC)CC2)=O)CC(N=[N+]=[N-])C1.C12CC(C1)CCNC2=O 61246,c1(C2(C(N3C(CNC(C(C4CCCO4)SCC)=O)CC3)=O)CC2)ncc(C)s1 61247,C#CCC(CC(=O)NC1(c2ccccc2)CCN(C(=O)CC(C)=C=C)C1)C1CC1 61248,C#Cc1ccc(C(=O)NC2CC(C)CN(C(c3cnc(O)o3)=O)C2)c(OC)c1 61249,c1(-c2n(-c3c(OC)cc(C)cc3)nc(C(C)OC)n2)noc2ccc(Cl)cc12 61250,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(C)O)CC2)C(C)C)c1 61251,N1(C(C2C(OC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61252,C1(CC)(NC(c2ccc(F)s2)=O)CCN(C(=O)CN2CCC2C)CC1 61253,C(=O)(CC(=O)N(CCCn1cc(CC(=O)O)nn1)C)N(C)C 61254,C1(C)(C2CCCC(C(=O)NC3(n4c(C)csc4=O)CC3)C2)NC(=O)NC1=O 61255,Cc1cc2ncc1S(=O)(=O)N2.N1(CC(C)N(C2(C)CC=CC2)C)CCCCC1 61256,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61257,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61258,C(=O)(CCCC(=O)NC1CCCN(C(=O)NC2CC3C=CC2C3)C1)NC 61259,c1(C(=O)NCCC2(NC(CCCC=C)=O)CCC2)coc2c(F)c(Cl)ccc12 61260,c1(C(N2CCC(O)(C(C)NC(C=C(C)C(C)C)=O)CC2)=O)cccn2nccc12 61261,N1(CC(=O)NCC2CC(NC(Cc3cc(C)[nH]n3)=O)C2)CCS(=O)CC1 61262,c1(C(C)F)ccc(C(=O)NCC2CCN2C(C2(C3CCCO3)CC2)=O)cc1 61263,C12(C(=O)NC(CN(C(C(C)NS(CC)(=O)=O)=O)C)C)CC=CC(C1)OC2 61264,c1(CNC(C2(NC(C(C)S(N)(=O)=O)=O)CCCC2)=O)cc2cc[nH]c2cn1 61265,c1(C(=O)NCC2OCC(CNC(c3ncn(CC)c3)=O)C2)c[nH]c2ccccc12 61266,N1(C(=O)CC2(N3CCCC3)COC2)CCC2CCCN(C(c3ccsc3)=O)C2C1 61267,c1(C(CC)C)nc(C)cc(=NCC2CN(C(c3cnc(C(N)=O)s3)=O)CC2C)[nH]1 61268,c1(C(C(=O)NC(CC=C)C)NC(=O)CC(C)NC=O)cccc(F)c1 61269,CC1COCCN1C(c1cccc(C(=O)NCCC#N)c1)C 61270,C(=O)(C1=CC(O)C(NC(c2ccc(C)cc2C)=O)C1)NCCOCC(=O)OC 61271,C(=O)(C1=CCCCCC1)NCC1C(C(N2CCN(CC)C(=O)C2)=O)CCO1 61272,C(C(O)C(=O)NC1CCC(CCC(=O)NCCN(CCCF)C)C1)=CC 61273,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61274,c1(OC)ccc2c(ccn2CC(=O)NCC(C)CN(C(=O)C(C)OC)C)c1 61275,Cc1cc(C(=O)NCCN(C)C(C2(O)CCC(C(F)(F)F)C2)=O)n(C)n1 61276,c1(OC)ccc(CCNC(=O)C(C)OC2(OC)CCCC2)cc1O 61277,c1(OCC)cnc(C(=O)NC2CCCC(NC(c3cc(C)cs3)=O)C2)c(Cl)c1 61278,Cc1cc(-n2cc(C3CCCN3C(C3CC(C(F)(F)F)C3)=O)nn2)ccc1Br 61279,C1(NC(C2C(C(=O)OC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61280,C1(CCNC(C2(OC(C)C)CCOC2)=O)CN(C(c2cccn2C)=O)CC1C 61281,N1(CCc2cn(-c3ccc(CC)cc3)nn2)C(=O)C2C(O)CCN2C1=O 61282,C1(NC(=O)NC2(c3ccccc3F)CCCC2)CC(=O)N2CCCCC12 61283,c1(N(CCN(C(C)C)C)C)cccc(S(=O)(=O)NC2CC2C)n1 61284,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)NCc1nnc(CC)s1 61285,C(=O)(CCC(C)(C)C)NCCN(C(C12CC1CNC2=O)=O)CC 61286,N1(C(c2c(C)nc(C3CCCOC3)s2)=O)CC2=C(C1)CN(C(c1ccns1)=O)C2 61287,C(C)(CC(C(=O)NC1CCN(C(C)=O)CC1)N1CCC(CCC(C)C)C1)SC 61288,N(C(=NCCN(C)C)NCC12CCCC1OCC2)C1CCC(C(=O)OC)CC1 61289,c1(C(CC(=O)NCCCOCCNC(C(CC=CC)C)=O)O)cc(Cl)cc(Cl)c1 61290,C#Cc1cncc(C(=O)NC(C(=O)NC(C#C)Cc2cn[nH]c2)C2CCCO2)c1 61291,CC(C)CC(C(=O)N1CC(NC(=O)CC2CCC(=O)N2)CC(C)(C)C1)C(C)C 61292,CC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccnc(-n3cccc3)c2)=O)C1 61293,N1(C(C(CCCNC(c2ncc(C)c(C)c2)=O)(C)C)=O)CCC2CCC(O)C1C2 61294,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61295,CCC(O)C(C)C(=O)NCC1CC(NC(=O)C(=Cc2cccs2)C)C1 61296,c1(CNC(C)=O)ccc(C(=O)NC(C)CCNC(c2ccn(C(F)(F)F)n2)=O)s1 61297,C=CCCC(C(=O)NC(C)(C)C=C)NC(=O)CCCCNC(C)=O 61298,n1(C(CC)C)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CN2CCOCC2)C1 61299,C12CCC(C1)C(=O)N2CCC1CC1.C1CCN(CCC)C1.S(=O)(=O)(CC1CC1)CN 61300,C1(CNC(=O)CC2CCS2(=O)=O)CCN(C(c2cnn(CCF)c2)=O)C12CC2 61301,c1(C(=O)NCC(c2ccccc2)NC(=O)Cc2cnoc2)ccc(F)cn1 61302,N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(C)O)C2 61303,Cn1cnc([N+](=O)[O-])c1NCC1CC(C)(C)CCC1C(F)(F)F 61304,CC1CC(C(=O)NC2(CC3CCC3)CC2)CN(C(c2ccn(CO)n2)=O)C1 61305,C1(NC(C2CC(C)(C(C)C)C2)=O)C2CC3C(C2)C13C(N1CCN(C(N)=O)CC1)=O 61306,Cc1noc(C)c1C(=O)NC(CNC(C1CC(n2ccnc2)C1)=O)CO 61307,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61308,N1(C(C2OCCN(C)C2)=O)CCC(F)(CNC(C2CC2(C)C)=O)CC1 61309,C1(CCNC(c2csc(Cl)n2)=O)CN(C(=O)CCCc2ccccc2)CCS1(=O)=O 61310,c1(C(=O)NC2CC(C)N(C(=O)COCc3cccnc3)C2)cccc(S(C)=O)c1 61311,c1(C(C(=O)NC2(C(N(CCSC)C)=O)CCC2)F)ccccc1 61312,c1(C(N(C)CCNC(=O)CC2CCC3(CCC3)O2)=O)cnc(O)c([N+](=O)[O-])c1 61313,c1(C(N2CCCC(Nc3ncccn3)C2)=O)cccc2sncc12 61314,CC1CCCC(C)N(C(C2CCC(CNC(=O)Cn3ccnn3)C2)=O)C1 61315,c1(C(=O)NC(C(C)NC(C2CCCS(=O)(=O)C2)=O)CO)ccc2ncccc2c1 61316,CN1CCN(C)C(CNC(=O)NC2CSCC2c2ccc(Cl)cc2)C1 61317,CC(C)C(Cc1ccccc1)C(=O)NCC1CN(C(c2cccnn2)=O)C1 61318,C1(NC(C(C)C(F)F)=O)CN(C(=O)Cc2cccc(O)c2F)CCC12CCC2 61319,Cc1ccc(C(=O)NCCCN(C(=O)CC2(C)CC2(F)Cl)C(C)C)c(O)c1 61320,Cc1nn(-c2ccccc2)cc1NC(=O)Cn1nccn1 61321,n1(CC2N(C(=O)C(O)Cn3cncn3)C2)nccc1C1(CC(=O)OCC)CC1 61322,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CC(C)(C)CN(C)C)C1 61323,Cc1nn(C)c(C)c1CC(=O)NCC1CCC(C)CN1C(=O)CCC1OCCO1 61324,CCC(C(=O)NC(CCCNC(C1CC1c1ccsc1)=O)c1ccccc1)SC 61325,c1(C(C)C)ncc(C(=O)NC2CCN(Cc3nc(-c4ccccc4)cs3)C2)[nH]1 61326,Cc1ccc(CC(N2CC(NC(c3cc(C)n(C)c3)=O)C3CC23)=O)cc1C 61327,c1(C(N2C(CNC(C3(O)CC(C)(C)C3)=O)CC(OC)C2)=O)c(C)ncn(C)c1=O 61328,C(=O)(CCCC(=O)NC(C)(CNC(c1coc2c1CCC2)=O)C(C)C)NCC 61329,C(=O)(C1Cc2ccccc21)NCC=CCNC(c1nccc2nn[nH]c12)=O 61330,c1(C(=O)NC2C(CNC(c3ccc(COC)o3)=O)CC2)cc(Cl)ccc1O 61331,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2C(C)SCCC2)=O)CCCC1 61332,C1(CNC(c2c(C)ccnc2)C2(C(=O)OC3CCCCC3)CC2)CCC(C)(C)CO1 61333,C(CCCCC(=O)N(C(C)CNC(C1CCC(OC(F)(F)F)CC1)=O)C)OCC 61334,N1(C(C2(C)CCCN(C(=O)CC(Cl)Cl)C2)=O)CC2CCNCC2C1 61335,C=CCC(CC)C(=O)N(C1CN(C(=O)CC(C)C(F)F)C1)C.C1(=O)CCN1 61336,CC1CC(c2ccccc2)CCN1C(=O)CCc1cn(C)cn1 61337,N1(C(c2c(C(C)C)cco2)=O)CC(C(=O)NCCn2cc(CO)nn2)=C(F)C1 61338,CC#CCCCC(=O)N1CCC(C(=O)NC2(CSC)CC2)C1 61339,C(CN=c1cc(C)[nH]c(=NCCOCC2CC2)[nH]1)(C1CCOCC1)OC 61340,C1(CNC(C2(N(C)C)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCO1 61341,N1(C(C(C)S)=O)CCc2cc(C(=O)NCC(C)(C)CCCl)ccc2C1 61342,S(=O)(=O)(c1cccc(F)c1)N(C1CC2CNC1C2)C(c1cccc(C)n1)CC 61343,C(=O)(CP(C)(C)=O)N(CCN(C(=O)COc1ccc(Cl)cc1)C(C)C)C 61344,CCCC(O)C(CO)NC(C1CCCC(NC(=O)CCCN(C)C)C1)=O 61345,C(=O)(N=c1[nH]nc(CC(C)C)s1)C1(COC)CCCCO1 61346,n1(CC(=O)NC(C2C(c3c(OC)cccc3)C2)C)cnc(C)cc1=O 61347,c1(OC)ccc(F)c(OC)c1C(=O)NCC(C)NC(=O)CCCNC(N)=O 61348,c1(C(=O)NC2CCC(NC(c3ccc(CC)c(N)c3)=O)C2)cncc2c1CCC2 61349,C1(NC(C=CC(CC)C)=O)CCC2CCN(C(=O)Cc3cc(C)cs3)C12 61350,CC1(C)CCN(c2nc(Cl)ncc2Cl)CC1CNC(c1nc(Cl)cs1)=O 61351,c1(CC(=O)N(C2CCN(C(C34CC(C)C3C4)=O)CC2F)C)ccc(O)c(Cl)c1 61352,c1(CC)ncnc(N2CC=C(CNC(C3(C)CCC(F)(F)C3)=O)CC2)c1F 61353,C1(F)(CNC(C2(C)CCOC2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61354,C12CC3CC1CN(C3)C(c1nccc(C(F)(F)F)n1)C(=O)N2.C(C(C)SC)OC 61355,C1(C(N2CCN(CC(c3cn(C)nc3)=O)C(=O)C2)=O)CCCN(CP(C)(C)=O)C1 61356,c1(C(N2C(CC)CN(C(=O)COC3(C)CCC3)CC2)=O)cc(C)c(C)nc1C 61357,C1(O)(C(=O)NCCCCc2cn(CC)nn2)CCNC1.C(C)(=O)N 61358,c1(C(N2CCCC(CNC(c3ccc(Cl)c(Cl)n3)=O)C2)=O)cnn2ccncc12 61359,C(=O)(C(CCCC(=O)OC)N1CCC2(CCSC2)CC1)NCCOC 61360,C1(OC)(CO)CCN(C(=O)C(CCN(C)C)NC(C2CSCC(=O)N2)=O)C1 61361,S(=O)(=O)(c1nc(NC2CCC2C)ccc1Br)N1CC(C)NC(=O)C1 61362,CC(C)(Cc1cnn[nH]1)C(=O)NC1CN(C(C2CS(=O)C2)=O)C(COC)C1 61363,N1(C(C2(CNC(=O)Cc3cnoc3)CC(=C)C2)=O)CCN(C)C(CC2CC2)C1 61364,c1(C(=O)NC2C(CNC(c3cnc(OCC)s3)=O)C2)ccccc1C(N)=O 61365,c1(NCC2(F)CCCCCC2)noc2c1COCC2 61366,Cc1ccc(CC(=O)NC2CC2NC(=O)C(C(C)C)NC=O)cn1 61367,C1(C(N(C(C)C(C)(C)O)C)=O)CC(=O)OC1C(C)(C)C 61368,c1(C(=O)NCCNC(C(c2ccccc2)NC(CC)=O)=O)n[nH]c(CC)n1 61369,C1(COC)CN(C(c2cnn(C)c2N)=O)CCN1C(c1ncccc1Br)=O 61370,c1(C(N(CC(C)NC(C2(C(=O)OCC)CC2)=O)C)=O)ccc2nnnn2c1 61371,c1(-c2nc(CCC)oc2)nc(C(c2ccccc2)C)nn1CCC 61372,N1(C(CCSCC=C)=O)CCCC(N(C(=O)CN(C)C(C)=O)CCF)C1 61373,C1(CC(=O)NCCN(C(=O)CCOc2cccnc2)CCC)COCC(C)O1 61374,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61375,C(C(=O)N1CC(O)(CN(C)C(C2CCSC2)=O)C1)(C(C)(C)C)NC(C)=O 61376,C12(C(N3CC(C)(NC(c4ccn(C(C)(C)C)n4)=O)C3)=O)CCCC1CS(=O)(=O)C2 61377,C1(=O)CCC(C)(C)C(=O)NCC2(F)CCC(C2)N1.CCC(C)C(=O)OC(C)(C)C 61378,C(=O)(C(F)(F)CC1CC1)N1CCC(CC(=O)NC2(C(C)C)CC(OC)C2)C1.CO 61379,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CNC(c1ccn(C)n1)=O 61380,c1(SCC(=O)N(CCCNCCNC(c2ccccn2)=O)C)ccccc1O 61381,CN1CCN(C(=O)CN2CCCNC2=O)CC1CNC(C1CC(F)(CO)C1)=O 61382,c1(OC)cc(C(N2CC(NC(c3sc(C)cc3Cl)=O)C(C)C2)=O)cc(N)c1N 61383,Cc1ccn(C)c1C(=O)NCC1(C(=O)NCCCCCN=[N+]=[N-])CC12CCC2 61384,c1(CCC2(C)CCOC2)cc(F)cc(Cl)c1.CC(C)S 61385,N1(C(C(C2CN(C(CC)=O)C2)O)=O)CCCOCC1 61386,c1(CNC)cccc(F)c1F.c1(C)cn(C(c2ccno2)C2CCCC2)nn1 61387,N1(C(=O)C=C2CCCC2)CCC2(CCCN(C(=O)Cc3ccc(O)nc3)C2)CC1 61388,c1(C(N(CCCNC(CC)=O)CC)=O)cc2c(OC)c(F)ccc2[nH]1 61389,S(=O)(=O)(c1ccn(C2CC2)n1)N1CC(C)(NC(=O)CN)OCC1 61390,C1(NCC2(NC(=O)CCC(C)C)CC2)CCCN(C(C)=O)C1 61391,N1(C(C(C)NC(=O)C(O)CN(C)C)=O)CCC(O)C12CCCC2 61392,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61393,C12(C(=O)NCC(CN(C)C(C3(C(F)F)CCC3)=O)O)COCC1C2(F)F 61394,c1(CNC(C2C(C)(C)CO2)=O)cccc(CNC(C23CCC(OC)C2C3)=O)c1 61395,c1(N(C(C)=O)C)ccccc1C(=O)NC1CCC(NC(c2nnc(C)s2)C)C1 61396,C1(C(=O)NCC2(CNC(C(C)O)=O)CCC2)(N(C)C)CCOCC1 61397,N1(C(C2CCC(N(C)C)CC2)=O)CC2CC1CN2C(=O)CN(CC(C)(C)C)C 61398,c1(C(=O)NCC2C(C(=O)NCC(C3CC3)OC)CCO2)nccc2cc[nH]c12 61399,C(=O)C(F)C(CC)CC.C(C)(C(=O)NCCN(CCOCCO)CC)O 61400,N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61401,C1(C(=O)NCC2CN(C(C(CC=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61402,Cc1cn2cc(C(=O)NC(C)CC(C)NC(C34CCN(CC3)CC4)=O)nc2s1 61403,C1(COC)(CNC(c2cn(C(C)C)nn2)=O)CN(C(C2CC2F)=O)C1 61404,C1(NC(C(C)OCCOC)=O)CCC12CN(C(=O)CSc1nncn1C1CC1)C2 61405,c1(SC)cc(C(=O)NC(CO)CC(O)c2ccccc2)ccn1 61406,C1(CNC(c2c(C)nn[nH]2)=O)CCCCN(C(C2COC(C)(C)CO2)=O)C1 61407,C1(COC)(NC(=O)CCCn2cccn2)CCN(C(c2ccc[n+]([O-])c2)=O)C1 61408,C1(CCNC(c2cnc(C)s2)=O)CCCCN1C(=O)C(F)Cc1ccccc1 61409,c1(N(C(C(C)CO)=O)C2CNCC2(F)F)nc2ccccc2s1 61410,N1(C(C2(C)C(C)CCCC2)=O)CCC(C(=O)N2CC(CNC(N)=O)C2)=C(F)C1 61411,CCC(CC)C(C)C(=O)NC1CCCCC1N(C)C(C1CCCCO1)=O 61412,c1(C(=O)NCCC2(O)CCN(C(C3(C#C)CC3)=O)C2)cc(OC)cc(Cl)c1 61413,c1(C(=O)NCC2N(C(CSCC(=O)OC)=O)CC2)cc2c(nn1)CCC2 61414,C1(C(=O)NCC(CNC(C(CCC)(C)C)=O)(C)OC)CCc2cnnn2C1 61415,c1(C(=O)CC)ccc(C(F)F)s1.C1(NC(c2cnc[nH]2)=O)CC(c2ccccc2)(N)C1 61416,c1(OCC)ccc(C(=O)NCCCN(C(=O)CCn2ncn(C)c2=O)CC)cc1 61417,C1(NC(C2(c3ccc(Cl)c(F)c3)CCCC2)=O)CC2CC1N(C(=O)CN1CCC1)C2 61418,CC1(C)CC1(Cl)C(=O)NCC1CCCN1C(c1cc(C2CCOCC2)no1)=O 61419,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61420,c1(C(N2C3C(NC(c4nc(C)n(C)n4)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61421,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3CCC(=O)N3)=O)CCC2C)=O)c1)NC 61422,N1(C(C(n2nnc(-c3ccccc3)n2)C)=O)CCN(C(=O)C=CCO)CC1CO 61423,c1(C(C2(CCNC(=O)OC(C)(C)C)N=N2)C)cccc(Br)n1 61424,C1(CN(C)C(c2c[nH]c(C(F)(F)F)c2)=O)CCN(C(C23CC2C3)=O)CC1 61425,C(C)(CNC(c1cnc(S)nc1)=O)(CC(C)C)NC(CC(=O)NCC)=O 61426,c1(COC(C)C)ccc(C(N2CC(NC(C3CCCC3C)=O)C2)=O)cc1 61427,C(=O)(C(C)CCCC(C)C)NCC1C(C(=O)NCC(=O)NCC#C)C1(C)C 61428,C1(N(C(C2C(CC)CC2)=O)CC)CCC(NC(=O)C(CC2CC2)OC)CC1 61429,c1(C(C(C)C)NC(=O)NC2COCC2F)ccc(C(F)(F)F)cc1 61430,Cc1cc(NC(=O)CCCCCN(C(=O)C(C)S(N)(=O)=O)C)cc(Cl)c1 61431,C1(NC(CC(=C)Br)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1F)C2 61432,CC1CCC(C)CN1C(c1ccc(CNC(=O)CN2CC3CCC2C3)nc1)=O 61433,c1(C(=O)NCC2(NC(C(c3ccc(Cl)cc3)C)=O)CCC2)csc2c1CCCC2 61434,C1(CC(=O)NCc2ccccc2Cl)CCCCN1C(CC(C)n1cc(Br)cn1)=O 61435,c1(CCC(=O)C(N2CCN(C(CN(C)CCO)=O)CC2)=O)nnc(S)nc1O 61436,C(=O)(C1=NN(CCO)C(=O)CC1)N1CCC(NC(c2c(C)cc(CC)o2)=O)C1C 61437,C1(C(N(c2ccc(Cl)cc2)CCOC)=O)CCc2nnc(C)n2C1 61438,C1(CC(=O)N(c2cn(CC)nc2)C)CCCN(C(=O)CCCC2CC2)C1 61439,N1(C(c2ccc(C)cc2)=O)C2CCC1C(C)C(NC(=O)CCC(C)O)C2 61440,C1(NC(CCOCCOCC)=O)C2CC3CN(C(C45CCN(CC4)C5)=O)C1C3C2 61441,c1(OC)cc(C(=O)N(C(C)CNC(c2cnc(C(C)C)o2)=O)C)cc(F)c1F 61442,c1(NC(C2(C)CN(C(c3cncc(F)c3)=O)C2)=O)cnc(I)cn1 61443,N1(C(=O)COc2ccc(Cl)cc2Cl)CCC2OCCN(C(C3CC=CC3)=O)C2C1 61444,c1(CNC(C(C)N(C)C)=O)ccc(CNC(C2CC3CC2CO3)=O)c(F)c1 61445,C1(CCC(=O)NC(CC)CC2CC2)CCCCC1 61446,c1(OC)cc(N)c(F)cc1C(=O)N(C(C)CCNC(C1CCC2(CC2)C1)=O)C 61447,c1(CCCNC(C(n2cc(N(C(C)C)C)nn2)C)=O)ccc(O)cc1C 61448,C1(CNC(C23CCC(C2)C(C2CC2)N3)=O)CC2(CCCC2)CO1 61449,C1(C)(C(N(CCCC(=O)NCc2nnnn2C2CC2)C)=O)COCCO1 61450,C1(=CC(=O)N(CC(CC)NC(C(C)OCC)=O)CC)CCC(C(C)(C)C)CC1 61451,C(C(CC(C)C)C(=O)NCC(C)(O)CC(C)C)NC(c1n[nH]c(CC)c1C)=O 61452,C1(NC(c2c(C)coc2)=O)CC2(CCN(C(=O)C#CC3(C)CC3)CC2)C1 61453,c1(C(=O)NC(CNC(C2(c3ccno3)CCC2)=O)CO)cncc([N+](=O)[O-])c1 61454,Cc1cnc(C(=O)NCC(C)(O)CNC(c2c[nH]c(=N)s2)=O)cc1Br 61455,C1(F)(CNC(C(C)(C)n2cnnn2)=O)CCN(C(c2csc(C#N)c2)=O)CC1 61456,C(C(CC1CCCC1)C(=O)N1CCC(C(C(C(OC)OC)=O)=O)C1)N 61457,c1(CC)ccc(C(N2CC(NC(=O)C3=CC(C)CC3)C3(CC3)C2)=O)cc1[N+](=O)[O-] 61458,CCN=c1cc(C(N2CC(O)(CN(C)C(c3ccc(O)c(F)c3)=O)C2)=O)cc[nH]1 61459,C1C(CC(C)C)NC(=O)c2ccc(cc2)-c2cn1nn2.c1(SC)ccncc1F 61460,n1(CC(N2CC(F)(CNC(=O)C3=NNC(C(F)F)C3)C2)=O)cc(Cl)c(O)nc1=O 61461,c1(OC(C(=O)N(CCC)CCNC(=O)CC(C)F)C)ccc(Cl)cc1C 61462,c1(SC)ccc(CN2CCC(C(N3CCN(CC(F)(F)F)CC3)=O)CC2)cc1 61463,c1(N2CC(C)OC(C3CC3)C2)[nH]c(=NCCS(C)=O)nc2scnc12 61464,C1(SC)CCCC1C(=O)NCC1(CC2CCN(C(C)C)C2)CC1 61465,C(=O)(CCC(F)(F)C(F)F)NCCCCC(C)NC(CC(C)OC)=O 61466,C(=O)(C1=CC2CCCC12)NCCOCCN(C)C(c1cnn(C)c1Cl)=O 61467,N1(CCC)CCC(C(C)NC(CONC(=O)C2(COC)CC2)=O)CC1 61468,C1(NC(CCCC)=O)CN(C(C2CCn3c(cnc3C)C2)=O)C2(CCCCC2)C1 61469,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61470,C12(CNC(c3c(C)nn(C)c3)=O)CCC(C1)N(C(C1CCC3CCC1O3)=O)C2 61471,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61472,C1(NC(CCC(C)C)=O)CC=C(C(=O)NCC2CCOC2=O)C1 61473,n1(CC)cnc2c(NC(C)C)[nH]c(=NCC(C(C)(C)C)N3CCOCC3)nc12 61474,C12(C(N(C)CC3(F)CCC3)=O)CC(CO1)N(C(C1OCCC1C)=O)C2 61475,CC1(NC(C23C=CC(CC2)C3)=O)CCN(C(c2cc(CO)on2)=O)C1 61476,Cc1cccc(C)c1OCC(=O)NCCC(C)NC(c1cn(C(C)C)cn1)=O 61477,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3nc(C)oc3C)=O)CC12 61478,CC1(C)CC(NC(c2snnc2C2CC2)=O)CCN(C(=O)Cc2ccsc2)C1 61479,C#Cc1cn(C)nc1C(=O)NCC1(NC(=O)COc2cc(C)ccc2F)CCOC1 61480,n1(-c2cc(C)cc(Br)c2)nc(O)c2c1NC(=O)C(c1ncccn1)O2 61481,c1(C(=O)NC(CCCC)CNC(=O)C(n2ccnc2C)C)cc(F)ccc1C 61482,c1(NCCCO)nc2ccccc2nc1N1CC2CSCC(C2)C1 61483,C1(NC(CC=CC=C)=O)CCN(C(=O)Cc2ncc(C)o2)C1(C)C 61484,Cn1c(O)nc2cc(C(N3C4CCC3CC(NC(C3(CO)CC3)=O)C4)=O)ccc12 61485,CN(CCCC(=O)NCC1(F)CCN(C(=O)CCc2nc(N(C)C)no2)C1)N=O 61486,c1(NC(C)CCO)[nH]c(=NCc2nc(Br)n(C)n2)nc2c1cnn2C 61487,C(=O)(CS(=O)(=O)C1CC1)NC(C)(CNC(c1ccccc1C1CCC1)=O)C1CC1 61488,C(c1cccnc1)=CC(=O)NCC1CCC(C(=O)NC2(c3onc(C)n3)CC2)O1 61489,N1(C(C2CCCC2)=O)CC2CCCN(C(=O)CSC(F)F)C2C1 61490,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1CNC(c1c[nH][nH]c1=N)=O)OC 61491,C1(N(C(C2(OC)CCCOC2)=O)C)CCCN(c2ccnc(CO)n2)CC1 61492,C1(C(=O)NCC2(F)CC(NC(=O)CC3OCCO3)C2)CCCn2cncc2C1 61493,C(=O)(N1CC(C)(O)CO1)c1cc(CNC(C2C(C(=C)C)OCC2)=O)on1 61494,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61495,c1(-c2cc(C(N3CCC(N(C(CC)=O)C)C3)=O)n[nH]2)cc(Cl)c(O)c(Cl)c1 61496,N(C)(C1CCc2c(F)cccc21)C(C(n1ncc(C#N)c1N)C)=O 61497,C1(CC(=O)NC(CCN(C(=O)Cc2cnco2)C)(C)C)CCCCC(=O)N1 61498,CC1(C)C(NC(=O)C(C2CCCCC2)F)CCN1C(=O)CC(F)(F)Cl 61499,N1(C(COC2C(CC)C2)=O)CC(NC(=O)CCNS(=O)(=O)CC)C(C)(C)C1 61500,C1(CNC(c2ccc(OC)c(F)c2Br)=O)(CO)COCC2CCCCN12 61501,c1(C(=O)NCC(C2CCC2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CCCC1)C2 61502,C1(NC(C(CCC)OCC)=O)COC2(C1)CN(C(c1cc3c([nH]1)CCCC3)=O)C2 61503,c1(C(N2CC(C)C(CNC(C3CCC=CO3)=O)C2)=O)cccc(Cl)c1N 61504,c1(OC)ccc(CC(N2CCN(C(C3Cc4nnsc4S3)=O)CC2C)=O)cc1F 61505,CC(CN=c1nc(C(C)(C)C)[nH]s1)N(C(=O)CC1CC2(CCOCC2)CO1)C 61506,C1(CNC(C2CCCC3CC23)=O)CCN(C(c2nnc(O)nc2O)=O)C12CCC2 61507,c1(C(N2CCN(C(C(CC=CCC)C)=O)C(C)C2)=O)cnc2c(C#N)cnn2c1 61508,c1(C(=O)NC(C2CCCN2)CC)ccc(CNC(=O)C(=O)N(C)C)s1 61509,c1(C(=O)NC(CN(C(C=CC2C(C)CCC2)=O)C)(C)C)nc(F)ccc1Cl 61510,C1(C(N(CC(C)(C)NC(=O)C=CC2CCCO2)C)=O)CCCC(=O)N1 61511,c1(N2CCN(C(c3cccc(N)c3)=O)CC2)nc2ccc(Br)cn2c1Cl 61512,C(=O)(C(C)(C)CN=c1[nH]c(=NCCOCC(F)F)[nH]c2cccnc12)NC 61513,C1(COCCNC(=O)CC2CCOC2)C2CN(Cc3ccncc3)CC12 61514,C1(C(=O)OCCC2CCC(CO)CC2)CC(C2CCC2)C1 61515,Cc1c(CC(=O)N(CCNC(=O)C2=CC(C)(C)C2)C(C)C)c(O)nc2[nH]nc(O)c12 61516,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61517,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)CO)n2)c(C)s1 61518,CC1(C)CCN(C(=O)CC2CSCCO2)CC1NC(=O)C(C1CCCCC1)=O 61519,CC(C)(O)C(NC(=O)CC1CC1(C)C)NC(=O)COC1CCCCC1 61520,C(N=c1ccc(C#N)c[nH]1)C1CCN(C(c2c(Cl)cn(CCC)n2)=O)C1 61521,C1(NC(COCC(=O)OC)=O)(CNC(C2CCC(=O)N2)=O)CCCCC1 61522,Cc1ccc(-c2cn(CCN(C(=O)C(F)n3ccnc3)CC3CC3)nn2)c(F)c1 61523,c1(C(=O)NCCCN(CC2(C)ON=C(C)C2)CC)coc(S(N)(=O)=O)c1 61524,C(C(C)C(F)(F)F)N(C(C1(C2N(C(CC3(C=C)CCC3)=O)CCC2)CC1)=O)C 61525,c1(C(=O)NCC(C2CCOC2)NC(=O)C=CCO)cnsc1 61526,CCN=C(NCc1cnn(C)c1C)N1CCC2(CCCC2)CC1 61527,CCC(C)C(C(=O)NC1CN(N2CCN(C(C)=O)CC2)CC1C)OC.C1(C=O)CC1(C)C 61528,CN1CCN(C(C2CNC(=O)N2)=O)CC1CNC(c1ccc(-c2ccco2)o1)=O 61529,Cc1oc(S(N)(=O)=O)cc1C(N1CC2(CCN(C(c3nocc3C(C)C)=O)C2)C1)=O 61530,CCS(=O)(=O)c1cccnc1NCC1CCCC12CCCO2 61531,C(=O)(C(C(C)(C)C)NC(=O)CC1CNC(=O)C1)NCCC=CCCC 61532,C1(CC2CCCC2)C(=O)N1C1CC1C.CCC 61533,N1(C(c2n(C(C)C)ccc2)=O)CCOC2(CCCN(C(C3(O)CCC3)=O)C2)C1 61534,c1(C(=O)NC2(CO)CN(C(CC3CNC(=O)O3)=O)C2)cc2n(n1)CCO2 61535,[SH](=O)(=O)C1CCCC1(F)F.CC1CC(O)CN1 61536,c1(C(C(=O)NC(C)CC2CCCN2c2cc(F)ncn2)(F)F)ccc(F)c(F)c1 61537,c1(OC)cccc(CN(C)CCOCCN(C)C(C2CC=CCC2)=O)n1 61538,c1(NC(=O)NC(c2ccc(N3CCCS3(=O)=O)cc2)C)ncc(C(F)F)cn1 61539,C1(CCNC(C2N(C(C)=O)CCC2)=O)CCN(C(C2(O)CN(C)C2)=O)CC1 61540,c1(C(=O)NC(C2CCN(C(=O)CCNC(=O)N(C)C)C2)(C)C)ccc2c(c1)OCO2 61541,CCC(CC(=O)NC1CCC(NC(=O)C(c2cccc(OC)c2)C)CC1)C(C)C 61542,c1(NC)cncc(C=CC(N2CCC23CN(C(c2cnc(OC)cn2)=O)C3)=O)c1 61543,C1(C(=O)OCC(c2ccccc2)OCC)CC(c2ccccc2)CN1 61544,CCCCC(C(=O)NCC1CCCCN1C(c1c[nH]nc1OCC)=O)C(C)C 61545,c1(C(=O)NCC(O)CNC(=O)C(F)CC2CCC2)nc(Br)n2ccccc12 61546,N1(C(CN(CC)CC)=O)CC2CCC2(CNC(c2c(C)ccnc2O)=O)C1 61547,C12(COC)COCCN1OC2=O.c1(NC(=O)OC(C)(C)C)c[nH]c(Br)c1 61548,C1(OCC=C)CCCCC1N=c1ccnc(Nc2cn3ccc(C)cc3n2)[nH]1 61549,n1(CCCN(C(C2=CC(C)(CC)C2)=O)CC)nc(O)c2ccccc2c1=O 61550,N1(C(c2cc(CC)on2)C(=O)NCCOC(F)F)CCCC(O)(C(=O)OC)C1 61551,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61552,n1(CCOC)nnnc1C(CCSC)NCC1CCCO1 61553,CC1(C)CCN(c2ccc(C#N)cn2)CC1.C1(=O)CCCn2cc(nn2)CN1C 61554,C(CCCC(O)C(=O)O)NC(=O)N(c1nc(CC(F)(F)F)cs1)CCO 61555,C(=O)(C#CC1CCCCO1)NC1C(CC)N(C(c2ccc3ccoc3c2)=O)CC1 61556,c1(SCC(=O)N(CCNC(c2cnsn2)=O)CC2CCCC2)ccc(F)cc1Cl 61557,N1(C(c2cnc(CC)s2)C(=O)NC(C)(C)CC)CC(=O)Nc2ccc(C#N)cc21 61558,c1(C(=O)NC(C(C)C)CNC(=O)CCc2cncnc2)cccnc1O 61559,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C)(C1CC1)OC)CCC1CC1 61560,c1(CC)nc(C(=O)NC(C)CN(C(=O)CCCNC(N)=O)C)c(Br)s1 61561,CC(CC(C)NC(=O)CC1CC2CCC1O2)N=c1nc(CN(C)C)[nH]s1 61562,CC(C)CCCC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61563,c1(C(=O)NC2CCCN(C(C3(C)C=CCC3)=O)CC2)cncc2c(O)nccc12 61564,C1(C)(C(=O)NCC(NOCC(C)(C)O)=O)CNC(=O)C1 61565,C(C(C)(C)CNC(=O)CCN1CCCC1=O)NC(C(C)NC(CC)=O)=O 61566,C1(N(C)C)CCC(C(N2CCCC2c2csc(CNC(C3CCO3)=O)n2)=O)CC1 61567,c1(C(N2CCC(NC(=O)C=Cc3ccccc3)CC2)=O)cc(OC(F)F)ncc1Cl 61568,C12(NC(c3c(SC)csc3)=O)CCCC1CN(C(=O)Cc1ccc(C(C)C)s1)C2 61569,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61570,C1(NC(c2c(Cl)cnc(C)n2)=O)COC2(CCCN(C(C3CCS3(=O)=O)=O)C2)C1 61571,C=C(NCc1cc(OC)no1)NC1CCOc2c(C)cccc21.OC 61572,N1(C(CCCCC(C(=O)OC)=O)=O)CCCC(O)(C(=O)OC)C1 61573,c1(OC)ccc(C(C(=O)NC2(C)CC2)N(C)Cc2ccccc2OC)nn1 61574,CCC(C(=O)OC)C(=O)NC(C)CCNC(c1cn(C(C)C)nc1C(F)(F)F)=O 61575,c1(C2CC(C=O)C2)cc(O)n[nH]1.C(C)(C)(C=CC)N(C(C)=O)CC 61576,O(NC(=O)CCCOCC(=O)NCC1CC1)CCCC 61577,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(=O)C(C(C)C)C3CCC3)C2)C1 61578,C1(CNC(C2(C(=O)OC)C3CC4C(C3)C24)=O)CCCCN1C(c1ncncc1Cl)=O 61579,CC1=C(C(=O)NC2C=CCN(C(=O)C3=CCCO3)C2)C(C)n2ncnc2N1C 61580,c1(C(=O)Nc2occ(C(=O)OCC)c2)c(C)nc(C(C)C)nc1O 61581,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)Cn2c(CCC)nnc2S)CC1 61582,n1(CC(C)C)nc(-c2ccoc2)nc1C(C)N(C)C.c12noc(n1)C2 61583,CC(C)CC(C(=O)N1CCC(C(=O)N(C)Cc2cocn2)CC1)N(C)C 61584,CC1N(C(=O)CC2N(C(C3CCCSC3)=O)CCC2(C)C)CCOC1(C)C 61585,C=C(C)C(CC(=O)N1CCC(F)(CNC(=O)CCCC2CC2)C1)OCC 61586,c1(C(N2CCC(CN(C(=O)CN3CCCC3C)C)C2)=O)cccc2sccc12 61587,C1(C)(OCC(=O)NCCCSC)CN(C(c2sccc2C)=O)C1 61588,Cc1cc2ncnc(NC3CC4CN(C(c5c(Cl)cnn5C)=O)CC34)c2[nH]1 61589,C(C(CNC(C1C2(CC2)C12CC2)=O)S(C)(=O)=O)NC(C(c1c(C)cccc1)C)=O 61590,c1(C(N(CC(C)NC(c2c(C)cc[nH]2)=O)C)=O)cc2ncn(C)c2cn1 61591,N1(C(c2cc3ccccc3nn2)C(=O)NC(C)C)CCNC(=O)C(F)(F)C1 61592,C1(CC)(CC)CC(NC(=O)C(O)C(F)(F)F)CN1C(c1ccn(C2CCC2)n1)=O 61593,c1(N2CC3CN(C(CCS(=O)(=O)NC)=O)CC3C2)cccc(F)c1[N+](=O)[O-] 61594,C1(C(=O)NCC2(CNC(CCC(C)OC)=O)CCCC2)Cc2nncn2C1 61595,CCCCCCCC(=O)N1CCCC1CCC(=O)OCC 61596,c1(C(=O)OC2CCC(CC)CC2)cc2cc3c(cc2[nH]1)OCCO3 61597,C1(O)(C(C)NC(C(CSC)C)=O)CCN(C(c2cc(Cl)cnc2C)=O)CC1 61598,C1(NC(CNC(=O)NC)=O)CN(C(C2(C)SCCCS2)=O)Cc2cccn2C1 61599,O=C(C(F)(F)C(F)n1ccnc1)NC(c1ccc(F)cc1)c1ccc(Cl)cc1 61600,c1(CNC(=O)CSCC2CCCCO2)ccc(C)cc1.C(=O)(CCc1cnc[nH]1)N 61601,CC(O)C(F)(F)C(=O)NC1CC(CNC(=O)Cc2ccc(C(F)(F)F)nc2)C1 61602,c1(CC(N2CC(CNC(C3CCC4CC4CC3)=O)C2)=O)c[nH]c2cccc(Cl)c12 61603,c1(N2CCC(C=C)C2)nc(N2CCC3(CCC(=O)N3)C2)nc2ccsc12 61604,c1(C(=O)NCCOCCCN(C(c2cc(CC)[nH]n2)=O)C)cc(F)ncc1OC 61605,C1(c2nnnn2C2CC(F)(F)C2)(Nc2c(COCC)cccn2)CCCC(C)(C)C1 61606,c1(N2C(CNCc3ccc(C(=O)OCC)o3)CCC2)ncnn2cc(Br)cc12 61607,c1(-c2nc(C3CCCC3)on2)c[nH]c(C(=O)NC2CC2CNC(C2(Br)CC2)=O)c1 61608,c1(C(c2nnnn2C2COC2)(C)OCC(C=C)OC)c(Cl)cc(F)cc1Br 61609,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 61610,N1(C(C2(CC)CCCN2C(=O)COc2ccccc2)=O)CCC(=O)N(C)CC1 61611,c1(C(C)(C)C)ccc(C(N2CCC(F)(C(=O)NCCC(F)(F)F)C2)=O)cc1 61612,CC1CC(=O)NCC1C(N1CCC(CC(=O)Nc2cncc(C(F)F)c2)CC1)=O 61613,C1(C(=O)NCCCCCC)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 61614,N1(C(=O)CSC(F)(F)F)CC2(C1)CN(C(=O)C=CCNc1ccccn1)CC2CO 61615,N1(C(C(=C)C)=O)CCCC(C(N2CCN(c3ccccc3)CC2)=O)C1 61616,N1(C(C(C)SCC)=O)CCCC(C)(C)C1NC(C1CCCN1C)=O 61617,CON=Cc1ccc(C(=O)NC2CCC(NC(=O)C(C)CCCC(C)C)C2)cc1 61618,c1(NC(C2SCCN(C(COC(C)(C)C)=O)C2)=O)c(F)ccc(F)c1Cl 61619,CCCCCCC(=O)NC(C1CCCC1)CNC(c1ccncc1C(F)F)=O 61620,Cc1cc(CNC(N2CCN(C3CC4(C3)CN(C)C4)CC2)=O)c(N)cc1F 61621,C(=O)(C1=CCS(=O)(=O)C1)NCCOC1CCN(C(c2nn(C)c(=O)cc2)=O)C1 61622,C(=O)(C1=CCCC1P(C)(C)=O)NC(C(C)NC(c1c(OC)cncc1)=O)CO 61623,c1(C(=O)NCC2C(NC(C(C(C)C)(C)O)=O)CCC2)cccc2cc[nH]c12 61624,C1(CC)CCCCN1C(=O)C(O)C1CN(C(=O)CCOCCOC)C1 61625,C1(CC(N2CCN(C(c3c[nH]c(=N)o3)=O)CC2)=O)Oc2ccccc2NC1=O 61626,N1(C(C2CC(=C)CN2C(=O)CCCSC)=O)CC2(C)CC1CCO2 61627,c1(OC)cc(C(=O)NCC(C(C)C)NC(C23CCC(F)(CO2)C3)=O)cnc1OC 61628,c1(CC)c(NC(C2CCCC2NCc2cc(Br)ccn2)=O)csc1C 61629,c1(-c2nn(C(CC)C)c(C(F)C3CC3)n2)ccc(N(C)C)c(F)c1 61630,C1(C)(C(=O)NCC2CCN(C(C)(C)C)C2)CCN(C(c2coc(Br)c2)=O)C1 61631,N1(C(C(CC2CCC2)NC(CC2C(C)(C)OCC2)=O)=O)CCC2(CCCO2)CC1 61632,CN1CCN(C(C(=O)NCC2CCCO2)C2CC2Cl)C(CN(C)C)C1 61633,C(=O)(CCCCC(C)(C)C)N1C2C(C(N(OC)C)=O)C(CC2O)C1 61634,C1(C)(NC(C2(NC(CC(C)C3CCCO3)=O)CC2)=O)CCOC(C)C1 61635,Cn1cnc2[nH]c(C(=O)NC3(CNC(=O)C(C)(C)F)CCC3)cc12 61636,c1(OC)cccc2cc(C(N3CCN(C(C4CC(OC)C4)=O)C(CF)C3)=O)[nH]c12 61637,N1(C(=O)CCN2C(=O)CCC2=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C2C1 61638,C(C(=O)NC1CCC(F)(F)CC1)(C(C)CC(C)(C)C)N(CC#C)C(C)C 61639,c1(C(=O)NC2C(NC(C3C(C)C3)=O)COC2)cccnc1O 61640,CCCCCCCCC(=O)Nc1cccc(S(=O)(=O)NCC(=O)NC2CC2)c1 61641,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 61642,C#CCC1(C)C(=O)N2CCC(O2)C(=O)N1CC.C(C)(C(F)F)=CCOC 61643,C1(C(NOCCCC=C)=O)CN(C(=O)CC=C(Cl)Cl)CC1C 61644,c1(C(N(C(C)CNC(c2cc3n(c2)CCSC3)=O)CC)=O)ccc(C)c(F)c1F 61645,Cc1cccc2c(C(=O)NCC3(C)CCCN(C(=O)Cc4nc[nH]n4)C3)coc12 61646,C(C(C)(O)C(=O)N1CC(n2cnnc2)C1)OC.C1C(C)(C)CC(=O)N1 61647,C1(NC(=O)CCn2cc(-c3cccc(Cl)c3)nn2)CC(C(=O)O)C12CCC2 61648,N1(C(CC(CN(C)C)NC(=O)CCc2cocn2)=O)CC2(CNC(=O)OC2)C1 61649,C1(CC)CCc2sc(C(=O)OCC3CN(C(=O)OC(C)(C)C)C3)cc2C1 61650,c1(C(N(C(C(C)NCC(C)C)=O)C(C)C(N)=O)C)ccccc1 61651,C1(NC(c2c[nH]nc2C=Cc2ccco2)=O)CC(OC(F)F)CN1 61652,C(c1ncc[nH]1)=CC(=O)NCCN(C(=O)C=Cc1cscn1)C 61653,CC1CNC(=O)CN1C(c1ccc(CO)s1)C(=O)NCc1cccc(Cl)c1 61654,Cc1cc(C)c2[nH]nc(C(N3CC(O)CCC3CO)=O)c2c1 61655,N12CCC(C(O)C1)C2.Cc1cc(C)n(-c2ccccc2OC(=O)C=C2CCC2)n1 61656,C(CCC(CCC)NC(=O)C=Cc1cncc(F)c1)NC(C(C=C)N(C)C)=O 61657,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 61658,C(=O)(C1=C(C#N)CCC1)N1C(CNC(COc2cccc(C)c2F)=O)COCC1 61659,CCC(C)(C)C(O)C(=O)N1CCC2CC1CN2C(c1ccc(Cn2cccn2)o1)=O 61660,N1(C(c2cccnc2CO)=O)CCC2(CC1)CN(C(C1C3CNC(=O)C13)=O)C2 61661,C1(CN(C)Cc2cn(-c3cncc(F)c3)nn2)COCCN1C(=O)COC1CC1 61662,C1(C(N2CCC(CF)C2)=O)(CNC(=O)CCc2cn[nH]c2)CC(F)(F)C1 61663,CC1(C)CC(C(N2CCC2c2cccc(Br)c2F)=O)CC(C)(C)N1 61664,c1(CC)ncc(C(=O)NC(C)CCN(C(=O)Cc2cccc(O)c2F)C)c(C)n1 61665,N1(C(C(=O)NCC)Cc2cccc(I)c2)CCN(CC(=C2CCCCC2)F)CC1 61666,CCCCC(C(=O)N1CCN(C)CC1C(=O)NC(CCC)C1CCCC1)C(C)C 61667,c1(C(N2CCC(N(C(C(C)NC(=O)OC)=O)C)C2)=O)ccc(O)nc1C 61668,C1(CNC(CC2CCC(C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CCCO1 61669,N1(C2(C(=O)OC)CC2)CCC(CNC(CC2(NC(C3SCCC3C)=O)CC2)=O)CC1 61670,C1(NC(COC(CC)(C)C)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 61671,N1(C(c2cc(O)n[nH]2)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ccc12)=O 61672,C1(C(=O)NCC2(CO)CCN(C(CC)=O)C2)CC(=O)NC(=O)N1.CC=O 61673,c1(C(=O)NC(C2CCN(C(=O)CSCc3cccs3)C2)C)ncc(Cl)s1 61674,c1(C(=O)NCC(CNC(CC(=O)NCC)=O)(C)O)c(C)cc(OC)cc1C 61675,C(CC(CNC(=O)CC1(C)CCC1)NC(c1cnnn1-c1ccccc1)=O)OC 61676,Cc1cnc2nccc(C(=O)NC(CNC(C3(O)CC3)=O)C(C)(C)C)c2c1 61677,Cc1nn(CCO)cc1C(=O)NC1CC(NC(=O)C(C)(O)C2CCOCC2)C1 61678,c1(SC)nc(N2CCC(CNC(c3cc(N(C)C)ccc3F)=O)C2(C)C)ncc1C 61679,CC(C(=O)NCC1(NC(=O)CC2CCCC(F)(F)C2)CCCC1)S(C)(=O)=O 61680,Cc1csc(C=CC(=O)NC2(C)CCN(C(=O)CCc3cncc(O)c3)C2)n1 61681,c1(C(c2cnn(C)c2)CC)nc(CC2CCC2)nn1-c1cccc(Cl)c1 61682,Cc1cc(C)c(NC(C2CCC(NCc3ccn(C)n3)C2)=O)c(Br)c1 61683,Cc1ccccc1C1(C(=O)NC2CCCC2)CC1.N12CCC1C2 61684,C1(NC(c2cccc(C(F)(F)C(F)(F)F)c2)=O)(CO)CCN(C(C2CC2(F)F)=O)C1 61685,Cc1cccc(C)c1OCCC(N1CCN(C(=O)CCc2nncs2)CC1C)=O 61686,c1(C(=O)NC23CC(NC(c4csc(C(F)F)c4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 61687,C(=O)(CC(C)C(C)(C)C)OCCN(C(C1C(C(C)C)CCO1)=O)C 61688,c1(CC)nc(=NC(C)CNC(=O)COCc2ccccc2)s[nH]1 61689,c1(OC)cc(C(=O)NC2CCC2CNC(C2CC2C(C)C)=O)cc2cccnc12 61690,N1(C(C(F)(F)C2(OC)CCC2)=O)CC(N(C)C(C2CC3(CC3)CO2)=O)C(F)C1 61691,c1(OCC)ccc(OCC)c(C#N)c1.C1(CN(C(=O)C)C)CCCO1.C1C(=O)O1 61692,CC1CN(C(=O)C(C)(Cl)Cl)CC(C)N(C(C2CCC3(CC2)N=N3)=O)C1 61693,c1(C(=O)NC2C(C)CN(C(C3CCCC3(C)C)=O)C2)cn2c(n1)SCC2 61694,C#CCCCC(C)C(=O)NCCN(CCOC)C(c1cc2cn[nH]c2cn1)=O 61695,C12(C(=O)NCC(CC)(C)CO)CCC(NC(c3cnc(C)cn3)=O)(CC1)C2 61696,N#Cc1cccc(NC(C2(CNS(=O)(=O)c3cn[nH]c3)CC2)=O)c1[N+](=O)[O-] 61697,N1(C(C2(C)CC(C)C2)=O)CCCCC1CNC(=O)CCc1ccc(F)cn1 61698,Cn1cc(CNC(N2CCCCC2c2cccs2)=O)c(Cl)n1 61699,c1(N2CCC(C(C)NC(=O)Nc3nnnn3C)C2)cccc2cnccc12 61700,C(=O)(CCCCCC#N)NC(CC#C)C(=O)N(C(C)C(C)(C)C)C 61701,CC(C)(C)C(Br)C(=O)N1CCCCC1Cn1cc(CCS(=O)(=O)N2CCCC2)nn1 61702,Cc1ncc(Cl)cc1CNC(=O)CCn1cc(C2CC(N3CCCCC3)C2)nn1 61703,c1(C(=O)OC)cncc(CNC(=O)C(C2CCOC2)NC(=O)C=CC2CC2)c1 61704,Cc1cc(C(N2CCN(C(C3CC3c3ccc(O)cc3)=O)CC2C)=O)cnc1Cl 61705,N1(C(C(C(C)C)F)=O)CCCOC(CNC(C2SC3C=CC2CC3)=O)C1 61706,C1(C(=O)NC2(COC)CN(C(C3CNC(=O)C3)=O)C2)C2CC3C(C2)C13 61707,c1(C(=O)NC2CN(C(c3c(=N)[nH]cnc3)=O)C(CO)C2)ccc(F)c(Cl)c1 61708,C(=O)(C(C)S(C)(=O)=O)N(CC(C)CNC(=O)COc1nn(C)cc1Br)C 61709,C(=O)(CCCC(=O)NC1COCCC1NC(c1cnc(C(C)(C)C)nc1)=O)OC 61710,c1(OC)cc(OCCOC)cc(N2CCCN(Cc3cccc(C)c3O)CC2)c1 61711,c1(CC)nsc(N)c1C(=O)N(C)CCC1CCN(C(=O)C(C)(C)C)CC1 61712,N1(C(C=CC(CC)=CC)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 61713,CC(C)C(C(=O)N(CCCNC(c1c[nH]c2cccnc12)=O)CCO)C(C)C 61714,CCCCC(C(=O)NCC1CCCCN1C)NC(=O)CCCSC 61715,C1(NC(C(C=C)O)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 61716,c1(NC(N2CCCC(C(=O)OC)C2)=O)cc(N(C)C)cc(F)c1F 61717,N1(C(c2c(OC)ccnc2)=O)CCOC(C)(CNC(C2CN(C)CCO2)=O)C1 61718,c1(CCC(=O)NCC(CC)N(C)C(C2CCOC(C)C2)=O)ccc(SC)cc1 61719,c1(C(=O)NC(CCN(C(c2c(C)[nH]nc2Cl)=O)C)C)ccc(S(C)=O)cc1 61720,C1(CNC(C2(C(C)C)CCCO2)=O)CC2(CCC2)CN1C(C1CC(=O)N1)=O 61721,C1(C(=O)NCCC(C)CCNC(c2c[nH]nc2Br)=O)(CC)CCOCC1 61722,C1(=O)C(CC2CCC2)NC(=O)CO1.C1(C)(O)CCCC1.C1(C(C)C)(OC=O)CC1 61723,N1(C(C(C)=CCC)=O)CCC2(CC1)CC(NC(C1CCC(C(=O)OCC)C1)=O)C2 61724,N1(C(CC(C)OC)=O)CCC(NC(=O)CSc2nnnn2C2CCCC2)C12CC2 61725,Cc1ccc(N)c(C(=O)NC(C2CC(NC(=O)CO)C2)C)c1 61726,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(=O)CC2CCC2(C)C)C1 61727,C#Cc1cc(C(=O)NCCN(C(=O)C(C)(C)COC)CC2CC2)cc(F)c1 61728,C#CC12CC(CN1C(C1(COC)CN(C(=O)C(C)CC(C)C)C1)=O)C2 61729,C(C(=O)N=c1cc[nH]cc1I)C1N(C(c2n(C)ncc2I)=O)CCC1 61730,C1(C(C(=O)NC(N2CCOCC2)CC)NC(=O)Cc2cncs2)CCOC1(C)C 61731,c1(-c2cn(C3CC(C(N(C45CC(C4)C5)CC)=O)C3)nn2)ccnc(F)c1 61732,c1(OC)cc(C=CC(N2CCCCC2c2n[nH]cc2C(N)=O)=O)sn1 61733,c1(C(=O)OC)cc(OC)cc(CNC2CCOC(C)(C)C2)n1 61734,c1(OC)cc(NC(C2CN(C(=O)CSC)CCN2C)=O)ccc1F 61735,C1(c2n(CCCCCC)nnn2)(NC(C)CCC=C(C)C)CC2CCC(C1)N2 61736,C1(NC(C=CCC(C)(C)NC(Cn2c(C)ncc2)=O)=O)CCSC(C)C1 61737,C1(NC(CCn2ncn(C)c2=O)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 61738,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 61739,C1(F)(CNC(C(CC)c2ccccc2)=O)CCN(C(c2sccc2C)=O)C1 61740,N1(C(c2cnn(C)n2)=O)CCC(C2CCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 61741,c1(COC)ccc(C(=O)NC(CNC(=O)CCOCCCC(C)C)CC)cc1 61742,C#CC1CCCN(C(c2ccc(C(=O)OC)nc2C)C(=O)NCCOC)C1 61743,c1(CC(N2C(C)C(NC(=O)CN(C)S(=O)(=O)N(C)C)CC2)=O)cc(F)ccc1O 61744,N1(C(C(CC#C)(C)C)=O)CC(NC(c2cc(OC(F)F)n(C)n2)=O)C(C2CC2)C1 61745,c1(CNC(c2ccccc2F)(C(=O)OC)C)cc(Cl)c2c(c1)OCCO2 61746,c1(C(=O)OC)ccc(C(=O)NCCCC(C)NC(=O)C=Cc2cc[nH]n2)o1 61747,N1(C(C2(C(=O)NC)CC2)=O)CC(CCNC(c2c(SC)cnn2C)=O)C(C)C1 61748,c1(C(=O)NCCC(F)(F)F)cccnc1CNC(=O)CNC(C1CCC1)=O 61749,C1(OC(C)(C)C)CN(C(=O)CSC2CC2)CC1CNC(C1(F)CCCOC1)=O 61750,C(N=c1cc(-c2ccccc2)nc[nH]1)C1C(NC(c2cn(CC)nc2)=O)CCC1 61751,c1(CC2N(C(c3c(CNC(=O)CN)cco3)=O)CC2)ccnn(C)c1=O.CN(C)C=O 61752,CCCC(CNC(C1CC1(F)F)=O)NC(c1cn(C2CC2)cn1)=O 61753,N1(C(c2ccn(CCC)n2)=O)CC2(CCC2)CC1CNC(=O)CS(=O)CC 61754,Cc1cc(S(=O)(=O)N2CCC(N3CCCNC3=O)C2)ccc1N1CCCS1(=O)=O 61755,N1(C(C=CCC)=O)CC2CC1CN2C(c1cccc(-c2cnn(C)c2)n1)=O 61756,C1(NC(C2CC(C)CN2C(=O)CSC(F)(F)F)=O)CC(C)N(C)CC1C 61757,CC(CCN=c1[nH]cnc2cc(F)c(F)cc12)NC(c1cc2n(n1)CCOC2)=O 61758,CC1CCN(C(=O)C(=O)N(CCCNC(C2CC2c2cn[nH]c2)=O)C)C1 61759,N1(C(C)C(=O)NC(C(N2CCCCCC2)=O)c2cccs2)CCC(C(C)CO)CC1 61760,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)NC(C1(CCCC)CC1)=O 61761,C(=O)(C(F)C(F)(F)F)NCC1CCC(NC(c2csc3cncn23)=O)CC1 61762,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC(CO)C1 61763,C#Cc1ccc(C)c(NC(C2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)c1 61764,CC1CN(C)C(C)CC1NC(c1cn(CCNC(=O)C(C)(O)C2CC2)nn1)=O 61765,c1(C(N(C2CN(C(c3ncoc3C(C)(C)C)=O)C2)C)=O)cc2sccc2n1C 61766,Cc1[nH]nc(C(N2CCOCC2CNC(=O)C(O)C2CC2)=O)c1N 61767,C12(C(N3CCC(C(=O)OCC)C3)=O)CCN(CC1)CC2.C1(COC=O)CC1CN 61768,c1(CNCCN(N(C)C2CC2)CC)ccc(S(=O)(=O)NC)cc1C#N 61769,c1(C(N2CCN(C(C(C#N)C3CC3)=O)CC2)=O)sc2ncccc2c1Cl 61770,c1(C(=O)NCCN(C(c2ncc(C)c(Cl)c2)=O)CC2CC2)cc2n(c1)CCSC2 61771,c1(C(=O)NCC2(CN(C(c3ccc(C)s3)=O)C)CC2)ccc(Cl)nc1N 61772,c1(OCC2(C(=O)OC)CNC2)nc2ccccc2o1.C12CC(F)CN(C1)C2=O 61773,C1(NC(Cc2nc(C)sc2)=O)CCC(NC(=O)CN(C2CCSC2)C)CC1 61774,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 61775,C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CCCCN(C)C 61776,C1(NC(c2c(C)cccc2)=O)CC(NC(c2ccc(CO)c(F)c2)=O)C12CCC2 61777,C1(NC(c2ncc(OC)cc2F)=O)COC2(CCC2)C1NC(=O)C1CC1 61778,C1(c2nnnn2CCC2CC2)(N)CCCCCC1F.Cc1nc(C2C3COCC23)n[nH]1 61779,N1(CC)CC(c2nnnn2CC2(C)CC2)(NCCCc2nccs2)CCC1=O 61780,C1(C(=O)NC(C(C)(C)NC(CC=CC=CCCCCC)=O)C)CNC(=O)N1C 61781,C1(CNC(C(O)=CCC)=O)CCCC1NC(c1cc(C(=O)OC)[nH]n1)=O 61782,C1(NC(c2c(O)nnc(C)c2C)=O)CCN(C(=O)COC(C)(C)C)CC12CCC2 61783,C(=O)(C(O)C(C)(C)C)NCC(C)(C(C)C)NC(C1(C(=O)OCC)CCC1)=O 61784,C(=O)(CCCC(C)C)N(C)CC1CCN(C(C(C)OC)=O)C1 61785,c12ccc(c(Cl)c1)-n1cc-2nn1.C1(CC)CC(CNC(=O)OC(C)(C)C)CC(C)O1 61786,CCCCC(C)N=c1[nH]c(N2CCN(CCC(C)(C)C)CC2)nc2c1CSC2 61787,C(CCCOC)(C(=O)Nc1cc(F)ccc1OC(F)F)NC(C(COC)C)=O 61788,N1(C(Cn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]cc2Br)C1 61789,CN1CCCC(C(=O)N(CC(N)=O)CCNC(c2[nH]ccc2C2CC2)=O)C1 61790,C(=O)(CCCC(C)(C)C#N)NC1CC(O)C1(C)C.c1(OC)cc(O)c(Cl)cc1S 61791,N1(C(c2c(OCCCC)cccc2)=O)CC2COCCC2(NC(=O)CCF)C1 61792,n1(CC(=O)NC2C3CN(C(Cc4c(C)nc[nH]4)=O)CC32)nc2ccccn2c1=O 61793,C1(C(=O)NCC(=O)OC)C2CCC(C2)N1C(C1(C)CCN(C)C1)=O 61794,N1(C(c2c(OCC)cccc2)=O)CCC2(CCCN2C(=O)CCc2cccs2)CC1 61795,c1(C(N2CCC(NC(CCC#CC)=O)CC2)=O)cc(OCC)ncc1Cl 61796,c1(CC)cc(C(=O)NC2CN(C(=O)CCC(C)(C)OC)CC23CC3)ccc1C 61797,CCC(CNC(=O)CC(C)CNC(c1nccnc1C(N)=O)=O)(CC)OC 61798,c1(CCC)cc(C(N2CCC(C(C)NC(c3cnc(CC)n3C)=O)C2)=O)nn1C 61799,N1(C(C(C)(F)F)=O)CCCC(N2CCN(C(C3C=CCC3)=O)CC2)C1 61800,c1(C(=O)NC2CC(NC(c3c(CCC)occ3)=O)C2)nc2n(c1Cl)CCCC2 61801,c1(C(=O)NC(CNC(C)=O)(C)CO)cc2c(s1)CC(C)(C)C2 61802,n1(C(CC)C)nc(C(=O)NCC2CCN(C(C3OCCOCC3)=O)CC2)cc1C 61803,c1(C(C(=O)N(CCCOC)CC2CC2)N2C3CCC2C3)nc(C(C)(C)C)ccn1 61804,C1(NC(c2c(CC)noc2)=O)CCN(C(c2ccccc2C2(C)CC2)=O)CC1C 61805,N1(C(c2cccc(-c3ccncc3)c2)=O)CCC(c2ccc(SC(F)(F)F)s2)CC1 61806,c1(C(=O)NCc2c(C(N3CC(CC#C)OCC3)=O)[nH]cc2)cc(C)nc(C)n1 61807,c1(NC(CNC(CCCN(C)C)=O)=O)ccccc1Oc1ccccc1 61808,C(=O)(CCCCC(C)C)NC(CCCCNC(C(C(C)C)OCC(C)C)=O)C 61809,C1(N(C(C(CC=C)(F)F)=O)C)CCCC2CN(C(=O)CC(C)(C)CC)CC12 61810,CCN=C(NCC1(C)CC1(F)F)N1CCc2c(Br)cccc2C1 61811,C1(O)(C(C)NC(=O)CC(C)c2ncco2)CCN(C(C2(CF)CCC2)=O)CC1 61812,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 61813,c1(NC)c(C(=O)NCC2(O)CN(C(C3CC4CCCC34)=O)C2)cccc1N 61814,C(=O)(C(C)CCCc1ccccc1)NCC1CCC(NC(C2C(CC)C2)=O)C1 61815,C1(C)(CNC(c2n(CC#C)cnn2)=O)CC(OC)CN1C(=O)CCCCCOC 61816,C1(NC(C#CC(C)(C)C)=O)CC2CC1CN(C(C1CC3(C1)CC(C#N)C3)=O)C2 61817,C12(C(=O)NCC=CCNC(C(C)NC(c3ccco3)=O)=O)CCCN(CCC1)C2 61818,N1(C(C=C2CCN(C)CC2)=O)CCCN(C(c2ccc(Cl)nc2N)=O)CC1 61819,CN1CC(C)(C(=O)NCCOCCN(C)C(c2nnn(C)n2)=O)CC1=O 61820,C1(CC(=O)NCC(C)O)COC2(CCN(Cc3ccc([N+](=O)[O-])cc3Cl)CC2)C1 61821,c1(OC)ccccc1OCCCC(=O)OCC(c1ccccc1)O 61822,N1(C(COCCC#C)=O)CCCC(F)(C(N2CCS(=O)C(C)C2)=O)C1 61823,c1(CC)cccc2c(CC(=O)NC3(C)CCN(C(C4(CCF)CC4)=O)C3)c[nH]c12 61824,c1(C(C2CC2)OC)ncc(NC(N2CC3C(C2)C3(C)C)=O)c(C)n1 61825,Cc1nn(CC(C)C)c(Cl)c1C(=O)NC1CC(C)N(Cc2ccccc2F)C1 61826,c1(C(=O)NC2CCC(NS(=O)(=O)c3ccc(Cl)s3)CC2)cc(Cl)nc(Cl)c1F 61827,CCCC(CNC(c1cc(Cc2ccccn2)[nH]n1)=O)NC(C1(O)CCC1)=O 61828,C(=O)(C(C)Cc1ccccc1)NCCN(CCOC)C(c1cnc(C(C)C)[nH]1)=O 61829,C1(C(=O)NC(C2CN(c3cnc(F)cn3)C2)C)CCC(N(C)C)CC1 61830,n1(CC(=O)NCC(C)(O)CNC(C2(CC(F)F)CC2)=O)cnc2c(N)ncnc12 61831,c1(C(=O)NCC(c2ccc(F)cc2)NC(C=CC(CC)C)=O)ncc(Cl)nc1Cl 61832,C1(NC(=O)CC2(c3ccccc3)CC2)COC2(C1)CN(C(=O)C1=CCCOCC1)C2 61833,N1(C(CC(C)c2ccco2)=O)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC1C2 61834,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 61835,N1(C(CSC2C(=O)OCC2)=O)C2CCCC1CN(C(c1csc(S)n1)=O)C2 61836,c1(C(=O)NCCOCCNC(c2c(C)nc(N)cn2)=O)cccc2scnc12 61837,c1(C(=O)NC(C(CCC)C)C(=O)OC(C)(C)C)n[nH]c2c1CONC2=O 61838,CC1CCCC(OC(C)C(N2CC3C(NC(=O)C=Cc4cnn(C)c4)C3C2)=O)C1 61839,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CCC2N(C(C2CCOC2)=O)C3)c1 61840,CC1CC(=O)NC(C(=O)NCc2cccc(NC(=O)C(=O)c3ccsc3)c2)C1 61841,N1(C(C2(F)C(C)C2)=O)CCc2[nH]nc(CNC(=O)C(c3ccc(F)cc3)O)c2C1 61842,CC(O)CCN=c1[nH]c(N2CCC(N3CCOCC3)C2)nc2c1COC2 61843,c1(SC)ccccc1-n1nc(CCO)nc1CC(F)(F)F.C(=O)CO 61844,c1(C(=O)OC(C)C(=O)Nc2cc(O)nc(=O)n2C2CC2)cc(F)c(F)cc1I 61845,C12(CCN3CCN(C(c4ccc(OC)cn4)=O)CC3)CCC(CC1)C2(C)C 61846,c1(CCC=O)c(C)noc1C.C(=O)(C(C)Cc1cccnc1)N(C(CC)C)CC 61847,C1(C(=O)NC2C(C(=O)OC)CC2)C(C)(C)CCN1C(=O)C(=Cc1ccccc1)C 61848,Cc1nc(C(=O)NC2(C(N3CCOCC3)=O)CCCC2C)c(C)o1 61849,c1(C(=O)NCC(=O)NC2CCC2C(=O)NC2CCCCC2)cccn1C1CC1 61850,C(C(O)C(F)(F)F)NC(C1N(C(c2cncc(OCCF)c2)=O)CCC1)=O 61851,N1(CC(=O)NCC2N(C(CCCSC)=O)CCC2C)CCN(C)C(=O)C1 61852,C=CCC(C(=O)N(C1CCN(C(c2ccc(SC)s2)=O)CC1)CC)C(C)C 61853,c12ccc(cc1)NC2(C)C.C1(OC)CCCC1C(=O)OCc1cccs1 61854,N1(C(C2(F)C(C)C2)=O)CC(NC(c2csc(-c3ccco3)n2)=O)C(O)C1 61855,C1(NC(C(C)OCCOC)=O)CN(C(c2ccnn2CC#N)=O)C(C)(C)C1 61856,CC1CC2(CCN(C(=O)CCc3ccc(S(C)=O)cc3)CC2)CN1C(c1ccccc1)=O 61857,C=CC(C)(O)CC(=O)N(C)CCN(C(=O)CCC1CCCCO1)C 61858,c1(C(N2CCCCC(NC(=O)C=C3CCOCC3)C2)=O)cc2n(n1)CCCN2 61859,CC1(OCC(=O)NC2CN(C(=O)CCc3cncs3)C2)CCCCCC1 61860,c1(C(=O)OCC)sc2ccncc2c1NC(CSc1ccc(C(=O)OC)o1)=O 61861,Cc1ccc(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)nc1 61862,N1(C(c2cccc(C(C)(C)C)c2)c2n(C)nnn2)CCC2C(CCC2(F)F)C1 61863,C1(NC(CC)=O)(CNC(=O)CNc2nc(C)cs2)CCCCC1C 61864,c1(NC(C(C2CCCO2)NC(CC(C=C)C)=O)=O)cccc([N+](=O)[O-])c1 61865,C1(C(=O)OC)CCCC1N(C(=O)C=CCN(C)C)C.C1CO1 61866,OCC(F)(F)CCCCN=C(NCc1ccon1)NC1CCC1 61867,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CO)c1C)=O 61868,C1(C(=O)NCCCOCCCNC(C(C)=CC2CC2)=O)CC(C2CC2)C1 61869,Cc1cc(NC(C2CCN2C(=O)CCc2cncn2C)=O)c(O)c(C)c1 61870,C=CC(CCC)CC(=O)NC1CC2(C1)CN(C(c1cc3n(n1)CC(F)C3)=O)C2 61871,Cc1nc(N(C)C)sc1C(=O)NC(C)C(C)NC(=O)CCF 61872,CCCCN=C(NCc1cccc(F)c1F)NCc1nc(C2CC2)n[nH]1 61873,C1(CNC(Cc2nc(CC)sc2)=O)CC2CCC1N2C(=O)C(C)(CC)CO 61874,C1(C(=O)NC2CC(CNC(C(C)NC(=O)C3CC3)=O)C2)CCNC(=O)C1 61875,CCCC(C(=O)OC)C(=O)N1CC(C2(NC(=O)CC3CCS(=O)(=O)C3)CC2)C1 61876,c1(N(CCC2CCS(=O)(=O)C2)CC)nnc(-c2cccnc2)n1CC(C)C 61877,Cc1nc(C=CC(=O)NCC2(C)CC(NC(C3CCC3)=O)C2)[nH]c1C 61878,c1(CC)cc2c(NCCN(C)C(C3SC4C=CC3CC4)=O)nc(C)nc2s1 61879,C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2ccc(F)cc2C#N)=O)CC1C 61880,N1(C(CC(C)(C)CNC(=O)C=CCN2CCCC2)=O)CCC(C2(O)CC2)CC1 61881,N1(C(c2c(-n3cc(C(C(C)C)O)nn3)cc(F)cc2)=O)CC(C)(C)C(O)C1(C)C 61882,C1(C)(C(=O)NCCCCNC(C(CCC)=CCC)=O)CCCCC1(F)F 61883,c1(C(=O)NC2C(OC)C2)cc(C)c(C#N)cn1.N12CCCC1C2=O 61884,N1(C(CCC)=O)CCC(CN(C(=O)C(C2CCOCC2)OC)CC)C1 61885,C1(NC(C2CCCN2C2CC2)=O)CCC2CCN(C(c3cnc(O)s3)=O)C1C2 61886,CCC(CC)C(F)C(=O)N1CCN(C(c2ncsc2Br)=O)C(CCO)C1 61887,N1(C(c2cnc(C)[nH]2)=O)CC2CN(C(=O)C=CCF)CCC2(CO)C1 61888,C(C1CCC(c2nnnn2CC(F)F)(Nc2cccc(OCF)c2)C1)=C(C)C 61889,C(c1ccc(OC)c(Cl)c1)=CC(=O)NCCOCCCNC(C=C(CC)C)=O 61890,c1(C(N2C(C(=O)Nc3c(Br)ncc(OC)c3)CC(F)C2)=O)ccc(C#N)cc1O 61891,C(=O)(N=c1cccn[nH]1)N1CC(C)C(NCc2ccc(F)cc2)CC1 61892,c1(NC(=O)NCCOc2ncccc2Cl)ccc2c(c1)CCOC2 61893,C12CN(CCC1(F)F)C2.c1(C(=O)NCCOCCOC)ccn(C)c1C 61894,N1(NCc2cc(CC)c(C)o2)C(=O)NC2CN(C(C)=O)CCC12 61895,N1(C(C(C2CCOC2)OC)=O)CC2CCC1C(NC(=O)CN1CCC(C)CC1)C2 61896,N1(C(CSCCCC)=O)CCCC1C(Cc1cn(C)nn1)(C)C.n1(C)cccn1 61897,S(=O)(=O)(c1ccc2occc2c1)NC(CCC(=O)OCC)C 61898,N1(C(C(C)=CC)=O)CCC2(NC(c3sc(N4CCCCC4)nc3Cl)=O)CC2C1 61899,CC1CCCN(S(=O)(=O)NCCOCC=CCF)C1 61900,c1(C(=O)OCC)cc(Br)ccc1NC(C1CN(Cc2cc(C)[nH]n2)CCC1O)=O 61901,c1(C(N2C(C(N(C(c3c(CC)nc[nH]3)=O)C)C)CCC2)=O)cnc(COC)nc1 61902,C1(CNC(C(CC)N(C)C)=O)CC2CCC1N(C(c1cn3cc(C)nc3s1)=O)C2 61903,c1(C(=O)NC2CC(NC(c3c(C)nc(CCC)s3)=O)C2)csc2ncnc(O)c12 61904,C(CC(C(=O)N1CC(C)(C(=O)NC(N)=O)C1)NC(C1C(OCC)CCC1)=O)OC 61905,c1(NC)cncc(C(=O)NC(C)CCCCNC(=O)CC2CCCO2)c1 61906,C(=O)(CCCCC(F)(F)F)N1C(C)CC(CNC(=O)CC23CCCN2CCC3)C1 61907,CCCC(C(O)C(=O)Nc1ccc(O)c(OC)c1)NC(C1CCCN1C(C)=O)=O 61908,n1(CC)c(C)nn(CC(=O)NCCCNC(c2ccc(C(N)=O)cc2)=O)c1=O 61909,C(=O)(C(F)(F)C(F)F)NCC1CN(C(c2c(C(C)C)nns2)=O)C(C)C1 61910,CCC(CN1CCCCC1CCOC)(CC)C(=O)NCC1CC1 61911,N#Cc1c(C2(c3ccc(C4CC4)cc3)CCO2)cccc1Cl.C12CCCCC1NC(=O)NC2 61912,C1(O)(C(N2CC(O)(C(C)NC(=O)COC(F)F)C2)=O)CCSCC1 61913,C1(CC)CCCC(N=c2nc(NC3CCSc4ccccc43)c3ccccc3[nH]2)C1 61914,CC(C)CC(CC(=O)NC1(CO)CCC(C)C1)NC(C1(C2CCCO2)CC1)=O 61915,c1(C(C)(C)C(=O)NCC2(O)CN(C(=O)Cc3cccs3)C2)ccc2c(c1)OCO2 61916,CC1CCC(NCC2CCN(C(=O)C(O)C(C)C)C2)CC1 61917,c1(OC)ccc(C(=O)NC2CC2NC(C2CCN(C)C2C)=O)c(N)c1F 61918,C1(SCC)C(C2CC2)CCN1C(=O)CC1CCC2CC12.CC1CC(C(=O)N)CCC1C 61919,c1(C(N2CC(COC)(NC(c3nccn3C)=O)C2)=O)cc(Cl)cn1C(C)C 61920,N1(C(=O)CCOC2CC2)CCCN(C(C2(C(F)(F)F)CC3CC3C2)=O)CC1 61921,c1(CNC(C(c2ncccc2C)N(CCCO)CCC)=O)ccc(C)cc1 61922,N1(C(C=CCOC)=O)CCC2(NC(c3cc(CO)on3)=O)CC2C1 61923,c1(NC(C2C3CCN(C(C4C(CC)C4)=O)C3C2)=O)nc2ccc([N+](=O)[O-])cc2[nH]1 61924,N1(C(CCCCCC#C)=O)CC2CS(=O)(=O)CC2(NC(c2ncn(C)n2)=O)C1 61925,C1(C(=O)OC)C(C)CCCN1C1CCN(c2ccccc2F)CC1 61926,c1(C(N2CC(CNC(C3(C)C=CCC3)=O)OCCC2)=O)ccc2nc(Cl)nn2c1 61927,CC(C)S(=O)(=O)C(C)C(=O)NC1(CNC(c2cc3c(nc2O)CCC3)=O)CC1 61928,c1(C(=O)NC(CNC(C(COC)COC)=O)CCOC)cc2oc(Cl)cc2[nH]1 61929,C1(C)(N)CC(N)C1.C1(C(C(=O)C(CNC(C2C(C)C2)=O)=O)O)CCOCC1 61930,c1(C(=O)NCC(CC=C)NC(c2cnc(Br)s2)=O)cc(F)ccc1NC 61931,C1(C(=O)NCC(C)N(C)C)CN(C(c2ccc(N3CC=CC3)cc2)=O)C2(CCC2)C1 61932,c1(NC(C(CC)=O)=O)cnc(Br)c(Cl)n1.c12csc(n1)NC2=O 61933,C1(C(=O)OC(c2nc(COC)cs2)C)C(C)(C)CN(C(=O)OC(C)(C)C)CC1(C)C 61934,c1(C2(NC(N(CC(F)(F)F)CCC)=O)CC2)ccc(Cl)cc1 61935,C1(C2CCC2)(C(=O)NC23CC(NC(C4(CC)CCOCC4)=O)(C2)C3)CC1(F)F 61936,n1(CC(=O)NC2(CCSCC(=O)NCc3cn[nH]c3)CCC2)ncccc1=O 61937,c1(C(=O)NCC(CC)(C)NC(=O)Cc2c[nH]nc2C)cc2c(cc1O)OCO2 61938,c1(C(=O)NCCCCNC(C(C)c2ccco2)=O)ncccc1N 61939,c1(-c2cn(C(C)C(=O)N3CCCC3c3ccccc3I)nn2)cc(F)c(F)c(F)c1 61940,Cc1cn2cc(C(=O)NCCC3(O)CN(C(=O)CCc4nc[nH]n4)C3)nc2s1 61941,c1(CC(=O)NCC2(OC)CN(C(C=NOC)=O)C2)sc(C)cc1C 61942,C(c1nc2ccccc2o1)=CC(N1CCC(C)C1CNC(=O)Cc1sccc1Cl)=O 61943,C1(COC)CN(C(=O)CCCC(=O)OC)CCN1C(C1CC(=O)N(C(C)C)C1)=O 61944,c1(C(N(C)Cc2cn(-c3ccc(C(=O)O)cc3)nn2)=O)ccnc(N(C)C)c1 61945,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 61946,N(C1CS(=O)(=O)N(C)c2ccccc21)C(N(c1ccc(F)cc1)CC(C)C)=O 61947,Cc1[nH]nc(Cl)c1C(N1CCC(C)(CNC(=O)CCc2cscn2)C1)=O 61948,CC1(C)CC(C)(C(=O)NCC2(O)CCOC2)CN1C(c1cncc(O)c1)=O 61949,N1(C(CN(C)C(C2(c3ccnn3C)CC2)=O)=O)CC(NC(N)=O)C2CC12 61950,Cc1c(Cl)c(C(N2CC3CC(NC(=O)OC(C)(C)C)C2C3)=O)nn1C 61951,c1(C(=O)NC(C)CNC(=O)C(C)n2cncn2)cccc2c1OCCN2C 61952,c1(C(=O)NC2(CF)CC2)ccc2nc(CCCNC(c3cc(Cl)cs3)=O)[nH]c2c1 61953,C1(CC)CCC(C)CC1C(=O)OCC1CCC(C)(C)CC1 61954,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 61955,C(C1c2ccccc2CN1C(=O)CCOCC(F)F)NC(C1CCOCC1)=O 61956,N1(C(C(C)c2ccsc2)=O)CC(NC(=O)CCc2cn(C)nn2)C(F)C1 61957,N1(C(C2C(CC)CN(C(=O)C(C)n3cnnn3)C2)=O)CCc2nc[nH]c2C1 61958,c1(SC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(C(C)C)C2)=O)c(O)n1 61959,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 61960,C1(NC(CSCC)=O)CC2CCC1N2C(c1cc(-c2cccc(Cl)c2)on1)=O 61961,CC(C)C(O)C(=O)N1CC(NC(=O)C=CC2CC2)C(c2ccnn2C)C1 61962,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 61963,C(=O)(C(C)(C)CCCF)NCCC1CC(NC(C(c2n(C)ncc2)O)=O)C1 61964,C1(C(=O)NCC)CCN(C(=O)NC(C)COC)C1 61965,c1(C(=O)NCC2CN(C(c3conc3C3CC3)=O)CCO2)cn2c(n1)SCC2 61966,C1(NC(CCOCCOCC)=O)CN(C(c2c[nH]cc2C)=O)Cc2nccn2C1 61967,CC1(CC(c2csc(C(F)F)n2)NC(c2ccccc2)=O)CCC(=O)NC1 61968,c1(C(N2CC3C(CNC(c4cnc(C(C)C)[nH]4)=O)(C3)C2)=O)ccc(CO)c(Cl)c1 61969,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)c1F 61970,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 61971,CCCCS(=O)(=O)CC(=O)N1CCC(O)(CN(C(=O)C(F)C2CCOC2)C)C1 61972,CC1(C(=O)NCc2ccc(C(F)(F)F)nc2)CCN(S(=O)(=O)CCCl)C1 61973,C(=O)(C(C)CCC(C)(C)C)N(C(C(CC)C)C(=O)N1CCN(C)CC1C)C 61974,N1(C(C2CCCN(CC)C2)=O)CC(CNC(C2CC(O)C2)=O)C(C)(C)C1 61975,c1(C(N(C(N(CCOC2CC2Cn2ccccc2=O)CC)=O)C)C)ccccc1Br 61976,CN=c1nc(N2CCCC(S(N)(=O)=O)C2)[nH]c(=NCC2CCC3(CC3)CO2)[nH]1 61977,c1(OC)cc(C2CC2)ccc1C(=O)NC1(C)CC(NC(=O)C(c2cncnc2)C)C1 61978,Cc1nn(C(C)C)cc1C(=O)NC1(CNC(C2(CO)CC(C)(C)C2)=O)CCC1 61979,C1(CNC(C)(C)C)CC12CN(C(=O)OC)C2.CC(C)C(Cc1ccccc1)NC=O 61980,Cc1nc(=NC(=O)CC2CN(C(=O)OC(C)(C)C)CCO2)s[nH]1.C 61981,Cn1ccnc1C(F)(F)C(=O)NCC1CC(NC(=O)C(C)(C)C2(O)CCOC2)C1 61982,c1(C(N(CCC)CCNC(C23CSCC2C3)=O)=O)cc(C(F)F)n(C)n1 61983,C1(C(N(C)CCn2cccn2)=O)COCC1NC(=O)Cn1cnnc1 61984,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3cscc3-n3cnnn3)=O)C2)C1 61985,C1(NC(N2CCCC2)=O)CCC2(CCCCN2C(=O)CC2CCCCO2)CC1 61986,C1(C(=O)NC2CCCC2CCO)CSCN1CC(c1ccccc1)(C)C 61987,c1(C(=O)NC2CC(CCNC(CN(C3CC3)CC)=O)C2)ccc2c(c1)ncn2C 61988,C1(CC(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCO2)CNC(=O)O1 61989,C1(C(=O)Nc2nc(-c3c(COC)cccc3)sc2)CCC(C)CC1C 61990,CCC(C)(C)CCCC(=O)N(CCCC(=O)NCC1CCCC(C)CC1)C 61991,CN(C)NC(=O)CCC(=O)NC1(C)CCCCC1C(=O)NCC(F)(F)CO 61992,Cc1cnc(CC(=O)N(CCNC(=O)C(F)(Cl)c2ccccc2)CC2CC2)s1 61993,Cc1cc(C(N2CCC(NC(=O)Cc3ccco3)C23CC3)=O)cc([N+](=O)[O-])c1Cl 61994,N1(C(c2cccc(C3(C(=O)OC)CC3)c2)=O)CC2CCN(C)C2C1 61995,CC1CCC(C)(CNC(C2(CO)CN(C(=O)CCCn3ccccc3=O)C2)=O)C1 61996,C(CCCCCNS(=O)(=O)Cc1ccncc1C(F)C(F)(F)F)N(C)C 61997,Cc1ccc(C(N2CCCCCC2CNC(=O)COCC(F)(F)F)=O)cc1N 61998,C1(NC(C2C(C)(C)C2(C)C)=O)CCC2CCN(C(c3cc(C(F)F)ns3)=O)C1C2 61999,O=NN1CCCCC1C(=O)NCCCCCCNC(C1CCCCN1N=O)=O 62000,N1(C(C(c2ccc(F)cc2)NC(C(C)CC#N)=O)=O)CCC12CCCOCC2 62001,C1(CC=C)(C(=O)NC2CCC2NC(=O)CN(C(=O)CCC)CC)CC=CC1 62002,N1(C(CSc2nc(C)[nH]n2)=O)CC2CC1CN2C(C1CCN(CC2CC2)CC1)=O 62003,C1(CNC(CCc2c(C)noc2Cl)=O)CC(C)CN(C(=O)C(C)(C)CN(C)C)C1 62004,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(c2cc(Cl)ns2)=O)CC(O)C1)=O 62005,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(C3CCCCO3)=O)CC2C1 62006,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1CCOC1 62007,Cc1nc(Br)sc1CNCCC1CCN(C(C2CCOC2)=O)CC1 62008,C1(O)(CN(C(=O)C(O)Cc2ccccc2)C)CCN(C(=O)Cn2cccc2)C1 62009,N1(C(C2C(C)(NC(CCc3cn(C)nn3)=O)CCCC2)=O)CCOC2(CCCC2)C1 62010,S(=O)(=O)(c1cccc(Cl)c1)N1C(C(=O)Nc2c(C)nc(I)cc2)CCC1 62011,C1(C(=O)NC(C(C)(C)C)CNC(=O)C=CSc2ccccc2)CCC2CC1CO2 62012,Cc1nsc2ncc(C(N3CC(CCCCNC(c4ccoc4)=O)C3)=O)cc12 62013,N1(C(=O)C2=NOCC2)CCC2(CCOC2)C(CNC(C2(Cl)CC2)=O)C1 62014,C1(CCC)CCCN(C(C2(F)CN(C(=O)CC3OCCCO3)C2)=O)C1 62015,C1(C(N(CCOCCCNC(c2c(C)coc2)=O)C)=O)CC2COCC2C1 62016,C1(N(C(=O)CNC2CC(CC(C(=O)C(F)C3CCOC3)=O)C2)CC)CCCCC1 62017,C1(C(=O)OC)CC(F)(F)CN1C(C1CCCN1C(c1cnnc(Cl)c1)=O)=O 62018,c1(C(N(CC(CC)NC(c2ccnnc2)=O)C)=O)ccc(C2CC2)o1 62019,C(=O)(C1=COCCC1)NCC(C(C)C)NC(C1(O)CCSC1)=O 62020,N12CC3CC1CN3C(=O)c1c(nccc1)NC2=O.C(CCCl)OCC1CC1 62021,c1(CC(=O)NCc2ncccc2Br)cc(=O)oc2cc(O)ccc12 62022,C1(CC=C)(C(N2CC(OCCNC(C3CC3(C)C)=O)C2)=O)CCOC1 62023,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(N3CCCC3)cc2)=O)CC1 62024,C1(C(=O)NCCCC2C=CS(=O)(=O)C2)NCCOC12CCC2 62025,c1(C(=O)NCC(C)N(C(=O)C=C2CCC2)C)ncn2cccnc12 62026,CC1(CS(C)(=O)=O)CN(C(=O)CN2CCCC2)C1.c12ccoc1CNC2=O 62027,c1(OC)c(C(=O)NCC(C)(C2CC2)NC(c2ccc(CO)s2)=O)csc1C 62028,C1(C(=O)NCC(C)(C2CCCC2)NC(c2scc(COC)c2)=O)CC2(CC2)CO1 62029,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCC2(CNC(=O)C=CC2(C)COC2)C1 62030,Cn1nc(C(=O)NC2(CF)CCN(C(C34CC(C)(C3)OC4C)=O)C2)cc1C#N 62031,C1(C(N(CC)CC)=O)CCN(C(=O)Cc2cncnc2O)C12CC2 62032,C1(CC(=O)OC)COCCN1C(c1cocn1)C(=O)NCc1cccc(Cl)c1 62033,c1(C(N(CCC(C)NC(=O)CC2CC3(CCC3)C2)C)=O)[nH]nc2ncnc(O)c12 62034,N1(C(c2cnc(C)s2)=O)CCN(C(C2CC(C)(C)C2C(F)(F)F)=O)C(CCO)C1 62035,c1(CCOC(C(COC)Oc2ccccc2)=O)cccc2nonc12 62036,C(=O)(C1CCCc2nn[nH]c21)N1CC(O)(CCNC(c2nc(C)nc(O)c2)=O)C1 62037,N1(CC)CCN(C(=O)Cc2ccc(CC(C)C)cc2)CC1=O 62038,C1(CC(=O)NC2(CN(C)C(C3(C)C=CCCC3)=O)CC2)CCCC(=O)C1 62039,N1(C(C2(COCC)CC2)=O)CC2(C1)CNCC(C)(C)O2.C1(COC)CCCS1(=O)=O 62040,CCCC(O)CC(=O)N1CCN(C(C2(C(F)(F)F)CC3CC3C2)=O)CC1 62041,CC(C(F)F)=CC(=O)NCC(C)N(C)C(C1(CCF)CC1)=O 62042,C1(C(=O)NC(C)CC2CC2)CN(C(=O)C(F)C(C)(C)O)CCN1C 62043,C1(C)(C(N2CC(CCCC)N(C(c3n[nH]cc3F)=O)CC2)=O)CCCNS1(=O)=O 62044,c1(CC(=O)NC2CC3(C2)CN(C(=O)C=C(Cl)Cl)C3)cc(F)cc([N+](=O)[O-])c1 62045,C1(C(N(C)CCn2cc(CCC(N)=O)nn2)=O)Cc2ccccc2C(=O)O1 62046,c1(C(=O)NCCN(C(CC2(C)OCCO2)=O)C2CC2)ccc(Br)cc1F 62047,c1(OCOC)cccc(C(=O)N(C(CNC(=O)CNC(C)=O)C2CC2)C)c1 62048,c1(C(=O)NCC(CO)NC(c2ccc3c(c2)CC3)=O)cc2n(n1)CCC2 62049,N1(C(=O)C=C(Cl)Cl)CCCC2(CCN(C(C3(C(F)(F)F)CCC3)=O)C2)C1 62050,Cc1cc(Cl)c(C(N2CC(NC(=O)CC3CCCN3C(C)C)CC2C)=O)cc1C 62051,C(c1ccccc1)=CCC1CCN(C(=O)C(O)C2CCC2)C1.O=C1CN(C2CC2)C(=O)N1 62052,C1(C(=O)NCC(CN(C(C=C(C)Cl)=O)C)C)(C(F)F)CCN(C)CC1 62053,N1(C(C2(OC)CCCCCC2)=O)CCCN(C(=O)CS(=O)(=O)C(C)C)CCC1 62054,C1(NC(C(N2CC(C)C2)C)=O)CCCC1CNC(C1(c2cccnc2)CCC1)=O 62055,CC1CCCC(NCc2cn(C3CN(C(C45CC6CC4C5C6)=O)CC3O)nn2)C1 62056,Cc1cc(C(=O)NC(C)(CO)C(=O)NCCN(CC(F)F)C)ncc1N 62057,c1(C(=O)NCC(=O)N(CC)CC)cc2cc(-c3cc(C)cs3)cnc2[nH]1 62058,c1(C(=O)NC(C)CN(C(=O)C(C)(C)N(C)C)C)nn(C)c(Cl)c1Br 62059,c1(CC)cnc(NC(c2ccc(C(N3CCC(N4CCC4)C3)=O)[nH]2)=O)nc1 62060,CC1(C)C(CNC(c2cccc(NC3CC3)c2)=O)CCN1C(N)=O 62061,CC1C(NC(c2cccc(Cl)c2)=O)CC2CCC1N2C(=O)CCCN(C)C(C)C 62062,CC1(c2cn(Cc3ccccc3F)nn2)CCCN1C(=O)C#CC(=O)N1CCCC1 62063,C1(n2nc(C)c(I)c2)CC2CCCC2N1CC(F)F 62064,C1(C(=O)NCCN(C2CCCC2)C(Cn2c(C)nnn2)=O)CCOCC1(C)C 62065,c1(CCC)ccc(C(N2CCC(NC(=O)CCCNC(N)=O)C2)=O)cc1[N+](=O)[O-] 62066,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62067,C(=O)(C(O)C(CCC)NC(c1cn(C(C)C)nn1)=O)NCCCCCC 62068,c1(OC)ccc2[nH]c(C(N3CCSC(C(=O)NCC(C)O)C3)=O)cc2c1 62069,N1(c2cc(NCC3COC(=O)N3)nc(C)n2)CC2CC(C1)N(C)C2 62070,C1(CNC(=O)C(=O)Nc2ncc[nH]2)(CC2CCCC2)CC1(F)F.C1CC(=O)N1 62071,N1(C(CCC)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62072,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)C=CCN2CCCC2)CC1(C)C 62073,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCN(C(Cc2ncc(C)s2)=O)CC(O)C1 62074,O=C(CCCC(=O)N1CCN(C(C2CCC(=O)CC2)=O)CC1)c1ccc(Cl)cc1 62075,c1(C(N(C2C(C)CN(C(=O)C(F)F)CC2)C)=O)nc2ccc(Br)cn2n1 62076,C1(C(=O)NCC(C)(F)CNC(=O)C(C2CCCCCC2)O)CCc2nncn2C1 62077,c1(CNC(=NCC)NCC2COC(C)(C)C2)nn(C)c2cccnc12 62078,CCCCC1C(=O)N2CCC(F)(C2)C(=O)N1.C(C(C)(C)C(=O)NC)OC 62079,C(=O)(CCCNC(c1cnn(C2COCC2N)c1)=O)OC 62080,N1(C(C(CSC)NC(C2CC=CC2)=O)=O)CC2C3C=CC(O3)C2C1 62081,NC1CC(O)CN(C(=O)Nc2cncc(-c3cncc(-c4ccccc4)n3)c2)C1 62082,C(=O)(C(C1=CCCCC1)N1CCC(C2CC(F)(F)C2)C1)N1CCCC(C)(C)C1 62083,N1(C(c2cccnc2)=O)CCCCC1c1cn(CCOC2CCCC=C2Br)nn1 62084,Cc1cccc(C)c1NC(=O)COCC(=O)NCC(=O)N(C)Cc1ccoc1 62085,C1(C(N(CCN(C(C)C)C(C2C=CCC2)=O)C)=O)(Cc2ccccc2)CCCO1 62086,c1(C(=O)NC2CC(CNC(C3CCC4CC34)=O)C2)ccc(=NCC2CC2)[nH]c1 62087,Cc1cc(N)c(C)nc1C(N1CC(CNC(=O)CSc2nc[nH]n2)C2(CC2)C1)=O 62088,N1(C(CN(CCC)C)=O)CCC(C)(C)C(CNC(=O)C(c2cn(C)nc2C)C)C1 62089,c1(COC)cccc2oc(-c3nc(-c4occc4C)no3)nc12.c12ccc-1cc2 62090,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62091,C1(OCC)CCC(C(c2ccccc2)NC(c2cc(-c3ccccc3)no2)=O)CC1 62092,c1(C(=O)NCCSC)csc(=NCc2cc(F)ccc2Br)[nH]1 62093,c1(C(N(CCOCCN(C(C(F)OC)=O)C)C)=O)cc(-c2ccc(C)s2)[nH]n1 62094,c1(C(N2CC(NC(CC(CC)OC)=O)C(SC)C2)=O)cc(C)c(N)cc1Cl 62095,c1(OC)cccc(CNC(=O)NC(CO)C(C)CO)c1OC 62096,c1(N2CC3CCN(C)C3C2)nc(N2CCn3ccnc3C2)nc2c1SCC2 62097,C(CCCCCC(=O)N1CC(CNC(C2OCCC2C)=O)CC1C)NC(C)=O 62098,c1(C(=O)NC(CNC(c2c(OCC)cccn2)=O)C(C)C)c(C)nc2sccn12 62099,C(=O)(C(CC(C)C)c1ccccc1)N1C(CNC(CCC=C)=O)CC(O)C1 62100,C(CC(C)C)(C(=O)OC(C)=O)ONC(CC1(NC(C2N(CC)CCCC2)=O)CC1)=O 62101,C12CCCN(C1)C(=O)C2(C)C.C(c1cnccn1)=CC(N1C(C=C)CC1)=O 62102,N1(C(=O)N(C2CC(F)(F)C2)Cc2cnc(C(C)C)s2)CC2COCC2(CO)C1 62103,C1(CN(C(c2cn(CCCC)nn2)=O)C)CCCCN1C(c1c[nH]ccc1=O)=O 62104,C1(C(=O)NC(CC=C)CNC(c2cnn(CC(F)F)n2)=O)CCC(N=[N+]=[N-])CC1 62105,C1(C(=O)NCCN(CCC)C(C)C)CC(F)(F)CN1C(=O)CC1CC2(CC2)CO1 62106,c1(C(=O)NCC23C(CN(C(CC4(OC)CC4)=O)C2)C3)ccc2nccn2n1 62107,CC(C)(C)C(O)C(=O)N1CC(CCNC(=O)C(N)=O)C1 62108,CCCCC(F)C(=O)N1CCC(CO)(NC(=O)COC(C)(C)C(F)(F)F)C1 62109,C1(C(N(C(C(=O)OCC#C)C)C2CC2)=O)CC2(O)C1(C)C2(C)C 62110,c1(C(=O)NCC(CO)NC(C(c2scc(C)n2)C)=O)cc(C)nc2ccccc12 62111,N1(C(C2N(C(C(CCSC)NC)=O)CC(C)C2)=O)CCOC(C#N)C1 62112,c1(C(c2n(CC(=C)C)nnn2)NCCC2CC2C)cn(C)nc1OC 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62201,c1(SC)cccc(CC(=O)NCCCC(C)NC(=O)CS)c1.c1(S)ncc[nH]1 62202,C1(CCC(=O)NC(c2nncs2)C)CCCCN1C(=O)C=CC1CC1 62203,C(C(F)C(=O)NCc1cc(C(C)C)no1)C1CN(C(CSCC)=O)C1 62204,c1(C(=O)NCC(CNC(C2(CC)CCNC2=O)=O)(C)F)n[nH]c2c1COCC2 62205,N1(C(C(CC=CC)C)=O)CC(NC(c2cnc(C)n2C)=O)C2(CCC2)C1 62206,C1(CC)CC(O)CN1C(c1cc[nH]n1)=O.c12scc(-c3ccccc3)c1C(=O)N2 62207,Cc1ccccc1OCCCC(=O)NCC1(F)CC(NC(C2(F)CC2)=O)C1 62208,Cc1c(NC(=O)C(C2CCCC(O)C2)(C)C)cc(CN)n1CCO 62209,c1(OC)cc(C)ccc1CCCC(=O)NC12CCCC(NC(=O)CCF)(C1)C2 62210,Cc1ccc([N+](=O)[O-])c(C(=O)N(CCCCN(CC(C)CO)C)C)c1 62211,C1(CCC(=O)N(C)CNCC(=O)NC2CCC2NC(=O)NC)CCCOC1 62212,c1(C(C)C)ccc(C(=O)NCC2(O)CC(NC(C3NC(=O)OC3C)=O)C2)nc1 62213,N1(C(C(c2cn(C)nc2)=O)=O)CCN(C)C(CNC(=O)Cn2cccn2)C1 62214,C1(C(=O)NC(CCN(C(C(=C(C)C2CC2)F)=O)C)C)CCCCC1O 62215,C1(C(N2CCC(CN(C(Cc3c(SC)cccc3)=O)C)C2)=O)CN(C)CC12CC2 62216,c1(C(=O)NCC(C(C)C)NC(c2nc(C(=O)OC)sc2)=O)ccc2cnnn2c1 62217,N1(C(C)C)CCC(NC(C2CCCN(C(=O)CCn3ccnc3)C2)=O)C1=O 62218,C1(CCNC(=O)NCC(O)CF)CCCCC12CC2 62219,c1(OC)cc(OC)nc(C(N2C3CCC2C(CNC(=O)CS(N)(=O)=O)C3)=O)n1 62220,c1(C(=O)NC(C(C)NC(CSc2ccc(OC)cc2)=O)C)cccc2nncn12 62221,c1(C(=O)NCC(CCOC)NC(c2[nH]c(O)nc2C)=O)cc2occc2[nH]1 62222,C1(C(N2C(CCC)(CO)CCC2)=O)CCC(C)(C)N(C(C2CC(=O)CCO2)=O)C1 62223,C1(NC(c2c(N)nccn2)=O)CC12CCN(C(c1ncccc1Cl)=O)C2 62224,CCC(CC(F)F)C(=O)N(CCCOCCN(C)C(c1cc(C)cc(C)n1)=O)C 62225,CCCC(C)C(=O)NCCN(C)CC.N1(C(C)=O)CC(OC(=N)O)C1 62226,C1(OCC(=O)NCC2(F)CCN(C(C(C)C3CC3)=O)C2)CCC(F)(F)CC1 62227,c1(CC)cc(C)c(C(N2CCC(C(C)C(N3CC(C)(N(C)C)C3)=O)C2)=O)o1 62228,Cn1nc(Br)cc1C(c1nnnn1C1COC1)NCCCOC1CCOC1 62229,c1(C(CC(=O)N(CC)CC)NC(=O)Cc2nccn2C)ccc(C#N)cc1 62230,CC1CN(C(c2cnn(CCO)c2)C(=O)NCCC#N)CC2(CCC2)O1 62231,c1(C(N2C(CNC(C3(C)C(C)(C)C3)=O)CC(F)C2)=O)ccc(O)c(Cl)c1 62232,C(N=c1nc(N2CCC(CC3CC3)C2)c2c([nH]1)CCS2)C1CN(CC(F)F)C1 62233,C1(C(C)CO)CCN(C(C2(C(C)C)CCCN2C(=O)CC2CCC(=O)N2)=O)CC1 62234,C(=O)(CCC(CC)OC)N(CC(C)NC(c1c(CCC)cccc1)=O)C 62235,C1(O)(CNC(C2CC(C)C2)=O)CCN(C(=O)C(F)CC2CC2)CC1.Cn1nnnc1 62236,c1(C(N2CC(O)(CN(C)C(c3cn(C4COCC4O)nn3)=O)C2)=O)snc(Cl)c1Cl 62237,C1(NC(C(C(C)C)OC)=O)CCN(C(=O)CCc2cnoc2)CC1(C)C 62238,C1(OC)CC(CNC(C2(C(F)F)CC(O)C2)=O)N(C(c2cc[nH]c2)=O)C1 62239,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(NC)nc2)=O)ccc(C)cc1SC 62240,N1(C(C2=C(C)CCC2)=O)CCC2CC2(C(N(C)C[Si](C)(C)C)=O)CC1 62241,C=C1CC2CCC(C1)N2C(C1CCC(CNC(C2CCCCO2)=O)C1)=O 62242,N1(C(c2c(C)snn2)=O)CCC(C2CCN(CC(C)(C)C)CC2)C1.C1C(=O)O1 62243,C1(C(C)C)CCC(NC(=O)C(=O)NCc2cccc(Cl)c2)C(=O)N1 62244,n1(CC)c(CNC(c2c(C(=O)NC3(F)CC3C(=O)OC)cnn2C)=O)cnc1C 62245,C=CCS(=O)(=O)CCN=c1nc(N2CC(CO)C3(CCC3)C2)c2[nH]ccc2[nH]1 62246,CC(CC(N)=O)C(=O)NCC(=C1CN(C(C2CC2C(F)(F)F)=O)C1)F 62247,C1(CC)C(C)OCCN1C(=O)CCC(C)(C)NC(=O)C(C1(C)CC1)N(C)C 62248,C1(CCC)CN(C(C2CCSC2C)=O)CC1NC(=O)C(N1CCCCC1)C 62249,CC(C)(C)C(C(=O)NCP(C)(C)=O)N(c1ccccc1)CN1C(=O)CCC1=O 62250,c1(C(=O)NC2CCN(C(c3nc(CC)oc3C)=O)C2C)cnn2c1C(=O)NCC2 62251,N1(C(c2scc(CNC(C(NOC)=O)=O)c2)=O)CC(C)(C2CCC2)C1 62252,c1(CCC(=O)N(CC(C)C)CC(=O)NCC2CCC2(F)F)ncccn1 62253,C1(C(N2CCC(NC(C3COCCO3)=O)C2)=O)COc2ccc(F)cc2C1 62254,c1(CCNC(=O)NCCCCCl)cc(O)nc(O)n1 62255,c1(C(N2CCC(N(C)C(c3ccc[nH]3)=O)C2)=O)cnc(C2CC2)nc1O 62256,c1(C(=O)NCCOC2CCN(C(c3c(C)nn[nH]3)=O)C2)cnc(O)n(C)c1=O 62257,C1(CC(N2CCC(C)(CNC(C3C(=C)C3)=O)CC2)=O)CCC2(CCC2)CO1 62258,Cc1cc(C(N2CC(C)(C(=O)Nc3ncc(C)cc3I)C2)=O)cc(C(F)(F)F)c1 62259,Cc1nc[nH]c1CNC1(CNC(C2C(Oc3ccncc3)C2)=O)CCOC1.C(=O)(C)N 62260,N1(C(Cc2c(CC)con2)=O)CC(NC(c2ccc(C)s2)=O)CC1C 62261,c1(C(N2C(CCNC(C(C)CC(N)=O)=O)COCC2)=O)ccc2c(c1)CCCC2 62262,CN1CCC(O)(C2(C(=O)NCC(C3CC3)N(C(=O)CS(C)(=O)=O)C)CC2)CC1 62263,Cc1nc(C(=O)Nc2ccc(C(=O)NCC3(c4cc[nH]c4)CC3)nc2)sc1C 62264,CC1CN(C(=O)CCC(C)(C)F)CCC1C(=O)NC(C)C(C)C(F)(F)F 62265,N1(C(C2C(C(N)=O)CC2)=O)CCCC2C(NC(c3cncc(Cl)c3Cl)=O)CC12 62266,C1(N(C(CSCC#C)=O)C)CCCCN(C(=O)CSCCC)C1 62267,C(=O)(C(F)CC1CCOC1)NCC=CC(=O)NC(C)(C)CC1CC1 62268,N1(C(C2CCN(C(C(N3CCN(C)CC3)C)=O)C2)=O)CCOCC1Cl 62269,N1(C(CCN(c2ccccc2)C)=O)CCC12CN(C(C1CCCN1N=O)=O)C2 62270,c1(OC)ccc(C(=O)NC2(CF)CCN(C(=O)C(COC(C)C)OC)C2)cn1 62271,N1(C(C2CCCC(=O)O2)=O)CCOC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC12 62272,C1(NC(C(C)CC(N)=O)=O)COC2(CCN(C(c3occ4c3CCC4)=O)CC2)C1 62273,C1(C(=O)NC(CNC(CCS(=O)(=O)N(C)C)=O)C(C)(C)C)CN2CCN1C(C)C2 62274,c1(C(=O)NC(C)(C)CCNC(C2CCS2(=O)=O)=O)ccc(C(O)CF)cc1 62275,N1(C(CN(C(C(C(=O)OC)OC)=O)CC2CC2)=O)CCN(C2CC2)C(C)C1 62276,S(=O)(=O)(c1cc(Br)cnc1N)N1CCN(C(C)C2CC2)CC1 62277,Cc1cc(F)cnc1C(N1CCCC(CNC(c2cn(C)ccc2=O)=O)CC1)=O 62278,CC1CC(CNC(=O)C(C)(C)c2ccccc2)CN1C(=O)CCOC1COC1 62279,c1(OC)cc(F)c(NC(C2CC(OC)CN2C(=O)CCOC)=O)cc1OC 62280,C(CCCC(=O)N1C(CNC(C2(C)CC2)=O)CC2CC12)OCCC=C 62281,C1(NC(CC)=O)CCCCC12CCCN(C(=O)C(c1ccccc1)OC(C)C)C2 62282,c1(SC)ccc(C)c(C(=O)NCC2=CCN(C(c3c(F)cccc3F)=O)CC2)c1 62283,C#Cc1ccccc1NC(C1CC(O)CN1C(=O)Cc1ccc(Cl)cc1)=O 62284,N12CC3C(C3C1)C2=O.c1(C(C)NC(=O)CC2(N3CCCC3)COC2)cc[nH]c1 62285,O=C1CCc2c(C(N3CCC(CCNC(C4(C5CC5)CC4)=O)C3)=O)cccc2N1 62286,C(=O)(C(CSCC)NC(C1CCOCS1)=O)NCCOCC 62287,Cc1cc(C(=O)NC(C(C)NC(=O)C=CSc2nc[nH]n2)C(C)C)c(O)nc1C 62288,C1(COC)(OC)CCN(C(=O)CC2CCCC(C)C2)C1.c12ccc(cn1)[nH]c2=O 62289,C(=O)(CCCC(F)(F)F)NC(C(C)C)(C)CNC(c1cc2n(c1)CCC2)=O 62290,C(=O)(C(C)(C)CCF)NCC1OCCN(C(COc2ccc(C)cc2)=O)C1 62291,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CC2)ccc(Cl)cn1 62292,c1(OC)ccc(CC(C)C(=O)NC(C)(C)C(C)NC(=O)CSC2CC2)cc1 62293,C(=O)(CCCS(C)(=O)=O)N1C(CNC(CC(c2cccs2)NC(C)=O)=O)CC1 62294,N1(C(c2cc(C)c(F)c(C)c2)=O)CCC2C(CCN2C(=O)C=Cc2ccsc2)C1 62295,C1(NC(CCN(C(c2c(CC)n(C)nc2)=O)C)=O)CC12CCCCCC2 62296,C1(C(=O)NCCCOCCCNC(C(n2ccc(C)n2)C)=O)CCCCCCC1 62297,c1(CC(=O)NCC=CCNC(=O)CC2CCCCC2O)ccc(O)cc1 62298,c1(NC(C2CC(=C)CN2C(=O)CCc2cccs2)=O)ccc(OC)nc1Br 62299,n1(CCC)cc(C(=O)NCCCCCNC(=O)C(C2CCC2)OC)nn1 62300,c1(CC)c(NC(c2ccn(CCOC)n2)=O)ncnc1Cl.C12CCN(C1)C2=O 62301,N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)CCc1nnc(C)n1C 62302,c1(CC)cccc(C(=O)NC2CC(CNC(c3c(C4CC4)cnn3C)=O)C2)c1F 62303,C(=O)(C1=CCC(NC(C2(C)COC(=O)N2)=O)C1)Nc1cc(C)sc1 62304,C=CCC(CNC(=O)CCn1cnnn1)C(=O)NCC1CCCCCCC1 62305,c1(-c2cc(C(=O)Nc3scc(COC)n3)ncc2)cc2ccccc2[nH]1 62306,c1(C(=O)NCC(C2CCCC2)NC(C2C3COCC23)=O)ccnc2ccsc12 62307,N1(C(c2cccc(SCC#N)c2)=O)CC(NC(C2CSC2)=O)C2(CCC2)C1 62308,N1(CC2C(C)CCCC2)C(=O)CN(CCn2cnnn2)C1=O 62309,N1(C(=O)NC2(C#C)CCC2)CCCC(CNC)C1 62310,c1(CN2CCNC2=O)nc(C(F)F)ns1.C(=O)(CN(C(C)(C)C)C)OCCC 62311,N1(C(c2cn(CCC)nn2)=O)CC2CCC(NC(=O)CN(C)CC)(C2)C1 62312,CCC(O)C(F)(F)C(=O)NCC1C2CN(C(C3(CNC(N)=O)CC3)=O)CC12 62313,c1(C(=O)NC2(CNC(c3c(CC)nns3)=O)CCCC2)cc2c(cn1)CCCC2 62314,C1(C(=O)NC(CNC(C2(CC)CCCO2)=O)CC(F)(F)F)CN2CCN1CC2C 62315,N1(C(CC2C(C)=NNC2=O)=O)CC=C(C(=O)N2CCCOCC2C)CC1 62316,N1(C(Cc2ccc(C#C)cc2)=O)CCC2CCCC12CNC(=O)CCN1CCC1 62317,C=CCCCCCCC(=O)N1CCC(CNC(=O)C(F)(F)c2cccnc2)CC1C 62318,C1(C(=O)NC2CCC(NC(CC3(C)CC3F)=O)CC2)CCCCCCC1 62319,C(=O)(CC1NC(=O)c2ccccc21)NCCCC(C)NC(c1c[nH]nc1F)=O 62320,CC1CN(C(c2cccc(N(C)C)n2)=O)CCC1CNC(C1CNC(=O)N1)=O 62321,c1(C(=O)NCC(C)CNC(c2cc(O)cc(F)c2F)=O)csc(S(N)(=O)=O)c1 62322,S(=O)(=O)(c1c[nH]c2ncccc12)NC(CN1C(=O)CCN(CCF)C1=O)C(F)F 62323,C1(CNC(C(C=CC)O)=O)N(C(C2CC3CCC2C3)=O)CCCC1(C)C 62324,N1(C(c2cscc2F)=O)CCCC2(C1)CN(C(C1CC(O)C13CCC3)=O)CCO2 62325,S(=O)(=O)(c1ccc(Cl)c(C(=O)NCC2CCCC(C3CC3)O2)c1Cl)N(C)C 62326,CC1CC(NC(C2(NC(c3ccnnc3O)=O)CCCC2)=O)CCO1 62327,c1(C(=O)OC)cc(=NCC2CCCCC2NC(c2cc(Br)ccc2Cl)=O)[nH]cn1 62328,Cc1ccc(Cl)c(C(N2CCC(CCNC(C3CCCCO3)=O)C2)=O)c1N 62329,C1(C2CCN(C(c3ccc4cncn4c3)=O)C2)(NC(C=CCC)=O)CC1 62330,C1(O)(CCNC(c2cc(C(C)=O)[nH]c2)=O)CCN(C(=O)CN2CCCCC2C)C1 62331,c1(N2C3CC(CO)CC2CC3)[nH]c(=NCCC(O)C2CC2)nc2sccc12 62332,C1(CNC(c2nccc(CC)c2)=O)COC(C)(C)CN1C(C1CC(F)C1)=O 62333,Cc1cc(C(=O)NCC(O)CCNC(=O)C(C)C2CCC2)c2c(n1)CCCC2=O 62334,C1(CCNC(CC=CC=C)=O)CN(C(=O)CCC(F)(F)F)CC(C)O1 62335,C1(CC(N2C(CNC(c3ncccc3Cl)=O)CC2)=O)CC2(CCC2)CCO1 62336,c1(C(N2CC3C(CNC(C(CSC)O)=O)C3C2)=O)cc2n(n1)CCC2 62337,C(=O)(C(F)C(C)C)Nc1nc(CNC(=O)NC)sc1.c1(C)ccc(Br)cc1 62338,c1(C(N(CCCNC(c2cnc(O)n2C)=O)CC)=O)cnn2c1OCCC2 62339,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62340,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62341,C1(C#N)(NC(Cc2c(SC)cccc2)=O)CCN(Cc2ccnn2C)C1 62342,C1(C(=O)OC)(CNC(=O)Nc2ccnn2-c2ccncc2)CCOC1 62343,N12CCCCC1COC(=O)C2=O.C(C(F)F)C(N(C1(CC(F)F)CC1)C)=O 62344,c1(NC(CC2(NC(CCC)=O)CCC2)=O)c(C)nn(C)c1SC 62345,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC(CCNC(c2nnnn2C)=O)CC1 62346,C1(NC(c2cc(C(C)C)no2)=O)CC(F)CN(C(c2ccc(CO)c(Cl)c2)=O)C1 62347,c1(C(N)=O)cn(CCNC(=O)C(O)CNC(c2ccc(Cl)o2)=O)cn1 62348,C(CCN(C)C)(C(=O)NC(C)(C)CCCO)NC(CC(=O)OC)=O 62349,CC(C)C(C(=O)NCCCN(C)C(C1(n2ccnn2)CC1)=O)Sc1nc[nH]n1 62350,N1(S(CC(=O)OCC)(=O)=O)CC2(CCCN2C(=O)C(C)(C)C)C1 62351,C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1c(C)n(C2CC2)cc1)=O 62352,c1(OCC)cnc(C(=O)NCCC2CN(C(=O)C(C)COC)CCO2)cn1 62353,CC1CCCCN1CCNC(=O)N(C)CCN(C)C(=O)C1CC1 62354,N1(C(C(COC)COC)=O)CCN(C(c2cc(Cl)c(C)cn2)=O)CC1C1CCC1 62355,N1(C(C2(CCC=C)CCCC2)=O)CCN(C(=O)C(C)N2CCCC2)C(C)C1 62356,c1(C(N(C2CCCC2)CCNC(C(C)NC(CC)(C)C)=O)=O)sccc1Br 62357,c1(N(C)C)ncc(Cl)c(CNC2(c3ccccc3)CC3(CC3)C2)n1 62358,c1(C(N(CC(=O)N(CC(=O)N(C)C)C)CC)=O)ccc(C#N)n1C 62359,N1(C(=O)NC2CCCOC2)C2CCC(C2)C1CNC1CCN(CC2CC2)C1 62360,CC(C(=O)NN1CCCC1C(=O)N(CCN=[N+]=[N-])CCO)=C1CCC1 62361,Cc1cc(C)n(CC(N2CCC(CC#N)C2)=O)c(=O)n1 62362,CCCC(CCC)(c1nnnn1C1CC1)NCCn1cnccc1=O 62363,CCCCCCC(=O)NC(C1CCCN1C(c1c(Cl)cncc1Cl)=O)C 62364,N1(CCN(C)C)CCC2C1CCCN2C(=O)CCC(=C)Cl 62365,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C2=COCC2)c(C)n1 62366,c1(C(=O)OC)cnc(N(C)CC2CCN(C(=O)C(C)CSC)C2)cc1C 62367,CC(C)C(O)C(=O)NC(C)C(CO)NC(c1cnn(C(F)(F)F)c1)=O 62368,C1(CC(=O)N(CC(C)(C)NC(c2cncc(OC)n2)=O)C)Cc2ccccc2C1 62369,CC(C)(CNCc1cccc2cc[nH]c12)CCS(C)(=O)=O 62370,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)C(C)C2CC2)C(CCO)C1 62371,N1(C(C(C)SC)=O)CCCC(C2CCN(C(=O)C(C3CCC(=O)N3)C)C2)C1 62372,c1(NC(c2ccc(NC(C3C(C(=O)OC)C3)=O)s2)=O)cn2c(C)cccc2n1 62373,C1(COC)(NC(=O)Cc2cnn(C)c2)CN(C(=O)C=CC(N)=O)C1 62374,CCC(CC)C(C)C(=O)NC1CCC(F)(CNC(c2n[nH]c(C)c2Cl)=O)C1 62375,C1(C(=O)NC2CC(CNC(c3c(C)csc3C)=O)C2)COc2cc(F)ccc2C1 62376,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)(C)C)cc(C)c2nc(C)cn2n1 62377,NS(=O)(=O)c1ccccc1CNC1CCCN(CCC2C3COC2C3=O)C1 62378,C1(CN(C)C(c2cccs2)=O)CC(O)CN1C(C1CCC(c2cc[nH]n2)O1)=O 62379,C#CC1(O)CCCN(C(=O)CC2CC3(CC3)CN2C(c2csc(C)c2C)=O)C1 62380,C1(CNC(CCC(C)O)=O)CCCC12CCN(C(=O)C(=O)C(C)(C)C)CC2 62381,Cc1cnn(C)c1CNC(C1CC1C#N)=O.C12(CCCC1)CC(=O)N2C 62382,C1(NC(c2cc(C)sn2)=O)C2CC1N(C(c1cccc(N)c1Br)=O)C2C 62383,c1(C(=O)NCC2N(C(C(C)C(F)F)=O)CCCCC2)cnn2cnccc12 62384,C(C(CC(=O)NC1CC(C)OC1=O)NC(C1SCC=C1C)=O)OC 62385,N1(C(c2c(C)cc(C)nc2)=O)CCN(C(c2[nH]cc(C)c2C)=O)C2CCC12 62386,Cc1cc(C(=O)NCc2cnc(C)n2-c2ccccc2OC(C)(C)C)ccc1C#N 62387,N1(C(=O)CCC2CC2(F)F)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 62388,N1(C(CC2CC(OC)C2)=O)CCC(O)C(NC(=O)C(c2ccc(C)cc2)(C)C)C1 62389,c1(C(N2CC(C)C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)=O)ccc(Cl)c(F)c1 62390,C(CN=C(NCc1cnco1)NCC1CCCCC1C)NC(CC)(C)C 62391,C#CCC(C(=O)NCc1nc(C)cs1)NC(c1sncc1C)=O 62392,C(=O)(C(O)CC(C)C)N1CC2C(NC(c3n[nH]c(C)c3Cl)=O)(C2)C1 62393,c1(OC)cc(C)cc(Br)c1-c1ncc(CC(=O)NNC(=O)Cc2ccc(F)cc2)[nH]1 62394,C(=O)(C1CCc2c[nH]nc21)NC1(C2CCN(C(c3c(OC)scc3)=O)C2)CC1 62395,CCCCC(=O)C(=O)N1CC(CNC(c2cc(C)ccc2Cl)=O)C(C)(C)C1 62396,N1(C(C2(C)CC2)=O)CCN(C2COCC2NC(c2cc(C3(C)CC3)on2)=O)CC1 62397,C1(NC(c2cnccc2Br)=O)C(CNC(=O)C2=CCCC2)CCC12CCC2 62398,N1(C(c2ncc(OCC)cc2Cl)=O)CC2CCC1CN2C(C1CSC(C)=N1)=O 62399,N1(C(C(=C(C)C2CC2)F)=O)C2CCC1CC(NC(C1CCn3nccc3C1)=O)C2 62400,C1(NC(c2cccn3ncnc23)=O)CN(C(=O)CC2OCCO2)C2(CCCC2)C1 62401,C(C(=O)N1CCC(C(N2C3CCC2CC3)=O)O1)c1c(=N)[nH][nH]c1 62402,C1(C)(C(N(CC(=O)N)C2CC2)=O)CC2CCC1CC2=O.Cc1ccc(S)cc1 62403,c1(C(=O)NCC2(C)CCN(C(=O)C(O)P(C)(C)=O)C2)nccc2ccsc12 62404,c1(C(N2CC(C)CC(C(N(CCC)CC)=O)C2)=O)c[nH]c2ccccc12 62405,c1(-c2nc(C(N(CC=C)C)C)on2)cccc(-c2csnn2)c1 62406,N1(C(C(C)CN2CCOCC2)=O)C(C)C2CC1C2NC(=O)C(C)(C)N(C)C 62407,CC(CC(=O)N1CCC(C2CCCN2C(c2ccc(CO)cn2)=O)C1)C(F)F 62408,C1(CNC(C)=O)(CNC(=O)C(Cc2ccccc2F)c2cncs2)CCCCC1 62409,CCC(CC(=O)NOC(C1CCCCC1)CO)N(C)C(C1CCOC1(C)C)=O 62410,n1(CC(CC2CCOCC2)NC2CCN(CC#CN)C2)ncc(O)nc1=O 62411,c1(CCN(C(=O)CSC(F)F)C)nc(C(N)=O)cs1 62412,n1(CCC)ncc(C(=O)NCC2CC(NC(C3CCCN3C)=O)C2)c1C 62413,C(C(C)(C)CN(C)C)NC(CN(C(=O)CCc1ncco1)C(C)C)=O 62414,CC(C(=O)NCCc1ccsc1)(C1CCC1)NC(C1CCOCC1)=O 62415,Cc1ccc(Cn2cc(CC3(C4N(C(CS)=O)CCC4)CC3)nn2)cc1.C1CC1 62416,S(=O)(=O)(c1cccs1)N(C(C)C(=O)N1CC(c2ccc(O)nn2)C1)CCO 62417,CCC(CC)C(C(=O)N(CCC(=O)NCc1ccc(C)s1)CCCO)OC 62418,C(C(=O)N1CCC(C(=O)N(CC(CC)CO)CC)O1)N(CCC)C 62419,c1(NC2CCC2)nc(Cl)ccc1F.CC(c1cccs1)=CC(=O)N1C2CC2C1=O 62420,Cn1ccc2ccc(C(N3CC(NC(C4CCOCC4)=O)C3)=O)cc12 62421,C1(C(=O)NCCCNC(C2C(C)CC2C)=O)CCCCNC1=O 62422,c1(NC(c2cccc(Cl)c2)CC)ncnc2c1CCO2 62423,c1(C(=O)OC)cnsc1NCCC(C)(C)NC(C1CN(c2ccccc2)C1)=O 62424,CS(=O)(=O)c1ccc(CN2CC3C(Nc4ncc(I)cn4)C3C2)c(F)c1 62425,N1(C(c2c(C)nc(O)nc2C)=O)CC2CCCC2(N=c2[nH]nc(C(C)C)o2)C1 62426,c1(C(N2CC(CC(=O)Nc3ccccn3)OCC2)=O)ccc2cccnn12 62427,Cc1oc(-c2ccco2)nc1C(=O)NC1CCN(C(=O)C(C)OCC(C)C)C1 62428,N1(CC)N=C(C(=O)N(C2CCC(NC(=O)C=C(C)C(C)(C)C)C2)C)CCC1=O 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62463,Cc1cc(C(=O)NC2(CCCNC(=O)CC3CCN(C)C3=O)CC2)cc(C)c1C 62464,C1(NC(c2c(OC)nsc2)=O)CCN(C(=O)CSC(F)F)C1C 62465,N1(C(Cc2cn(C)nc2)=O)C2CCC1CC(CNC(C1CC(C)(C)CO1)=O)C2 62466,c1(OCC)ncc(C(=O)NCC2CCCCC2NC(C2CNC(=O)N2)=O)cn1 62467,Cc1c(NC(C2(c3ccc(F)c(F)c3)CC2C)=O)cccc1C(F)(F)F 62468,Cc1cnc(C(=O)NCC2CN(C(=O)C(=O)NCCC(N)=O)C3CC23)c(C)c1 62469,O=C(C(O)C(F)F)NCC1CC1CNC(=O)CCc1nnc(C(F)F)o1 62470,Cc1[nH]nc(C(=O)NCCN(C(=O)CCCCN2CCCCC2)C2CC2)c1C 62471,c1(C(N(CC(C)NC(C2CC3CCC2C3)=O)C)=O)cnc2c(c1)N(C)CCO2 62472,C(=O)(C(C)C(=O)N1CCC=CC1C(=O)N(CC(O)CO)C)OC 62473,C1(NC(=O)C(C)(C)C2CCCO2)CCCCC1CNCc1c(C)non1 62474,C(=O)(C(O)C(F)(F)F)NC(COC)CC(=O)NCC12CCC(CC1)C2 62475,c1(C(=O)NC2CC(NC(c3cc(C)c(C)s3)=O)C2)cnn2c1CC(C)CC2 62476,C(C)(C(=O)N1CC(O)(CCNC(C2(C3CCOCC3)CCC2)=O)C1)(C(C)C)OC 62477,c1(N(CC2C(C)CCC2)CC2CC2)c(F)ccc(N)c1Br 62478,CCCCC(CNC(=O)NC1CC(OCC(=O)C2CC2)C1)NC(=O)C(C)S 62479,c1(C(N)=O)ccccc1C(=O)NCC1CCC1NC(=O)C=Cc1cnccn1 62480,N1(C(C(CC=CC)C)=O)CCN(C(c2nccn2C(C)C)=O)CC1CC(F)F 62481,C1(NC(CC(=C)C)=O)COC2CN(C(c3sccc3NS(C)(=O)=O)=O)CC12 62482,C1(C(=O)NCCC2(OC)CN(C(C(C=C)(F)F)=O)C2)CCC2CCC(=O)N12 62483,c1(C(=O)NCC2OCCN(C(C=CC)=O)C2)cc(C(C)C)cc(Br)c1 62484,c1(C(N2CC(NC(CN(C3CCCC3)C)=O)C3C2C3)=O)n[nH]c2c1CCSC2 62485,C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(N2CCOC3CC23)=O)(OC)C1 62486,c1(N(C(=O)Cc2ccc(C)cc2C)CC)nc2ccccc2o1 62487,c1(C(=O)NC2CC(NC(c3cccc(OC(F)F)c3)=O)C2)cc(CO)cc(Cl)c1 62488,CCC(CC(=O)N1CC(O)(C(F)C(N2CCC(OCCF)CC2)=O)C1)OC 62489,c1(CCC(N2CC(CNC(C(C)(Cl)Cl)=O)C(O)CC2)=O)cc(F)c(F)c(F)c1 62490,c1(OCCN(C(C2COCCO2)C(=O)OCC2CC2)CCC)ccccc1 62491,c1(OC)cc2c(=O)c(C(N3CCC4(CCC(O)C4)C3)=O)c[nH]c2cc1C(C)=O 62492,N12CCCC1CNCC1C(C1)C2=O.C(=O)(C(C)C1CCCC1)OC 62493,c1(-n2cc(C3(OC)CN(C(C(C)N(C)CC)=O)C3)nn2)ccc(F)cc1NC(N)=O 62494,C(=O)(C(C)CC(C)(F)F)N1CCC(CCNC(CNC(C(C)C)=O)=O)CC1 62495,CCC(C)CC(C)C(=O)NCC1(C(N2CCN(CCO)CC2C)=O)CCC1 62496,c1(O)c(F)cc(F)cc1Br.Cc1cnc(NC(C2CCN(CCO)C2)=O)cn1 62497,N1(C(c2ccc(C)cc2F)=O)CCCN(C(c2sccc2CO)=O)C(C)C1 62498,CC1(NC(=O)C(F)C2CCOC2)CCCN(C(=O)C=CI)C1 62499,N1(C(C(CC=C)NC(=O)Cc2ccoc2C)=O)CCS(=N)(=O)CC1 62500,N1(C(C2=CCN(C(C3(C(=O)OC)CCCO3)=O)C2)=O)CC2C3CCC(C3)C12 62501,C1(C(N(C(CC(=O)N(C)Cc2ccc(C)cn2)(C)C)C)=O)CC2(CCCO2)C1 62502,CC(O)CCCCCC(=O)NCCN(c1ncccc1C(F)(F)F)C 62503,N1(C(COC(C)=O)=O)CCCCC2(CCN(C(=O)C=Cc3cnn(C)c3C)C2)C1 62504,CC(C)CCC(=O)NCC(C)(CO)NC(c1ccc(OCCOC)nc1)=O 62505,c1(C(=O)NCC2C(C3CC3)CCN2C(C2CCCCO2)=O)cccc2sccc12 62506,c1(C(=O)NCCCOC)ncc(N)nc1C.c12nccc(n1)N1CCC(C1)N2C 62507,C1(NC(CC=C)=O)CN(C(=O)CN(CC(C)(C)C)C)C2(CCC2)C1 62508,C1(NC(C(C)Cn2ccnc2)=O)CCS(=O)(=O)C12CN(c1nnc(O)s1)C2 62509,C(=O)(CCCC(=O)N(C)C)NCC(C)(CO)NC(C(CNC(C)=O)C)=O 62510,N1(C(CSCC)=O)CCC(NC(c2ccc3c(c2)CCC(O)C3)=O)C(F)(F)CC1 62511,C1(CN(C(=O)C(F)C2CCCC2)CC)CCCN(C(C2CC2C(C)(C)C)=O)C1 62512,C(CCC(C)(C)C(=O)NCC1CCCNC1=O)NC(C(CC(=O)OC)C)=O 62513,Cc1cc(C(N2CCC(CO)(CNC(=O)Cc3sccc3C)C2)=O)cc(N)c1 62514,c1(CNC(=NCCCN2C(=O)NCC2)NC2CCC2)cc2c(s1)CCCC2 62515,N1(C(C2(c3ccccc3)CCCC2)=O)CC(O)C(O)C(O)C1CNC(=O)C1CC1 62516,c12ccc(cn1)OCCCN(C)C2=O.c1(C(C(C)C)O)ccc(F)cn1 62517,C1(NC(C2(C)CC(=C)C2)=O)CN(C(=O)C(O)CC(C)C)C2(CCC2)C1 62518,Cc1ccc(C(C)C)cc1C(=O)NC(C)CC1CN(C(=O)C(O)CN(C)C)C1 62519,C1(C(N2CCN(C(CN(CCOC)C)=O)C(CF)C2)=O)CCC(N=[N+]=[N-])CC1 62520,c1(C(N2C3CN(C(C=CS(CC)(=O)=O)=O)CC2CCC3)=O)cc2ccc(Cl)cc2s1 62521,c1(NC(c2scc(CNC(COCCC#C)=O)c2)=O)cc2n(n1)CCO2 62522,C1(C(N(C(C)C(N2CCCC2CC(=O)NC)=O)CC#C)=O)CCC(C#C)C1 62523,c1(NC(CC=C=C)=O)ccc(Cl)c(Cl)c1.C12CN(CC1C)C(=O)CNC2=O 62524,CCCCC#CC(C)(C)NC(C1CN(C(C2(C)CCCC2O)=O)CC1C)=O 62525,C1(C(N(CCCNC(=O)C#CC2CCCC2)CC)=O)CCCN1S(=N)(=O)N(C)C 62526,c1(C(=O)NC2CC3(CN(C(C(COC)OC)=O)C3)C2)nccc(C#N)c1F 62527,C(=O)(C(CC)CCOCC)NC1(CC=C)CCN(S(=O)(=O)CCOC)C1 62528,C(C(=O)N1CCC2CC12)(C(C)(C)O)N(C(CC1(CCC=C)CC1)=O)CC 62529,C1(NC(C(CSC)c2ccccc2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1(C)C 62530,C(=O)(C(C(C)C)CC1(CC(=O)NCC)CC1)NCC(CCC)OCC 62531,c1(CCC(=O)NCC2CN(CCNC(CSCC)=O)C2)ccc(F)cc1Cl 62532,C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(=O)C(F)=C2CCCC2)C1 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62550,O=C1NCCc2occ(NC(=O)C(N3CCCC(CN4CCCC4=O)C3)=O)c21 62551,Cc1nc2[nH][nH]cc-2c(=NCCC2CCCN(C(=O)CCC(F)F)C2)n1 62552,c1(C(N(CC(C)NC(=O)CC2CCC(C)(C)CO2)CC)=O)c(F)ccc(N)c1F 62553,C(=O)(C(CC)C(F)(F)F)N1CC(F)(C2CN(C(C(C=C)CC)=O)C2)C1.c12cn(nn1)C2 62554,C1(C2=CC=CC=CC(CC)(NC(CN(C)OC)=O)CCOCCO2)CCC(=O)N1 62555,CC(CC(F)F)C(=O)NC1C2CN(C(=O)Cc3cccc(O)c3F)CC12 62556,C1(CC(=O)NCC(C)(C2CC2)NC(c2ccc(SC)o2)=O)CCCCC1CO 62557,C(CCSC)(C(=O)NC1(CC(=O)NOC(C)C(=O)OC)CC1)OC.C(C)(=O)N 62558,Nc1cc(F)ccc1C(=O)NC1COCC1NC(C1CC1C(F)F)=O 62559,C1(NC(=O)NCCn2cc(CCc3ccccc3)nn2)CCn2ncnc2C1 62560,O=C(C(F)C1CCCC1)NCC1CCC1NC(=O)C(O)C1CC1 62561,N1(C(C2C(C(N)=O)C2)=O)CC2(CO)CC1(C(=O)NC1CCC3CC13)C2 62562,N1(C(c2c(O)ccc(C)c2)=O)CCCN(C(=O)C(O)Cc2cnc[nH]2)C(C)C1 62563,N1(C(CC(COC)C)=O)CC2(CC(NC(=O)CC3CSCCO3)C2)C1 62564,c1(C(=O)NCC(C2CCC2)NC(C(C=C=C)C)=O)cnc(C)c(C)c1 62565,N1(C(c2cn3ccsc3n2)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 62566,C(=O)(C1=C(F)CN(C(=O)CCS(N)(=O)=O)CC1)N(C)CCN1CCCC1 62567,c1(OC)cc(NC(C2CC2NC(c2ncccc2S(C)(=O)=O)=O)=O)c(Br)cc1F 62568,C1(NC(CCOCC(C)C)=O)C2CC(O)C1N(C(C1(C)CC(=O)N(C)C1)=O)C2 62569,Cc1cc(NC(=O)CCCNC(N)=O)ccc1NC(=O)CCc1cnn[nH]1 62570,c1(CC)nc(=N)[nH]c(=NCC2CCCN(C(C3OCC(C)C3C)=O)C2)[nH]1 62571,CC(C)(C)C(C)(O)C(=O)NC1CC(F)CN(C(=O)Cn2cc(F)ccc2=O)C1 62572,N1(C(C2(NC(c3c(C)nc(O)cc3)=O)CC2(C)C)=O)CCCN(C)CCC1 62573,c1(C(=O)NC(CC)CNC(c2cc(C3CC3)on2)=O)c(C)noc1CC(C)C 62574,CC(C)CC(C(=O)N(C)CCN1CCCCC1)NC(=O)C(C)n1cccc1 62575,C1(CC(=O)NCC(N(C(c2c(C)snn2)=O)C)C2CC2)CCS(=O)(=O)CC1 62576,C(=O)(C1CCCc2c(O)cccc21)NC(CCCC)CNC(c1c[nH]cc1Br)=O 62577,S(=O)(=O)(CCC(=O)NC(C(=O)NCC1(C)CNC(=O)O1)c1cccs1)NC 62578,Cc1cc(C(C)C(=O)NC2C=CC(CNC(=O)CC(C)(C)F)C2)cc(F)c1 62579,C=C(C)CCCC(=O)NCC(C1CCN(C(c2coc(C(N)=O)c2)=O)CC1)F 62580,c1(C(=O)NCCC(O)CNC(c2n[nH]c3c2COC3)=O)ncnc(O)c1F 62581,C1(CNC(C(C)SCC)=O)CCC2(CN(C(c3oc(Br)cc3C)=O)C2)O1 62582,CC1(CNC(c2cccc(O)n2)=O)CCN(C(C2CCC2C(=O)OC)=O)CC1 62583,c1(C(C)C)cnc(O)c(C(N2CC(CNC(C3CC(OC(F)(F)F)C3)=O)C2)=O)c1 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62619,N#Cc1cnc(C(N2CC3CC(NC(C4CCC(=O)NC4)=O)CC3C2)=O)c(Cl)c1 62620,c1(NC(c2n(C)cc(NC(c3cc(Cl)ncc3F)=O)c2)=O)cc(Br)cc(F)c1O 62621,CCC(C)CCC(=O)N1CCCCC1CCNC(c1cc(C)on1)=O 62622,c1(CC)nc(C(N2CCCC2(C(=O)NCCn2cccn2)COC)=O)c(C)o1 62623,c1(C(=O)NC2CCCN(C(Cc3onc(C)n3)=O)C2C)ccc2c(c1)CCOC2 62624,c1(C(N(CCCNC(=O)OC)C)=O)ccccc1OCC(=O)OC 62625,C1(C(=O)NCc2c(C(=O)NC(C)(C)CCCF)n(C)nc2)CN2CCC1CC2 62626,c1(CC(=O)NC(C)C(CO)NC(C2CCC(=O)C2)=O)csc2c(F)cccc12 62627,c1(OC)cc(C(N2CCC(n3cc(C4CC4CO)nn3)C2)=O)cnc1Cl 62628,c1(C(N2CCC(C)(C(=O)NCC(N3CCCCC3C)=O)C2)=O)cc(F)cc(I)c1 62629,C1(C2CN(C(C3C(O)C(=O)N(C)C3)=O)C2)(NC(C(C)NC(N)=O)=O)CC1 62630,C=CC1OCCC1C(=O)NC1(C(=O)N(C)CC2CC2(C)C)CCC1 62631,c1(C(=O)NCC23CC2CN(C(=O)CSc2ccoc2)C3)ccc(C2CC2)cc1F 62632,C12CCCC3(CCN(CC3)C1=O)O2.C(CC(=O)NC(C1CC1)C1CC1)OC(C)C 62633,C1(C(N(CCN(C)C(c2ccc(CC(C)(C)O)s2)=O)C)=O)C(F)(F)C12CC2 62634,c1(SC)cccc(C(=O)NCC(C(C)C)NC(C2C(Cl)(Cl)C23CC3)=O)c1 62635,c1(C(=O)NC2(C)CCN(C(=O)CNC=O)C2)ccc2ncccc2n1 62636,Cc1ccc(CC(N2CCC(F)C(NC(c3cc(Cl)c(Cl)n3C)=O)C2)=O)cc1C 62637,N1(c2nccc(C#N)n2)CC2CCC(NCc3ccc4nc(O)[nH]c4c3)CC2C1 62638,C12(C(=O)NCCC(C)N(C(CC(CCC)(C)C)=O)C)CCCN(C1)S(=O)(=O)C2 62639,c1(C(=O)NC2CC(N(C(CCC(C)N(C)C)=O)C)C2)nn(C)c2ccc(F)cc12 62640,n1(CNC2C3CN(CC(F)(F)F)CC23)ccc(=O)n(C)c1=O.C12CC(C1)C(=O)N2C 62641,CCC(C(=O)OC)C(=O)NC1COCCC1NC(c1cnn(C2CC2)c1)=O 62642,c1(N(C)CCC(c2ccccc2)CO)ccc(S(=O)(=O)N2CCSC2)c(Cl)c1 62643,Cc1nn(C)cc1NC(=O)CN(C(=O)CCCC#N)C 62644,N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(CCN2C(=O)C(O)C2CCCC2)C1 62645,Cc1cnccc1C=CC(N1CC=CC(NC(C2CCNC(=O)C2)=O)C1)=O 62646,C(CC(CNC(c1n[nH]cc1C1CC1)=O)NC(=O)COCC(C)(C)C)OC 62647,N1(C(CN(C(C)=O)C)=O)CC(OC)CC1CCN(C(=O)C1=COCC1)CC(C)(C)C 62648,N1(C(c2c(Cl)nc(N(C)C)s2)=O)CC(CNC(=O)C(C)(O)C(C)C)CC1(C)C 62649,C12(C(=O)NCCC(C)NC(=O)C=CCOC3CCOCC3)CCOC(C)(C1)C2 62650,c1(C(=O)NCC2(C(F)(F)F)CC2(F)F)ccccc1C1CC1(F)F 62651,CC1Cc2cc(S(=O)(=O)N3CC4COC(=O)C4C3)ccc2O1 62652,C1(C)(NC(C(C)C)Cn2cccn2)C2CNCC12 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62722,c1(C(=O)NC2C(CNC(Cc3nc(CC)sc3)=O)C2)cc(O)c2ccccc2c1 62723,N1(C(CCCCN(C)C)=O)CCCCC2(C1)CN(C(=O)C(Cl)=CCl)C2 62724,c1(C(=O)NCC2N(CC(=O)NC3CC(CF)C3)CCC2)ccc(OC(F)(F)F)cc1 62725,c1(NC(C2C3(CN(C(C(C)S)=O)C3)C2)=O)cn2nc(Cl)ccc2n1 62726,c1(NC(CCc2ccc(C)cc2Br)=O)nn(C)c(C(C)C)c1S(N)(=O)=O 62727,CCCCCCC(C)CC(=O)N1CC(F)CC1CN(C(=O)C#CC(C)(C)O)C 62728,c1(C(=O)NCC(C)N(C(CCc2c(C)cccc2)=O)C)cc2c(C)sc(C)c2s1 62729,C1(CC)(NC(=O)C(C(C)O)c2ccccc2)CCN(C(=O)CN(C)C(C)C)CC1 62730,C(=O)(C(=O)N=c1ccn(CCO)[nH]1)N(CCC(N1CCN(C)CC1C)=O)CC(F)(F)F 62731,C1(CNC(c2c(C)sc(Cl)n2)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCN1C 62732,N1(C(C(CC)O)=O)CCC(CCNC(=O)COCc2nc[nH]n2)C(F)(F)CC1 62733,c1(C(=O)NCC2CCC(NC(C(COC)O)=O)C2)cc(NC(C)=O)cc(Cl)c1 62734,C1(C(=O)Nc2cn(CCC)nc2)CCCN(C(=O)C(=CC2CCCC2)C)C1 62735,C(CNC(=O)CC(n1nc(C)cc1C)C)(CC)(CC)NC(C(C)=CC)=O 62736,N=c1[nH]c2cc(C(=O)NC3CC(F)(CNC(c4ccc(Cl)c(F)c4)=O)C3)ccc2s1 62737,N1(C(C(C(C)(C)O)F)=O)CC(CNC(C2CCCC2)=O)CC12CCOCC2 62738,c1(N2CC(CNC(C3(C)CS(=O)(=O)C3)=O)OCC2)ncccc1[N+](=O)[O-] 62739,c1(C(C)CC(N2CCN(C(=O)CC(O)CN(C)C)CC2)=O)c(F)cccc1F 62740,C1(CC)CCCC1C(=O)NC1(CC=CC(=O)NCCCCc2cnc[nH]2)CCC1 62741,c1(NC(=O)NC2C(NC(COc3ccc(C)cc3)=O)COC2)cc(F)ccc1F 62742,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 62743,c1(C(=O)NC2(C)CN(C(=O)C(F)(F)c3ncccn3)C2)scc(Cl)c1Cl 62744,c1(NC(N2CCCC(C)(C(F)F)C2)=O)n[nH]c2c1CC(C(C)(C)C)CC2 62745,C(=O)(C(C)C(C)(C)c1ccccc1)N(CC(CNC(CC(COC)C)=O)C)C 62746,C1(C(=O)OC)CC(N(C)C)CN(C(c2nc(C(C)C)cs2)C(=O)OC)C1 62747,C1(CCNC(c2ccc(C(F)F)o2)=O)COCCN1C(=O)CCN1CCOCC1 62748,Cn1cc2cc(C(=O)NCCC(C)(C)CNC(c3c[nH]c(=N)o3)=O)ccc2n1 62749,C1(CNC(CC2(C=C)CC2)=O)C2CCC(C2)N1C(c1cccc(NC(=O)NC)c1)=O 62750,c1(C(N2C(C)(CNC(COCC(=O)NC)=O)CCC2)=O)cc(Cl)c(C)cc1OC 62751,C(=O)(CC1COc2cc(O)ccc21)N1C2CC(CN(C(C(CCC)(C)C)=O)C2)C1 62752,c1(C(=O)NCC(=C)CCNC(=O)C(CC)NC(C)=O)cc2sccc2s1 62753,C1(SCC(C)NCCOC(=O)C(C)(C)c2ccccc2)CCCC(O)C1 62754,c1(NC(C2C3CN(CCOCC4CCCC4)CC23)=O)c(Cl)nnc(Cl)c1Cl 62755,C#CCCCCCC(=O)NC1CCC(NC(C2(O)CCOC2)=O)C1 62756,c1(NCCCN2C(C)CCC2)nc(N2CCC(CN(C)C)C2)nc2c1ncn2C 62757,N1(C(CC(CC)SC)=O)CC(NC(c2conc2SC)=O)CC12CCOCC2 62758,N1(C(c2c[nH]c(=N)o2)=O)CCC2(C1)CN(C(c1cscc1Br)=O)CCO2 62759,N#Cc1c[nH]c(C(=O)NC2CN(C(c3cccc(OC(F)(F)F)c3)=O)CC2F)c1 62760,Cc1ccc(C=CC(=O)NCCCCNC(=O)Cc2ccc(OC3CC3)cc2)o1 62761,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCCc2ncccc2F)C(C2CC2)C1 62762,N1(C(CCCCCOCC)=O)CCOC2(C1)CN(C(=O)C(CSC)OC)C2 62763,CON(CCC(=O)Nc1cnn(C)c1O)C(=O)c1cc(C)c[nH]1 62764,C1(C(N2C(C#C)CC2)=O)C2CCC(C2)N1C(=O)Cn1c(C)ccc1C 62765,Cc1ccc(C=CC(=O)NC2CC(C(F)C(=O)NCc3ccc(C)o3)C2)o1 62766,C(CCCCC(=O)NCC1=CCCN(C(=O)C(F)(F)CO)C1)N(C)C 62767,CCCC(C)(C)CC(=O)NC1CC=C(C(=O)NC(c2ccnn2C)CC)C1 62768,CCCCC(C)CCC(=O)NC(CCC(=O)N(CC(=O)NCC)C)C(C)C 62769,C(C)(C(=O)N(O)Cc1cn(-c2ncccn2)nn1)OCC=C 62770,c1(C(N(CCCN(C)C)CCNC(c2c(OC)n[nH]c2)=O)=O)nc(C)sc1Br 62771,N1(C(c2c(C)nc(Br)cc2)=O)CC2(CCN(Cc3cccc4[nH]ccc34)CC2)C1 62772,c1(OC)cccc2c1C(C(=O)N1CC(OC)C1)CC2=O.C(=O)(COCC(F)F)O 62773,N1(C(c2cnc(SC(C)C)nc2)=O)CCCC(O)(CNC(=O)C(C)(Cl)Cl)C1 62774,C(=O)(N1OC2CCC1CC2)C1N(C(C(CC)c2ccccc2)=O)CCC1(C)C 62775,c1(OC(C)=O)ccc(F)cc1C(=O)N(C)C.C12CC(CN1C1CCCC1)OC2 62776,c1(OC)cnc(C(=O)NCC2CCN2C(C2CC2C2CCCO2)=O)cn1 62777,CCC(C)(C)C(O)C(=O)N1CC(N(C(=O)Cn2ccc(C(F)F)n2)C)C(C)(C)C1 62778,c1(-c2cn(C3C(NC(C(C=C=C)C)=O)COC3)nn2)cc(F)c(F)cc1F 62779,N1(C(c2c(C(C)C)ncs2)=O)CCCC(C(C)(C)C)C1.C12CCCC1C(=O)N2 62780,c1(OC)ccc2cc(CN3CCCC(C(=O)N=c4cnc(I)c[nH]4)C3)oc2c1 62781,C1(CNC(CC2(NC(C3(CC(C)C)CC3)=O)CCOC2)=O)CC12CCCCC2 62782,c1(NCCOC)ncccc1C(=O)NCC1CCC1NC(C1CC=CC1)=O 62783,c1(OC)ccc(C(N2CC(C)CC2C(N2CC(NS(C)(=O)=O)C2)=O)=O)cn1 62784,C1(NC(N(C2(C)CCOCC2)C)=O)CN(C)CCN1C 62785,c1(SCC(=O)N)ccccc1CC(=O)NCC1C(CCOC(C)=O)C1.C1(C)CC1 62786,c1(N2CCC(NC(C(c3ccccc3)OCC(C)C)=O)C2)ncccc1C#N 62787,N1(C(CC(=O)NCC)=O)CC2ON=C(CNC(c3cncc(F)c3)=O)C2C1 62788,C1(NC(c2coc3c2COC3)=O)CC2(CCN(C(C3(CO)CC3(F)F)=O)CC2)C1 62789,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(F)cc1)C2 62790,N1(C(=O)CC2(c3ccccc3)CC2)CC2CCN(C(C3(O)CC3)=O)CC2C1 62791,N1(C(CCN(C)C)=O)CC2C(CN(C)C(C3CCC(C(N)=O)N3C)=O)C2C1 62792,CC1N(C(C2CCN(C(=O)c3cncnc3)O2)=O)CCCC1(C)C 62793,c1(C(C)C)ncc(Br)c(=NC2CC2C(=O)NCCn2ccnn2)[nH]1 62794,N1(C(CP(C)(C)=O)=O)CCC2(CC2)CC1C(N1CCC(c2cccnc2)CC1)=O 62795,Cc1cnc(C(=O)NC2(C)CCCN(C(=O)CC3CCOC3)C2)c(Br)c1 62796,C1(OC)CC(NC(=O)CO)C12CCN(C(=O)CCSCc1cccc(Cl)c1)CC2 62797,C1(CC(N2CCCC2Cc2cn(CCOCCO)nn2)=O)(OC)CCCC1 62798,N#Cc1cccc(C(O)C(=O)NCc2ccnc(OC3CCCCC3)c2)c1 62799,O=C(C1=CCCSC1)NC1CC(NC(=O)C(C2(O)CCCCC2)(F)F)C1 62800,Cc1cncc(C)c1NCc1ccc(C(F)(F)F)cc1 62801,C12(C(=O)NCC3CCN(CC)C3)CC(CCO1)N(C(=O)C(F)C(F)(F)F)C2 62802,C(CNC(c1cnc(S)n1C)=O)(CC(C)C)NC(COCc1cc(C)on1)=O 62803,C1(C)(C(=O)NCCCCN(C(C2CC(C)N(C)C2)=O)C)CCC2CC2C1 62804,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 62805,c1(C(=O)NC2C(NC(C3(CC#C)CCCOC3)=O)CC2)nnc2ccccn12 62806,c1(SC)c(C(N2CC3(C2)CN(C(c2nc(C4CC4)cs2)=O)C3)=O)cccc1Br 62807,c1(C(N(CCCN(C(COCCOCC#C)=O)C)C)=O)ccncc1Br 62808,N1(C(C)=O)CCN(CC(N2CC(NC(C3CC34CCC4)=O)C2)=O)CC1.C1(C)CO1 62809,N1(C(C(C(CC)C)O)=O)CC2CCC(N(C(=O)C=Cc3cccs3)C)C2C1 62810,CCN1C(=O)Cc2cc(NC(N3CC(O)CC(C)(C)C3)=O)ccc21 62811,N1(C(C(C2(O)CCC2)NC(c2nc(CC)oc2C)=O)=O)CCc2nnnn2CC1 62812,C1(CCNC(c2c(SC)n(C)nc2)=O)CC(F)(F)CN1C(c1cn[nH]c1)=O 62813,C(=O)(C(F)C(C)CC(C)(C)C)N(CCC)CCNC(=O)C(C1CCCCCC1)O 62814,Cc1ccc(CN2CCN(C3CN(C4(c5csc(O)n5)CC4)C3)CC2)cc1 62815,C(CNC(=O)CC1CC(F)(F)C1)(CC(=O)N(C)Cc1ncc[nH]1)OC 62816,c1(C(=O)NCc2c(CNC(C3CCC(C)(C)C3)=O)cccn2)cnc(N)c(N)c1 62817,CC1CSCCN1C(=O)CCN(C)C(C1CCCSC1)=O 62818,N1(C(C(C)C)=O)CCCC1(C)C(=O)NCc1nncs1 62819,C1(C(=O)NC(CN(C(c2sc(CO)nc2C)=O)CC)C)CCC2(CCOCC2)O1 62820,C1(NC(C(C)=C2CC2)=O)CC2CC(NC(=O)C=Cc3cncn3C)CC2C1 62821,Cc1nccc(C(=O)NCCN(C)C(c2cc(C3CCCCC3)on2)=O)c1C 62822,c1(C(C2CC2)NC(C(=O)NCCCC=CC)=O)c[nH]c2cc(OC)ccc12 62823,Cc1nc2ccccc2cc1C(=O)NCC(CO)NC(=O)C(O)CC[S+](C)C 62824,CC1(CC2CCCCC2)CC(F)(F)CN1Cc1nc(-c2ccc(Cl)s2)no1 62825,C1(CC(N2CC(CNC(N)=O)C2)=O)CCCCN1C(=O)C(F)n1ccnc1 62826,C(=O)(C1CCCn2cc(C(F)(F)F)nc21)OCCCOC(=O)C1CC1 62827,Cc1cc(-c2noc(COc3sc(C)cc3Br)n2)n(C)n1 62828,C1(NC(C)=O)CC(C(N2CCN(C(c3ccncc3)=O)CC2)=O)C12CCOCC2 62829,CC1CCCCC1CCNC(c1cc(CNC(=O)CCC2(C)CC2)[nH]n1)=O 62830,c1(C(=O)NCC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C2)ccc2nc(O)oc2c1 62831,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(c1cccnc1CO)=O 62832,c1(C(=O)NCC2N(C(=O)CC3CCNC3=O)CCN(C)C2)cncc2ccsc12 62833,c1(C(=O)NC(C)CCNC(=O)C(F)F)cc(Cl)cc2c1CCC2 62834,N1(C(C2CN(C(CCSCCC)=O)CC2(C)C)=O)CC2OC(=O)N(C)C2C1 62835,C1(C(=O)NCCCS(C)=O)CCN(C(=O)CCn2ccnc2)C12CC2 62836,C1(NC(C(CC)O)=O)CC(F)CN(C(c2ccccc2C2CCCC2)=O)C1 62837,CC(C)CC(O)C(=O)NC(C)CNC(=O)Cc1ncn(C(C)C)n1 62838,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(C2CCC2)=O)CC1COC 62839,C1(C(C)NC(Cc2ncc(CC)[nH]2)=O)CN(C(=O)CCn2ccnn2)CCO1 62840,N1(C(C(C)n2ccnn2)=O)CCC(CO)C(NC(C23CC(F)(C2)C3)=O)C1 62841,C1(C(=O)NCC2(CNC(c3ccc4nccn4c3)=O)CC2)CCC2(CCC2)CC1 62842,c1(NC(=NCCC2OCC(C(=O)OC)O2)NC2CC2)cccc(OCC)c1.C(CO)S 62843,N1(C(CC(C)(C)N(C)C)=O)Cc2nccn2CC(NC(C2(F)CCCOC2)=O)C1 62844,O=C1CC(C(=O)N2CCOCC(CNC(c3cccc(C(F)F)c3Cl)=O)C2)=NN1 62845,c1(C(=O)NC2(C(=O)NC3(CC)CCOC3)CCC2)ccnc(C)n1 62846,N1(C(C(CC)C)=O)CCCOC(CNC(c2ccccc2CN2CCCC2=O)=O)C1 62847,CC1(C)C(C(=O)NCC2(F)CC(NC(C3CCOC(C(F)F)C3)=O)C2)C1C#N 62848,Cn1c(CCC(=O)N2OC3C=CC2CC3)nc2ccccc12 62849,c1(C(N(C2CCN(C(c3sc(NC4CC4)nc3C)=O)C2)CC)=O)ccc(Cl)nc1 62850,C(=O)(CCCCC(F)F)N1C(CNC(c2cc[n+]([O-])cc2)=O)C(C2CC2)CC1 62851,C1(NC(C(c2ccc(C)s2)C)=O)C=CCN(C(=O)Cc2cnnn2C)C1 62852,C(C)(CNC(=O)C(C)SC(C)C)(C(C)C)NC(Cn1c(C)nnn1)=O 62853,CC1(C)C(NC(=O)C=CC2CCOC2)CCN1C(C12CCC(C)(CO1)C2)=O 62854,c1(CNC(=O)CC2CCCN(S(=O)(=O)C(F)(F)F)C2)cncnc1O 62855,c1(C(N2CCC(C(N(C)CC3(O)CCC3)=O)C2)=O)ncc(F)cc1N 62856,c1(NC(CN2CCC(C(=O)OC)(OCC)C2)=O)c(Cl)ccnc1C 62857,C1(C(=O)NCC2CN(C(c3c(OC)cncn3)=O)CC2O)CC2(CCOC2)C1 62858,c1(C(=O)NC2CC(O)(CNC(c3c(C)cc[nH]3)=O)C2)nc(C2CC2)ncc1Cl 62859,N1(C(C2C(OC)C2)=O)CCC(C)C(CNC(c2c[nH]cc2C(N)=O)=O)C1 62860,c1(OC)cc(C(=O)NCC2CCN2C(C2CC(CF)C2)=O)cc([N+](=O)[O-])c1Cl 62861,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 62862,c1(C(C)C)nc(NCCCC2CC2)cc(=NC(C)C2CCCC2)[nH]1.c1(S)ccccc1C 62863,N1(C(c2n(C(C)C)ncn2)=O)CC(NC(=O)CSc2ccccc2F)CC1C 62864,c1(C(N(CCNC(=O)Cc2ccsc2)C2CC2)=O)cccc(F)c1Br 62865,CCC(C)(C(=O)Nc1cccc(NC(c2cc(Cl)no2)=O)c1)OC 62866,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 62867,N(C1CN(C(=O)C(CC)ON)CCc2ccccc21)C(C1(C=C)CCOCC1)=O 62868,C#CCCCC(C)C(=O)NC(COCC=C)C(=O)NC(c1ncccn1)C 62869,c1(OC)cc2cc(C(=O)Oc3cccc(-c4nc(C)ns4)c3)[nH]c2cc1C(=O)O 62870,C(=O)(CC1=NN(C)C(=O)C1)N(C1C(C)CN(C(c2cc3ccsc3s2)=O)CC1)C 62871,N1(CCC)CC(C(N2CCCC(CN(c3nccc(CO)n3)C)C2)=O)CC1=O 62872,Cn1ccc2ccc(C(=O)NCC3CCC(NC(C4CC4(F)F)=O)CC3)cc12 62873,c1(C(=O)NCC2(C)CCCN2C(C2CS(=O)(=O)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 62874,n1(CC(n2cc(-c3cccc(Br)c3F)nn2)=O)ncn2cccc2c1=O 62875,c1(C(=O)OC)ncccc1CN1CCC(F)(C(=O)Nc2ccc(SC)nc2)C1 62876,c1(C2CN(C(C3OCCCO3)=O)C2)ccc(Br)nc1 62877,CCCC(C)(CC)C(=O)N1CC(NC(=O)CNC=O)C(C)(C)C1 62878,C1(NC(c2c(NC)scn2)=O)CCCC(C(N2CCCCC2CCCO)=O)CC1 62879,C(CCCCC(=O)NCCC(C)CCNC(=O)Cc1c(O)ncnc1O)SC 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62934,c1c[nH]c(=O)cn1.C1(CN)COC(CNC(C2(C(=O)SC)CCC2)=O)C1 62935,C1(NC(C=C(C)C(F)F)=O)CC2CCCC(C1)N2C(C1(C(F)F)CC(F)(F)C1)=O 62936,c1(C(C(=O)NC2CC(C)(C)C2)NCC(CCOC)(C)C)cc(Cl)cc(Cl)c1 62937,N(C1CC2CCCc3cccc1c32)C(C1(COC)CC1(F)F)=O 62938,N1(C(C2N(C(CCC(=O)NC)=O)CCC2)=O)CCC(C(=O)NOCC)C(C)(C)C1 62939,C1(C)(NC(C=C(C)CNC(=O)Cn2cnnn2)=O)CC2(CCC2)C1 62940,c1(C(N2CC(C)C(NC(=O)CN3CC4CC4C3)CC2)=O)ccc(S(N)(=O)=O)[nH]1 62941,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 62942,c1(C(=O)NC(CNC(C2C(C)(C(C)C)C2)=O)(C)C)ccc2nn[nH]c2c1 62943,N1(C(Cn2ccc(C)n2)=O)CCC(NC(=O)OC(C)(C)C)C1C(C)C 62944,N1(C(COC2(C)CCOCC2)=O)CC2COCC2(NC(C2CCCN2C(C)C)=O)C1 62945,N1(C(c2[nH]nc([N+](=O)[O-])c2Cl)=O)CCCC2C1CCCN2C(=O)C=CC1CC1 62946,N1(CC)CC2CCC1CN2C(c1ccc(CO)cc1F)C(=O)NCCCF 62947,c1(CC(=O)NC2CCC(NC(CN(C)CC)=O)C2)ccccc1[N+](=O)[O-] 62948,c1(C(=O)NC(C2CN(C(C3(C#N)CCCO3)=O)C2)C)cc2nccnc2cc1F 62949,c1(C(C)O)ccc2c(c1)OCO2.c12cn(nn1)CCC(=O)NCCCSC2 62950,C1(OC)(CNC(C2COC(=O)N2)=O)CCN(C(=O)Cn2ccccc2=O)C1 62951,c1(C(N2CC(CNC(C3COCCO3)=O)C(O)C2)=O)nc2ncccn2n1 62952,c1(OC)cccc2[nH]cc(C(N3CCOC(C(N4CC5C(C4)C5(C)C)=O)C3)=O)c12 62953,C(=O)(C1=C(Cl)CCOC1)NC1CN(C(C(C)OCCOCC)=O)C(C)C1 62954,c1(NC(COC)C2CC2)nc(=NC2CC2c2ccc(F)c(Cl)c2)[nH]c2c(C)nn(C)c12 62955,c1(C(=O)NCCN(C(=O)C=Cc2cccs2)C2CC2)cc2ccc(Cl)c(F)c2[nH]1 62956,c1(C(=O)OC)ccc(N(C)Cc2ccc(Cl)cc2)cc1Cl.C12CCN1C2=O 62957,C(C(CC(C)C)C(=O)NC1(n2ccnn2)CC1)NC(c1nnc(C2CCC2)s1)C 62958,N1(C(c2n(CC)ccn2)=O)CC2CC1C2NC(c1ncccc1OC)=O 62959,C1(CNC(C2(CCC)CC2)=O)CC(OC)CN1C(=O)CC(C)C1CCC1 62960,c1(N2CCC(CC)(CO)C2)nc(=NC(C)c2cc(F)ccc2Br)[nH]c2cc[nH]c12 62961,N1(CC(C)C)CCC(C(N2CCC(NC(=O)CC3CN(C)CC3O)C2)=O)CC1 62962,Cc1cnc(N2CC3CC(NC(C4CNC(=O)N4)=O)CC2C3)c([N+](=O)[O-])c1 62963,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 62964,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 62965,c1(C(=O)NC2CN(C(c3n(C(C)C)ncc3)=O)CC2O)c(Cl)nc2ccccn12 62966,C1(NC(c2c(OC)c[nH]n2)=O)CCC(CNC(=O)Cc2cncn2C2CC2)CC1 62967,c1(CN2C(CC(=O)NC3(C#N)CCOCC3)CCC2)c[nH]c2nc(Cl)ccc12 62968,C(C(C(=O)NC1CCC1NC(=O)Cc1cccc2nsnc12)C(C)(C)C)OCC 62969,C(C(C)(C)CC(=O)NC(C1CCN(C(N)=O)CC1)C)NC(n1cnnc1O)=O 62970,N1(C(CCOCC#C)=O)CCC(NC(=O)C(CC)N(C)C)C(CO)CC1 62971,Cc1ccc(C(C2(N(C)C)COC2)NC(=O)C(n2cc(C)cn2)C)cc1 62972,c1(CCC(=O)NCC2N(C(C(C=C)O)=O)CCOC2)cc(F)c(Cl)cc1Cl 62973,c1(C(=O)NCC2N(C)CCN(C(c3ccoc3CO)=O)C2)c2c(nn1C)CCC2 62974,C1(C(=O)NC(c2nc(CC)on2)C)CCCCCCN1C(=O)CC1C=CCC1 62975,C(=O)(C(F)CCC(C)C)N1CC(NC(c2[nH]cc(C)c2)=O)C(O)C1 62976,c1(C(=O)OCC)ccc(N2CC(CNC(=O)CCCOC(N)=O)C(O)C2)nc1 62977,N1(C(c2c(C)n[nH]c2)=O)CCCC(C(C)NC(=O)Cc2cc(Cl)cs2)C1 62978,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(N)cnn1C)=O 62979,N1(C(C(C)C2CC2)=O)CCOCC(CNC(=O)C(F)=CC2CC2)C1 62980,CCC(C)C(O)CN1CCC(CC(=O)NCc2ccc(OC(F)(F)F)cc2)C1 62981,N1(C(C(CCF)NC(c2ccn(C3CC3)n2)=O)=O)CCCC2CNC(=O)C12 62982,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 62983,C1(C#N)(C(=O)NCCC(C)NC(C(C)N2CCCC2)=O)CCSCC1 62984,N1(C(c2ccc(C)c(C)c2)=O)CCC2(C1)CN(C(=O)Cc1cc[nH]n1)CCO2 62985,Cc1cn2nc(C(=O)N(C3CN(C(c4cccc(C(C)C)n4)=O)C3)C)cc2c(=O)[nH]1 62986,C1(C(=O)NCC(CCOC)NC(c2cnccn2)=O)CCN(C(C)C)CC1 62987,Cn1cnc(NC2CCN(C(=O)CCCC3CC3)C2)cc1=O 62988,C1(C(=O)OC(=O)CN(C)C(=O)OCCCC)CCN(C(C2CC2F)=O)CC1C 62989,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(C)n2)C1)=O 62990,C(C1CCOC1)=CC(=O)NCCC(O)CNC(=O)C(F)(F)C1CCCCC1 62991,CC(C)(CC(=O)NOCC1CCCCC1)n1cc(-c2cncnc2)nn1 62992,C(=O)(C#CC1CCCC1)N(CCNC(CN(S(N(C)C)(=O)=O)C)=O)C1CC1 62993,C(CN=C(NCc1ccnc(C#N)c1)N(C)CC1CCN1C)OCC 62994,C1(C(=O)NCC(C)(C)NC(c2nc(OCC)sn2)=O)NC(=O)CC1C(F)(F)F 62995,c1(COC(c2n(C)nc(Br)c2)=O)cc(S(C)(=O)=O)cs1 62996,CC1OC2(C(=O)N(C3CCN(C(=O)CN4CCN(C(N)=O)CC4)CC3)C)CCC1C2 62997,CCC1=C(C(=O)N2CCC(CC(=O)NCC3OCCC3(C)C)CC2)CCCO1 62998,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CC(C)(C)SC)CC1(F)F 62999,C1(C(=O)NC2C(NC(CC3CN(C(C)=O)C3)=O)C2)CCCCC1C(F)(F)F 63000,c1(SCC(=O)N(CC(CC)NC(c2cccs2)=O)C)ccccc1N=NN(C)C 63001,n1(CCC(=O)NCCCN(C2CC2)CC)c(CC)nnc1S 63002,N1(C(COCCC)=O)CCC(C)C(NC(=O)COc2ccc(C(N)=O)cc2)C1 63003,Cn1ccc2[nH]c(C(N3CCC(F)(F)C(NC(C45CC6CC4C5C6)=O)C3)=O)cc12 63004,c1(NC(CCC2CCN(C(=O)CC3CSC3)C2)=O)cccc(F)c1O 63005,c1(CNC2CC(NC(c3ccccc3-c3ccsc3)=O)C2)cc(F)ccc1Cl 63006,c1(C(=O)NCC(C)NC(c2c(CC)cc(F)cc2)=O)cc2cncn2c(O)n1 63007,Cc1cccc(C(N2CC3(NC(c4ccsn4)=O)CCC2C3)=O)c1Cl 63008,c1(CC(=O)NCC2C(NC(COCCC#C)=O)CC2)coc2c(C)c(Cl)ccc12 63009,c1(C(=O)NCC2(NC(=O)CN3CCCC3=O)CCC2)cccc2cccc(O)c12 63010,N1(C(CNC(=O)OC)=O)CC(CNC(=O)C(C)(C)C2CC2)C(O)C1 63011,N1(C(C(C)CF)=O)CC(F)(F)CC1CNC(=O)Cc1cn(C)nc1C(F)(F)F 63012,N(C(=NCc1ccc(Cl)cc1)NC1CC1F)CCC1(C)CC1 63013,C(CC(C)(C)C)(C(=O)N1CC(C2CC2C(N2CCCC23CC3)=O)C1)OC 63014,c1(OC)nc(N2CCC(CCOC(=O)C3=CCOC3)C2)ncc1OC 63015,C(=O)(C1=CCC(F)(F)CC1)NC1CC(F)(CNC(CC(=C)C)=O)C1 63016,N1(C(CCCC=C)=O)C(CC(=O)NC2CCCCCC2C)C2CCCC12 63017,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)N(CC(=O)OC(C)C)C 63018,C(=O)(CCC(C)CN(C)C)NC1CN(C(COCc2onc(C)n2)=O)C(C)C1 63019,C1(CNC(c2ccoc2Cl)=O)CCN(C(=O)C(c2ccccc2)O)CC1 63020,c1(C(=O)NCC2CCN(C(C(CC)=CC)=O)C2(C)C)cccc(C)c1CCC 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63039,c1(C(=O)NC23CN(C(C(C4CC4)OCC)=O)C(C2)C3)c(C)nn2c1CCCC2 63040,N1(C(c2ccc(OC)c(Br)c2F)C(=O)NCS(N)(=O)=O)CCC2(COC(=O)N2)C1 63041,c1(C(=O)NC2(CNC(CCCOCC=C)=O)CCC2)ccc(N)c(Cl)n1 63042,C=CCC(F)(F)C(=O)NCC1CC(C)N(C(=O)C#CC2CC2)C1 63043,O=S(=O)(CCO)CCSC1CCCCCCC1 63044,c1(C(=O)NCC2(COCC)N(C(CC=CC)=O)CCC2)cc2n(n1)CCC2 63045,c1(C(N2CC(NC(C34CC(C3)S(=O)(=O)C4)=O)C3CC3C2)=O)ccnc2ncccc12 63046,c1(OCC(N2C(CNC(=O)CCCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63047,c1(C(=O)NC(C(C)NC(c2c(OC)ccc(F)c2)=O)C)cccn2ccnc12 63048,c1(CSC)ccc(C(=O)NC2CC(CNC(c3cccc(C)c3)=O)C2)cc1 63049,N1(CCNC(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 63050,C12(C(=O)NCC3N(C)CCN(C(CC(C(=C)C)O)=O)C3)C3CC(CC13)C2(F)F 63051,C(=O)(C(C)CC)NC(C(=O)NCC(CSCC)O)c1ccoc1 63052,c1(N2C(CNC(c3cc(CCC)[nH]n3)=O)CC(F)(F)C2)ccc(S(C)(=O)=O)cn1 63053,C1(C(=O)NCc2cn(CCOCc3ccc(Cl)cc3)nn2)CC2(CCC2O)C1 63054,CN=c1cc(C(=O)N(C(C)C(N2CCCC(C)(N(C)C)C2)=O)C)cc[nH]1 63055,c1(C(=O)NC2C(NC(c3cn(CCO)nn3)=O)CC2)cccc2cnsc12 63056,CC(CCNC(=O)C(F)F)CCNC(c1cccc(-c2ccc(F)cc2)n1)=O 63057,c1(NCC2CCN(C)C2)ncccc1S(=O)(=O)NC1COC2(CCC2)C1 63058,C(C(C)(C)C(=O)NCC(O)CC(=O)NC(C1CSC1)C)NC(C)=O 63059,c1(C(N2CC(NC(CCC#C)=O)CC(F)(F)C2)=O)c(F)cc(OC)c(F)c1F 63060,C1(C(=O)NC2CN(C(c3c(CCC)nsc3N)=O)C2)CC2(CCCC2)CO1 63061,C1(NC(C2CCOC2)=O)CN(Cc2ccc(-c3ccccc3)nc2)CC(F)(F)C1 63062,C12(COC)CC(C(N3CC(N(C(=O)CCc4cccnc4)CCO)C3)=O)(C1)C2 63063,N#Cc1ccnc(C(=O)NC(C2CCOC2)CNC(=O)CC2CSC2)c1F 63064,C(=O)(CCCCC(F)(F)F)NCC(n1cc(COC(C)=O)nn1)(C)C 63065,C=CC(C)(C)C(=O)N1CCC(O)(C(C)NC(c2[nH]ccc2COC)=O)C1 63066,C12(NC(Cc3n(C)ncc3Cl)=O)CCN(C(c3cc4sccc4s3)=O)CC1C2 63067,N1(C(Cn2cnc(=N)[nH]2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1CCO 63068,Cc1cc(C)c2[nH]c(CC3CCN3C(=O)OC(C)(C)C)nc2c1.S1(=O)(=O)CCN1 63069,c1(OC)cc(C(=O)Nc2ccc(CCc3ccccc3)cc2)cc(OC)c1OC 63070,Cc1cc(O)ncc1NC(=O)CC1C2CCCC2N1C(=O)CC(C)C(F)F 63071,N1(C(CN(C(C2CC3(CC(C)C3)C2)=O)C)=O)CCN(C)C(C)C1C 63072,Cc1csc(C(=O)N(C2CCN(C(c3c(C4CC4)noc3C(C)C)=O)C2)C)c1C 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63090,c1(C(=O)OC)ccc(C)nc1N1CCCCC(NC(=O)CCCCN(C)C)C1 63091,CC(CC(=O)NCCN(C(=O)Cc1ccccc1)C1CC1)n1ccnc1 63092,C1(NC(Cn2ncc(C#C)c2)=O)CC(CNC(=O)CC2CC3C=CC2C3)CC1O 63093,Cc1nc(C(=O)NCCC2(NC(=O)CN(C3CCC3)C)CC2)n[nH]1 63094,C1(C)(C(=O)NC(C2CN(c3ncccc3S(C)(=O)=O)CCO2)C)CCCCNC1=O 63095,C1(C(=O)NC2CC(CCNC(c3c(CC)ocn3)=O)C2)CCCC(C)(C)O1 63096,CCC(F)(F)CC(=O)NCc1ncoc1CCNC(=O)C(C)(O)CCC 63097,C1(CNC(c2c(CC)nco2)=O)CN(C(c2cc(F)ccc2CC)=O)CC1(F)F 63098,c1(C(N2CC3CC(O)CC3C2)=O)cc2nc[nH]c2cc1F 63099,Cc1ccc(C(=O)NCC(C)NC(=O)C(c2c(C)n[nH]c2C)C)c(N)c1Br 63100,C1(NC(C2(C(C)C)CCCN2C(=O)C=C(C)C)=O)CCC2CC1CO2 63101,Cc1cc(C(=O)N(CC(O)CN(C(=O)CC(C)F)C)C)nn1-c1ccc(Cl)cc1 63102,C1(C)(C(=O)NCC2(OC)CN(C(CCC(=O)OCC)=O)C2)CCCCC1C 63103,c1(C(N2C3CN(C(C4COCC4O)=O)CC2C3)=O)c(F)ccc2c1OCC2 63104,C(CC)(CC(=O)NCC(C)C(C)C)NC(c1cn(CC=C)nc1)=O 63105,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(=O)Cc1ccsn1)C2 63106,CC(CC(=O)NCC1CC1NC(=O)CC(=O)NC1CC1)P(C)(C)=O 63107,Cc1ccc(NC(C2CCCCN2c2ncnc3occc23)=O)c(F)c1F 63108,C1(CNC(C(CC)N(CC)CC)=O)CC(C)CN(C(C2(CCF)CC2)=O)C1 63109,c1(C(N2C(C(N(CCC#C)C)=O)CC3(CC3)C2)=O)cccc2c1CCC2 63110,C1(C2(C(=O)OC)CC2)COC2(CCC2)CN1N1C2CCCC1CC2 63111,CCCCCC(O)C(C)C(=O)N1CCCC(CNC(C2(CSC)CC2)=O)CC1 63112,C(C1CCC(C)CC1)=C(C)C(=O)N(c1ccc(N2CCOCC2)cc1)C(C)C 63113,CC1(C(=O)NC2CC2CNC(=O)Cn2ccc(-c3ccccc3)c2)CCCCO1 63114,N1(C(C2N(CCC)CCC2)=O)CCC(CNC(c2cc(C)nc(C)n2)=O)C1(C)C 63115,N1(C(CCSCCCC)=O)CCN(C(=O)CSC(F)F)CC1CCOC 63116,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63117,CC1CN(C(C2CC(F)(c3ccccc3)C2)=O)CC1n1cc(-c2cncn2C)nn1 63118,C1(C)(C(N(CCN(C(C(CCCC)O)=O)C)C(C)C)=O)CCCCCCC1 63119,c1(CN(C(C2CCN(c3nccc(C#N)n3)C2)=O)CC)ccc2ncnn2c1 63120,C(=O)(C(F)C(F)(F)F)NCCC1CC(NC(c2cc(C)n(C3CC3)n2)=O)C1 63121,CC1CC(C(=O)N(CC(C)NC(C2CN(c3nnnn3C)C2)=O)C)CCS1 63122,c1(C(N)=O)ccc(NC(=O)NCc2cnn(CCF)c2)c(F)c1 63123,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63124,N1(C(CN(CC(=O)NC)C)=O)CCN(C(=O)CCc2cncn2C)CC1C1CC1 63125,C1(CNC(C2C(C)CCCC2)=O)CC(C)CN(C(c2ccnn2CC2CC2)=O)C1 63126,N1(C(C2(CC=C)CCN(C(=O)COC3(C)CCCC3)C2)=O)CC2(CCC(=O)N2)C1 63127,N1(C(CCOCCOC)=O)CC(NC(c2cncc(F)c2)=O)CC1C 63128,CN1CCc2cc(C(=O)NCCN3CCN(C(=O)C(N)=O)CC3)ccc21 63129,C#CCCCOC.C1(=O)CN1CC.C1(=O)COCCN1C.C(C=C)O 63130,C(CN=C(NCCC1CCCCO1)N1CC2CC1CS2(=O)=O)C1(CO)CCC1 63131,N1(C(COCCC)=O)CC(C)(CNC(c2ccnc(C)n2)=O)CC1(C)C 63132,c1(C(=O)NCC(CNC(CCC(C)C#N)=O)(C)F)cc2n(n1)CCCN2 63133,C(N=c1[nH]c(Cl)ncc1Cl)C1N(C(CCCc2ccc(OC)cc2)=O)CCCC1 63134,Cc1ccc(C(C(=O)O)NC(=O)NCC2(c3ccc(O)nc3)CC2)cc1C 63135,c1(COC)nc(NCCF)cc(=NCC(c2ccc(OC(F)F)cc2)SC)[nH]1 63136,N1(C(C)=O)CCC(C2CCCN(C(C3CCCCCNC3=O)=O)C2)C1 63137,Cc1cc(=NC2CC2C2CCCCC2)[nH]c(NC2COc3ccc(C)cc32)n1 63138,N1(C(C2C(C#C)C2)=O)CCN(C(=O)C(N2CCN(CC)CC2)=O)CC1CC 63139,C1(C)(CCC(=O)N(C)CC2(NC(c3csc(CC4CC4)n3)=O)CC2)CCC(=O)N1 63140,C12(NC(C(CC)C)=O)CCC(C(=O)NCCN3CC(N(C)C)C3)(CC1)C2 63141,N1(C(C(CCC)OCC)=O)CC(C2(NC(c3cnc(Cl)c(N)c3)=O)CC2)C1 63142,O=C1NC(=O)N2CCN(C(=O)C(=O)C3(C4CCC(F)(F)C4)CCC3)CC12 63143,N1(C(CN2CC(C(N)=O)C2)=O)CCN(C(C2CC2C2CC2)=O)CC1 63144,C12(C(=O)NCC3(O)CN(C(CC4CC(=C)C4)=O)C3)CC(C(C)(C)OC)(C1)C2 63145,N1(C(C2CC(N(C)C)C2)=O)CC(NCc2cc(Br)c([N+](=O)[O-])s2)CC(F)(F)C1 63146,C1(O)(CNC(=O)CCCCc2ccc(F)cc2)CCCN(C(=O)CC2CCC2)C1 63147,C1(C2(O)CN(C(C3CCc4nnnn4C3)=O)C2)(CNC(c2cc(C)no2)=O)CC1 63148,c1(CC)[nH]nc(C(=O)NCCN(C(=O)Cn2ncccc2=O)C(C)C)c1Br 63149,C#CCCCCCC(=O)N1CC(OC)C(NC(C2(CC)CNC(=O)C2)=O)C1 63150,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63151,N1(C(CC2N(C(c3nc(CC)sc3)=O)CCC2)=O)CCCSCC1C 63152,c1(C(=O)OCC)cnn2c1CC(NC(c1ccc(F)c(F)c1C)=O)CC2 63153,C1(NC2(CC(=O)NC(C3CCCC3)C)CCC2)CCN(C(=O)C(F)(F)C2CC2)C1 63154,C12(C(=O)NC3CCN(C(C(CC)C)=O)CC3)CC3CC(CC1C3)C2 63155,C1(C(C)NC(=O)CN(C(N)=O)CC)(CNC(CCNC(C)=O)=O)CCCC1 63156,CC(CC(F)(F)F)C(=O)N(C1CN(C(C2CC(n3cnnc3)C2)=O)CCC1O)C 63157,Cc1csc(C(=O)NCC2CN(C(C)=O)CC2C)c1Br 63158,c1(-n2cc(C(=O)NC)nn2)cccc(NC(c2ccoc2)C)c1 63159,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)NCCS(=O)(=O)N(C)C)[nH]1 63160,C(C(=O)N(CC(C)C(=O)NCc1c(CC)noc1C)C)(C(C)C)OCC 63161,N1(C(c2ccc(OC)c(Cl)c2)=O)CCN(C(C2CC=CC2)=O)CC(C)(F)C1 63162,N1(C(=O)C=CCO)CCC2CCN(c3ncc(Br)c(O)n3)CC2C1 63163,c1(C(N(C(CN(C(C2(CCC=C)CCCC2)=O)C)C)C)=O)nccc(Cl)c1O 63164,c1(N(CCN(CC)CC)CC)cc(Cl)c(F)cc1S(N)(=O)=O 63165,CCCCC(CC)C(=O)NCC1CCCN(C(=O)CC2CCOC(C)(C)C2)C1 63166,N1(CC(=O)NC2CCOCC2NC(=O)COC2CC=CC2)C(=O)CCC1=O 63167,Cc1cc(C(N2CCC(F)(C(N3CCC3CN=[N+]=[N-])=O)CC2)=O)nc(O)n1 63168,c1(SCCn2nc(C)c(C(N3CCOCC3C3(C)CC3)=O)c2)ccc(F)cc1F 63169,C(=O)(CC(C)(C)C(=O)NC1CCC(NC(=O)CC2CCC(C)(C)O2)C1)OC 63170,C1(NC(c2ccco2)=O)CN(C(=O)COc2cc(Cl)ccn2)CC12CCC2 63171,CC1CC=CCC1C(N1CC(O)(C(C(N2CCN(C3CN(C)C3)CC2)=O)F)C1)=O 63172,C1(N2CCN(Cc3ccc(C)cc3)CC2)CN(C(=O)C2(c3ccccc3)CC2)NC1=O 63173,N1(C(COCCC=C)=O)CCCC2(NC(c3ccc(CO)c(C)c3)=O)CCCC12 63174,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2C)cnc2c(c1)NCC(=O)N2 63175,N1(C(CNS(N(C)C)(=O)=O)=O)CCCN(C(c2ccsc2Cl)=O)C(CO)C1 63176,C1(N(C(CCOCCN(C(C=CCC)=O)C)=O)C)CCCCN(C)C1 63177,c1(C(c2ccccc2)C2CC2C(=O)NC(C)CCN(C)CC)ncsc1Br 63178,C=CCC(CC(=O)NCC(O)CC)NC(C1(Cl)CC1)=O 63179,C1(C(=O)NCCCC(=O)N(C)C)CCC2(CC2)N1C(C1CCCN1C)=O 63180,Cn1c(C(=O)NCC2CCCCN2C(=O)CCC2CCCO2)ccc1C1CCCO1 63181,c1(C(=O)NC2(c3ccccc3)CN(C(C3CC3F)=O)C2)ccc(F)cc1 63182,C=C1CC(C)NC(=O)OC(=O)C1.C1(C(C)NC(=O)OC)CCS(=O)(=O)C1 63183,c1(C(N2C(C(=O)Nc3cc(C)c(F)nc3)CC3CC32)=O)ccc2c(c1)C(=O)CC2 63184,N12CCC(CC1)N(C)C2=O.c1(CCC)nnnn1CC(=O)Nc1csnc1Cl 63185,N1(Cc2c(C)nc(Cl)cc2)CCC2(CC1)CC2NC(c1ccc(C#N)cn1)=O 63186,N1(C(CC(C)(C)C)=O)CCN(C(=O)C=CC2CC2)C(C2CC2)C1 63187,C(=O)(C(CC(C)C)N(C(c1cnsc1C)=O)C1CC1)NCc1nc(CC)sc1 63188,CC1CCN(C(C2(c3ccccc3)CC(F)C2)=O)CCN1C(=O)C=CC(F)(F)F 63189,Cc1nccn1CCCC(=O)N.C1(C(N)=O)CCC(CCC(N2CC(O)(CO)C2)=O)C1 63190,C(=O)(CC(C)C(C)(C)C)NCN1CCC(C=C)(C(=O)NC2(CC#C)CC2)C1 63191,c1(CNC(N2CC(Cc3cccnc3)C2)=O)cccc(OC(F)(F)F)c1 63192,C1(NC(c2c(C)nn(C)n2)=O)CN(C(c2ccc(F)c(CO)c2)=O)CC1N=[N+]=[N-] 63193,c12cc(C)nc(n1)N1CCC(CC=C)(C1)NC2=O.C#CCCCC(=O)OCC 63194,CC1(C)CN(C(c2csnn2)=O)CCC1C(=O)NC1CN(C(N)=O)C(C)(C)C1 63195,C(=O)CCC(C)(C)C(=O)N1CCC(F)C(O)C1 63196,c1(C(=O)NC2CC(NC(c3ccn4c3CCCC4)=O)C2)cnn2c(=O)cc[nH]c12 63197,C1(C(=O)NC(CCNC(C(C)C2(O)CCC2)=O)(C)C)CC2CCC1O2 63198,C(=O)(C(F)CC(C)(C)N)NCC(C)(C)OCCNC(C1(COC)CC1)=O 63199,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63200,C(=O)(C(C)(O)C(C)(C)C)NCC1N(C(Cc2ccc(SC)cc2)=O)CC1 63201,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63202,c1(C(=O)NC(C)CCN(C)C(C2CC2C)=O)cc(-c2ccncc2)nn1C 63203,c1(C(=O)NCC23CC(CNC(C4(N(C)C)CCC4)=O)(C2)C3)cccc2c1OCC2 63204,Cc1cncc(CCC(=O)NC(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63205,N12CCN(C(=O)C1)CC2=O.c1(NC(C=CC(=O)N(C)C)=O)cnc(N(C)C)nc1 63206,c1(NC(=O)NC2CCN(C(C3CC4CC3CC4O)=O)CC2)c(Cl)cccc1Cl 63207,c1(OCC)ccc(C(N)=O)cc1S(=O)(=O)NCCC1CCS(=O)(=O)N1 63208,C12(OC)CCC(CN(C3CCOC3)CC3CC3)(CC1)C2 63209,c1(C(=O)NCCCCC2CCCN(C(C=C(C)Cl)=O)C2)ccc(C(F)F)nc1 63210,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCCC2)cccc2cncn12 63211,N1(C(c2n(CC)ccc2)=O)CCC(NC(C2(CCF)CCC2)=O)C(C)C1 63212,c1(NC(=O)NC(C2CCSC2)C#C)cc(C)cc([N+](=O)[O-])c1 63213,C(=O)(C(F)C(C)(F)F)NC(C(=O)N1CC(OC)C1)(C)CC1CC1 63214,c1(C(N2CCN(C3(C(=O)NC4CC(OC)C4)CC3)CC2)=O)c(Cl)cc(Cl)nc1N 63215,C(=O)(C(C)(C)CCCO)N(C)CC1CCCN1C(c1ccc(CO)cc1)=O 63216,N1(CC2N(C(c3n(CC)ncc3)C(=O)NCCOC)CCOC2)C(=O)CCC1=O 63217,c1(C(=O)NCCC(C(C)C)NC(C(CC(=O)OC)C)=O)cc2cn[nH]c2cn1 63218,O=C(C1CCCc2scnc21)NCC1CCN(C(=O)CCc2ccco2)C12CC2 63219,C1(C(C)NC(C2(NC(C)C)CC2)=O)CCCN(C(C2CC2C(C)O)=O)C1 63220,C1(N(C(=O)COCP(C)(C)=O)C)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CC2 63221,C12(C(=O)OCC)C3C4C1C1C2C3C41C(=O)N(CC(C)CNC=O)C 63222,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1C 63223,N1(C(C(CC)(C)F)=O)CCCCC(NC(c2ccsc2Br)=O)CC1 63224,Cc1c(C(N2CCCN(C(C3CCCO3)=O)CC2)=O)[nH]c2cc(F)ccc12 63225,C(=O)(CCC(=O)NC(C1CCCO1)=O)NCCN(CCC)CC 63226,C1(CNC(c2c(CC)occ2)=O)CC(C)CN(C(C2(CCO)CC2)=O)C1 63227,C1(NC(c2n(C)ccn2)=O)CN(C(C2CC2C(C)(F)F)=O)C(C)(C)C1 63228,c1(C(=O)NC2(CCNC(c3nccc(CC)c3F)=O)CC2)ccc2sncc2c1 63229,N1(C(C=C(CCC)C)=O)CCC(N(C(=O)Cc2c(C)cccc2F)C)C2(CC2)C1 63230,C1(CC(=O)NC2CC=CC2)(NC(C2CC2Cl)=O)CCCC1 63231,C1(NC(C2(CC=C)COC2)=O)CCC(NC(c2cnc(Br)s2)=O)C1 63232,c1(CC)c(C(=O)NCCNC(=O)CCCc2nc(C)no2)cccc1Br 63233,c1(C(N2C(CNC(c3c(C)coc3)=O)CC2)=O)c(C)nn(C(C)C)c1Cl 63234,Cc1nsc(CC(=O)NCC2(NC(=O)CC3CCCO3)CCOC2)n1 63235,N1(C(c2[nH]cc(C)c2)=O)CC(N)C2(CCOCC2)C1 63236,C1(NC(c2nc(C)c(C)s2)=O)CCCN(C(=O)C(N2CCCC(C)C2)=O)CC1 63237,S(=O)(=O)(c1ccc(=NCCC2CCSC2)[nH]c1)NC1CC(C)(C)SCC1 63238,Cc1cc(C(=O)NCC2COC(CNC(=O)Cc3n[nH]c(C)n3)C2)nc(O)n1 63239,CC1N(C(c2cccnc2-c2ccc(F)c(F)c2)=O)CCC1(C)C 63240,C=C(Cl)CCC(=O)NC(C1CC=CCC1)C(=O)N(CC(C)CC)C 63241,N1(C(C(N2CCCCC2=O)C)=O)CCC(F)(CNC(c2cn(CCO)nc2Cl)=O)C1 63242,c1(CNC(=O)NC(CC)CCOC)cc(Br)c(C)s1 63243,N1(C(C2(OC)CCC2)=O)CC(CNC(c2cc(OC)nc(OC)c2)=O)C(C)(C)C1 63244,c1(NC(c2ccc(C(=O)NC)cc2)=O)cccc(F)c1CO 63245,CC1CC(C)(C(=O)Nc2cccc(C(N3CC4CC3C4)=O)c2)CCO1 63246,CC(C)C(O)C(=O)NC(C)(CSC)C(=O)NCc1cnn(C)c1O 63247,Cc1conc1C(=O)NC(C)C(c1ccccc1)NC(C1CSC1)=O 63248,CC(=O)CCCCC(=O)N1CC=CC1(C)C(=O)NCC(C)CC(F)(F)F 63249,C1(C)(C(N2CCC(O)(C(C)NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)CCC2CC2C1 63250,c1(CC(=O)NCC2(C)CCN(C(C3(CO)COC3)=O)C2)ccc(S(N)(=O)=O)cc1 63251,C1(OC)CC(NC(=O)CCNC(=O)CN2CCNC2=O)C12CCC2 63252,C12(CC(=O)NCC(C)(C)CNC(=O)CC3(C)CC3(F)F)CCC(CC1)C2(C)C 63253,CC1CCC(O)CN1C(c1nc(Br)n(C)n1)C(=O)NCc1cccc(Cl)c1 63254,N1(C(C(CCN(C)C)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63255,c1(-c2nc(NC(C3C(NC(C=C)=O)CCC3)=O)sc2)cnc(-c2nc(C)no2)nc1 63256,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63257,c1(CC(=O)N(CCOC)Cc2nc(C3CCCCC3)no2)cccc(F)c1 63258,N1(C(C(C)OC2CCOC2)=O)CCC2(CCN(C(C3CCC(O)CC3)=O)CC2)C1 63259,C(C(C)(C)CC(=O)N1CCC(C)C(C)C1)NC(COCCCOC)=O 63260,N1(CC2N(C)CCCC2)CCC(NC(=O)Cc2ccc(Br)cc2F)C(C)(C)C1 63261,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CC)CC12CCC2 63262,CN1CCN(C(=O)NC2CN(c3ncnc4cc[nH]c34)CCO2)CCC1=O 63263,C1(=CC(=O)NC2(CNC(C(C=C)O)=O)CC2)CCC(C)CC1 63264,C(CCCCCC(=O)OC(F)(F)F)N(C(C)(C)C)C.c12ccccc1NC1CC21 63265,N1(C(C)C)CCCC(C(=O)NCC2CN(C(=O)COC(F)F)CC2C(F)(F)F)C1 63266,Cc1noc2c1C(c1nnnn1C(C)C)NCCCCC2.c1(C)ccc(F)nc1 63267,c1(OC)ccc(I)c(C(=O)NC2CC2C(=O)Nc2ncc(Cl)cc2F)c1 63268,c1(CC)ccc(Cl)c(C(N2CCC(CNC(C3(OC)CCCC3)=O)C(C)C2)=O)c1 63269,C1(CNC(CCCC#CC)=O)CC2CCCC(C1)N2C(c1ncn(C)n1)=O 63270,N1(C(C(C(CC)O)C)=O)C(CNC(=O)CC(C)(C)C)CC2CCCCC12 63271,C1(CNC(c2occ(C)c2C)=O)CN(C(=O)COC2CCCOC2)CCC1(F)F 63272,Cc1cc(C(=O)NCC2CCCN(C(=O)C=CCCc3ccccc3)C2)n(C)n1 63273,N1(C(C2(C)C(C)(C)C2)=O)CC2CC(CNC(C3CC4(CC4)CO3)=O)C2C1 63274,C1(C(C(N2CC(O)(CC=C)C2)=O)F)CCC(NC(=O)CC(C)c2ccco2)CC1 63275,Cc1nc(=N)[nH]c(=NCCCCNC(=O)CSC(C)C)[nH]1 63276,c1(C(C)OC)nc(NC2CCCCC2NC(=O)C(C)NC(C)(C)C)cc(Cl)n1 63277,c1(C(=O)NC(CNC(C(n2ccc(C3CC3)n2)C)=O)C)cc(C(N)=O)ccc1F 63278,N1(C(c2cn(CCC=C)nn2)=O)CC(C2CCCN(C(C3CCCCO3)=O)C2)C1 63279,c1(C(=O)NCC2N(C(c3cnc(OC)nc3)=O)CC(O)C2)cnc2[nH]nnc2c1 63280,C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)NC1CC2COCC(C1)C2)C1(C)CC1 63281,CCCCCC(O)CNC(C1(CC=C)CCCN1C(=O)C(O)CC)=O 63282,c1(CC)cnc(C(N2CCCC2(C)C(=O)NC(C)CCC2CC2)=O)nc1 63283,c1(C(N2CC(C)(CNC(CC=C(C)C)=O)C(C)C2)=O)cccc2nccn12 63284,C1(CNC(c2cncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC12CCOC2 63285,CCC(CCOC)C(=O)NCC(CNC(=O)Cn1ccnc1C)OC 63286,c1(C(C2CC2)OC)nc(CC(F)C(F)(F)F)n(-c2ccc(Cl)cc2)n1 63287,C(=O)(C(F)(F)C(C)O)NCCC1(OC)CN(C(=O)C(C2CCOCC2)C)C1 63288,c1(OCC(=O)N(C2CCN(C(=O)OCC(C)(C)C)CC2)CCC)ccc(F)c(C)c1 63289,c1(SCCC2CNS(=O)(=O)C2)cccc2c1OCO2 63290,CCCC(CNC(C1CCCSC1)=O)NC(c1cnc(C(F)F)s1)=O 63291,C(=O)(C(C)C(C)(C)C)N1CC(NC(CSc2n(CC)ccn2)=O)C1 63292,Cc1ncc(C(=O)NCCCN(C(=O)CCC(C)(C)C)CC2CC2)c(C(C)C)n1 63293,c1(C(c2n(CCCOC)nnn2)NC2(CC(N)=O)CC2)ccc(C(C)(C)C)cc1 63294,C1(NC(CCC(C)NC(c2c(C)scc2)=O)=O)C2C3CCC(C3)C12 63295,S(=O)(=O)(c1cccc(N2CCCN(C)CC2)n1)NC1CC(OC)(OC)C1 63296,C1(NC(=O)Cc2ccsc2)CC(F)(F)CC1NC(C1(O)CCC1)=O 63297,CC(C)C(CN(C)C)C(=O)N1CCC1CN(C1CCC1)C(C1CCN1)=O 63298,C1(n2cc(-c3cccc(CN(C)S(N)(=O)=O)c3)nn2)CC2CCC(C1)C2F 63299,C1(C(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)CC2COCC(C1)C2 63300,c1(C(N2CCCC(n3cc(CNC(C(C)C)=O)nn3)C2)=O)ncc(Br)cc1Br 63301,C(=O)(C1=CCC(NC(=O)C(CC=C)OC)C1)N(CC#C)CCF 63302,N1(C(CCC#C)=O)CCC2(CC1)C(N(C)C(c1cn(CCOC)nn1)=O)CS2(=O)=O 63303,C(=O)(CCC(C)(C)OC)NC1C(NC(C(C(C)C)Oc2ccccc2)=O)CC1 63304,C1(COC)(NC(=O)CC2CCC(C)(C)C2)CCN(C(c2cscn2)=O)C1 63305,C1(C)(CNC(C(C)Cc2cnn(C)c2)=O)CCCN(C(=O)C(C)(Cl)Cl)C1 63306,C(c1cccc(F)c1)=CC(=O)N(CC(C)O)CCNC(CN(C)CC)=O 63307,Cc1cc(=O)c2cc(NC(=O)NC3CCN(c4ccc(F)cc4F)C3)ccc2[nH]1 63308,CC1(C#CC(=O)N2CC3CN(C(c4cncc(Cl)c4)=O)CCC23)CCCO1 63309,C1(C)(C(N(CC(C)(C)NC(C(Cn2ccc(C)n2)C)=O)C)=O)CCC(C)(C)CC1 63310,C1(CC)CCN(C(=O)CC(C)n2ccnc2)C1CNC(C1C2CCCCC12)=O 63311,C1(CCN(c2ccc(Br)cc2)CC(C)C)CS(=O)(=O)CC1O.c12csc(n1)NC2=O 63312,C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 63313,O=C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)Sc1cc2cccc(Cl)c2o1 63314,Cc1cc(N)c(C(=O)NCC2CC2CNC(=O)C(C)CC2CCCC2)c(F)c1 63315,C1(OCC)CC(NC(=O)C=CC(F)(F)F)C12CCC2 63316,N1(C(C(c2ccccc2)C)=O)CC2(CCCCN2C(c2cnc(S)n2C)=O)C1 63317,C(CC(C)C(=O)NC1(CNC(CCc2ccc(SC)o2)=O)CC1)=CC 63318,c1(CC(N2CCC(C(C)(C)NC(CC(=C)Br)=O)C2)=O)nc2ncccn2n1 63319,C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C)CCC2C(C)C)=O)C12CC2 63320,C1(NC(CN(c2ncccn2)C)=O)CC2CCC1N2C(C1CCN(C2CC2)C1=O)=O 63321,C(=O)(CC(C)C(=O)NCC(C)NC(c1coc(Br)c1)=O)OCC 63322,CC1(C)CN(C(=O)C(C2CC2)NC(=O)C(C2CCCCC2)F)CCC1O 63323,C(C(CC)(CC)C(N)=O)NC(CN(CC#C)C(c1cccnc1S)=O)=O 63324,C1(NC(C2CCCCC2)=O)CC2CCC1N(C(c1ccn(C3CC3)n1)=O)C2 63325,C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(CCSCCC)=O)C1 63326,N#Cc1ccc(F)cc1NC(c1c[nH]c(C(N2CCCCC2)=O)c1)=O 63327,c1(C(=O)OC)cc(NC(c2csc(NC(c3cnc(C)nc3)=O)n2)=O)ccc1O 63328,CONC(=O)C(C)CNC(C1CC1C(F)F)=O 63329,C1(C(C)CNSC(F)(F)F)CCCCN1C(=O)C(C)CSC(F)(F)F 63330,C1(NC(c2scnc2C2CC2)=O)CN(C(=O)CC2OCCCO2)Cc2nccn2C1 63331,C(=O)(C(C)CNC(=O)C(CC1CCOCC1)NC(=O)C(C)C#N)NC 63332,CC1C(NC(C2CC(F)(F)C2)=O)CCN1C(=O)CC(=O)N(C)C 63333,C1(C(=O)NCC2CCCCC2CN)CCN(CC2(S(C)(=O)=O)CC2)CC1F 63334,c1(OC)nc(N(CC(C)CNC(c2ccc3cncn3c2)=O)C)c(Cl)cc1C 63335,CC1(C)CCc2c1n[nH]c2C(=O)NCC1CN(C(=O)CCn2ccnc2)CCO1 63336,C1(NC(C(C)C)=O)CCN(C(c2ccc(C(=O)NC3CC3)o2)=O)CC1 63337,C1(N(C(CS(=O)(=O)NC)=O)C)CCCCN(C(c2nnc(S)n2C)=O)C1 63338,CCC(CCCC(=O)NC(C)CC1CCOC1)NC(=O)CCc1ncnn1C 63339,C(CCCCCOC)NC(C1(CC)CN(C(c2cc(CC)no2)=O)C1)=O 63340,c1(C(=O)OC)cc(C)sc1NC(C1CN(C(=O)C(C)Cc2c(C)noc2C)C1)=O 63341,C1(NC(C2CC23CCC3)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C12CCC2 63342,N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(CO)C1 63343,N1(C(CCN(C(C2(CC(C)C)CCOC2)=O)CCO)=O)CC2(CNC(=O)N2C)C1 63344,CC(CC(=O)NCC(C1CC1)NC(c1cnn(C)c1Cl)=O)C(F)F 63345,CCCCC(CNC(c1cncc(F)c1)=O)NC(=O)Cn1ccnn1 63346,CC(CS(C)(=O)=O)C(=O)N1CCC(C)C(NC(=O)C(c2ccccc2Cl)C)C1 63347,C(=O)(CCC(CC)CC)NC(CC(C)NC(COCCCC)=O)C 63348,c1(CCC(=O)NC2(CNC(C3=CC(C)CC3)=O)CC2)ccc2ncccc2c1 63349,N#CC1CN(C(=O)C=CCC2(NC(c3cnncc3O)=O)CCC2)CC12CCC2 63350,C(=O)(CC(C)CCC=C(C)C)NCC1C=CC(NC(c2ccc(OC)s2)=O)C1 63351,c1(N(C)C)ccc(F)cc1C(=O)NC1CC(CNC(c2cnn(C3CC3)c2)=O)C1 63352,C1(C(N(CCO)CC)=O)CC(O)CCN1C(=O)C1=NOC(C)C1 63353,CC1(C)CN(C(c2cc[nH]n2)=O)CC1NC(c1cccc(Cl)n1)=O 63354,CCCS(=O)(=O)CC(=O)NCCC(O)CNC(c1cc(OC)cs1)=O 63355,c1(C(c2nc(-c3ccncc3)nn2C2CCC2)OCC)cccc(OC)c1 63356,N1(C(C(C)NC(CC)=O)=O)CCC(NC(c2ccc(C)cc2F)=O)C12CC2 63357,N1(C(CC(C(C)C)C)=O)CCCCC(C2CN(C(C3(C(F)(F)F)CC3)=O)C2)C1 63358,c1(C(N2CC(C)N(C(c3ccno3)=O)CC2)=O)cc2c(F)ccc(Cl)c2[nH]1 63359,c1(CN(C2(OC)C(OCC)COC2)CCO)cc(C)c(C)cc1C 63360,CC(C(=O)NC1(CC(=O)NCCC2CC2C)CC1)C1CCC1 63361,C(C(C)(O)C(=O)N1CCC(F)(C(=O)NCC2=CCCOC2)C1)OC 63362,c1(CC(N2CCC(C(C)NC(c3c(C)n[nH]c3)=O)C2)=O)ccn2cncc2c1 63363,c1(C(=O)NC(C)C(CO)NC(c2cccc3sncc23)=O)cccc([N+](=O)[O-])c1 63364,c1(N(CCOCCCC)C)ncnc(N2CCOC(C)(CSC)C2)c1C 63365,c1(CN2CCC(CC(=O)NC(C3COCCO3)C)CC2)c(F)cccc1Cl 63366,c1(C(=O)NCC2CN(C(C(C)O)=O)C(C)(C)C2)cccc2c1OCCCO2 63367,O=C(C#CC1CCCO1)NC1CCCC1CNC(c1cc(O)nc(C2CC2)n1)=O 63368,c1(C(=O)OC)cc(NCC2CCN(C(=O)C(C)(C)CF)C2)cc(C(F)(F)F)n1 63369,C1(CC(=O)NCC(C)NC(CN(C(CCOCC)=O)C)=O)CCN(C)CC1 63370,N1(C(Cc2nc(COC)sc2)=O)CC(C)C(NC(=O)CN2CCOCC2)C1C 63371,C(=O)(C(CCC(N)=O)OC)N1C(Cn2cc(-c3ccc(CC)nc3F)nn2)CCC1 63372,CC(C)(C)CCCC(=O)NC1CCC1NC(C1(CC#N)CCCCC1)=O 63373,c1(CC)coc(C(C(=O)NCCCOCCOC)N(CCCN(C)C)C)n1 63374,CCCCC(O)C(=O)NC1CCCC1NC(=O)CC1(O)CCCN(C)C1 63375,N1(C(CC2(OC)CC2)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)CC(F)C1 63376,C(=O)(C(=O)N=S(C)(C)=O)N1CCCC(N(C(CCCCCC)=O)C)CC1 63377,N1(C(C(CC)CC)=O)CC(CNC(c2ccnc(C)c2C)=O)OC2(CCC2)C1 63378,N(C1c2ccccc2OCC1CNC(C)=O)C(Cc1cc(OC)c(O)c(Br)c1)=O 63379,CCC(C(=O)N1CC2CCC(CNC(C3CCCC34CCC4)=O)(C2)C1)C(F)(F)F 63380,C1(CCNC(c2c(COC)cccn2)=O)CC2CCC(C1)N2C(=O)CCSC 63381,n1(CC)cncc1C(=O)N(CCNC(C1(CCSC)CCC1)=O)C1CC1 63382,c1(C(N(CCN(C)C)C)=O)csc(=NC(CCO)C2CC2)[nH]1 63383,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63384,CCCCC(O)C(=O)N1CCN(C(c2ccc(F)c(O)c2)=O)C(CCC)C1 63385,c1(OC)ncc(C(N2CC3CC2(CNC(=O)C(C)c2ccco2)C3)=O)cc1C 63386,Cc1ccc2c(=NCCC3CC=CC3)[nH]c(=NC(C)c3ccccc3)[nH]c2c1 63387,C1(OC)CN(C(=O)CCN2CCCCC2)CCC1NC(c1csc(O)n1)=O 63388,c1(CNC(C=CSC)=O)ccccc1CNC(c1coc(O)n1)=O 63389,Cc1cc(C(N2CCN(C(c3cnc(O)c(Br)c3)=O)C(C)C2)=O)nnc1Br 63390,c1(C(C(=O)NCCN(C(=O)CCN2CCCCC2=O)CC)C)nnc(S)nc1C 63391,N1(C(C(C=C)(F)F)=O)CC(C(=O)Nc2ccc(C)cc2F)C2(CC2)C1 63392,N1(C(c2n(C)cnc2)=O)CCCC(C2CN(C(=O)CCCC3CCCO3)C2)C1 63393,CC(C)(O)C(F)C(=O)NCC1CC(F)(F)CN1C(=O)CCCn1ccnc1 63394,c1(C(N2C(CNC(C34OCCC(C)(C3)C4)=O)CCC2)=O)cccc2c1COCC2 63395,c1(C(C)COC2CC2)nc(-c2cccc(N)n2)nn1C1CCCCC1O 63396,N1(C(c2ccc(COC)[nH]2)=O)CCC2(COC(CNC(=O)Cc3nc[nH]n3)C2)C1 63397,C1(NC(C2N(C(C)=O)CCC2)=O)CCC(CNC(c2cnnn2C)=O)CC1 63398,C1(CCC)(NC(=O)CCn2nc(C)cc2C)CCCN(C(=O)C(C2CC2)OC)C1 63399,c1(C(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2)cccn2ccnc12 63400,c1(N2CCC(CNC(C3CCCC(F)(F)C3)=O)C2)cnc(Cl)cc1[N+](=O)[O-] 63401,C(CNC(c1n[nH]c(C)c1F)=O)(CC(F)(F)F)NC(COCCCCC)=O 63402,c1(C(N(CCC(=O)N2CCC2)C)=O)ccc(S(=O)(=O)N2CCCCC2)cc1.CN 63403,c1(C(=O)NC(c2nnnn2C2CC2)C)csc(C(c2ccccc2)N)n1 63404,Cc1cc(C)n(NC(=O)C2CCN(S(=O)(=O)c3cnn(C)c3F)C2)c(=O)n1 63405,CCC(F)(F)C(=O)N1CC(O)(CNC(=O)C=Cc2csc(C(F)(F)F)c2)C1 63406,C(=O)(CCCCCC#N)N.C(=O)(CNC(=O)C=C)NCCCC 63407,C1(F)(C(=O)NC2CC(C)N(C(C3CN(C)C3)=O)CC2)CCC(F)(F)CC1 63408,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63409,Cc1cccc(OCC(N2CCC(CO)(NC(=O)CC(C)(F)F)CC2)=O)c1F 63410,N1(C(C(C)SCC)=O)CCCC2CN(C(c3ccc(CC(C)C)s3)=O)CC12 63411,Cc1ccc(C(=O)NC(c2n[nH]cc2C(N2CC3CC3C2)=O)C2CC2)cc1 63412,c1(C(N2CCC(n3cc(-c4ncc(Br)cn4)nn3)C2)=O)cccc2oc(O)nc12 63413,c1(C(C)C)ccc(NC(=O)C(c2ccn(C)n2)NC(=O)C=Cc2ccoc2)cn1 63414,c1(NC(CC2(C(=O)OCC)CCC2)=O)ccccc1NC(=O)C(C1CCC1)OC 63415,c1(C(C(=O)N(CCCNC(C2CCCCC2)=O)CC)OC(C)C)cccc(Cl)c1 63416,C1(CC)OCCC1NC(=O)CCCNC(=O)CNC=O 63417,C1(CC(N(C)OC2CCCC2)=O)CN(C(C2CC2c2ccccc2)=O)CC12CC2 63418,C(CC(C)C(=O)NC12CC(C(=O)N(C(CC)CC)C)(C1)C2)=CCC 63419,CCCCCC(F)C(=O)N1CC=C(C(=O)N2CCCC(CCOC)CC2)CC1 63420,C1(N(C(C)C(=O)NC2CC2)C(=O)CC2(O)CCOCC2)CCOC(CO)C1 63421,c1(CNC(C(c2ccc(F)c(Cl)c2)N)=O)cc(C(F)(F)F)ccc1Cl 63422,C1(NC(C2(C)CCN2Cc2cc(C#N)ccn2)=O)CCC2(CC1)OCCO2 63423,C12(NC(C3C(C#C)C3)=O)CCC(CC1)N(C(=O)CN1CCCNC1=O)C2 63424,Cc1nn(C)cc1S(=O)(=O)N1CC2CN(C(c3ccnc(Cl)n3)=O)C2C1 63425,C1(C(N(C2CCCN(C(=O)Cc3cscn3)C2)C)=O)CCCCCCC1 63426,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3Cl)=O)C2)=O)CC1 63427,CC1CCC(O)(C(N2CCN(C(C)C(=O)N3CC=CC3)CC2)=O)CC1 63428,C(C)(C(=O)N(C)Cc1cccnc1)(C1CCOCC1)OC 63429,Cc1cccnc1CCC(N1CCCC(C(C)NC(=O)C=CC=C(C)C)C1)=O 63430,Cc1nc(N2CCCC2CN(C)C)c(C)c(C)n1.C12CN(CC1C(N)=O)C2=O 63431,c1(C(=O)NC(CNC(C(=O)NC(C)C)=O)C(C)C)cc(Cl)cc(Cl)c1Cl 63432,Cc1cnc(C)c(NC(C2(F)CC=CCC2)=O)c1 63433,C1(C(=O)NCCCC(=C)C)CC2CCC1N2C(=O)C=C=C(C)C 63434,N1(C(c2c(N)non2)=O)CC2CCCC(CNC(C3CCC(=O)NC3)=O)C2C1 63435,CCCCCCC(C)C(=O)NCC(C)N(C)C(c1c(C)cnnc1O)=O 63436,c1(C(=O)NC(CN(C)C(c2ccccc2)=O)(C)C)ccc(Br)cc1 63437,Cc1scc(CC(=O)NC2CN(C(c3cc(O)ncn3)=O)CC2CO)c1C 63438,CC(C)C(C(=O)NC1(C)CC2(CCC2)C1)C(C)NC(c1cc(C#N)ccc1N)=O 63439,N1(C(C(COC2CC2)NC(C)=O)=O)CC(NC(=O)C=CCF)C(O)C1 63440,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N(CCN(C(C1C(C)C1C)=O)CC)CC 63441,c1(OCC)cccc(CC(=O)NCCNC(c2ccnc(OCCO)c2)=O)c1 63442,N1(C(CSCCC)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2(C)C)C1 63443,c1(OCC#C)cc(Cl)ccc1CN1CCC1 63444,Cc1nccnc1C(N1CCC(CC(=O)N(C(C)C)CC2CCC2)C1)=O 63445,C1(CC(NOCCCN(C)C)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)C1(C)C 63446,C1(C(C(=O)N(CCCN(C)C)C)NC(=O)CCn2cccc2)CC=CCC1 63447,c1(C(=O)Nc2c(C)cc(NC(C3OCCO3)=O)cc2)cnc2c(N)cccc2c1 63448,C1(C(N2CC(CCC)C(NC(c3cc[nH]n3)=O)C2)=O)CSc2ccccc2O1 63449,N1(Cc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63450,Cc1ccsc1CC(=O)NCC1CC(NC(c2nocc2CC(N)=O)=O)C1 63451,C1(C(NOCCC(C)C)=O)CCC(O)CN1C(C1(C)CCCCC1)=O 63452,N1(C(c2n(CC)ncc2)=O)CC(C(=O)N(CC(C)OC)CC)CC12CCC2 63453,C1(CC(C)C)(C(=O)N(CCCCN(C(=O)Cc2cccn2C)C)C)CCCCC1 63454,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63455,O=C(C1=CC2(CCOC2)C1)NC1CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CC12CCC2 63456,C(=O)(CC1CCOc2ccccc21)N1CC(CNC(C(C)CF)=O)C(C)C1 63457,C1(C(=O)NCC2CCCN(C(=O)CCC3CCC3)C2)(OC)CS(=O)(=O)C1 63458,C(c1ccc(F)c(F)c1)=CC(N1CC(C)C(NC(=O)CN2CCCNC2=O)C1)=O 63459,C(CCCCC(=O)N1CCC12CN(C(c1cc(Cl)c(Cl)n1C)=O)C2)N(C)C 63460,CC1CC(C(=O)NCCC2CCN(C(=O)CN3CCCNC3=O)C2)CCS1 63461,CN1CC(C(N2CCCCC2c2cn(C3CCOCC3)nn2)=O)Cc2ccccc21 63462,CCC(C(=O)N1CC(C(C)NC(C2CCCO2)=O)C1)C(C)(C)CC 63463,c1(NCCSCC=C)cc(=NCC(CC#N)c2ccccc2)[nH]c(CC(C)C)n1 63464,c1(OC)cc(CN2CC(NC(c3ccc(C(F)(F)F)nc3Br)=O)C2)ccc1O 63465,C12=CC=C(C=C1)C2NC(C)C1CC1.c1(CCOC(C)C)nnnn1C 63466,S(=O)(=O)(C1CCN(C(=N)N2CC(O)C2)CC1)NC.c12ccccc1CC=CC2 63467,N1(C(c2c(OC)ccs2)=O)CCC2CCCC12C(N1CCCC1(CO)CO)=O 63468,C1(CC)CN(C(c2c(Cl)cccc2Cl)=O)CCN1Cc1cccc(Cl)n1 63469,C(=O)(CCCCC(N)=O)N1CC(CC(C)NC(=O)Cc2ccnc(Cl)c2F)C1 63470,c1(SC)ncccc1S(C)(=O)=NC(=O)C1CCc2ccccc2C(C)C1 63471,C12(C)CC13CCN(CC3)c1cccc(n1)CNC2=O.c1(CC)ocnc1C1CC1 63472,Cc1c(C(N2CCC(F)(CNC(=O)C(O)Cn3cncn3)C2)=O)ccc2n[nH]cc12 63473,c1(C(=O)OCC)ccc(NC(C23CC(CC(C)C)(CO2)C3)=O)nc1Cl 63474,CC1CN(C=O)CC(C)N(C(C2CC(=O)N2)=O)C1.c1(N)nn(C)c2c1CCC2 63475,C=CC(CC(=O)NC(C)CCCCNC(=O)CCNC(=O)CO)c1ccccc1 63476,c1(C(=O)NC(C2CN(C(C=CCC)=O)C2)C)cc(=O)c2c(Br)cccc2o1 63477,C1(N(C(=O)COCc2nnc(O)s2)C)CCN(C(=O)Cc2ccn(C)n2)CC1 63478,N1(C(C2C(C(=O)OC)C2)=O)CC(CNc2nc(C#N)c(Cl)s2)C2(CCC2)C1 63479,C=CCCC(CC(C)C)C(=O)N(CCNC(=O)C(C(C)C)NC(=O)OC)CC 63480,C1(C(CNC(CN(CCCC)C)=O)C)CCN(C(C)=O)CC1.C1(=O)C(F)N1 63481,C1(NC(c2cnn3c2OCC3)=O)CC2CCC(C1)N2C(=O)CC1(O)CCC1 63482,Cc1n[nH]c(C)c1C(C)NC(=O)C(C1CCCC1)NC(c1cc(C(N)=O)[nH]n1)=O 63483,C1(CC)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(=O)C(C)n1ccnc1 63484,C(=O)(C1=C(Cl)CCC1)N1C(C)CC1.C1(CC(=O)NCC)COCC(C)(C)O1 63485,c1(CNCCC(CC)C)cc(=NCC(Cc2ccccc2F)CO)[nH]c(C)n1 63486,CC1CC(C)CN(C(=O)COC(=O)CCC2OCCO2)C1 63487,C1(C(=O)OC)CCCC2(CCN(C(=O)CC3CCC4CNCC34)CC2)O1 63488,n1(CC(=O)NC2C(C)CN(C(=O)CSc3ccccn3)C2)ccc([N+](=O)[O-])n1 63489,Cc1ccc(C(=O)N(CCC(C)NC(c2cnn(CC(=O)O)c2)=O)C)cc1F 63490,CN1CCC2(CCN(C(=O)C(C(C)(C)O)NC(C3COCCO3)=O)C2)C1 63491,N1(c2ccc(C3CCC(=O)NC3=O)cc2)Cc2ccccc2CC1CCO 63492,Cc1cnc(C(=O)NC2CCN(Cc3cc(Cl)ccc3Cl)CC2C)c(C)c1 63493,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(C#N)CCCCCC1)=O)C2 63494,C1(N(CCNC(C(C)N(C)C(C2C=CCC2)=O)=O)C)CCOC1(C)C 63495,c1(N(C)CC2N(C(CC(CCCC)CC)=O)CCC2)nc2cc(F)c(F)cc2s1 63496,N1(C(c2ccn(CCC)n2)=O)CC2(CCC2)CC1CNC(c1cc(C)c(C)[nH]1)=O 63497,c12ccc(F)cc1O2.C1(C(=O)OC(C)C)COCC1C(F)(F)F 63498,c1(C(N(C)CC2(NC(=O)CSC3CCCO3)CC2)=O)cnn2ccncc12 63499,CCC(C)(C)C(=O)N1CCC(N(C(=O)C(C)(C)N2CCCCC2)C)CC1 63500,N1(C(CC2(OC)CC2)=O)CC(CNC(=O)CSC2CC2)C2(CC2)C1 63501,c1(C(=O)NCCC2CCCN(C(=O)CC3CSC3)C2)ccc2cnoc2c1 63502,N1(C(CC2(C(C)C)CCC2)=O)CC2CC1(CNC(=O)CNC(c1cncnc1)=O)C2 63503,c1(NC(CC2CCN(C(c3n(C)ncn3)=O)C2)=O)ncc(Br)cc1Br 63504,c1(C(N2CC(NC(C3CCCC4CC34)=O)C2)=O)ccc2c(c1)OCCO2 63505,C1(C(=O)OCC)CCN(C(c2ccc(-c3ccc(F)c(C#N)c3)o2)=O)C12COC2 63506,C(=O)(CCNC(=O)CCC1(C)CC1)N(CC(=O)NCCOC)CC=C 63507,C=Cc1ccc(C(N2CCC(C(CC)NC(=O)Cc3cc[nH]c3)CC2)=O)cc1 63508,c1(CC(=O)NC2(CCO)CN(C(C3(n4cccn4)CCC3)=O)C2)ccc(Cl)cc1 63509,N1(C(=O)Cn2cc(NC(=O)CN3CCCC3)cn2)CC2CCC(O)C(O)C12 63510,C1(C)(CNC(CCOC(C)C)=O)CCCN1C(=O)CCc1cn(C)nn1 63511,c1(C(=O)NCC2N(C(c3c(OC)c[nH]n3)=O)CC2)[nH]c(-c2cccc(C)c2)nc1C 63512,C(c1ccc(F)c(F)c1)=CC(N1C2CN(C(c3ccc(OC)nc3)=O)C(C2)C1)=O.CO 63513,N1(C(C2CN(C(N)=O)C2)=O)CC2CCCC2C1C(N1CCC(n2cnnn2)C1)=O 63514,N1(C(c2c(C)ccc(Cl)c2)=O)CCC2(CC1)OCCC2NC(C1CC(C)C1)=O 63515,S(=O)(=O)(c1cc(F)ccc1C)NC1CN(Cc2cccc(NC(C)=O)n2)CC12CC2 63516,N1(C(C(C)S(N)(=O)=O)=O)Cc2ccccc2C1CNC(C1CC2(C1)CC21CC1)=O 63517,c1(OC)cccc2c(C(N3CC(NC(c4cccnc4F)=O)C3)=O)coc12 63518,C1(C(N2CC(C(C(=O)N(c3ccc(F)cc3)C)O)C2)=O)C2CCC(C2)C1C 63519,c1(C(CO)CNCC2CCOCC2)ccc2c(c1)OCCO2 63520,C1(C)(CNC(C2(OCC)CCC2)=O)CCCN(C(c2cc(C(N)=O)ccn2)=O)C1 63521,c1(C(N2CC(N(C)C)C(F)C2)=O)cnc2n1CCN(C(c1ccc(O)cc1Cl)=O)C2 63522,c1(OC(C(=O)NCC(C)N(C(c2c(CC)nco2)=O)CC)C)ccc(F)c(F)c1 63523,C1(NC(CCCCCC#C)=O)CC2(CCCCN2C(=O)C(F)CCC)C1 63524,C1(C(=O)NCCC2(O)CN(C(CCSC)=O)C2)CC2CC(C1)CC(F)(F)C2 63525,C1(C(=O)NCCC2CCN(C(CNC(c3n(C)ncc3)=O)=O)C2)CC2(C1)CC2F 63526,N1(C(C(CC)OCC)=O)CCC2(CC(C(=O)NCCC(C)C)=NO2)C1 63527,CN1CCC(C(N2CC(n3cnnn3)C2)=O)(NC(C2CC=CCO2)=O)C1 63528,CCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)C(n1cc(C)cn1)C 63529,c1(C(=O)NC2CN(C(CSCC(C)=O)=O)C2)ccc(-c2ccccc2)[nH]1 63530,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCC2)CC1CNC(C1C=CC=CC=C1)=O 63531,c1(C(=O)NC2CN(C(c3nnn(CC)c3C)=O)CC2O)cc2n(n1)CC(F)C2 63532,n1(CCC(=O)NC2CN(C(c3c(C)nns3)=O)CC2F)cnc([N+](=O)[O-])c1 63533,C=C1CCC(C(=O)N(C)CCOCCCNC(C23CCC2C3)=O)CC1 63534,c1(C(C(=O)NCCOC)NC)cnc(C(C)(C)C)[nH]1.c1(CC(=O)OC)ccccn1 63535,CCCCC1CO1.C(C)(CC(C)C)NC(=O)CCCN(C(N)=O)C 63536,c1(C(N2CCC(N(C(C(CC)O)=O)C)C3(C2)CC3)=O)cc2cccnc2cc1F 63537,N1(C(CCNS(C)(=O)=O)=O)CCCC12CN(Cc1ccco1)C2 63538,c1(C(=O)NC2CC(C)N(C(=O)CCCCC#N)CC2)ccc2c(c1)CCC=C2 63539,Cc1ncc(C(N2CCN(C3CCN(C(c4ncoc4C)=O)C3)CC2)=O)c(=O)[nH]1 63540,c1(C(=O)NCC(C)(C)NC(=O)C2=COCC2)c[nH]nc1S(N)(=O)=O 63541,N1(C(Cc2c(C)occ2)=O)CCC2CN(C(=O)CSc3cccs3)C2C1 63542,c1(CNC(C2N(C(Cc3nc(C)sc3C)=O)CCCC2)=O)cc(C)ccc1O 63543,CC1(C)CN(C(=O)Cc2ccccc2O)C(CNC(=O)CCc2ncc[nH]2)CO1 63544,c1(C(N(CC(C)CNC(C2CS(=O)(=O)C2)=O)C)=O)noc2c1CC(C)(C)CC2 63545,N1(CC(C(N2CCC(C)(CC)C2)=O)NC(=O)OCC)CCS(=O)(=O)CC1 63546,c1(C(N2CC(CNC(c3ccncc3O)=O)C3C2C3)=O)ccc2snnc2c1 63547,C1(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2)C2CC2)CCC2(CCOCC2)C1 63548,C12(C(C)C)CC(CO1)N(C(c1cc(Cl)nn1C)C(=O)NC1CC1)C2 63549,C(=O)(CC(C)C)NCC1(CC(=O)N(C(CCC)C)CC)CC1 63550,c1(C(=O)NC(C(C)(C)NC(C(CC)C#N)=O)C)ccc(Br)c(OC)c1 63551,N1(C(C2C(C(N)=O)COC2)=O)CC2CCCC2(NC(=O)CCOCC(F)F)C1 63552,c1(C(C)N(CCO)C=O)ccccc1Cl.c1(C(CCCC(=O)N)O)ccccc1 63553,C=CC1(CS(=O)(=O)NCC2CCCN2C2CCC(C)(C)CC2)CCCCC1 63554,C1(C(N2CCC(C(=O)NC(C(C)C)(C)CO)C2C)=O)CC2C(C1)C2(F)F 63555,C1(NC(c2cccnn2)=O)CCCCN(C(C2C3CC4C(C3=O)C24)=O)C1 63556,C1(C(=O)OC)C=CCC(C(=O)NCC(O)CNC(=O)COc2cccnc2)C1 63557,Cc1cn2cc(CC(=O)NCC3CC3NC(c3cnn4c3N(C)CC4)=O)nc2s1 63558,c1(C(N2CCN(C(C3(O)C(C)(C)C3)=O)CC2)=O)ccnc2[nH]ncc12 63559,c1(C(N2CCN(C(C(CC(C)=O)C)=O)C(CO)C2)=O)cc2n(c1)CCSC2 63560,N1(C(CNC(=O)NC2C(=O)NCC2)=O)CCC(CF)(NC(C2CCCOC2)=O)C1 63561,C(=O)(CC(CC)CC)N1CC(C(=O)NCC2CN(C(C(CC#C)C)=O)C2)OCC1 63562,C(=O)(CC(C)CC(C)(C)C)N1CC(C2N(C(c3sc(C)c(O)n3)=O)CCC2)(O)C1 63563,c1(NC(CC2(CNCC(=O)NCC)CCOC2)=O)cc(C(C)(C)C)nc(SC)n1 63564,N1(C(CCS(CC)=O)=O)CCC(C)N(C(=O)CN2CCCCC2=O)CC1 63565,C1(NC(C2C(c3nc(C)sc3)C2)=O)CCC(N(C(=O)Cn2cnnn2)CCO)CC1 63566,C1(NC(COCC=C)=O)CN(C(C2CCCC(O)C2)=O)CC2(CCC2)C1 63567,c1(C(=O)O)ccc(C)c(O)c1.N1(C(C)(C)OC)CC(C(N2CCCC2C)=O)CC1=O 63568,C#Cc1cccc(NC(=O)NC(c2ccccc2C)C)c1Cl 63569,C(=O)(C#CC1CCOCC1)NC(C1CN(C(C2CCc3nnnn3CC2)=O)C1)C 63570,c1(C(=O)NC2CC3(C(NC(C(C)c4ccsc4)=O)C3)C2)c(F)ccc(F)c1Cl 63571,C1(OCCn2cc(C3N(C(=O)OC(C)(C)C)CCCC3)nn2)CC2(CCC2)C1O 63572,C(C(C(=O)N(C)C)N1CCC(OCCC(=O)OC)CC1)(C1CC1)OCC 63573,c1(COC)nc(NCCC2(OC)CCS(=O)(=O)C2)cc(=NCCc2cnc(C)o2)[nH]1 63574,c1(C(=O)NCC(=C2CN(C(COCCC#C)=O)C2)F)ccc2[nH]ccc2c1 63575,C#CCC(C)(C(=O)N(C)CC1(c2cc[nH]n2)CC1)NC(C1CCC(C)(CC)O1)=O 63576,N1(c2nnc(C(C(CC)C)(C)C)n2C)CCc2ncn(C)c2CC1 63577,C1(CNC(c2nc(C)n(-c3nc[nH]n3)n2)=O)COCCN(C(C2CC2(F)F)=O)C1 63578,C1(CC(=O)NCCC(CCNc2nccc(C(C)(C)C)n2)(F)F)CCCNC(=O)C1 63579,c1(C(=O)NC2C(NC(c3[nH]cc(C)c3)=O)CCC2)ccc(N(C)C)nn1 63580,C1(C(=O)N(C)C(C2CCCC2)C)(OC)CCN(C(=O)CN2C(=O)CCC2=O)C1 63581,N1(C(CCCOC(C)=O)=O)CC(CC(=O)N(C2CCCC2(C)O)C)CC1(C)C 63582,C1(N(C(c2cc(CC)no2)=O)CCO)CCN(C(C23CCCCC2C3)=O)CC1 63583,c1(C(=O)NCC(C)CN(C)C(c2cnc(C#N)cn2)=O)ccc(C(F)F)cc1F 63584,N1(C(C(=O)NCCCC)C)CC(C(C(=O)NCC)N(C)C)(OC(C)(C)C)C1 63585,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(c1ccn(CCF)n1)=O 63586,C1(NC(C(CC)O)=O)CC=C(C(=O)N2CC(OC(=O)NC)C2)C1 63587,c1(C(N(C2CCSC2)CCNC(C2CN3CCN2CC3)=O)=O)cccc(Cl)c1Cl 63588,c1(C(N2CCc3ncsc3C2)C(=O)NC(C)C)cccc2occc12 63589,CCC(F)(F)CC(=O)NC1CN(C(=O)C=CCF)CC1C(F)F 63590,N1(C(C(CCC)CNC(c2cc(C(C)=O)on2)=O)=O)CCOCC(F)(F)C1 63591,C=CC(CC)CC(=O)N1C2CCC1C(NC(=O)C1=CCCCC1)C2 63592,C1(COC)(NC(c2nc(C)nn2C)=O)CCN(C(=O)C(F)OC(C)C)CC1 63593,N#CC1CN(C(C2(c3c(F)cccc3Cl)CC2)=O)CC1NC(=O)CO 63594,Cc1ccc(F)cc1C(=O)C(=O)N(C1CCN(C(C2(C#N)CC23CCC3)=O)C1)C 63595,CC1CCN(C(=O)CCOCC(F)F)CC1CNC(c1ccc(F)c(Cl)n1)=O 63596,c1(C(=O)NC2C(NC(c3cccc(OC)n3)=O)COCC2)cc2n(n1)CCCN2 63597,C1(C(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)CCCOC1c1ncc[nH]1 63598,c1(C(=O)NCC(C)(C)NC(c2c(CC)scc2)=O)ccn2cc(C)nc2c1 63599,c1(NCC(=O)NCCNC(C(C)NC(C)=O)=O)ccc(Sc2ccccc2)cc1 63600,c1(C(N2CCCC(C(N(C3CNCC(C)C3)C)=O)C2)=O)ccc2cc[nH]c2n1 63601,c1(C(=O)NC(CNC(CC(=O)NCC)=O)C(C)C(C)C)cc2nnn(C)c2s1 63602,N12CCN(CC1)C(C)C2=O.C1(CC(N2CCC(NCC)CC2)=O)C(=O)ON=C1C 63603,c1(C(N2CC(SC)C(NC(=O)Cc3cccn3C)C2)=O)n[nH]c2ccc(Cl)cc12 63604,C(=O)(C1=CC2C=CC1C2)N1C(CO)CC(NC(CCC=CC(C)C)=O)C1 63605,c12nc3n(n1)CCCC3NC(=O)N(C)C2.n1(C2(O)CN(CC)C2)nc(C)cc1C 63606,C1(=O)CC(C(C)(C)C)N1C(=O)CN(C1CCCC1)C.Cc1c[nH]c(C(=O)OC)c1 63607,N1(C(CN2CCC(OC)C2)=O)CC=C(C(=O)NCc2cscc2C)C1 63608,C1(C2(O)CCN(c3nc4cccc(F)c4o3)CC2)(NC(C23CC(C)C2C3)=O)CC1 63609,C12(C(=O)NCC3N(C(=O)C=C(Cl)Cl)CC=C3)CC3CC(C1)CC(O)(C3)C2 63610,c1(CC(=O)NCCC2(O)CCN(C(=O)C3=C(Cl)CC3)C2)cn2cc(F)ccc2n1 63611,Cc1nc(-c2ccccc2)[nH]c1C(C)N(C(=O)OCc1ccsc1)C1CC1 63612,c1(C(N(CCOC)CCNC(=O)C(C)SC(F)(F)F)=O)ccoc1Cl 63613,C(=O)(C1=CC2C=CC(C1)C2)N(C)CC1(O)CN(C(c2c(CC)non2)=O)C1 63614,C(=O)(CC1COc2ccccc21)NCC(CC=C)NC(=O)CCc1cnn[nH]1 63615,N1(c2nnc(OC)n2C2CC2)CCC2(CCC2N2CCC23CCCCC3)CC1.O=CO 63616,N1(C(C(n2ncc(C)c2)C)=O)CCC2C(C1)CN2C(C1C2CC3C(C2=O)C13)=O 63617,c1(C(N2CC(CC=C)(C(=O)NCC(=O)NC)C2)=O)ccn2cnnc2c1 63618,N#CC1(CC(=O)NC2CCCCN(C(=O)C(F)CC3CCCC3)C2)CCOCC1 63619,c1(CC)ccc(O)c(C(=O)NC2CC(NC(c3cn(C4CC4)nc3C)=O)C2)c1 63620,N1(C(c2cccc(Cl)c2C)C(=O)NCCC)CCN2C(=O)C(=O)NCC2C1 63621,C1(CC(=O)NC(CC)(C)CNC(=O)CCc2csc(=N)[nH]2)CC2CCC1O2 63622,C=CC(CC)CC(=O)NCCC1CC(OC)CN1C(=O)Cc1cc[nH]c1 63623,N1(C(C2CC(O)(CNC(C(C#C)(C)C)=O)C2)=O)CCC(O)(C=C)C1 63624,c1(NC(c2nc(-c3cn(CCC)nc3)sc2)=O)ccc(O)cc1C 63625,C1(CN(C(C(=O)NC(C(=O)OCC)C)CC2CCCCO2)C)C(C)(C)C1(C)C 63626,Cc1cn(-c2ccccc2)[nH]c1=NC(=O)C(=O)NCC12CC(I)(C1)C2 63627,CC1CN(C(C2CCC2C(C)(C)C)=O)CCC1CNC(C1(c2cccs2)CC1)=O 63628,c1(C(N2C(C(C)C)CN(C(c3cc(=O)cc[nH]3)=O)CC2)=O)cc(S(C)(=O)=O)cs1 63629,c1(NC(=O)CNc2ncccn2)cc2ccc(-c3ccccc3O)cc2[nH]1 63630,N1(Cc2nc(C)on2)CC2C(C(=O)NC(C)Cc3ccccc3F)C2C1 63631,C1(C)(NC(C(C)SCCCC)=O)CCCN(C(c2ccc(Cl)c(OC)c2)=O)C1 63632,c1(COC)nc(C)c(C(=O)NCC2CCC(NC(=O)Cn3cnnn3)C2)s1 63633,C1(C(=O)NC2CC(C)(CNC(Cc3ccc(C)nc3)=O)C2)CCC2(CCC2)O1 63634,c1(CCN(C(=O)CN(C(=O)CC2CCOC2)CC2CCC2)C)nccs1 63635,N1(C(C2CC3(CC(NC(=O)Cc4cccs4)C3)C2)=O)CCC2(CCOC2=O)C1 63636,c1(CNC(C2C(CNC(CC(C)c3ccco3)=O)C2)=O)ccc(S(C)(=O)=O)cc1 63637,Cc1ccc(C)c(NC(=O)CC=CCNC(c2scnc2C)=O)c1 63638,CC(C)(C)CCCC(=O)NCC12CN(C(C3CCCN3C3CC3)=O)CC(F)(C1)C2 63639,CCC(CC)C(F)C(=O)NC1CN(C(=O)COC(F)(F)F)CC1(C)C 63640,C#Cc1cnc(NC2CCCCC2CNC(C2CCCC(=O)N2)=O)nc1 63641,CCC(CC)CCC(=O)N1CC2CC1CN2C(=O)CC1CC1(C)C 63642,C1(NC(CN(C(=O)CCc2ncco2)CCC)=O)CCC(C(C)O)CC1 63643,c1(CC)[nH]nc(Cl)c1C(=O)N(C1CCN(C(c2cnc(C)s2)=O)C1)C 63644,N1(C(C(=O)NC(C)CNC(=O)CC2CC=CCC2)C)C(=O)NC2(CCCC2)C1=O 63645,C1(OC)CC(CCNC(=O)CCN2CCC2)N(C(c2coc(O)n2)=O)C1 63646,C1(NC(C2CC(CC)C2)=O)(CO)CCN(C(c2ccnc(Cl)c2OC)=O)CC1 63647,N1(C(c2cc(COC)no2)=O)CCC2CN(C(=O)CC(F)(F)Cl)CCC2C1 63648,c1(NC(=NCCN2C(C)CCS(=O)(=O)C2)NC2CCC2)cc(Cl)c2c(c1)OCO2 63649,N1(C(C2CC(C)CN2C(c2ccnc(CO)c2)=O)=O)CCN2C(=O)OCC2C1 63650,C1(CNC(C2(C#C)CCCC2)=O)CC2(CCC2)CN1C(=O)C(CC)C1CC1 63651,c1(C(=O)NCCCc2cn(CCOC3CCOC3)nn2)cc(O)cc(O)c1 63652,C(CN=c1[nH]c(Cl)nc2c1CCC2)(C1CCC1)OC1CC1.N12CCOCC(C1)C2=O 63653,C1(COC)CCN(C(=O)C(C)(C2CC2)N(C(=O)CCCC2CCCO2)C)C1 63654,Cc1cc(=NCc2ccns2)[nH]c(N2CCC(C(C)C#N)CC2)n1 63655,C1(NC(c2ccc(C3(OC)CCC3)cc2)=O)CCN(C(=O)CC(N)=O)CC1(C)C 63656,C(CC(F)(F)C(F)F)NC(c1c(CC)cccc1)C(=O)OC 63657,c1(C2(C(=O)NC)CCC2)ccc(Cl)c(C(=O)OC)c1.N12CCC(C1)OC(C)C2=O.CC 63658,C1(N(C(C2(CC(C)(C)O)CCC2)C(=O)OC)Cc2ccccc2)CCCC1(F)F 63659,C1(C(N2CC(C(C)NC(c3ccn(C)n3)=O)C2)=O)CCc2ccc(F)cc2O1 63660,CC(CF)C(=O)NC1(C)CN(C(=O)C(c2ccccc2)C)C1 63661,N1(C(CNC(N2CCCOC2=O)=O)=O)CCCc2[nH]nc(CO)c21 63662,Cn1nc(Br)c2ncnc(NC3CCN(C(c4nsc5ccccc45)=O)CC3O)c12 63663,CC1Cc2cc(C(=O)NC3CC(F)(CNC(C4CC=CCC4)=O)C3)ccc2O1 63664,C1(CNC(C(CCC)=CCC)=O)CCN(C(c2cn(CC(F)F)cn2)=O)C(C)C1 63665,N1(C(C(C)NC(C)=O)=O)CC(C(=O)NCC(C)C(=O)NC2CC2)(CC)C1 63666,C(=O)(C(F)(F)C(F)(F)C(F)F)NCCC(CNC(=O)CCCC1CCCCC1)O 63667,C1(C(=O)NCC2CCN2C(C2CC(OC3CC3)C2)=O)CC=CCO1 63668,N1(C(CCCCCOC)=O)CC2CC(C(N3CCC(CC(F)F)C3)=O)C(C2)C1 63669,N1(C(C(OC)OC)=O)CC(NC(c2ccc(F)c(Cl)c2)=O)CC(C)C1 63670,c1(OC)ccc2nc(CNCC(=O)NCCc3cccc(Br)c3)[nH]c2c1 63671,C1(CNC(C2(OC(C)C)CCC2)=O)CN(C(C2CCCN2C)=O)CC12CC2 63672,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(C)C(CNC(c2c(C)ncn2C)=O)C1 63673,c1(OC)c(C)cc(NC(N2C3CCC2CC(Oc2nccc(Br)n2)C3)=O)cc1C 63674,C#CCC(C(=O)N1CC(C(C)C)N1CC)NC(C1CCOC1(C)C)=O 63675,N1(C(C(C2CC2)SC)=O)CC2CC(C1)C2NC(=O)CSCCNc1ccccc1 63676,C(=O)(CCC(=O)C(C)(C)C)N(C(C)C)CCN(C)C(C12CSCC1C2)=O 63677,C#CCC(O)C(=O)N(C(C(=O)NC(c1nn(C)cc1O)C)C1CC1)C 63678,CC(N=c1nc(CC2CC2)[nH]s1)C1CCCN(C(=O)CC2CCSC2)C1 63679,CCC1CNC(=O)C2=NC(=N)NC(=N1)N2.c1(CC(=O)NC)cc(Cl)cs1 63680,N1(C(CC(CCCC)NC(=O)COCCC(C)C)=O)CC(C)(C)C2CCCC12 63681,C1(C(C)NC(=O)COC2CCC2)CCN(C(C2CCCCC2O)=O)CC1 63682,C(=O)(C(C)(C)CN(C)C(C1CCOC(CC)C1)=O)NC(CCC)c1ccco1 63683,N1(C(CC2CC(SC)C2)=O)CCN(C(c2cncc(C)n2)=O)C2(CC2)C1 63684,C(=O)(CC(C1CC1)NC(C1OCCC1NC(=O)C(C)N1CCCC1)=O)OCC 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63702,CC(C)(C)CCCCC(=O)NC12COC(C1)C(NC(c1cncc3c1CCC3)=O)C2 63703,c1(C(N2CCCC2c2cc(Cl)sc2Cl)=O)c(O)ncc2c1CCC2 63704,N1(C(C(CC#C)NC(=O)CN2CCC(=O)CC2)=O)CC2CCC=CC12 63705,N1(C(C(=O)NC2CC(NC(CC(C)C)=O)C2)C)CCP(C)(=O)CC1 63706,N1(C(C(C)N(C(=O)C(F)CC(C)(C)C)CCO)=O)CCc2ncncc2C1 63707,c1(C(N2CC(C(C)NC(C3CCCC3C)=O)OCC2)=O)csc([N+](=O)[O-])c1 63708,N1(C(c2cc(C)sc2)=O)CC2CCC1C(CNC(c1cc(Cl)ccc1F)=O)C2 63709,CCCCCC(F)C(=O)NC1(C(=O)NC2(C)CC2(C)C)CC1C 63710,C=CC(CCC)CC(=O)N1CC(N(C(C2CCOC2C)=O)C)(COC)C1 63711,N1(C(CCOCC#C)=O)CCC(NC(=O)COCCOCC)C1 63712,N1(C(C2CCCC(C)C2)=O)CCCC2(CCCN2C(=O)CC2CCS(=O)(=O)C2)C1 63713,C1(OC)CCCC(CC(N2CC(O)(CN(C(=O)COc3ccon3)C)C2)=O)C1 63714,C1(CNC(=NC)NCc2cc(C3CCC3)no2)CC[Si](C)(C)C1 63715,Cc1cc(NC(=O)CC2COCCN2Cc2cnc(C3CC3)nc2)n(CCO)n1 63716,C(N1CC(C)C1c1ccccc1)c1n(CC(NOC(CC)(C)CN(C)C)=O)nnn1 63717,c1(C2(C(N3C(CNC(C4(COC)COC4)=O)C=CC3)=O)CC2)ccc(Cl)cc1 63718,Cc1nnc(NC2CC(NC(=O)CCC3CCCO3)C23CCC3)c(C#N)c1C 63719,c1(OCC=C(C)C)ccc(NC(=O)C(N2CCC(C3OCC3(F)F)CC2)=O)cc1 63720,N1(C(C2CCC(CCCCC)O2)=O)CC=C(CNC(=O)CC2CC2(C)C)CC1 63721,C1(C(N(CCC)CCC)=O)CC2CN(C(C3(C)CCC(=O)CC3)=O)CC2C1 63722,c1(C(=O)NC2CCN(C(c3cnc(Cl)s3)=O)C2)ccc(F)c(-n2cccc2)c1 63723,C1(NC(C2(CCCC)COC2)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC1(C)C 63724,C1(c2nn(C)c(O)c2)CCN(N2CC(CS(C)(=O)=O)C2)C1 63725,CCN=c1[nH]cc(C(=O)Oc2ccc(CCNC(C)=O)cc2)s1 63726,C1(CNC(CC2(N(C)C(c3ccc(F)cn3)=O)CC2)=O)CC2(CCC2)CO1 63727,C(=O)(CC1OCc2ncccc21)ONC(=O)C=CC(=O)NCC1CCCCO1 63728,CCCCCC(=O)NC(CO)CCCCNC(=O)CNC(=O)C(CC)C(C)O 63729,C=CCC(CC(F)F)NC(c1ncoc1CNC(=O)C(C)CCCC)=O 63730,C(N=c1cc[nH]cc1[N+](=O)[O-])C1C(C)CN(C(=O)Cn2cc(C3CC3)nn2)C1 63731,N1(C(C(c2c(C)ccc(F)c2)(F)F)=O)CC2CCCC(CNC(=O)C(C)O)(C2)C1 63732,C1(NC(c2[nH]n(C)c(=O)n2)=O)CCOC12CCN(C(c1cncs1)=O)CC2 63733,c1(CC(=O)NC2(CC=C)CN(C(=O)CC3COCCO3)C2)cc(F)ccc1O 63734,N1(C(CC)=O)CC2CC(C(=O)NCC3CC(c4cccc(F)c4)C3)CC1C2 63735,c1(C(N2C3C(NC(CCn4ccc(C)n4)=O)C(C3)C2)=O)cn2cc(Cl)cnc2n1 63736,CCCCC(F)C(=O)N1CC2CC1CC2NC(c1ccc(CO)o1)=O 63737,C1(O)(C(C=C)NC(=O)C(C2CCOC2)NC(=O)COC(C)C)CCSC1 63738,c1(C(=O)NC(CNC(C2(OC(C)C)CCC2)=O)CO)cc2sccc2n1C 63739,c1(CC(=O)NC2CCN(Cc3cnc(F)c(F)c3)CC2)cccc(Cl)c1F 63740,C(=O)(C1COc2ccccc21)NCC1N(C(C(C(CC)C)O)=O)CC(C)(C)C1 63741,c1(C(=O)NC2CC3CN(C(c4nncc(OC)c4)=O)C2C3)ccc2nccn2c1 63742,c1(C(N(CC(CC)NC(=O)CCc2nc[nH]n2)C)=O)ncc(C)cn1 63743,c1(SC)ncc(C(N2CC(CNC(C3CN4CCN3CC4)=O)CC2C)=O)c(O)n1 63744,C(CO)(C(=O)N1CCC(C(N2CC(c3ccon3)C2)=O)C1)OC 63745,n1(CC(=O)NCC(C)OCC)cc(Br)ccc1=O.C12(CC=CCC1)C(=O)N2 63746,N1(C(c2onc(C(C)OC)n2)=O)CCN(C(=O)C=CC2CCOC2)CC1 63747,N1(C(C(CC2CN(C(CCCOC)=O)C2)F)=O)CC(C)(C#N)C1 63748,S(=O)(=O)(c1cc(S(C)(=O)=O)c(C)o1)N1CCC(N(CC)CC)CC1 63749,CC1(C)CN(C(=O)COCC(F)(F)F)CC1CNC(c1cnc(N)c(Cl)c1)=O 63750,N1(C(C2(COCC)CCC2)=O)CCC(CNC(=O)C(C)S)(COC)CC1 63751,N1(C(COCCOCC#C)=O)CCCCC1C(=O)Nc1cccnc1Br 63752,c1(C(N(C)CCN2CCN(C(=O)CC3CC(F)C3)CC2)=O)cc(N)cc(O)c1 63753,C1(C(N2CC(C)C(NC(=O)CCC(C)(F)F)CC2)=O)CC2(C1)C(F)(F)C21CC1 63754,CC(C)CC(O)C(C)C(=O)NC(C(=O)N1CC(n2cnnn2)C1)c1ccco1 63755,c1(C(N2C(CCNC(c3c(C)ncs3)=O)C(C)CCC2)=O)ccc2ncnn2c1 63756,C1(C(=O)NC(C)CCN(C(=O)CCc2cnn[nH]2)C)CCCN(C)C1 63757,CC1CC=CCC1C(=O)NC(CNC(=O)Cc1cc(-c2cccs2)[nH]n1)C1CC1 63758,c1(OC(C)C)cc(C(=O)N(C)CC2CCCN2C(c2c(O)noc2C)=O)ncn1 63759,Cc1cccc(C=CC(=O)NCCNC(CSCCC(O)C(C)(C)C)=O)c1 63760,Cn1nc(C(N2CCSCC2CCNC(C2CCC2(C)C)=O)=O)cc1C(F)F 63761,c1(C(N2CCC3(NC(c4ccc(C)nc4)=O)C(C2)C3)=O)cccc2c1NCC2 63762,n1(C(C)C)ncc2c(NC(CCO)C3CCC3)[nH]c(=NCCc3cn[nH]c3)nc12 63763,N1(C(CCCC(C)C)=O)Cc2nccn2CC(NC(C2CCC(N(C)C)C2)=O)C1 63764,c1(C(N2CC3(C(C(=O)Nc4n(C)nc(C)c4Cl)C3)C2)=O)cc(C#N)ccc1F 63765,c1(C(=O)OCc2cc(C)cc(C)c2)cc(S(=O)(=O)N2CCOCC2)cn1C 63766,C1(C(N(CCN(C2CCN(C)CC2)C)C)=O)CCC2(CCC2)CC1 63767,c1(C(N2CCC(C(C(=O)NCCC(=O)NCC)F)C2)=O)cc(C)ccc1O 63768,N1(C(C2C(C)C2C)=O)CC(O)(C(C)(C)CNC(=O)Cc2cc(C(C)C)no2)C1 63769,Cc1cc(=NC(=O)C(=O)C(C)(C)CCCNC(=O)CCN(C)C)[nH]n1C 63770,C1(C(NOCC(CC)NC(C2CCCOC2)=O)=O)(OC)CC(O)C1 63771,c1(C(N2CC(CN(C)C(c3nn(C)cc3C(F)F)=O)C2)=O)ncccc1F 63772,Cc1oc(C(c2nnnn2C(C)C)NC2C=CCC2)cc1CSC 63773,c1(CC(N2C(C)CCC(C)C2)=O)cc2ccccc2oc1=O 63774,c1(OC)ccc(O)cc1C(=O)C(N1CCCCC(NC(=O)C2=CCCCC2)C1)=O 63775,c1(C(N2CC(CN(C(=O)C(C3CCOCC3)O)C)C2)=O)ccn(C)n1 63776,CC(O)CCCC(=O)NC1CN(C(C2(C(=O)OC(C)(C)C)CCC2)=O)C(C)(C)C1 63777,C1(CCNC(c2ccc(CC)o2)=O)CN(C(=O)CCc2ccc(C)o2)CCCO1 63778,c1(CCC)cccc(C(=O)N(C2CN(C(=O)CC3(F)CCC3)C2)C)c1 63779,C1(NC(C2(COC)CN(C(c3cnsc3)=O)C2)=O)CC(=O)N(C)C1 63780,C1(O)(CCNC(CNC(=O)OCC)=O)CCN(C(=O)C(C(C)C)n2cnnn2)C1 63781,C1(SC)CN(C(C2C(C)(C)C2(F)F)=O)CC1NC(=O)CN1CCOCC1=O 63782,Cc1cc(C(=O)NC2C3CCN(C(=O)Cc4ccc(O)c(C)c4)C23)ccc1F 63783,N1(C(C(=O)NCCOCCOC)=O)CCCCC(NC(c2nn(C)cc2Cl)=O)C1 63784,N1(C(C(CC)NC(N)=O)=O)CCC12CN(C(=O)CC1CCC(O)C1)C2 63785,C1(CNC(C(COCC)C)=O)Cc2ccccc2CN1C(C1(F)CCCC1)=O 63786,C1(C(N2CC(CNC(C(C)OCC(C)C)=O)OCCC2)=O)CCc2ncsc2C1 63787,c1(C(=O)NCC2(OC)CN(C(=O)CC3(C)OCCO3)C2)cccc(S(N)(=O)=O)c1 63788,c1(C(N2CC(NC(CCCc3ncc(C)o3)=O)C(C)C2)=O)cnc2cc[nH]c2c1 63789,c1(C(N2CCC(NC(C3CCCC3(F)F)=O)(CF)C2)=O)ccn2c(O)nnc2c1 63790,C1(N(CCOC)C)CCN(C(=O)C(c2csc(C3CCCC3)n2)C)CC1 63791,C(CNC(c1ccon1)=O)(CC(F)(F)F)NC(Cc1ccc(OC)nc1)=O 63792,C1(C(=O)NC(C)CNC(c2nc[nH]c2C(F)(F)F)=O)CN2CCCCC2CO1 63793,Cc1ccccc1C=CC(=O)NCCN(C(C1CCOC1)=O)C1CC1 63794,C=CCCCC(C(=O)NCC1CCCN1C(C)C)NC(c1c[nH]c(=NC)o1)=O 63795,c1(NC)scnc1C(=O)NC(CO)C(C)NC(=O)C(CC)OC 63796,C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)C(C)Oc1ccccc1Cl 63797,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 63798,C1(NC(c2n(CC(C)C)ncc2)=O)CC2(C1)CC2NC(C1=CC=C2CC12)=O 63799,C12(CNC(C3CCCC4CC34)=O)CN(C(c3cn[nH]c3)=O)CC(F)(C1)C2 63800,C1(S(N)(=O)=O)(NC(c2cnn(C)c2C(=O)OC2CN(C3CC3)C2)=O)CCCC1 63801,N1(C(C(CCC)C)=O)CC(C2CCCCN(C(=O)CCC3CC3(C)C)C2)C1 63802,c1(C(=O)OC)cccc2cccc(CNc3cc(OC)c(OC)c(I)c3)c12 63803,c1(N2CC=C(C)CC2)nc2cc[nH]c2c(=NC(C)c2cccnc2OC)[nH]1 63804,c1(SCC)cc(Br)ccc1C(=O)NCC1CC1NC(c1csc(CC)n1)=O 63805,N1(C(c2noc3ncccc23)=O)CC2CCC1CN2C(c1cc(Cl)cnc1Cl)=O 63806,C1(NC(CC(C)c2ccco2)=O)CC12CCN(C(=O)C(C)(C)CCC#N)CC2 63807,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(NC(=O)CCF)CCOC1 63808,C1(CC(C)(C)C)CN(C(C2CCC(C(N)=O)C2)=O)CCN1C(c1cnsn1)=O 63809,C(=O)(CCCCCNC(=O)NCCSCCCO)NC1C(CCC)CCCC1 63810,C(=O)(C(C)CNC(=O)C(Cc1cc[nH]n1)NC(C1CC1C#N)=O)NC 63811,N1(C(C2C(C)CC(=O)CC2)=O)CC(NC(C2CCCCC2)=O)C2CCCCC12 63812,C(CCCCCNC(CC1(OCC)CCC1)=O)NC(C1CCC(N(C)C)C1)=O 63813,c1(OC)cc(SCC(N2CC(CNC(C3CCC(C)(C)CO3)=O)C2)=O)cc(F)c1 63814,CC(Cc1ccc(Cl)cc1)CC(=O)NC(C)(CNC(=O)C=Cc1nccs1)CO 63815,CC(CCC(C)(C)C)C(=O)N1CCN(CCN(C)C(c2cc(Cl)ccn2)=O)CC1 63816,N1(C(Cc2c(COC)cccc2)=O)CC2(CCN(C(C3CCN(C)C3C)=O)C2)C1 63817,CC1CCCC(CNC(c2cc(CNC(c3cc(Cl)n[nH]3)=O)nn2C)=O)CC1 63818,C1(C(N(C(C#C)C2CCC2)C)=O)CSCCN1C(=O)C(O)C1CCC1 63819,C1(CC(=O)NC2(CO)CC(OC)C2)CCCCN1C(=O)CC1CCC(C)(C)C1 63820,c1(-c2cn(C(C(=O)OC)C)nn2)ccc(NC(=O)C(C)COC(C)C)c(Br)c1 63821,N1(C(c2ccc(OC)o2)=O)CCCC(C2CCCCN2C(C2CCCOC2)=O)C1 63822,CC1OCCC1CCc1ccn(CC(F)F)n1.C1CCCN(C)C(=O)N1 63823,CCCC(F)F.C(=O)(C(C)n1cccn1)NCCCN(CCCN)C 63824,c1(CC(=O)NCCOCCN(C(c2c(C)cc(CO)o2)=O)C)ccc(F)c(F)c1 63825,C(=O)(C(CC(C)(C)C)NC(c1ccc(F)cn1)=O)N(CCCCCC=C)C 63826,N1(CC(C)CCO)CCOCC(C(C2(O)CCCCC2)NC(=O)OC(C)(C)C)C1 63827,Cc1nn(C)cc1S(=O)(=O)NC1CC1C(=O)Nc1cc(OC(F)F)cc(O)c1 63828,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 63829,N1(C(c2cnc(OC)nc2C)=O)CC2CC(NC(C3CN(C(C)=O)C3)=O)CC1C2 63830,C1(C)(CCC(=O)N(CC(CC)OC)C)CCCN1C(=O)CN(CC)CC 63831,C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1(O)CN(C(CC2CCN(C)C2)=O)C1 63832,C1(CNC(=O)CCCC2CCCC2)CC2CCC1N(C(c1cccnn1)=O)C2 63833,C#CCCCCCNC(c1ccc(CNC(=O)CC2CCCC(O)C2)nc1)=O 63834,c1(C(=O)NC(C(CO)NC(c2n(CC)ccc2)=O)C)cnc(N)cn1 63835,c1(C(=O)NCC2CCCN2C(=O)COC2CCCCCC2)ccc2ncsc2c1 63836,N1(C(C)C)CC(NC(c2cc(CNC(C3CC3F)=O)[nH]n2)=O)CC1=O 63837,C(CC(CC)CC)(c1n(-c2ccccc2)nnn1)OC.C(F)F 63838,c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CCCC2)ncc2[nH]ncc2n1 63839,N1(C(C(CC)SC)=O)CCC(CN(C(=O)Cc2cc(CC)nn2C)C)CC1.C(C)=O 63840,C(C(C(=O)NC1(CC(=O)N(CCC(O)CO)C)CCC1)OC)OC 63841,Cc1cccc2c(CN3CCC=C(C(=O)NCc4nccnc4Cl)C3)c[nH]c12 63842,C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC=C)NC(=O)Cc1cn(C2CC2)nn1 63843,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 63844,Cc1cc(=NCCc2nncs2)[nH]c(N(C)C(C)C2CC2)n1 63845,CCCC(CCC)C(=O)N(C1CCCC(NC(c2cc(CCCO)on2)=O)C1)C 63846,CC1CCCCC1(C)C(=O)NCCN(CCOCCO)C(c1nn(C)cc1N)=O 63847,c1(N2C(C(=O)NCCCNC=O)CC(O)C2)ncnc2c1cc(I)n2C.CCO 63848,C1(C(=O)NCC(CC)CC)CN(C(C2(OC(C)=O)CC2)=O)CC1(C)C 63849,N#Cc1cc(CN2CCNC(C(=O)NCc3ccsc3)C2)ccc1F 63850,c1(N2CC3CN(C(c4cc(C)nc(C)c4)=O)C3C2)ncnc2n[nH]cc12 63851,c1(COC)cccc(C(=O)NCC2(C(c3cnn(CCSC)c3)=O)CCCC2)c1C 63852,Nc1cc(C(N2CCN(C(=O)CCCN3CCCC3)CC2C2CC2)=O)cc(O)c1 63853,c1(CNC(C(c2cn(-c3cccc(C(N)=O)c3)nn2)C)=O)ncc(Cl)nc1N(C)C 63854,C1(NC(c2c(C)[nH]nc2Cl)=O)CCN(C(c2ccc(C3CC3)c(F)c2)=O)C(C)C1 63855,c1(-c2cn(CCN(C(=O)C(O)C(C)C)CC)nn2)c(F)cccc1Br 63856,c1(C(=O)Nc2c(C)nccc2)c[nH]c2cc(-c3ccsc3C)cnc12 63857,c1(CC(=O)NCC(CC=C)NC(c2cc(Cl)no2)=O)cn2ccsc2n1 63858,c1(C(N2CCC(N(C(CSCC)=O)CC)C2)=O)nnc(O)c(Br)c1O 63859,C(=O)(C1=CCC(C)(C)CC1)NCC(C)NC(c1cccc(N2CCCCC2)c1)=O 63860,C1(C(=O)NC2(C)CN(C(C(C3CCC3)OC)=O)C2)CC2CCC(C1)C2O 63861,c1(CNC(=O)CCc2cccc(O)c2)cnc2c(C(=O)O)cnn2c1 63862,n1(CC)ccc(CC(=O)NC2(CCNC(C3CC=CCC3)=O)CCC2)n1 63863,N1(C(C(C=C)C)=O)CCN(C(c2cn(C)nn2)C(=O)NCC2CC2)CC1 63864,Cc1cnn(C)c1CNC(=O)C(C1CC1)NC(c1ccc(OC(C)C)nn1)=O 63865,c1(C(=O)NC2(CCNC(C(C(C)(C)C)SC)=O)CCCC2)cc(C)c(N)cc1Cl 63866,c1(C(N2C(C3(N(C)Cc4ccc(C(=O)N)[nH]4)CC3)CCC2)=O)ncncc1Cl 63867,N1(C(C2CCN(C(C3CCC(CC)CC3)=O)C2)=O)CCCNC(=O)C12CC2 63868,c1(C(c2ccccc2OCC#N)CC)nc(-c2nc[nH]n2)nn1CC1CCCO1 63869,c1(C(N2C3(C(=O)NC4CC(C)(O)C4)CC(C2)C3)=O)cc(C#N)ccc1N 63870,C1(=O)C(O)(CC)CN2C=NN=NC2(CC)C(=O)NCC(CC=C)N1 63871,C1(CC(=O)NCC2CCN(C(=O)NC)C2)CCCCN1C(c1ccc(F)s1)=O 63872,C1(CC(=O)NCC2C(CC)CCO2)CCCCN1C(C1CC(N(C)C)C1)=O 63873,N1(C(Cc2cccc(OC)n2)=O)CCN(C(c2cn(C)cn2)=O)CC1CC(F)F 63874,C(CCCC(C)(C)C)NC(CC(CNC(C1CC1(C)C)=O)OC)=O 63875,Cc1nn(C)c(C)c1CCC(=O)NC1CCC(F)(CNC(C23COCC2C3)=O)C1 63876,c1(COC)nc(NCCc2cccc(C#N)c2)cc(=NCC2(C(C)C)CC2)[nH]1 63877,C(=O)(CC1=CCCCC1)N(C)CC1N(C(C2(OC)CC2)=O)CCC1 63878,C1(NC(c2cc3n(n2)CCOC3)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC12CCC2 63879,C1(SCC)CC2CCC(C1C)N2C(=O)C(C)OC(c1cnn(C(C)C)c1)=O 63880,C(N=c1ccc(C#N)c[nH]1)C1CN(C(C(C(C)C)SCC)=O)CC1C 63881,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 63882,Cc1nc(C(=O)N(C)CC2CCCCN2C(=O)Cn2ncccc2=O)c(C)s1 63883,N1(C(CCOCC#C)=O)CCCN(CCNC(c2ncnc3cc[nH]c23)=O)CC1 63884,CCC(F)(F)CN(C(=O)C(N1CCCC1C1CC=CCC1)=O)CCOC 63885,c1(CNC(C2CCCN(C(C34COC(C5CC5)(C3)C4)=O)C2)=O)ccccc1Br 63886,Cc1cnc2n1CC(C(N1CCOCC1CN(C)C(c1nncs1)=O)=O)CC2 63887,c1(NC(CC2C(C)OCC2)C)ccc(C(=O)NCCSCc2ccccc2)cn1 63888,CC1(C)CCCN(C(=O)Cc2n[nH]cc2Br)C1CNC(c1scnc1Cl)=O 63889,CCC(CN(C)C)CC(=O)NC1(CNC(C)=O)CN(C(C2CC(OC)C2)=O)C1 63890,c1(C(=O)NC2CCCC(NC(c3ccc(CC)o3)=O)C2)ccc2ccccc2c1 63891,C1(NC(C2CN(C(CC)=O)C2)=O)CCC2CCN(C(c3csnc3C)=O)C1C2 63892,N1(C(C2C(NC(CC(C)CN(C)C)=O)CC2)=O)CCCCC(CO)C1 63893,N1(C(=O)CN2CSCC2=O)CC2(CCCC2)C1C(=O)NC1CCC2CCC1C2 63894,C(c1ccc(OC2CCCC2)cc1)=CC(=O)N(C(CNC(CC(C)C)=O)(C)C)C 63895,C(=O)(C(C)(C)CN(C)C)N1C(CNS(CC=C)(=O)=O)CC1 63896,C1(N(C(CCOCCOC)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1C 63897,N1(C(=O)COCC2CCOC2)CC2(C1)CN(C(=O)C(F)N1CCC1)C2 63898,C1(NC(C=CC)=O)CC2CN(C(=O)CC(c3c(C)nn(C)c3C)=O)CCN2C1=O 63899,N1(C(c2nnc(C)s2)=O)CC2(CO)CC1(CNC(c1cc(C(F)(F)F)cs1)=O)C2 63900,C1(C(=O)NCC2CC(CNC(C3CN(C)C3)=O)C2)CCOC(=O)CC1 63901,C1(CNC(=O)CC2CCC3CC3C2)CC2COCC2N1C(c1ccc(Cl)s1)=O 63902,c1(C(N2CC(C(C)NC(=O)CCC3(C)N=N3)OCC2)=O)ccc2nc(O)[nH]c2c1 63903,N1(C(C)C)CCCCC1C(=O)N(CCCNC(=O)C(C1CCOCC1)C)C 63904,C(=O)(C(F)C(C)(F)F)NCc1cc(C(N2C(C)(CCC)CC2)=O)no1 63905,N1(C(c2cc(C)oc2C)=O)CCCOC(CNC(=O)C(C2CCOCC2)F)C1 63906,C(=O)(CC1=CCOCC1)N1C(CCNC(CCC(=O)N(C(C)C)C)=O)CSCC1 63907,CCC(CC)C(F)C(=O)NCCCC(O)C(=O)N(CCF)C1CC1 63908,N1(C(c2[nH]cc(C)c2)=O)CCC(NC(=O)COc2ccc(F)nc2)CC1C1CC1 63909,Cc1cc(=O)oc(C)c1C(=O)NCC(C(C)C)NC(C1CCCCC1O)=O 63910,C(=O)(C(O)CCNC(=O)Cn1cnnc1O)NC1CC(C=C)C1 63911,c1(CC)ccccc1CC(=O)NC1CCC(NC(C2(CC)CC2)=O)CC1 63912,N1(C(CC(C)C)=O)CCCC1C=CC(=O)NCCC(F)(F)Cl 63913,N1(C(Cc2scc(C)n2)=O)CCCC(C)C1CNC(=O)Cc1cnoc1 63914,c1cc(Cl)ccn1.C(=O)(C(C)N(CCNC(=O)SC)C(C)C)NCCOCCC=C 63915,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(C(C)=O)cc2)cc(N)cc(F)c1 63916,C(=O)(CC(CC)C(C)C)N1CCN(C(CCC=CC)=O)C(CCOC)C1 63917,N(C1CC(C)n2ccnc21)CC(COC)Oc1ccccc1 63918,C(CCCC(=O)NC1CCCC1NC(=O)C(c1ccc(Cl)s1)=O)SC 63919,c1(SC)nc(NCCN(C(=O)C(CC(C)C)N(C)C)C(C)C)cc(Cl)n1 63920,CN1C(=O)CCC1C(=O)NC12CC(C(=O)NC(CC3CCCO3)CO)(C1)C2 63921,C(C(C(=O)NC1CC(N(C(=O)CC#N)C)C1)C(C)(C)C)N(C)C 63922,C(c1cocn1)=CC(=O)NC1(CC(=O)NCCSCCOC)CCC1 63923,c1(CC)cc(C(N2CCC(OCCNC(=O)C(C)SC)C2)=O)c2c(c1)CCO2 63924,c1(OCC=CC(N2CC(N(C)C(C3CC3F)=O)C2)=O)ccccc1 63925,c1(C(=O)NCC(CNC(=O)CC2C=CS(=O)(=O)C2)OC)nnn2c1CCCC2 63926,C(N=c1ccnc(C2CCCC2)[nH]1)C1(NC(c2c(C(C)N)ocn2)=O)CC1 63927,c1(OC)cc(C)c(C(C)(OC)NC(=O)C(C2CC2)OC(C)(C)C)cn1.C1CN1 63928,c1(OC)c(Br)cc(CN2C(C(=O)NCCc3ccc(I)cc3)CC3CC23)cc1Br 63929,C(C(C(C)C)NC(=O)OC(C)(C)C)NC(=O)C(C#N)=CCNC(C=CCC)=O 63930,CC(C)(C(=O)NC(C1CCC(NC2CCCC2)C1)C1CC1)C1CC1 63931,c1(N2CCCCC(NC(C3C(C)CC(=O)N3)=O)C2)ncnc2c(F)cccc12 63932,c1(C(N2CCCC(COC)C2)C(=O)NCC2CCCO2)n[nH]c2cc(Cl)ccc12 63933,Cc1cnn(CCNC(C2N(C(=O)C(CO)NC(=O)C(C)C)C(C)C2)=O)c1 63934,C1(OCC)CC(NC(=NCCC(=O)N(C)C)NCC2CC2)C12CCOCC2 63935,C1(C(=O)NCC2OCCN(C(c3cc(CC)oc3C)=O)C2)COC2COCC2O1 63936,CC1(C)CCCN(C(=O)Cc2ccccn2)C1CNC(c1nccc(Cl)c1F)=O 63937,c1(C(C)C)cccc(CC(=O)NCCN(C(=O)C(O)C(F)F)CC2CC2)c1 63938,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 63939,CCC(CC(=O)NCC1CN(C(=O)C=C(C)C(F)F)C2COCC2O1)C(C)(C)C 63940,C(CO)(C(=O)NC(CNC(C1CNC(=O)C1)=O)C1CCC1)N(C)C 63941,c1(CC(=O)NC(C2CCN(C(=O)C3=CCOC3)CC2)C)cn2ccsc2n1 63942,Cn1cnc2c(C(=O)N(CCCNC(C3CC3C(=O)N)=O)CCO)ccnc12 63943,C1(NC(C(CC)N(C)C)=O)CN(C(c2csc(C(C)OC)n2)=O)CC1C 63944,C12(NC(c3csnn3)=O)CCOC(CNC(C3C=CC=CC=C3)=O)(C1)C2 63945,c1(Cn2cc(C(C)NC(c3ccc(Cl)nc3O)=O)nn2)cc(F)c(F)cc1F 63946,C1(CC(=O)NC2CCN(C(=O)CC34CCCC3C4)C2)(CC=C)CCCC1 63947,C1(NC(CC=C)=O)CCCCC1CNC(c1cn(CCc2ccccc2)cn1)=O 63948,C(=O)(CCC(C(=O)NCCn1cc(CC(=O)O)nn1)N(C)C)OC 63949,N1(C(c2c(CC)c[nH]n2)=O)CC(OC)C2(CC2)C1.C12(CCOC1)C(=O)N2 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64020,C1(CNC(Cc2cc(C)[nH]n2)=O)CN(C(c2csc(C)n2)=O)C2CCN1C2 64021,c1(CC(=O)N(C)CCn2cc(CN3CCCC(F)C3)nn2)ccc2nsnc2c1 64022,c1(C(=O)NCCCC2CNC2)cc2c(Br)cnn2cn1 64023,Cc1cccc(C=CCC(=O)NCCC(C)N(C)C(C2CC2C#N)=O)c1 64024,c1(C2C(=O)NC(C#N)N(C)CCCN2C)ccoc1C.C(C)(C)(C)C1CC1 64025,CS(=O)(=O)c1cnn(CC(N2CC(NC(c3ccsn3)=O)C(O)C2)=O)c1 64026,c1(CC)ccc(F)cc1C(=O)NCC1(C(F)F)CCN(C(c2ccnn2C)=O)C1 64027,C12(NC(Cc3cnc(OC)nc3)=O)CCC1CN(C(c1ccc(Cl)cc1O)=O)C2 64028,C1(CNC(C(C)CO)=O)CC2COCC2N1C(C1CCC(F)C1)=O 64029,c1(C(=O)NCCN(C(c2nc(C(C)C)sc2)=O)C2CC2)ncccc1O 64030,N1(C(C)=O)CCC12CCC2.c1(C2c3nnnn32)cccc(Cl)n1.C1CN1 64031,c1(CCC)nc(C(C)NC(=O)CC2C(NC(c3sccc3F)=O)CC2O)no1 64032,c1(C(N2CC(CNC(C(CC)C(C)C)=O)(OC)C2)=O)ccc2c(c1)COC2 64033,C(C)(C(C)NC(=O)C(C1CC1)N(C)C(C1(n2cccn2)CC1)=O)SC 64034,c1(C(=O)NC(CNC(c2ccc(OC(C)C)nc2)=O)(C)C)[nH]nc([N+](=O)[O-])c1Cl 64035,C1(NC(CN(C)C(c2ccco2)=O)=O)CC2CC1CN(C(=O)C1=CCCS1)C2 64036,Cc1ccc(OCCC(=O)NC(CNC(c2c(C)cnn2C)=O)C2CC2)c(C)c1 64037,c1(C(N2CC(C(=O)NC(CCC=C)CO)OCC2)=O)ccc2nonc2c1 64038,c1(C(=O)OC)cnc(C)nc1CN1CCC(N(C(CCC(=C)C)=O)CC)C1 64039,c12cccc(n1)NC(=O)C1CCN(C1)C2=O.c1(C(=O)OC)nc[nH]c1OC 64040,c1(C(N(CCCC(N2CCCC(CSC)C2)=O)CC)=O)cc(Cl)cnc1C 64041,c1(N(C)C)ccc(NC(C2CC3CC3N2C(c2cnc(O)[nH]2)=O)=O)cc1F 64042,c1(C(C(N2C(C(=O)NC(C(C)O)CO)CCC2)=O)(C)C)ccccc1F 64043,Cc1ncnc(O)c1C(=O)NC1CCN(C(=O)Cn2cncn2)C1(C)C 64044,C1(NC(CCc2cccc(OCC)c2)=O)CCCCCN(C(=O)C(F)=CCCF)C1 64045,C1(C(=O)NC(CNC(CCCN(CCCC)CCCC)=O)C)CC12CCOC2 64046,C12(NC(c3c(C)nsc3)=O)CCC(CN(C(c3scc4c3OCCO4)=O)C1)C2 64047,C=CCC(C(=O)NCC1CC(F)(CNC(=O)CC(O)CN(C)C)C1)OC 64048,c1(C(=O)Nc2c(NC(C(CC)O)=O)cc(OC)cc2)cnc2c(NC)cccn12 64049,n1(CC)cc(C(N2CC(CNC(=O)Cc3ccoc3C)C3(CC3)C2)=O)ccc1=O 64050,C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(N2C(C)CCCC2)=O)C1 64051,N1(C(C2CC(C#N)C2)=O)CCCCC1CNC(c1ccc(Cl)[nH]1)=O 64052,c1(C(=O)NCCC(C)(C)NC(C2C(C)C2)=O)nc(OCC(F)F)ccc1Cl 64053,C(CCC(=O)N(C1CCC(NC(=O)COC2(C)CCCC2)C1)C)N(C)C 64054,C=CC(C)(CC)C(=O)N1CC(OC)C(NC(=O)C(F)(F)c2cscn2)C1 64055,O(C1Cc2ccccc21)C(=O)NC(COCCCCC)=O 64056,c1(C(=O)NC(C(C(=O)OCc2c(OC)nn(C)c2)C)C)cn(C)c(=O)cn1 64057,C(CCC1CC1)(C(=O)NC1CC(N2CCCC2)C1)NC(C=CC(=O)N(C)C)=O 64058,Cc1cc(O)c(F)cc1CN1CCOC(c2cn(CC3(O)CCC3)nn2)C1 64059,C1(C)(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C)C)CCC(=O)NC1 64060,c1(C(C(=O)NCCOC)N(C)Cc2cncn2C)csc2c1CCCC2 64061,C(=O)(N=c1ccc(Cl)n[nH]1)c1ccc(NC(C(CCC)(C)C)=O)c(OC)n1 64062,c1(NC(CCC=C)=O)cccc(C(=O)NC(=O)CCc2ccnnc2)c1 64063,C1(F)(CNC(c2ccc(CC)s2)=O)CCCN(Cc2cccc(C)n2)C1 64064,C1(NC(C=COCC)=O)CN(C(=O)C=CI)CC2(CCOCC2)C1 64065,C1(NC(C(C)C)=O)CN(C(=O)C(F)C2CCCC2)C2(CCOCC2)C1 64066,CC1(C)NC(=O)N(CC(N2CCC2CNC(=O)COc2ccon2)=O)C1=O 64067,c1(NC(=O)C(=O)N2CCC2)cc2cc(C(=O)OC)ccc2oc1=O 64068,CCC(C)CC(=O)C(=O)N1C(C(N2CCCC(C(=O)OC)C2)=O)CCC12CC2 64069,C1(C)(c2cn(CC34N(C(CC5CCN(C)C5=O)=O)CC(C3)C4)nn2)CC2(CCC2)C1 64070,CCC(C(=O)N1CCCC1C(C)(C)NC(c1ccc[nH]1)=O)N(C)C 64071,N12CCOC(C)(C1)CNC(=O)C2.c12cc(on1)CNC2=O.C1(C(=O)C2CC2)CCC1 64072,CN1CCN(CC2CCC(O)C(C)(C)O2)c2cc(C(=O)O)ccc21 64073,c1(OC)ccccc1C(=O)N(CC(C)NC(c1coc(C2CCC2)n1)=O)C 64074,C(C(C(C)C(C)C)NC(c1cnn(C(F)(F)F)c1)=O)NC(C(COC)(C)C)=O 64075,C1(CC(=O)NCc2coc(O)n2)CCCCN1C(c1ccccc1Cl)=O 64076,c1(NC(c2n(C(CC)C)nnn2)C2(CC(N)=O)CC2)cnc(CN(C)C)nc1 64077,C1(C(=O)NC(C(=O)N(CCCCO)C)CC2CCCC2)CCC2(CC1)CC2 64078,C1(NC(C(C)(C(C)C)NC(C)=O)=O)CC2(CCCCN2C(C2CCOCC2)=O)C1 64079,Cc1cc(C)c(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)O)C)c(O)n1 64080,Cc1cnc2ccccc2c1C(=O)NC1CC1NC(=O)Cc1ccno1 64081,C1(CNC(C=CC)=O)CN(C(=O)CCOc2cc(Cl)ccc2Cl)CC12CC2 64082,c1(CC(C)NCCN(C(=O)OC)Cc2ccccc2)cccc(SC)c1.C(F)(F)F 64083,C1(NC(c2cocc2Br)=O)CN(C(C23CCCCC2C3)=O)CC2(CCC2)C1 64084,N1(C(C(C)(F)F)=O)CC2CCC(CNC(C3CSC3)=O)C2C1 64085,C(=O)(C1CCc2ccccc21)NCC1(NC(CC2CC(C)C2)=O)CCC1 64086,CC1CCCCN1Cc1ccccc1NC(=O)NCc1cn(CCCCCO)nn1 64087,N1(C(c2ccc(NC)cc2)=O)CCCC12CN(C(=O)Nn1nc(C)cc1C)C2 64088,C1(C(N2C(C)C(NC(c3ncnn3C)=O)CCC2)=O)CCc2nncn2C1 64089,c1(OC)cccc2sc(C(=O)N(CCCNC(=O)C(C)SC)CC(C)C)cc12 64090,c1(CC(=O)N(C2CCCN(C(C=CCC)=O)C2)CCO)c(Cl)cccc1Cl 64091,CCCC(C(=O)NCC12CC(CO1)N(C(C1CCC(CCC)CC1)=O)C2)C(C)C 64092,c1(C(=O)NC(C)(CNC2CC2C#N)C2CCC2)ccc(N2CCC2)nc1 64093,CCCC(C)N=c1[nH]c(=NCc2nocc2C(C)(C)C)[nH]c2c1CCC2 64094,CC(C)(O)CCC(=O)NCCCCCNC(c1ccnn1C1CCC1)=O 64095,N1(C(C2CC=C(C)CC2)=O)CC2CCN(C(c3ccoc3CC(N)=O)=O)CC2C1 64096,CC1C(NC(c2cnn(C)c2N)=O)CCCN1C(=O)CNS(N)(=O)=O 64097,c1(CNC(C(=O)NC(COCC)C(C)C)=O)cnc(O)c(F)c1 64098,Cc1cc(C(=O)NC(C(=O)NCC2CSC2)C(C)O)cc(O)c1 64099,c1(CC)ccccc1OCCC(=O)NC1CCCN(C(c2cc(C)c[nH]2)=O)C1 64100,Cc1ncncc1C(=O)NC1CCCC1C(=O)NCC1CCN(C)C1 64101,C1(NC(C(C)SC)=O)CCOC12CCN(C(c1cc(Cl)c(F)cc1N)=O)CC2 64102,C(=O)(N=c1c(C)c[nH]cc1Br)c1cccc(N2CCC(NC(C)=O)C2)c1 64103,N1(C(C2(CC(C)=O)CC2)=O)CCC(CNC(c2cc(C(F)F)[nH]n2)=O)C(F)(F)C1 64104,C1(NC(CSCCC)=O)CC(C)CN(C(=O)C(O)C(C)CC)C1 64105,Cc1ccc(CNC(C2C(C)CN2C(=O)C=Cc2cscn2)=O)c(C)c1 64106,N1(C(c2c(C(C)=O)ccs2)=O)CCCN(C(c2c[nH]nc2C)=O)C(CN(C)C)C1 64107,c1(C(N2CCC=C(F)C2)C(=O)NCCC#N)ccc2cccnc2n1 64108,c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)C(CN(C)C)C(C)C)cc1C 64109,c1(C(=O)NC2(CC#C)CCOC2)cnc(CNC(C2(C)CCOC2)=O)nc1 64110,c1(C(=O)NC(c2c(C)n[nH]c2C)CC(=O)O)cc2ncccc2[nH]1 64111,N1(Cc2c(C)con2)CCC(C2CCCN(C(=O)CCn3cc(C)cn3)C2)C1 64112,S(=O)(=O)(c1csc2ccccc12)N1C2CN(C(COC)=O)C(CC2)C1 64113,c1(S)ncc(C2CC(N(CCCOCCO)C(=O)OC(C)(C)C)C(O)C2)cn1 64114,C1(C#N)(NC(=O)NCc2c(F)cc(C)c(Cl)n2)CC2CCC(C2)C1 64115,C(=O)(CC(C(F)(F)F)N(C)C)N1CC(C)C2(C1)CC2.C(=O)(CCc1cnco1)NC 64116,Cc1ccc(OCCC(=O)NC2CN(C(=O)Cn3ccnn3)CC2(F)F)c(C)c1 64117,Cn1ccc2nc(NC3(C#N)CCN(c4ncccn4)C3)ncc12 64118,c1(NC(C2(C)N(C(c3ccc(OC)c(Br)c3)=O)CC2)=O)cc(Cl)cc(Cl)c1O 64119,N1(c2n(CCOCC=C)c(Cc3sccc3Br)nn2)CCc2ncnc(O)c2CC1 64120,C1(C(=O)NCC2N(C(C3=NOC(C(C)(C)C)C3)=O)CC2)CCC2(CCC2)CO1 64121,c1(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccc(Br)cn2)ncncc1Cl 64122,C1(NC(CC(=C=C)C)=O)CC2CN(C(=O)CC3CC(N(C)C)C3)CC2C1 64123,C1(NC(c2ccn(CC)n2)=O)CC2CC1N(C(c1cc(CC(C)C)on1)=O)C2 64124,N1(C(c2c(O)ccc(C)n2)=O)CCC2(CC1)CC2NC(c1ccoc1C1CC1)=O 64125,C(=O)(CC(C)CC(=O)OC)NC(CCC)C(=O)N(CC)Cc1ccco1 64126,C1(C(N2CC(N3C(=O)C3(C)C3CC3)C2)=O)C2CC3C(C2=O)C13.COCO 64127,N1(C(C(=O)OC)CCc2ccc(Cl)cc2)CCCN(C(C)C(N)=O)CC1 64128,c1(C(=O)OC)cncc(C(N2CC(F)CC2CNC(=O)CCC=C(C)C)=O)c1 64129,CCC(C(=O)NCC1(CCNC(c2sc(C)nc2C)=O)CC1)C(C)C 64130,C#CCCCCCCC(=O)NCC(C)(C1CCC1)NC(C1CCOC(C)(C)C1)=O 64131,N1(C(CC=C)=O)CCC2C(NC(c3cc(Cl)cnc3OC)=O)C2CC1 64132,c1(CC(=O)NCCCCC(CO)NC(C2C(CC)C2)=O)cnc2ccccc2c1 64133,c1(C(N2CCN(C(CS(=O)(=O)NCC)=O)C(C)C2)=O)cc(Cl)cc(C)c1O 64134,c1(C(N2CCCC(NC(CNC(CC)=O)=O)(CO)C2)=O)cc2c(C)cccn2c1 64135,C(=O)(CC(C)CC(C)(C)C)NC1(c2ccccc2-c2c(C)c(Cl)ccc2)CC1 64136,C12(C)CCCN1C2=O.n1(CC)cc(CNC(=O)CCCC2CC2C)nn1 64137,C=C1CCN(C(c2nocc2CC)=O)C(C(N2CCCC(O)C2C)=O)C1 64138,C(=O)(CC(F)(F)C(F)(F)F)N1CC2C(N3CCCC(OC)CC3)C(CC2)C1 64139,N1(C(C(Cc2cc[nH]n2)NC(COCCC)=O)=O)CCCC(C2CCC2)C1 64140,Cn1cc(N)c(-c2nc(CCn3nccn3)nn2-c2ccccc2)n1 64141,c1(OC(CNC(C2(Br)CC2)=O)C(=O)O)ccc2c(c1)OCCO2 64142,Cc1ccc(Br)c(Cc2nc(-c3ccco3)nn2Cc2cccnc2)n1 64143,C1(NC(C(c2ccccc2)OCC)=O)CCN(C(c2cnc(Cl)nc2)=O)CC1 64144,C1(F)(C(=O)OC)CCCN(C(=O)NCC(c2ccc(O)cc2)O)C1 64145,c1(C(C)C)cc(C(N2CCC(CNC(c3ccnc(Cl)c3N)=O)C2)=O)cc(O)n1 64146,c1(C(N(CC(C)NC(=O)C#CC2CCCOC2)C)=O)ccc(Cl)cc1[N+](=O)[O-] 64147,c1(OCC)c(NC(=O)NC2CCCC(c3ccc(Cl)cc3)C2)cccc1F 64148,N12CCC(C(F)C1)C2=O.C(=O)(C(C(C)C)SC(C)C)NCCN(S(CC)(=O)=O)C 64149,N#Cc1ccnc(N2CCN(C(=O)Nc3ccccc3C3CCCCC3)CC2)c1 64150,C(=O)(CC(CC)NC(=O)C=CC1CCCC1)NCC(CC)OC 64151,Cc1ccc(C=CC(=O)NC2(C)CCN(C(c3cc(C(C)(F)F)on3)=O)C2)nc1 64152,N1(C(C2(c3cnc(SC)s3)CC2)=O)CCc2c(-c3ccccc3)cccc21.C(C)=O 64153,c1(NC2CN(C(CC(C)C3CC3)=O)C2)ncnc(CN(C)C)c1[N+](=O)[O-] 64154,C(=O)(C1CC=Cc2ccccc21)NC1CC(NC(c2c(C)nccc2)=O)C(O)C1 64155,N1(C(c2cc(CC(C)C)on2)=O)CC(CNC(c2nsnc2O)=O)CC1(C)C 64156,Cn1c(=O)n(C)c2c(C(N3CC(CO)(NC(=O)COCCF)C3)=O)cccc12 64157,N1(C(CC(CNC(c2cc(CCC)on2)=O)O)=O)CC(C)C12CCOCC2 64158,CC1CC(C#N)CN1.C1(n2cc(C34CC(C(=O)N)(C3)C4)nn2)CC2C(C1)C2(F)F 64159,c1(SCC)cccc(C(=O)NC2CC2NC(=O)CCSC)c1 64160,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(OC)n[nH]2)=O)cncc(Cl)c1Cl 64161,C1(NC(=O)COC2CCCC2)COC2(C1)CN(C(=O)C=CBr)C2 64162,C(CC(F)(F)F)CC=CC(=O)N(C)CC=CC(=O)N(C(=O)CCn1cccn1)C 64163,C1(NC(c2ccc(CC)s2)=O)CCCN(C(=O)C(C)(C)N2CCOCC2)C1 64164,N1(C(C(C)n2cnnn2)=O)CCC2(CC1)CCN2C(c1ccccn1)=O 64165,C1(C(=O)NCC2C(NC(c3c(CC)nco3)=O)CC2)CCCCN1N=O 64166,C(c1ccc(Cl)s1)=CC(=O)NC(CNC(C=CCN(C)CC)=O)(C)CO 64167,c1(CN(CCNc2ccc[n+]([O-])c2)CC)cccc2c[nH]nc12 64168,C1(NC(CC(=O)NCC)=O)COCCN(C(C2CCCN2C2CCCC2)=O)C1 64169,c1(OC)ccccc1C(F)(F)C(=O)NCC1C=CC(NC(=O)C=NOC)C1 64170,CN1CCC(=CC(N2CC(N(C)C(c3ncccc3Cl)=O)C(O)C2)=O)CC1 64171,CC1(C)CC(C(=O)N2CCC(NC(c3ccc(C(F)(F)F)nn3)=O)C2)=NO1 64172,c1(N2CCCC(C)(C)C2)nc2c(c(=NCCc3cc(F)c(F)c(F)c3)[nH]1)COC2 64173,C1(CC=C)(NC(c2cccc3c2CCOC3)=O)CC2CN(c3ncccn3)CC2C1 64174,Cc1nc(-c2ccc(C(=O)N(C(C)CNC(c3cnns3)=O)C)cc2)[nH]c1C 64175,Cc1cc(Cl)cc(C)c1O.C1(OC(CNC(CCC(=O)N)=O)C2CC2)CCCCC1 64176,CCS(=O)CC(=O)NCC(N1CCN(C(=O)C(C)(C)C2CC2)CC1)C(F)F 64177,N1(C(=O)NC(CCCOCC)C)CCN(C(=O)CNC(=O)C(C)(C)C)CC1 64178,c1(CC)noc(CCCC(=O)NC(C)CN(C(=O)CC#N)CC)n1 64179,CC1(C=CC(=O)NCC2CN(C(C3(CCF)CC3)=O)CC2(F)F)CCOCC1 64180,CCCC(C(=O)N(C)CCOCCNC(c1cncc(OC)n1)=O)S(N)(=O)=O 64181,C(=O)(C(c1ccco1)NC(=O)CC1CCOC1)N(C)CC1CCCS1 64182,N1(C(C(C)=CCC2CC2)=O)CCC(OCCNC(=O)Cc2cccnc2)C1 64183,C(C1CC2(CCC2)C1)SC.N12CCC(O)C1CC(N1CCCCC1)CC2=O.C1CN1 64184,N1(C(C(CC)C)=O)CCCC(C)(NC(=O)CCc2cccnc2Cl)C1 64185,N1(CCOC(C)C)CCc2cc(OCc3ccccc3C(F)(F)F)ccc21 64186,C(=O)(CC(O)C(Cl)(Cl)Cl)NCCN(C(=O)C(O)C1CCCC1)CCC 64187,C1(C)(C(N(C2CCCCC2)C)=O)CCCC1NC(=O)CNC1CC2(CSC2)C1 64188,C1(C(N2CCC3C(CCN3Cc3nccnc3Cl)C2)=O)CCCC2CCCCC12 64189,c1(OC)ccc(C=CC(=O)NC2CC(O)CN(C(c3ccc(F)o3)=O)C2)cc1 64190,c1(C(N2CC(c3cn(CC)nc3)C(C)(C)C2)=O)ccc2ccccc2n1 64191,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)C2)=O)cnn2ccc(O)nc12 64192,C(CCN=C(NCC1COc2ccccc21)N1CCC(F)C1)SC 64193,C1(C(=O)NCC=CCNC(c2c(C(C)(C)C)[nH]cn2)=O)CN2CCCC1(C)C2 64194,C1(C(=O)OCC)CC(S(C)(=O)=NC(=O)CCc2cc(OC)ccc2OCC)CCO1 64195,CC1=C(C(=O)N2CC(NC(C3(O)COC3)=O)CC23CCC3)C(=O)OC1(C)C 64196,c1(C(=O)NC(CC)CNC(C2CC2OC(C)=O)=O)cc(C#N)[nH]c1C 64197,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(c2n(CC)ccn2)=O)C(N=[N+]=[N-])C1 64198,c1(C(N2CCN(CC3CC3)CC2)C(=O)NCC)c(C)nn(-c2ccccc2)c1Cl 64199,C(=O)(C(C)(C)C1=CCSCC1)NCC1N(C)CCN(C(c2csc(O)n2)=O)C1 64200,c1(C(N2CCN(C(COCCOCC)=O)CC2)=O)cc(C)c(O)c(N)c1 64201,Cc1nc2ncccn2c1C(N1CCC(NC(C2CCOCC2)=O)C(O)C1)=O 64202,c1(CC)cnoc1C(=O)N(CCC(=O)NCc1csc(C)c1)C 64203,c1(NC)ccc(C2CC2)cc1.C12(CCN(c3nc(C4CCCC4)ns3)C1)CC(=O)N2 64204,c1(OC)cccc(C(O)C(=O)N(C)CC2COCCN2C(c2cnc(O)o2)=O)c1 64205,N1(C(CCc2nnc(CSC)o2)=O)CC2CC(NCC3(C)C=CCCC3)C2C1 64206,N1(C(C(C)CNC(C2CCC(=O)N(C)C2)=O)=O)CCC12CCCSC2 64207,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)(C(C)C)NC(c1c(C)n(C(C)C)nc1)=O 64208,N1(C(c2ccc(C)o2)=O)CCC2(NC(c3c(Cl)c(C)nn3C)=O)CCCCCC12 64209,N1(CC(=O)NC2CCC2)CCN(Cc2cccc(Br)c2)CC1 64210,C1(CCOC)(NC(=O)CN(C)C)CCN(C(C(C(=O)NC2CCOCC2)CO)=O)C1 64211,C1(NC(C(C)N(CC)CC)=O)CN(C(c2cc(CO)[nH]n2)=O)C2CCCC12 64212,CC1CC(C(N(C=O)Cc2ccccc2C2CC2)=O)C1(C)C 64213,C(=O)(CC(O)CC(C)C)Nc1c(C)cc(NC(C2C3C4CCC(C4)C23)=O)cc1 64214,N1(C(C(CC)(C)C)=O)CCc2c(c(CNC(C3(F)CCOCC3)=O)nn2C)C1 64215,c1(C(N2C(CN(C(c3coc(C#N)c3)=O)CC)CCC2)=O)ccc([N+](=O)[O-])c(C)c1 64216,C1(C(=O)NC2COCCN(C(=O)C3=CCCC3)C2)CCn2nnnc2C1 64217,CCCC(C)C(=O)NC(CN(C(=O)CNC(c1cccc(C)c1)=O)C)(CO)CO 64218,c1(OC)ccc(C(N2CC(OC)CC2CNC(=O)C(F)=C2CCC2)=O)c(O)c1F 64219,CC(C)CC(CC(=O)NC1C2CCCCC12)NC(C1CCCSC1)=O 64220,c1(C(=O)NCCN(C(CCCC(C)=O)=O)C2CCCC2)[nH]c2c(c1C)CCCC2 64221,c1(C(=O)OCC)sc(C)cc1NC(=O)NC1CC(C)CO1 64222,c1(C(C(=O)NCCC)N(CC(=O)OC(C)C)C)cc(OC)ccc1Br 64223,c1(C(=O)NCCC2CCN(C(=O)CCn3cncn3)CC2)c(F)ccc(Cl)c1Cl 64224,c1(NC2C(C)CN(C(C3CCCN3S(C)(=O)=O)=O)CC2C)ncc(C#N)cc1F 64225,C1(C(N2CC(C)OC(C)C2)=O)CC12CCN(Cc1cn[nH]c1)CC2 64226,O=C(C1=CC2CCC(C1)C2)NCC1(F)CCN(C(=O)C(O)CN2CCCC2)C1 64227,C1(CC(=O)N(C2CCC2)CCNC(C)=O)CCC(N(C)CCO)CC1 64228,N1(C(C(c2cn(C3(C)C(C)CCCC3)nn2)(C)N(C)C)=O)CCc2cccnc2C1 64229,C1(NC(c2c(CC)nc[nH]2)=O)CCC(NC(C2(C)CC=CCO2)=O)CC1 64230,C1(CC(=O)N(CCOCC(=O)NC2CCSCC2)C2CC2)CCCOCC1 64231,CC1CCC(CNCc2ccccc2)C(=O)N1.C1CC2(C1)CC(N)C2 64232,c1(-c2ccc(CNc3ncc(C(=O)OCC)cn3)s2)c[nH]c2ncc(OC)cc12 64233,C(=O)(CC(F)(F)F)NCC1CC(F)(CNC(CCCc2onc(C)n2)=O)C1 64234,C(=O)(CS(C)(=O)=O)NCc1c(CCNC(CC(C)F)=O)ocn1 64235,CC(CCCNC(C1(Cl)CC1(F)F)=O)NC(=O)C(C)(C)Oc1ccccn1 64236,c1(COCC)nc(-c2ccnc(C)c2)n(-c2cccc(F)c2)n1 64237,C1(C(=O)NCCN(C(=O)CCOCC(C)C)CC)(OCC)CCCCC1.C1(C)CC1 64238,N(C1c2cc(F)c(F)cc2CC1C)C(C(C1CCCCCC1)C)=O 64239,C1(C(N2CC(NC(C(C(C)(C)C)SC)=O)C(O)C2)=O)=CC(F)=CC(=O)CC1C 64240,c1(C(c2sccc2Cl)C(=O)NCCNC(C2CC(C)(F)C2)=O)ccc(F)cc1 64241,N#Cc1ccc(C(=O)NC2COCC2NC(=O)CCc2ccncc2)cc1F 64242,c1(CC(=O)NCC(C)NC(c2cn(C)ccc2=O)=O)c(F)cncc1Cl 64243,C1(=CC(N2C(C(C)NC(CCc3cnc(C)o3)=O)CCC2)=O)CCCCC1(C)C 64244,C=CC(C)C(C)C(=O)NCCCN(C(=O)C(C)(C)F)C1(C2CC2)CC1 64245,C12CCN(CC1)C2=O.C(=O)(CC(O)C1CC1)N(CC(c1ccccc1)N(C)C)C 64246,CCC(C)CC(C(=O)N1CCC(O)C(C)(C)C1)NC(=O)CC(C)N(C)C 64247,N1(C(C2(CC)CCOCC2)=O)CCOC2(CCN(C(C3CCSC3)=O)CC2)C1 64248,C1(C(=O)NC2CC(NC(C(C)=CC)=O)C23CCC3)CC2CCC(C1)C2=O 64249,N1(C(CN)=O)CCN(C(C2C(C)(C)C2)C2CC2)CC1.c1nnnn1C1CCC1 64250,c1(CC)ccc(CN=C(NCCSC)NC2CC2C2CC2)cc1 64251,c1(CN2CC(C(=O)Nc3c(OC)ccc(Cl)c3)SCC2)cc2ccoc2cn1 64252,c1(C(=O)NCC2CCCN(C(C3CCC(F)CC3)=O)C2)ccc2cccnc2n1 64253,c1(C(=O)NCC2C(NC(=O)CCC3CCOC3)CC2)cc(F)cc2nn[nH]c12 64254,n1(C(C)C)nccc1SCC(=O)NC(c1ccccc1)c1cccs1 64255,N1(CC(=O)NC2CC(F)(CNC(C(C)C3CC3)=O)C2)CCC(O)CC1 64256,C1(NC(c2n(CC)nnc2)=O)(CF)CCN(C(=O)CN2CC3C=CC2C3)C1 64257,c1(C(=O)NCC(CNC(C2NC(=O)OC2)=O)C(F)(F)F)cnc2c(c1)CCCO2 64258,C12(NC(c3n(C(C)C)ccn3)=O)CCCCC1(CNC(C13CC4CC1C3C4)=O)C2 64259,c1(N(C)CC2COCCO2)ncccc1S(=O)(=O)N(C)Cc1c(C)ccs1 64260,C1(OC)CC(CC(=O)NC2CC(O)(CO)C2)N(C(C2CC2(C)C)=O)C1 64261,CC1=CCC(C(=O)NCCNc2cnc(F)cn2)CC1 64262,CCC(CN(CCNC(C1CC12CCC2)=O)CC)CC(=O)NC 64263,C(CCCCC(=O)NCC1(NC(=O)CCC2CC2CC2CC2)CCOC1)=CC 64264,N1(C(c2ccc(C)s2)=O)CC2(CCOCC2)CC1CNC(=O)CC(C)C 64265,CCC(C)CCCC(=O)N1CC2C(CN(C(=O)CSc3ccc(F)cc3)C)C2C1 64266,C(=O)(C(C)CC(C)(F)F)N1CCC(O)(c2cccc(C)c2)CC1 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64285,c1(C(N(CCCNC(=O)C=CC2CCOC2)CCC)=O)cccc(Cl)c1 64286,C1(CNC(COCC)=O)CCC12CCN(C(=O)C(c1cccc(C)c1)=O)CC2 64287,c1(N2CCC(CCC)(NC(=O)C(COC)OC)CC2)cnc2ccccc2n1 64288,c1(OCCCCCNC(CN(C)C)Cc2nnnn2C(C)(C)C)cccc(F)c1 64289,CC1OCCN(C(C2C3CCC(F)(F)C23)=O)C1C(N1CC2(CC(O)C2)C1)=O 64290,O=C(Cc1cccc(OCCF)c1)N=c1[nH]n(-c2ncccc2Cl)c2ccccc12 64291,C#CC1CCN(C(c2cc(OCC)ns2)C(=O)NCCC2CC2)C1 64292,C(N=c1cc(C)nc(Cl)[nH]1)c1c(CNC(C(C(CC)O)C)=O)cccc1 64293,C1(OC)CCN(C(=O)CC(C)(C)C)C1NC(=O)CCCN(C)C(C)=O 64294,C(=O)(CC(Cc1ccc(C)cc1)NCc1nc(-c2ccc(Cl)cc2)no1)OC 64295,CC(C(=O)N1CC(O)CC1CC(=O)N(CC(C1CCCC1)O)C)C(F)(F)F 64296,c1(C(=O)NCCC2CCCN2C(=O)COCCF)cc2ccc(Cl)c(F)c2[nH]1 64297,c1(C(N2C3CN(C(C4CC(=O)NCC4)=O)C(CC3)C2)=O)c(Cl)ccc2c[nH]nc12 64298,C1(C)(C(=O)Sc2ccccc2Br)CCN(Cc2cn(C(C)CO)nn2)CC1 64299,C(C)(CO)(C(=O)N1CCC1(C)CC(=O)NCC1C=CCCC1)OC 64300,C1(NC(=O)C(c2ccccc2)O)CC2CC1CN(C(C1(F)CCCC1)=O)C2 64301,C1(C)(COC(C)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1C.C(CC(=O)NC)O 64302,n1(CC(=O)NCC#CCNC(C2CC(C)SCC2)=O)ccc(=O)n(C)c1=O 64303,c1(C(C(=O)NC(CC)(C)CNC(C2(OC)CCC2)=O)O)cccc(Cl)c1 64304,C1(NC(C(CO)NC(C(C)C)=O)=O)CCN(C(=O)CNC=O)C12CCC2 64305,N1(C(c2c(CNC(C3CC(=O)NCC3)=O)ccs2)=O)CC2COCC(C2)C1 64306,Cc1c(NC(=O)N=c2nc(C3CCCOC3)[nH]s2)oc2ccccc2c1=O 64307,NS(=O)(=O)CCCCCCC(=O)NC1CC1NC(=O)C(c1ccccc1F)F 64308,c1(C(=O)NC(C)CC(C)NC(=O)CCC2CC2(C)C)ccncc1Cl 64309,N1(C(C2CCCN(CC)C2)=O)CCN(C(c2cccnc2N)=O)C(CC#N)C1 64310,c1(CC)cc2c(N(CCNC(c3ccnc(Cl)c3F)=O)CC)ncnc2s1 64311,Cc1scc(CC(C(O)CO)NC(=O)NC2(c3ccccc3)CCC2)c1C 64312,S(=O)(=O)(c1cccc(N2CCCOC(C)C2)n1)NCC(C1CCCCC1)OC 64313,N1(C(CCCOCC)=O)CCN(Cc2cn(CCOC3CCOC3)nn2)CC1 64314,Cc1n[nH]c(C)c1C(=O)N(C)Cc1ccccc1CNC(C1C(C)(C)C1(C)C)=O 64315,C1(C(=O)NC(C2CC2C(=O)NC(C)(C)CCF)C)C(O)C2CCOC12 64316,C12(C(=O)NC(CCOC)C)COC(C1)C(NC(=O)C=CC1CCCCC1)C2 64317,C1(C(=O)NC2CC(CN(C)C)C2)CCC2(CC2)N1C(=O)CC1CCC(=O)NC1 64318,CCC(C)C(CC(=O)Nc1c(OC)cccc1C)NC(=O)C(C)C(=O)OC 64319,c1(C(N2C(CNC(c3cn(C)nn3)=O)CCC2)=O)c(O)cccc1O 64320,N1(C(C(C)C2CC2)=O)CC(O)CC1CNC(=O)CC(=O)NC(=O)C=CC1CCCC1 64321,CC1CC(c2nc(Cc3ccc(C(C)(C)C)cc3)nn2C)=NN1C(c1ccccc1)=O 64322,N1(C(CCCC#CC)=O)C2CCC1C(C)C(NC(=O)C=CC(C)(C)SC)C2 64323,c1(C(=O)NCCC(C(C)C)NC(CNC(COC)=O)=O)cccn2[nH]c(=N)nc12 64324,c1(C(=O)NCCC(C(C)C)NC(C=CSC)=O)cc2cccc(F)c2o1 64325,CC1CCC(C(N2CCN(C3CCN(C(C4SCCS4)=O)CC3)CC2)=O)NC1=O 64326,N1(C(C(c2cn(C)nn2)NC(CN(C)C(N)=O)=O)=O)CCC=C(Cl)C1 64327,c1(C(=O)NCC(C)NC(c2ccc(NC(C)=O)cc2)=O)sc2ccccc2c1C 64328,CCC(C)(CCC(C)C)C(=O)N1CCC(CF)(NC(=O)CC2(O)CCCC2)C1 64329,c1(OC(C)C(=O)NC2CCC2NC(c2ccc(N)c(N)n2)=O)ccc(F)c(F)c1 64330,N1(C(c2ccc(CNC(c3scc(OC)c3)=O)cc2)=O)CCC2C(C(N)=O)C2C1 64331,c1(C(c2n(CC(=C)C)nnn2)NC(C(C)C)C2CC2)cnc2cccnn12 64332,CC1(C)CCCC(CC(=O)NC(C2CN(C(=O)CSc3ccccc3)C2)(C)C)O1 64333,CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CN2CSCC2=O)CC1O 64334,c1(N(C)C)ccc(CNC2CNC(=O)C2)cc1S(=O)(=O)NC1C2CCC(F)(F)C12 64335,c1(C(=O)NCc2ccc(NC3CCO3)cc2)ccc(CC)c([N+](=O)[O-])c1 64336,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CCCN(C(C3CNC(=O)N3C)=O)C2)C1 64337,c12cnc3[nH]c(cc3c1)N(C)CC(=O)c1cc-2ccc1F.C(C1CC1)OC.OC 64338,N1(C(C2C(F)(C(=O)OC)C2)=O)CCOC2(C1)CN(C(c1ccnnc1O)=O)C2 64339,CC1CC(NC(C2CCO2)=O)CN(C(=O)C(F)(F)C(F)F)C1 64340,Cc1cnc2c(cnn2CC(=O)NC2CCCN(C(c3cccs3)=O)CC2)c1 64341,c1(CC(=O)N(C2CC2)CC2N(C(C(C)OC)=O)CCCC2)cccc(Cl)c1OC 64342,c1(NC(=O)OC)ccccc1C(=O)NCC(CC)N(C)C(C1CC1C(C)C)=O 64343,c1(CNC2CN(CC(N3CCC(CC(=O)OC)C3)=O)C2)ccc2c(c1)COC2 64344,C(c1cc(C)cc(C)c1)=CC(=O)N(CCN(C(C(C(C=C)C)C)=O)C)C(C)C 64345,C1(NC(c2oc(C)c(CO)c2)=O)C2CC3C1C3C2C(N1CCC(C)C1)=O 64346,CCC(C)(CO)C(=O)N1CCCC(N(C)C(c2ccc(COC)c(N)c2)=O)C1 64347,c1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)COC2)cc(C)ccc1Cl 64348,CC1(C)CC(NC(C2C(O)CCN2C(=O)CC#N)=O)C12CCC2 64349,Cc1ccc(CCC(=O)NCC2CCC2CNC(=O)CCC(=O)N(C)C)cn1 64350,c1(C(N2CCOC(C)(CC)C2)C(=O)NCCOCC)ccc(C)c(I)c1 64351,C(=O)(C1=NOCC1)N(C(CCNC(C1CC(CC)C1)=O)C)C 64352,N1(C(=O)CC2CC=CCC2)CC2=C(C1)CN(C(=O)CC1CCC(F)(F)C1)C2 64353,Cc1cn2cc(C(=O)NC(C)CN(C)C(C3CCc4nncn4C3)=O)ccc2n1 64354,N1(C(COCCCC)=O)CC(NC(=O)C(C)(C)CF)C(SC)C1 64355,c1(NCCOCCC)nc2ccc(OCC(=O)OC)cc2s1 64356,C#CC(C)(C)C(=O)NCCC1CN(C(=O)CC(C)(C)O)CC1C 64357,c1(C(=O)NCCN(C(c2nc(C(C)(F)F)cs2)=O)CC)cc2c(nc1O)CCCC2 64358,c1(CC)[nH]c(C(=O)NC(C)(CNC(C2CCOC2)=O)c2cccs2)nc1Cl 64359,O=C1CC(C(=O)NCCC2COCCN2C(C2CC(O)(C(F)(F)F)C2)=O)CCN1 64360,CCCCCCCNC(=O)C(C1CCCO1)NC(=O)C=C(C)C(C)C 64361,C1(NC(C2CCC(CC)CC2)=O)CN(C(C2CC2(C)CC)=O)Cc2nccn2C1 64362,Cc1ccccc1C=CC(=O)Nc1nnc(CC(=O)Nc2cccc(F)n2)s1 64363,C(CN=C(NC1CC1(c1ccc(C2CC2)c(F)c1)C)N1CCC(C)(C)C1)OC 64364,C1(C(=O)NC(CC(C)C)CNC(=O)Cc2cnoc2)CCc2cn(C)nc2C1 64365,C(=O)(CCCCC(N)=O)N1CCN(C(c2c(F)ccc(N(C)C)c2)=O)CC1CF 64366,N1(C(C(C)C)=O)CCC(C2CCN(C(=O)C(F)C3CCC3)CC2)C1 64367,c1(C(=O)NC2C(C(N3C(C)COCC3)=O)CCC2)cc(I)ccc1F 64368,Cc1[nH]cc(NC(N2CCCC2CSc2ccc3c(c2)CCC3)=O)c(=O)c1Cl 64369,c12cn(nn1)Cc1ncoc1-2.C(=O)(C(C)(C)C)NCC(=O)N(C)CCO 64370,C(CCCCNC(C1CCCC1Cc1ccccc1)=O)OC 64371,C(=O)(CCCCCC(C)C)NCCCN(C(C=Cc1c(C)noc1C)=O)C1CC1 64372,C(CCCCC(=O)NC1(C(=O)NC(C)(C)COCCSC)CCSC1)OC 64373,C1(=O)NNC(=O)c2ccc(cc2)CN1.CCC(COC)CO 64374,CC1(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1NC(=O)CCc1nc[nH]n1 64375,N1(C(CN2CCCC(CC)C2)=O)CC(CNC(=O)Cc2c[nH]nc2C)CC1(C)C 64376,c1(C(N2C(C)(C(N3CCN(C)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 64377,Cc1cc(CN2CC3CC3(C(=O)Nc3cc(C(F)(F)F)c(Br)cn3)C2)ccc1Br 64378,c1(-n2cc(C(=O)NCC3C(C)CCC3C)nn2)cccc(F)c1Cl 64379,C1(NC(=O)C2=CCN(C(c3ccc(CO)s3)=O)C2)CC2CCCC(C1)C2 64380,CC1CC2CC(C(=O)NC3CCCC3(C)NC(=O)Cc3c[nH]nc3O)(C2)O1 64381,c1(OC)cncc(C(=O)NCCC(C)NC(=O)C(O)CCc2ccccc2)c1 64382,c1(C(=O)N)c(OCC2CC2OC)cccc1F.N1(CC)CCC(C(=O)CCN)CC1 64383,Cc1cccc(C(=O)N(CCCCCNC(c2cnn(C(F)F)c2)=O)C)c1O 64384,N1(C(C(CC=C)(F)F)=O)CCCCCC(NC(C2(C)CCC(F)(F)C2)=O)C1 64385,Cc1ccc(C)n1CC(N1CC(O)(C(C)NC(c2cnn(C3CC3C)c2)=O)C1)=O 64386,N1(c2n(CC)nnn2)CCC(CCCC)CC(C)(C)C1.[nH]1ncccc1=O 64387,C1(OC)(CNC(=O)COC)CCN(C(=O)CCNC(=O)OC2CC(F)(F)C2)C1 64388,c1(C(=O)NC(CC#C)(C)C(=O)NCCCN=[N+]=[N-])ccc2cc[nH]c2n1 64389,N1(C(c2c(C#C)c[nH]n2)=O)C2CCC1CC(F)(CNC(C1(O)CCOC1)=O)C2 64390,Cc1cc(C)[nH]c(=NCc2cn(C)nc2CNC(=O)CC2CCCC2C)n1 64391,N1(C(Cc2c(Cl)cn(C)n2)=O)CC(NC(=O)Cc2cncs2)C(C2CC2)C1 64392,Cc1cc(=O)n(C)nc1C(N1CCCCC1C(C)NC(=O)C(C)(Cl)Cl)=O 64393,c1(C(N(CCCCN(C)C(C2CCC2)=O)C)=O)n[nH]c2c1CCCCC2 64394,Cc1nn(CCc2ccccc2)c(C)c1C(N1CC(C)CCC1C)=O 64395,Cc1ccc(O)c(NC(=O)CCC(C)(C)NC(C2CCCCO2)=O)c1 64396,C1(CC#C)(NC(=O)CCc2ccsc2)CCN(C(=O)COCCCF)C1 64397,N1(C(=O)Cc2ccc(O)cc2)CCC(CO)CC1CNC(C12CC3CC1C2C3)=O 64398,C1(C(=O)NCc2c[nH]nc2NC(C23CCCC2(C(=O)OC)C3)=O)(CC)CCOCC1 64399,N1(C(C(CCS(C)=O)O)=O)CCN(C(c2cnns2)=O)C2(CCC2)C1 64400,C(CCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1)NC(C)=O 64401,C1(CNC(Cc2cc(OCC)no2)=O)CC2COCC2N1c1cccc(F)c1 64402,CCCC(C)CC(=O)NCCC1CCN(C(c2cc(C)nc(OC)n2)=O)C1 64403,N1(C(C2C(=C)CC2)=O)CC(CCn2cc(-c3c(Br)cnn3C)nn2)C(C)C1 64404,Cc1cc(O)nc(C)c1C(=O)NCC(c1ccccc1)CNC(=O)CC#N 64405,c1(C(=O)OCc2ccc(-c3ccc(OC)cc3)nc2)cnc(Cl)cc1F 64406,CC#CCC(C(=O)NC(c1cn(C)nc1C)C)NC(c1cn(C(C)C)nn1)=O 64407,C1(NC(=O)CC2CC3(CCC3)C2)CCN(C(=O)CS(=O)(=O)CC2CCCO2)CC1F 64408,C(CC(C(=O)NC1CC(n2cccn2)C1)NC(C1COC(C)C1)=O)SC 64409,C1(CNC(=O)CC2CC2C2CC2)CCCN(C(=O)Cc2ccsc2)CC1 64410,Cc1cncc(CC(N2CC(=O)CC2C(=O)NCc2cnc(C(C)C)[nH]2)=O)c1 64411,c1(CC(c2n(CC=C)nnn2)NCC(C)C)ccc(OC)cc1OC 64412,c1(C(=O)NC2COCCN(C(C(C)(Cl)Cl)=O)C2)cccc2cnsc12 64413,S(=O)(=O)(c1ccc(Cl)cc1)NC1CCN(C(c2ccc(Cl)nc2O)=O)CC1O 64414,Cc1ccc(C(N2CC(NC(=O)C(C(C)C)NC(=O)NCCC)C2)=O)c(C)c1 64415,Cn1ncc2c1CN(C(=O)C1=CCN(C(=O)NC3CC3c3ccccc3)C1)C2=O 64416,C12CC(C1)NC(=O)COC2.C1(C(N)=O)CCOC1.C12(CC1)C(=O)N2 64417,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64418,C1(C(=O)NC(CCC(C)C)C)CC1C1CN(C(C2(O)CCCC2)=O)C1 64419,CCC(C(=O)NCC1(O)CN(C(=O)CC2CCC(O)C2)C1)SC 64420,c1(C(=O)NC2C(C)CN(C(c3cccnc3Cl)=O)C2)cn2cccc(Br)c2n1 64421,c1(CCCCN)cc2ncccc2[nH]1.CC(C)(C(=O)N1CCCC1)c1cn(C)nn1 64422,C1(CN(C[Si](C)(C)C)CC)CCCN(S(N)(=O)=O)C1 64423,CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CCO1 64424,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3c(N)sc(C)c3C)=O)CCC2C1 64425,N1(C(C2CC(Nc3ccn4ncc(Br)c4n3)C2)=O)CCC2(CCNC2=O)CC1 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64443,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64444,CCC(C)(C)C(C)(NC(c1csc(Br)c1)c1nnnn1-c1cnn(C)c1)SC 64445,C(C(C(=O)NCCOCC(CC)CC)C1CCCCC1)OCC 64446,C1(C(=O)NC(C(=O)NCCOCC)Cc2cn(C)nn2)(OC)CCC(C)C1 64447,N1(C(C2CC(C)C2)=O)CC(NC(c2c(-c3cccs3)cnn2C)=O)CC2(CC2)C1 64448,c1(OCCCC)n[nH]cc1CN(C)C(C1CCCO1)=O 64449,c1(N(C(=O)NCCC2(OC)CC2)CC)csc(NC(=O)OC(C)(C)C)c1 64450,c1(C(=O)NC(C(C)NC(c2cc(OC)ns2)=O)C)cccc(C(C)(F)F)n1 64451,N1(C(C(C(C)(C)C)NC(C(COC(C)=O)C)=O)=O)CC2(CNC(=O)N2)C1 64452,N12CC3CCN(CC3C1)C(=O)COC(=O)C1(CCC1)CC2=O.C1(C)(COC)CCC1 64453,C1(C)(CNC(Cc2ncc(C)o2)=O)CCCN1C(c1csc(Cl)n1)=O 64454,C1(CC(=O)NC)CCN(C(=O)CC2CCC2)C(C)C1.C12CCN(C1)C2=O 64455,N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)CC1C1CC1 64456,C(=O)(C(O)CC[S+](C)C)NCC(C)(C)NC(CN(c1cccc(Cl)c1)C)=O 64457,N1(C(C2(C=C)CC2)=O)CCc2c(CNC(=O)CCCSC)cccc2C1 64458,C1(CC(=O)OC)(C(F)(F)F)CC2CC2C1.C1(=O)CC2(CC2)N1CCN.N(C)C 64459,C(=O)(C(C)(F)C(C)(C)F)N1CCC(NC(C(C(=C)C)(C)C)=O)CC1C 64460,C1(NC(CCOCC)=O)CCCCCC1C(=O)NCCC1CCSC1 64461,Cc1ccc(-c2ccc(CN(CC(O)CO)C)cc2)cc1F 64462,C1(C(=O)NCC2(OCC)CC2)CCCCN1C(C1(C)CCC(=O)N1)=O 64463,c1(C(N(CCCCNC(CC2C(OC)CC2)=O)C)=O)cnn(CC(F)(F)F)c1C 64464,c1(CC)ccc(C(N2CCC(OCCNC(=O)C(C)CO)C2)=O)cc1C(F)(F)F 64465,C1(N(C(=O)NC(C)CC2CCC2)CC)CCC(C(c2sccc2Cl)C)CC1 64466,n1(CC)c(C(=O)NCC2CCN2C(=O)CCCC(C)=O)cccc1=O 64467,c1(CN(C(=O)NC2C(CCC)CCC2)CC)nccc(=O)n1C 64468,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(C3CCCO3)=O)C2)CC1 64469,N1(CC(N2C(C(=O)O)CCC(F)C2)=O)C(=O)C(=O)N(Cc2ccccc2)C1=O 64470,CC1(C)CC(C)(CO)CN1C(C1CC(=O)CN1C(C1(C(C)(C)O)CC1)=O)=O 64471,Cc1cncc(NC(C2C=CCN2C(c2nnn(C)c2C(F)F)=O)=O)c1 64472,C1(C(N2C(CCC=C)CCC2)=O)CC(O)CN1C(C12CC(CO)(C1)C2)=O 64473,N1(c2snc(C(C)OCC)n2)CCC2CC(CNC(=O)C=CCF)CCC2C1 64474,N1(C(CCOCCC)=O)CC(NC(c2[nH]nnc2CC)=O)CC1(C)COC 64475,Cn1cc(Cl)c(C(=O)NCCc2ocnc2CNC(=O)CC2CCC3CC23)n1 64476,c1(CN(C(=O)C(=O)N(C)CC2(O)CCC2)C(C)C)ccc(Cl)cc1 64477,Cc1nc(C(=O)N(C2CCN(C(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)C2)CCO)sc1C 64478,Cn1ccc(=O)cc1C(=O)NC1CC1C(=O)Oc1ncccc1C(F)F 64479,C1(C(=O)NCC(CC=C)(C)C)CCCN(C(C2CCC2(OC)OC)=O)CC1 64480,C(C)(c1cnn(C)c1)=CC(=O)NC(c1ccc(OCC#N)cc1)C(=O)OC 64481,c1(C(=O)NC(c2noc(-c3ccccc3)n2)C)c(Br)cnn1-c1ncccn1 64482,CC(CSc1ccccc1)C(=O)NC1CCC1CNC(=O)CCc1ccc[nH]1 64483,CC1CN(C(c2conc2C2CC2)=O)CC1NC(=O)Cn1nnc(=O)[nH]1 64484,c1(C(C(=O)NC(C2N(C(c3c(OC)n[nH]c3)=O)CCC2)C)O)ccc(Cl)cc1F 64485,S(=O)(=O)(c1ccc(F)c(C(=O)NC(CNC(=O)CC2(O)CCC2)CO)c1)N(C)C 64486,C1(CC(=O)NCCN2CCOCC2)CN(C(=O)C=Cc2ccncc2)CCO1 64487,C(=O)(CC(C)CC(C)C)N1CCN(CC(C)NC(C=Cc2ccc(C)o2)=O)CC1 64488,c1(C(=O)NCCC(C)N(C(CCC(=O)OC)=O)C)ccc(C)cc1Br 64489,c1(NC2CCOC2)cc(N2CCN(CCc3noc(C(C)SC)n3)CC2)ncn1 64490,c1(CC(=O)OC)nocc1CNC(C)C(=O)NC(c1ccccn1)C1CCCC1 64491,n1(CC)cnc2nc(=NC(CC)n3ccnc3)[nH]c(N(CC(C)OC)C)c12 64492,N1(C(C(C2CC2)OCC)=O)CCCC12CCN(C(c1c(C)cccc1O)=O)C2 64493,Cc1nc(CC(=O)N(C2CCCN(C(c3ccc(CO)cc3)=O)C2)C)c(Cl)s1 64494,CC(C)C(C(C)NC(c1ocnc1-c1ccccc1)=O)NC(c1cnc[nH]1)=O 64495,Cc1cn2c(n1)CCC(NC(=O)NCc1ccnn1Cc1ccccc1)C2 64496,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64497,c1(NC(=O)NCC2(C)CC(C)(C)C2)ccc2ccc(Br)cc2c1 64498,c1(NC2CC(C)CC(C)C2)nccc(=NCCCCC2CCCCC2)[nH]1 64499,C1(CN(C23CCCCC2C3)C)CCC2(CCCCC2)O1 64500,N1(C(CCOCC)=O)CC(NC(c2nc(C(F)(F)F)sc2C)=O)C2CCCCC12 64501,CC1CCC(CC(=O)NCC2(CN(C(=O)CN3CCNC3=O)C)CC2)C1 64502,c1(C(=O)OCC)conc1C(=O)NCCOC1(C(=O)N(C)CC)CC1 64503,N1(C(c2c(C)n(C(C)C)nc2)=O)CCCC(N(C(=O)Cc2ccnn2C)C)CC1 64504,S(=O)(=O)(c1cccnc1NC1CC1)N(C(C)CCc1ccccn1)CC1CCCS1 64505,C1(C(=O)NC2CC(CCC(=O)N(C)CC3CCSC3)C2)CC2CCC1C2 64506,O=CN1CCN(C(=O)Cn2cc(CNC(C3CCC(=O)C3)=O)nn2)CC1 64507,N1(C(C2C3(CCN(C(C4N(C)CCCC4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64508,CC(F)(F)C(C)(C)CS(=O)(=O)NCCc1cncc(Br)c1 64509,c1(CCNC(=O)Nc2cnn(CC)n2)cccc(OC)c1OCC(F)(F)F 64510,c1(C(N2CC(CNC(c3cncc(OC)c3)=O)OCC2)=O)cn2nc(C)sc2n1 64511,c1(OC)n[nH]c(C(N2CCCC2C2CCN(C(=O)C(C)(C)CF)C2)=O)c1Br 64512,Cc1nc(C)n(CC(N2CCC(C(F)F)(CNC(c3c[nH]nc3Br)=O)C2)=O)n1 64513,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64514,CC1CN(CC(=O)N(C)Cc2ccc(OC(F)F)nc2)Cc2nncn21 64515,CC1OC(C)(C)OC1(C)C(=O)NCc1ncoc1CNC(=O)CCCC(F)(F)F 64516,c1(N2CCC(CC(=O)OC)C2)cc(C)nc(NC(N2CCCC2C(N)=O)=O)n1 64517,Cc1ccc(C(=O)NC(C)CNC(c2cncc(C3CC3)c2)=O)c(C(C)C)n1 64518,C=CC(C)(O)CC(=O)NCCC1(NC(=O)C(C(C)(C)O)OC)CCC1 64519,N1(C(c2c(C)n(C)cn2)=O)C(CC(=O)NCc2nncn2C(C)C)C2CCCC12 64520,N1(C(C(C(C)O)(C)C)=O)CC2(CC(C(N3CCOC(C#N)C3)=O)CO2)C1 64521,C1(CNC(CCCCCC)=O)CC2(CCN(C(C3CC(CN(C)C)C3)=O)C2)CO1 64522,c1(C(CCOCC(F)(F)F)NCC(c2ccccc2Cl)(C)C)cccc(Cl)c1 64523,N1(C(c2cc(CCC)[nH]n2)=O)C(C)CC2CN(C(c3cc(COC)[nH]n3)=O)CC12 64524,C1(C)(C(=O)NCC(N(C(C2C(c3nc(C)[nH]n3)C2)=O)C)C2CC2)CCC(C)C1 64525,Cc1cnc(C(=O)N(C(C)CN(C)C(c2cnc(Br)s2)=O)C)c(F)c1 64526,c1(CNC(C(=O)N(CC(N)=O)C)=O)nc2ccc([N+](=O)[O-])cc2[nH]1 64527,N1(C(c2nc(C)nn2C)=O)CCC(CNC(=O)COCCN(C)C)C1(C)C 64528,c1(CNC2CCC(CC(=O)NC(C3CCCCO3)CC)C2)cc(C#N)ccn1 64529,c1(OCC(N2CCOCC2C2CCCOC2)=O)ccc2nc(Cl)ccc2c1 64530,c1(C(=O)NCC2COC(CNC(=O)C(F)n3ccnc3)C2)ccnc2[nH]ncc12 64531,N1(C(c2cn(CC=C)nc2)=O)CCCOC(CNC(C2CCC(CC)C2)=O)C1 64532,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(c3ccncc3Br)=O)O2)C1 64533,c1(NC2CN(C(c3c(CC)nn(C)c3)=O)C(C)C2)c([N+](=O)[O-])c(C)nn1CC 64534,N1(C(c2ccc(OC)s2)=O)CCC2CCN(C(=O)CCN3CCOC3=O)C2C1 64535,C(=O)(C(CO)C(C)(C)C)N1CCN(CCN(C(c2c(COC)cco2)=O)C)CC1 64536,O=C(C#CC1CCOC1)NC1CC2CCC1CC2NC(=O)CSC(F)F 64537,c1(NC(c2n(C(CC)(C)C)nnn2)(C)C(C)OC)ccc2nncn2c1 64538,C(CCCCCC(=O)N(C)Cc1cc(OC)no1)NC(C(C=C)O)=O 64539,c1(CC)cc(C(N2CC3C(NC(c4cc(C(C)=O)[nH]n4)=O)C3C2)=O)c(C)o1 64540,CC(CC(C)(C)C)C(=O)N1CCCC1C(N1CCC(CC2CC2)CC1)=O 64541,C(N=c1nc2scnc2c(N2CCC3(CCC3)C2)[nH]1)C1(C)C(C)(C)C1(C)C 64542,c1(NC2CC(OCC)C2)nccc(=NC(CC)CC(F)(F)F)[nH]1 64543,C#CC1CN(C(=O)C(C)CC)CCN1C(=O)CSc1nncn1C1CC1 64544,c1(C(N2CC(O)(CNC(C(C)N(C)Cc3ccccc3)=O)C2)=O)nc(=O)n(C)[nH]1 64545,c1(CC(=O)N(CCCNC(C2CCC(C)S2)=O)C(C)C)ccc2ccoc2c1 64546,CC(C(=O)N1CC(N(C)C(c2ccc(CF)cc2)=O)C2(CC2)C1)C(C)(F)F 64547,c1(CC(=O)NC(C)CNC(=O)CC2(CO)CCC2)cccc(N2CCOC2=O)c1 64548,S(=O)(=O)(c1c(C)noc1C)NCc1oc(C(=O)OC)c(C)c1 64549,N1(C(c2c(CNC(C3C(=O)NCCC3)=O)cc[nH]2)=O)CC2(CCC2)CC1CO 64550,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CCSC2)=O)CC1 64551,c1(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)cccc2c1CCCN2 64552,C#CCCCC(C)C(=O)NCC1CN(C(c2ccc(F)o2)=O)C1 64553,c1(C(N(CCCNC(=O)CC(O)C2CCCC2)CC)=O)ncccc1OC 64554,c1(OC)ccnc(C(=O)NC(CO)CC(O)c2ccccc2)c1F 64555,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(c1cc(F)n[nH]1)=O 64556,N1(C(C(C)OC)=O)CC2(CCN(CCc3ccc(F)c(C)c3)CC2)C1 64557,C(=O)(CCN(OC)C(=O)C12CCC(CC1F)C2)NCc1n(CC)ncn1 64558,CC1CC(NC(=O)CC2CC(CF)C2)CN1C(C1CC1(C)C(F)F)=O 64559,c1(C(=O)NC2CCN(C(CC(C)F)=O)C23CC3)nccc2ccsc12 64560,C#CCC(CC(=O)N1CCC(C)=C(C)C1)NC(c1c[nH]c(=NC)s1)=O 64561,C1(C(C)NC(CCOCCOC)=O)CCCN1C(=O)C(C1(O)CCC1)SC 64562,C=CCCC(C(=O)NCC(C#N)CC)NC(c1cccnc1O)=O 64563,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 64564,c1(C(=O)NC(CC=C)CO)cccnc1CNC(=O)C(c1ccnn1C)C 64565,c1(C(N2CC(C(=O)OC)CN(C)CC2)=O)c(F)cc(C(F)(F)F)c(N)c1F 64566,c1(NC(=O)NC2CCN(CCOC)C2)csc2c1CCCC2 64567,c1(OCC(=O)NC2CCC(NC(c3ccn(C(C)(C)C)n3)=O)C2)cccc(F)c1 64568,CC1(NC(c2ccc(-n3cccc3)cc2)=O)CCN(C(=O)C(F)n2cccn2)C1 64569,C1(C(=O)OC)CC(F)CN(C(c2c(C(C(=O)OC)NC3(C)CC3)cnn2C)=O)C1 64570,Cc1n[nH]c(C)c1C(c1ccc(F)cc1)NCC(=O)OCC1CCOC1 64571,c1(N2CC(C(C)NC(=O)CC(c3ccc(F)cc3)O)C2)ccc(Br)cc1[N+](=O)[O-] 64572,C(CCN=c1[nH]c(=NC(C)CC(=O)N(C)C)c2ncccc2[nH]1)(OC)OC 64573,c1(C(=O)NC2(C)CCN(C(C3CCN(CCC)CC3)=O)C2)cc(Cl)c(F)cc1Cl 64574,CC1CCN(C(=O)C(C2CCOCC2)O)CC1NC(c1cc(C(N)=O)cn1C)=O 64575,C(CNC(c1cc(OC)cc(C)n1)=O)(CC(F)(F)F)NC(C(COC)O)=O 64576,c1(CC(=O)NC2C(CNC(Cn3c(C)ncc3)=O)CC2)nc2c([nH]1)CCCC2 64577,C1(CC)C(CC(=O)NC2(C3CCCN3C(c3csc(O)n3)=O)CC2)C1(F)F 64578,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(CC)c(=O)c2)=O)CC1 64579,C(CN1C(=O)Cc2ccccc21)OC(c1cnn(C)c1C1CC1)=O 64580,N1(C(C(CSC)OC)=O)CCCC(C(=O)NOCC(O)C(C)C)(CO)C1 64581,Cc1oc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C 64582,c1(N2C(C(C)(C)NC(c3scc(C)c3Cl)=O)CCC2)ncnc2c1cnn2C 64583,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nnnc1C)C2 64584,C=CCN=C(NCC1(C(=O)OC)CCCC(C)(C)C1)N1CCOC(C)(C)C1 64585,N1(C(COCC=C)=O)CCC(C2OCCC2NC(=O)CNS(=O)(=O)NC)CC1 64586,CCC(C(O)C(C)C)NC(=O)CCNC(c1ccc(Br)cc1)=O 64587,C1(C(=O)NCC2C(NC(C3C(C)(CC)C3)=O)CCC2)Cc2ccccc2N1C 64588,c1(C(CNC(C2CC2CF)=O)NC(C(C)N(C)C)=O)ccc(Br)cc1 64589,C#CCC(CC(=O)NC1CCCC(CC)C1)NC(=O)C(C)(C)CO 64590,C=CCCCC(=O)N1CC2C(NC(c3c[nH]cc3C(C)(C)C)=O)C2C1 64591,N1(C(C(n2cc(Br)cn2)C)=O)CCCCC1CN(C)C(c1c[nH]nc1F)=O 64592,C1(OC)CCC12CC(C(=O)NC(C1CN(C(=O)CC(O)C3CC3)C1)C)C2 64593,CN1CC(C(=O)NCC2CCC(NC(c3ccccc3OC3CC3)=O)CC2)CC1=O 64594,c1(CC)nn(C)cc1C(=O)N(C)CC1CCC(=O)N1 64595,CCC(C)C(C(=O)NCC1=CCN(C(=O)Cn2ccnc2C)CC1)OC 64596,C1(NC(C2(OC)CCN(C(C3CN4CCC3CC4)=O)C2)=O)CN(C)CC1(F)F 64597,c1(C(=O)NCC)cccc(C(N2CC(NC(=O)CC3COCCO3)C(F)C2)=O)c1 64598,c1(OC)ccc(C(C)NCc2ccc(-c3cccs3)c(F)c2)cc1C 64599,N1(C(C2C(CNC(C(C3CCC3)OCC)=O)C2)=O)CCOC(C23COC(C2)C3)C1 64600,c1(C(=O)OC(C(=O)Nc2c(C)ncc(C)n2)C(C)C)cc(C)ccc1[N+](=O)[O-] 64601,c1(C(=O)NCC(CNC(c2c(C)[nH][nH]c2=N)=O)OC)sccc1S(N)(=O)=O 64602,N1(C(CCSCC)=O)CCCC(C)(NC(=O)CCOc2ccccc2C(N)=O)C1 64603,n1(CC(=O)N(CCCNC(=O)CP(C)(C)=O)CCC)cccc(Br)c1=O 64604,C=CCC(CC)C(=O)NCc1cccc(NC(C2CC(NC(=O)C(C)C)C2)=O)c1 64605,C(=O)(CCC(C(=O)NC1CCOC1)N1CCOCC1c1ncnn1C)OCC 64606,C1(C(=O)NCC(CC)NC(=O)CN2CCCC2CO)(COC)CCOCC1 64607,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)C(C1(C)CC1)C)OC 64608,CC1(CNC(=O)CNC(C2CCC2)=O)CCCN1C(c1cc(C(N)=O)c[nH]1)=O 64609,C(C(CO)C(C)C)NC(C1C(C(C)NC(c2c(C)cns2)=O)C1)=O 64610,c1(N2CCN(C)C(CN)C2)nc(N2CCCC(C)(CN(C)C)C2)nc2c1CCC2 64611,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 64612,CC1COc2c(C(=O)NCC(O)CNC(c3ccccc3Br)=O)cnn2C1 64613,CC(C)C(O)CC(=O)N1CCN(C)C(CNC(C2CCC(N(C)C)CC2)=O)C1 64614,c1(CC)cnn(C)c1C(=O)NCCOCC(=O)NCCC1CCCC(C)C1 64615,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C2CCCOC12 64616,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 64617,c1(NCC(=O)N(C2CN(C(C3(C4CCCO4)CCC3)=O)C2)C)ccc(C#N)cc1 64618,c1(C(=O)NCC(CNC(=O)COc2ccccc2)O)cccc2cccc(O)c12 64619,C1(F)(CNC(c2c(Cl)cc(C)s2)=O)CCCN(C(=O)C(O)C2CCC2)C1 64620,S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2ncc(Cl)cc2Cl)C1 64621,CS(=O)(=O)c1cccnc1C(=O)NCC1(CNC(C2CC23CC(O)C3)=O)CC1 64622,c1(NC(=O)NC)ccc(NC(=S)NCCCCl)cn1 64623,c1(CC)cnc(C(C)NC(c2ccncc2)c2nnnn2C(C)C)[nH]1 64624,C=CCC(CC(=O)Nc1cnc(C2CC2)nc1)NC(C1CC(=O)N(C)C1)=O 64625,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 64626,C(=O)(CC(C)P(C)(C)=O)N1CCN(C(c2cc(C)cc(N)c2)=O)CC1CCN(C)C 64627,Cn1c(C(=O)NCC2CC(NC(=O)CC3CCCC(=O)C3)C2)cnc1O 64628,C1(CN(C)C)CC(O)CN1C(c1n[nH]cc1CNC(=O)CC1CC(=O)C1)=O 64629,n1(CCC)ncc(C(N2CCCCC2CCN(C)C(C2CCS2(=O)=O)=O)=O)c1Cl 64630,C1(N(C(CCC=C)=O)CC(F)(F)F)CC2(CCN(C(=O)C=CC(C)C)CC2)C1 64631,COn1cnc(C)c1C(=O)NC(C)C(C)NC(=O)C(c1cc(F)cc(Cl)c1)(F)F 64632,c1(C(=O)NCCN(C(C(C)OCC(C)C)=O)C(C)C)cc(S(C)(=O)=O)ccc1Cl 64633,C#CCCCCC(=O)N1CCC(NC(=O)CCc2cccc(OC)n2)C(F)C1 64634,N1(C(Cc2c(CC)con2)=O)CC(NC(C2CCO2)=O)C(O)C1 64635,c1(C(N(C2CCN(C(CCCC)=O)C2)CCO)=O)c(C)cccc1C 64636,c1(C(=O)NCCOCCCNC(C(C)SCCCC)=O)cc(Cl)ncc1O 64637,c1(C(=O)NC(CNC(=O)CC2CCOC2)C2CC2)cnc2sccn2c1=O 64638,CCC(C)CC(=O)N(C1CC(NC(=O)Cc2sc(C)nc2C)C1)C 64639,C(=O)(CC1CCc2ccc(O)cc21)NC1c2cccc(OC)c2CCC1 64640,CC1(C)COCCC1C(=O)NC1CN(C(=O)COCCOC(F)F)CC1O 64641,N1(C(c2c(C)nccc2)=O)CCC2CC2(C(=O)NCC2(O)CC2)CC1 64642,Cc1[nH][nH]c(=N)c1C(N1CCC(CN(C)C(c2cnc(CC(C)C)[nH]2)=O)C1)=O 64643,N1(C(C(N2C(C#C)CCC2)=O)=O)CCN(C)CC1C 64644,C1(C(=O)NCC2(O)CN(C(=O)C(C)C)C2)(CC)CCC(O)CC1 64645,C1(CN(C(=O)CCO)CC)CCCCN1C(=O)CC=CC(C)(C)C.C(C)(C)=C 64646,c1(C(N(CC(C)(C)NC(c2cnc(CC)nc2O)=O)C)=O)occ2c1CCOC2 64647,CCC(C(=O)NC(Cn1cncn1)C(=O)NCCCCCN(C)C)N(C)C 64648,c1(OC)cc(NCCCCNC(=O)Cc2nncn2C(C)C)c(Cl)cc1[N+](=O)[O-] 64649,C(=O)(CC(C)NC(c1sccc1SC)=O)OCC 64650,Cc1cc(C(=O)N(C(C)CNC(=O)C(O)c2ccsc2)C)c(C)n1C(C)C 64651,n1(CC)nc(C(=O)NC2CN(C(=O)C(F)N3CCCC3)CC2C)cc1C1CC1 64652,c1(C(=O)NCCNC(C(C)OCCCC)=O)ccc(CNC(=O)C2CC2)cc1 64653,C(=O)(C#CC(=O)NC(C)C)N1CCC(N(C(=O)C(C)n2ccnc2)CCC)C1 64654,C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(Cc2cn(C(C)C)nc2)=O)CC1C#N 64655,C1(C(N2CCC(N(C(=O)CSS(C)(=O)=O)CCC)C2)=O)CCC([N+](=O)[O-])CC1 64656,c1(C(=O)OC)cccc2cc(C(=O)N=c3[nH]nc(Cl)cc3Br)sc12 64657,c1(C(N2C(CC(C)C)CCCC2)C(=O)NC2COC2)cccn2ccnc12 64658,N1(C(C(CC)F)=O)CC2(C)CC1(C(=O)NCC(CO)C1CC1)C2 64659,N1(C(C(CCC)C)=O)CCN(C(=O)COC(C)C)CC1C 64660,N1(C(C2(CC=C)CN(C(=O)COCC3COCCN3C)C2)=O)CCN(CCO)CC1 64661,C1(C(=O)NCC2CC(SC)C2)(COC)CN(C(=O)C(=Cc2ccco2)C)C1 64662,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(c2oc(CC)nc2C)=O)C(C)CC1C 64663,c1(C(=O)NCC2(NC(COCCC)=O)CCC2)ccc(C(N)=O)cc1 64664,c1(C(N2C(C(=O)NCCN(C(=O)OC(C)(C)C)CC)CCC2)=O)ncccc1F 64665,N1(C(C(C(C)OC)OC)=O)CCN(C(=O)C=Cc2ccc(C)cn2)C2CCC12 64666,Cc1cc(C(c2nnnn2-c2ccc(F)cc2)NC2(CCF)CC2)c(C)cc1Br 64667,Cn1cnc2ccc(C(N3CCN(C(c4ccon4)=O)C(C4CC4)C3)=O)cc12 64668,CC1(C(=O)NCC2(F)CCN(C(c3ccc(CO)nc3)=O)C2)CCCCCC1 64669,C1(C)(C(=O)NC2(CSC)CCC2)CC(OC(C)C)CN1C(=O)CCC(C)C 64670,Cc1cc(C(=O)NCCCN(C(=O)CCCCC#N)C2CC2)c(C)n1-c1ccon1 64671,C1(N(C(=O)CC2(O)CCCOC2)C)CCN(c2nccc(N3CCCC3)n2)CC1 64672,C1(C(N2CCC(CNC(=O)OC(C)(C)C)C2)Cc2ccccc2)COC(C)(C)C1O 64673,c1(C(=O)NCCCC(C)NC(C2CCC=CCC2)=O)cc(F)c2c(c1)CCC2 64674,c1(C(C(=O)NC)NN(CC(F)(F)F)CCOC)ccc(C)c(F)c1F 64675,C1(Cc2scc(COC)c2)CCCN(CC(=O)NCC(=O)NC2CCOCC2)C1 64676,C(C(F)(F)C(=O)NC(C)CN(C(c1cc(-c2ccco2)on1)=O)CC)OC 64677,C(CN=c1[nH]c2cc(Br)cnc2s1)C1N(C(c2c(OC)nsc2)=O)CCCCC1 64678,C1(c2[nH]c(N3CC4CC4C3)nc(=NC)n2)CCCOC12CCCC2 64679,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 64680,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2Cl)=O)C1 64681,C#CC1CN(C(C23CC(CN(C(C4(F)CCC4)=O)C2)C3)=O)CCO1 64682,c1(C(=O)NCC(C)NC(C(C)n2cccc2)=O)cc2c(F)c(Cl)ccc2[nH]1 64683,C1(NC(Cc2ccc(C)c(Br)c2)=O)CC2(CCC(NC(=O)C(F)=CCCF)CC2)C1 64684,C(CCC(C)(C)C(=O)N1CC(O)C(O)CO1)NC(C(c1cnn(C)c1)C)=O 64685,Cn1[nH]nnc1=NCC1(CNC(=O)C2CC2)CCC1 64686,c1(C(N2CCC(O)(C(CNC(C=CC)=O)C)C2)=O)ccc2nc[nH]c2c1F 64687,N1(C(C(C)N(C)C)=O)CC2CCN(C(c3ccc4cc[nH]c4n3)=O)CCC2C1 64688,c1(C(N2CCC3(CCO3)C2)C(=O)NCCSC)ccc(-c2cccs2)cc1F 64689,c1(OC)cc(C(N2CC(C)(NC(c3csnc3OC)=O)C2)=O)c2c(c1)CCO2 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64708,C1(CNC(C2N(C)C(=O)OC2)=O)CN(C(C2(C)C=CCCC2)=O)CCC1(F)F 64709,c12cc(Cl)cnc1c1c[nH]nc1c(=O)[nH]2.c1(CNC)cc(F)ccc1F 64710,c12cc(C)sc1NC2=O.c1(-n2cc(C(C)(C)SC)nn2)ccccc1OCCF 64711,C1(C(=O)NC2CC(N(C(=O)C(C3CCCCC3)N(C)C)C)C2)CN2CCC1C2 64712,C(CCCCCC(=O)N1CC2CC(O)CC1C2)NC(c1nccc(Cl)c1F)=O 64713,C1(C(N(CCCN(C(=O)CCn2cnnn2)C)C)=O)CCCNC1=O 64714,C1(NC(C(C)OC)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 64715,c1(C(=O)NCC2CN(C(C(CC(C)C)OC)=O)CC2(F)F)scc2c1OCCO2 64716,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 64717,CC1N(N2CCOC(c3noc(-c4ccccc4)n3)C2)C2CCCC12 64718,C12(NC(C(F)=CCC)=O)CN(C(=O)CCC3CCCCC3)C(COC)(C1)C2 64719,C1(N(C(C2CCN(C(Cc3c(CC)con3)=O)C2)=O)C)CCCC1C#N 64720,N1(C(c2ncc(C)nc2)=O)CC2CCC1C(Nc1ncnc(Cl)c1C)C2 64721,N1(C(c2cccc(OC)c2O)=O)CCC(NC(C2(CF)CCC2)=O)C(CO)CC1 64722,c1(C(=O)NC(C(=O)NCCc2cnc(C)[nH]2)Cc2ccoc2)cnc(Cl)n1C 64723,N1(C(C)=O)CCC(C)(C(N2CC(NC(C3(C)CCNC3=O)=O)CC(F)C2)=O)CC1 64724,C(C(C)C)(C(C(=O)NCc1ccccc1Br)N1CCC(O)C(O)C1)OC 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65007,C1(CC(=O)NCC(CO)NC(C(C)NS(C)(=O)=O)=O)CCC(O)C1 65008,N(C1CCSc2ccc(Cl)cc21)C(Cn1c(C)nnc1)=O 65009,C(CCCCC(=O)N(C1CCN(C(=O)CC2CC(C)C2)C1)CCOC)=CC 65010,c1(C(N2CCCC(C)C2)CN2CCCC(C(=O)N(C)C)C2)ccc2[nH]nc(Cl)c2c1 65011,c1(C(N2CCC(N(C(C3CCCCC3F)=O)CC)CC2)=O)cccc(N)c1C 65012,C1(NCCNC(c2ccc(C)cc2)=O)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65013,c1(C(=O)NCCNC(C(C)=C2CCCC2)=O)ccccc1-c1nc(C)no1 65014,c1(C(N2C(CNC(CCC(=O)NC)=O)CC(F)(F)C2)=O)c(C)nc2ncnn2c1C 65015,c1(OC)ccc(C(N2CCC3CCC23)C(=O)NCCSc2ccccc2)c(Cl)c1O 65016,C(C(C)(C)CNC(=O)C(C)(C)N(C)C)NC(CNS(CC)(=O)=O)=O 65017,N1(C(CC2C(C)=NNC2=O)=O)CC2(C=C(C(=O)NCc3cccnc3F)CO2)C1 65018,c1(C(=O)NCC2(CNC(C3C(C)C3C)=O)CC2)cnc[nH]c1=N 65019,c1(C(=O)NC(C2(O)CCN(C(=O)C3=C(Cl)CC3)CC2)C)ccc(Cl)c(Cl)c1 65020,c1(C(C)C)cccc(C(N2CCC(CCNC(C3CCC3CF)=O)CC2)=O)c1F 65021,C(=O)(C(C#N)C(C)C)NCCCC1OCCN(C(c2cc(OC)no2)=O)C1 65022,N1(C(CC)=O)CCCC(C)(C)C1CNC(c1ccc(-c2ccc(Cl)s2)cn1)=O 65023,Cc1cc(C(N2CC(C)CCC2C(=O)Nc2cc(F)c(F)cc2I)=O)c(O)c(C)c1 65024,CC(C)(C)S(=O)(=O)CC(=O)NCC(N1CCN(C(=O)C=C2CC2)CC1)C(F)F 65025,C1(OC2(Nc3c(Br)cccc3)CC2)CN2CCC1(F)CC2 65026,C(=O)(C(C(C)NC(c1ccc2[nH]ccc2c1)=O)C(C)C)N(CC(C(C)C)OC)C 65027,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65028,N1(C(CC2C(C)(C)C2)=O)Cc2[nH]nc(C(N3CCCC3)=O)c2C1 65029,CC(C)(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(c1cn(C2CC2)nn1)=O 65030,c1(COCC)nc(Cl)cc(=NCC2(C(=O)Nc3c(C(F)(F)F)cnn3C)CC2)[nH]1 65031,CCCCC(C(=O)NC(COC)CC(N1CC2(CCC(=O)NC2)C1)=O)C(C)C 65032,CCC(CC(=O)NOCC1CCC(NC(C)=O)CC1)CC(C)C 65033,c1(OC)cc(NCC(F)F)cc(Cl)c1O.C(C(=O)NNC(=O)O)S 65034,c1(SCC(N2CCC(C)(C)C2)=O)ccc(F)c(S(=O)(=O)N(C)C)c1 65035,CCC1=NOC(CNC(C2CCC(NC(c3c[nH]nc3OC)=O)CC2)=O)C1 65036,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65037,C#CC(CNC(C1CCN1C(=O)C(O)C1CC1)=O)CC 65038,c1(C2(C(N(C3CN(C(c4c(C)[nH]cc4)=O)CC3F)C)=O)CC2)ccc(Cl)c(F)c1 65039,N1(C(Cn2nc(C)oc2=O)=O)CCC(C2CC2)C1C(N1CC(c2nc(=O)o[nH]2)C1)=O 65040,c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)sccc1Cl 65041,c1(NCC(CCC)(C)CO)ncc(C)cc1S(=O)(=O)NC(c1cccc(F)c1C)C 65042,c1(C(C)OCC)cccc(-c2nc(N(C)CC)n(C3CCSC3)n2)c1 65043,c1(C(=O)NCC(CC(C)C)NC(N)=O)ccc(S(=O)(=O)NC(C2(C)CCC2)=O)s1 65044,Cc1nc(C(N2CC(NC(=O)CN3CCSCC3)C(O)C2)=O)cn1C(F)F 65045,N1(C(C(=O)NCC(C)C)CCc2ccccc2)C2CC1N(C)C(=O)C2(C)C 65046,N1(C(C(=O)NCC)=O)CCN(C(=O)NC2CN(C)CC2c2ccccc2)CC1 65047,c1(C(N2CCCCC2CCO)C(=O)NCCC)cccc2ccnn12 65048,C1(C(=O)NC(CNC(c2nnc(-c3ccccc3)s2)=O)CO)CCCSC1 65049,c1(C(C(=O)NC2COC2)N(C)Cc2ccc(SC)cc2)cc(F)ncc1C 65050,CC(C(C)C(=O)N(C1CCCC1)C)NC(C1CN(C)CCO1)=O 65051,c1(C(=O)NCC(C(=O)N(C2CC(O)C2)C)CC2CC2)n[nH]cc1[N+](=O)[O-] 65052,C1(N(C(=O)C(N)=O)C)CCN(C2CCCN(C(=O)CC3CC4CC4C3)C2)CC1 65053,c1(OC)ccc(C(C)=CC(=O)NCC23CC2CN(C(=O)C=CC=C(C)C)C3)cc1 65054,c1(C(=O)NC(C(C)C)CO)ccnc(NC(=O)CCc2ncccc2F)c1 65055,N1(C(CC2OCCN(C(c3ccc(C)c(O)c3)=O)C2)=O)CC(C)C12CCOCC2 65056,Cc1cc(C(N2CCCC(CNC(=O)C=CC3CC3)C2)=O)cc(S(C)(=O)=O)c1F 65057,C(c1ccccc1OC)=CC(=O)NCC(=C)CCNC(c1cnsn1)=O 65058,c1(CCC(=O)NCC2N(C(=O)C(C)(C)CF)CCN(C)C2)ccc2c(c1)OCO2 65059,CCN=C(NC(C1(O)CCOC1)C1CCCC1)NC1CCN(c2cnn(C)c2)C1 65060,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnc(C2CC2)s1)=O 65061,C(C)(C(C)(C)NC(=O)CCc1cn(C)nn1)NC(C1(CC#C)CC1)=O 65062,c1(CC)ccsc1C(C(=O)NCc1ccco1)N(C1CC1)C(C)C1CC1 65063,C(=O)(C(C(C)C)C(C)C)N1CCC(C(N(C(CC)CN)C)=O)O1 65064,c1(C(C(=O)OC)=O)cn(C)nc1C(N1CCC(NC(=O)Cc2csc(C)c2)C1)=O 65065,c1(C(N(CC(C)NC(=O)CCSC)CC)=O)cc(Cl)cc(Cl)c1O 65066,C(N=c1ncc(C(F)F)c[nH]1)C1N(C(C)C)CCCC1.C12CC(C1)NC2=O 65067,Cc1cnc(C(N2CCC3(CC3NC(=O)CCC(=O)N(C)C(C)C)C2)=O)c(C)c1 65068,c1(CCC(=O)NCC2(CN(C(C3C(CC)CC3)=O)C)CC2)ncccn1 65069,c1(N(CCN(C)C(c2cc(F)c(CO)c(F)c2)=O)C)ncccc1S(C)(=O)=O 65070,C(C)(C(CC(=O)NCCOC1CC1)NC(C1CC(C(C)C)=NO1)=O)OC 65071,C1(CC(=O)NC(C(=O)N(CC(O)CF)CC)CC2CCC2)CC(=O)NC1=O 65072,c1(OC)c(C(=O)NC(C)(CNC(c2ccc(C3CC3)cn2)=O)C(C)C)csc1Cl 65073,CC1C(NC(C2CCCCC2O)=O)CCCN1C(C1CC(=O)N1)=O 65074,CNS(=O)(=O)N1CCN(CC(=O)NC23CC4CC(C2)CC(O)(C4)C3)CC1 65075,N1(C(C(CC)N(C)C)=O)Cc2occ(C(=O)NC3CC4C=CC3CC4)c2C1 65076,c1(C(N(CCNC(CC(=O)NCC)=O)C(C)C)=O)cccc2cnnc(O)c12 65077,C(=O)(C1=CCS(=O)(=O)C1)NCC(C(C)C)(C)NC(=O)C(C)CN1CCCCC1 65078,CC(C)C(CO)C(=O)N1CCCCC1CN(C(=O)C(C)CC1CCCO1)C 65079,C1(NC(CN2CCN(C)CC2)=O)COCCN(C(=O)CCCC2CCCC(=O)N2)C1 65080,N1(C(CC2(C#N)CCC2)=O)CCCC(NC(=O)COCCCF)C1 65081,CN1CC=C(CC(=O)N2C3CCC2CC(NC(c2cc(C(N)=O)[nH]n2)=O)C3)CC1 65082,CCC(C)(C)C(O)C(=O)NCC1CN(C(C2CC3(CCCO3)C2)=O)CC1O 65083,C1(CC#C)(C(=O)NCCN2CCC(CO)C2)CCCN1C(=O)CSC(F)(F)F 65084,c1(C(N2C(C(C)(C)NC(c3cccc(F)n3)=O)CCC2)=O)ccc2cc[nH]c2c1 65085,C1(C(=O)NC(CN(C(c2cc(COC)on2)=O)C)C)(C(=O)OC)CCCNS1(=O)=O 65086,c1(C(N(CCNC(C(CC#C)C)=O)CC)=O)n[nH]c2ccc(F)cc12 65087,N1(C(C2N(C)CC(F)C2)=O)C(C(N2CC3CC2CS3)=O)CCC12CC2 65088,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC=C(Cl)Cl)C1 65089,C1(CC(N2CCCC(CCNC(=O)CC3OCCCO3)C2)=O)CN2CCN1CC2 65090,C1(C(C(N2CCCC(NC(Cc3n(C)ncc3)=O)C2)=O)O)CCS(=O)(=O)CC1 65091,Cc1cc(C(=O)NCC(C2CCOC2)NC(c2cc(CO)n(C)n2)=O)ccn1 65092,C(C)(CO)(C(=O)N(CCC(=O)NCC1CCCOCC1)C)OC 65093,Cc1cc(C)c(C#N)c(NCCc2csc(C)n2)n1 65094,C1(NC(N2CCSCC2)=O)CC(Cc2ccc(-n3[nH]cnc3=O)cc2)C12CCC2 65095,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)N(C)C 65096,Cc1sncc1C(=O)NCCCNC(C1CC1(C)C)=O 65097,c1(CC(=O)NC(CCO)C(F)F)cccc2c1CCN(C(=O)CO)C2 65098,C1(C(=O)NCC(C)OC)(OC)CCN(C(=O)Cc2ccc(Br)cc2F)CC1 65099,c1(CN(C2CCCC3(CNC3)C2)c2c(F)cccc2Cl)cnc2n1CCCCC2 65100,CC1C(NC(=O)C(C)Cc2cnc[nH]2)CCCN1C(c1nn(C(F)F)cc1Cl)=O 65101,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65102,c1(C(N(CC(C)NC(=O)C2=C(Cl)CCC2)C)=O)ccc2c(c1)CCCC2=O 65103,c1(C(N2CC(CC(C)NC(C3CCN(CC)C3)=O)C2)=O)cc2cncn2c(O)n1 65104,N1(C(=O)CCN2CCOCC2)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65105,CC1CC(CNC(=O)CCOC2COC2)CN(C(C2CCCS2)=O)C1 65106,CC(C)CCCCN(C(=O)C(CC1CC1)NC(c1cncn1C)=O)C 65107,N1(C(CCCOCC)=O)CC2(CCC2)CC1C(=O)N(CC(C)(C)CO)CC 65108,c1(CCC)nsc(N(C(c2nccn2C2CC2)=O)CC2CCNCC2)n1 65109,c1(CC)nc(C)c(C(N2CCCCC2CN(C(=O)Cn2cnnn2)C)=O)c(C)n1 65110,N1(CC(=O)N(C2CCOC2)CC)CCCCC1C(=O)Oc1csnn1 65111,C(=O)(C(O)(C(F)(F)F)C1CC1)N1C(CCNC(=O)Cn2cnnc2O)COCC1 65112,N1(CCOC(C2CCOC2)CNC(C(C)(C)C2CCCO2)=O)Cc2ccccc2C1 65113,N1(C(c2nc(CNC(C(C(C)C)OC)=O)cs2)=O)CCN(C)CC1C 65114,n1(CC)cc(NC(C2(OC(C3(COCC)C=CCC3)=O)CCC2)=O)c(C)n1 65115,N1(CC)CC(C(=O)NC(CC)CC(=O)NCC2(CCOC)CCCC2)CC1=O 65116,N1(C(c2ccc(CC)o2)=O)CC(NC(=O)Cc2ccsn2)C2CC12 65117,Cn1cc(C(c2ccco2)NC(c2nnnn2Cc2cccs2)c2ncco2)cn1 65118,N1(C(c2cc(C)sc2C)=O)CCC(CNC(=O)CCOCCN(C)C)C12CC2 65119,C1(CCC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)CN1CCC(C)(C)C1 65120,CCC(CC)C(CNC(=O)N(C)Cc1cccc(F)c1F)OC 65121,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65122,c1(C(=O)NC2(CNC(C3(C)CCN(C)CC3)=O)CCC2)n[nH]c2c1COCC2 65123,CC1=NOC2(CCN(c3cc(C(C)(F)F)ncn3)CC2)C1 65124,C1(Nc2ccc(C(=O)OC)cn2)(CNC(=O)Cn2cnnc2)CCCCC1C 65125,c1(Cc2cn(CC(=O)N(C(c3ccccc3)C)C3CC3)nc2)cc(Cl)ccc1Cl 65126,c1(N(C2CCNC2)Cc2c(C)nc(COC)s2)ncc2[nH]ncc2n1 65127,C(CC(O)CNC(c1ccc(C(F)(F)F)[nH]1)=O)NC(C=CCC)=O 65128,C=CCCN=C(NCC1CC12CCSCC2)NCC1(F)CCC(CO)CC1 65129,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65130,c1(C(N2CC(CC)(NC(=O)CCCS(N)(=O)=O)C2)=O)cnc2ccc(OC)nn12 65131,C=CCC(C)(C)CC1C(=O)C2C3(CCN1CC3)c1c(cccc1)NC2=O.CC=C 65132,C(=O)(CC1=CCCC1)NC1(CC=C)CCN(C(C2CC3CCC3C2)=O)C1 65133,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(c2cc(COC)on2)=O)CCN1C 65134,c1(CN2C(CCCC)CSCC2)ccnc(-c2nn[nH]n2)c1F 65135,N1(C(C(CCC)OCC)=O)C2CCC1CN(CCc1cccc(Cl)c1)CC2 65136,N1(C(c2cc(C)sc2)=O)C2CCC(C(=O)NCc3cncc(Cl)c3)C1CC2 65137,c1(C(=O)NC2CC(CNC(C(CC)(C)O)=O)C2(C)C)ccc(OC(F)F)c(Cl)c1 65138,CC1CC(CNC(=O)CCP(C)(C)=O)CN(C(c2ccc(Cl)c(N)c2)=O)C1 65139,N1(C(C=CCC)=O)CCN2CCOCC2(CNC(C2COCCO2)=O)C1 65140,c1(C(=O)NC(C)CO)ccccc1SCc1nnc(S)n1C.C12CN(C1)C2=O 65141,N1(C(c2c(C)ccnc2O)=O)CC2(CCCC2NC(=O)CSC(F)F)C1 65142,CC(C)C(C)(C)C(=O)NCC1(C)CCN(C(c2cnn(C3CC3)c2)=O)C1 65143,Cc1nnc2n1CCCC2C(=O)NC1CCC(CNC(c2cn(C)nn2)=O)CC1 65144,CON1CC(C(=O)N(CCC(=O)OCC=CCF)C(C)(C)C)CC1=O 65145,CON(CCC(=O)Nc1ccc2c(c1)OCO2)C(=O)CN1CC2(CC(O)C2)C1 65146,C1(NC(C(C)OCCOCC)=O)CC2CN(C(c3nc(O)sc3C)=O)CC2C1 65147,C1(NC(C2C(CC)C2)=O)CCCC1NC(=O)CC(=O)NCC(F)(F)F 65148,O=C1NCc2c(CS)cccc21.c1(COC(C2(O)CC2)=O)ccco1 65149,c1(OC(C)C)cccc(C(=O)NCC2CCC(NC(c3ccc(F)cc3)=O)C2)c1 65150,N1(C(C(C)CCF)=O)CC(S(C)(=N)=O)C1.C(C)(C(=O)N)NC(=O)NC 65151,CCCCCC(O)CC(=O)NC1CC(CNS(=O)(=O)CC2CCC2)C1 65152,c1(-c2ccc(F)nc2F)ccc(NCc2ccncc2F)c(F)c1F 65153,c1(OCCC)ccc(C=CC(=O)NC2CC3CCC(C2)N3)c(OC)c1 65154,C(CC(=O)NCC1CC(SC)C1)N(C(=O)CC1CC1(C)C)CC 65155,c1(C(N2CC(CC)N(C(c3csc(C)n3)=O)CC2)=O)cncc(S(C)(=O)=O)c1 65156,CC(C)C(C(C)NC(=O)CCC(F)F)NC(=O)CCCN(C)C(N)=O 65157,Cc1cc(O)ncc1C(N1CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1)=O 65158,Cc1ccc(NC2CCCCC2NC(=O)CCCF)c([N+](=O)[O-])c1 65159,C1(NC(CC2(OC)CCOCC2)=O)CCC2(CC1)CN(C(=O)C(C(C)C)SC)C2 65160,c1(CC)nc(N2CCCC(NC(=O)Cc3ccccc3F)CC2)cc(C#N)n1 65161,N#Cc1cncc(CC(=O)NCC2CCN2C(=O)CC2CC3CCC2CC3)c1 65162,N1(C(=O)Cc2nccs2)CC2CC2(CNC(C2(N3CCCC3)CCC2)=O)C1 65163,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65164,C1(CNC(c2cc(C)n(C(C)C)n2)=O)CN(C(=O)Cc2csnn2)C2CCN1C2 65165,C1(NC(C(C)C)=O)CCCC1(C)C(N(C)N)=O.C(=O)(CCc1ccco1)NC1CC1CC.C 65166,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65167,C1(NC(C(C)c2ccsc2)=O)CC2CCC1N2C(=O)COc1ccc(F)cn1 65168,C1(C(=O)NCCN(C(=O)C(O)CNC(=O)OC(C)(C)C)C)CNC(=O)N1 65169,N1(C(C(C)(O)c2ccccc2)=O)CCN(C(=O)NC2CC3C(C2)C3(F)F)CC(O)C1 65170,C#CC1(O)CCCN(C(=O)CNC(=O)CNC(c2ccsc2C)=O)C1 65171,C(=O)(C#CC1CCCCO1)NCCCC1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 65172,CC1(C)C(C(=O)NC2CCC(NC(c3c[nH]nc3F)=O)CC2)CCS1(=O)=O 65173,[N-]=[N+]=NCCC(=O)NC1(C(=O)NCC(O)CO)CC(CO)C1 65174,Cc1cnn(CC(N2CCC(C)(CCNC(=O)COC3COC3)C2)=O)c(=O)c1 65175,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65176,c1(C(=O)NC2CC(CC(=O)NC3C(c4n(C)ncc4)C3)C2)cccc(F)c1O 65177,C(CC(=O)NOCCC1CCCO1)(C1CC1)NC(C1CCC(N(C)C)CC1)=O 65178,N1(C(c2cncc(C)n2)=O)CCCC2C(CCCN2C(=O)COC2(C)CCC2)C1 65179,C1(NC(=O)NCC=C(C)C)CCN(C(=O)COC(C)(C)C)C12CCC2 65180,N1(C(C2(C)CC=CCC2)=O)CC2(CC2)CC1CNC(=O)CC1CC2(CCC2)CO1 65181,Cc1cc(C(=O)NCC2CN(C(=O)Cn3cnnc3O)CC2C)c(Cl)cn1 65182,c1(CNC(c2cc(C(=O)NCC3CCCO3)[nH]n2)=O)csc(C(F)F)n1 65183,C=CCC(CC=C)C(=O)NCC1CCCN(C(C2(OC)CS(=O)(=O)C2)=O)CC1 65184,C(=O)(C1CCCc2nncn21)NC1CCC(NC(C2(C)CC(C#N)C2)=O)CC1 65185,N1(C(c2c(C)coc2)=O)CCN2C(=O)C(NC(=O)Cc3ncnn3C)CC2C1 65186,O=C1CC(CC(=O)N2CC3CC3(CNC(=O)C(O)Cc3ccccc3Cl)C2)=NN1 65187,c1(SCCC(=O)N(CCCO)CCNS(CC)(=O)=O)ccccc1 65188,C(=O)(CC1=CCOCC1)N(CCC(=O)N1CC(N(CCCO)C)C1)CC#C 65189,c1(C(N(CCNC(=O)C=CC=C(Cl)Cl)CC2CC2)=O)cccc2nccn12 65190,C(c1cnc2ccccc2n1)=CC(N1CC(C(C)NC(c2nc(Cl)cs2)=O)C1)=O 65191,c1(C(=O)OC)cc(C(=O)NC23CC2CN(Cc2cnc(C4CC4)[nH]2)C3)cc(Cl)c1 65192,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65193,C1(CC)(NC(=O)Cc2c[nH]nc2O)CN(C(=O)CC2(C)CC2(Cl)Cl)C1 65194,Cc1ccc(C(N2CCC(O)C(NC(c3c(F)cnn3C(C)C)=O)C2)=O)c(=O)n1C 65195,CC1CN(C)CCN1C(=O)C(C)OC(c1cccnc1)C 65196,c1(C(C)(C)C)n[nH]c(=NCC(C)(C)NC(c2cnc(F)c(F)c2)=O)s1 65197,Cc1ncsc1C=CC(N1CCC(CN(C(=O)C(C)CF)C)C1)=O 65198,N1(CC(N2C(CNC(=O)Cc3ncncc3Cl)CCC2)=O)CCc2ccccc2C1 65199,Fc1ccc(CCCNc2cccnc2C(F)(F)CF)cc1 65200,N1(C(CC(C)OC)=O)CC(C2(NC(c3ccc(Cl)cc3C(F)F)=O)CC2)C1 65201,S(=O)(=O)(c1c[nH]ccc1=NCC1CCCS1(=O)=O)NC(c1ncc(OC)cc1C)C 65202,Cc1ccc2nc(C(=O)NCC3(CNC(C4CCC5CC45)=O)CC3)ccc2c1 65203,N1(S(C(C)C)(=O)=O)CCN(C(C2CCCSC2)C(=O)NCCC(F)(F)F)CC1 65204,N1(C(c2c(C)cccc2Cl)=O)CC2(CCN(C(=O)CC(C)(F)F)CC2CO)C1 65205,C1(C(=O)NCCC2(C(=O)NCC3(O)CCC(C)C3)CC2)CN2CCN1CC2 65206,C(=O)(C(C)(F)C(=O)N1CCCC(CNC(c2nc(OC)ccc2C)=O)C1)OC 65207,CS(=O)(=O)C1(C(=O)NCC2(CCNC(C3CC(N=[N+]=[N-])C3)=O)CC2)CC1 65208,c1(N2CCC(C(=O)OCC3OCCC(C)C3)CC2)cccc(Cl)c1F 65209,C(=O)(C(C)(C)C)NC(C)CN(C(=O)CNC(=O)C(=O)NC1CC=CCC1)C 65210,N1(C(c2nc(C)n(C)c2)=O)CCN(C)C(CNC(c2cn3c(n2)CCC3)=O)C1 65211,N1(C(=O)C=CC2CCCO2)CCOCC(OC(F)(F)F)C1.O(C(F)F)C 65212,C(C1=NOC2CCCCC12)NC(C1CCC2N(C(CCC=C)=O)C1CC2)=O 65213,C1(NC(C2C(CC)CC2)=O)CCCCCN(C(=O)C=C(C)C)C1 65214,c1(NC(C2CC(OC)C23CCC3)=O)ccc2c(c1)N(C)CCC2 65215,C1(NC(C(CC)SC)=O)CC(C)CN1C(=O)CC1CCCC(C)C1 65216,Cc1n[nH]c(C)c1C1CC1C(N1CCC(n2cc(-c3scnc3C)nn2)CC1)=O 65217,N1(C(c2cc(C)oc2C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1 65218,CCCC(C(O)C(=O)N1CCOCC1CCC)NC(c1c(F)ccc(F)c1F)=O 65219,N1(C(CCCC#C)=O)CCCCCC1CNC(c1cc(C)nnc1CC)=O 65220,N1(C(C2NCCN(C(c3scc(C)c3C)=O)C2)=O)CCCC(C)(O)C1 65221,N1(C(=O)NC2CCCC2C2CC2)CCC2CCC(C1)O2 65222,C(=O)(C1=CC2(CCOCC2)C1)NCC1(C(C)(C)O)CN(C(C(CC)(C)F)=O)C1 65223,c1(C(N2CC(C)C(NC(c3ccc(O)nn3)=O)CC2)=O)c(Cl)ccc(Cl)c1O 65224,c1(C(=O)NCCCCCNC(C=CCN(C)CC)=O)cccc(COC)c1F 65225,N1(C(CCC)C)CC(C(=O)NCCNC(=O)CC(c2ccc(Cl)cc2)O)CC1=O 65226,Cn1ccnc1CNC(=O)C(N)Cc1ccoc1 65227,C(=O)(C(C)C(C)NC(c1ccc[nH]1)=O)NCCC(=O)N(CC)CC 65228,N#Cc1c(F)cc(C(=O)NC2CCN(C(=O)CCCCc3cnc[nH]3)C2)cc1F 65229,CC1C(C(=O)NCCCCCCF)CCCN1C(C1CCCC(=O)N1C)=O 65230,CC1CC(NC(=O)COc2ccccc2NC(=O)CO)CCN1CC(=O)N(C)C 65231,C1(C)(CC)C=C(C(=O)N2CCOC(CC)C2)C1.N12CCOCC1CC2=O 65232,CON1CC(C(=O)NC(C(N2CCC(C)(CCO)C2)=O)C2CC2)CC1=O 65233,C(=O)(C(C)(O)CCN(C)C)N1CC(C(C(=O)NCCC(C)(C)OC)O)C1 65234,c1(CC(C(N2CC(CC(C3CC3)OC)C(CO)C2)C(=O)OC)C)ccccc1Br 65235,N1(C(CN(C)C(C2CCCCC23CC3)=O)=O)CCCCC(NC(=O)C2CC2)C1 65236,c1(C(=O)NC(CCNC(c2nn(C)c(C#N)c2)=O)(C)C)c(Cl)ccc(F)c1F 65237,CC(CCCCNC(=O)COCc1ncnn1C)NC(=O)C=CSc1nc[nH]n1 65238,C#Cc1cnc(N2CCCC(CO)(NC(=O)C=Cc3cnc(C)s3)C2)nc1 65239,n1(Cc2nc(C)on2)nnc(CNC(C2(N=[N+]=[N-])CC2)=O)c1C 65240,Cc1ccc(C=CC(N2CCC(C(=O)NCC3CN(C(=O)CC4CC4)C3)CC2)=O)o1 65241,C1(C(=O)Nc2c(C#C)c[nH]n2)CC2CN(C(=O)C(F)OC(F)(F)F)CC12 65242,c1(C(=O)OCC2C(C)C2NC(c2cc(O)nc(O)n2)=O)ccc(F)c2ccncc12 65243,Cc1cc(Cl)c(Br)cc1S(=O)(=O)N(C1Cc2ccccc2N1)C1CC2CC1CN2 65244,c1(C(=O)NCC(CNC(=O)C(F)(F)c2nccs2)OC)cccc(F)c1N 65245,c1(NC(=O)NCC2CN(C)C(=O)C2)cccc2c1COCC2 65246,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65247,C(CS(=O)(=O)CC(=O)NCC(C)(CNC(c1c(C)ncn1O)=O)OC)OC 65248,C(=O)(CCCCNC(C1CC(C)C1)=O)NC(C(=O)OC)CC1CC1.C1(C)CC1 65249,c1(C(=O)NC2CN(C(C(OC)OC)=O)C2)cc(C)n(-c2nc(C)cs2)c1C 65250,c1(OCC)ccc(CCC(=O)NC(C)CCN(C)C(c2nonc2N)=O)cn1 65251,c1(C(N2CCN(C3(CCC(=O)N4CCCC4)CC3)CC2)=O)ccc2nc[nH]c2n1 65252,C(=O)(C(C)(O)C(C)C)NCC(C(N1CC(CC#C)OCC1)=O)Cc1cnn(C)c1 65253,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65254,CCC(CC(=O)NC1CCCN(C(=O)CCC(=O)c2ccccn2)C1C)C(C)C 65255,c1(C(N2CCC(CC=C)(NC(c3cc[nH]n3)=O)C2)=O)c(F)c(N)cc(Cl)c1F 65256,c1(C(C)NC(c2nc(CN3CCCCC3C)cs2)=O)cnn2c1NCCC2 65257,CN1CCC(F)(CNC(=O)C(C)(CO)NC(C2CNC(=O)N2)=O)C1 65258,CC1OCCCC1C(=O)N(C)C.c12nnn(C)c1C(=O)NOCC(=O)NC2 65259,C1(NC(=O)COC2CC(F)(F)C2)(CF)CCN(C(=O)CC2CCC(=O)O2)C1 65260,Nc1ccc(-c2nc(NCCn3cnnn3)cs2)nc1 65261,CCCC(CNC(=O)CC(C)n1cccn1)C(=O)NC1(C2(OC)CCC2)CC1 65262,c1(C(=O)NCCCCCCNC(CN(CC)CC)=O)ccc(C2CC2)c(C)c1 65263,C=CCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65264,c1(C(N2CCC(C(=O)NCCNC(CCC#C)=O)CC2)=O)cccc2nncn12 65265,C1(NC(c2c(C)cnnc2)=O)(CNC(=O)CCOCC(F)F)CCCCC1C 65266,N1(CC2(OCC)CCSC2)CCC(=O)N(CCCc2cccnc2)C1=O 65267,C1(C(=O)NC(CC)CN(C(=O)C(C2CCC2)OC)C)CCS1(=O)=O 65268,CN1CCc2[nH]nc(-c3nc(C4CC=CCC4)no3)c2C1 65269,c1(OC(=O)NCC2CCC(C3CC3)O2)ccc(Br)cc1.CC1CS1 65270,N1(C(C(C)Sc2ccco2)=O)CC2CN(C(C3CC4(CCC4)CN3)=O)CC2C1 65271,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65272,c1(C(=O)NC(c2ccccc2)C(C)c2cccs2)cnn(-c2ccccn2)c1 65273,Cn1cnc2[nH]c(C(=O)NC3CC(C)(NC(=O)CC4CC5COCC45)C3)cc12 65274,C1(CCC(=O)N(C)CC2CC2)CCN(C(=O)CC2COCC2O)C1 65275,c1(C(N2CCC(CNC(CCC=CC)=O)C2)=O)cc(C)c(N)cc1F 65276,C1(C(N(C)CC2CCOC2)=O)CC2(CC2)CN1C(=O)C=CC1CC1 65277,C=CCC(C)(C)CC(=O)NC(C)(C)C(C)NC(c1cn(C)c(C(F)F)n1)=O 65278,Cc1nnc(NC(=O)NCc2ccc(CCC(N)=O)cc2)n1C 65279,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CC4CCC3C43CC3)=O)C2C1 65280,c1(CC(=O)N(CC(C)N(C(C(C)NS(CCC)(=O)=O)=O)C)C)cn(C)nc1Cl 65281,C1(Cc2cn(CC(=C)O)nn2)CCCCN1C(c1scnc1CC)=O 65282,c1(C(N2C3C(NC(COCC(=O)NC)=O)C(C3)C2)=O)ccc2ncccn12 65283,N1(C(C(C)CN(C(=O)Cc2ccon2)C)=O)CC2(CCC(=O)NC2)C1 65284,c1(C(N2C3CN(C(c4c(C)nccc4)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65285,CC1=NOC(C(=O)NC(CNC(C2CCCN2C2CCOCC2)=O)C(C)(C)C)C1C 65286,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)C)=O 65287,c1(CCC(=O)NCC(CN(C(c2nc(CCC)sc2)=O)C)O)nnc(S)nc1O 65288,C(=O)(N=c1[nH]c(Cl)ncc1SC)C1CN(C(CC(C=C)C)=O)C(C)CC1 65289,N12CCCCC1C2.c1(C(C)=O)ncc(-c2cn(CCN(C)C)nn2)s1 65290,c1(C(=O)NC2CC3(CN(C(C(C(C)C)C)=O)C3)C2)ccc2c(c1F)CCC2 65291,CCC(C)(C#N)C(=O)NCC12CC(NC(c3cnc(C(=O)OC)s3)=O)(C1)C2 65292,c1(N(C(C2CC(NC(=O)CCc3nc(O)n[nH]3)C2)=O)CC)ccccc1F 65293,N1(C(C(N2CCN(C)CC2)C)=O)CC(NC(C23CCCN2CCC3)=O)CCC1C 65294,N1(C(=O)CCC2CCCC2)C(C(=O)NCCC2(C3CC3)CCC2)CCC1C1CC1 65295,C1(C(N2CC(OC)(CNC(C3C4COCC34)=O)C2)=O)CC(C)OC1C 65296,c1(CC)cc(C(=O)NC(C)Cc2cccc(CNC(c3cocn3)=O)c2)c(C)o1 65297,C1(NC(=O)Cc2ccc(C3CCCC3)cc2)CC(NC(c2cocn2)=O)CC1O 65298,c1(CN2C(C)CCC2C(=O)Nc2ccccn2)ccc(F)c(Br)c1F 65299,C1(C)(C(N2CC(NC(CCC(=C)Cl)=O)CC23CCC3)=O)CCC2(CC1)OCCO2 65300,c1(OC)nn(C)c(Br)c1C(=O)NCCCN(C)C(C1(C)CC1F)=O 65301,C(CC(=O)N1CC2(CSC2)C1)(C(F)(F)F)NC(=O)C=Cc1cscn1 65302,Nc1ccnn1CC(=O)NCCC1CN(C(c2occc2-c2ccccc2)=O)C1 65303,c1(CN(CCSC(=N)N)Cc2ccc(F)cc2)nc2cnccc2s1 65304,CN=c1[nH]c(N(CC(=O)NC2CCS(=O)(=O)CC2)C)ncc1Cl 65305,N1(C(CCCOC(F)(F)F)=O)CC2(CC(NC(N)=O)CO2)C1.C12CC(F)(C1)NC2=O 65306,Cc1cc(Br)c(F)cc1C(=O)NC1CC(NC(=O)CCOC(C)C)C1 65307,C1(OCC)CC2(C1)CC2C(N1CC(OCCOCNC(=O)CN2CCC2C)C1)=O 65308,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCC(C)(F)F)C1 65309,CC1CCCC(CC(=O)NC(C2CCN(C(c3ccn(CCF)n3)=O)CC2)C)O1 65310,c1(C(=O)NCC(c2ccccc2)CNC(C2C=CCC2)=O)cc(C2(O)COC2)on1 65311,C(C(CNC(C1(c2ncccc2F)CC1)=O)C(F)(F)F)NC(CN1CC(C)C1)=O 65312,C1(NC(CSCCNC(C2C(=C)C2)=O)=O)CC1(C)C 65313,C1(C(N(CC)Cc2ccnc(O)c2)=O)CC12CCN(C1CCC(=O)NC1=O)CC2 65314,CN=c1cc(C(N2CCC(C)(NC(C3CCC(C(N)=O)N3C)=O)CC2)=O)cc[nH]1 65315,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(=O)COC1CCOC1)CCO2 65316,c1(CN)cn(C)nc1.c1(C(c2ccccc2)SC)nnnn1C1CCOC1 65317,CCC(C(=O)Nc1cccc(C(C)(C)C)n1)C(C)C 65318,C1(C(N2CC(N(C)C(c3ccc(F)cc3F)=O)C2)=O)CCc2cncn2C1 65319,Cc1ccc(C(c2ccncc2)NC(=O)NCC2CC2c2ccco2)cc1 65320,C1(NC(C=CC(C)(C)SC)=O)COCCC1NC(=O)C(C)(O)C1CC1 65321,c1(C(=O)NC2(CCOC)CCN(C(=O)C3=CCCO3)C2)cc(Cl)ccc1C 65322,C1(CCNC(C2(CC#C)CCCO2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC1 65323,C12CCC3(CN(C3)C1=O)O2.c1(NC(C(C)NS(CCC)(=O)=O)=O)cc(C)n(C)n1 65324,CC1CCCC1C(N1CC(O)(CNC(=O)Cc2ccsn2)C1)=O 65325,C1(CC(N2CCC(CCNC(C3(CC)CCOCC3)=O)C2)=O)CCCS(=O)(=O)C1 65326,Cc1ncncc1C(=O)N(CC(=O)NC1CCN(C2CCC2)C1)C 65327,C1(N(CC#C)C(c2ccnc(C3CC3)n2)=O)CCN(C(C2CC=CCC2)=O)CC1 65328,C(=O)(C(C)=NOCC#N)NCC(CC)N(C(=O)C(C(C)C)OC)C 65329,N1(Cc2cn(C)nc2Cl)CC(=O)N(CC2(C3CCCCC3)CCCC2)C1=O 65330,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NC(C1(OC)CCC1)C 65331,Cc1cc(=O)oc(C)c1C(=O)NCC1CC1NC(=O)Cc1ccccc1Br 65332,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65333,c1(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)CC)scnc1Cl 65334,c1(C(=O)NCC(CNC(c2cccc(COC(C)C)c2)=O)(C)O)cnc(Cl)cc1Cl 65335,CCCC(CCC)C(=O)N1CCC(C(=O)N(C(C)CC(C)C)C)O1 65336,C1(CCNC(C2CC(=O)NC2)=O)CCCCN1C(=O)CCNc1cnccn1 65337,c1(OCC(=O)N(CC2CC(F)CN2C(=O)C2=CCC2)CC2CC2)cccc(Cl)c1 65338,c1(NC(=O)OC(C)(C)C)ccc(F)c(C=O)c1.C12CC1COC2=O 65339,N1(C(C=C(C)C2CC2)=O)CCC(C2CCCN(C(=O)CN3CCN(C)CC3)C2)C1 65340,C(CC(F)F)(C(=O)NCCN1CCCCC1C)NC(CC=C)=O 65341,c1(C(N2CCC(N(CCC)C(c3oc(C)nc3C)=O)C2)=O)ccc(CC)nc1O 65342,c1(Cc2cn(C(C3CCOCC3)CC)nn2)coc2ccccc12 65343,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(CC(C)C)s1)=O 65344,C=CC(C)(CC)C(=O)NCc1ccc(CNC(=O)C(C)NC(=O)CC)cc1 65345,n1(C(C)(C)C)cc(Br)c(C(=O)Nc2ccccc2C(O)C(F)(F)F)n1 65346,c1(C(N(CC(C)CNC(C2C3CCCCCC23)=O)C)=O)cccc2c1C(=O)NC2 65347,c1(C(=O)N(C2(CNC(c3cncs3)=O)CCCC2)C2CC2)cc2n(c1)CCSC2 65348,C1(NC(C2CCCC(=O)N2)=O)CC2(C1)CN(Cc1cc(O)ncc1Br)C2 65349,C(=O)(CC(CC)CC)N(CCC(=O)NCC(CCC)NC(N)=O)CC 65350,C1(C(C)C)CN(C(=O)Cc2occc2C)CC1NC(c1ccc(CCF)cc1)=O 65351,C1(OC2CC(CC(=O)NCC)C2)CCN(C(=O)COCc2cccnc2)C1 65352,Cc1c(C(=O)NC(c2ccccc2F)CNC(c2cscn2)=O)cnn1CCO 65353,CCC(C)CC(C)C(=O)NCC=CCNC(c1n[nH]c(C)c1Cl)=O 65354,c1(C(=O)NCCCCNC(C2C(c3c(C)cccc3)C2)=O)ccc(F)c(C)c1O 65355,Cc1cnc2n1CC(C(=O)NCC(F)CNC(c1csc(Br)c1)=O)CC2 65356,C(=O)(CCP(C)(C)=O)NC1C(=O)NCC1.C(C)(COCCO)=CC 65357,c1(C(=O)NC2CN(C(C3(C)CC3)=O)C2)ccc(Cl)c(CC2CCCO2)c1 65358,c1(OC)cccc(Br)c1CNC(=O)CCNc1cnc[nH]1.N12CCC(CC1)C2C 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65480,CC1(C)CCC(CC(=O)NCc2cc(C(=O)NCC3CCCO3)n[nH]2)C1 65481,C1(C(N(CC(C)C)Cc2ccncc2)=O)CCCCC1CNC(C1CCC(O)C1)=O 65482,O=C1COC2(CCN(c3nc(N4CCC=C(F)C4)c4cccc(F)c4n3)CC2)N1 65483,C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1CCN(C(c2c(C)csc2)=O)C1 65484,N1(C(N(C)CCN(C)C(C2(C)CC2Br)=O)=O)CCOCC1 65485,C12(NC(C(c3ccccc3)N(C)C)=O)CC(C1)N(C(c1cccnc1O)=O)C2 65486,N1(C(c2ccc(CSC)cc2)=O)CC2CC(NC(=O)CCC3CCCO3)CC1C2 65487,C1(NC(C2OCCN(C)C2)=O)COCCN(C(=O)CN2CCSCC2)C1 65488,C1(CNC(C(C2CC(C)(C)C2)OC)=O)(CO)CCN(C(c2ccc(Cl)s2)=O)C1 65489,C(=O)(CCC(C)(C)C)N(CC(C)C)CC(=O)NCC1(CO)CCOC1 65490,c1(C(N)=O)cc(N2CCC(CC3CCCN3)CC2)cc([N+](=O)[O-])c1 65491,c1(C2C(C(=O)OC)CC(F)(F)C2)cc(C)nc2nc(C)nn12 65492,N1(C(C(C)O)=O)CC(CNC(=O)C(=O)Nc2ccc(Br)cc2)C2(CCC2)C1 65493,Cc1cc(C(=O)NCC(O)CNC(C2NC(=O)OC2C)=O)ccc1C1CC1 65494,N1(c2cc(NCc3cc(C)ncc3)ncn2)CCc2cccc(Cl)c2C1 65495,N1(C(CC(C)SC)=O)CCC(NC(=O)CCc2ccc(F)cc2F)C2(CCC2)C1 65496,C1(NC(C(C)SCC)=O)(CF)CCN(C(=O)CCc2cncc(Br)c2)C1 65497,C(=O)(CCC(C)(C)C)NCC(CN(C(CCc1scc(C)n1)=O)C)O 65498,N1(C(C(C)(C)c2cccnc2)=O)CC2CCC2(CNC(=O)CCc2nccs2)C1 65499,c1(C(N2CCC(NC(C34CC(COC)(OC3)C4)=O)CC2)=O)nn(C)c(C)c1Br 65500,c1(C(=O)NCC(C2CCC2)NC(c2nccc(CC)c2)=O)cnc2n1CCC2 65501,c1(CN2CCC(NC(c3c(C)nc(OC)s3)=O)C(F)C2)ccc([N+](=O)[O-])cn1 65502,Cc1ccc(C)n1CC(=O)NC(C)CN(C(=O)CC1CC(=O)NC1=O)C 65503,CCC(C)(COC)C(=O)NC(C)CCCNC(c1ccn(C(C)C)n1)=O 65504,C1(C(=O)NC(C2CCCN2C(c2cnc(C(C)(C)C)o2)=O)C)CS(=O)(=O)C1 65505,CCCCCCC(C)NC(C1(C)CN(C(=O)CCc2cccc(O)c2)C1)=O 65506,Cc1cc2c(CC(=O)NC3CC(NC(c4cc(C5CC5)sn4)=O)C3)csc2s1 65507,C=CCC(CC(=O)N(CCCF)C)NC(c1coc(N(C)C)n1)=O 65508,C12(OC)CCCCC(C(N3CCC(NC(=O)CCCF)C(CO)CC3)=O)(C1)C2 65509,C1(C(=O)NCC2(NC(CC3(C=C)CCC3)=O)CC2)CCC(=O)NC1CC 65510,N1(C(c2nn(C)c(Cl)c2)=O)CCC(F)CC1C(=O)NCCc1ccncn1 65511,C1(C(N(CCCNC(C2(F)CCCC2)=O)C)=O)Cc2cccc(OC(F)F)c2O1 65512,c1(C(N(C)CC2COCCN2C(C2CC23CCC3)=O)=O)cc2c(nn1)CCCO2 65513,c1(C(=O)NCCN(C)C(C2C=CCCC2)=O)nn(C(C)(C)C)cc1Br 65514,c1(C(=O)NC2(CNS(C)(=O)=O)CN(CC)C2)cc(NC(C)C)ccc1C 65515,CC1=C(C(=O)N2CCCC2C(C)NC(C2CC3COCC(C2)C3)=O)CCS1(=O)=O 65516,c1(C(=O)NCC2(NC(=O)CC(=O)Nc3nccs3)CC2)cc([N+](=O)[O-])c[nH]1 65517,C(N=c1[nH]c(N2CCCOCC2)nc(=N)[nH]1)c1cc(C)c(Cl)cc1 65518,N1(c2ccnc(C(C)C)n2)CCCC(C)(CNC(=O)CC2(C)CC2(Cl)Cl)C1 65519,c1(OC)ccc(Cl)cc1C(=O)N(C1CCC(NC(=O)C(C)(C)c2cnc[nH]2)C1)C 65520,C1(C2(C(N(CCN(C(=O)C=Cc3ccco3)C)C)=O)CC2)CCN2CCOCC12 65521,N1(C(C(C#N)C2CC2)=O)CCC2(C1)CN(C(c1cnc3[nH]ncc3c1)=O)C2 65522,c1(C(=O)NC2(CNC(CC#N)=O)CCC2)cc2n(n1)CCCNC2=O 65523,N1(C(=O)C=Cc2cncc(O)c2)CC2CCC1CN2C(C1CC1(CC)CCO)=O 65524,Cn1c(C(=O)NC2(C3CCC3)CC2)ccc1C#N.N12CCOC(C1)C2=O 65525,N1(C(C2CCCN(C)C2)C(=O)NC2CCCCCC2)CCCCC2(CCC2)C1 65526,C1(NC(C(C)NC(c2ccoc2)=O)=O)CC2CC1N(C(=O)NC1CCC1)C2 65527,N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCCCn2cncn2)=C(F)C1 65528,Cc1cccc(C(=O)NC(C)CCN(C)C(c2ccccc2Br)=O)c1C 65529,[N-]=[N+]=NC1CN(C(=O)CC2CCCCC23CC3)CC1NC(=O)Cc1cccnc1Cl 65530,C(CC(C)(O)CNC(=O)C(O)CNC(C1CCCN1C(C)C)=O)OC 65531,N1(C(C(CC)OCC)=O)CCC(C)(CNC(c2cnc(C)[nH]2)=O)C1 65532,C(C)(CCC(=O)NCCN(C1CCCC1)C(c1cnc(C(C)(C)C)[nH]1)=O)OC 65533,c1(NC(c2n(C)c(N3CCC(c4ccon4)CC3)nn2)=O)ccc(Cl)c(F)c1F 65534,N1(C(C2CN(C(C)C)C2)=O)CCC(C)(C(=O)N(CC(Cl)Cl)C)C1 65535,C(C)(C(C)C(=O)N1CCOC(CC)C1)NC(c1ncn(CC)c1)=O 65536,c1(C(N(C2CCN(C(=O)CC3CCNC3=O)C2)CCC)=O)ccc(CC2CC2)s1 65537,c1(C(=O)NCC(C)CNC(c2nsnc2O)=O)sc2sccc2c1Cl 65538,C(=O)(CCCCCCCC)N1C(CNC(c2c(CC)c(C)sc2)=O)CC(O)C1 65539,C#CCCCCC(=O)NCC(CNC(C1CCCC(O)C1)=O)C(F)(F)F 65540,N1(C(CC23C(CN(C(CC(C)OC)=O)C2)CC3)=O)CCC(C#N)CC12CC2 65541,C1(C2(O)CN(C(c3cc(C)cc(C(F)F)c3)=O)C2)(CNC(CCOC)=O)CC1 65542,N1(C(c2c(COC)ocn2)=O)CC(C)CN(C(=O)CC(F)F)C(C)C1 65543,C(=O)(C1CCCc2ncccc21)N1CCC(N(C(CC)=O)CCO)CC1 65544,c1(C(N2CCOCC2CCNC(c2ccsc2Cl)=O)=O)cnc2sccn2c1=O 65545,N1(C(c2cc(CNC(CSCCC(C)C)=O)[nH]n2)=O)CCN(C)C(CO)C1 65546,c1(NC(c2nc(CC)c(C)s2)c2nnnn2CCOC)cnn2c1C(=O)NCC2 65547,N1(C(C2CN(CC)c3c2cccc3)=O)C2CCC1CN(C(C1CCC1)=O)C2 65548,C(=O)(CCCCCC(C)C)N(CCOC)CCNC(=O)C#CC1CCOC1 65549,C(CS(C)(=O)=O)NC1C(C(=O)OCC=CCC)CC1 65550,c1(N(C2(CC(=O)O)CCC2)CC2CC2)cccc(Br)c1OC(F)(F)F 65551,CCC1=NOC(C(N2CCCC(N(CCF)C(c3cn(C)cn3)=O)C2)=O)C1 65552,N1(C(c2c(C)nn(C(C)C)c2)=O)CCC(CNC(=O)COC2(C)CCC2)C(C)C1 65553,c1(OC)cc(C(=O)N(C)CCN(C)C(c2cc(N)ccn2)=O)cc2cnn(C)c12 65554,c1(CNC(C2CCN(Cc3cc(O)cc(Br)c3)C2)=O)ccc2c(c1)C(=O)CC2 65555,CONC(=O)CNC(C1(F)CN(C(=O)CC(=O)C(C)C)C1)=O 65556,C1(C(=O)NC2CN(C(c3c(CC)noc3)=O)CC2C)CC2CCCC(C1)C2 65557,CC(C)CC(=O)C(=O)NC1CCCC(C(N2CCCC2C(=O)N(C)C)=O)C1 65558,c1(N(CC(=O)N(CC2CC(=C)C2)CC)CC)n[nH]c2c1COC2 65559,C1(CC)CN(C(=O)C(CCCOC)NC(CCC=CC)=O)CCN1C 65560,CC1CC(NC(=O)Cc2csnn2)CN1C(=O)CCCN1CCOC1=O 65561,c1(C(=O)NC2C=CCN(C(=O)C(C3(O)CCCCC3)(F)F)C2)cc(F)ccc1F 65562,CC(C)C(C(=O)NC(C)(CO)C1CCC1)N(C)C 65563,c1(SC)cc(C(=O)NC(C)C(C)NC(c2conc2-c2ccccc2)=O)c(C)o1 65564,Cc1ccc2nc(C(=O)NCC(C)CNC(c3ccn4ccsc34)=O)ccc2c1 65565,CC(C)(CNC(C1CC(CC2CC2)C1)=O)CC(=O)NCc1cc(O)ccc1F 65566,C(C(C)(O)CC(=O)NCC1(CNC(=O)CC(F)F)CC1)OC 65567,c1(C(=O)NCC(C2CCCCC2)NC(C(C)NC(N)=O)=O)cc2scc(Cl)c2[nH]1 65568,C1(OC)CN(C(N2CSCC2=O)=O)CC1NC(=O)CC1CCN(C)CC1 65569,c1(OCCNC(N(C2CCN(C(=O)OC(C)(C)C)C2)C)=O)cccc(Br)c1Br 65570,CN1CC=CCC1CC(N1CC(N(C(=O)Cc2ccsc2)C)C(O)C1)=O 65571,C1(CNC(c2cc(OCC)no2)=O)CCCN(C(=O)Cc2ccccc2F)C1 65572,c1(C(C(=O)NC2CC(C(=O)OC)C2)N(CCC)C)csc(C(C)(C)C)n1 65573,C(C(C(C)(C)C)NC(c1cc(C)ns1)=O)NC(c1ccc(C)o1)=O 65574,CCC(C)C(O)C(=O)N1CCC(CNC(=O)CO)C12CC2 65575,CCCCCCC(=O)NCC1(C)CCC(NC(=O)Cc2scnc2C)C1 65576,N1(C(C2CCC(OC)CC2)=O)CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1 65577,N1(C(=O)COCC2CC2)CC2(CCN(CC3C=CCCC3)CC2)C1 65578,Cc1[nH]cc(C(N2CC=CC(NC(C3(O)CC4CCC3C4)=O)C2)=O)c(=O)c1Cl 65579,CC1=NS(=O)(=O)NC=C1C(=O)N1CC2CC1C2NC(=O)CC(O)C(C)C 65580,C(=O)(CC(C)(O)COC)N(CC(CC)NC(=O)C=Cc1cc[nH]c1)C 65581,N1(C(C(C)OCC)=O)CCN(C(=O)CCCOC(C)(C)C)C(CC)C1 65582,CC(CC(C)(C)C)N=c1[nH]c(=N)[nH]c(=NCc2csc3ccc(Cl)cc23)[nH]1 65583,c1(CCC)nnc(Cn2nc(C)cc2C)n1CC(C)(C)SCc1ccccn1 65584,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(OCC(=O)NCc2c(OC)cccc2)C1 65585,C1(C(=O)NC2CC3(C(C(=O)NC4CC(CC(=O)OC)C4)C3)C2)CCCCC(=O)C1 65586,CC1CC(C(N)=O)CN(C(=O)NC(=O)OC(C)(C)C)C1.C12CCC=CC1N2 65587,C1(NC(C(C)=C(C)C)=O)CCN(C(c2csc(C)n2)=O)C(c2ccccc2)C1 65588,CCC(O)C(C)C(=O)NCCCN(C1CCCC1)C(c1cnc(C2CC2)[nH]1)=O 65589,N1(C(C(NOC)=O)=O)CCCC1C1CCCN1C(c1c(OC)ccnc1O)=O 65590,N1(C(C2(c3cccc(-c4c(C)ccs4)c3)CC2)=O)CCC2(CC1)OCCO2 65591,c1(C(CC)CC)cn(C2CCN(C(c3cn(-c4nccs4)nn3)=O)C2)nn1 65592,c1(OC)cnc(F)c(C(N2CCC(CC(=O)Nc3cncc(F)c3I)CC2)=O)c1 65593,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)N(C)CC1CCOC1 65594,c1(C(=O)NCC2(NC(C3(C=C)CC3)=O)CCC2)c(Cl)c(-c2ccccc2)nn1C 65595,C1(NC(C2CCC(C)S2)=O)(CNC(c2cncc(F)c2Cl)=O)CC2CCC1CC2 65596,c1(N(C(C2N(C(C(C3CCCC3)OC)=O)CC(F)C2)=O)C)ccc(O)cc1C 65597,Cc1cc(CC(N2CC(NC(C3CC(C)(O)C3)=O)CC2(C)C)=O)cc(C)c1 65598,C(=O)(CC(O)C(C)C)NCCN(C(=O)Cn1ccc(O)nc1=O)CC 65599,N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(C2CCC2)nc1)=O 65600,Cc1ccc(-c2cn(CC(CC(C)C)NC(C3CCC(CO)O3)=O)nn2)cc1C 65601,c1(C(N2C(CNC(C(C)(C)O)=O)CC2)=O)ccc2nnc(C(F)F)n2c1 65602,N1(C(=O)Cc2cnc3ncccn23)CCN(CCNC(=O)CC(F)(F)F)CC(O)C1 65603,C1(CNC(CSCC=C)=O)COCC1NC(=O)CSCCC#N 65604,C(=O)(C#CC1CCCC1)NC1(COC)CCCN(C(=O)C(=C2CCCCC2)F)C1 65605,CC(C)C1=CCC(NC(C2(NC(=O)C=Cc3ccncc3)CCN(C)C2)=O)CC1 65606,C(=O)(CC#CC(C)=O)N1C(C(=O)NC(c2ccccc2)C#C)COCC1 65607,C1(CNC(C(C(C)O)(F)F)=O)CC2(CO1)CN(C(=O)C(F)(F)CO)C2 65608,C(=O)(CCC(C)(C)F)OC(C1CCCC1OC)C(=O)OC 65609,n1(SCC)ncc(NC(C)=O)c1C.N12CCN(CC1)C(=O)N(C)CC2 65610,N1(CC2CCC(C)O2)CCC2(CCCCC2NC(c2cc3occc3[nH]2)=O)CC1 65611,N1(C(C2C(OC)CC2)=O)CC(NC(c2ccc(Cl)c(F)c2N)=O)C2(CCC2)C1 65612,N1(C(C(N2CCOCC2)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 65613,CC1CC(C(=O)NCC2C3CN(C(c4ccc(Cl)nn4)=O)CC23)CCC1C 65614,N1(C(C(C)SC(C)C)=O)CCN(C(c2ccc(CO)s2)=O)CC1CO 65615,C1(C#N)(C(N2CC(CC)(NC(c3cncc(CO)c3)=O)C2)=O)CCN(C)CC1 65616,c1(OC)ccc(C(N2CCCC2(C)CNC(C2CC2OC)=O)=O)cc1[N+](=O)[O-] 65617,C(=O)(C(C1(C)CC1)NC(=O)C(C)N(CC(C)C)C(C)C)NC(C(C)SC)=O 65618,NS(=O)(=O)N1CCCC(C(=O)NCC(O)CNC(c2c[nH]c(C(N)=O)c2)=O)C1 65619,c1(CC(=O)NCCCC2C(C)(C)CCN(CC)C(=O)C2)scnc1C 65620,CCCCCCCCCCCN(C)C(C1CCN(C(=O)C(C)CCCC)C1)=O 65621,Cc1ccccc1C=CC(=O)NC(C)CCN(C)C(C1CC2CC2C1)=O 65622,c1(C(N2CCC(NC(CN(CC)CC)=O)C(O)C2)=O)cccc2c1OCCO2 65623,c1(SC)cc(C)c(C(N2CC(CNC(C3(C)CCOC3C)=O)C(O)C2)=O)o1 65624,CC1N(CCN2CCCNCC2)CCOC1(C)C 65625,CCCCC(C(=O)NCC(CC(N1CC(CO)CC(C)(C)C1)=O)OC)C(C)C 65626,C(C)(CC(=O)NC1CCCC1NC(c1cc(N)c(F)cc1F)=O)(C(F)F)N(C)C 65627,C1(C(=O)NC2CC(C(=O)NCC3CN4CCC3C4)C2)CC2(CCO1)CC2 65628,C1(NCCc2n[nH]c(=NC)s2)CCC(O)CN(C(c2c[nH]c3ccccc23)=O)C1 65629,n1(C(C)C)nccc1CN1C(CN(c2cnns2)C(=O)NC2CCCO2)CCC1 65630,C1(NC(C(CC)C)=O)CCCC(C(=O)Nc2ccc(Br)cn2)C1 65631,CC1(C)CN(C(C(=O)NCCC2CC2)CCCC2CC2)C2COCC12 65632,N1(C(c2c(C)ncs2)=O)CCC2(CC1)CCN(C(c1csc(C)c1C)=O)C2 65633,c1(CC(=O)NC(CNC(C)=O)CO)ccc(Cl)s1 65634,Cn1cnc2nc(=NCc3ncc(F)cc3F)[nH]c(NCc3cccc(Cl)c3F)c12 65635,C=CCC(CC(F)F)C(=O)N1CC=CC(NC(c2sncc2C)=O)C1 65636,C12(C(=O)NC(C3CCCN(C(c4cnc(Cl)s4)=O)C3)C)CC3CC(C(=O)N1)C2C3 65637,c1(C(=O)NCCCC(=O)NCC(CO)C2CCC2)ccc(F)cc1[N+](=O)[O-] 65638,C1(=O)NNc2nccnc2N1.Cc1noc2ccc(CNC(=O)C(F)(F)F)cc12 65639,c1(OC)ncccc1C(N1CC(CNC(C2(n3cc(Cl)cn3)CC2)=O)CC1C)=O 65640,C1(C(N2CCC(O)(CNC(COCC#C)=O)C2)=O)CCc2nnn(C)c2C1 65641,c1(C(=O)NC2CCN(C(C(CCC)C)=O)C(C)(C)C2)cc(C)cc2c1OCC2 65642,C#CCC(C)(CC)C(=O)NC1COCCC1C(N1CCOC(C)C1)=O 65643,CCC(CC(=O)NC1CCC(NC(=O)C(C)(C)CN(C)C)C1)C1CCC1 65644,c1(CNC(C(C=C=C)C)=O)nc2c(s1)CN(C(C1(C(=O)OC)CC1C)=O)CC2 65645,c1(C(N2CCC(N(C(c3sc(O)nc3C)=O)CC)CC2)=O)ccc2ncccc2c1 65646,CC1(C)CCOC(C(N2CCC(C3CC(NC(=O)CC#N)CCO3)CC2)=O)C1 65647,O=C(CC(F)(F)c1ccccc1)NCC(O)CNC(=O)C(O)CF 65648,c1(C(=O)NCC2(F)CCN(C(C3CC(OCC)C3)=O)C2)ccc(C)c(C)c1 65649,C12(C(=O)NCCC(C)(C)CNC(C3CN(C(N)=O)C3)=O)CCCCC1OCC2 65650,C1(C(=O)NCc2nccn2C)(NC(CN(C(C)=O)C)=O)CCC(C)CC1 65651,C(CC(=O)N(C1(CC(=O)NCC(C)CN2CCCC2)CC1)C)OC 65652,C1(NC(C(CC)c2ccccc2)=O)CCCCC1NC(c1cc(C)n(CC)n1)=O 65653,C1(CCNC(CC2CC(OCC)C2)=O)CN(C(c2ncn(CC)n2)=O)CC1C 65654,C1(NC(C(C)(C)CF)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC1c1ccccc1 65655,c1(C(N(C)CC2CCCCN2C(=O)C(C)(C)C2CC2)=O)cnc2ccccc2n1 65656,C1(CC)CN(C(=O)C=Cc2cnccn2)CCN1Cc1nc(Cl)ccc1Cl 65657,C(CCOCCO)(C(=O)N1CC([N+](=O)[O-])(O)C1)NC(=O)C#CC1CC1 65658,c1(NC(C2N(C(C=CC(C)C)=O)CC(O)CC2)=O)cnc(C)c(C#N)c1 65659,c1(N2CCC(N3CCC(=O)NC3=O)C2)cc(=O)n2ccccc2n1 65660,C1(O)(CNC(C2CCC(=C)CC2)=O)CCCN(C(c2ccc(Br)cc2F)=O)C1 65661,c1(OCC)cc(C(=O)NC(CCN(C(=O)C(C)OC)C)C(C)(C)C)oc(=O)c1 65662,N1(C(c2c(C)n(CCC(C)C)nc2)=O)CCCC(NC(C2CC(C)(F)C2)=O)C1C 65663,c1(C(=O)NC2C(NC(c3cc(C)sn3)=O)CCC2)ccc2c(c1)CN(C)C2 65664,c1(C(N2CCC(NC(c3cncc(C(C)C)c3)=O)CC2)=O)nnn2c1CCC2 65665,c1(C(=O)NC(c2ccsc2Cl)COC)cnn2c(Cl)cccc12 65666,Cn1cc(C(=O)NC2C3CC(NC(=O)CCC4CCC4)CC23)nc1C=O 65667,c1(C(N2CCC(CNC(C3(C(CC)=O)CC3)=O)C2)=O)ncccc1-n1cccn1 65668,C(=O)(C1=CCCCC1C)NC(CNC(c1occ(C)c1)=O)Cc1ccccc1 65669,Cc1nc(Cl)ccc1S(=O)(=O)NCC1CN(Cc2cccc(O)c2O)CCO1 65670,c1(-c2c(CC(N)=O)csc2)ccc2c(c1)CN(Cc1ccc(F)cc1)CC2 65671,Cc1cc(F)c(Cl)cc1C(=O)NCC(C)CN(C)C(c1ccc(C#N)nc1O)=O 65672,c1(C(=O)NCC2C(N(C)C)CN(C(C3CCCO3)=O)C2)cc(C#N)c(C)cn1 65673,N1(C(C=CCC)=O)CCN(C(c2cnn(CC)c2CC)=O)C(CC)C1 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65692,c1(CC#N)ccsc1C(=O)NC(CNC(c1ccc(Cl)o1)=O)C1CC1 65693,C(=O)(C(=O)N=S(C)(C)=O)N1CC(NC(CC2CCC(C)CC2)=O)C(C)CC1 65694,N1(C(c2n(C)nc(Br)c2)=O)CCOC2(CCCCC2NC(C2CCOCC2)=O)C1 65695,CCCC(CCC)C(=O)NC(CNC(=O)COc1ccccc1CC)C(C)(C)C 65696,N1(C(CC)=O)CC(NC(c2cccnc2OC)=O)CC2(CCOCC2)C1 65697,N1(C(=O)NOCC(F)F)CCC(OC2CCOC2)CC1 65698,N1(CCC#C)CCCC1C(=O)NCCN(CCC)C(c1coc(CCC)n1)=O 65699,CC1CN(C(C2(O)CCSC2)=O)CC1CCNC(c1cc(-c2ccoc2)on1)=O 65700,c1(-c2cn(C)nc2)ccccc1NCC1CN(c2ccc(F)cc2)C1 65701,N1(c2ccc(C)s2)CC(C(N2CC3CC2(c2ccnn2C)C3)=O)CCC1=O 65702,C1(C(=O)NCc2cn(CC(=O)NCC(O)C(F)(F)F)nn2)CC2C(C1)C2(F)F 65703,C1(N(C(C2CC=CCO2)=O)CC)CCN(C(=O)C(F)OC(F)(F)F)CC1 65704,c1(CC(C(=O)N(C(C)CNC(C2CC2F)=O)C)C)ccc([N+](=O)[O-])cc1 65705,Cc1cccc2[nH]cc(C(=O)NC34CC3CN(C(C3CCC3)=O)C4)c12 65706,C1(=O)CCC(F)(F)C(=O)C(=O)C(F)C(=O)NCCN1CC(=O)OC.OC 65707,C1(C(=O)NC(C(C)C)c2nc[nH]n2)CCN(C(=O)CC(=O)NCC2CC2)CC1O 65708,C1(CC(=O)NC2(C)CCN(C(=O)Cc3n[nH]c(=N)s3)CC2)CSc2ccccc2O1 65709,c1(CC(=O)NCC(CNC(C2(C)CC2)=O)O)ccc(N(C)C)cc1 65710,N1(C(c2c(CC)noc2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 65711,c1(SC)nccc(=NC(CNC(c2n[nH]cc2C2CCC2)=O)C(C)C(C)C)[nH]1 65712,CC(=O)CCN=C(NCCc1ccc(Cl)o1)NC1CN(C(=O)OC(C)(C)C)C1 65713,c1(NCC(C)(C2CC2)OC)nc(N2CCOC(c3ccccn3)C2)nc2sccc12 65714,C#CCC(CC(F)F)C(=O)NC1COCCC1N1CCCC1 65715,O=C(C1c2c[nH]nc2CN1C(c1cnc(O)o1)=O)NC1C2COCC12 65716,c1(C(N2C(C3(NC(COCCC)=O)CC3)CCCC2)=O)ccc2cnccc2n1 65717,C(=O)(C1=CCCSC1)N1CC(N(CC(=O)Nc2ccc(F)cc2)C)C1 65718,C1(NC(C2CC(Nc3ccnc(NCC4CC4)n3)C2)=O)CCOCC1F 65719,CCC(C)CC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1 65720,N1(C(Cc2c(C)ccs2)=O)C(C(=O)NCC(=O)NC(C)C)CC2CC12 65721,C#Cc1ccc(C(=O)N(C)CCOCCNC(=O)Cc2n[nH]c(=NC)s2)cc1 65722,C12(C(=O)NCC(=O)NC(c3ccc(F)c(F)c3)C(C)C)CCCN1CCC2 65723,C1(C(=O)NC2CCN(C(C(C)c3ccco3)=O)C2)CN2CCN1CC2 65724,C1(C(=O)NC2CC(Cn3ccnn3)C2)CCC(C#N)C1.C12CC(C1)C(=O)N(C)C2 65725,CCCCC(C)CCC(=O)NC1(COC)CCN(C(=O)CC2CC=CCC2)C1 65726,C(=O)(C(F)CCC(C)(C)C)N(C1(C(N2CCC(C(=O)NC)C2C)=O)CC1)C 65727,C1(CC(=O)NCC(CN(C(CC=C(C)C)=O)C)C)CCCC1C 65728,Cc1nnc(O)c(C(=O)NC2CN(C(c3cncnc3C(C)C)=O)CCC2C)c1C 65729,C1(NC(c2cc(CNC(C(CC)(C)OC)=O)sc2)=O)CCCCCC1F 65730,c1(C(N2CCN(CC(=O)NCCC(C)(C)C)CC2)=O)ncc(F)cc1N.C(N)(=O)N 65731,C1(CC(=O)NC(C)C(=O)NCC(C2CC2)OC)(CC)CCO1 65732,N1(C(C(C=C)(C)CCOC)=O)CCOC2(CCN(C(c3cncnc3C)=O)C2)C1 65733,N1(C(c2c(C)onc2-c2ccccn2)=O)CC2CC1CN2C(c1coc(Cl)c1)=O 65734,N1(C(COC(C)=O)=O)CCC(F)(C(=O)NC(Cn2cccn2)CO)CC1 65735,N1(C(C(C)CO)=O)CCN(C(=O)CSc2nc[nH]n2)CC1c1ccccc1Cl 65736,C1(NC(CCc2cc(C)no2)=O)CCN(C(c2cc(C)cnc2Cl)=O)CC1(C)C 65737,C1(C2(O)CN(C(C3(C(F)F)CCOC3)=O)C2)(CNC(=O)C2=C(Cl)CCC2)CC1 65738,C1(C(C)NC(=O)CC2CC2(F)F)CCCN(C(=O)CC2CC(F)(F)C2)C1 65739,N1(C(=O)CCc2cccnc2F)C2CCC1CN(Cc1ccc(O)c(O)c1O)C2 65740,c1(NC(CC)C)ccnc(N(C)C(=S)Nc2ccc(F)cc2)c1 65741,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(=O)CCn2ccccc2=O)CC(F)C1 65742,c1(OC)c(F)cc(C(=O)NC2(CNC(c3nc(Br)cs3)=O)COC2)cc1F 65743,CCCCC(O)CC(=O)N1CC(C)(C)CC1C(=O)NC1CCCC1N=[N+]=[N-] 65744,N1(CCNC(COCCC=C)=O)CCC(NC(c2sccc2OC)=O)CC1 65745,c1(OC(CN2C(NC(C(CC)=O)=O)CCC2)=O)cc(C(F)(F)F)cc(C(F)(F)F)c1 65746,C(CCC(O)C(=O)NC1(CC2CC2)CCC1)NC(=O)C(O)C1CCC1 65747,S(=O)(=O)(c1cccnc1NCCc1nnc(O)o1)NCC(C(C)(C)C)O 65748,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 65749,C(C(CO)C(C)CC)NC(C(Cn1cncn1)NC(c1n(C=C)nnc1)=O)=O 65750,c1(C(N2CCC(CNC(C3(N(C)C)CC3)=O)C2)=O)cccc2c1CCCC2 65751,C(=O)(C(F)C1=CCCCC1)NCCOCCN(C(Cc1c(C)cccc1C)=O)C 65752,N1(C(c2cnn(C3COC3)c2)=O)CC2(C(=O)O)CC1(CNC(=O)C(F)F)CC2 65753,N1(C(CC=C)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)C2(COC2)C1 65754,c1(C(=O)NC(CC)C(=O)NCc2ncnn2C)cc(C)cc(C#N)c1 65755,c1(C(C)OC(C2CCCN2C(=O)OC(C)(C)C)=O)cccc(C(F)(F)F)n1 65756,N1(C(CC2CCC(NC(C3CCCC3O)=O)C2)=O)CC(CO)C(O)C1 65757,c1(NC(=O)NCc2cc(=N)[nH]cc2)nc2ncccc2o1 65758,c1(C(=O)NCc2c(C3CN(C(C(C=C)O)=O)C3)ocn2)ccc(C2CC2)cc1C 65759,Cc1n[nH]cc1C(=O)NC1CCC(NC(C2(c3ccccc3)CCCC2)=O)C1 65760,CC(C)C(CCNC(=O)CCOCCN(C(=O)Cc1ccno1)C)OC 65761,c1(CC)nc(C#N)cc(=NC(C)C2CCN(C(C3CCC(N=[N+]=[N-])C3)=O)C2)[nH]1 65762,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 65763,Cc1n[nH]c2nc(O)c(C(=O)NC3(CNC(=O)C=CC(C)C)CCOC3)cc12 65764,N1(C(C(C)OCCC=C)=O)CC(O)C(O)C1C(=O)NC1CC(=C)CC1 65765,N1(C(CCC)=O)CCCC1CNC(C1(C(F)F)CC(O)C1)=O 65766,CC1(C)CN(C(=O)C(C2CCOCC2)O)CC1CNC(c1ccc(F)c(F)c1)=O 65767,C1(NC(C2N(CC)CCCC2)=O)CC2CCC(C1)N2C(c1c[nH]c(=NC)s1)=O 65768,c1(OC)cncc(C(=O)NC(C2CCN(C(=O)CC3CCC(=O)N3)C2)(C)C)n1 65769,c1(OCC(=O)N(C2CCCN(C(C3CC3F)=O)C2)CC)ccc(C(C)=O)c(Cl)c1 65770,c12sc3ccccc3c1CNC2=O.N1(C(C2(C)CC2)=O)CCC2(N(C)C)CC2C1 65771,CC1C(NC(=O)C(C)(C)C)C(C)CCN1C(=O)Nc1ccc(F)cc1I 65772,CC1CC(NC(=O)CCc2ncc(F)cn2)CN1C(c1ccnc(C(F)F)c1)=O 65773,c1(C(N(C2CCCN(C(=O)C(O)C(F)F)CC2)CC)=O)nc(C)c(C)nc1C 65774,N1(C(c2ccc(COC)cc2)C(=O)NCC=C)CC(C)OC(C)C1C 65775,N1(CC(=O)NCCCCNC(CCNC(=O)NC)=O)CCCC1C 65776,C1(NC(c2cccc(SCCC)c2)=O)CCN(C(c2cccc(CC)n2)=O)CC1O 65777,C1(CC)CN(C(C2(F)CC2)=O)CCC1NC(C1CCC(CCO)CC1)=O 65778,c1(NC(=O)C(N2CCCC(Cc3ccccc3)C2)=O)cc(Cl)cnc1Br 65779,C1(CNC(C2C(C=C)CC2)=O)CCCN(C(=O)CN(c2cncc(CC)c2)C)C1 65780,C(N=c1[nH]cnc2c1SCCC2)C1OCCN(C(c2c(C)nns2)=O)C1 65781,C(C(O)CCNC(=O)Cc1csc(C2CCCCC2)n1)NC(=O)CCF 65782,c1(C(=O)NC(CCCC)CNC(=O)C=Cc2ccnn2C)ccc(C#N)n1C 65783,N1(C(C2CC3(CCC3)C2)=O)CCN(CC2CCCN(C(c3cscn3)=O)C2)CC1 65784,c1(C(N2CCC(C)(NC(c3cnc(N(C)C)nc3)=O)C2)=O)cnc(O)cc1O 65785,c1(C(=O)NC2CC(NC(C3(S(N)(=O)=O)CC3)=O)CC2O)c(F)ccc2n[nH]cc12 65786,Cc1ccnc(C(N2CCCC2(C)C(N2CCCC(OC3CC3)C2)=O)=O)c1 65787,C12(C(N3CC(NC(C(=Cc4cccs4)C)=O)(CO)C3)=O)CCC(CO1)C2 65788,N1(C(C(=O)NCC)=O)CCC(C)(C)C1C(=O)N(C1CCC(C)(C)C1)C 65789,c1(NC(C2CN(C(c3n(C)c(S)nn3)=O)CC2F)=O)cccc2c1CCO2 65790,C1(C)(C(N(C(C)C(=O)O)CC)=O)CCN(C(c2csc(F)c2)=O)CC1 65791,CCC(C(=O)N(CCCNC(C1CCC(=O)NC1)=O)CCO)C(C)(C)CC 65792,c1(C(=O)NCCC(Cc2ccc[nH]2)NC(CC=CCC)=O)ccc(C#N)cn1 65793,c1(C(=O)NC2(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)n[nH]c2c1CSCC2 65794,c1(O)cccc(Br)c1.C1(C)(OCC(=O)NCC2C(C(C)NC=O)C2)CCC1 65795,c1(C(=O)NCC(C)NC(C2CCCC2C)=O)ccc2c(c1)B(O)OC2 65796,N1(C(=O)Cc2cnc[nH]2)CCC(CC2CC2)CC1.C1CO1 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65987,C(=O)(C(F)C(C)(F)F)NCCCOCCC(=O)NC(c1nc(O)n[nH]1)(C)C 65988,CC1COCCN1C1CC(NC(=O)NC(c2ccccc2)C)C1 65989,N1(C(CC=CC=C)=O)CC2CCN(C(C3CC(=O)N(O)C3)=O)CC(C2)C1 65990,CC(C(=O)NCC1(CNC(c2cc(N)c(F)c(F)c2F)=O)CC1)C(C)C(C)(C)C 65991,c1(C(c2ccnn2-c2ccccc2Cl)NC(C)CCC2CCCC2)ccc(F)cc1 65992,n1(CC)nccc1C=CC(=O)NCC(C)(C)CN(C)C(c1cc(=O)cc[nH]1)=O 65993,C(CCSC)(C(=O)OCCCSCC)NC(c1cc(-c2ccoc2)[nH]n1)=O 65994,C1(C2C(CC(=O)NC(C(N3C(COC)CC3)=O)c3ccoc3)C2)CCOC1=O 65995,c1(CCC(=O)N(CC(C)N(C(C(C)O)=O)C)C)ccc(Cl)cc1Cl 65996,CCC(C)(C)C(O)C(=O)NCC1CCN(CC(=O)NC(C)Cc2cccs2)C1 65997,N1(C(CC(C)C)=O)CCc2c(ncn2C)C12CCN(C(=O)CC(C)C)C2 65998,C1(CC(=O)NCCCN(C(=O)CCC2CCCO2)C(C)C)CCCOCC1 65999,c1(C(=O)OC)cc2c([nH]1)CCN(C(=O)CSc1ccc(N)c(C(F)(F)F)c1)C2 66000,C1(NC(=O)C=Cc2ccccc2Cl)CCSC12CN(C(=O)Cn1ncnn1)C2 66001,C12(C(=O)NCc3n(CCC)ccn3)CC(CN1C(c1nc(Cl)cs1)=O)C2 66002,C1(CNC(C(C)(C)OC)=O)CCCCN1C(C1CC(C(F)(F)F)C1)=O 66003,N1(C(C)C)CC(C(=O)N(CCCNC(=O)C(C)(C)n2cncn2)C)CC1=O 66004,C=C(C)CCCC(=O)NC(CNC(C1CCCN(CCC)C1)=O)CC 66005,C1(CNC(C(C)OCC2CC(C(=O)NC3CCCC3)CO2)=O)CC2(CCC2)C1 66006,C1(=O)C(C(C)C)NCCN1CC#C.c1(OCC(=O)NC)cccnc1 66007,c1(CNC(=O)CC2(CO)CC2)ccc2c(c1)CN(C(C1(F)CCCOC1)=O)C2 66008,CC1CC(C)(C(=O)NCc2cccc(NS(C)(=O)=O)c2)CC(C)O1 66009,N1(C(CCCC)=O)CCC(NC(=O)CCc2ccccn2)C1C(C)(C)C 66010,Cc1ccc(C2CC2)c(NC2CCC3CCC2O3)c1 66011,c1(C(N(C2CC2)CCCNC(CCS(C)=O)=O)=O)cc2scc(Cl)c2[nH]1 66012,C1(CC=C)CCCCN1.c1(CC)cn(C(=O)O)cn1 66013,c1(C2C(C(N(CCCCNC(=O)CCF)C)=O)C2)nccc2ccccc12 66014,C1(C)(COCC)CCCN(C(C2CC2CC(C)C)=O)C1.C12(CC1)CC(=O)N2 66015,CC1C(NC(=O)CC=Cc2cccc(F)c2)C(C)CCN1C(=O)C1CC1 66016,N1(C(CCC#CC)=O)CCCCC1C1CCCN1C(c1cc(C)ccn1)=O 66017,C#CCC(CC#C)C(=O)N1CCCCC(CNC(c2sc(C)cc2OC)=O)C1 66018,C1(C(=O)NC(C2(CNC(=O)C(C)(C)C(N)=O)CC2)C)SC2C=CC1CC2 66019,C1(C(N2CC(C)C(Nc3ncnc4sccc34)C2)=O)CCCC(F)(F)CC1 66020,N(C1CCCc2ccnc(Cl)c21)C(C(C1CCOCC1)N(C=O)Cc1ccco1)=O 66021,C1(C(=O)NC(c2n(CC)ncn2)C)CC(N=[N+]=[N-])CN1C(=O)Cc1ccsn1 66022,C12(N(C(CN(C)CC)=O)C3CCC3)CCN(C(c3ccccc3)=O)CC1C2 66023,CC1CCC(C)(N2CCCC2)C1.C12(C)CCN(C1)CC(=O)C(=O)CCn1cc2nn1 66024,c1(CNC(c2c(C)snc2)=O)cccc(C(=O)N(CC(F)F)C2CCC2)n1 66025,C(C)(C(CC(=O)NC1(C)CC(C)(C)C1)NC(=O)C(C)C(F)(F)F)OC 66026,CC1CN(C(c2ccc(Br)o2)=O)CC1NC(c1cn(C(C)(C)C)nn1)=O 66027,C1(NC(c2c(C)n(C)cn2)=O)CC2CCC(C1)N2C(=O)CC1OC(=O)NC1(C)C 66028,N1(C(COC)=O)CC(NC(=O)CCCOC(C)C)CC12CCCOC2 66029,N1(C(c2n(CC=C)ccc2)=O)CC(O)CC1CNC(=O)COCCOCC 66030,c1(CC(C(=O)NC2(CF)CC2)NC(Cc2ncc(CC)[nH]2)=O)ccccc1Br 66031,C12(CNC(CCC(CC)C)=O)COCCN1CCN(C(C1(C)CCOCC1)=O)C2 66032,N1(C(C(=O)NC2CC2)=O)CCC(C(N2CCC(CC(F)F)C2)=O)(CO)C1 66033,c1(NC(C2CCCC(NCc3ccc(F)c(Br)c3F)C2)=O)cc2ccccc2[nH]1 66034,Cc1n[nH]c2cnc(C(=O)NC3CC(CNC(=O)C=C4CCN(C)CC4)C3)cc12 66035,N1(C(C2CN(N(C3CC(C#N)C3)C(COCC)=O)C2)=O)CCC(CN(C)C)C1 66036,c1(C(N2CCCC(N(C(C(CC)SC)=O)CC)C2)=O)cnc2c(cnn2C)c1N 66037,c1(C(N2CCC(CCNC(c3cnc(C(N)=O)s3)=O)C2)=O)cnc2n1CCS2 66038,C1(NC(C(CC)Oc2cccc(F)c2)=O)CCN(C(C2(C)C=CCC2)=O)CC1C 66039,C1(CC)C(NC(=O)CN(CC(C)(C)C)C)CCCN1C(=O)C(C)CC(N)=O 66040,N1(Cc2ccc(OC(C)C)nc2)CCC(=O)N(Cc2ccc(Cl)o2)C1=O 66041,N1(C(CC(=O)NCC)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CC2 66042,c1(C(C)NC(=O)CC2CCCCCC2)ncccc1NC(C1CCCCO1)=O 66043,C1(C)(C(N(CCCCN(C(=O)CCc2ccncc2)C)C)=O)COC(=O)OC1 66044,CCCCCC(O)CC(=O)NC(CNC(C1(C(F)(F)F)CC1)=O)(CC)CC 66045,C1(NC(c2cc(C3CC3)cnc2Cl)=O)CCC2CCN(C(c3csnn3)=O)C1C2 66046,CCCCCCN(C(C1CC(C)(NC(=O)C(OC)OC)C1)=O)CC 66047,c1(C(N(CCCN(C(C2CC(SC)C2)=O)C)C)=O)c[nH]c2cccc(F)c12 66048,C1(NC(C2C(C)CC2)=O)CCC(N(C)C(c2cnsc2)=O)CC1 66049,CCC(=O)CCC(=O)N1C(CC(=O)NC(C2CCOCC2)C)C2CCCC12 66050,N1(C(C(C(C)C)SC)=O)CC2CCCC(C1)N2c1ncccc1C 66051,c1(C(=O)NC(C)CC2CCC2)ccccc1.C12CC1C2 66052,N1(C(Cc2ncc(CC)[nH]2)=O)CCCC(N(C(=O)CC2CCOCC2)CCF)C1 66053,N1(C(CC2(C)CC2(Cl)Cl)=O)CC(NC(c2ccnc(OC(F)F)c2)=O)CC1CO 66054,C1(CNC(C(=O)NCC)=O)CN(C(=O)Cc2ccc(CC)c(C)c2)CC12CC2 66055,c1(C(N2CCC(C(CO)NC(CCC(C)SC)=O)CC2)=O)ccc2occc2n1 66056,C(=O)(C(O)C(F)(F)F)NCC1C(C=O)C1.C1(C(N(CC)CC)=O)CCOCC1 66057,C12(C(=O)NCc3nc(C)[nH]n3)CC(CN(C(C3CCSC3)=O)C1)C2 66058,c1(N(CCN(C)C(c2cnn(-c3ccccc3)n2)=O)C)cnc(C(F)F)cn1 66059,Cc1cccc(C)c1C(N1CCCC(Nc2cc(Cl)ncn2)C1)=O 66060,C(CC(C)C(=O)NC1CCCCC1C(=O)NOCc1[nH]c(C)nc1C)=CCC 66061,N1(C(c2c(Cl)cn(CC)n2)=O)CCCC(CCNC(=O)CN2CC(C)(C)C2)CC1 66062,C1(CC(=O)NCC(CC)NC(C2(c3ccno3)CCC2)=O)CC(C)(C)CO1 66063,CC1CN(C(=O)CO)CCC1NC(c1nn(C)nc1Br)=O 66064,c1(OC)cc(C)cc(-c2cn(C3(CC(O)C4CCC4)CC3)nn2)c1C(=O)O 66065,Cc1cc(C(F)(F)F)nc(NC(C2CSC(=O)N2)=O)n1 66066,N1(C(CCC(=C)Br)=O)Cc2ccccc2C(NC(c2cnc(C)nc2C)=O)C1 66067,c1(C(N2CCC(C)C2CNC(=O)CSC2CCOC2=O)=O)ccc2nncn2c1 66068,N1(C(CC=CCCCCC)=O)CCCC1C=CC(=O)NC(c1nnc(C)o1)C 66069,CC(C)S(=O)(=O)CCCn1c(-c2ccc(SC(F)F)s2)nnc1C1CCCC(O)C1 66070,C1(NC(C2(C(C)NC(c3cncc(Cl)c3)=O)CC2)=O)CCN(C)CC1C#N 66071,c1(C(=O)OC)scc(C)c1NC(N1CCC(C(=O)N(C)C(C)C)C1)=O 66072,C1(NC(C2CCCNS2(=O)=O)=O)CCC2CC1CN2C(c1ccncc1)=O 66073,n1(CC(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)cnc([N+](=O)[O-])c1 66074,CC1(C)CCCCC1C(=O)NCC1CC(NC(C2CCC23CCC3)=O)C1 66075,N1(C(c2scc(C)c2)=O)CC=CCC1C(N1CC(CC2CCCC2)C1)=O 66076,Cc1[nH]nc(C(F)F)c1C(=O)NCC(C#N)CCNC(=O)N(C(C)(C)C)C(C)C 66077,C1(F)(CNC(C(C)SC)=O)CCN(C(=O)C(C)(O)C2CC2)CC1 66078,C(=O)(C(C)(C)CCC#N)NC1CCC(CNC(C(CSC)O)=O)CC1 66079,N(C1CCc2ccccc21)C(C1(C)N(C(C2CN(C(C)=O)C2)=O)CC(O)C1)=O 66080,c1(C(N2CC(OCCC(=O)NCC(F)F)C2)=O)nc2cc(F)ccc2s1.C1CO1 66081,N12CC3(C1)CN(C(=O)CO)CC3COC(C)C2=O.CC(C)C=CC=O 66082,C1(CC(=O)NCCCNC(C2COCCC2(F)F)=O)CCn2cncc2C1 66083,Cc1cccc(C(F)C(=O)NCC(C)N(C(=O)CN2CC3CC3C2)C)c1 66084,Cn1cnc2c(NCC3C4CN(C(c5ncoc5C5CCC5)=O)CC34)ncnc12 66085,c1(C(N2CCC(C(=O)OCC)C2)=O)cccnc1OCC.C1(C)CN1 66086,Cc1ccc(C(=O)NCCCN(C(C2CCS2(=O)=O)=O)C2CC2)cc1 66087,N1(C(c2c(C)noc2C)=O)C2CCC(C(=O)NCCC3CCCCC3)C1CC2 66088,C(=O)(CCN=c1cc[nH]c2ccc(C#N)cc12)NC(C)C 66089,N1(CC)N=C(C(=O)NCC(C)NC(c2cc(C)nc(N(C)C)n2)=O)CCC1=O 66090,c1(C(=O)NC2(CNC(C3(SC)CC3)=O)CCC2)cc2ccc(Cl)cc2c(O)n1 66091,C(=O)(C(CC(C)C)NC(=O)CC(COC)NC(=O)C(C1CCCCC1)O)NC 66092,c1(C(=O)NCC(C)NC(C2(N(C)C)CC2)=O)cc(-c2ccccn2)on1 66093,C(C(C)(CC)C(=O)Nc1cnc(C(C)C)nc1)NC(c1ccc(NC)cn1)=O 66094,c1(C(=O)NC(CC(F)F)C(=O)NCC(Cl)=CCl)ccc2n[nH]cc2c1 66095,c1(CC(=O)N(CCCN(C(=O)C(C)(C)C2(O)CCOC2)C)C)ccn(C(F)F)n1 66096,N1(C(c2c(OC)nccc2)=O)CC(O)C(O)C1CNC(C12COC(CF)(C1)C2)=O 66097,N1(C(c2n(CC)nc(C)c2)=O)CCCCC(N(C)C(C2CC(OC)C2)=O)C1 66098,N1(C(C2C(C=C)CC2)=O)CCN(C(C2CCN(C(=O)OCC)CC2)=O)CC(O)C1 66099,Cn1cccc(C(N2CCC(CO)(NC(C3CCC4CC34)=O)C2)=O)c1=O 66100,C#Cc1cccc(CC(=O)NC(CCC=C)C(=O)NC(CCF)C(=O)OC)c1 66101,Cc1ccccc1-n1nc(C(C)C2CC2)nc1-c1cnc(C(C)(C)C)nc1 66102,c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)=CC)CC2)ccc2c(c1)C(=O)NC2=O 66103,C(=O)(N1OC2CCC1C2)C1C2(CCN(C(c3c(C)cc[nH]3)=O)C2)C1 66104,N1(C(CCC=CCCC)=O)C(CNC(=O)C(C)SC)CC2CCCC12 66105,c1(C(=O)NCC(CN(C(C2(CC(C)C)CCC2)=O)C)O)ccc(Cl)nn1 66106,C(=O)(CCC(C)(C)N(C)C)N(C(C)CNC(=O)CC1CC1C(=O)OC(C)(C)C)C 66107,c1(C(N(C(CCNC(c2cc(C(C)C)[nH]n2)=O)C)C)=O)cc2cccn2c(O)n1 66108,C1(CNC(Cc2ccn(CC(C)C)n2)=O)CCN(C(=O)CN(C)C(N)=O)C1(C)C 66109,CCC(C)C(C)(O)CNC(=O)C(C)(CNC(c1ccc(C)n1C)=O)CC 66110,N1(C(CCS(CC)=O)=O)CCCC2CN(C(C3(F)CCC3)=O)CC12 66111,C(=O)(C1=C(C(F)Cl)N(c2cccc(Br)c2)C(=O)NC1c1ccc(F)cn1)OCC 66112,c1(-c2ccccc2)nccc(C(=O)NC2C(NC(CCOC)=O)CCC2)n1 66113,c1(C(=O)NC(C)C(CO)NC(C2(C)CCCCCCC2)=O)ccc(F)c(F)c1F 66114,S(=O)(=O)(c1cccnc1N1CCc2oc(C)nc2C1)NC(CCC)CC 66115,c1(CN(CC(CC)O)C)ncccc1S(=O)(=O)N1CCN(C(C)(C)C)CC1 66116,CC(F)(F)CN=c1[nH]c(=NCC2CCCCS2)[nH]c2c1CSC2 66117,c1(CNC(C(N2CCC(O)CC2)C)=O)cccc(C(N2CC(CN(C)C)C2)=O)n1 66118,c1(CC(N2C(CNC(C3CCCOC3)=O)C=CC2)=O)c[nH]c2ccc(Cl)cc12 66119,N1(C(C)=O)CCCC2CN(C(=O)C=CSCc3ccco3)CC12 66120,c1(C(=O)NCC(N(C(c2cn(C(C)C)nc2)=O)C)C2CC2)cc2cccnc2s1 66121,c1(C(C)C)ccc(C(=O)NCC2CC2NC(c2c(Br)nnn2C)=O)c(O)n1 66122,N1(C(C(CNC(=O)Cn2cccn2)OC)=O)CCCCC1CC(N)=O 66123,C1(C(N2CC(C3(NC(CC(C)CN(C)C)=O)CC3)C2)=O)CCC(S(N)(=O)=O)CC1 66124,N12CCN(C(=NCCOC)N1)CC2(F)F.CC(C)(C)OC(=O)NC1CCC1 66125,c1(C(=O)NCC(C2CC2)NC(C2CC(CC)C2)=O)cn(C)c(=O)n1C 66126,C(=O)(C(CCOCCO)NC(c1cccc(O)c1)=O)N(CCC(=O)NC)C 66127,c1(C(N(CCn2cc(-c3ncoc3C)nn2)CC)=O)cc2nc[nH]c2cc1N 66128,CC1=CCSC1C(=O)NCC1CCC1C(=O)NCc1ccsc1 66129,c1(C(=O)NC2CC(NC(C(CC)OC)=O)CC2O)cc(F)c(OC)c(F)c1 66130,C1(CNC(CC2N(C(C(CC)NC(C)=O)=O)CCC2)=O)OC(=O)CC1(C)C 66131,N1(C(CC(C)(C)NC(=O)C=CC2CCCC2)=O)CCC(C)(CCO)CC1 66132,N1(C(COC(C)C)=O)CCC(CN(C(=O)C(C2CCOC2)OC(C)C)C)CC1 66133,N1(C(C2(CC#C)CCOC2)=O)C2CCC1CC(NC(=O)Cc1csc(S)n1)C2 66134,c1(C(=O)NCC2(F)CCCN(Cc3n(C)ccc3)C2)cc2ccccc2o1 66135,C1(C2CC2)(CNC(=O)Cn2nnc(C(C)(C)C)n2)CCN(C(=O)Cn2cncn2)C1 66136,N1(C(CSCC)=O)C2CCC1CC(CC(C)NC(c1c(C)c[nH]c1C(N)=O)=O)C2 66137,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCC(NC(c2cnc[nH]2)=O)C(F)C1 66138,c1(CNC(c2ccc(C#N)s2)=O)coc2c1CN(C(=O)COc1ccsn1)C2 66139,c1(C(=O)NCC(CC=C)NC(=O)CC2CC2(C)C)cncc(Cl)c1C 66140,c1(N2CCC(COC)C2)nc(N(C)CCN2CCOCC2)nc2c1ncn2C 66141,CC(CCC(=O)NC(c1ccccc1)C)NC(C1CNC(=O)O1)=O 66142,C(c1cccnc1)=CC(=O)NCCN(CCCN(C)C)C(c1c(C)c[nH]n1)=O 66143,c1(OC)cncc(CNC2(c3nnnn3C)COC(CC(C)C)C2)c1 66144,C=C1CC2CCCC(C1)N2C(CC1OCCO1)C(=O)OC 66145,N1(S(C2(CC=C)CC2)(=O)=O)CCc2ccccc2C1CNc1c(C)ccnc1Cl 66146,c1(-c2n(CC)ncc2)ccc(C#N)c(F)c1.C12CN(CCO1)c1cc(ncn1)NC2 66147,C1(NC(C(c2cncnc2)C)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 66148,C12(NC(C(C)OCCCC)=O)CCOC(CNC(=O)C(C)(C)CC3CCC3)(C1)C2 66149,Cc1ccc(OCC(=O)NC2CC(NC(c3cncc(Cl)c3)=O)C2)cc1 66150,C(=O)(CCCCc1ccc(F)cc1)NCC(C)(CO)NC(=O)CCc1ccco1 66151,c1(CC)cc(N(CCCNC(C2CC(c3ccccc3F)C2)=O)C(C)C)ncn1 66152,C=CC1OCCC1C(N1CCC(CN(C)C(c2ocnc2C)=O)C1)=O 66153,CC1(C)CCCCC1NC(C1CCN(C(c2ncncc2Cl)=O)CCO1)=O 66154,C1(C(=O)NC2(COC)CCN(C(=O)Cc3conc3C)C2)CC2C=CCC(C1)C2 66155,c1(C(=O)NC(COCC)C(=O)NCCN=[N+]=[N-])cccc(C)n1 66156,C(=O)(C(C(C)(C)C)n1cc(C2CCCCCC2)nn1)NC(C)CC1CC1 66157,C1(CNC(=O)C=CBr)CC12CCN(C(C1C3CNC(=O)C13)=O)CC2 66158,CC(C)C1=NOC(C)(C(N2CC=CC(NC(=O)C(c3cccc(Cl)c3)O)C2)=O)C1 66159,N1(C(CC(C)SC)=O)CCC(O)C(N(C)C(C2SC3C=CC2CC3)=O)C1 66160,N1(C(C(CC2CC2)OC)=O)CCS(=N)(=O)C(C)C1 66161,C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(c2nncs2)=O)C1 66162,C1(NC(C2OCCC(C)C2)=O)COCCN(C(=O)C=Cc2cnc[nH]2)C1 66163,Cc1cc(CC(=O)NC2CCN(C(C3CC(C)(C)C3)=O)CC2O)cc(F)c1 66164,C1(CNC(COCC(=C)C)=O)CCN(C(=O)Cn2nc(O)ccc2=O)CC1C 66165,C(=O)(C(C(C)(C)C)NC(=O)C(C)OC)NC1CCC(C(=O)OC)C1 66166,c1(C(=O)NC2C=CC(C(=O)OCC)C2)ccc(F)nc1C 66167,C#CCCCC(=O)NCC1CCN(C(=O)C=CCOc2ccccc2)C1 66168,C1(=O)C(C(C)(C)C)n2cc(nn2)CN1.C(=O)(C=C(C)Cl)NCCOCCOC 66169,C1(CCC=C)(C(=O)NCc2sccc2C)CN(C(=O)CCn2ccnn2)C1 66170,CCC(CCC(=O)NC1CCCN(C(C)C)C1)NC(c1ccnc(CO)c1)=O 66171,C1(C(=O)NC2CCCC(NC(CN(C)C)=O)C2)C2CC3CC(C2)CC1C3 66172,C1(N(C=O)Cc2cc(C)ns2)CCc2ccccc2NC1 66173,CC(C)C(C(=O)NCC1CN(C(=O)CN2CCCCC2=O)CC1O)N1CCCCC1 66174,N1(C(c2c(OC)cccc2OC)=O)CCC2(C1)CN(c1ccnc(C)n1)C2 66175,c1(C(=O)NCC(C2CCOC2)NC(CCC(C)(C)OC)=O)ccc2cc[nH]c2n1 66176,c1(C2(C(=O)NCCCNC(=O)C(O)CN3CCCC3)CCC2)c(F)cccc1F 66177,C1(CC)CCC(C(=O)NC2(C(=O)NCC3(C)CC3)CSC2)O1 66178,c1(OC)cc(Cl)ccc1C(N1CCCCC1C(=O)NCCc1ccccc1O)=O 66179,N1(C(c2nc(CC)sc2N)=O)CCCCC(NC(=O)CCOC(C)=O)C1 66180,c1(C(=O)NCC(CNC(=O)CN2CCOC2=O)O)cccc(F)c1O 66181,Cc1sc2ncc(C(=O)NCC(=C3CN(C(=O)C(C)(C)C)C3)F)n2c1C 66182,C=CCC(C)C(=O)N1CCCCC1C1(NC(=O)C(CC2CCCCC2)CC)CC1 66183,c1(CN(C(c2cc(C)oc2C)C)C)ccc(F)c(O)c1F 66184,CCC1=NOC(CC(=O)NC2CN(C(=O)CN(C)Cc3nnc(C)n3C)C2)C1 66185,c1(C(N2CCCC(CCNC(C3CS(=O)C3)=O)C2)=O)cncc(C(F)F)c1 66186,C12(CNC(C3(C)CC(C)C3)=O)CCCCC1N(C(c1cnc[nH]c1=N)=O)CC2 66187,c1(CNC(c2n(CC)nnn2)(C)CCI)ccc(Br)c(F)c1 66188,Cc1cc(C(N2CC(CN(C3CCCC3)C)C3(CC3)C2)=O)nnc1O 66189,N(C1CCSc2ccc(Br)cc21)CC(C)(C)OCC1CC1 66190,N1(C(C(C)Cc2ccccc2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 66191,C1(C2(CO)N=N2)CCC(C)(C)C1.N1(C(C)=O)CC(CNC(N)=O)C1 66192,C1(NC(C=CC)=O)CN(C(c2ccc3cncn3c2)=O)CC(C)(C)C1 66193,c1(OCC)cc(C(=O)NCC(CNC(c2ccc(Br)cc2)=O)OC)cc(Br)c1 66194,N12CCC(O)(C1)C(C)CNC(=O)C1CC(C1)CC2=O.C(=O)(CCSC)NC(C)=O.CO 66195,c1(CC)scnc1C(=O)NC1CCC1NC(=O)CNC(c1ccoc1)=O 66196,c1(CC(=O)OC)ccc(OC(F)(F)C(F)(F)F)c(NC(C)CCN)c1 66197,N1(C(C2(COC)CCCO2)=O)CCC(C)C(CNC(=O)C=C(C)C(F)F)C1 66198,CCCCCCC(C)(C)C(=O)N1CCCC12CCN(C(C1CC3(CC3)CO1)=O)C2 66199,N1(C(C=C)=O)CCC2CCCC12C(=O)NC 66200,N1(C(C(CC)CC)=O)CCC(C2CCN(C(=O)COC)CC2)CC1 66201,N1(C(C2C(C)(CC)C2)=O)CC2CC(NC(=O)C(C)SC(C)C)(C2)C1 66202,Cn1ccc(CCC(=O)NCC(c2ccccc2)NC(=O)CCCC2CCCC2)c1 66203,N1(C(C2(CC)CCOC2)=O)CC2CCC2(CC(N2CC(CN(C)C)C2)=O)C1 66204,C(=O)(C1=CCCOC1)N(C1CCCC(N(C(=O)Cn2cc(Cl)cn2)C)C1)C 66205,C1(CNC(C2(CC=C)CCCCC2)=O)CCC2CN(C(c3cnn[nH]3)=O)CC12 66206,c1(C(=O)N(CC(C)N(C(=O)C(=O)NC2CC2)CC)CC)coc2ccc(O)cc12 66207,c1(C(=O)NCC2C(CNC(c3cc(OC)c(O)nc3)=O)C2)cncc([N+](=O)[O-])c1 66208,CC1CN(C(=O)Cc2cc(Cl)cs2)CC(C)N(C(C2CCCC2(F)F)=O)C1 66209,c1(CN2C(C(=O)NCc3cccc(C)c3O)CC(=C)C2)cn2cc(Cl)ccc2n1 66210,C(=O)(CCCC(N)=O)NC1CN(C(C=CCOC)=O)C(C)C1 66211,C12CSCN1C2=O.C1(C(C)O)CN(C(=O)C(=O)NC2CC2)C1 66212,C1(OC)CN(C(c2n[nH]c(C)c2Cl)=O)CC1NC(c1nc(C(C)(C)C)no1)=O 66213,C1(O)(CNC(CC#N)=O)CCCN(C(c2cccc(C(F)(F)F)n2)=O)C1 66214,C(=O)(C(CCC(N)=O)NC(N)=O)NCC1CN(C(CN(C(C)=O)C)=O)CC1C 66215,N1(C(C(CC)O)=O)CCC(O)(C(C)NC(C2CCC(C(N)=O)CC2)=O)C1 66216,N1(C(Cc2nc(C)sc2)=O)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C(C)C1 66217,c1(C(=O)OC)cnc(N2CCOC(C(C)NC(=O)COC(C)C)C2)nc1 66218,Cc1cnn(CCNC(=O)C(CC2CCC2)NC(=O)C(=O)N(C)C)c1.C(CN)S 66219,c1(C(N2CC(C(=O)NC(c3ncc(C)o3)C)C2)=O)ccccc1C#N 66220,C12(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N3CCCC3)CCCC1CC(=O)C2 66221,CC1CC(CNC(=O)C(=O)N(C)C)CN1C(c1ccccc1N1CCCC1)=O 66222,C#CCC(CC(=O)OC)NC(=O)C(C(C)CC)N(C(=O)C(C)c1cc[nH]n1)C 66223,c1(-c2n(CC=C)c(N(CCCO)CCOC)nn2)c(OC)ccc2ccccc12 66224,c1(C(=O)NC2CC(NC(c3c(C)nc(C)nc3C)=O)C2)ccc2oc(O)nc2n1 66225,c12cn(C)c(n1)C(=O)NCC1CCN1C2=O.c1(OCC)cccs1.C(F)F 66226,c1(C(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)cnc2cccnn12 66227,CC1CC(NC(=O)C(C)OCC2CC2)CN(C(=O)C=Cc2ccc(F)cc2)C1 66228,C(=O)(C(C)(CO)NC(c1cc(Cl)cs1)=O)N(CC(C)OC)C.C(C(F)(F)F)S 66229,CC(C(=O)NCC1(F)CC(NC(=O)COCP(C)(C)=O)C1)C(=O)OC 66230,CCC(CC(=O)N1CC(F)(CNC(C2(c3cc[nH]n3)CCC2)=O)C1)c1ccccc1 66231,c1(NC(C2C(C)C2c2cccs2)=O)ccccc1C(=O)N(C)C 66232,c1(C(C(=O)N(CC(C)CNC(C2CCOC2)=O)C)O)cnn(C)c1 66233,C1(N(C)C)CN(C(c2cccnc2CO)=O)CC1(C)C.C12CC(C1)NC(=O)CO2 66234,CCC(CC(=O)NC1CCCN(C(c2ccc3occc3n2)=O)C1)C(F)F 66235,Cc1ccc(C(=O)NCC2CCC(NC(=O)C=Cc3cccnc3)C2)cn1 66236,c1(C(N2CCCC(N(C(=O)C(O)P(C)(C)=O)CC)C2)=O)ccc2oc(=N)[nH]c2c1 66237,c1(C(N(C2CCC(NC(c3ccsc3)=O)C2)C)=O)cccc(-n2cccc2)c1 66238,C(CCC(=O)N(CC(C)NC(=O)C(C)CN1CCCCC1)CCO)N(C(C)=O)C 66239,C1(N(C(C(C)OCCOC)=O)C)CCCC2CN(C(=O)CCc3cccs3)CC12 66240,C1(CC)C(NC(c2c[nH]c(=N)o2)=O)CCN1C(=O)CC1CC2(CC2)CO1 66241,N1(C(CC2OCC(C)(C)C2)=O)CCCCCC(NC(c2cc3cc(Cl)sc3[nH]2)=O)C1 66242,C1(N(C(c2ccn(C)c2)=O)CC)CCCN(C(=O)C=Cc2ccc(Cl)cc2)CC1 66243,C(CC(CC)C(=O)NC12CCC1CN(C(c1ccc(OC)nc1Cl)=O)C2)=CC 66244,N1(C(C(=O)NCC)=O)CCN(C(C2CCC2(C)C(F)F)=O)C(c2cnn(C)c2)C1 66245,Cc1cccc(C(N2CCCC2C2CCCN(C(=O)C(=O)N(C)C)C2)=O)n1 66246,N1(C(C2CCN(c3c(C)cncn3)CC2)=O)CCC(O)(CO)CC1 66247,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2(C#N)CC2)CCC12CCOCC2 66248,C12(C(N3C(CNC(CCN(C)CCO)=O)CC3)=O)CSC(C1)C2 66249,c1(C(=O)NC(CCNC(COCCC#C)=O)C)cc(Cl)cc2ccccc12 66250,C(C)(C(=O)NC1(COCC)CSC1)ONC(=O)COC(C1CCOC1)C 66251,Cc1nc[nH]c1CC(O)C(=O)N(CCNC(=O)CNS(N)(=O)=O)CC1CC1 66252,C1(NC(c2ccc(C)c(O)c2)=O)CC2CCC(C1)N2C(c1cnoc1)=O 66253,c1(OC)cc(C)c(C(N2CCCC2C(C)NC(=O)C#CC2(C)CC2)=O)nc1Br 66254,N1(C(C2CCCN(CCNC(=O)OC)C2)=O)CC(=O)C(N)C12CCC2 66255,c1(COC)ccoc1C(=O)NCC(CNC(=O)Cn1cc(Cl)cn1)CO 66256,C1(C)(CNC(C(C2CCCCC2)C)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1 66257,C1(CC(=O)NC2(CC=C)CN(C(=O)COCC)C2)CC(c2ccccc2)=NO1 66258,C1(CC(=O)NCC2CCCC(C)C2)CC(C)(C)CN1C(=O)CC1C=CCC1 66259,N1(C(CN2C(=O)NCC2)=O)CCN2C(=O)OCCC2C1 66260,c1(NCCC(C)C)ncccc1S(=O)(=O)NCC(c1ccc(Cl)cc1)CO 66261,C(=O)(CC(C(F)(F)F)c1ccon1)N(CCCNC(C1=NOC(C)C1)=O)C 66262,c1(CC)[nH]nc(C(N2CC(OC)C(NC(c3ccc(CC)[nH]3)=O)C2)=O)c1[N+](=O)[O-] 66263,c1(CC(=O)NC2C(C)CN(C(c3cc(C(C)(C)C)on3)=O)C2)ccc2c(c1)CC2 66264,CC1CCOC(C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C)C1 66265,C=CCC(C(=O)NCc1cnc(OCC)nc1)NC(c1ccnc(C)n1)=O 66266,C1(NC(c2cnc(C)nc2)=O)CC2(CCN(Cc3nccnc3Cl)CC2)C1 66267,c1(C2(N)CCOCC2)c[nH]c2cccc(C(N3CCC4(CCCO4)CC3)=O)c12 66268,c1(CC)nccnc1C(=O)NC1C=CCN(C(=O)CC2(C)CCCCC2)C1 66269,C(=O)(C(C)CCCC(C)C)N(CC(CC)NC(=O)CC1CC(=O)NC(=O)C1)C 66270,CC(C)CS(=O)(=O)N1CCCCC1C(=O)NC1CCC(N)CC1 66271,N1(C(c2cccc(C(=O)NC)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66272,OCCCCN=c1[nH]c(=NCC2C3COCC23)c2ccccc2[nH]1 66273,C12(C(N(CCCCNC(=O)CCCN3CCCC3)C)=O)CC(C)(CCO1)C2 66274,C1(NC(C(CCC)O)=O)CCCCCN(C(=O)C(=Cc2ccccc2)OC)C1 66275,Cc1ccc(C)c(C(=O)NCC2CCN(C(=O)C(C)Cc3ccccc3)C2)c1N 66276,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66277,C1(C(N(CCCC)C2CC2)=O)CCC(C)(C)N(C(=O)CCOC(C)=O)C1 66278,Cc1ccn2cc(C(N3CCCC34CN(C(=O)Cc3nc(C)cs3)C4)=O)nc2c1 66279,c1(CN(C2CC23CN(c2ncc(F)c(C)n2)C3)CC)cc(C(F)(F)F)cc(F)c1 66280,S(=O)(=O)(c1cc(C)cnc1N1CCC(Oc2ccccc2)CC1)N(CCNC)C 66281,C#Cc1cnn(C)c1C(N1CCCC(CC(=O)NCCC(O)CCC)CC1)=O 66282,C1(C)(CC)CC(NC(=O)C=CCN(C)C(c2[nH]ccc2C)=O)CCO1 66283,c1(C(N(C2(C(=O)NC3(COC)CC3)CC2)C)=O)sccc1C1CC1 66284,N1(S(=O)(=O)c2ccccc2)CCN(S(=O)(=O)Cc2cccnc2)CC(O)C1.CN 66285,C1(CC(=O)OC)CS(=O)CCN1Cc1cccc(Br)c1O 66286,C1(C(=O)Nc2ccc(SC)nc2)CCc2nc(-c3ccc4cc[nH]c4c3)sc2C1 66287,C1(N(C)C)CC(CC(=O)NCC(C)(C2CC2)NC(=O)Cc2cnc[nH]2)C1 66288,N1(C(C=C)=O)CCCC(C(=O)NC(c2cccc(OCC)c2)CO)C1 66289,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCc2cnc[nH]2)CC12CCC2 66290,C1(NC(=O)Cc2ccnc(Cl)c2)CN(Cc2cccnc2O)CC1(F)F 66291,c1(OCC)ccc(CO)cc1-c1ccc(NCC2(C(=O)O)CCC2)o1 66292,CCCCC(CNC(C1CC(=O)N(C(C)C)C1)=O)NC(=O)C(c1ccccc1)=O 66293,c1(C(C)OC(C2(C)CCCC2=O)=O)ccc2ncsc2c1 66294,N1(C(CC2C(CC)C2)=O)CCC(F)(CNC(=O)C(Cc2ccc(F)cc2)NC)C1 66295,Cc1cc(Cl)ccc1CNC(C1COCCN1C(c1cn(C)cc1C)=O)=O 66296,C1(C2CN(C(C(=O)NC(c3nnc(O)n3C)C)=O)C2)CN(C)CCO1 66297,Cc1c(C(N2CCC(N(C(=O)C=CCCC=C(C)C)C)CC2)=O)cccc1CO 66298,Cn1cc(C(F)(F)F)nc1C(=O)NCC1CCN(C2CC2)CC1 66299,N1(C(CN2CCC(C)(C)C2)=O)CC2(NC(=O)COCC3CCC3)CCC1CC2 66300,C(=O)(C(=O)N=S(C)(C)=O)NCC1CCC(NC(C(C)Cc2ccccc2)=O)C1 66301,CC1(C)CCCCC(OC(c2cnoc2-c2cccs2)=O)C1 66302,C1(C(N2CCCC2CC2CC2)=O)CCCC2CC12 66303,Cc1cc(C(N2CCN(C(C3(C(N)=O)CC3)=O)CC2C)=O)c(C)n1-c1nccs1 66304,c1(C(=O)OC)cccc(C2(C(=O)N(CC(C)NC(=O)C(CCO)SC)C)CC2)c1 66305,N1(C(C2(C)CCC(C)C2)=O)CC(C(=O)OCC(C)(C)C)C2(CCC2)C1 66306,C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(C(CC=CC)C)=O)CC2O)CCOCC1 66307,Cc1cnc(O)c(CNC2CCC(C(N3CC(C)(C(=O)OC)C3)=O)C2)c1 66308,c1(NC2CCCN(C(C3CC4(C3)CC4(F)F)=O)C2)ncc([N+](=O)[O-])cc1Br 66309,C1(NC(C2(COC(C)C)CC2)=O)C=CCN(C(=O)C(c2cccc(Cl)c2)C)C1 66310,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66311,c1(N(c2ccc(C)cn2)CCCC)ccc(COC)cc1 66312,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66313,CCC(CC)CC(=O)N1CCN(C(c2cn3ccsc3n2)=O)CC1CCOC 66314,c1(C(N2CCN(C)C(CNC(=O)COCC3CCC3)C2)=O)cc2ccncc2s1 66315,N1(C(c2ccc(SC)o2)=O)CC(OC)C(NC(=O)CNC(=O)CC(C)(C)C)C1 66316,C1(C2CCN(C(=O)C=C3SCC(=O)N3C)C2)(NC(C(C)S(N)(=O)=O)=O)CC1 66317,N1(c2cc(N(C)Cc3ccsc3)nc(C)n2)CCCc2ccc(C(N)=O)cc21 66318,C1(NC(CC2C(C)C2)=O)CCC(NC(c2ccnc(OCCO)c2)=O)CC1 66319,c1(CNC(N(C(c2ccncc2)C)C)=O)nc2c(o1)CCSC2 66320,c1(SCC)ccc(Cl)cc1C(N1CC2C(CNC(C3(C(=O)OC)CC3)=O)C2C1)=O 66321,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66322,N1(C(=O)Nc2c(C)ccc(OCCC(N)=O)c2)CCCNC(=O)C(F)(F)C1 66323,c1(NC(N(C(CC(CC)C)C)CC)=O)cnc2ncnc(O)c2c1 66324,c1(C(N2CCC(CNC(c3nn(C)c(Cl)c3)=O)C2(C)C)=O)ccc2ncsc2c1 66325,Cc1cc(N)cnc1C(=O)NCCNC(=O)CCC1CC(C)(C)CO1 66326,CC1SCCN(C(c2cccc(Nc3ccccc3)n2)=O)C1c1ccccc1 66327,C=CCC(C)(C)C(=O)NCc1ccc(CNC(C2CCC3CC3CC2)=O)cc1 66328,c1(CN2CCC(CC(=O)OC)C2)c[nH]nc1NC(C(C)=CC=C)=O 66329,C1(NC(C2(CC=C)CC2)=O)CN(C(=O)C(CC)N(CC)CC)CC(C)(C)C1 66330,c1(OC(C)C)cc(-c2cccc(NC(c3ccsc3CO)=O)n2)ccn1 66331,CCCC(C(=O)OC)C(=O)N(C(C)CN(C)C(c1sc(C)nc1C(C)(C)C)=O)C 66332,N1(C(C2CCC(C(C)C)N2C(c2cc(CO)[nH]n2)=O)=O)CCC(N(C)OC)CC1 66333,N1(C(C(COCC)(C)C)=O)CC(C(=O)NC2CC23CC(OC)C3)CC(C)(C)C1 66334,C1(O)(C(C)C)CCCN(C(=O)CC2CCCCN2C(=O)CC2(O)CCCOC2)C1 66335,CC1(C)C(NC(=O)C=CCF)CC1C(=O)NCC(Cl)Cl 66336,Cc1cc(CN=C(NCC(c2ccoc2)N2CCCC2)NCC2CC2)c(C)s1 66337,C(CCC(C)C(=O)N(C1CC(NC(=O)C(F)(F)OC(C)=O)C1)C)OC 66338,c1(OCCNC(C)=O)cccc(Br)c1C(=O)NC1CC1C 66339,C1(NC(C(=O)NCCNC(C)=O)=O)CN(C(C2CC2[N+](=O)[O-])=O)CC2(CCC2)O1 66340,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(O)c2)C)(C)C)C(=O)CNC1=O 66341,C1(NC(C2CC3(CCC3)CO2)=O)CCN(C(C2CCCC23CC3)=O)CC1F 66342,c1(C(=O)NC(CC(=O)NC(c2cn(CC)nc2)C)C(F)F)c[nH]c2ccncc12 66343,C1(NC(c2ccc(C=C)cc2)=O)CCN(C(c2cnn(C)c2C)=O)C12CCC2 66344,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66345,N1(C(C(C)(C)c2ncco2)=O)CCCC(CN)CC1.C1(S)CCCO1 66346,c1(C(N2CC(OCC)(CNC(C3CN(C4CCOC4)C3)=O)C2)=O)ccc(C)cc1 66347,c1(-n2cc(C(N(C3CCCC3O)C(C)C)=O)nn2)ccc(I)c(Cl)c1 66348,C(C(C)(C)C(=O)NCCC1CCN(C(C2CN(C(C)C)CCO2)=O)C1)OC 66349,N1(C(C(C=CC)O)=O)CCN(C(C2(C(F)F)CCOC2)=O)CC1CC(=O)NC 66350,c1(N2CC3C(C(=O)OC)(C3)C2)nc2ccccc2o1 66351,CCC(CC(=O)NCCc1ccc(CNC(C2CSCCS2)=O)cc1)C(C)(C)C 66352,c1(C(=O)NC2(CO)CN(C(c3ncn(CC)c3)=O)C2)ccc2cccnc2n1 66353,c1(CCSC(F)(F)F)ccc(OC(C)(C)COC)c(C)c1.n12nnnc1C2CC 66354,CON=Cc1ccc(C(N2CCC3CN(C(=O)Cc4cc[nH]c4)C3C2)=O)cc1 66355,C(=O)(N=c1[nH]c(Cl)c(I)nc1Br)C1CCCN(C(c2cc(O)c(O)c(O)c2)=O)C1 66356,N#Cc1ccc(CCC(=O)N)cc1.C1(C(F)(F)F)CCCNC1 66357,c12ccccc1C2NC(=O)CN(C)C.C(=O)(C(C)(C)CF)NCC(=O)OC 66358,Cc1cc(C)c(C(N2CC(CNC(=O)C(C)S(C)(=O)=O)C2)=O)c(=O)o1 66359,c1(CC(=O)NCC2CN(C(c3c(OC)c[nH]n3)=O)C2)ccc(C)c(Cl)c1 66360,c1(C(=O)NC(CNC(c2n(CC)ncc2)=O)C2CC2)cnc2ccc(Br)cn12 66361,CC(C)CC(C(=O)OC)N(C)C.C1(=O)C(CO)N1.C1(=O)C(C)N1.C(N)(=O)N 66362,N1(C(C(C)Cn2cccn2)=O)CCCOC(CNC(c2cnn[nH]2)=O)C1 66363,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(C2CCCC(=O)CC2)=O)CC1 66364,C12(CNC(c3ncc[nH]c3=O)=O)CCC(C1)N(C(C1(O)CC1)=O)C2 66365,C(C(C(=O)N1CC(C)(CC(=O)NCCC(C)CO)C1)OC)OC 66366,C(=O)(C1=CCCN(C(c2ccc(F)c(F)c2F)=O)C1)NCC(CO)OC 66367,c1(N2CC(N(C(=O)Cn3ncnn3)CC3CC3)C2)nccc(-c2ccsc2)n1 66368,Cc1nc(C(C)NC(C2CC2C(=O)OC(C)(C)C)=O)oc1C 66369,CC1(C)C(CNC(=O)C(CC2CCC2)NC(C2CNC(=O)O2)=O)C1(C)C 66370,N1(C(C2=CC(O)C(NC(c3nncc(OC)c3)=O)C2)=O)CCCC(C2(C)CC2)C1 66371,C1(O)(C(N2CCCC(CNC(=O)CCc3ccsc3)C2)=O)CN2CCC1CC2 66372,CCC(C)CC(=O)C(=O)NCc1c(C(=O)NOC(c2ccccc2)C)cccc1F 66373,Cc1nc(NCC2CCC(C(=O)Nc3ncc(C(F)F)s3)C2)c(C)c(O)n1 66374,c1(COC)cc(CSc2ccccc2OCC2CCOC2)ccc1F 66375,N1(C(=O)C(O)c2ccsc2)CCC(F)(F)C(CNC(c2cn(C(F)F)cn2)=O)C1 66376,CCC(CS(=O)(=O)c1ccccc1)NC(=O)Nc1nocc1Cl 66377,C1(NC(=O)COCC(F)F)CN(C(C2(F)C3CCCCC23)=O)CC1C1CC1 66378,n1(CC)nc(C(=O)NC2(C(=O)NCCCn3nccn3)CCCC2C)cc1C 66379,N1(C(c2c(C)ncnc2C)=O)CC2(CC(NC(=O)C#CC3CC3)c3nccn32)C1 66380,N(C(=NCCF)NC1CCOc2c(F)ccc(F)c21)C(C1CCC(CN(C)C)O1)=O 66381,CC1CCCCN1C(=O)CCNC(=O)NCCc1cn(C)nn1 66382,c1(OCC)cccc(C(=O)N(C)CC2CCN(C(c3cnn(C)c3OC)=O)C2)c1 66383,c1(C(=O)NC2CCCN(C(C(n3cc(Cl)cn3)C)=O)C2)c(Cl)cccc1[N+](=O)[O-] 66384,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C)=O)C1C2 66385,CC1CCN(C(=O)CCCNC(c2cc(C3CC3)on2)=O)C1 66386,c1(CSC)cc(Br)ccc1NC(=O)N(C1CC2CCC1C2)Cc1ccccc1F 66387,C1(CNC(c2cc(C3CC3)cc(F)c2)=O)CC2C(O)CC2O1 66388,CC12CCCC1N(C(=O)CC1(C(F)(F)F)CC1)CCN(C(=O)Cc1cnc[nH]1)C2 66389,CC1CCN(C(c2ccc(CF)cc2)=O)CC1NC(=O)COC1CCCCC1 66390,C1(C)(C(=O)NCC2C(C(=O)NCC(C3CCCCC3)C)CC2)CC(F)C1 66391,C#Cc1cccc(C(=O)NC2(OC)CC(C(N3CC(N4CCC4)C3)=O)C2)c1 66392,C1(NC(Cc2cc(CC)no2)=O)COC2(CCN(C(C3(C)COCCO3)=O)C2)C1 66393,c1(CC(C)C(=O)NCCN(C)C(C2CC3CC3C2)=O)ccc(C(C)(C)C)cc1 66394,Cc1c(C(=O)NC23CC(NC(c4cn(C)nn4)=O)(C2)C3)oc2ccc(Br)cc12 66395,N1(C(c2c(C)[nH]cc2)=O)CCCC(NC(c2n[nH]cc2-c2ccccc2)=O)C1C 66396,c1(C(=O)NC(CNC(=O)Cc2ccc(O)nc2)C2CC2)cc2cccn2c(O)n1 66397,N1(C(C)C(=O)NC(=O)Nc2ncc(Cl)cc2Cl)CC(CO)OC2COCC12 66398,c1(C(=O)NCC2(C)C(C)CN(C(=O)C(F)=CC3CC3)C2)nc2ccccc2cc1Cl 66399,C1(C(CCNC(CCC)=O)(C)O)CCN(C(=O)C#CC2CC2)CC1 66400,c1(C2(C)CC2N(C(c2sc(Br)nc2Cl)C(=O)NC2CCOC2)C)cccc(F)c1 66401,c1(C(C(=O)NC2CC(F)(CNC(C(C)O)=O)C2)(C)C)ccccc1F 66402,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C(F)C(C)(C)O)CC1 66403,CC(CC(F)F)C(=O)NC1CC2(C1)CN(C(=O)C(C)Cc1ccnn1C)C2 66404,Cc1cc(C(N2CCC(Cn3cc(C(C)O)nn3)C2)=O)c2c(c1)CCC2 66405,C1(NC(C2C(C)(CC)C2)=O)(COC)CCN(C(=O)C=Cc2ccc(C)nc2)CC1 66406,C(=O)(CCCC(C)NC(c1ccncc1Cl)=O)Nc1cc(C)oc1C 66407,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66408,N1(C(c2cccc(CN=[N+]=[N-])c2)C(=O)NCCN2CCOCC2)CC2(CCOC2)C1 66409,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66410,CC(O)CC(C)(C)CN(C)CC1(CO)CCN(C(=O)OC(C)(C)C)CC1 66411,c1(C(N2CC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)cc2nn[nH]c2cc1F 66412,N1(C(C=CC)=O)CCC(CN2CCN(C(c3ccc(OC)nn3)=O)CC2)CC1 66413,C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66414,Cc1cc(C(N2CCCC2CN(C(c2cc(Cl)ccc2O)=O)C2CC2)=O)cc(O)n1 66415,C1(OC)CC(C(N(C2CCN(C(C3(CCCC)CCC3)=O)CC2)C)=O)C12CCC2 66416,C1(OC)CN(C(=O)C(c2cccs2)SC)CCC1NC(c1cc[nH]c1C)=O 66417,C1(OC)(CNC(c2cc(-c3ccco3)nn2C)=O)CCN(C(=O)C=C(C)Cl)C1 66418,N1(C(CC(CC(=O)NC)C)=O)CC2CC3CC2C1C3NC(=O)CCCSC 66419,C(=O)(C1=CN=C2N=CNN2C1)N(C1CCCN(C(C(C)(C)OC(C)C)=O)C1)C 66420,N1(C(C=CCC(C)(C)NC(C=CCOC)=O)=O)CCC2CN(C)CC2C1 66421,c1(OC)cccc(C)c1C(=O)NCCCC1CCCCN1C(=O)C(O)C(C)(C)C 66422,Cc1cncc2cc(C(N3CC4CCC(C3)N4C(=O)C(C)C3CC3)=O)sc12 66423,CC1(C)C(NC(=O)COCC(=O)OC(C)(C)C)CC1CNC(c1cc(F)cs1)=O 66424,n1(CC(=O)NC23CC(CCF)(C2)C3)cnc([N+](=O)[O-])c1 66425,N1(C(C(C)(C2CCC2)NC(C(CC2CCC2)OC)=O)=O)CCCCC(N(C)C)C1 66426,c1(C(=O)NC2CCN(C(c3n(CC)ccc3)=O)C2)ccc2c(c1)N(C)C(=O)CO2 66427,C(=O)(CC(C(F)(F)F)OC)NC(CCNC(C1CN(CC)C(=O)CC1)=O)(C)C 66428,Cc1cc(N(CCN)C(c2ccc(O)c(F)c2Cl)=O)c(I)cc1Cl 66429,C(=O)(CC(O)CC1CC1)NC(CNC(C1C(=C)C1)=O)(C)Cn1cccn1 66430,C12(C(=O)NCc3ccc(CN(C)C(C45CC(O)C4C5)=O)cc3)CCCC1CCC2 66431,Cc1noc(C)c1C(N1CSCC1C(=O)NCCC1(C)CC1)=O 66432,CC1(C)CCC(NC(C2CC(NC(N)=O)C2)=O)C(CNC(c2ccccn2)=O)C1 66433,c1(Cn2cc(C(C)(C)F)nn2)cc([N+](=O)[O-])ccc1Br 66434,CC(C)(C)C(=O)C(=O)N1CCC(C)(NC(=O)C(N2CCCC2)C2CC2)C1 66435,C1(C(=O)NCCC(C)CCNC(=O)Cc2cc[nH]n2)CN2CCN1CC2 66436,c1(NCC(CO)NC(=O)NCC(N2CCCC2)=O)ccc2cccnc2c1Cl 66437,Cc1nc2ccccc2n1CC(=O)NC1C=CCN(C(=O)CC2OCCC2(C)C)C1 66438,C1(C(=O)NC(CO)C(=O)NC2C3COCC23)CC2(CCC2)CO1 66439,N1(C(C2(CC)CCC2)=O)CC2(C1)CN(C(=O)C(c1ccccc1F)(C)OC)C2 66440,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)C3)=O)CC1C2 66441,CC1(C)CC(C(=O)NC2(CC3CCC3)CC2)=NO1.C12(CC1)C(=O)N2 66442,N1(C(CCCNC(=O)OC)=O)CCCC(CN(C)C(C2CCCCN2C)=O)C1 66443,C(=O)(CC(C(C)(C)C)NC(c1cnn(C)c1SC)=O)NCC(CC)(F)F 66444,C1(C(=O)NCC(C)N(C(C(C)n2ccnc2)=O)C)C(c2ccncc2)C1(C)C 66445,c1(NC(C2CN(C(=O)CCc3ccnc(Cl)c3)C2)=O)ccc2scnc2c1 66446,c1(NC(C2C(NC(c3cc(Cl)cc(Cl)n3)=O)CCC2)=O)ncc(F)cc1Br 66447,C(=O)(C(Cc1cccc(Br)c1)CC(C)C)NC.C12CCN(CC1F)C2=O 66448,C1(NC(c2c(CC)scc2)=O)CCN(C(c2ccccn2)=O)C(C)C1 66449,c1(OC)nccc(=NC2CC23CCC(NC(c2scc(C)c2Cl)=O)CC3)[nH]1 66450,c1(C(N2CCCCC(CNC(C3=NNC(=O)C3)=O)C2)=O)ccc(F)c2ccsc12 66451,[SH](=O)(=O)c1ccc(C2OCCO2)cc1.CC(C)(C)OC(=O)NC1CNC1=O.C1CC1 66452,C12(C(N(C3CCCN(C(C(CC)COC)=O)CC3)C)=O)CCCC(=O)N1CCC2 66453,C(=O)(C(C(C)C)NC(C1CCCCC1NC(c1cccc(CO)c1)=O)=O)OC 66454,CCCCC(CNC(=O)C(C(C)C)N(C)C)NC(c1cnn(C)c1Cl)=O 66455,c1(CNC(C2CC2NC(C23CCN(CC2)C3)=O)=O)cc(F)ccc1-n1cccn1 66456,N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C1C2 66457,C(=O)(CC(F)(F)C(F)F)NCC(CNC(=O)C(Cc1cccc(Cl)c1)C1CC1)O 66458,C=C(C)C(C)(C)C(=O)Nc1c[nH]nc1-c1cccnc1.C12CC(C1)CC(=O)N2 66459,CC1(c2cn(-c3nccs3)nn2)CC2CCC(C1)N2C(c1ccc(Cl)cc1Br)=O 66460,c1(N2C(c3cc(F)c(-n4cccn4)c(F)c3)CCCC2)ccnc2c(Cl)cnn12 66461,CC(C)(CNC(=O)COC1CCC1)CC(=O)NCc1cc[nH]n1 66462,C1(CC(=O)N(CC(C)N(C(C)=O)C)C)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66463,c1(-c2c(C)noc2)nc(CCn2cc(Cl)cn2)nn1CC(C)(C)C 66464,C12(NC(C(C)OCC#C)=O)CCC(C1)N(C(=O)CCCC(=O)NC)C2 66465,c1(C(N2C(C(C)(C)C)CCC2)C(=O)Nc2cccc(Br)c2)ccc2c(c1)OCO2 66466,C12CCC(CC1)O2.C(C(=O)NC(C1(CC2CCC2)CC1)=O)SCCOC 66467,CC1CC(C(=O)NCc2cn(CCNC(=O)CSc3ccc(F)cc3)nn2)=NO1 66468,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66469,c1(OC)ccc(CN2CCN(CC(=O)Nc3noc(C)n3)C(C)C2)cc1[N+](=O)[O-] 66470,C1(NC(C2(COC)CCOC2)=O)CCN(C(c2ccc(O)nc2)=O)C1C.C1CC1 66471,N1(C(c2ccc(CCC)cc2)=O)CC(NC(c2nc(C)no2)=O)C(C)(C)C1 66472,c1(C(N2CCN(C(c3c(C)nco3)=O)C3C2CC3)=O)cc2ccsc2c(O)n1 66473,c1(NC(CC=C)=O)cc(-n2cc(C3C(C)CCN3C(C)=O)nn2)ccc1Cl 66474,c1(C(=O)NC2C(CC)N(C(c3ccc(C4CC4)s3)=O)CC2)ccc(N=[N+]=[N-])cc1 66475,c1(C(C(=O)NCCC2CC2)N(CC(=O)OCC)CC(C)C)ccc(Br)c(F)c1 66476,Cn1ncc(Cl)c1C(=O)NC1C2CN(C(=O)CCN3CCOCC3=O)CC12 66477,C(C)(CC(C)N=c1[nH]c2ncc(Cl)cc2o1)NC(c1c[nH]c2cccc(C)c21)=O 66478,N1(C(CSC)=O)CCCC(CCC(=O)NCC(N2CCC(C)CC2)=O)C1 66479,N1(C(C(CC)C(=O)OC)=O)CC2CCCCN2CC1CNC(=O)C(=O)NC(C)C 66480,C(C(O)CC(=O)NCC1CNC(=O)C1)NC(Cc1c(C)ocn1)=O 66481,c1(C(N2CCC(OCCNC(C(C)SC)=O)C2)=O)ccc(-c2ccco2)nc1C 66482,CC(C)C(C(=O)N(CCCCNC(=O)C=CCN(C)C)C)ONC(=O)OC(C)(C)C 66483,C(CC(C)C(=O)NCC1CCCN1C(=O)C(C)OC(C)(C)C)=CC 66484,N1(C(C2C=CCS2)=O)CCC2CN(C(=O)CCN3CCC3)C2C1 66485,C1(CNC(c2nnc(C)s2)=O)CCCC2CN(C(=O)C(C)OCC(C)C)CC12 66486,Cn1cc(C(CNC(=O)CSn2cc(Cl)cn2)NC(c2c[nH]nc2Br)=O)cn1 66487,c1(OC)ccccc1-c1noc(CNC2CCCC(c3ccc(Cl)cc3)C2)n1 66488,C1(C)(C(N(CC(CC)CC)C2CC2)=O)CCCN(C(c2cnc(C)n2C)=O)C1 66489,c1(OC)cc(C(N2CCC(NC(c3ccc(N)cc3Cl)=O)C2)=O)cc([N+](=O)[O-])c1 66490,Cc1cccc(O)c1C(N1CCCC(CN(S(=O)(=O)CCCl)C)C1)=O 66491,CC1CN(C(c2ccnc3c2ccn3C)=O)CC(C)N(C(=O)C(Cl)=CCl)C1 66492,C1(C(=O)NC2CCOCC2)CCOCC1C(=O)NCC1CC2(CSC2)C1 66493,c1(CC(=O)NCCN(C)C(C2C3COCC23)=O)cccc([N+](=O)[O-])c1C 66494,CC1CN(C(C2CC=CCC2NC(C23CCCN2CCC3)=O)=O)CCCO1 66495,N1(C(C(C)(N(C(C(C)N2CCC2)=O)C)C2CC2)=O)CCCC(F)(CO)C1 66496,C(=O)(C1=CCCCC1C)N1CC(N(C(c2c(C)nc(-c3ccco3)o2)=O)C)C1 66497,c1(C(C2CCOC2)NC(=O)C(=O)NCCO)ccccc1NS(C)(=O)=O 66498,N1(C(c2c(C)nc(CCC)s2)=O)CC2(CCCC2NC(C2CCCN2CC)=O)C1 66499,C1(N(C(c2cnc(Cl)c(C)c2)C(=O)NCC)Cc2ccco2)CCCCCCC1 66500,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)NC(C(=O)OCC)C1CC1 66501,C1(NC(C2CCN(C(C)=O)CC2)=O)CC2C1CCN2C(=O)Nc1ccccn1 66502,Cc1nc(SCc2ccc(F)cc2)n(CC2CCOCC2)c1C 66503,CCCC(C=O)C(=O)N(C)CCN(C)CCN(CC)CC.N1(C(C)=O)C2CCC1COC2 66504,Cc1cc(NCC(CN2CCN(c3nc(I)cnc3I)CC2)O)ccc1[N+](=O)[O-] 66505,c1(C(=O)NCC(C2CC2)NC(c2n(CCOC)ncc2)=O)ncc(CC)nc1Cl 66506,CC(C)CC(O)CC(=O)NCc1ccc(C(=O)NCCN(C2CCCC2)C)o1 66507,C12(OC)CCC1CN(C=O)C2.C1(N)CCN(C(=O)CCCC2CCC2)C1(C)C 66508,Cc1c(C(N2CCSCC2CCNC(C2CN(C)C2)=O)=O)sc2nccn12 66509,N1(C(C2N(C(CCC(C)SC)=O)CC(=O)C2)=O)CCc2nc(C)[nH]c2C1 66510,c1(C(N(C2CCN(C(c3cnco3)=O)C2)CCC)=O)nocc1C 66511,c1(C(N2CC(c3ccccc3)(C(C)=O)C2)C(=O)NCCCF)cc(Br)cc(C)n1 66512,O=C(CC1COc2ccccc21)NCC1(F)CN(C(=O)C=Cc2ccco2)C1 66513,N1(C(C(CC#C)C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66514,N1(C(CC2CCC(=O)NC2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66515,Cc1cccn(CC(=O)NCCCCc2ccccc2Br)c1=O 66516,CN=c1ccc(C(N2CC(CC(F)C(=O)NCC(=O)N3CCCO3)C2)=O)c[nH]1 66517,O=C(C(F)C1=CCCCC1)NC1CCN(C(c2ccoc2)=O)C1C(C)(C)C 66518,c12nnc(-c3cccs3)n1CCN2CCC#C.c1(S)ccccc1 66519,CCCCCC(O)C(=O)NC1CC(CO)N(C(C2CC2c2ccc(Cl)cc2)=O)C1 66520,c1(C(C)C)ccc(C(=O)NCC2CC(CNC(=O)C(CC)N(C)C)C2)cc1Cl 66521,C1(CC(=O)NCC2CCN(C(C3CC(C)C3)=O)C2)CCC(=O)N1 66522,C1(C(=O)Nc2c(-c3n(C)ncc3)n[nH]c2)CCN(C(C2COC(=O)N2)=O)C1(C)C 66523,S(=O)(=O)(c1cccnc1)N1CC(C(=O)NC2CCCC(OCC)C2)C(O)CC1 66524,N1(CC(=O)NCCCC(C)(C)C)CCC2(O)CCOCC2C1 66525,c1(CC)nc(-c2nc[nH]n2)sc1C(=O)NC1CN(C(=O)C(F)(F)CC2CC2)CC1O 66526,CC(C)(CC=Cc1cccs1)NC(C1CC(Br)C1)=O 66527,c1(-n2c(C3(NCC(C)C)CCCOCC3)nnn2)ccc2c(c1)OCCO2 66528,N1(C(CCCCOCC)=O)C2CCC1CN(C(c1cc(C(F)F)n(C)n1)=O)CC2 66529,N1(C(c2ccc(C(C)(C)C)s2)=O)CC2CCN(C(c3cccc(F)c3)=O)CC2C1 66530,N1(C(c2nnc(C)c(C)c2-c2ccnn2C)=O)CCc2cc(Br)c(Cl)cc2C1 66531,C1(CNC(c2nncc(OC)c2)=O)CC2(CO1)CN(C(=O)CCc1cnco1)C2 66532,N1(C(C)=O)CCCN(C(=O)NCc2cnc(Cl)c(Br)c2)C(C)C1 66533,Cc1nc(C=CC(=O)NC2COCCN(C(C3(C4CC4)CC3)=O)C2)[nH]c1C 66534,CN1CCCCC1C(N1CCC1C(=O)NC1(C(O)CO)CC1)=O 66535,c1(NC(c2cc(C(=O)NC3CCCSC3)on2)=O)ccc(CCOCC)nc1 66536,C1(NC(CNC(CC(=O)NCC)=O)=O)CCCCN(C(c2ocnc2CC)=O)C1 66537,C1(C(=O)NCCNC(C2(OCC)CC2)=O)CC12CCOC2 66538,C(=O)(C1CCc2c[nH]nc21)N(CCCNC(c1ccn(C2CCC2)n1)=O)C 66539,c1(C(N2CC(C)N(C(=O)CC3CCCC34CC4)CC2)=O)ccc(O)c2ncccc12 66540,C1(NC(C2CCCC3(CNC3)C2)=O)CCC2(CCN(C(=O)CS(=O)(=O)C3CC3)CC2)C1 66541,Cc1cccc(C=CCN(Cc2nonc2C)CC2CC2)n1 66542,Cc1cc(C(=O)NCC2CN(C(C3(O)CCC3)=O)CC2C)c(Cl)cn1 66543,n1(CC(=O)OC)cc(C(=O)NCCC2CN(C(C3(O)COC3)=O)C2)nn1 66544,N1(C(c2c(CC)occ2)=O)CCC(C)(C(=O)N(CCC(N)=O)C)C1 66545,C(=O)(NNC(=O)c1cncc(OC(F)(F)F)c1)Nc1nc(OC)sc1 66546,c1(NC(=O)Nc2ccc(C3CS(=O)(=O)CC(=O)N3)cc2)ccc2ncccc2n1 66547,C(CC(=O)NCCCCCCF)(C(F)F)NC(CC(C)c1ccco1)=O 66548,C1(C)(C(=O)NCC(=CC(=O)NCCCC2C(C)C2)C)CC(=O)C1 66549,C1(NC(=O)COc2ccccn2)CCCN(C(c2cc(C(=O)C3CC3)on2)=O)C1 66550,Cc1nccc(C(N2CCC(C(C)C)C2CNC(=O)Cc2ccc(F)cc2)=O)c1C 66551,C(CC(=O)NC1CC2C(NC(c3cccc(N)c3F)=O)C2C1)(C(F)(F)F)OC 66552,CC(CC(F)F)C(=O)NCC(O)CNC(c1ccnc(C(F)(F)F)c1)=O 66553,N1(c2n(CC(=C)C)c(-c3cscc3SC)nn2)CCC2C(C)CCC2C1 66554,N1(C(C)C(=O)NC(C2(O)CN(C(C3CCC(=O)O3)=O)C2)C)CCCCCC1 66555,N1(C(CCOCCC)=O)CCC2(CC1)CC(NC(=O)C(C1CCCO1)C1CC1)C2 66556,C1(O)(C(C)NC(=O)Cc2cnoc2)CCN(C(=O)CCCN2C(=O)CCC2=O)C1 66557,CC1CCN(C(=O)Cc2conc2C2CC2)CC1NC(=O)CCc1ccccc1 66558,n1(COC)ncc(C(=O)NCCCCCNC(=O)C(F)OC(F)(F)F)c1C1CC1 66559,N1(C(=O)CCCn2cncn2)CC(C(N2CCS(=O)(=O)CC2)=O)C(F)(F)C1 66560,c1(C(C(=O)NCCC=CC)NC(=O)CC2CC2c2ccccc2)ccccc1 66561,CC(C)C(O)CNC(=O)C(c1ccoc1)NC(=O)C(C)n1cccn1 66562,C1(C(=O)NC(CN(C)C)CCO)(CC)CCCN1C(C1CC(N=[N+]=[N-])C1)=O 66563,Cc1cnc2c(C(=O)NCC(CO)NC(=O)Cc3ccc(C)o3)c(C)nn2c1 66564,N1(C(C(C)=NOCC#N)=O)CC(C(N2CCc3ncsc3C2)=O)C(C2CC2)C1 66565,c1(CNC(C23CC(c4ccccc4)(C2)C3)=O)cn(Cc2ccc(Cl)s2)nn1 66566,c1(C(N2CC(O)(C(C)NC(C(C)Cc3cnc[nH]3)=O)C2)=O)ncnc2c1CCC2 66567,C1(C(N(CC(C)(C)C)C)=O)CCCN(C(=O)Cc2cnn(C)c2)CC1 66568,CC(CC(F)F)C(=O)NC1CC=CCC1C(N1CC(O)(CCO)C1)=O 66569,c1(C(=O)NCCNC(c2c(C)cccc2Br)=O)ccc2nc(N(C)C)[nH]c2c1 66570,c1(CCN2CCN(C)CC2)c(F)cc(C(N2CCC(C(=O)OC)C2)=O)cc1F 66571,CCCC(CNC(=O)CC(COC)NC(c1ccn(CC)n1)=O)CCO 66572,CN1CC2CC2(C(=O)NCC2CCCCC(n3cc(CSC)nn3)C2)S1(=O)=O.C(=O)O 66573,N1(C(C2(F)CCS(=O)(=O)C2)=O)CCC2(CC1)CN(c1ccnc3ncnn13)CCO2 66574,c1(OC(C)C)ccc(CCC(=O)NCC(C)N(C(=O)C=Cc2cnc[nH]2)C)cc1 66575,Cc1ccc(-c2csc(NC(=O)CN3CC(F)CC3CO)n2)cc1 66576,Cc1cnc(NC(C)(CN(C)C)C2CC2)c(S(=O)(=O)NCC2CCC(C)C2)c1 66577,C1(C)(C(=O)NCCCNC(C2(NC(C)C)CC2)=O)CCOC1 66578,n1(CC)ccc(C(=O)NCC2CCC(NC(C3(OCC)CCOCC3)=O)C2)c1C 66579,C1(C(C(=O)N(C2CCN(C(c3cscc3Cl)=O)C2)C)O)CCOCC1 66580,c1(C(=O)NC2CC(NC(=O)Cn3cccn3)CC2O)cc(F)c(F)c(Cl)c1 66581,C1(NC(C(NOC)=O)=O)CC(NC(c2ccc(C)cn2)=O)C12CCOCC2 66582,N1(C(C2CCCN(C)C2)=O)CCC2(CC(NC(C3(C)CCC3)=O)C2)C1 66583,C1(NC(c2ccc(OC)o2)=O)CCCN(C(c2sc(CC(C)C)nc2C)=O)C1C 66584,c1(C(C2CC2)(C2CC2)NCc2cc(C)on2)sc(N2CCCCC2)nc1C 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66744,CC(C)(CC(=O)NCC1CC12CC2)NC(C1CCC=CO1)=O 66745,c1(C(CNC(C2CC(OC)C2)=O)NC(=O)C(C)=C2CC2)ccc(C)cc1 66746,N1(C(C(C)N(C(=O)Cc2nnc(C)s2)CC)=O)CC2(C=CCO2)C1 66747,S(=O)(=O)(c1ccc(C#N)c(NCCCCF)c1)NC1C(C)CCC1 66748,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C(=O)C(C)CF)CCC12CCC2 66749,C1(NC(CCC(C)OC)=O)CN(C(=O)CCn2nc(C)cc2C)CC2CC12 66750,C1(NC(CC=C)=O)CCCN(C(c2cn(CCc3ccccn3)nn2)=O)C1C 66751,c1(C(=O)NC2CN(C(CCC3N(C)CCCC3)=O)CC2F)cc(N)cc(O)c1 66752,N1(CCn2c(SC)nnc2N2CCCCCC2)CCCC(Cc2ccccc2)C1 66753,N12CC(C3CC13)NC(=O)c1ncoc1C2=O.c1(CCC)csc(C)n1 66754,c1(C(=O)NCC2(F)CN(C(=O)CCC3CC(F)(F)C3)C2)cncc([N+](=O)[O-])c1 66755,CN1C(=O)Cc2c(C(=O)NCC3(F)CN(C(C4CCS(=O)(=O)C4)=O)C3)cccc21 66756,c1(C(N2C(CNC(C3C(C=C(C)C)C3(C)C)=O)CCC2)=O)ccc2ncncc2c1 66757,C(=O)(CC(C)C(=O)OC)NCCN(C(=O)Cc1cc(F)ccc1F)CCOC 66758,C1(O)(CNC(C2(CC=C)CCC2)=O)CN(C(=O)C(C)OCC2CCCO2)C1 66759,C(=O)(C(C(C)(C)N(C)C)C1CCCC1)NC1C(C(=O)OC)N(CC2CC2)CC1 66760,c1(CC)[nH]c(=N)sc1C(=O)NCCCCN(C(=O)C(C)C1CCCO1)C 66761,c1(C(C)C(N2CCCC(NC)C2)=O)ccc(S(=O)(=O)N(C2CCC2)C)cc1.N(C)C 66762,N1(C(CC2CCC(C)CC2)=O)CC(NC(=O)CCCC2CCCO2)CC(C)C1 66763,c1(SCC(=O)NCC(CC)NC(=O)C(C)OC)ccc(C)cc1 66764,Cc1c(Br)ccc(NC(=O)C(=O)NCCN(C)C)c1I 66765,Cc1cc2cc(C(=O)NCCN(C)C(C3(CF)CC3)=O)c(Cl)cc2[nH]1 66766,C1(C(=O)NC2CCC(CCC(=O)N(C)CC3(C)CCOC3)C2)(OC)CCOC1 66767,C(=O)(CC(CC1CC1)NC(=O)C(CC)OC)N1C(CCC#C)CCC1 66768,N1(C(C(C)S(N)(=O)=O)=O)CC2(C1)CN(C(=O)CC(C)(C)C)CC2CO 66769,C1(C)(OCC)CCN(C(C23COC(C(=O)NCC4CC4COC)(C2)C3)=O)CC1 66770,Cc1nc(CNc2nccs2)sc1C(=O)OCC1CCOC(C)C1 66771,N1(C(C2Cc3cscc3C2)=O)CCCCC2(C1)CN(C(=O)CCn1cccn1)C2 66772,C1(C(C(=O)N(CC=C)CCOC)NC(c2cnco2)=O)CC=CCC1 66773,c1(C(CNC(C)=O)NC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 66774,N1CC(NC(=O)C=CCCC(C)C)CCC1C.C=C1CC(CC(=O)OC)C1 66775,c1(C(C)NC(N2CCC2CC(CO)C(=O)O)=O)ccccc1C 66776,Cc1nc2cccc(C(=O)NC3COCC3CNC(C3CC(CN(C)C)C3)=O)c2[nH]1 66777,c1(C(CNC(C2(F)CCN(Cc3cnc(Cl)nc3)C2)=O)O)ccc(F)cc1 66778,c1(NCCCC(=O)NCc2nc(SC)nc(O)c2)ccc2c(c1)CCO2 66779,C12(CC)CC(CN1C(=O)COc1cnn(C)c1)NC2=O.C(CC(C)C)OCC=O.CC 66780,C1(CC(=O)NCC(C)NC(c2cc(C3CC3)n(C)n2)=O)COC2CC1C2 66781,c1(OC)c(NC(C23CC2CN(c2nccc(C#N)n2)C3)=O)ncnc1Cl 66782,N1(C(c2n(OC)cnc2C)=O)CCC2(CC1)CC(CNC(=O)C(F)C1CCC1)C2 66783,S(=O)(=O)(CCCCCS(=O)(=O)N=c1ccc(Br)c(N)[nH]1)N1C(N2CCN(C)C(=O)C2)CC1 66784,C123CCCCC1CN(C2)Cc1cn(nn1)C3.C1(C(=O)OC)OCCN(C)C1=O 66785,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 66786,C1(NC(C2(SC)CCC2)=O)COC2(CCN(C(c3ocnc3C(F)F)=O)CC2)C1 66787,N1(C(c2c(C)c(Cl)ccn2)=O)CC(C)N(C(=O)CC(F)(F)C(F)F)CC1C 66788,CC1C(CO)CCCN1C(=O)CCN(CCCO)C(c1ccc(Cl)s1)=O 66789,N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NCC3(C#N)CC3)C2)C1 66790,N(C(=NCCCCC(F)(F)F)NCC1(O)CCSC1)C(CCF)C 66791,C1(N(C)C(c2cccc3ccccc23)C2CC2)CC(C2CCCCC2)CCN1 66792,CC(C)C(O)CNC(=O)C(CC1CC1)NC(=O)CNC=O 66793,c1(OCC)ccc(Cl)c(NC(C2CCN2CCC2CCCC2)=O)n1 66794,N(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)C(Cn1c(C)nnn1)=O 66795,CC1CCCC(CC(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)C1 66796,CC(C(=O)N1CCOC(CCCNC(c2ccc(F)c(N)c2)=O)C1)C(F)(F)F 66797,c1(N2CCC(C(N(C(COC)(C)C)C)=O)C(O)C2)cc(C#N)nc(C2CC2)n1 66798,c1(C(N2CCN(C(COC)=O)C(c3ccncc3)C2)=O)cc2ccc(F)c(F)c2o1 66799,C1(c2cn(CC)nc2)CN(C(=O)Cc2cnn(C3CC3)c2Cl)CCO1 66800,C1(NC(CC(C)(C)N(C(c2c(C)coc2)=O)C)=O)CN(C)CC1(F)F 66801,C(=O)(CCN(C)C(C1CC1C)=O)NCC1C(C(=O)OCC)C1 66802,C1(CCC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1(C)CCSC1 66803,C1(NC(C=CC)=O)(CF)CCN(CCNC(c2conc2C2CCCC2)=O)C1 66804,Cc1cccnc1C(C(=O)N(C)CC1CCOC1)NC(=O)OC(C)(C)C 66805,C(C)(CCCC(=O)N(C)CC1CC1(C)C)NC(c1c(C)sc(Cl)n1)=O 66806,C1(NC(C2C(CC)CCN2C(c2nccnc2N)=O)=O)CCCC(C)(C)C1 66807,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 66808,c1(C(=O)NCC2CN(C(COCC(=C)C)=O)C2)c(N)cccc1Cl 66809,N1(C(Cc2c(C)occ2)=O)CC2CN(C(=O)COc3ccc(F)cc3)CC2(C)C1 66810,c1(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccc2nc(S)oc2c1 66811,C1(C(=O)NC(CC#C)CC(F)F)CCN(C(c2cnn(C(F)F)c2)=O)C12CCC2 66812,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 66813,N(C(=NCCCNS(C)(=O)=O)NCC1CCCCO1)C(CC)C 66814,CC1=C(C(=O)NC2CC3CC(NC(C4CCS(=O)CC4)=O)CC3C2)CCCC1 66815,CC1CCCN(C(c2c(NCCC3(C)CCCO3)cccc2)=O)C1 66816,c1(C(N2C(CCCNC(C3N(C(C)=O)CCC3)=O)CCC2)=O)c[nH]c(C)c(Cl)c1=O 66817,Cc1cnc(S(C)(=O)=O)nc1N1CCC(CC(=O)NC2(Cl)CC2)C1 66818,C(CC(C(=O)N1CC(O)C(O)C1)NC(C1SCC=C1C)=O)SC 66819,c1(C(C)NC(C(C)OCCC=C)=O)nc(CC=C)n[nH]1 66820,C1(C)(C(=O)NC2C=NN(C)C2=O)CN(c2cc(-c3ccccc3)ncn2)CCO1 66821,CC1CCN(C(=O)CCc2c(Cl)cncc2Cl)CC1NC(=O)C=CC1CC1 66822,c1(C(=O)NC(CCCC)CNC(=O)Cn2c(C)csc2=O)cnc2[nH]nnc2c1 66823,C1(CNC(C(C)N(C)C)=O)CCCC1NC(C1CCC2CC12)=O 66824,c1(NC(C2CN(C(=O)COc3ccsc3)CCO2)C)ccc(F)cc1[N+](=O)[O-] 66825,c1(C(=O)NCCC(C)NC(CC(CCC=C(C)C)C)=O)cc2c(C)cccc2o1 66826,C1(CNC(CC=CC=C)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 66827,N1(C(C2CCOCC2)=O)CCC(N(C(C2(C3CCCO3)CC2)=O)C2CC2)C(F)C1 66828,C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NC1CC(NC(C(CC(=O)OC)C)=O)C1 66829,N1(C(C2(CC)COC2)=O)CCCC2(CCN(C(c3ccc4nonc4c3)=O)C2)C1 66830,C1(N(C)C(c2ccc(C(F)(F)F)o2)=O)CN(C(c2ncsc2C2CC2)=O)CC1F 66831,c1(CC(C)NC(=O)Nc2nc(Cc3ccccc3)ns2)cc(Cl)ccc1Br 66832,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CCC)oc2)=O)CC1 66833,C(=O)(C1=CS(=O)(=O)CCC1)NC(C(C)NC(=O)CCC1CC1CC1CC1)C 66834,n1(CC)cnc2nc(N3CCN(C)C4(CCC4)C3)nc(N(CC(F)(F)CC)C)c12 66835,CCC(CC(C)CO)NC(=O)CC1CCN1C(C1CC(N=[N+]=[N-])C1)=O 66836,CCS(=O)(=O)CC(=O)NCCN(C(=O)C1=CCC1)C(C)C 66837,CCC(CNC(=O)CC1CCCC1NC(=O)CCC(=O)N(C)C)C(C)C 66838,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCF)C2 66839,C1(NC(c2ncc(OC)nc2)=O)CCCN(C(=O)CN2CC3CCC2C3)CC1CO 66840,C(=O)(C(C)(C)CC(F)(F)F)NCCC(C)NC(Cc1c(CC)noc1CC)=O 66841,c1(C(=O)NC2C(C)(C)CN(C(=O)CCSC(F)(F)F)C2)ccnc2c1CCN2 66842,C(=O)(CN=c1[nH]c(C)cs1)NC1CCC(CNC(c2cc(OC)nc(Cl)c2)=O)C1 66843,N1(C2CN(C(=O)NCC3CC3c3ccco3)C2)CCCS1(=O)=O 66844,c1(OCC(=O)NC2CCOC2C(F)F)ccc(C2CC2)cc1Cl 66845,c1(NC(C(F)OC)=O)cccc(NC(c2cn(C(C)C)nn2)=O)c1 66846,C1(C(C)C)CN(C(=O)CC(C)c2ccncc2)CCN1C(C1(C)CC1(C)C)=O 66847,C12CCCN1N(C)CC(C)NC2=O.c1(C=O)ccccc1.C1(C=O)COC(=O)N1 66848,C(=O)(C(F)C(F)(F)F)N(CC(C)NC(c1ccc(C(F)(F)F)cc1F)=O)C 66849,CN1CCC(C(=O)NC2(CCNC(C3CCC(F)C3)=O)CCC2)CC1=O 66850,N1(C(C(C)(C)NC(C2CCCOC2)C)=O)CC(C#N)(S(C)(=O)=O)C1 66851,C(c1ccc(F)nc1)=CC(=O)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)C 66852,C1(NC(c2ccc(CNC(C)=O)cc2)=O)CCCN(C(c2nscc2N)=O)CC1 66853,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)Cc1cn[nH]c1 66854,C(=O)(C(C)(O)C(F)(F)F)N1C(CCNC(C2CCCCC2)=O)CC(OC)C1 66855,C(CCC(CCC)CN(c1n[nH]c2c1CCC2)C(C)=O)NC(C=CCC)=O 66856,C1(CNC(C(C)SCC)=O)(CO)CCCN(C(C2CCCN2C(C)=O)=O)C1 66857,C(=O)(CC1=CCOCC1)NC1CCC(CNC(c2nc(C)n(C)c2)=O)CC1 66858,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 66859,Cc1cc2ccccc2nc1C(N1CC2CCN(c3nncs3)CC2C1)=O 66860,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 66861,c1(NC2C(C(N3CCOCC3)=O)CCCC2)cc2ncnn2cn1 66862,N1(C(CC2(OC)CCC2)=O)CCOCC(NC(c2ccc(CO)c(F)c2)=O)C1 66863,N1(C(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(=O)C(c1cccc(C)c1)F 66864,c1(C(=O)OC)cc(OC(C)=O)c(C)cc1NC(=O)COC(c1scc(C)c1C)=O 66865,c1(C(N2CC(C)OC(CCNC(=O)C3=CCCCO3)C2)=O)cc(C#N)ccc1F 66866,c1(C(=O)NC2(CO)CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 66867,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(O)CN2CCCC2)C)C1 66868,C1(C(=O)NC(C(=O)NC2CC(O)C2)c2cccs2)CN2CCCC1C2 66869,CC(Cc1ccccn1)N=c1[nH]c(=NC(CF)c2cncs2)[nH]c2ccc(Cl)cc12 66870,Cn1ccc(-n2cc(CC3CCCN3C(c3ncc(Br)s3)=O)nn2)cc1=O 66871,C1(C(N(CC(N2CC(C#C)C2)=O)CC)=O)CCOC1C(=C)C 66872,c1(C(N2CCN(C(CCC=CC)=O)C(CO)C2)=O)nsc2ccc(C)cc12 66873,C1(C(N2CC(C(C)NC(C3CCSC3)=O)C2)=O)CC(=O)c2ccccc2O1 66874,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 66875,C(=O)(C#CC1CCCOC1)NCCOCCN(C(CC(C(=O)OC)C)=O)C 66876,CCC(C)C(C)(O)CN(C(=O)C(CC(C)C)ONC(C1CC12CCCC2)=O)C1CC1 66877,N1(CC=CC(=O)N(CCCN(C(=O)C(C)C(C)C)CC)CC)CCCCC1 66878,CC1CCCC(O)(CNC(=O)NCCn2cc(C(C)(C)NC(C)(C)C)nn2)C1 66879,N1(C(C(CCC)C)=O)CCCC(C)(NC(=O)CCSc2n[nH]c(C)n2)C1 66880,c1(SCC)ncccc1C(=O)N(CC(C)(C)NC(=O)CSCCC#N)C 66881,Cc1ccc(Cl)c(C(=O)NCC2CCN(C(C3CC4CC4C3)=O)C23CC3)c1N 66882,C1(OC)CC(CNC(=O)CC(C)(C)C)N(C(=O)CCn2cncn2)C1 66883,CCCC(O)C(CO)NC(=O)CC1CCCC(NC(=O)CCc2cnn(C)c2)C1 66884,C(=O)(C(F)C(C)(C)O)NC(C1CCN(C(=O)CCNC(=O)C=CCl)CC1)(C)C 66885,N1(C(C2NC(=O)OC2)=O)CCC=C(CNC(=O)CCc2nncs2)C1 66886,N(C(=NCc1cccs1)NC1CC12CCCC2)C(C)C1CC1 66887,c1(OC)cc(C(=O)N(C)Cc2ccccc2O)cc(C)c1 66888,c1(CNC(C(=O)NC2CCC(OC(C)(C)C)CC2)=O)ccc(Cl)cc1Cl 66889,C12(C(=O)NCC(C(C)O)O)CC(C(=O)OC(C)(C)C)(C1)C1(CCOCC1)O2 66890,N#Cc1cc(C(=O)NC23CCN(C(c4ccc(CO)s4)=O)CC2C3)c(O)cc1N 66891,C1(CC)(NC(=O)Cc2cccc(F)c2)CCN(C(C2CNC(=O)N2)=O)C1 66892,N1(C(C(CC(F)F)N(C(C=C(CC)CC)=O)C)=O)CC2CC(C1)C2(C)C 66893,N1(C(c2c[nH]nc2C2CC2)=O)CCOCC(n2cc(C(=O)N)nn2)C1.[nH]1cccn1 66894,N(C(=NCCc1ccccn1)NC1CCC1)C1CCC(C2(O)CCC2)C1 66895,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(=O)Cc3cnco3)CC2)c1 66896,c1(CCN2C3CCN(C3)C2=O)cncc(Cl)n1.c1(N(C)C)ccccc1 66897,C1(CC)CN(C(=O)Nc2cnc(-c3ccsc3)cn2)CC1SC 66898,Cc1cc(CO)cc(Cn2ccnc2C)c1.n12cc(nn1)C1CN(C1)C(=O)CC2 66899,CCCC(CC)CC(=O)N1CC2CCC(C1)N2c1nc(Cl)ncc1C 66900,C1(NC(CN(CC(=O)NC(C)C)C)=O)CN(C(=O)C(C)CN(C)C)CC1F 66901,N1(C(c2ccc(CNC(=O)CCCN3CCNCC3)cc2)=O)CCC2CC2C1 66902,C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)(C)N(C)C)CCC1CO 66903,C1(COC)CC(CNC(C2CC2C(C)(C)C)=O)N(C(=O)COCC(C)C)C1 66904,c1(CN(C)C(C23COCC(C2)C3)=O)ccccc1CNC(C1(F)CC=CCC1)=O 66905,c1(C(=O)NC2(CCNC(C3(CC#C)CCCO3)=O)CCC2)nnn2c1COCC2 66906,C(=O)(C(C)(C)C(C)(C)C)N(C1CN(C(C2C(C(=O)OCC)CC2)=O)C1)C 66907,Nc1ncc(C(N2CC(CCCCNC(c3ccco3)=O)C2)=O)cc1Br 66908,c1(C(=O)NC2CCC(N(C(=O)CCc3cccc(F)c3)C)C2)nccc(N)c1Cl 66909,c1(C(N2CCN(C(=O)OC(C)(C)C)CC2C(F)F)=O)cc(F)cc2nccnc12 66910,Cc1ccc(F)c(CN2CCN(Cc3cnc(Cl)c(Cl)c3)CC2)c1Br 66911,C12(CCSC1)C(=O)N2.C1(C#N)(CC(=O)NC2(CC(=O)OC)CC2)CCC1 66912,C(=O)(C(C)(C)C(=O)NC(C1CCCCN1C(c1cc(Cl)cn1C)=O)C)OCC 66913,C1(C(C)NC(=O)CNC(=O)C2CC2)CCN(C(=O)CC(=O)N)C1.C1(CCO)CCC1 66914,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1C1CC1)=O.c12cc(on1)CNC2=O 66915,C1(C(N(C(C)CNC(=O)CCn2cncn2)CC)=O)CC(C2CCC2)C1 66916,c1(OC)cc(C(N)=O)ccc1-c1cn(CCC(=O)NCCCCCl)nn1 66917,Cc1[nH]c2ccccc2c1CC(N1CCC2(C1)CN(C(C13CCC(C1)C3)=O)C2)=O 66918,C=CCC(C(=O)N1CC(CNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 66919,c1(CC(=O)NC2CN(C(c3c(C)noc3C)=O)C2)cc(F)cc(C#N)c1 66920,c1(NC(CN(C(C2C(C(=O)OCC)C2)=O)C)C)cc(CC)nc(C)n1 66921,N1(C(=O)CCN2CCC2)CCCCC(CNC(=O)CNc2ncccn2)C1 66922,N1(C(CC=C)=O)CC(CN(C)C(c2cc(Br)ccc2C)=O)C2(CC2)C1 66923,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2F)=O)CC12CC2 66924,C12(CCCCC1C)C(=O)N2.C1(OCC)(CNC(=O)CCOC)CCC1.N(C)C1CC1 66925,C(CCC(C)(C)C(=O)O)N(C(c1ncc(F)c(C2CCC2)n1)=O)CC 66926,N1(C(C=CC(=O)N(C)C)=O)CCCC(N(C(=O)C(F)Cc2ccccc2)C)C1 66927,c1(C(=O)OC)ccccc1NC(c1nccc(NC(c2ccccc2)C)n1)(C)C 66928,CC(C)CCC(CO)NC(c1sccc1CNC(c1ccnc(O)c1)=O)=O 66929,CC1CN(C(=O)Cc2cc(C3CC3)nn2C)CC1NC(C1CCC(=O)N1C)=O 66930,c1(C(C(=O)N(CCNC(C2CCCOC2C)=O)CC)C)cccc2ccccc12 66931,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 66932,c1(N(C)Cc2ccccc2CNC(=O)C=C2CCCCC2)ncc([N+](=O)[O-])cn1 66933,c1(C(=O)OC)ccccc1Cn1cc(CCC2CCCN2C(=O)C2=CCCC2)nn1 66934,c1(C(=O)NCC(C)(C2CC2)NC(c2nncs2)=O)ccc(-n2ccnn2)cc1 66935,n1(C(CC)CC)nccc1C(=O)NCC1CC1CNC(=O)CNC=O 66936,C(CCN(C)C(c1cnc(C2CC2)s1)=O)(C(C)C)NC(c1ccc(CCC)[nH]1)=O 66937,Cc1csc2ccc(CC(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 66938,C(N=c1cc(NCC2CCCO2)nc(-c2ccccc2)[nH]1)c1nccc(SC)c1 66939,C1(C(=O)NCC(CNC(c2ccc(OC)s2)=O)O)COc2ccc(Cl)cc2O1 66940,C1(C(C(=O)NCC2CC(CCC)C2)NC(=O)CCC2CC2)CC=CCC1 66941,C(CC(C(C)(C)C)NC(c1ccnc(C(F)F)c1)=O)N(C)C(C1CC=CCC1)=O 66942,N1(C(C(C)SC(C)C)=O)CC2(CCCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 66943,N1(C(c2ccc(Cl)c(F)c2)C(=O)NC)CCOC2CS(=O)(=O)CC12 66944,Cc1nc(C(N2CCC(CCC(C)(C)C)(NC(C3C4CCC34)=O)C2)=O)oc1C 66945,C#Cc1ccc(CC(=O)N(CCC(=O)NCCN2CCC(=O)CC2)CCCO)cc1 66946,C1(OC)CCC(CC(N2CC(n3cc(C(=O)OC(C)C)nn3)C2)=O)CC1 66947,Cc1cc(F)c(F)cc1C(N1CCC2CC12C(=O)Nc1ncc(Br)nc1Cl)=O 66948,c1(C(=O)NC2C3CN(C(c4ccc(C#N)o4)=O)CC32)cc([N+](=O)[O-])cc(O)c1O 66949,C1(CC)CN(C(=O)Cc2cccnc2)CCC1NC(c1sncc1C)=O 66950,N1(C(CCS(=O)(=O)N(C)C)=O)CCOC2(C1)CN(C(C1(Cl)CC1(C)C)=O)C2 66951,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 66952,C1(CC(=O)NCC(CO)NC(=O)CNc2ccccc2)CCCCCC1 66953,Cc1ccccc1C=CC(N1CSCC1C(N1CCCCC(CO)C1)=O)=O 66954,C1(CC)CC2(CCCN2C(=O)C(CCCCC)NC(=O)OC(C)(C)C)C1 66955,N1(C(C2(CC=C)CCN(C(c3csnc3OC)=O)C2)=O)CCC2(CCSC2)C1 66956,N1(C(c2ccc(CC)cn2)C(=O)NC(C)C)CC(C)(C)OC2(CCC2)C1 66957,c1(C(N2CC3CN(C(C(C)(C)C(F)F)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 66958,N1(C(CCC#N)=O)CC2CS(=O)(=O)CC2(NC(C2CC2c2ccc(F)cc2F)=O)C1 66959,N1(C(C2C(C)OCC2)=O)C2CCC1CN(C(=O)C(c1ccccn1)C)C2 66960,c1(OC)c(C(=O)NC2OCCN(C)C2=O)ccnc1Cl.C12CCCN(C1)C2=O 66961,C1(NC(c2c(C)nnn2C)=O)CC2CC(C1)N(C(=O)Cc1cncc(F)c1)C2 66962,Cc1cc(C(=O)NC(C)CCCNC(c2ccc(Cl)o2)=O)cc(C)c1N 66963,C1(C(=O)NCc2cc(C(=O)NCC(C)OC(F)F)sc2)CCC(N=[N+]=[N-])C1 66964,c1(NC(C2CC(F)CN2C(C2CCOC2)=O)=O)cnc(Br)nc1 66965,c1(C(=O)NC2(CCNC(CCc3cn(C)nc3)=O)CC2)cnc2[nH]ccc2n1 66966,C1CN=C(NCC(C)OC)NC12CC2.c1(N)cnccc1Cl.c1(OC)ccccc1C 66967,C1(CNC(C(Cc2ccccc2)OC)=O)CN(C(C2OCCO2)=O)CCO1 66968,CC(C)C(C)C(CNC(=O)COC1(C)CCC1)NC(c1cc(C#N)cs1)=O 66969,c1(NC)cccc(C(=O)N(CCCC(N2CC(O)(C(F)(F)F)C2)=O)CCO)n1 66970,C(C(N=c1[nH]c(=NCC2CCCS2)[nH]c2cc(C(F)(F)F)ccc12)C1CC1)OC 66971,c1(COC(c2ccc(-c3nnn(CCSCC)n3)o2)=O)cc(C)cc(Br)c1O 66972,c1(C(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)cnc(O)c2ccccc12 66973,N1(C(C2CCCN2Cc2ccco2)=O)CCC2(CCCc3ccccc32)C1 66974,c1(C2(C(N3CC(C#C)C3)=O)CC(C(=O)OC(C)(C)C)C2)cccc(Cl)c1F 66975,C1(C)(C(=O)NCC(C)C=O)CC(N)C1.C(=O)(C(COC(C)(C)C)OC)OC 66976,c1(CC(N2CC(C)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)ccc2sccc2c1 66977,N1(C(c2c(CC)cns2)=O)CC2=C(C1)CN(C(c1cc(C)c(C)[nH]1)=O)C2 66978,CC(CCC(C)(C)C)C(=O)NCC=CC(=O)NC(C)Cn1cnnc1 66979,C1(CCCNC(COCC(C2CCC2)OC)=O)CCCCO1 66980,C1(C(=O)OC)(NC2(CC(=O)NC3CCCC(C(F)(F)F)C3)CCC2)CCCCC1 66981,c1(C(CNC(N(CCOC)Cc2noc(=N)[nH]2)=O)O)ccc(O)cc1 66982,N1(C(CSCCOC)=O)CC2CCN(C(c3ccc(C4CC4)nc3C)=O)CC12 66983,O=C(C1=NOC2(CCC2)C1)N1CC(C2CC2C(=O)NCC23CCC(CC2)CC3)C1 66984,c1(C(=O)NCC2CN(C(Cn3c(C)ccn3)=O)CC2C)ccc2nc(=N)[nH]n2c1 66985,C(c1cncc2ccccc12)=CC(=O)NC(C1N(C(CC(C)C)=O)CCC1)(C)C 66986,C1(NC(c2nc(CCC)oc2)=O)CC(N=c2[nH]c3cccnc3s2)C1 66987,C12(C(=O)NC(C(=O)N(C(C)C)C)CC3CCC3)CCC(CC1)C2 66988,CCS(=O)c1ccccc1C(=O)NCC1CC1NC(c1nccc2ccsc12)=O 66989,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 66990,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 66991,Cc1ccc(CNC(C2CCN(C(=O)CN3CCCCC3)CC2)=O)c(F)c1F 66992,C=CCC(C)C(=O)N(CCCCNC(C1(C(=O)NC)CCCOC1)=O)C 66993,CCC(O)C(C)(C)C(=O)NCC1(O)CC(C(=O)N(CCC(F)(F)F)C)C1 66994,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2c(Cl)cn(CCC)n2)=O)CCN(C)C1 66995,Cc1c(C(=O)NCCCOc2ccccc2)noc1-c1ccccc1 66996,C1(CNC(c2c(C)cco2)=O)CC2(CCO1)CCN(C(C1C3COCC13)=O)C2 66997,c1(C(=O)NCCOCCN(C(c2ccc(C)c(O)n2)=O)C)ccc2nccn2n1 66998,C12CCCN1NC(=O)C1CN(CC1F)C2=O.CCC(C1CC1)SC 66999,c1(C(N2CCCCC(CC(=O)NCc3ccc(C)nc3)C2)=O)c[nH]c2cnccc12 67000,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCC2)=O)C1 67001,CC1(F)CCC(C(N2CC=CC2Cn2cc(C3CCCSCC3)nn2)=O)CC1 67002,C1(C(=O)NCCN(CCC)C(c2cc(C)ccc2OC)=O)CCC2C1C2(F)F 67003,N1(C(CC(C)(C)n2cc(S)nn2)=O)CCCC(O)(CC#N)C1.C1(F)CCOC1 67004,N1(CC(=O)NC(=O)NCC=C)CCC(C)(NC(=O)Cn2cc(C#N)cn2)C1 67005,c1(N(C(C(=O)NC(C)CC2CCC(C(F)(F)F)CC2)=O)C)ccc(F)c(F)c1 67006,C1(NC(C(CN(C)C)O)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1CO 67007,C(=O)(C1CCc2ccccc21)N1CCCC(N(C(c2c(C)cco2)=O)C)CC1 67008,N1(OC(c2ccsc2C(=O)O)=O)CCN(Cc2n(C)nnc2)CC1 67009,C1(NC(C2(C3CC3)CC2)=O)CN(C(C(C)Sc2ccccc2)=O)CCC1N 67010,c1(NC)ccc2[nH]c(C)c(C(=O)NCCCC3(NC(=O)OC(C)(C)C)CC3)c2c1 67011,N1(C(c2c(C)cn(C)n2)=O)CCC(O)(C(C)NC(=O)C(C)n2ccnc2)CC1 67012,C(=O)(CCCCC(C)(C)C)Nc1c(C)ccs1.C1(=O)C(N)CCCN1.C1(C)CC1 67013,C=CCC(CC)C(=O)NC(c1cccc(Cl)c1)CNC(C1(O)CC(C)(C)C1)=O 67014,C1(C)(CC(C)(C)c2ccccc2)N2CCC(C2)O1.CCCCCCNCC1CC1 67015,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67016,N12CCC(O)C1NC2=O.Cc1cnsc1C(N1CCC1C1CCOCC1)=O 67017,C(=O)(CCC(=O)N(C)C)N(C1CCN(C(C23CC(C)(C2)C3)=O)C1)CCC 67018,C=CCCCCC(=O)NC(CNC(C1CCCC(C)(C)O1)=O)CO 67019,C(C(=O)N1CC(F)(F)C1C1CC1)(C(C)(C)C)N(C(Cc1c(C)nccc1)=O)C1CC1 67020,Cc1c(Br)ccc(F)c1C(N1CCOCC(C(=O)NCCC(C)CO)C1)=O 67021,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)Cc2ccon2)CC(F)C1 67022,O=C1CNC(=O)C(CC(=O)NCCN2CCN(C(=O)CNC=O)CC2)N1 67023,C1(C)(C(N2CC(SC)C(n3cc(CCc4nn[nH]n4)nn3)C2)=O)CCCCNC1=O 67024,C(C1c2ccccc2CN1C(C1CC2COCC2C1)=O)NC(C1N(C=O)CCC1)=O 67025,C1(CC)CN(C(=O)CSCC(F)F)CC1C(=O)NCC(Br)=C(C)C 67026,N1(C(C2CC3CC3N2C(c2ccc(CO)c(F)c2)=O)=O)CCCC2CCCCC12 67027,c1(NC(c2nc(OC(C)=O)sc2)=O)ccc2nc(Br)sc2c1.C12CC1CNC2=O 67028,C(=O)(C(F)C(C)(F)F)NCc1ccc(C(N(CC#C)CC2CCC2)=O)s1 67029,N1(C(c2ccc(OC)s2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1CC1CC1 67030,C1(NC(=O)NC)CCCC(NC(=O)C(N2CCCC2c2sccc2C)=O)C1 67031,C12(CC(N3CCC4CC34)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67032,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67033,c1(OC)c(F)cc(CN2CCN(C(c3ccc(F)cc3Cl)=O)C(CO)C2)cc1Cl 67034,C=CCC(CNC(=O)CN(CC)CC)C(=O)N1CCC(CCO)C1 67035,C(CC1=CCN(C(c2cc(F)c(Cl)cc2Cl)=O)CC1)NC(=O)C(F)CC1CCC1 67036,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CC1C)C 67037,C#CCC(C)(C(=O)NCC1CC(=O)N(C)C1)NC(=O)C(c1ccccc1)=O 67038,C(C(N=[N+]=[N-])C(=O)NCC(CNC(=O)CCC1CCC1)C(F)(F)F)OCC 67039,C1(CC(=O)N(C2CCN(C(C3(F)CCC3)=O)C2)CC)CC2(CC2)CO1 67040,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67041,c1(C(=O)NC(CNC(C=CCC)=O)C2CCC2)cnc(CC2CC2)s1 67042,C1(C(=O)NC2CCC(NC(C3CC34CCC4)=O)CC2)CC2CSCC(C1)C2 67043,N(C(=NCCSC)N(C)Cc1cc(F)c(C)cc1F)C(C1CCCO1)COC 67044,C#CC1CN(C(=O)C(c2c(C)cccc2Br)NC(=O)CCCCN(C)C)CCO1 67045,Cc1c(Br)noc1C(N1CCC(n2cc(C(=O)NCCN(C)C)nn2)C1)=O 67046,C(CCNC(CC1CC(=C)C1)=O)(C(=O)N(c1ccccn1)C)CCN1CCCC1 67047,c1(C(=O)NCC(CNC(c2cc(CCC)nn2C)=O)(C)C)cc2occc2[nH]1 67048,C(=O)(CCCCCSC)NCC1(CCCNC(C(CC=C)C)=O)CCCC1 67049,N1(C(CCC#C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67050,c1(C(N2C(COC)CCC2)=O)c(NC(=O)C(C)CBr)cccc1F 67051,c1(C(=O)NC(CNC(c2cc(C)c(C)o2)=O)C2CC2)ccn2nccc2n1 67052,CC(C)C1=NOC(C(N2CC=CC2CNC(=O)CCC23CCC(CC2)C3)=O)C1 67053,C12CC13CCN(CC3)C1(CC1)CN2.N1(c2ncn(C)c(=O)c2)CC2CCC(C1)N2C 67054,c1(N2CCCC(CNC(C)=O)C2)ccc(S(=O)(=O)NCCCCO)c(Cl)c1 67055,CC(C)(C)C#CC(=O)NCC1CCCCN1C(=O)CC1CCC(=O)O1 67056,N1(C(C(CCC)OC)=O)CC2CCCC1(CNC(C1CC13CC3)=O)C2 67057,N1(C(c2c(OC)ccs2)=O)CC2(C1)CN(Cc1cccc(Cl)c1O)CC2CO 67058,Nc1c(C(=O)NC2CC2NC(C2CCC(N(C)C)CC2)=O)cccc1[N+](=O)[O-] 67059,c1(C(=O)N(C2(C)CN(C(C(CC)NC(C)=O)=O)C2)CC)c(C)nc2ccccn12 67060,C=C(C)C(O)CC(=O)NCCC1CN(C(=O)CCCc2nc(CC)no2)CCO1 67061,c1(C(N(C)CCNC(c2cc(F)c(F)cc2Cl)=O)=O)cc2n(n1)CCNC2=O 67062,c1(C(N2CCN(C(CCC(C)OC)=O)C(CCO)C2)=O)nc2ncccn2n1 67063,c1(NC(=O)NC(c2cncc(C)n2)C2CC=CCC2)cc(C(F)(F)F)ccc1I 67064,C(=O)(CC(CC)C(F)F)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67065,C(=O)(C(F)CCC(C)(C)C)NC1(C(C)C)CCN(C(c2c(CC)ccs2)=O)C1 67066,C#CCC(CC(F)F)C(=O)NC(C(=O)NCC1=C(C)CCOC1)C(C)CC 67067,N1(C(c2cc(OC)no2)=O)C(C(=O)Nc2sncc2C#N)CC2CC12 67068,CN(C(=NCC1C=CCCC1)NC1CCC1)Cc1ccco1 67069,c1(CC(=O)NC2CC(NC(c3ccsc3)=O)CC2O)n[nH]c2ccccc12 67070,c1(C(=O)NCC2N(C(c3c(C)c(N)ccc3)=O)CCC2C)[nH]nc2ncnc(O)c12 67071,c1(CC(=O)NCCC(C)NC(c2c(F)ccc(CC)c2)=O)cnn2c1CCCC2 67072,C1(=O)C(C)(CC#C)N1.C(=O)(CCC=C(C)C)NCCSCCOC#C 67073,CC1=C(C(=O)NCC(C(C)C)NC(C2CCCCN2N=O)=O)SCCO1 67074,c1(C(N2CC(C(C)(C)O)(CNC(C=NOC)=O)C2)=O)nc(C)c(C)nc1C 67075,Cc1cccc(C)c1C(=O)NCC1(C)CCN(C(C2CCC(O)CN2C)=O)CC1 67076,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67077,c1(NC(CN2CCN(C(C=CCCC)=O)CC2)=O)cnc2c(C)nsc2c1 67078,Cc1cccc(N2CCC(N3CCC(n4cc(-c5cnn(C)c5N)nn4)C3)C2=O)c1 67079,C(F)(c1ccccc1)=CC(=O)NCC1CC(O)CN1C(c1cc(C2CC2)no1)=O 67080,c1(CC(=O)NCC(C2(O)CN(C(C(C)=C3CC3)=O)C2)C)ccncc1C 67081,N1(C(C=C(CC)CC)=O)CC2CC(NC(C3CC3c3ccccc3Cl)=O)CC1C2 67082,CC(C)C(F)C(=O)NCCN(C(C1CC(=C(F)F)C1)=O)C1CC1 67083,C(CN=c1cc[nH]c(C(F)(F)F)c1)NCC(N1CCC(NS(=O)(=O)C2CC2)CC1)=O 67084,c1(C(N(CC(C)NC(=O)C(C(C)O)N(C)C)CC)=O)cnc(N)c(Cl)c1 67085,N1(S(CC(=O)OCC)(=O)=O)CCC2CN(C(=O)Nc3nnc4n3CCC4)CC2C1 67086,C(=O)(C1=NOCC1)NCCC(CNC(c1c(CCCC)ocn1)=O)OC 67087,c1(C(=O)NCCC(=O)N(CC#C)CC2CCOC2)cccc(C#N)c1 67088,CCC(C#N)C(=O)Nc1cccc(NC(=O)C=CC(=O)NC2CCCCO2)c1 67089,C12(C(=O)OC)CCCC(CNC3CC4(C3)CC(N3CCOCC3)C4)(C1)OC2 67090,C(CCS(C)(=O)=O)(C(=O)NC(CNC(C1(c2ncccc2F)CC1)=O)CO)OC 67091,C12(C(N3CCC(CCNC(c4cc(C#N)[nH]c4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 67092,Cc1ccccc1CCC1CCCN(C(=O)NCCCCc2cncnc2)C1 67093,C1(OC)(CNC(c2cc(C3CC3)on2)=O)CCN(C(C2CCCCO2)=O)CC1 67094,Cc1ccc(C)c(C(=O)NCC2(C)CCCN(C(=O)CCC3CCC(=O)N3)C2)n1 67095,C1(CNC(C(C=C)OC)=O)COC(C)(C)CN1C(c1ncc(F)cc1F)=O 67096,Cc1cc(C(=O)N(CC(O)CNC(=O)C=CC2CC2)C)cc(O)n1 67097,c1(C(N(CCN(C(C2CCC(C)NC2=O)=O)C)C)=O)cccc2c1CCN2 67098,n1(CC(=O)N(C2CCN(C(=O)CC3CCC4CC34)C2)CC)nc(C)oc1=O 67099,c1(C(N2CC(C3(NC(C(C)SCCC)=O)CC3)C2)=O)cc(C)c(OC)c(Cl)c1 67100,C(=O)(CCS(=O)(=O)Cc1ccccc1)NCC1C(C)CN(C(=O)C#CC2CCC2)C1 67101,Cc1cc(C(=O)NC(C2CN(C(C34CC(C(F)(F)F)(C3)C4)=O)C2)C)on1 67102,N1(C(C(C)S(N)(=O)=O)=O)CCC(C2CC2)(CNC(=O)CCc2ccc(O)nc2)C1 67103,C1(C(N(CC(C)NC(=O)COCCC)CC)=O)COC1.C1C(=O)N1 67104,CCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)C(CO)N(C)C)CC1 67105,C1(C(N(CC(C)N(C(Cc2scc(C)c2)=O)C)C)=O)C(C)(C)C1(F)F 67106,c1(CCNC(=O)NC(CC(=O)NC(CCC=C)C)C2CC2)nc2ccccc2s1 67107,C(=O)(CCCCCN(C(=O)CC1CC(F)(F)C1)C)NC1CCN(C)C1 67108,c1(N2C(CNC(c3ccc(F)cc3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67109,N1(C(CCSc2ccc(C)cc2)=O)CC2CCC1CN2C(=O)C(C(C)O)N(C)C 67110,CCCC(O)C(=O)NC(C1CCN(C(=O)COCCc2ccc(Cl)s2)C1)C 67111,n1(CC#C)c(C)cc(C(=O)NCC2(O)CN(C(c3cn(C)nc3O)=O)C2)c1C 67112,C1(NC(CS(N)(=O)=O)=O)CN(C(c2ccc(-n3ccnn3)cc2)=O)C2CCCCC12 67113,c1(C(C)C(N2CC3(CC3C(=O)NCc3cncc(Cl)c3)C2)=O)ccc(Br)cc1F 67114,C(c1ccc(SC)cc1)=CC(=O)NCC1(C(C)(C)O)CN(C(C(CSC)OC)=O)C1 67115,c1(C(=O)NC(CN(C(C2(C)CC(C(F)(F)F)C2)=O)CC)C)ccn2nccc2n1 67116,CCC(CC)C(C)C(=O)N(CCC(=O)NCc1csc(C)n1)CCCO 67117,N1(C(C(N2CCCCCC2)C)=O)CCCC(CCNC(C2CC(CF)C2)=O)C1 67118,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67119,C1(NC(C(C2CC2)SC)=O)(CO)CN(C(c2ccc(C(C)=O)o2)=O)C1 67120,c1(CC)nnc2n1CCCC2C(=O)N1CC(NCc2cccc(Br)c2)C1 67121,CC1CCCC(C)N1C(c1ccc(CN2CCC(C(C)CN(C)C)CC2)[nH]1)=O 67122,N1(C(C2CCCN(c3c(Br)cnc(C(C)(C)C)n3)C2)=O)CCc2nocc2C1 67123,c1(CCC(N2CC(O)(CN(C(C(C)OCC)=O)C)C2)=O)ccnc(C)n1 67124,c1(OCC)cccc(Cl)c1C(=O)NC1CCCC(NC(=O)C(CC(C)C)OC)C1 67125,C1(CNC(c2[nH]cc(C)c2)=O)C(C)CCCN1C(c1sc(Br)cc1C)=O 67126,c1(CC(=O)NCCC(=C)CNC(=O)C(c2ccnn2C)C)csc2nc(C)cn12 67127,c1(C(c2nnnn2C2CCC2)NC(CC)C2CCC2)ccnn1CCC 67128,CC(C(C)(C)NC(=O)CCCn1cncn1)NC(=O)COCCc1ccccc1 67129,c1(CC)nnc2n1NC2C1CCCC1.c1(CCC2(C)CC2)cccc(C)n1 67130,C(=O)(C1=CCCCC1P(C)(C)=O)NCC(CNC(C(C)(C)c1ccns1)=O)CO 67131,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67132,N1(C(c2nc(OCC)sn2)=O)CC(NC(=O)CC(C)c2cccnc2)C(C)(C)C1 67133,Cn1nnc2c1CCN(C(=O)CCCCCNC(=O)C(C)(F)C(C)(C)F)C2 67134,Cc1c(C(=O)NCC(C)NC(C23CC2COC3(C)C)=O)cncc1Cl 67135,C1(CC)C(C)CCN1C(C1CC(NC(=O)C(C2CCC2)OC)CCO1)=O 67136,C1(C(=O)NC2CC(N(C)C(C3CC(O)C3)=O)C2)CCc2cnn(C)c2C1 67137,c1(OCC(=O)NCC(C(C)C)NC(=O)C(O)c2cnc[nH]2)cccc(Br)c1 67138,N1(C(C)=O)CCC(C(=O)N(CC(O)CN(C(=O)Cc2ncc(Cl)s2)C)C)CC1 67139,N1(C(CC23C(CN(C(c4c(CC)con4)=O)C2)CC3)=O)CC(=O)NCC12CC2 67140,c1(C(N)=O)ccc([N+](=O)[O-])c(N(CCNc2ccc([N+](=O)[O-])o2)C2CC2)c1 67141,N1(C(C(CCSC)O)=O)CC2CCN(C(c3cccc(Cl)c3N)=O)CCC2C1 67142,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CN2CCCC2=O)CC1O 67143,C1(C(=O)NC(c2onc(C)n2)CO)CC(C)CN1C(C1(O)CCCC1)=O 67144,C1(CNC(C(CC)OC)=O)CN(C(=O)CCNc2ccccn2)CCC1(C)C 67145,c1(-n2ccc(C(=O)NC3C(NC(=O)C=Cc4cscn4)C3)n2)ccccc1Cl 67146,c1(-n2ncc(C)c2)cccc(C(=O)NCCN(C)C(c2oc(CO)nc2C)=O)c1 67147,C(CCCCCCC(=O)N1CC2CC(NC(=O)C(c3ccccn3)O)C1C2)SC 67148,c1(C(=O)NCC2CCC(NC(c3ccc(C)nc3C)=O)C2)cc(C)cc(C)c1N 67149,C#CCC(CC(=O)NC1CCC(N(C(=O)C(C)=CC)C)C1)c1ccccc1 67150,C(=O)(CCCC(C)(C)C)N1CC(CNC(c2n(C(C)C)ncn2)=O)C1 67151,c1(C(N(CCNC(c2c(O)cc(C)nn2)=O)C2CC2)=O)c(C)nc2ccccn12 67152,N1(C(C2(CC)CCOC2)=O)CCC(CC(C)NC(C2SCC=C2C)=O)CC1 67153,CC1CCCC(CNC(c2cc(CNC(C3(O)CC3)=O)no2)=O)C1 67154,c1(NC(=O)C(N2CCCCC(CO)C2)=O)cc(N2CCCC2)cc(F)c1 67155,N1(C(CC(C)(C)OC)=O)CC(C)N(C(C2(C)CC3CCC2O3)=O)C(C)C1 67156,C1(C)(CNC(CCc2cn(C)nn2)=O)CCC(NC(=O)COCc2ccnn2C)C1 67157,c1(CC)ccc(Cl)c(C(=O)NC(C)C(C)NC(c2oc(CO)cc2C)=O)c1 67158,c1(OC)cc(OC)cc(N(C(c2cnc(C(C)O)s2)C(=O)NC2(C)CC2)C)c1 67159,C1(NC(=O)CCc2cccc(Cl)c2)CN(C(c2cc(F)c[nH]2)=O)CCC1O 67160,CC1(OCCOCCNC(=O)COC)CN(C2CCN(C(=O)C3CC3)C2)C1=O 67161,c1(CS(=O)(=O)NC2(C)CCN(C(=O)OC(C)(C)C)C2)cnc(O)nc1O 67162,C1(C)(C=O)CC2C=CC1C2.Cc1cccnc1OCC1CCC(C(=O)NC)CC1 67163,c1(NC)ncnc(OC)c1C(=O)NC1CC1CCNC(C12CC(C)(CCO1)C2)=O 67164,CCC(CC)(CCNC(=O)CN(C)C(C)=O)NC(=O)CC1CCCOC1C(C)C 67165,CCC(C)CCCCC(=O)N1CCC(NC(C2CCCC(C)(C)C2)=O)C(C)(C)C1 67166,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67167,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67168,c1(N2CCC(CC)OCC2)nc(N2CCSC(c3cccs3)C2)c2c(n1)CCS2 67169,Cc1nc(NC(=NCC2CCCN2C)NC(c2cccc(F)c2)C)cc(C#N)n1 67170,c1(C(N2C(C(C)(C)NC(=O)CCC3CCC3)CCC2)=O)ccc2nc[nH]c2c1F 67171,C1(N(C(=O)CC2(COC)CC2)CC)CCN(C(=O)CCCc2ccc(C)s2)C1 67172,C(C(F)(F)C(C)(C)O)NC(C1(CNC(C(COC)O)=O)CC(C)(C)C1)=O 67173,CC(O)(C(=O)N1C2CCC(C2)C1C(N1CC2CCC1C2)=O)C(F)(F)F 67174,C(=O)(CS(=O)C(F)(F)F)N(CCCN(C)C(C1CCN1C(C)(C)C)=O)C 67175,CCCCCC(F)C(=O)N(CCCN(C)C(c1cc(F)c(N)cc1F)=O)C 67176,CN1CC(C(=O)NC(C2CCN(C(C3CC(C)(O)C3)=O)CC2)CO)CC1=O 67177,N1(C(C(CC)F)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])c(CC)nn1C)=O)CC2 67178,CC1(C)CC(NC(=O)CNC(=O)C2CC2)CN(C(C2CC2Cl)=O)C1 67179,CCC(O)C(C)(C)C(=O)NCC(CC(=O)N(CC(C)(CC)OC)C)OC 67180,n1(Cc2c(C)noc2C)ncc2cc(I)ccc12 67181,c1(C(=O)NCC2(F)CN(C(C(C(C)O)C)=O)C2)cn2cc(Cl)cnc2n1 67182,C1(n2cc(CO)nn2)(C(=O)OC)CCN(C(=O)NCc2[nH]ccc(=O)c2O)CC1 67183,C1(C(=O)NCCCC(C)NC(=O)CCCC2CCCCC2)(CO)CCCCO1 67184,Cc1ccccc1-n1cc(CN2CCC(O)CC2)cn1.N12CCC(CC1)NC2=O 67185,CC#CCC(C(=O)Nc1cnccc1OC)NC(=O)CCC1CC(OC)C1 67186,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]c1 67187,c1(CN(C)C(C2CCC(F)CC2)=O)cc2ccsc2n1C 67188,N1(C(C(c2cncnc2)C)=O)CCC(NC(=O)C=Cc2ccco2)C12CCC2 67189,N1(C(CCCC)=O)CCC(C)C1CNC(=O)CCc1ncc(Br)cn1 67190,C1(C)(CN(C(=O)CCN(C(=O)CC2CCCC2)CCO)C)CCCC1O 67191,S(=O)(=O)(c1ccc(NCCN2CCCCC2)cc1Br)NC(c1ccccc1F)C 67192,c1(OC(C(=O)NC(CNC(Cc2cnn(CC)n2)=O)CO)C)cccc(Cl)c1 67193,C(CNC(CCCC=C)=O)(C(C)C(C)C)NC(=O)Cc1sc(SC)nc1C 67194,C#CC1(C(=O)NC(c2ccnn2C)C)CCN(C(c2csc(C)n2)=O)C1 67195,C1(CNC(C(CCOC)NC(c2cnncc2O)=O)=O)CC2CCCC2C1 67196,Cc1ccc(C#CC(=O)NCCC2CCOCO2)cc1 67197,C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCSC2)=O)C2CCCC12 67198,C(c1ccncc1)=CC(=O)NC1(C(N2CC(F)(F)C2CCOC)=O)CCCCC1 67199,O=C(C1=NOC2(CCOC2)C1)N1CCC2CCN(C(=O)C(F)F)CC12 67200,c1(C(=O)NCC2CN(C(CC3CC(C)C3)=O)C(C)C2)ccc(Br)c(F)c1F 67201,c1(C(=O)NC23CC(NC(C4COC(=O)C4)=O)(C2)C3)cnn2ncccc12 67202,N1(C(C=CCN(CCC(F)(F)F)CC)=O)CC(NC(=O)C(F)(F)CO)CCC(O)C1 67203,c1(CC)ncoc1C(=O)NC(C(=O)N(C)Cc1nnc(O)o1)C1CCC1 67204,Cc1c(Cl)sc2nc(Cl)c(CNC(c3ccccn3)CO)cc12 67205,C1(C(=O)NCCOC2CCN(C(c3cnc(C(F)F)s3)=O)C2)CC2CCC1CC2 67206,N1(C(COCC(C)C)=O)CCCC(CNC(=O)C(n2ccc(C3CC3)n2)C)C1 67207,C1(C(=O)NCC2=CCC2)(CC)CCN(C(=O)CN2CC(C)(C)C2)C1 67208,c1(C2CC(c3onc(-c4c(C)ncnc4C)n3)OCC2)cc(=O)n(C2CC2)c(O)n1 67209,C1(C(N2CCOCC(NC(=O)Cc3ccoc3)C2)=O)CC2CCCC(C1)C2=O 67210,N1(C(C(C)Cc2ccccc2)=O)C2CC1CN(C(c1nc(C(C)(C)C)no1)=O)C2 67211,N1(C(c2cc(OCC)n[nH]2)=O)CCN(C(=O)COC2CCCC2O)C2(CC2)C1 67212,C1(NC(C2CC(CC)C2)=O)COCCN(C(c2c(N)cccc2Cl)=O)C1 67213,CC1CCOC(C(=O)NCCC2CC(NC(c3cc(=O)cc[nH]3)=O)C2)C1 67214,C1(NC(c2ccnc(N3CCC3)n2)=O)CCCN(C(=O)Cc2ccoc2)C1 67215,C1(OC)(CNC(=O)Cc2ccccc2)CCN(C(=O)CC2CCC(=O)NC2)C1 67216,N1(N(c2cc(CO)[nH]n2)C)CC(CNC=O)CC1(C)C.C1(C(F)(F)F)(C=O)CCC1 67217,C(=O)(CCCCC1CC1)NC(CC)CNC(=O)CNC(=O)Nc1ccccc1 67218,N1(C(c2c(CC)con2)=O)CCN(C(=O)C(C(C)(C)C)SC)C(CO)C1 67219,N1(C(C(C(C)C)OC(F)F)=O)CC2(C=C(C(=O)N(CCCO)C)CO2)C1 67220,N12CCCN(CC1)C(C(=O)OC)c1cc2ncn1.C1(OC)CCC1 67221,c1(OCCc2nn(C(COC)C)c(-c3sccc3Cl)n2)c(C)cccc1Cl 67222,c1(C(N(CC(O)CNC(=O)C(F)C(F)(F)F)C)=O)ccc(C#N)cc1 67223,C1(NC(C(Br)=C(C)C)=O)CC2(CCCCN2C(=O)CCCn2cncn2)C1 67224,N1(C(=O)COC)CCC2(CCCN(C(c3ccccc3)=O)C2)C1.C1CCOC1=O 67225,CCC(C)C(=O)N(CCCOCCN(C(=O)C(C)(C)c1ccccc1)CC)C 67226,C(=O)(C1=CCCOCC1)NC1(C(=O)N(C)Cc2ccsc2)C(C)CCC1 67227,N1(C(C(c2ccccc2)NC(C)=O)=O)CCOCC1CNC(C1CC(F)(F)C1)=O 67228,N1(CC(=O)NC(C)(CNC(=O)C(c2ccccc2)F)C2CCC2)C(=O)CCC1=O 67229,c1ccc2c(c1)nc(CN1CCOC(c3ccc(Cl)s3)C1)n2CC1CCOC1 67230,C1(CNC(C(CC=CC)N(C)C)=O)CN(C(=O)CC2CC(OC)C2)CC1(C)C 67231,N1(C(CSCCCC)=O)CCCCC(CCC(N2CCC(F)(C#N)C2)=O)C1 67232,c1(C(N(C2CCN(C(=O)C#CC3CC3)C2)CC)=O)cn(C(C)C)nc1C 67233,c1(-c2nnn(C)n2)cccc(C2CC2)n1.N1CCOC(c2ncn[nH]2)C1 67234,S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCC(C)(C(=O)Nc2ccc(O)cc2O)C1 67235,C1(NC(Cc2n(C(C)C)cnn2)=O)CCC(C)N(C(=O)CC2CCCO2)C1 67236,N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(c2ccc(C(C)C)s2)=O)C(CO)C1 67237,CC1=C(C(=O)N2C(C)CCC2(C)C)C(C)n2nnnc2N1C 67238,CCCCCCC(C)NC(c1coc(CNC(=O)C(CO)OC)n1)=O 67239,N1(C(C)=O)CCCC(C(=O)NC2CN(C(=O)Nc3n[nH]c(Br)n3)C2)C1 67240,c1(C(N2CC3CCCN(C(C(C)OC)=O)C3C2)=O)ccc2c(Cl)nccc2c1 67241,C(=O)(CCC(F)(F)C(F)F)NC1CN(C(c2ccn(CCC)n2)=O)CC(O)C1 67242,c1(CNCc2cccc(OC)c2OC(F)F)ccc(C)c(F)c1F 67243,c1(NC)ccc(C(N2CC(O)(C3CCCN3C(=O)CCOC)C2)=O)cn1 67244,C12(C(N(CCCN(C(CC(C)CF)=O)C)C)=O)CCCCC(F)(C1)C2 67245,c1(C(=O)NC2C(C)N(C(=O)C3=CCCO3)CCC2)nn2c(c1Br)CCC2 67246,c1(C(=O)NCC2CN(C(=O)C(F)CC3CC3)CCO2)cc2ccccc2o1 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67404,C12OCCC1NC2=O.CCCCNC.C1(C=O)(CC2CCC2)CC1 67405,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67406,N1(C(C2(CC)CC2)=O)CCC(C(=O)NCC(=O)NC2CCCC2)C(C)(C)C1 67407,c1(C(C(=O)OC)NC(C)CCO)ccc(Cl)c(C)c1 67408,c1(C(C(=O)NCCOC)NC(N(CC#C)C2CC2)=O)cc(Cl)ccc1Cl 67409,N1(C(C(C)C(=O)N2CCOCC2)=O)CCCCCC(NC(C2CC2C2CC2)=O)C1 67410,N1(C(C2N(C(c3cn(C(C)C)nc3)=O)CC(O)C2)=O)CCCCC(CO)C1 67411,C(=O)(CC(C)(C)CNC(c1scc(C)c1C)=O)N1C(C(N)=O)CC(OC)C1 67412,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67413,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67414,C(=O)(C1=CCC(NC(=O)CC2COCCO2)C1)NC(c1cncs1)C 67415,N1(C(CCC=C(C)C)=O)Cc2[nH]nc(C(N3CCCCC3C3CCC3)=O)c2C1 67416,C1(NC(CCS(=O)(=O)NC)=O)(CNC(c2ncccc2Cl)=O)CC2CCC1CC2 67417,c1(OC)ccc(OCCC2CC2)c(C(F)(F)C(=O)NC2Cc3nccn3C2)c1 67418,C12(C(N(CCNC(c3ccc(CO)cc3F)=O)C3CC3)=O)CC3CC(C1)C(=O)C(C3)C2 67419,C1(C(=O)OCCCO)CN(S(=O)(=O)CC2CCC2)CCC1c1ccccc1 67420,N1(C(C2(c3cn(CC4CCCN4)nn3)CC2)=O)CCCC12CCOC2=O.CS 67421,C1(C)(OCC(=O)NCC(C)CNC(C2CCCSC2)=O)CCOCC1 67422,c1(C(=O)NC2CC2)cnc(-c2cn(-c3ccccc3)nn2)cn1 67423,C1(CCNC(CCCC)=O)CCCCN1C(=O)COCc1nc(CC)no1 67424,CCC(CC)C(C(=O)N1CCC(C)(C)C1C(=O)NC(C)CCc1cn[nH]c1)OC 67425,CC1CCN(C(c2cnn(C)c2C(F)F)=O)CC1NC(C1CC(F)(CO)C1)=O 67426,c1(C(=O)NC(C2N(C(C(C3CC3)OC)=O)CCC2)C)cc(Cl)c2[nH]c(O)nc2c1 67427,c1(C(=O)NC(C2CCN(C(CN(C(C)C)C)=O)C2)C)ccnc(CN(C)C)c1 67428,c1(C(c2n(C3(C)CC3)nnn2)NCC2CCC3(CC3)C2)cccc2sccc12 67429,c1(CC(=O)NCCC(C)NC(=O)CCSCc2nccn2C)ncc(Cl)s1 67430,c1(NC(=O)C(N2CC(O)(NCCCSC(F)(F)F)C2)=O)cc(F)ccc1F 67431,c1(C(N(C)CCC2CCCCN2C(C23CCC2C3)=O)=O)cnn(C)c1S(N)(=O)=O 67432,C1(NC(COCC)=O)C2COCC1CN(C(=O)Cc1coc3ccc(F)cc13)C2 67433,c1(C(=O)NCC(CNC(Cc2cn(CC)nn2)=O)(C)C)noc2cc(F)ccc12 67434,CC(CC(=O)NCC1CCCS1)N(C(C1COCC1C(N)=O)=O)C 67435,CCCC(CCC)C(=O)N(C1CCN(C(C2(COC)CCCC2)=O)C1)C 67436,c1(OC)ccc(CC(N2CCC(CNC(=O)C(CCO)N(C)C)C2(C)C)=O)cc1O 67437,c1(C(N(CCC(C(C)C)NC(CC=C)=O)C)=O)cc2cc3c(cc2[nH]1)OCCO3 67438,C1(NC(C)=O)CN(C(C2CCCN(CCC#N)C2)=O)Cc2nccn2C1 67439,CC(C)C(C)(O)CNC(c1ncoc1CNC(=O)C=Cc1cccnc1)=O 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67457,CC(Cc1cnc[nH]1)C(=O)N(C1CCN(C(C2CC(F)(F)C2)=O)C1)C 67458,c1(OC)ccc(C(=O)NC(CNC(=O)CC(C)(C)CO)C(C)(C)C)cc1F 67459,c1(C(=O)NCCCNC(C(C)OCCC#C)=O)c(OC)ccc(F)c1Br 67460,CC1(C)OCCC1C(N1CC(OC2CCN(C(=O)COCC3CC3)CC2)C1)=O 67461,c1(C(N(CCCNC(=O)CC2(C)CC2F)CC)=O)cnc(C(C)C)nc1O 67462,N1(C(c2c(CC)cccc2)=O)CCCC(C)C1CNC(=O)CC1CCS(=O)(=O)C1 67463,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2nocc2Cl)=O)CCC12CCC2 67464,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67465,N1(C(c2n[nH]cc2C(N2CCCC(O)C2)=O)=O)CCOC(C(F)(F)F)CC1 67466,c1(-c2cn(C3C(C(N4CCN(CCOC)CC4)=O)C3)nn2)cccc(C)c1O 67467,C(CC(=O)NC(c1cn(-c2cccc(Br)c2)nn1)C)(C(F)(F)F)NC(C)=O 67468,C(C1CCCN1C(=O)C=CC1CC1)=CC(N1CC(C)(NC(=O)NC)C1)=O 67469,c1(NCC23N(C(=O)OC(C)(C)C)CCC2CCC3)ccc2ccc(Br)cc2n1 67470,N1(C(C2CCCN(CC)C2)=O)CCC(C(N)=O)C(O)C1.C12CCC(O1)C(=O)N2 67471,C(CCCC(=O)N1CCOC(CCO)C1)NC(C(C=C)O)=O 67472,c1(CC(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)ccnc(F)c1F 67473,C1(CNC(C2CCS2(=O)=O)=O)CCC(NC(c2cc(C(F)F)on2)=O)C1 67474,c1(-c2cn(CCN(C)C(C3CCC(=O)N3)=O)nn2)cccc(Cl)c1Cl 67475,S(=O)(=O)(c1cccs1)NC1CC(C(N(C(C)C(N2CCOC(CO)C2)=O)C)=O)C1 67476,C1(NC(CCCOc2cccc(C)c2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1F 67477,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67478,C1(CCNC(c2n(C)ncc2)=O)COCCN1C(C12CCC1C2)=O 67479,CC(CN(C)C)CC(=O)NCC1(C)CN(C(=O)CCF)C1 67480,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67481,c1c2ccc(cc2)n1.c1(CCC)nocc1C(=O)NC1CCN(S(=O)(=O)CC)C1 67482,N1(C(C(S(C(C)C)(=O)=O)C)=O)CC23CCCCC2(C1)CN(C(=O)CC#N)C3 67483,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(CF)C3)CC2(C)C)co1 67484,CC(C)C(CNC(c1cc(C(N)=O)c[nH]1)=O)NC(c1cnn(C2CC2(F)F)c1)=O 67485,N1(C(c2c(C)c[nH]n2)=O)Cc2ccccc2C(NC(C2CC3C(C2)C3(C)C)=O)C1 67486,CC1CN(CCNC(N2CC(C)CCC2c2ccccc2)=O)S(=O)(=O)C1 67487,N(C)(C1=CCC2(CC1)OCCO2)Cc1ccc(OC(C)C)cc1 67488,C1(C(N2C(C)(OC)CC2)=O)CCCN(C(=O)C(C)(F)c2ccon2)C1 67489,c1(C(=O)NC(C)CNC(c2cc(CCO)on2)=O)ccc2c(c1)C(=O)CCCC2 67490,C1(CNC(C=CCNC(CC(C)c2ccco2)=O)=O)CCCOC1(C)C 67491,C1(N(C(c2ccc(C(C)=O)s2)=O)C)CN(C(=O)CCn2cccnc2=O)CC1O 67492,c1(C(N2CC(O)CC2c2cccs2)C(=O)NC(c2cccs2)C)ccccc1Br 67493,c1(C(N2CC(C)(C(=O)Nc3nc(C(F)(F)F)ccc3Br)C2)=O)ccc(Br)cc1O 67494,CCCC(CC)C(=O)N1CCC(CC(=O)NCCc2ccsc2)C1(C)C 67495,C(=O)(CC1CCc2ccccc21)N1CCN(C(CC(=O)NCC2CC2)=O)CC(O)C1 67496,C1(C(=O)NCCF)CC2CC2N1C(C1C=CCC1)=O 67497,c1(CC(=O)NC2C(NC(C3(C(C)C)CC3)=O)C2)cccc(Br)c1 67498,C(=O)(CCP(C)(C)=O)NC(C(=O)NC(CC=C)Cc1cn[nH]c1)C(C)C 67499,c1(OCC2CCN(Cc3n(C)ncc3Cl)CC2)ncnc(Cl)c1-c1ccc(Cl)cc1 67500,N1(C(C=C(COCCC=C)C)CCCC)CCN(C(C)=O)CC1CCC 67501,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67502,c1(NC(C2(C(=O)OCC)CC2)=O)c(N2CCC(N(C)C)C(C)C2)ncnc1Cl 67503,C1(NC(=O)C=Cc2cccs2)CC2CCC(C1)N2C(C1CCCCN1C1CC1)=O 67504,C12CC3CCC(C1)N3C(=O)C2.CC1(C)CC(C(=O)NC2CN(C(N)=O)C2)CO1 67505,c1(OCC)ncccc1C(C(=O)NC1CCCCC1)N(C(C)C(F)F)C 67506,C1(c2n(CCOCC)nnn2)(NC2(C)CCS(=O)(=O)CC2)CC2COCC2C1 67507,C(=O)(CC1=NNC(=O)C1)NC1CCN(CCNC(CC2(C=C)CCC2)=O)CC1 67508,c1(-c2nc(C3C(=O)N(C4CC4)CC3)n(-n3cncn3)n2)csc2ccc(F)cc12 67509,C(C)(C(C)(C)C(=O)N(C1C(C)(C)C1(C)C)C)NC(c1ccc(CC)[nH]1)=O 67510,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67511,CC1Cc2cccc(C(=O)NC3(CNC(c4ccc(F)cc4)=O)CCC3)c2O1 67512,C1(COC)CC(O)CN1C(=O)C(COC)NC(C1CC1C(C)(C)C)=O 67513,C1(NC(=O)Cc2c[nH]nc2O)C=CCN(C(C2(F)CC2c2ccccc2)=O)C1 67514,C(CN=c1[nH]c2c(c(=NC(C)CC(N)=O)[nH]1)SCC2)C1CCCN(CCC)C1 67515,CCC(O)CC(=O)N1CC(NC(=O)C(C)Oc2cccc(CO)c2)C1 67516,N1(C(CCNC(C)=O)=O)CCCC12CCCN(S(=O)(=O)CC#N)CC2 67517,C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1C1CC1 67518,C(=O)(CCC(C)(C)NC(=O)Cc1cncn1C)N(C1CCCC(O)C1)C 67519,c1(C(=O)NC2CN(C(c3c(CC)noc3)=O)C(C)CC2)cnc(O)c([N+](=O)[O-])c1 67520,C(=O)(C1=CC(O)C(NC(=O)CN2CCCCC2C)C1)N1CCC(CC(C)C)C1 67521,c1(C(=O)NCC(CNC(COC(CC)C)=O)CO)cncc(C(C)(C)C)c1 67522,C(CC(=O)NC1CC(O)C1)N(C(=O)COC1CC1(F)F)CC.C1CN1 67523,N=c1ccc(C(=O)NC(CNC(c2cccc(OCC(N)=O)c2)=O)C2CC2)c[nH]1 67524,C1(NC(C(c2ccc(C)s2)C)=O)CC2(C1)CC(CNC(C1(C)CCSCC1)=O)C2 67525,CCS(=O)C1CCCC(NC(=O)C(=O)Nc2cc3ccccc3n2C)C1 67526,N1(C(CCC#CC)=O)CCN(C(=O)C=CC(F)(F)F)CC2CCCCC12 67527,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67528,C1(CNC(CC(=O)N(C)C)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CCC2 67529,C(=O)(C(O)C1CN(C(c2ccoc2)=O)C1)N(C1CCC1)C 67530,c1(CCCn2cc(COCc3c(F)cccc3)nn2)ccc(Br)c(Cl)c1F 67531,c1(C(N(C(C(=O)N(CC(C(C)C)OC)C)C2CC2)C)=O)cccc(C)c1O 67532,c1(CC(n2cc(C(CC)NC(C3(C)CNC(=O)C3)=O)nn2)C)cc(F)ccc1F 67533,C1(C(=O)NC2CN(C(c3ccc(-n4ccnc4)cc3)=O)C2)CC2(CCC2O)C1 67534,C(=O)(CC1=CCOCC1)NCC1C(C(=O)NCc2cccc(OC)n2)CC1 67535,N#Cc1ccc(Br)c(C(N2CCC(F)(C(=O)Nc3c(F)cc(F)cc3Cl)C2)=O)c1 67536,c1(C(N2CC(CNC(C(C)NC)=O)OCC2)=O)cc(Cl)cc(Cl)c1OC 67537,C1(CNC(c2csc(-c3ccsc3)n2)=O)CC2(C1)CN(C(=O)CCF)C2 67538,c1(C(N2CCC(C(=O)NC(C)C)C2)=O)cnc2ncc(C(C)(C)C)cn12 67539,C(C(C(=O)NCC1(F)CCCC1)N(C)C)NC(C(C)n1cccn1)=O 67540,c1(C2N(c3n(CCC(=O)NC)c(CC(C)C)nn3)CCOC2)nc2ccccc2s1 67541,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncc(F)cn1 67542,CCCCCCC(CC)(CC)C(=O)NC(C)CC1CN(C(=O)C(F)C(C)(C)O)C1 67543,N1(C(C2CN(C(CNC(CC(C)(C)C)=O)=O)CC2O)=O)CC(S(N)(=O)=O)C1 67544,CC(=O)N1CCC(C(N2CCCC2C(N2CC3C(C2)C3(F)F)=O)=O)O1 67545,c1(C(=O)NCC(CN(C(c2nc(C)sc2C)=O)C)C)cc(N)cc(O)c1C 67546,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C1CCN(C(C2CC(=O)NCC2)=O)C1)CCO 67547,c1(C(C)NCc2cnc3c(c2)CCCC3)ccc2c(c1)OCCO2 67548,C(=O)(CC(O)CC(C)C)NCC(C1CCN(C(c2c(C)cccc2Cl)=O)CC1)C 67549,C(=O)(Nn1cnnc1COC)C1N(C(Cn2ncc(CC)c2)=O)CCCC1 67550,CCC(C)CCCCC(=O)NC(C)(CNC(=O)CNC1CC2CCC1C2)C1CC1 67551,C1(C(=O)NCC(C)Cn2ccnc2)CC(=O)CN1C(C1OCCC1(C)C)=O 67552,N1(C(C(C)Oc2ccccc2)=O)CCC(CNC(=O)CC(F)(F)F)C(C)C1 67553,c1(CC(=O)NC(CN(C(=O)CCCC(C)C(C)C)C)(C)C)cn(C)nc1C(F)(F)F 67554,N1(C(CN(CC#C)C(C2CN3CCN2CC3)=O)=O)CC2CC(C(N)=O)C(C2)C1 67555,c1(C(C)C)cc(C(=O)NCC(CO)NC(=O)Cc2cccc(Cl)c2F)cc(O)n1 67556,C1(C)(C(N2CCCC(CN(C(=O)C=CC=C(Cl)Cl)CC)C2)=O)CCC(=O)CC1 67557,C(=O)(CC(C(F)F)NC(C1CSC1)=O)N(C)Cc1ccns1 67558,Cc1ccc(C2(C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)CCC2)cc1 67559,c1([SH](CC(C2CC2)OC)CC=CC)cccc(OC)c1 67560,Cn1cnc2c(C(=O)NCC(CO)NC(=O)Cc3nc(F)c(F)cc3F)cccc12 67561,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 67562,c1(N(C)C)cccc(C(N2CC=CC(NC(c3cc(Cl)cs3)=O)C2)=O)n1 67563,c1(C(N2C(C(C)(C)NC(C(CN(C)C)O)=O)CCC2)=O)c[nH]nc1[N+](=O)[O-] 67564,CCCC(C)(C)C(=O)NC1CCCC(CNC(=O)C=Cc2nc(C(C)(C)C)cs2)C1 67565,c1(C(C(=O)N(C2CC(C)(C)C2)CCNC(c2c(C)snc2)=O)C)ccc(F)cc1F 67566,Cc1cc(NC(N2CCCC2Cc2ccncc2)=O)c(C)n1Cn1cncn1 67567,CC(C)C(F)C(=O)NCC12CC(CN1C(=O)C(C)(C)c1cccs1)C2 67568,N1(C(c2onc(C)n2)=O)CCN(C(=O)C(c2ccccc2F)O)C(COCC)C1 67569,c1(CNCC2CCC(C(N)=O)O2)ccc(-c2ccccc2)nc1 67570,C1(NC(C(C(C)C)n2cncn2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC(O)C1 67571,C1(CNC(=O)C(O)c2ccco2)(CN(C)C)CCCC1.C12CC1C(=O)NC2C 67572,C(=O)(C#Cc1ccccc1)NC(CC)CNC(=O)CC(C(F)F)N(C)C 67573,c1(OC)cc(C)c(CN2CC(CCNC(=O)C(=O)NC)CC2=O)cc1OC 67574,C1(NC(=O)Cc2cnoc2)CCC2CCN(C(c3coc(Br)c3)=O)C12 67575,CC1=C(CNC(C2COCCN(S(=O)(=O)CCN)C2)=O)SCCO1 67576,c1(C(=O)NCC2(C)CCN(C(C3C(C#C)C3)=O)CC2)cc(C)c(F)cc1F 67577,c1(C(=O)NCC2C(NC(C(C)N3CCC3)=O)C2)ccc(O)cc1[N+](=O)[O-] 67578,N1(C(c2n(CCC)ncc2)=O)CCN(C(c2ccc(O)cc2F)=O)C(C2CC2)C1 67579,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 67580,C(=O)(C(C)(C1C(C(=O)OC(C)(C)C)CC1)NC(=O)NC1CCN(C)C1)OC 67581,N1(CC(=O)NC)C(=S)NC(c2cc(-c3nccs3)cs2)C2=C1CCN(CC)C2=O 67582,CC1CN(C(=O)CCCN(C)C)CC1(C)CNC(c1ccc(CN(C)C)cc1)=O 67583,C12(C(N3CCC(C(N4C(CCC=C)C4)=O)(COC)C3)=O)CCC(CO)(CC1)C2 67584,N1(C(C2C(C)(C)C2)=O)CC(=O)NCC1C(N1CC(C(C)C)C1C(C)C)=O 67585,N1(C(c2nnc(O)o2)C)CC(NC(=O)CC2CCCCC2)CCC1C 67586,c1(C(N2CCC(C(C)(C)NC(CC(C)SC)=O)CC2)=O)n[nH]c2c1CCCCC2 67587,c1(OCCCC)ccc(CCOC(=O)C(c2cnn(CC)c2)C)cc1 67588,C1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCCC2)C2CC3CC(C2)CC1C3 67589,c1(C(N2CCC(N(C(=O)CN3CCC3C)CC#C)CC2)=O)ccc(O)c(F)c1 67590,C12(C(=O)NC(C)CN(C)C(c3ccccc3CO)=O)CC1COC2(C)C 67591,Cc1nn2cc(N(C)C(=O)OCC=CCNC(=O)CC3CCC(C)O3)nc2s1 67592,C1(O)(CC=C)CCN(C(C2C(NC(=O)CCc3cncnc3)C2(C)C)=O)CC1 67593,C1(C(N2CC(C(C)C)C2)=O)CCN(C(C2CC23CCOCC3)=O)C12CCC2 67594,C1(NC(N(C(C)=O)Cc2cc(C)oc2C)=O)CCCN(CCN2CCCC2)C1 67595,C(CC(=O)NCC(F)(F)Cl)(CC(C)C)NC(Cc1c(C)scc1)=O 67596,C(=O)(CC(O)C(C)(C)C)N1CCC(F)(CNC(c2ccc(C)nc2)=O)CC1 67597,C=CCC(CC)C(=O)NC1(COC)CCN(C(=O)CC2(O)CCCOC2)C1 67598,c1(C(=O)NCC2(C)CCC(NC(C(=C(C)C3CC3)F)=O)C2)ccc2cc[nH]c2n1 67599,CCC(C(=O)N(CC(c1ccccc1)NC(=O)CCc1cnn[nH]1)C)OC 67600,C(=O)(C(C)(C)N(C)C)N1C(C(N(C(C=C)C2CCC2)C)=O)CC1 67601,N1(C(C2C(C)CC2)=O)CCC(CO)(CNC(C2CC=CC2)=O)CC1 67602,N1(C(N2CC(n3cc(S(C)(=O)=O)cn3)C2)=O)CC(C(=O)NC(C)(C)C)C2(CC2)C1 67603,C1(CNC(C=CC(C)NC(C=CC(C)(C)SC)=O)=O)CCOC(C)C1 67604,C(=O)(C1=CC2(CCOC2)C1)N1CC2C(CNC(c3c(C)nncc3)=O)C2C1 67605,N1(Cc2c(OCC)ccc(Br)c2)CC2CCN(C(c3cc(C(C)C)on3)=O)C2C1 67606,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 67607,c1(C(=O)NC2(C(=O)NC34CC(C3)C4)CC2)cc(OC)c(N)c(OC)c1.C(C)(C)COC 67608,C1(CNC(C(c2cccc(Cl)c2)C)=O)CN(C(C2CC(=O)C2(C)C)=O)CCCO1 67609,Cc1cnc(C)c(C(=O)NCCC(C)CCNC(c2ccc(Cl)s2)=O)c1 67610,N1(C(c2cc(C)no2)=O)CCCN(C(c2ccnn2CCF)=O)CC1C 67611,Cc1ccncc1CCC(N1CCC(CC(N2CCC(CN(C)C)CC2)=O)C1)=O 67612,c1(C(=O)NCCC(N)C2CCC2)ccc2nc(S)[nH]c2c1 67613,CC(C)CN=C(NCc1ccc(CC(C)C)cc1)N1CCC(N(C)C)C1 67614,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 67615,c1(C=O)cc(N)ccc1O.C1(C(=O)NCCN(C)C2CC2)CCCC(CF)C1 67616,CCC(C(=O)NCC1(NC(=O)CCc2cccnc2)CCC1)C(C)C 67617,C1(C(=O)OC)N(C(=O)CCC2(C)CCN2C(C2CC(CF)C2)=O)CC1(C)C 67618,C(=O)(CCC(F)(F)C(F)F)NCCCNC(CCc1nc(C)sc1)=O 67619,c1(CC)ccc(C(=O)NC(CNC(C2CC2(F)F)=O)CC)cc1[N+](=O)[O-] 67620,c1(C(N(C)Cc2cccc(Br)n2)=O)cccc2nccn12 67621,C1(OC)(CNC(=O)CN(C2CCSC2)C)CCN(C(C2C3CC4C(C3)C24)=O)CC1 67622,CC(C(=O)N1CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C2(CC2)C1)S(N)(=O)=O 67623,C(=O)(CCCCCOC)NC(CC)(C)CNC(=O)CCCC1CCCCC1 67624,CC1(C(=O)NC(C2CCCCC2)CNC(C2CCCCS2)=O)CC2(CCC2)C1 67625,O=C1CCC(O)CN1Cc1cn(CC2CCN(C(C3CCCCS3(=O)=O)=O)C2)nn1 67626,CCC(C)CC(C(=O)NCCCn1cc(C)cn1)NC(c1cnc2n1CCC2)=O 67627,C(N=c1[nH]cnc(Cl)c1Br)C1(CNC(CCCC(C)C)=O)CC12CCC2 67628,N1(CC)CCCC1C(=O)NC1CC(NC(=O)CSC2CCCC2)C1 67629,N1(C(C(C)Cc2ccc(Cl)cc2Cl)=O)CCC12CN(Cc1ncccc1O)C2 67630,CC(C)CC(O)CC(=O)NCCn1cc(C(=O)N(C)CC2(O)CCCCC2)cn1 67631,C1(C(=O)NC(CNC(COC(C)(C)C)=O)C2CCC2)CC2(C1)CC21CCC1 67632,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 67633,C1(C(=O)NCCN(C(=O)Cc2sccc2Cl)CCC)(NC)CCCCC1C 67634,CCC(C(=O)N(CCNC(=O)C(C1CCCCC1)SC(C)(C)C)C1CC1)N(C)C 67635,C1(C(N(C(C)C)CCNC(=O)Cc2cnn(C3CC3)c2)=O)CCCCC1(F)F 67636,C1(C(=O)NC(CCCC)CNC(C2(CO)CCCC2)=O)CCCCC12OCCO2 67637,CCC(O)C(=O)N(C)CC1CCN(C(=O)CCNC(C2CCCCC2)=O)C1 67638,C(=O)(C(C)C(O)CCCC)N1C(CC(=O)N(CC#C)C2CC2)CCC1 67639,c1(CC)ccnc(N(C)C)c1.c12n[nH]cc1C(=O)N(CC)C(C)CNC2=O 67640,N1(C(Cc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=CC3CCC3)C2C1 67641,N1(C(c2ncc(C)nc2)=O)CCC(C2(NC(C34CC3CCC4(F)F)=O)CC2)CC1 67642,C=C(C)C1OCCC1CNC(=O)CC(CNC(c1cc(C)c(N)cn1)=O)OC 67643,c1(CC(=O)NC(C(c2ccccc2F)NC(CC=C=C)=O)C)cn(C)nc1CC 67644,c1(OC)ccc(C(=O)N(CCCN(C)C(c2sccc2C)=O)C)nc1OC 67645,C=C1CCN(C(c2cccs2)=O)C(C(=O)NCc2cc(C)ccc2O)C1 67646,C#CCC(C)C(=O)N1CC(COC)(NC(c2cn(CCO)nc2C)=O)C1 67647,c12cc(Cl)ccc1O2.N1(C(CN(C)C)=O)CCN(C(=O)C(O)C2CCCC2)CC1 67648,c1(C(=O)NCC(CNC(C(CC(=C)C)OC(C)=O)=O)OC)cc(=O)c(OC)cn1C 67649,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ccn(C)n2)C(CC)C1 67650,c1(OC)nc(C(N2CC(CCNC(=O)C=Cc3cn(C)nn3)C2)=O)cc(O)n1 67651,C1(C(=O)NC2C(C)CCN(c3cc(CC)nc(CC)n3)C2)CCC2(CCC2)C1 67652,N1(C(C2CC=C(C)CC2)=O)CCCC(O)(CNC(c2c[nH]c(=N)nc2C)=O)C1 67653,c1(C(=O)NC2CN(C(=O)CCc3nccs3)CC2O)ccc(F)cc1Br 67654,c1(C(=O)NC2CCCC(NC(C(C)CC(N)=O)=O)C2)cc(Cl)c(F)cc1O 67655,c1(-n2c(C(CSC)(C)NC(c3nncs3)C3CC3)nnn2)c(C)cc(C)cc1C 67656,CC1(CNC(c2ccsn2)=O)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 67657,c1(C(C(=O)NC2CC2)N(C(CC)C(=O)OC)C)cnc2ccnn2c1 67658,c1(C(N2CC(NC(CC(CC)O)=O)(CO)C2)=O)cccc(C(N)=O)c1OC 67659,CC1(C)CCCCC1C(N1CCOCC1CC(N1CCC(O)(C(F)F)C1)=O)=O 67660,C1(NC(C2CC(OC)CN2C(=O)C(C)Cc2ccco2)=O)CCC(C2CC2)CC1 67661,C1(NC(COc2c(CC)cccc2)=O)CCN(C(=O)CCC2CCOC2)CC1C 67662,C1(c2nnnn2C2CC2)(NC(c2cn(Cc3ccccc3)cn2)=O)COCCO1 67663,c1(C(N(CC(CNC(CCC2CC(C)C2)=O)O)C)=O)ccc(=O)n(C)n1 67664,Cn1[nH]c(=NC(=O)C2(CCC#N)CC2)s1.n12cc(nn1)CCN1CC2C1 67665,C1(C(N(CC(COC)O)C)=O)CC(NC(C2(O)CCSC2)=O)CCO1 67666,c1(C(N2CCN(C(c3c(C)cns3)=O)CC2C)=O)ccc(S(C)=O)cc1 67667,N1(S(CC2(C)CC2(F)F)(=O)=O)CCC12CCNC2=O 67668,c1(CC(=O)NCC(C)(C)NC(c2ccnn2-c2ccncc2)=O)ccccc1F 67669,C1(C2CCN(C(c3cccnc3N)=O)C2)(NC(C(C2CC2)SC)=O)CC1 67670,C1(C)(C(=O)NCC2CC(OCC)C2)CCCN(C(c2cc(C3CCC3)on2)=O)C1 67671,Cc1ccc(CN(C(C2CCC(C)O2)C(=O)NCC2CCOC2)C)c(Br)c1 67672,C1(CNC(c2cc(C(C)C)on2)=O)CC2(CC2)CN1C(=O)CC1CCC=CCC1 67673,C1(NC(Cn2c(C)nc(C)n2)=O)COC2(CCN(C(c3nnn(C)c3C)=O)C2)C1 67674,C(N=c1[nH]c(N2CCC3CC3C2)nc(=N)[nH]1)C1(CCC=C)CC1 67675,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCOCCC)=O)C2)C1 67676,C(c1ccc(-c2ccccc2)cc1)=CC(=O)NC1CC(NC(C=CS(C)=O)=O)C1 67677,C(=O)(C1CCCc2ncnn21)N1CC2(CC(NC(C(CC(C)C)OC)=O)C2)C1 67678,C1(NC(c2c(CC)onc2)=O)CCN(C(=O)CC2(C(F)(F)F)CC2)CCC1(F)F 67679,N1(C(C2C(C)=C2)=O)CC(NC(=O)CC2CCCCCC2)C2(CCOCC2)C1 67680,C=CCC(C)(C)CC(=O)N1CCN(C(c2cnc(CC)nc2)=O)CC(CO)C1 67681,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2NC(=O)CN2CCCC(CC)C2)C1 67682,CC1(CNC(C2CCCC2)=O)CCN(C(=O)C2=CCCSC2)CC1 67683,c1(CC)c(C(=O)NCCC(O)CNC(=O)CN2C(=O)CNC2=O)cnn1C 67684,N1(C(CSCCC)=O)C2CCC(C(N3CC(N(C)C)C(C(N)=O)C3)=O)C1CC2 67685,C12CCCN(C1)CCCCCC2.C1(C(=O)NCc2ccco2)CCCN1CC1CC1 67686,C1(=O)NNC(=O)CC12CCCC2.C(C(C)(C)C(=O)N)C(C)=O.CCN 67687,N1(C(CC(CC#C)NC(=O)C(CC=C)NC(C)=O)=O)CCn2nccc2C1 67688,N#Cc1ccccc1C=CC(N1CC(NC(=O)CCc2ncc[nH]2)C(O)C1)=O 67689,C(C(C)C(F)C(=O)N(C1CCCC1C)C)NC(c1n(CCC)ccc1)=O 67690,N1(C(C(C2CCCO2)OC)=O)CC(O)(C2(CNC(C3(Br)CC3)=O)CC2)C1 67691,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(c1cc(C(F)(F)F)cs1)=O)CC)(C)C 67692,C(CCCCC(=O)N1CC(NC(=O)CC(C)n2cccc2)C(C)C1)=CC 67693,C1(C(N(CCNC(CCC(C)SC)=O)CC2CC2)=O)COCC2(CCC2)O1 67694,C1(C(=O)NCC=CCNC(c2c(C)oc(Br)c2)=O)CC2CCC1NC2=O 67695,C(=O)(CCCC(F)F)N1CC2C(NC(=O)CCCN3C(=O)CCC3=O)C2C1 67696,C1(NC(C2(CCNC(c3cncs3)=O)CCCC2)=O)CCCOC12CCC2 67697,C(c1cccnc1)=CC(N1CC(CC(C(=O)N(CC#C)CCO)F)C1)=O 67698,S(=O)(=O)(c1[nH]c(=NCc2c(C)c(C)nn(C)c2=O)ccc1Br)NCCOC 67699,C(=O)(CC(=O)N1CCC(NCCC2CC2)C1)N(C)C.c1(=O)c(=O)n1C1CCCC1 67700,C(=O)(CN=c1ccc(C#N)c[nH]1)NC1CCC(NC(C(CCC)C)=O)CC1 67701,C(=O)(CC(F)(F)C(F)(F)F)N1C(C(C)NC(c2cncs2)=O)CCC1 67702,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 67703,CC(CCNC(C1CC=CCC1NC(c1cc(Cl)ns1)=O)=O)C(C)(C)C 67704,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NC(C2CCCC2)C)O1 67705,O=C1COC2CN(C(c3cccc(C(F)(F)F)n3)C(=O)NC3COC3)CC2N1 67706,C1(F)(CNC(c2c(C)con2)=O)CCC(NC(c2nccnc2C)=O)C1 67707,N1(C(C(C)N(C(C)=O)C)=O)CC=CC(C(N2CCC2(C(=O)O)C(C)C)=O)C1 67708,Cc1c(C(=O)NC(CNC(=O)C(CC(C)C)C(N)=O)C(C)C)sc2nnc(S)n12 67709,C(CC(C)C)(C(=O)NC1CCN(C(=O)Cc2c[nH]c(=N)[nH]2)C1(C)C)OC 67710,C1(CCC)(NC(c2ccc(C(F)F)o2)=O)CCCN(C(c2cccc(C)n2)=O)C1 67711,C1(C(=O)NCc2ccoc2C2CC2)CCN(C(=O)C=CCN2CCCC2)C1C1CC1 67712,c1(-c2c(C)cc(F)c(CN3CC(F)(F)C3)c2)ccc2nnc(-c3ccnnc3)n2c1 67713,C(C(CN(C)CC1(CCOCC)CC1)OC)OC 67714,N1(C(C(CC2CCC2)NC(c2ccco2)=O)=O)CCC(C(F)F)CC1 67715,C1(C)(NC(C2(OC)CC2)=O)CCN(C(c2oc(C)nc2C(F)F)=O)CC1 67716,CC(C)C(CCN(C(=O)CC#N)C)NC(=O)C(C(C)O)c1ccccc1 67717,CC1CN(C)CCC1N=c1[nH]c(=NCC2(C(C)(F)F)CC2)c2c(F)cccc2[nH]1 67718,c1(C(N(C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)C)=O)cccc(F)c1C(F)F 67719,C1(C(=O)NC(CN(C)C(C2CC(C)(C)O2)=O)(C)C)CC2(CC2)C1 67720,C1(F)(C(N2CCCC(CCNC(CCCN(C(C)C)C)=O)C2)=O)CCC(C)CC1 67721,c1(C(C(N2CCC(CNC(c3sccc3F)=O)C2)=O)OCC)ccccc1F 67722,CC1=C(C(=O)N(CC(C)O)CCNC(c2cc(F)cnc2O)=O)SCCO1 67723,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 67724,N(C1CCc2ccccc21)C(CCCCNC(=O)C=CC1CCOC1)=O 67725,c1(C(N2CCC(OCC(N3C(C)CC3CO)=O)C2)=O)cc(C#N)n(C)n1 67726,c1(C(N2C(CC(C)O)CCC2)=O)cccc(S(=O)(=O)N(C)Cc2cc(O)no2)c1 67727,c1(CC)nc(CC(N2CCC(C(C)NC(C3CC34CCC4)=O)C2)=O)cs1 67728,c1(C(N2C(C)CC2C(=O)N(C)C)=O)nn(C)nc1-n1cc(-c2ccnc(Cl)c2)nn1 67729,c1(C2CC(Cl)C2)nc(CN2CCOCC2)nn1CC1CCCCO1 67730,N1(CCCC)CCN(C(c2c(C)cnn2CC)C(=O)NC)CC1 67731,Cc1c[nH]cc1C(=O)NCCC(=O)NC1COCC1F 67732,N1(S(C2CC(c3c(OC)ccc(F)c3)C2)(=O)=O)CCc2ccc(Cl)nc2C1 67733,c1(OC)c(C)csc1C(N1CCCC1CCNC(=O)CCCc1cccs1)=O 67734,c1(C(=O)OC)ncc(F)cc1F.c12nsc(n1)N1CC(C(N)=O)(C1)CNC2=O 67735,c1(NC(c2scc(C(C(=O)OCC)(F)F)n2)=O)ccc(C#N)c([N+](=O)[O-])c1 67736,C1(NC(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(c1nnn3c1CCC3)=O)C2 67737,C1(CNC(c2cn(CCC)nn2)=O)CCC(C)N(C(c2ccnn2CCC)=O)C1 67738,CCC(C(=O)OC(C)(C)C)C(=O)NC(C)(C)CN(C(=O)C(C(C)C)OC)C 67739,c1(C(N2C(CNC(CCOC)=O)CCCC2)=O)ccc(C2CC2)c(F)c1C 67740,C(=O)(CC(CNC(C1C=CCCC1)=O)C1CCC1)NC(C#C)(C)C 67741,C12(C(N3CC(NC(c4cnc(=N)[nH]c4)=O)C(C(F)(F)F)C3)=O)CC3CC1C2C3O 67742,c1(NC2CCN(CC(=O)OCC)C2)ncc(F)cn1 67743,N1(C(CCCC=C)=O)CCC2CCN(C(C3CCC(=O)N3CCC)=O)CC12 67744,C12(C(N(C(C)C)CCNC(=O)CCNC(N)=O)=O)CC(C)C1C2 67745,c1(C(=O)NCc2cccc(C#N)n2)cnc(F)cc1CNc1[nH]cc(C(N)=O)c1 67746,C1(N(C(CN(C)C)=O)C)CN(C(C2CCCN2C(C2CCC2)=O)=O)CC1F 67747,C1(O)(C(N2CCC(CCNC(CCCC)=O)C2)=O)CCCCC1 67748,C(=O)(CCCCCC(C)(C)C)N1CCC(NC(c2ccnc(N(C)C)n2)=O)CC1 67749,CC(N=c1ncc(I)c[nH]1)C1CCCN(C(=O)C(C)(O)c2ccccc2)C1 67750,c1(C(=O)NCCC(=C)CNC(=O)CC2CCCOC2)ccccc1SC 67751,C1(CCC)(NC(=O)CC(C)COC)CCCN(C(c2cc(Cl)no2)=O)C1 67752,C1=C2N(C(=O)CC(C)CC1)CC2c1ccccc1.c1(CNC(C)C)cnn(C)c1C 67753,N1(C(COC)=O)CCC2(CCCC2NC(c2cnc(Cl)c(N)c2)=O)C1 67754,c1(C(=O)NCC2C(C)CN(C(=O)CCSCC(N)=O)C2)nn(C)c2ccccc12 67755,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCCCC1 67756,C1(C(=O)NCCC(C)(C)NC(C(CSC)C)=O)CC2C(C1)C2(C)C 67757,C(=O)(C(O)CNC(C1CC1(C)C(F)F)=O)N(C(C)CO)C1CC1 67758,n1(C(CC)C)nc(C(=O)N(CCNC(=O)C=Cc2csc(C)n2)C(C)C)cc1C 67759,C(=O)(C(F)C(=O)NC(c1cccc(Cl)c1)CNC(=O)CSC(C)(C)C)OCC 67760,c1(C(=O)NC2CN(C(C3(OC)CC3)=O)C(C)CC2)csc2cccnc12 67761,c1(NC(C2C(NCc3c(C(=O)O)cccc3)C2)=O)nc(Cl)c(Br)cc1O 67762,c1(N(C2CCCN(C(CCC(C)NC3C(=C)C3)=O)C2)C)snc(C)c1C#N 67763,C1(N(C)C)CN(C(c2cocc2Br)C(=O)NC2CCOCC2)CC12CC2 67764,c1(NC(=O)CC2CC(NC(N3CCC(F)C(F)(F)C3)=O)C2)ccc2c(c1)CCC2 67765,c1(OC)cccc2c(C(N3CCC(C)C(CNC(C)=O)C3)=O)coc12 67766,Cc1c(CNC(=O)CCCNC(c2ccccc2CO)=O)cccc1O 67767,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)[nH]c2cc[nH]c12)C1OCCN(C)C1 67768,c1(C(N(C(C)C(=O)NCC(O)CO)CC)=O)ncc2ccccn12 67769,C1(CC=C)(NC(=O)C(O)CSC)CC2CCC(C1)N2C(c1cnoc1C(C)C)=O 67770,C1(CC(=O)NC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)C(C)CC1CC1 67771,C1(C(=O)NCC2(CO)C(C)(C)C2)CCOCCN1C(c1ccc(C#N)o1)=O 67772,c1(-c2cn(C3CC(NC(CSS(C)(=O)=O)=O)C3)nn2)cc(F)c(F)c(F)c1 67773,c1(C(N(CCn2cc(CNC3CCC(=O)NC3)nn2)CC)=O)coc2ccccc12 67774,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccnc(OC)c3)=O)C2)cc(F)c1 67775,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CCNC(C1CC(C)(C)C1)=O)=O 67776,Cc1ccc(C=CCC(=O)NC(C)CCNC(=O)Cn2ncc(Cl)c2C)cc1 67777,C1(CCC(=O)NCC(CC)C(C)C)CCN(C(=O)CC2CCC(=O)C2)C1(C)C 67778,c1(OC)cccc(NC(=O)N(C)C(c2cccc(OC(F)(F)F)c2)C)c1OC 67779,N1(C(c2c(COC)cco2)=O)Cc2ccccc2C(CNC(c2cnn[nH]2)=O)C1 67780,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 67781,CCC(CC(=O)NCCC(=O)N(C(C)(C)CC(C)C)C)CC(C)C 67782,N1(C(=O)Cn2cnnn2)CCC2CCCC(C1)N2C(=O)CCN1CCCC1 67783,CS(=O)(=O)c1cnc(NC(=O)NC2(c3ccc(F)cc3)CC3(CC3)C2)nc1 67784,C1(NC(c2cn(C)c(=O)n2C)=O)CC(C2CCN(C(c3cnc(N)cn3)=O)C2)C1 67785,CC(C)(O)C(F)C(=O)N1CCOC(C2CN(C(c3cncc(N)n3)=O)C2)C1 67786,N1(C(c2cncc(C)n2)=O)CCC(C2CCN(C(C3CC3Cl)=O)CC2)CC1 67787,CC1(C)CN(C(c2ccon2)=O)CC1NC(c1cc(-n2ccnc2)cs1)=O 67788,CCCCS(=O)(=O)NC(N(C)CCCc1cn(-c2ccccc2Cl)nn1)=O 67789,N1(C(Cn2c(CCC)ncc2)=O)CC2(CCC2NC(c2cc(=O)cc[nH]2)=O)C1 67790,C1(NC(C(CSC)(C)C)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 67791,CN1CCC(C(=O)NCNC(=O)OC(C)(C)C)CC1.C1(C(C)(C)C)CNC(=O)CO1 67792,C1(C2CCN(C)CC2)(C(=O)NCC(N(C)C(C2CC2F)=O)C2CC2)CC1 67793,CC1CCCC(OCC(=O)NCC(C2CCCC2)NC(c2ccsc2)=O)C1 67794,CC1(C(=O)NCc2cccc(Cl)c2F)CCCN(Cc2nccs2)C1 67795,c1(CC(=O)NCCNC(CCCN(CCOC)C)=O)ccc(OC(F)F)c(F)c1 67796,c1(OC)nc(C(N2CCC(=CCNC(=O)C(c3ccccc3)O)CC2)=O)sc1C 67797,N1(C(c2n[nH]cc2C(F)(F)F)=O)CC(N=c2[nH]nc(CO)s2)C2(CCC2)C1 67798,N1(C(C)=O)CCCC(O)(C(N2CC(O)(CNC(=O)CNc3ccsc3)C2)=O)C1 67799,CCC(CC)CC(=O)NCC1CN(C)CCN1C(c1cc(C)nn1C(C)C)=O 67800,n1(COC)nccc1C(N1CCC(OCC(=O)NC(C)Cc2ccnn2C)C1)=O 67801,c1(-n2c(-c3[nH]cc(CC)c3)nc(-c3ccoc3C)n2)nc2ccccc2n1CC 67802,C(=O)(CC(=O)NCC1CC(NC(c2c[nH]nc2Cl)=O)C1)NCC 67803,N1(C(C)=O)CCN(C(=O)CCCn2cc(C(C3CC3)C3CC3C(=O)O)nn2)CC1 67804,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CCN2CCCS2(=O)=O)CC(O)C1)=O 67805,N=c1[nH]cc(C(=O)NCC(F)CNC(c2cscc2F)=O)c2cc[nH]c12 67806,C1(C(NOCCOCC)=O)CCC(O)CN1C(c1cnncc1O)=O 67807,N1(C(c2cc(C)cc(C)n2)=O)CC2(CCC1)CN(C)CCO2 67808,c1(C(=O)NCCCNC(c2cccc(N)c2F)=O)c[nH]c2ccc(F)cc12 67809,c1(NC)snc(C)c1C(=O)NCC12CC1CN(C(C1CN(C(=O)NC)C1)=O)C2 67810,c1(CNCC2CCC(NC(c3cccc(Cl)c3)=O)CC2)ccc(C#N)cc1[N+](=O)[O-] 67811,C1(C2(O)CCOCC2)(CS(N2C(C(=O)OCC)C(O)CC2)(=O)=O)CC1 67812,c1(OC(C)C)cccc(C=CC(=O)NC(c2c(C)noc2C)CNC(=O)CO)c1 67813,c1(C(=O)NCCCNC(C2CCC2n2ccnc2)=O)cccc(C2CCC2)c1 67814,Cc1cnc(C(C)N(C(=O)C(C2CCCCC2)C)C)s1 67815,N1(C(c2c(C)ccs2)=O)CCC(NC(c2cc(C(F)(F)F)ccc2N)=O)CC1C 67816,C(=O)(C(C)(CC)CO)NCC(CC=C)NC(c1ncc(C(F)(F)F)cc1Cl)=O 67817,CC1CCCN(C(C)CNC(=O)N(c2ccccc2)c2conc2C2CCCO2)C1 67818,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 67819,C#CCC(C)(CC)C(=O)N1CCCCC(C(N2CCc3ncsc3C2)=O)C1 67820,C(c1ccc2occc2c1)=CC(=O)NC1C(NC(C(C(C)O)C)=O)CCC1 67821,C(=O)(CC(C)CC(F)(F)F)N1C(CNC(C(F)=CCC)=O)CCC1 67822,CCC(CCCC(F)(F)F)NCc1csc(Br)c1Cl 67823,C1(C(=O)NCCCCOCCCNC(C2(CF)CCC2)=O)COCC1C(F)(F)F 67824,c1(SCC(=O)NC2CN(C(c3cc(Cl)c[nH]3)=O)CC2O)ccc2c(c1)CCC2 67825,C(CNC(c1ccc(CO)nc1)=O)(CC(F)(F)F)NC(COCC(=O)NC)=O 67826,c1(CC(=O)NC(CC(C)NC(c2cnn(C)c2C(F)F)=O)C)ccc(F)c(F)c1 67827,C(=O)(C1=CCCSC1)NC(C(C)C)CNC(=O)COC1CCCOC1 67828,C1(NC(c2cn(CC=C)nn2)=O)CN(C(=O)C2=CCCCO2)C2(CCCCC2)C1 67829,c1(C(=O)NC(CCCNC(C2(CCC)CC2)=O)C)cc(C)nn1CC(F)F 67830,N1(C(CCC#CC)=O)CC2CCC1CN(C(c1cccc(OC(C)C)c1F)=O)C2 67831,Cc1cc(C)n2nc(C(C)NCCOc3cccc(Br)c3Cl)nc2n1 67832,c1(SCCC)ccc(Cl)cc1C(=O)NCC(CC)NC(=O)C(F)CC1CCC1 67833,C12(NC(COC(CC)(C)C)=O)CCC(F)(F)CC1CN(C(=O)C(F)C(C)(C)O)C2 67834,c1(C(=O)NC2CC(NC(c3nc(C)sc3C)=O)C2)ccc2nn[nH]c2c1O 67835,c12cc(Br)ccc1S(=O)(=O)NCC(C)N2.C12(COCCOC)CC(C)(CCO1)C2 67836,C1(NC(C(C)C)=O)CCN(C(c2csc(C(F)F)c2)=O)CC1C(C)C 67837,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 67838,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)C(F)C3CCC3)C1)C2 67839,O=S(=O)(c1cccc(NCC2=NOC3CCCC23)c1)N1CC2CC1C1CC21 67840,c1(CNC(N2C(C3(C=C)CCC3)CCC2)=O)c(F)ccc2c1OCC2 67841,C12(CNC(C=CCOC)=O)CC1CN(C(C1CC(C)(F)C1)=O)C2 67842,C(=O)(CCCCCOC)NCC1C(C(N2CCC(=C)C2)=O)C1 67843,c1(C(N2CCC(CNC(C(C(C)C)N(C)C)=O)CC2)=O)cc(=O)c(=O)[nH][nH]1 67844,C1(NC(C(C)SC)=O)COCC1NC(c1ccoc1I)=O 67845,CC(CO)(C(F)F)NC(=O)CSCCNC(C1OC2CCC1C2)=O 67846,c1(C(=O)NCC2CN(C(CC(C=C)C)=O)CC2O)n[nH]c2c1CS(=O)(=O)CC2 67847,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 67848,N1(C(C=C2CCC(C)CC2)=O)CCC(O)(CN(C)CCO)CC1 67849,c1(Cn2c(C(CC)NC(C)CCC(C)C)nnn2)cc(C(F)(F)F)ccc1C#N 67850,C#CC1CCC(CN2CC(N(c3ccccc3)C)C2)CC1 67851,CC(C)(C)C(CC(=O)OC(C)(C)C)C(=O)ON1CCCOC(=O)C1 67852,C1(NC(CC2CN(C)C2)=O)CN(C(c2cncn2C2CCOCC2)=O)CCC1O 67853,c1(C(=O)NCC(C)(C2CC2)NC(=O)CC2(O)CCOC2)cnn2c(=O)cc[nH]c12 67854,C1(CNC(C2CC(C)OCC2)=O)CC2(CCN(C(=O)COC3CCOCC3)C2)CO1 67855,Cc1[nH]c(C)c(C(=O)NCC2=CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)c1C 67856,C1(CNC(CS(=O)(=O)NC)=O)CCC2(CCC2)CN1C(c1cncn(C)c1=O)=O 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67998,C1(O)(CN(C(Cc2ccc(C)nc2)=O)C)CCN(C(=O)C(C)(C)CC#N)CC1 67999,N1(C(c2n[nH]c3c2CCC3)=O)CCC2C(CCN2C(=O)CCC2CCOC2)C1 68000,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2C3)CCc2nnnn2CC1 68001,Cc1nn(CC(=O)NC(C(=O)NCCCC(F)F)C(C)C)c(=O)o1 68002,n1(CCn2c(-c3c(Cl)n[nH]c3)nc(C3CCCO3)n2)nnc2ccccc12 68003,C=CCC(C)C(=O)NC(c1ccc(CNC(=O)CCc2cnn(C)n2)cc1)C 68004,c1(C(N2CCC(CN(C(=O)C(N3CCC(O)CC3)C)C)C2)=O)cn2c(n1)CCC2 68005,C1(C(=O)NC2CCN(C(c3c(OC)csc3)=O)C2)C2CC1(c1ccccc1)CO2 68006,C1(C(N(CCC(C)NC(c2cc(C3CC3)ccc2F)=O)C)=O)CCC(C)(C)CO1 68007,C1(C(N2CCN(C(CC#N)=O)C(CC(F)F)C2)=O)CC2CC(O)C(C1)C2 68008,Cc1cnc(C(=O)NC2CCC(C(=O)N(C3CC3)Cc3ccccc3F)C2)cn1 68009,Cc1cncc(C(N2CCCC2CCCNC(=O)C(C)OCC2CC2)=O)c1C 68010,Cc1ccc(Cl)cc1NC(=O)C(=O)NCCC1CC1C 68011,c1(CCCC(=O)N(CCNC(C=CC)=O)CCSC)cccc(Cl)n1 68012,c1(CC(=O)NCC=CCNC(C2C(COC)C2)=O)ccc(F)c(Cl)c1 68013,N1(C(C(CCC)CNC(=O)CN2CC(C)(C)C2)=O)CCC2(CCCOC2)C1 68014,Cc1nc(N(C)C)cc(N2CCCC(N(CC(F)(F)Br)C)C2)n1 68015,c12ccc(C)c(c1)NC2=O.c1(OC)ccccc1C(N1CCCCC1CC#N)C 68016,c1(C(N2CCC(NC(C(C)OCC#C)=O)CC2C)=O)cc2nc[nH]c2cc1F 68017,C(=O)(C(C)(F)C(=O)N1CC=CC(C(N2CCOC(CN(C)C)C2)=O)C1)OC 68018,C1(C(c2nnnn2C(C)C)C)CC(C)(C)C1NC1C2CC21.c1cnn(C)c1C.OC 68019,N1(C(=O)NCc2cc(C(=O)OCC)n[nH]2)CC(=O)N2CCCCC2C1 68020,C1(C(=O)NCC2(Cl)CC2(F)F)COC2(C1)CN(C(=O)CCSC1CCC1)C2 68021,c1(C(N2CC3CC(NC(CC=CC=C)=O)CC3C2)=O)csc(N=S(C)(C)=O)n1 68022,C#Cc1ccc(C(N2CCC3CC23C(=O)NC(c2cnn(C)c2)C)=O)nc1 68023,CCCCCCCCC(=O)NC1CCC(NCc2csc3ccccc23)CC1 68024,N1(C(CCC)=O)CCCC(C(=O)NCCN(C)C(c2ncsc2CC)=O)C1 68025,c1(N2CCN(C(CC)=O)CC2)ncc2c(n1)CN(Cc1ncc(C3CC3C)o1)C2 68026,c1(C(=O)NC2CC(NC(C(C)=C3CCCC3)=O)C23CCC3)cc(C)cc(Cl)c1N 68027,C1(C(C)C)CC(NC(C2CC(C)(O)C2)=O)CO1 68028,Cc1cccnc1CCC(=O)NC(CNC(c1cnc[nH]1)=O)(CO)CO 68029,c1(-c2n(CCc3c(OC)cccc3)nc(C3CC3)n2)cc2cccc(OC)c2[nH]1 68030,C(CCCCC(=O)NC1CCCC1(C)CO)N(C(C1N(C(C)C)CCC1)=O)C 68031,c1(C2C(C(N(CC(C)(C)NC(c3ccc(C4CC4)o3)=O)C)=O)C2)ccccc1F 68032,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)CCN(C)C)CC1c1ccnn1C 68033,C(CCCCC(=O)N1CC(C2(NC(C34CCCC3CCC4)=O)CC2)C1)NC(N)=O 68034,C1(NC(c2c(OC)c(C)cc(C)c2)=O)CC2(CN(C(=O)CCCC#N)C1)CCO2 68035,C1(C(C(=O)NCC(=O)OC(C)C)NC(=O)CN(C)C(N)=O)CC=CCC1 68036,Cc1ccc2ccccc2c1C(c1nnc(S(N)(=O)=O)s1)NC(=O)OC(C)C 68037,C1(CCC)CN(C(=O)C(c2c(C)n[nH]c2C)C)CC1CNC(=O)CSC(F)(F)F 68038,N1(C(c2c(C)ocn2)=O)CC2(CCOCC2C(=O)Nc2cc(CO)ccc2F)C1 68039,c1(OCCC)ccc(-c2cn(CC(=O)NC(C)N=c3[nH]ncs3)nn2)cc1OC 68040,c1(-c2nc(C(C)OC)nn2CC(C)C2CC2)scc2c1OCCO2 68041,N1(C(CC(CC)C)=O)CCCCCCC1C(=O)NCc1noc(CC)n1 68042,c1(SC)ccc(C(N2CC(NC(=O)CC(c3cccs3)N(C)C)C2)=O)cc1 68043,CC(CC(C)(F)F)C(=O)NC1CCC1NC(=O)CNC(=O)CNC(N)=O 68044,Cc1cnncc1C(=O)NC(CC1CC1)CC(=O)NCC(N1CCOCC1)=O 68045,C1(C(N(C2CCN(C(=O)Cc3sccc3C)C2)CC)=O)Cc2nccnc2C1 68046,c1(C(N2CCC(C)C2CNC(c2cnc(N(C)C)o2)=O)=O)cc2cccnn2n1 68047,c12cc(ccc1OC)CCO2.O(NC(=O)NC(C)C1CC1)CC(=C)C 68048,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68049,N1(C(C2=C(C)OCCC2)=O)CCOC2(C1)CN(C(=O)CC13COC(CF)(C1)C3)C2 68050,c1(NC(C(=O)NC(C)(CC2CCCCC2)CO)=O)ncc(Br)cc1Cl 68051,c1(C2(N(C(C#C)=O)C)CCC2)cc(C2CC2)ccn1 68052,c1(C(=O)NC2CCC(N(C(=O)C=Cc3ccc[nH]3)C)C2)cnnc(O)c1 68053,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68054,C1(C(=O)NC(CC)CNC(=O)CC(C)CC)CCn2c(Br)cnc2C1 68055,c1(NC(CCC=C)C)ccc(S(=O)(=O)NCCc2ccncc2Cl)cc1Cl 68056,C1(CC)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)CCCc2ccccc2F)CC1 68057,C1(CNC(CC=CC)=O)CN(C(c2ccc3c(c2)CC3)=O)CCN1C 68058,C1(COC(c2ccccn2)=O)CN(Cc2ccccc2Br)CCO1 68059,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=C(C)C 68060,c1(OCC)cncc(C(=O)NC2CC(CO)N(C(=O)Cc3cc(Cl)cs3)C2)c1 68061,CC1CCc2[nH]c(C(N3CCOC(CNC(c4ccnnc4O)=O)C3)=O)cc2C1 68062,c1(C(=O)NC2(C)CCN(C(=O)C#CC3CCCO3)C2)ccc([N+](=O)[O-])cc1 68063,c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)ccn(C)c(=O)c1 68064,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68065,c1(C(N2CC(C)(CNC(c3c(OC)n[nH]c3)=O)C(C)C2)=O)c(F)ccc(C)c1Cl 68066,C1(C(C)C)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)CC(F)F 68067,C(=O)(C1CCc2nccn21)N1CC(C)C(NC(=O)CC2(n3cccn3)CC2)C1 68068,C(=O)(C(Cc1ccccc1)CC)NCC1C(CNC(CCCOCC)=O)CC1 68069,c1(N(C)CC)ccc(C(=O)NCCC(C)(C)CNC(=O)C(C)(C)F)cc1 68070,C(CCSC)(C(=O)NCCCN(C(c1ccc(C)o1)=O)Cc1ccccc1)OC 68071,c1(-c2cccc(CNC(=O)OC(C)(C)C)c2)nc(-c2cccs2)nc2[nH]ccc12 68072,N1(C(C2(NC(C(C)OCC#C)=O)CCOCC2)=O)CC2CC(C)C2C1 68073,C(=O)(CCCC(=O)N(C1(c2ccon2)COC1)C)c1ccc(OC)cc1 68074,c1(OC)ccccc1CC(=O)N(CC(C)N(C1CC1OC)C(c1nocc1C)=O)C 68075,C(C1=NOC2CN(C(=O)CCN3CCOCC3)CC12)NC(c1cc(OC)no1)=O 68076,C1(CC(N)=O)(NC(CNS(NC)(=O)=O)=O)CCN(C(C2CC23CC(F)(F)C3)=O)CC1 68077,C(C(C)(C)C(C)(F)F)(c1n(CCOCC)nnn1)NCc1ncsn1 68078,c1(C(N2CCC(C)(C(=O)NC(C(F)F)C3CC3)C2)=O)cc2ncccc2[nH]1 68079,C1(C(=O)NC(C)(C)C)C2CCC(C2)C1C(F)(F)F.CN1CCNCC1 68080,c1(C(=O)NC2C(C)CN(C(=O)C(=O)NCC(F)(F)F)CC2)cc2cn[nH]c2cn1 68081,c1(N2CCC(CC(=O)NCC(C(=O)NCCOC)C)C2)cc(CO)ncn1 68082,c1(C(=O)NC(CN(C(C2CCOC(=O)N2)=O)CC)C)ccc(COC(C)C)cc1 68083,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68084,C1(C(=O)NC2CCC(NC(CCC)=O)C2)COCCN1CC 68085,C1(CC(NOCCCOC)=O)CN(C(=O)C2=CCSC2)CC12CC2 68086,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)C(F)F)C1)F 68087,c1(C(N(CCNC(C(c2cccc(N)c2)NC(C)=O)=O)C)C)cccc(F)c1 68088,C(CC(=O)N1CCCC1)OCCNC(COCC(=O)NC)=O 68089,C(c1cnc[nH]1)=CC(=O)NCC(CN(C(=O)Cc1cocn1)C)O 68090,N1(C(C(C)CF)=O)CC2(CCN(C3CCc4ccc(Br)cc43)CC2)S1(=O)=O 68091,c1(C(=O)NC(CC)CNC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68092,N1(C(c2cc(SC)ncc2)=O)CCN(C(C23CC(C)C2C3)=O)CC1CC1CC1 68093,N(C1CCc2ccc(F)c(F)c21)C(c1cnc(C)c(C)c1C)C 68094,N1(C(C2(CC#C)CCCC2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68095,Cc1nc2n(c1COC(c1c(C)nc3sc(C)cn13)=O)CCCC2 68096,c1(C(=O)NC2CCCN(C(CCCCCOC)=O)C2)cccc2c1CCCO2.C(C)=O 68097,CC(C)C(C)C(=O)N1CCOC(CNC(=O)Cc2cncnc2O)C1 68098,N1(C(C2(Cl)CC23CCC3)=O)CC2CCC(CNC(C3(C4CC4)CC3)=O)(C2)C1 68099,C(=O)(C(CC(F)F)N(C)C(c1ccc(F)cc1F)=O)N(CCCSC)C 68100,C1(NC(c2ccc(-c3ccccc3)cc2)=O)CCCN(C(c2ccncc2F)=O)C1 68101,C1(C(=O)NC2CC(C)N(C(C3(O)CCOC3)=O)C2)COc2ccccc2C1 68102,N1(C(C(CC2CCOCC2)NC(c2cc(C3CC3)on2)=O)=O)CC2COCC2C1 68103,N#CC1(C(N2CC3(CC3)CC2C(=O)NCC2CC23CC3(F)F)=O)CCOCC1 68104,C=C(C)CCC(=O)N1CCC(N(C(=O)C(=Cc2cnc[nH]2)C)C)CC1 68105,C#Cc1cccc(CC(N2CC(C(=O)NCc3ccc([N+](=O)[O-])o3)CC(C)C2)=O)c1 68106,C1(F)(CNC(c2csnc2Cl)=O)CCN(C(C2CCC(N(C)C)C2)=O)CC1 68107,N1(CC(N2C(CN(C(CC)=O)C)CCCC2)=O)C(=O)C(=O)N(C)C1=O 68108,N1(CCNC(C2CC(NC(c3scc(C(C)=O)c3)=O)C2)=O)CCN(C)CC1 68109,C1(CNC(=O)NC(C)C2CC2)CCCC(C(F)(F)F)C1 68110,c1(N2CCC(NC(C(CCC)(C)O)=O)C(C)C2)ncc2ncnc-2[nH]1 68111,c1(C(N2C(CNC(C3(OC)CC3)=O)C(C)CCC2)=O)cccc2c1CC(C)(C)C2 68112,Cc1ccc(Cl)c(C(=O)NC(CO)CCCNC(=O)C=CC2(C)COC2)c1 68113,C1(CC)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)CCC(C)(C)F 68114,C1(C(N2CC(NC(C(C)=C3CCCC3)=O)C(O)C2)=O)Cc2ccccc2S1 68115,N1(CC(C(=O)OC)(C)C)CC2CCCCCC2(C#N)C1 68116,C1(NC(C(C)CC2CCC2)=O)CCCC12CN(C(c1sc(F)cc1Cl)=O)C2 68117,C(=O)(CC(C(=O)N1CC(NC(=O)C=Cc2ccsc2)C1)NC(C)=O)OC 68118,c1(N(C)C)cncc(C(=O)NC(c2nnnn2CC(F)F)CCC2CCCO2)c1 68119,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCO3)=O)C4)=O)cc2o1 68120,c1(C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)ncc(Cl)nc1Cl 68121,C(C(CC(=O)N1CCOC(C(C)(C)C)C1)OC)NC(CC=C)=O 68122,CCCC(O)CN=c1[nH]c(=NCCCCCC(C)(C)OC)[nH]c2c1COC2 68123,C(=O)(C1=NNC(=O)CC1)N1CCC(C(C)NC(c2ncnn2C)=O)C1 68124,C=CCC(C(=O)N1CC(OCC(=O)NCC2(CC)CC2)C1)c1ccccc1 68125,N1(C(=O)CCC2CCOC2)CCCCC(C(=O)NC2(C3CC3)CCCC2)C1 68126,N1(C(c2cc(C)ncn2)=O)C2CCC1C(NC(=O)C(C1CCOCC1)N(C)C)C2 68127,c1(C(N2C3CC(NC(c4cc[n+]([O-])cc4)=O)(C3)C2)=O)cnc(O)c2cncn12 68128,Cc1csc(=NCC(=O)N(C2CN(C(C3CS(=O)(=O)C3)=O)C2)C)[nH]1 68129,N1(C(=O)Cn2cnnn2)CCN(C(C2CC3(CCC3)CO2)=O)C(CCO)C1 68130,N1(C(CC2CN(C(c3ccc(COC)cc3)=O)C2)=O)C2CCC1CC(F)(F)C2 68131,c1(N(C)CC2CCN(C(CC)=O)C2)[nH]c(=NC(C)c2cncs2)nc2sccc12 68132,Cc1cc(C(=O)NCC(N2CCN(C(c3csnn3)=O)CC2)=O)c(Cl)cn1 68133,C1(C(=O)Nc2c(CNC(C3(NC(=O)OC)CCC3)=O)c[nH]n2)CCC12CCCO2 68134,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68135,N1(C(c2ccn(COC)n2)=O)CCN(C(c2cc(COC)on2)=O)CC1CO 68136,C(C)(CC(C)NC(c1ccnn1C1CCCC1)=O)NC(CN(CCOC)C)=O.C1CCC1.O 68137,c1(C(N2CCCC(CNC(C3(SC)CCC3)=O)C2)=O)cc(C)nc(O)c1 68138,N1(C(CC2(CN(C)C)CC2(F)F)=O)CCN(C)C(CNC(C2CSCCS2)=O)C1 68139,CCCC(C(=O)NCC1(NC(c2ccc(S(N)(=O)=O)[nH]2)=O)CCOCC1)C(C)C 68140,Cc1[nH]c(C#N)cc1C(=O)NC(c1nocc1C(=O)NCCOCC(F)F)C 68141,C1(N(CC(=O)N(C)Cc2cncs2)C(C2C(C)C2)=O)CC(C#N)C1 68142,N1(C(CN(C(=O)C(c2ccc(Br)cc2)CO)CC)=O)CCCC(CO)C1 68143,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ncc[nH]2)c1)=O 68144,Cc1cc(C)n(CC(=O)NCC2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)n1 68145,C1(N(C(c2nccs2)=O)NC(=O)COC)C=CCN(CC)C1.c1(C)c(CO)noc1C 68146,N1(C(CC(C)=C(C)C)=O)CCCC(C)(C(=O)Nc2cccc(Cl)c2)C1 68147,C(CC)(CC)(CCNC(=O)Cc1cc(C)no1)NC(c1c(C(=O)OC)c[nH]c1C)=O 68148,C1(N(C(CNC(C(C)C)=O)=O)C)CN(C(c2ccc(OC3CC3)cc2)=O)CC1F 68149,C#CCC(C)(C(=O)NCc1ccc(O)cc1)NC(C1CCCC1F)=O 68150,CCC(CC(F)(F)F)NC(C1(CCNC(=O)C=Cc2cc[nH]n2)CC1)=O 68151,Cc1cncc(C(N2CCC(CCNC(c3nncs3)=O)C2)=O)c1 68152,C1(N(C(c2c(CC)[nH]cc2)=O)C)CCN(C(=O)C=Cc2cncnc2O)CC1C 68153,c1(C(N2CCC(N(C(COCC(C)C)=O)C)C2)=O)cc(N)cc(F)c1 68154,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68155,Cc1ccc(F)c(C(=O)NCCCN(CCCNC(C2CC3CC3C2)=O)C)c1F 68156,C1(NC(=O)CSCc2ccccc2)CCN(C(c2cscn2)=O)CCC1CCO 68157,c1(C(=O)OC)ccc(N(C)C)cc1F.C12(CCC1)NC(=O)CC1(CC1)C(=O)N2 68158,N1(C(C2C(C)CC2)=O)CCCC2CCN(C(=O)C=Cc3nccs3)CC12 68159,C1(NC(COCc2c(C)ncs2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68160,C1(NC(c2cc3c(nn2)CCC3)=O)CCSC12CN(C(C1CC1F)=O)C2 68161,C(CCCCNC(=O)C(O)C1CCCC1)NC(C(c1ccccc1)NC(C)=O)=O 68162,Cn1cc(C(N2CC3CC(NC(=O)C(O)C4CC4)C2C3)=O)c2ccccc12 68163,CC(c1ccccc1F)=CC(N1CC(N(C)C(C2COCCN2C)=O)C1)=O 68164,C1(C(=O)NCCSC(C)(C)C)CNCCN1Cc1csc(Cl)n1 68165,N1(C(CCCN(C(C)=O)C)=O)CC2CCC1CC2NC(C1CCC(C2CC2)O1)=O 68166,C1(C(CO)NC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68167,c1(CC(=O)NC2CCC(CSc3ccncc3)C2)ccc(C(F)(F)F)cc1[N+](=O)[O-] 68168,C1(C(=O)NCC(C)N(C)C(c2nc(CC3CCCCC3)cs2)=O)CC2C=CC1C2 68169,c1(CCC(N2CC(C(C)NC(=O)C(CC)N3CCCC3=O)C2)=O)c(C)noc1C 68170,C1(NC(=O)Cc2cccs2)CC2CCC1CN2C(C1C2CCCCC12)=O 68171,C#CCCCCCCCC(=O)N(CCNC(=O)Cc1csnn1)CCOCCO 68172,C(=O)(CC(C)CC(C)(C)C)NCCC(=O)NCc1ncc(C)cn1 68173,CN=c1ccc(C(=O)NC(C)(C(N2CCC(F)(CF)C2)=O)C2CCC2)c[nH]1 68174,N1(C(C(C(C)NC(=O)CN2CCN(C)CC2)(C)C)=O)CCC2CCCC2CC1 68175,C1(C(=O)NC23C(CN(C(C4(CC(=O)OC)CC4)=O)C2)C3)CCc2nc(C)[nH]c2C1 68176,Cc1nc(CCC(=O)NCC2C3CN(C(=O)Cc4ccc(F)nc4)CC23)oc1C 68177,c1(C(N(C(C(=O)NC(CCC)c2ccco2)C)C2CC2)=O)snc(C)c1N 68178,CN1CCC(C(=O)NCCOC(F)F)(NC(=O)Cc2cnns2)C1 68179,c1(N(C)Cc2cn(C(c3ccc(OC)cc3)C)nn2)c(F)cc([N+](=O)[O-])cc1F 68180,c1(C(N2CCCC(C(C)NC(C=CCC)=O)C2)=O)cccc2c1OC(C)C2 68181,CCC(C)(C(=O)N1CC(CNC(=O)C(C)(C)C2CCOC2)(OC)C1)OC 68182,N1(C(C=CCC)=O)CC(NC(=O)C=Cc2ccccn2)CC1(C)COC 68183,CC(C(C)(C)NC(C1CCCCO1)=O)NC(c1cnc(C(C)(C)C)[nH]1)=O 68184,c1(C(=O)NC(CC2CN(C(c3cc(C)[nH]n3)=O)C2)C)cc2sccc2s1 68185,O(C1C(=O)Nc2c1ccc(Br)c2F)CCC(C)C 68186,N1(C(=O)C(C2CCN(C(=O)C(C)(C)OC)C2)F)CCCC(C)(C)C1C.CCCN 68187,N1(CCCCOC)CC2CCC1CN2C(C1CC(NC(=O)OC)CCO1)=O 68188,N1(C(C2(CC=C)CCN(C(=O)C(C)OCCC(C)C)C2)=O)CCC(O)CC(C)C1 68189,N1(CC)CCN(C(C2CCN(C(=O)CCCC(C)=O)C(C)C2)=O)C(C)C1 68190,c1(SCC(=O)N(C2CCCC(NC(=O)CNC3CCC3)C2)C)ccc(C#N)cc1 68191,N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)C2=C(C)CC2)CC1(C)C 68192,CCCCCCOCC(=O)NCC1(NC(=O)CCc2cnc(O)[nH]2)CCOC1 68193,CN1CCC(C(N2CCC(C(c3ccco3)=O)C2)C(=O)NC(C)(C)C)CC1 68194,c1(OCC)cc(CNC2CC(NC(c3cc(Cl)ccc3Br)=O)C2)cc(F)c1 68195,C1(NC(c2cncc(F)c2)=O)CN(C(=O)C#CC2CCCO2)C2(CCC2)C1 68196,C1(CN(C(=O)C(C)N2CCCC2)CC)CCCN1C(=O)C(C1CC1)SC 68197,C1(C2CC2)(CNC(C2(OC)CS(=O)(=O)C2)=O)CCN(c2nc3ccccc3o2)C1 68198,c1(C(=O)NC2C(CNC(COCC(=O)NC)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 68199,N1(C(N(C)C)=O)CC2CN(C(C3COCCN(C(=O)CC4CC4)C3)=O)CCC12 68200,C1(C#CC(=O)NC23CC(NC(=O)CN4CCC(=O)NC4=O)(C2)C3)(CC)COC1 68201,N1(C(c2c(C)nc[nH]2)=O)CC(NC(C2(O)CC2)=O)CC2(CC2)C1.c12ccc(cc1)s2 68202,C1(C(C)(C)O)(CC=CC)CN(C(=O)CCC)C1.O(C(F)(F)F)OC(C1(C)CC1)=O 68203,c1(C(=O)NCc2c(C(=O)NC(CC#C)CO)[nH]cc2)c[nH]c2ncccc12 68204,Cn1c(O)nc2cc(C(=O)NC3CN(C(=O)CC(O)C4CC4)CC3(C)C)ccc12 68205,Cc1noc2ncc(C(=O)NC3CC4CC3N(C(c3ncccn3)=O)C4)cc12 68206,CC1(C)CC(C)(CNC(c2nn[nH]c2Cl)=O)CN1C(=O)CN1CC2CC2C1 68207,c1(N2CCN(C(C(C)C3CC3)=O)CC2C)cc(=O)n2cc(Cl)ccc2n1 68208,Cc1ccc(NC(=O)CN(c2ccccc2)C(C#N)C2CC2)c2[nH]cc(C#N)c12 68209,C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C)CC1)C(C1ON=C(C(C)C)C1)=O 68210,Cc1cc(C(=O)N(C2CN(C(C3CCOC(=O)N3)=O)CC2F)C)oc1C 68211,C(=O)(C1=CC2C=CC1C2)N(CC(C)CNC(=O)CC1(C)CCCC1)C 68212,C1(NC(COC(C)=O)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68213,C1(=CC(=O)NC(CCC)CCCNC(=O)C(C)CF)CC2CCC(C1)N2C 68214,C#CCCCCCCC(=O)NC1CC(NC(c2ocnc2CC)=O)CC1O 68215,N1(C(CN(C(C#CC)=O)C)=O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 68216,C(=O)(C1=CC2C=CC1C2)NC1(C(N2CCC(CC)C(O)C2)=O)CC1(C)C 68217,c1(C(N2C(CNC(C3(C)CC3(F)F)=O)COCC2)=O)ccc(Cl)cc1O 68218,c1(C(=O)NCCCN(C(=O)CCc2cc[nH]n2)CC)ccnc(Cl)c1Cl 68219,c1(CC(C)C)cccc(C(=O)NC2CCC2NC(C2CC2c2cccc(Cl)c2)=O)c1 68220,N1(C(C(C(C)C)c2ccc(-n3ccc(C)n3)s2)=O)CC(O)C(O)C(O)C1CO 68221,C1(NC(C2CC(OC)C2)=O)CN(C(=O)C2=CCOC2)CC1C(F)F 68222,c1(NC(NOCC(=O)NC(CCCC)COC)=O)ccc(F)cc1F 68223,c1(-c2ccc(CNCCSC(=N)N)cn2)ccc(F)c(F)c1 68224,c1(CC(N2CC(F)(CNC(C3(COC)CCCC3)=O)C2)=O)cc(F)ccc1C 68225,C1(NC(C2C(CNC(c3cn(C(C)C)nc3)=O)CCO2)=O)C(=O)NCCC1C 68226,C1(C2CC2)(C(N2CC(CC)(CC)C2)=O)CN(C(=O)Cn2nc(C)oc2=O)C1 68227,c1(C(=O)NCCCCN(C)C(c2ccc(N(C)C)cc2)=O)ccc2ccnn2c1 68228,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68229,C(C)(N=c1ccnc(NCC2CC2(C)C)[nH]1)c1ccc(SC)cc1 68230,CCC(C)CCC(=O)NCC(C)(CNC(c1ccc(F)cn1)=O)OC 68231,CCC(CC(=O)NCC1COC(CNC(=O)C=CCOC(C)(C)C)C1)C(F)F 68232,C(=O)(C#CC(C)(C)CN(C(C#C)C)C)NC(=O)CN(C)CCO 68233,C(=O)(C1=C(Cl)CCC1)N1C(C(C)(C)CNC(=O)CCOC2CCOC2)CCC1 68234,C1(n2cc(C(C3CCCOC3)=O)nn2)CCN(CC(C2CC(=O)NC2=O)=O)CC1.CN 68235,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68236,CC(C)CCCC(C)C(=O)N(CC(C)N(C)C(C1Cc2c(F)cccc2O1)=O)C 68237,N1(C(C(COC)C)=O)CCN(C(C2CC23CCOC3)=O)CC1C 68238,Cc1c(C(=O)NCC2C3CC2N(C(C2CCCN2N=O)=O)C3)cncc1N 68239,C=CCCCCCC(=O)NC1(C2CN(C(=O)C(F)(F)CO)C2)CC1 68240,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(=O)CCC2CCOC2)C1 68241,C1(C(N(C2CCN(C(=O)CCC(C)N(C)C)C2)CC)=O)C(C)(C)C1(C)C 68242,N1(CC(=O)NC2CN(C(=O)CC3CC=CC3)CC2C(F)(F)F)CCS(=O)(=O)CC1 68243,C1(CN(C)C(C2CCCCC2)=O)COCCN1C(c1cocc1C(N)=O)=O 68244,Cc1cc(=N)[nH]cc1C(=O)NCC1(CCNC(=O)C(C)(C)C(C)C)CC1 68245,c1(CC)nc(C(=O)NCc2cc(C(N3CC(CC)C(O)C3)=O)[nH]c2)c(C)o1 68246,N1(C(C2C(C)=C2)=O)CCC(NC(c2ncccc2OC(C)C)=O)C(C)C1 68247,C(C1NC(=O)c2ccccc21)Nc1nccc(=NCC2CN(C)C(=O)C2)[nH]1 68248,N1(C(C(C)=CC)=O)CC(O)(C2CCN(C(c3cc(C)c(C)cc3Cl)=O)CC2)C1 68249,N1(C(C2CN(C(c3c(C)nc(O)s3)=O)C(C)(C)C2)=O)C2CCC1CC(=O)NC2 68250,c1(C(N2CCCC(N(C(CC=C=C)=O)C)C2)=O)c(C)oc(C)c1C 68251,N1(C(C2C(CC)CN(C)CC2)=O)CC2=C(C1)CN(C(c1ccoc1Cl)=O)C2 68252,c1(NC(=O)Nc2cc(C)sn2)cccc(CC2CC2)c1 68253,C1(C(N(OC)C)=O)CN(C(C2(OC(C)=O)CCC2)C(=O)NC2CCCC2)CC1F 68254,C1(C)(CNC(CC(C)CF)=O)CCCN(C(c2cc(NC(N)=O)ccc2O)=O)C1 68255,c1(OC)cc(NC(C2(F)CCN(C(c3c(Cl)ccnc3Br)=O)C2)=O)nc(Br)c1 68256,c1(C(N2CCC(NC(c3ccncn3)=O)CC2)=O)c(F)cc(I)cc1F 68257,c1(C(N2CC(CNC(COC(C)(C)C)=O)OCC2)=O)ccnc2[nH]ncc12 68258,C(=O)(C#CC1CCCC1)N(CC)CC.CCCC(F)(F)C(=O)N(CC)CC 68259,C(C(C)(C)CC(=O)N1CCC(OCC(N)=O)C1)NC(CN(C)C)=O 68260,C#CC(C)NC(=O)CN(CCN(C)C)CC1CCC1 68261,C1(NC(c2ccc(CC)cc2)=O)CN(C(=O)CNS(=O)(=O)CC)C2CCCCC12 68262,N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C2C1 68263,c1(C(N(C2CCN(C(C3(C)CC(C)(C)C3)=O)C2)C)=O)ccc(P(C)(C)=O)cn1 68264,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(Cl)cc2Br)=O)C1)=O 68265,C1(NC(C(C2CC2)NC(CCNC(N)=O)=O)=O)CN2CCC1(C)CC2 68266,N1(C(CC2N(Cc3c(C)cccc3)CCC2)=O)CCc2cc([N+](=O)[O-])ccc2C1 68267,CC1CN(C(=O)C#CC(C)(C)C)CCC1N(C)C(c1cccc(NS(N)(=O)=O)n1)=O 68268,c1(C(=O)NCc2c(CN(C(C(C)C)=O)C3CC3)cccc2)cc2n(n1)CCCC2 68269,N12CCOC(CC1)C2=O.CC(C)CCSCC(=O)N(C1(C(N)=O)CCC1)C 68270,c1(C(N(C2CCCC2)CCNC(c2c(C)[nH]cc2)=O)=O)cc(C)n(C(C)C)c1C 68271,C(=O)(C1=NOC(CN(CC(CC(=O)OC)O)C)C1)Nc1ccc(F)cc1 68272,C1(C(N2CCN(C(c3cncs3)=O)C(C3CCCC3)C2)=O)CC2OC1C1CC21 68273,Cc1cccc(OCC(=O)NC2(CO)CCN(C(=O)CCC#N)C2)c1C 68274,c1(OC)cc(CONC(=O)NC2CC(C)(C)C2)cc(OC)c1OC 68275,C(C(C(=O)N1CC[Si](C)(C)CC1)C(C)(C)C)N(C(=O)COCc1nc[nH]n1)C 68276,C1(NC(c2cccnn2)=O)CC1C1CCCN(C(c2cccc(CF)c2)=O)C1 68277,c1(C(N2CC(C)N(C(=O)CCCC(N)=O)CCC2)=O)cc(N)c2ccccc2n1 68278,C1(OC)CC(CC(=O)NCCN2CCCOCC2)N(C(C2CCC2C(F)F)=O)C1 68279,N1(C(C=CCOC)=O)CC2CCCC2(CNC(=O)CCCCNC(N)=O)C1 68280,c1(C(N2CCCC(N(C)C(C3CCCC3(C)C)=O)CC2)=O)nc2ncccn2n1 68281,N1(C(C2C(C=C)C2)=O)CCC(O)(CNC(C2CCC(N(C)C)CC2)=O)CC1 68282,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3ccc(O)nc3)=O)cc2c1 68283,c1(OCC(=O)NC(CN(C(=O)C(n2ccc(C)n2)C)CC)C)ccccc1F 68284,N1(C(CCCC#C)=O)CCn2cc(C(=O)NCCCCN(C)C(C)C)nc2C1 68285,CC1CC(CNC(=O)C(F)=CC2CC2)CN1C(=O)Cn1cnc(C#N)n1 68286,O=Cc1cccc(CN2CC3(CCC(C(=O)Nc4cc(F)ncn4)O3)C2)c1Br 68287,C1(C(=O)NC(C(=O)NCCC2CC=CC2)C2(C)CC2)(CO)CCCO1 68288,c1(CS(=O)(=O)N(CCC)CCC)cccc(F)c1 68289,N1(C(C2CC(C)(C)NCC2)=O)CC(C)(C)C(O)C1(C)C 68290,C12(NC(C3CCCN3C(C3CC34CC4)=O)=O)CCCCC1C2 68291,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C2=CCSC2)CC(C)(C)C1 68292,C1(CC)(NC(=O)C(c2ccc(C)cc2)N(C)C)CS(=O)(=O)C1 68293,c1(CN2CCC(NC(c3cccc(C(F)(F)F)c3)=O)CC2)c(Cl)cc(Cl)cc1Cl 68294,C(=O)(C1CCCc2cccnc21)NC1CC2(CN(C(C3C(C)=NOC3=O)=O)C2)C1 68295,c1(C(C)OCC)nc(CC(=O)NC(C)CCNC(=O)C(C)Cc2cnn(C)c2)cs1 68296,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68297,CCCCC(C(=O)NC(C1CCCCN1C(=O)CN(C)C)C)C(C)C 68298,n1(CC(=O)N(C(c2ccccc2)CNC(c2cnnn2C)=O)C)nnc(C2CC2)n1 68299,C(CCCCCNC(c1c(Br)noc1C)=O)NC(C(n1ncc(C)c1)C)=O 68300,C(CCCC(=O)OC)(C(=O)NC1CC1)N1CCCC(COC)C1 68301,C(=O)(C(C)(F)C(C)(C)F)NC(CC)CNC(c1ccc(C)cc1O)=O 68302,Cc1cc(C(C)NC(=O)CNC(=O)CNC(=O)CNC(N)=O)c(C)o1 68303,C(=O)(C1CCc2cc(OC)ccc21)NCCNC(CCCOCCC)=O 68304,N1(C(C2C(C=C)OCC2)=O)CCC2(CCCN2CC(=O)NC(=O)NC2CC2)CC1 68305,CC1=CCCN(C(=O)CC2CCCCN2C(C2=CC=N[IH]2)=O)C1 68306,S(=O)(=O)(c1cn(C2CCOCC2)nc1C)N(C)CCc1cn(CCCF)nn1 68307,C(=O)(C(O)CC(C)(C)C)NCC(C)(C(C)C)NC(c1c(C)nn(C(C)(C)C)c1)=O 68308,C1(C(=O)NCCC(=O)NC(CC)C)CCOCC1NC(C1OC2CCC1C2)=O 68309,c1(C(C)(C)NC(=O)NCC2C(C)(C)C2)ccn2c(O)nnc2c1 68310,C(C(COC)C(=O)NC(CO)C(=O)N(C)CC1CCOC1C)OC 68311,c1(C(=O)NC2CC(NC(c3cc(Cl)ccn3)=O)C2)ccc(Cl)cc1F 68312,C12(NC(COCC)=O)CC(COc3ccc(Cl)c(C)c3)(CN1C(C1CC1C)=O)C2 68313,C1(C(=O)NCCC(C(=O)NC)N)CC2CC1C(O)C2O.CCC(=O)CCC=O 68314,C1(CNC(CC2(OC)CCC2)=O)CN(C(C2CCO2)=O)CC12CC2 68315,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(Cc3ccc(Cl)cc3)C2C1 68316,c1(-c2nc(C(C)C)on2)ccc(C(=O)NC2CCCC2C(=O)O)cc1 68317,C(C(=O)NCc1cn(C2CN(C(=O)CC(C)C)C2)nn1)(C(C)(C)C)NC(C)=O 68318,N1(C(C2(F)CCN(C(C(C)C(C)(C)C)=O)C2)=O)CCCCN(C)CC1 68319,c1(-c2occ(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68320,Cc1cc(CCNC(C2CCCC2n2cc(C3CCOC3)nn2)=O)cc(C)c1Br 68321,C1(NC(C2C(OC(C)=O)C2)=O)CN(c2nnco2)C1 68322,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68323,C1(C(N2CC(N3CCN(C(c4nc(C)[nH]n4)=O)CC3)C2)=O)CC(C2CCCC2)C1 68324,c1(N(CCC2N(C(C)=O)CCC2)CCn2cnccc2=O)cc(O)cc(N)c1C 68325,C1(=O)C(OC)CCN1.c1(CCN2CCC(OCC)C2)ccc[n+]([O-])c1 68326,C=CCC(C)C(=O)NC(CNC(c1ccnc(OC(C)CC)c1)=O)CC 68327,N1(C(CC(C)C)=O)CCC2(CCCCC2NC(=O)C(C2CCOCC2)C)CC1 68328,N1(C(C2(C=C)CCN(C(=O)COCC3CC3)C2)=O)CC2CC(C)(C)C2C1 68329,O(C=C(C#N)C(=O)NCC(C)NC(=O)Cn1cncn1)CC 68330,c1(OC)c(CNC2CCN(CCNC(=O)CCN3CCCC3)CC2)cccc1Br 68331,Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(n3cccn3)C2)=O)nc(C)n1 68332,C(C)(CCC(=O)NC1CC1CNC(=O)CC1CC1(C)C)OC 68333,Cc1nc(-c2ccc(C(N3CCC(NCCCO)C3)=O)cc2)nc(O)c1C 68334,CC(=O)CCCC(=O)Nc1cc(-c2cn(CCC(F)(F)Cl)nn2)ccn1 68335,C#CC1CCCC(NC(C2(OC)CCN(C(=O)CC3CCC(O)C3)CC2)=O)C1 68336,N1(C(c2c(CC)c[nH]n2)=O)CC2CCC2(CNC(C23CC(C2)S(=O)(=O)C3)=O)C1 68337,N1(C(C(C)NC(N)=O)=O)CC(CNC(=O)Cn2nccn2)C(c2ccccc2)C1 68338,C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)N(CCCCC=C)C)CC1 68339,c1(C(=O)NCCNC(CC(C)C)=O)ccc2ccoc2c1.C1(=O)CCNCCN1 68340,C1(CCNC(C(CC)(F)F)=O)C(C)CCCN1C(=O)COc1cccc(F)c1 68341,C1(N(C)C)CNC1=O.C1(C(=O)NCCNS(C)(=O)=O)CCCO1 68342,S(=O)(=O)(c1cccc(Br)n1)N1CCCC(C)(C(=O)NCC2CCNCC2)C1 68343,C1(NC(C(CCC)C)=O)CCC12CCN(C(c1c[nH]c(=NC)s1)=O)CC2 68344,C1(NC(C2(OC)CC2)=O)CCCC2CN(C(c3noc4cc(F)ccc34)=O)CC12 68345,N1(C(c2c(-c3c(C)cccc3)noc2C)=O)CC(C)CCC1C(=O)O 68346,CCCCCCC(=O)N(c1cccc(Cl)c1OC)CCCCN1CCCC1 68347,C1(OC)COc2c(C(N3CCCC3CN(C)C(c3scnc3Cl)=O)=O)cnn2C1 68348,O=c1cc(-c2nnc(NC(=O)C3CC3)o2)oc2cc(F)ccc12 68349,Fc1ccc(Br)c(Cn2cc(CCC3CC3)nn2)c1F 68350,c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)Cc3cnccn3)C2)cc1Cl 68351,CC1CC(NC(=O)Cc2ccsc2Cl)CN1C(C1SCCS1)=O 68352,Cc1nc(Cl)nc(N2CC(NC(=O)CC3CCCC(F)(F)C3)CC2C)c1[N+](=O)[O-] 68353,CC(C)(C#N)CCC(=O)NC1(CNC(c2cc3ccccc3o2)=O)CCOC1 68354,C1(CNC(C2CCC(CC)CC2)=O)CN(C(=O)CC(O)C(C)(C)C)CC(C)(C)C1 68355,C12CCC(C)N1C2.c1(-n2c(CC)ncc2)ccc(Br)cn1 68356,c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)cn(C)cc(Br)c1=O 68357,C=CC(C)C(=O)NCC(c1ccccc1)NC(=O)C(F)(F)C1CCCC1 68358,c1(C(=O)NC2CCN(C(C(c3cnccn3)C)=O)C2)cc(Cl)c([N+](=O)[O-])cc1F 68359,CC1=NOC(C)(C(N2CC3C(NC(c4cccc(C(F)F)n4)=O)C3C2)=O)C1 68360,c1(C(c2ccccn2)NC(c2ccc(C3CC3)cn2)=O)ccccc1F 68361,CC1CC(NC(C2(F)CC2c2ccccc2)=O)CCN1C(c1ccc(Cl)cc1F)=O 68362,c1(C(C(=O)NC(C)Cn2cc(CN3CCSCC3)nn2)(F)F)ccc(Cl)cc1Cl 68363,C(C(O)C(=O)NCCCN(CCCNC(=O)C(=O)N(C)C)C)SC 68364,C1(CC)CN(C(C2CC3CC3CC2C)=O)CCN1C(c1ccccc1F)=O 68365,C1(CC(C)NC(C=C(C)C(C)C)=O)CCN(C(c2cc(C3CC3)no2)=O)CC1 68366,CCC(CCCC(=O)NC1(C)CCCC1(F)F)NC(=O)Cc1c(C)ncnc1C 68367,C#Cc1ccc(NC(=O)NC2COCC2C(=O)OC(C)(C)C)cc1OC 68368,C1(CNC(COCC(C)C)=O)CC(F)CN1C(=O)CC1CCCO1 68369,C=CCCCC(C(=O)NCC(C)F)NC(c1cc(C)on1)=O 68370,n1(CC=C)nnnc1C1(NC2CC2c2cnn(C3CCOCC3)c2)CCCC1 68371,c1(C(=O)NCC2(NC(c3n(CC)c(O)nc3)=O)CCCC2)cc(S(C)(=O)=O)co1 68372,c1(C(=O)NCC(=O)NCCC(C)NC(c2cccc(=O)o2)=O)ccc(N)cc1 68373,C(C)(C)(C(C)CC(=O)N1CCC2CC12)NC(C(C)C(F)F)=O 68374,Cn1c(NCC2CC(NC(=O)CN3CC(=O)NC3=O)C2)c(C#N)c(=O)n(C)c1=O 68375,CCCC(C)CC(=O)NCC1(F)CC(NC(=O)CCSc2ccccc2C)C1 68376,C1(CNC(=O)NC2(CC)CCC2)CCN(C(=O)CCOC)C1 68377,Cc1cc(-n2cc(CONC(C3CCCC(NC(N)=O)CC3)=O)nn2)cc(C)c1 68378,C1(NC(c2scc(OC)c2OC)=O)CC2(C1)CN(C(C1CC1(C)C)=O)C2 68379,C1(OC)CCC2(CCN(C(C3(C(C)C)CCN(C(=O)C4=CCOCC4)C3)=O)C2)C1 68380,c1(C(=O)NC(CC(C)NC(C(C=C)CC)=O)C)cccc2ccoc12 68381,c1(COC)csc(C(N2CCC(C(C)(C)NCC3CC3(Cl)Cl)C2)=O)c1 68382,C(=O)(CS(=O)c1ccc(Cl)cc1)NC(C1CN(C(=O)OC(C)(C)C)C1)C 68383,c1(COC)ccc(C(N2CCCC(NC(c3cscc3Cl)=O)C2)=O)cc1 68384,CN1CCN(C(=O)CCc2ccc(O)c(Cl)c2)CC1CNC(=O)CCN1CCC1 68385,C1(CN2C(C(CO)(F)F)CCC2)CC(c2ccccc2)CO1 68386,N1(C(C2(COC)CC=CC2)=O)CC2(CC(NC(=O)CN3CCOCC3=O)CO2)C1 68387,C1(C)(C(=O)OCCc2n(SC)ncc2)CCc2ccccc21 68388,n1(CC)ccnc1C=CC(=O)N(C)CCN(C(=O)C(O)CCSC)C(C)C 68389,N1(C(C(CC)C)=O)CCC(NC(=O)CN(C2CCCC2O)C)C1C 68390,Cc1ccc2[nH]c(-c3cccc4[nH]cc(C(=O)Nc5onc(C)c5Cl)c34)cc2c1 68391,C1(NC(c2n(CC)c(O)nc2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1C 68392,N1(C(C(C)SCCCC)=O)CCC(C)(CCNC(C2CCC(F)C2)=O)CC1 68393,C1(N(C(CCOCC)=O)C)CN(C(=O)CCNC(=O)Cc2ccccc2)CC1O 68394,CON1CC(C(=O)NC2CCCCC2NC(c2c[nH]nc2Br)=O)CC1=O 68395,c1(-n2c(C3CC3)nnn2)ccc2c(c1)CCC2.c12cc(sn1)C(c1occc1)N2 68396,CC1(C(N2CC3CC(C2)C3NC(=O)CCCc2cnn[nH]2)=O)CCNC(=O)C1 68397,C(C)(C)(CCCCC(=O)NC1CCC(NC(c2cscc2OC)=O)C1)OC 68398,C1(CSC)C(=O)N1.C1(CCSCC(=O)S)(C(=O)OC(C)(C)C)CCC1.c1(CO)cccs1 68399,C1(F)(C(=O)NCC2(OC)CCN(C(COCCCC)=O)C2)CCC(C)CC1 68400,c1(C(C(=O)NCC(CNC(=O)C(O)C(F)F)OC)O)cc(F)c(F)c(F)c1 68401,N1(C(c2cncc(C#C)c2)=O)CCC(C(=O)NCCC(=O)NC(C)C)CC1(C)C 68402,c1(SCC(=O)NC(CNC(c2nc(C(C)OC)oc2)=O)C)ccccc1O 68403,C(=O)(C#CC1CC1)NC(c1ocnc1CO)CNC(c1c[nH]nc1OC(F)F)=O 68404,C(=O)(C(C(C)C)NC(=O)CC1CCC(=O)N1)NCC(C#C)(C)C 68405,C(CC1CC1)(CC(=O)O)Nn1cc(CN(C)Cc2ccc(N)cc2)nn1 68406,c1(C(=O)NC(C)(C)CNC(=O)COCCCF)ccc(OCCO)cc1 68407,c1(C(=O)Nc2ncc(-c3cc(OC)ncc3)s2)c(C)cc(Br)cc1F 68408,C1(NC(C(CC)C)=O)CCCCN(C(=O)CCSc2ccc(O)cc2)C1 68409,c1(C(=O)NCCN(C(COc2cn(C)nc2)=O)C2CC2)cccc(C#N)c1Br 68410,c1(CNCC2CC(=O)NC2=O)c(F)ccc(O)c1F 68411,c1(CNC(C(Cc2ccccc2)OC)=O)cccc(NC(C2CC=CCO2)=O)c1 68412,C1(C(=O)NCCCCCCNC(C(Cc2ccccc2)OC)=O)CC2CCC1CC2 68413,C12(C(N(CCC(=O)NCC)C)=O)CC1CN(C(=O)CCCOC(C)=O)C2 68414,C(CC(C(=O)NCC(C)N(C)C(c1ccc(C(F)(F)CF)cc1)=O)OC)OC 68415,CN1CCC(NC(=O)NC2CCCC2O)C1C(C)(C)C 68416,Cc1[nH]nc(Cl)c1C(N1CC(n2cc(NC(=O)CC=C(Cl)Cl)cn2)C1)=O 68417,C1(NC(C2C(CC)CCC2)=O)CC12CCN(C(=O)Cc1ccccn1)C2 68418,N1(C(CC2CC(SC)C2)=O)CC2CCC1CC2NC(c1ncnc(C)c1C)=O 68419,C1(CC=C)(NC(=O)COC(=O)CO)CCCN(C(=O)Cc2cncs2)C1 68420,c1(C(=O)NCC2N(C(C3(COC)CC3)=O)CC(OC)C2)ccc(OC)nc1OC 68421,N1(C(c2c(OC)scc2)=O)CC(CNC(=O)CC2(C)CCC2)C(C(F)(F)F)C1 68422,Cc1cnc(CCCNC(=O)CNC(C2(O)CN(C(N)=O)C2)=O)[nH]1 68423,c1(CC(=O)NC(CNC(C(C)OCCOC)=O)CO)cnccc1C(F)(F)F 68424,Cc1cc(COC(c2ncc(-c3ccncc3)s2)=O)cc2c1CCC2 68425,c1(C(=O)NCC(CNC(c2nc(CCCC)sc2)=O)C)cc(C#N)cn1C 68426,c1(COC(C)C)ccc([N+](=O)[O-])cc1.c12ccccc1-c1cc(ccn1)NC2 68427,C(CC(=O)NCC1CCN1C(C1CC(=C2CC2)C1)=O)(C(F)(F)F)OC 68428,O=C(C1=C(Cl)CCC1)NC(C(N1CC2(CCC2)C1)=O)C1(O)CCC1 68429,CC1CCCN(C(c2ccc(C#N)[nH]2)=O)C1CCNC(c1cccc(CO)n1)=O 68430,C1(C2CC2)(NC(c2c(C)ncs2)=O)CCN(C(c2cc(C)n(C(F)F)n2)=O)C1 68431,C1(CCC)CCCC1C(=O)NCCC(O)CNC(=O)C=CCOC(C)(C)C 68432,C1(C(C(=O)NC(C(=O)OCC)C2CCC2)F)CCN(C(c2conc2C)=O)C1 68433,c1(NC(CN(C(=O)CC2CCC(=O)N2C)C(C)=O)=O)ccnc(Br)c1N 68434,C1(=O)CC(O)C(C)NCC(C)N1CC.c1(C(=O)OC(C)(C)C)cnc(Cl)s1.C(C)=O 68435,c1(C(=O)NC(C2CCCC2)CNC(CCCc2scc(C)n2)=O)ccnc(C)n1 68436,N1(C(C(=Cc2ccccc2)CC)=O)CCOCC(CNC(=O)C=NOC)C1 68437,c1(C2(C(=O)NOCc3ccccc3F)CC(=O)N2)ccc(OC(F)(F)F)cc1 68438,C1(CC(=O)NCCC(C(C)C)NC(=O)C(C)(C)C2CC2)SC2=NCCN2C1=O 68439,c1(NCCCN(C(CCc2onc(COC)n2)=O)C)ncnc(O)c1Br 68440,c1(CC(=O)NC(C2CCN(C(c3cncc(F)c3)=O)CC2)C)ccc(F)cc1F 68441,C(=O)(CC(C)CC(=O)OC)NC1C(NC(C(CC)N(C)C)=O)COC1 68442,c1(C(C(=O)NC2C(OC)CNC2)(C)C)cccc(Cl)c1 68443,c1(N2C(C)CC(CNC(c3csc4ccccc34)=O)C2)ncnc2c1ncn2C 68444,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CCCCC1CC)=O)C2 68445,C12(C(N3C(CN(C)C(c4cnc(Br)s4)=O)CCC3)=O)CCC(C)(C1)OC2 68446,C(C(C)(C)CCCNC(C(F)(F)F)C1CCCCC1)OC 68447,c1(CN(C2CCC(C)CC2)C(=O)C(=O)Nc2cccc(C)c2)c(F)cccc1F 68448,N1(C(C2CCc3nnc(O)n3C2)=O)CCC2C(CCCN2C(c2cc[nH]c2)=O)C1 68449,C(=O)(C(=O)N=c1ncn(-c2cc(Cl)cc(Cl)c2)[nH]1)NC1C(C)C2CCC1C2 68450,Cc1ccc(C2(CNCCn3cc(C(c4cc(C)nn4C)(C)C)nn3)CC2)cn1 68451,C1(N(C(c2ncc(F)cc2F)=O)CC)CCCN(C(=O)COC2CCOC2)CC1 68452,C12(NC(C(C)OC)=O)CCCC1N(C(=O)CC=CC(C)(C)C)CC2 68453,Cn1nc(O)cc1C(=O)NC(C)(C)CNC(=O)Cc1csc(-c2ccoc2)n1 68454,C=C(C)C1OCCC1CNC(=O)CN(C(=O)Cn1ccc(C)n1)C1CCC1 68455,Cc1ccc2c(C(=O)NCC(C)(CO)NC(C34CCCC3C4(F)F)=O)onc2c1 68456,c1(OC)cc(SC)ccc1-c1cc(CN2CCC(C)CC2)ccn1 68457,C(=O)(C(F)(F)F)NCC(=O)N(CCN(C(=O)Cc1cccn1C)CC)CC 68458,C=CC1CN(C(=O)C(C)P(C)(C)=O)CC1NC(c1nccnc1C)=O 68459,c1(C(=O)NCC2CCC(C)N(C(=O)C(=O)N(C)C)C2)cccc2c1ncn2C 68460,C1(NC(CCc2onc(C)n2)=O)COCCN(C(C2COC(=O)N2)=O)C1 68461,N1(C(C2C(COC)CC2)=O)CCCC(O)(CNC(c2cn(C)nc2C(C)C)=O)C1 68462,O=C(NNc1cccc2c1CCCC2)Nc1cccc(-c2ncc[nH]2)c1 68463,c1(CC(=O)NCC(CCC)NC(=O)C(C)(CO)OC)cnc(Cl)cc1C 68464,N1(C(C(CO)OC)=O)CCCC2(C1)CN(C(=O)C(C)=C1CCC1)C2 68465,C12(C(=O)NCC3(CCNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68466,C12(C(=O)NCC3C(NC(C4(CS(N)(=O)=O)COC4)=O)C3)CCCC(=O)N1CCC2 68467,C1(N(C)C(c2csc(O)n2)=O)CCC2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 68468,N1(C(C(c2cccnc2)C)=O)CC(C)N(C(=O)CC(C)(C)C)C(C)C1 68469,C1(CNC(CSCC#C)=O)CC2COCC2N1C(=O)CCCCN(C)C(C)=O 68470,C1(NC(C(CC)NC(N)=O)=O)CC(OC)CN(C(=O)Cc2c(O)ncnc2O)C1 68471,C1(C(C(=O)N(CC(CC)O)C)F)CCN(C(=O)C(F)n2ccnc2)C1 68472,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68473,c1(CN=[N+]=[N-])ccc(C(F)(F)F)cc1.C12(CCCC1)NC(=O)N2 68474,c1(C(=O)NCC=CCNC(C(C)OCc2ccccc2)=O)cccc(Cl)c1Cl 68475,CC(C)CC(CC(C)C)C(=O)NC1(c2ccc(Br)cc2Br)CNC1 68476,c1(SC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3COCC3O)C2)nn1C 68477,c1(CNC(C(C2N(C(C(=O)OCC)C)CCC2)C)=O)nncn1CC 68478,N1(CC)CC(NC(C2C(CNC(c3ccc(=N)[nH]n3)=O)C2(C)C)=O)CC1=O 68479,Cc1ccc(C(=O)NC2CC3CC(NC(=O)Cc4ccc(F)cn4)CC23)nc1F 68480,N1(C(C(C)(Cl)Cl)=O)CCC(CF)(NC(c2c[nH]nc2F)=O)C1 68481,C(=O)(CCCC(F)(F)F)N1CCC(CC(=O)N(C2CCC(F)(F)C2)C)C1 68482,N1(C(c2cn(CC)nn2)=O)CC2CCC1CN2C(=O)CN(C1CC1)CC 68483,N1(C(C(C)(F)F)=O)C(C(=O)NCc2nc(CO)n[nH]2)CCC12CC2 68484,c1(C(N(C2CCN(C(=O)C(O)CC(F)(F)F)C2)C)=O)ncn2ccccc12 68485,c1(CC)cccc2c(C(=O)NC(C)(CNC(=O)CCC(N)=O)CO)c[nH]c12 68486,c1(OC)ncc(C(=O)NC2CCC(NC(c3scc(C)c3Cl)=O)C2)cc1Br 68487,N1(C(C(C)OCC)=O)CC=C(CC(=O)NC2CCN(C3CCCC3)C2)CC1 68488,N1(C(C=Cc2c(C)noc2C)=O)CC2CC(O)C1C2NC(C1CCSCC1)=O 68489,C(C(F)(F)C(=O)NCC1CC(C(=O)NCC(Cl)C(C)(F)F)C1)OC 68490,C1(O)(CC(=O)NCCNC(C2(CN(C(C)C)C)CC2)=O)CCCC1 68491,C1(NC(C2(OC)CC(CF)C2)=O)CC2CC(NC(=O)CCc3nocc3C)CC12 68492,C=CCCC(F)(F)C(=O)N(CCCCNC(=O)CNc1cn2cc(C)nc2s1)CC=O 68493,CC1(C)CC(CC(N2CC3CC2CN3C(=O)Cn2cnnc2O)=O)C(=O)O1 68494,C1(C(=O)NCCc2cc(C)ns2)CCN(C(=O)CC2CCCO2)O1 68495,C=CCCCCCCC(=O)NCC1(NC(c2noc3cc(Cl)ccc23)=O)CCC1 68496,N1(C(C)=O)CC2(C1)CN(C(c1cc(C(N)=O)c[nH]1)=O)C2.c1(C=O)ccco1 68497,C(C(C)(CC(C)C)NC(c1cnc(O)o1)=O)NC(C(CC)(C)C)=O 68498,c1(C(C)C)cccc(NC(=O)CCC2COCCN2C(C2CCCN(C)C2)=O)c1 68499,N1(C(C2CC(OC)C2)C(=O)NC(C)(C)C(F)(F)F)CCCC(SC)C1 68500,S(=O)(=O)(c1c[nH]c(=NCCC#CBr)cc1C)N1C(CCCCC)CCOCC1 68501,CN1CC2CCCN(CCCn3cc(C4CC4)nn3)C2C1 68502,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CCCC2)CCC(CCOC)CC1 68503,CC(C)(C)C#CC(=O)NCC(CC(=O)NCC1OC(=O)CC1(C)C)OC 68504,c1(CNC(C2CCC3CC(C)ON3C2)=O)ccc2c(c1)CN=S2(C)=O 68505,c1(CC(=O)NC(C2CCCN(C(c3ccc(C)o3)=O)C2)C)c(C)cc(C)nc1O 68506,C1(OC)(CNC(=O)CC2CCN2C(=O)C(C)C(C)(C)C)CCCCCC1 68507,C12(CSC)CC(C(=O)NCC(C)CC(=O)NCCCN(C)C)(CO1)C2 68508,c1(CC(=O)N(CC(C)NC(c2csc(C(C)OC)n2)=O)CC)ccccc1C 68509,C1(CNC(C(CC(C)C)F)=O)CCCC2CN(C(=O)C3=CCCOCC3)CC12 68510,N1(C(C2CC3CC(=O)C2O3)C(=O)NCC=C)CCOCC(C2CC2)C1 68511,c1(SC)cccc(C(N2CCC(CNC(c3c[nH]c(Br)c3)=O)C2)=O)c1 68512,C(C)(C)(CCCNC(C1(CCF)CCC1)=O)NC(C(CC)n1cncn1)=O 68513,C1(C)(C(=O)NCCNC(C)=O)CCCN(C(C2(CC(=O)O)COC2)=O)C1 68514,C1(NC(=O)Cc2cnc[nH]2)C2CC1N(C(c1ccc(O)nc1)=O)C2 68515,Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CN2CCSCC2)ccc1O 68516,c1(C(N2CCN(C(C3(CN(C)C)CC3)=O)C3C2C3)=O)c(F)c(F)cc(F)c1F 68517,C(CC(C)C)(CC(C)C)OCCNC(CCN(C(COCC)=O)C)=O 68518,C(=O)(C(CC(C)C)C(N)=O)NC(CC#C)C(N1CCOC(C)C1CO)=O 68519,N1(C(COC(C)=O)=O)CCCC(c2n[nH]cc2NC(c2oc(CN)cc2C)=O)C1 68520,N1(C(=O)CCOC2CCOC2)CCC2CN(C(C3CCC(F)(F)CS3)=O)CC2CC1 68521,c1(OC)ccc2c(c1)C(C)(C)N(C(=O)CCC1(C)N=N1)CC2 68522,CCCCCCC(C)CC(=O)NC1CCN(C(=O)CCC2CC(F)(F)C2)C1C 68523,C1(NC(C(C)CN)=O)CC12CCNCC2.C1(=O)C(c2cccs2)N1 68524,CC(C)(C)CCC(=O)NC1(CO)CCN(C(=O)CC2CCNC(=O)C2)CC1 68525,c1(C(N2CCCN(C(c3c(C)ncs3)=O)CC2C)=O)sc2[nH]cnc(=O)c2c1C 68526,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68527,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68528,C(CN=[N+]=[N-])N(C(C1(CNC(=O)C=C2CCC2)CC1)=O)CC 68529,c1(C(CC)(C)C)cccc(N(C(=O)C(N2CCCC(COC)C2)=O)C)c1 68530,c1(C(=O)NC(C(=O)N(CCOC)CCO)CC2CC2)cccc2c1OCC2 68531,CCC(C)C(CC(=O)NC1CCCSC1)NC(=O)Cn1ccnc1 68532,N1(CCN(C2CC3CS(=O)(=O)CC3C2)OCC)CCC2(CC1)CC2(C#N)CO 68533,c1(CNCCC(CCC)(C)C)cccc2c1CC(=O)N2 68534,C1(CNC(C=CC(C)C)=O)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 68535,C=CCC(C(=O)NC1(C)CC(NC(C2CC2c2ccc(F)cc2Cl)=O)C1)C(C)C 68536,N1(C(CC=C)=O)CCC(O)(C(C)NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 68537,C(C(O)C(F)(F)F)N(C(C1C(CNC(c2cc(C)[nH]c2)=O)C1(C)C)=O)C(C)C 68538,c1(OCC)cc(CC(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 68539,CC(C)C1=NOC(C(=O)NC2COCC2C(=O)NCC23CCC(CC2)O3)C1 68540,C(=O)(CCCCCCOC(CCC=C)=O)N.CCCO 68541,C1(NC(c2c(CC)noc2)=O)CCCC12CN(C(=O)CCc1cnco1)C2 68542,C(=O)(C(CNC(c1ccsn1)=O)CC(C)C)NC(c1nc[nH]n1)CC 68543,c1(-c2c(C(=O)NCC#CC)cccc2)ccc(SC(C)C)c(F)c1 68544,N12CC(C3(CCC3)C1)C(=O)NC(C(=O)OCC)C2=O.n1(CCOC)cnnc1 68545,Cc1nc(O)[nH]c1C(=O)NC(C)CNC(=O)Cc1ccsc1C 68546,CC1CN(C(c2ccccc2C)=O)CC1NC(=O)CN(S(C)(=O)=O)C.CC(F)F 68547,c1(C(N(C2CCCN(C(CCN(C)C)=O)C2)C)=O)ccc([Si](C)(C)C)s1 68548,C1(C(N2CC(CNC(C3(CC)CCOC3)=O)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] 68549,N1(C(CCOCCN(C(c2c(OC)nn(C)c2)=O)C)=O)CCC(C)(C2CC2)C1 68550,C=CC(C)(O)CC(=O)N(CC(=O)NC(c1ccccn1)CC)CC 68551,N1(CC)CCN(C(c2ccc(F)cn2)C(=O)NCC(=O)OCC2CCOC2)CC1 68552,CCN=C(NCc1ccc(CCCCC)o1)N1CCC2CCCOC2C1 68553,C1(CNCC(C)CNC(c2ccco2)=O)CC2CCCC(C1)C2 68554,C(CCCC(=O)NCC1(C(=O)Nc2conc2C)CC12CCC2)OC 68555,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 68556,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)Cn1nnnc1C)C2 68557,N1(C(C(=O)NCC2CC2)=O)CCC2CC12C(N1CCN(CCF)CC1)=O 68558,c1(C(C)=O)ccc(C(=O)NC(C2CCCN2C(=O)Cc2cc(C)no2)C)cc1 68559,C1(C(=O)NC2CCN(C(C3COC(=O)O3)=O)CC2)CCc2ncncc2C1 68560,C1(NC(C(c2cn(CC)nc2)(F)F)=O)CC(C)N(C(=O)CSCCOC)C1 68561,C1(C(=O)NC(C2N(C(C(=CC3CCCC3)C)=O)CCC2)C)CCCCCS1(=O)=O 68562,C1(NC(C(CC)Br)=O)CC(N=c2cc(C)nc(OC)[nH]2)C1 68563,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(c1cc(C(N)=O)[nH]n1)=O 68564,c12ccc(Cl)cc1NC2=O.Cn1cc(COCc2cn(CC(C)(C)C)nn2)cn1 68565,c1(C(=O)NCCCC2(NC(CC=C=C)=O)CC2)cccc2c(C)[nH]nc12 68566,C1(NC(=O)NC(c2ccc(Br)cc2)C)CCCN(C(=O)C(Cl)Cl)CC1 68567,C(=O)(C1=CCCCO1)N(C1CN(C(C(F)=CC)=O)CC1O)C 68568,C1(OC)CN(C(C23CC(C2)C3)=O)CCC1NC(c1cc(B(O)O)co1)=O 68569,N1(C(C(C=C)O)=O)CCC(C(=O)NCC(O)CC2CCC2)(CO)C1 68570,CCCC(C(O)C(=O)NC1CCC(C)CC1)NC(=O)C(C(C)CC)N(C)C 68571,N1(C(C(=O)NCCC(=O)NC(C)C(=O)NC2CC2)C2CC2C)CCC(C2CC2)CC1 68572,C12(C(N3CC(C)C(CNC(=O)Cc4cnc[nH]4)C3)=O)CCC(CF)(C1)OC2 68573,C1(CNC(c2c(CC)ccs2)=O)CCN(C(c2oc(C)cc2C)=O)CC1CC 68574,N1(C(C(c2ccc(C)cc2)=O)=O)CCCC(NC(c2cnn[nH]2)=O)C(F)C1 68575,C1(C)(C(N2CC(OCCC(=O)N(c3cc(C(N)=O)co3)C)C2)=O)CCCCCC1 68576,c1(C(=O)NCC(=O)N(CC(CCC)C)C)nccnc1OC 68577,C1(CC(=O)NCCCOC=C)CCN(Cc2cn(C)nn2)C1 68578,CCCCCCC(=O)NC(CCOCC)C(=O)N1CCC(CC2CC2)C1 68579,c1(CC)c[nH]nc1C(=O)NCC(C1CC1)N(C(=O)CCN1CCC(F)C1)C 68580,Cc1ncc(CC(=O)N(C(C)CN(C)C(c2sccc2C2CC2)=O)C)s1 68581,c1(C(=O)NCC(c2ncc(C)o2)N2CCOCC2)ccc(F)c(F)c1 68582,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2cnnn2C)=O)CC1C 68583,C1(C(=O)NC(CNC(C2(C#N)CC(C)(C)C2)=O)CO)CSc2ccccc2O1 68584,N1(C(C(CCC)CC(C)C)=O)CCC(C2(O)CCN(C(=O)CNC(=O)NC)C2)CC1 68585,C1(C(=O)OC)CCCCCN1C(C(=O)NC1CC1)C1CC1 68586,c1(C(=O)OCC(O)Cc2cn(CCCN(C)S(N)(=O)=O)nn2)ccc2c(c1)CCO2 68587,N1(NC(C2C(NC(c3ccc(C#C)o3)=O)CCCC2)=O)CCCCC(C)C1 68588,C1(C(=O)NCCC(C(=O)N(C)C)C)CC(C)(C)CN1C(C1CCC1)=O 68589,C(CCC(C)CC(=O)N1CC(NC(C2CCOCC2)=O)C2CC2C1)=C(C)C 68590,C1(CCNC(c2c(CC)onc2)=O)CN(C(=O)C(c2cccc(C)c2)C)CC1C 68591,C1(CC2(c3ccccc3C)CC2)CN(C(=O)CCn2cc(SCC)nn2)CCO1 68592,N1(C(Cc2c(SC)ccc(F)c2)=O)CC2(CCCC(CNC(C3(O)CC3)=O)O2)C1 68593,C1(NC(c2nc(C)c(C)s2)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1O 68594,C1(c2nnnn2C2CC2)(NCC(COC)SC)CSC(C)(C)C1 68595,CSC1=C(C(=O)NCC2CN(C(C3COC(=O)C3)=O)CCN2C)CCCC1 68596,c1(N2CC3C(CN4CC(C(N)=O)(CC)C4)C3C2)nc(Cl)nc(C)c1[N+](=O)[O-] 68597,C1(CC(NOCC(=C)C)=O)COCCN1C(=O)Cc1cn(CC)nn1 68598,C1(c2cn(C)nn2)C(C(=O)NOCc2ccc(-n3cnnn3)cc2)CC(=O)N1C 68599,N1(C(C2N(C(C)C)CCC2)=O)CC(CNC(=O)Cc2csnn2)CC1(C)C 68600,c1(CCCC(=O)NCC2(O)CCN(C(=O)C3CC3)CC2)c[nH]c2ccccc12 68601,C1(NC(c2cn3ccnc3s2)=O)CN(C(=O)C=CC2CCC2)C2(CCCOC2)C1 68602,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC(C)n3cccn3)=O)CC1C2 68603,C(=O)(C(C)(C)CC(F)F)NCc1cncc(C(=O)NCCC(C(=O)OC)C)c1 68604,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 68605,c12ccc(cc1)C(=O)NC2.C1(CCOC)(N(C)C)CCOC1 68606,c1(C(=O)NC2(CNC(=O)CC3COCC3O)CC(OC)C2)nccc2ccn(C)c12 68607,N1(Cc2cn(CC)nc2)CCOC(CC(=O)Nc2cncc(OC(F)F)c2)C1 68608,C1(O)(CCNC(c2ccc(Cl)cn2)=O)CCN(C(C2CCC2CF)=O)CC1 68609,Cc1cc(=NC2CC(C)N(CC(C)Cn3cccn3)C2)[nH]c(C(F)(F)F)n1 68610,CC1(C)CN(C(CC23CCC2CN(C(=O)CC2CCOC2=O)C3)=O)CCC1O 68611,C1(C(N(C2CCN(C(c3cc(C(C)OC)on3)=O)C2)CC=C)=O)CCCC1CC 68612,CN(C)S(=O)(=O)NCC(=O)OCCN(C)C.C1(C)(C)CCCN1c1nccc(O)n1 68613,c1(OCC(=O)NC2CC(CNC(C(C)Cn3cccn3)=O)C2)ccc(Cl)c(F)c1 68614,c1(-c2cnc(-c3nc(C)nn3C3CCOC3(C)C)nc2)ccc2c(c1)OCO2 68615,C(C(C(C)C(C)C)NC(C1(N2CCOCC2)CCCC1)=O)NC(CC1CC(=C)C1)=O 68616,CCC(C)CCC(=O)NCC(O)C(=O)NC1(CC)CCOCC1 68617,c1(C(=O)Nc2ncccc2C2CCOCC2)cccc2c1C1CCC2O1 68618,C(=O)(C1CCc2ccccc21)N1CCC(C)(CNC(CCC(C)(C)O)=O)CC1 68619,N1(C(C=CCOCCOC)=O)CCN(C(C2CC23CCC3)=O)CC(CO)C1 68620,Cc1cccnc1C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cncs1 68621,N1(CC(N2CC(=C(CNC(C3C(C(C)(C)C)C3)=O)F)C2)=O)CC2CCC1C2 68622,C(=O)(C(CC(C)C)C(C)C)N1CC(CCCC)N(C(=O)C(C)N2CCCC2)CC1 68623,C1(CCOC)CCCN(C(CC2CCCCN2C)C(=O)NCc2ccccc2)C1 68624,N1(C(C(CC)C)=O)CCC2(CCCN(C(c3ccc(OC)c(OC)c3)=O)C2)C1 68625,Cc1nccc(C(N2CCCC(NC(C3CC(C4CCC4)C3)=O)C2)=O)c1N 68626,c1(CN2C(C(N3CC4(CCC4)C3)=O)CCC2)c(O)cccc1F 68627,N#CCCCCCNC(=O)CC1(CNC(c2ccncc2O)=O)CC1 68628,C#CCC(CC(F)F)NC(C1(C)CN(C(c2cncc(OC)c2)=O)C1)=O 68629,C1(CCNC(C2N(C)CCCC2)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 68630,c1(C(N(CC(C)NC(c2cncc(OC)c2)=O)C)=O)cn2nccc2nc1C 68631,c1(C(N2CC(F)(C(=O)NC3(C)CC(O)C3)C2)=O)cc(C#N)ccc1N 68632,CON=Cc1ccc(C(=O)NCC(C(C)C)NC(=O)CC2CCCC23CC3)cc1 68633,c1(OC)ccc(C)cc1C(N1CCC(CNC(=O)C(C)c2ccsn2)C1)=O 68634,c1(C(N2CC(CCCCNC(C3C(=C)C3)=O)C2)=O)ccc(=O)n(CCOC)c1 68635,Cc1[nH]c2ccc(F)cc2c1C(=O)NCCNC(=O)CCCc1ccc(F)cc1 68636,c1(CC(N2CCC(=C(C)C#N)C2)=O)ccc2c(c1)OCO2.C1CCC(=O)NCC1 68637,c1(C(N2CCC(O)(CNC(Cc3nn(C)c(Cl)c3)=O)C2)=O)cc(N)cnc1Cl 68638,CC1CCCc2nc(C(N3CC(CCNC(=O)CNC(=O)C(C)(C)C)C3)=O)cn21 68639,C1(NC(Cc2c(OC)ccnc2)=O)CC(O)CN(C(=O)CSc2cnn(C)c2)C1 68640,N1(C(CC2(OC)CCC2)=O)CCC2(NC(c3cccc(=O)o3)=O)CC2C1 68641,C1(C(=O)NC(CC)CN(C(=O)CCC2(C)CC2)C)CCN(c2ncccn2)C1 68642,C1(CC(N2CCC(N(C(=O)CCSCC)CC)C2)=O)CCc2ccccc2C1=O 68643,C(=O)(CCCCCC#N)N1C(C)CC(CCNC(=O)CCC(N)=O)CC1 68644,C(=O)(CCCN=c1nccc[nH]1)N(C)CC1CN(C(c2csc(Cl)n2)=O)CCO1 68645,Cc1ncnc(C(=O)NC2CCC(NC(c3cc(C(C)(C)C)ccn3)=O)C2)c1C 68646,C(C(=O)NCC(C)(CO)NC(c1ccc(NC(C)=O)s1)=O)(C(C)(C)C)SC 68647,c1(C(=O)NCC(NOCC)=O)cccnc1CNC(=O)Cc1ccc(C)o1 68648,Cc1cc2ncc(C(N3CCC(C)C(NC(c4nonc4N)=O)C3)=O)c(C)n2n1 68649,C(=O)(N1CC(O)CCO1)C1CCN(C(C2(C)C=CCCC2)=O)C1 68650,c1(C(N(C)CC2CN(C(=O)CCOC3COC3)C2)=O)ccc(Cl)c(F)c1 68651,C(N=c1ccc(S(=O)(=O)NC2(Cc3cccnc3)CC2)c[nH]1)c1nc(C)sc1 68652,c1(C(N2C(CC)COCC2)=O)cc(C)cc2ccoc12.n1(CC(=O)OC)cc(CN)nn1 68653,N#Cc1ccc(C(N2CCCCC2)NC(=O)C(F)(F)F)cc1O.N12CCC1NC2=O 68654,c1(C(N(C(C)CN2CCSCC2)C)=O)cc(Cl)cc([N+](=O)[O-])c1 68655,C(=O)(C(CC1CCOCC1)C(F)(F)F)NCCNC(=O)CCc1ccoc1 68656,c1(CNC(NCC2C(C)C2)=NCC23CC(C(N)=O)(CO2)C3)ccc2c(c1)OCC2 68657,CC1CC=C(C(=O)NCCCC2CCCN2c2nn(C)cc2[N+](=O)[O-])CC1 68658,c1(N(C)CC)ccc(F)c(C(=O)NC(CNC(=O)CCc2cnn[nH]2)CC)c1 68659,c1(NC(=O)OC(C)(C)C)c(F)ccc(SC2CCCC3(CC3)C2)c1F 68660,C(C(C(C)C)NC(=O)CCC1CCCN1)N(C(CC)=O)CC 68661,C1(C(=O)NCC#CCNC(c2c(OC)cc(C)cn2)=O)CCCC1S(C)(=O)=O 68662,c1(C(N(CCCCNC(C2C(C)CCC2)=O)C)=O)nn(C)cc1N 68663,N1(C(C(C)SCC)=O)CCN(C(c2cnn(CC)c2)=O)CC1COC 68664,C1(NC(CC)=O)CCC2CN(CC(=O)NC3CC3c3cccc(Br)c3)CCC2C1 68665,c1(C(C)(C)C)cc(Br)cc(Br)c1C(=O)NCc1n[nH]cc1C(N)=O 68666,C=CCCCC(C(=O)N(C)Cc1ocnc1C)NC(=O)CN1CCN(C)CC1 68667,Cc1ccc(SCCC(=O)NC2CCN(C(C3CC3C(F)F)=O)C2C)cc1C 68668,c1(C(N2Cc3ncsc3C2)C(=O)NCCOC)cc2ncccc2o1 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68755,c1(C(N(CC(C)NC(=O)CCCC#N)C)=O)ccc(-n2cccn2)cc1 68756,c12ccc(cc1Cl)S(=O)(=O)N2.C1(CNC2CCC(C)CC2)Cc2ccccc2CO1 68757,c1(C(=O)NCCC(C)N(C(=O)CC2CCN(C)C2=O)C)cc(N)c(F)c(F)c1F 68758,c1(OC)cc(OC)c(CNC2CC=CC(C(N3CC4CC4C3)=O)C2)cc1OC 68759,Cc1nc(-c2ccc(C3CCC3)cc2)ccc1C(=O)NCCOc1ccccc1 68760,N1(C(c2cn(CC)nc2C(C)C)=O)CC(C(=O)O)OC(C)C1 68761,C(C)(C)(CC(=O)NC(CNC(=O)Cc1ccno1)CC(C)C)OC 68762,c1(C(C)=O)c(Cl)nc[nH]c1=NCC1(F)CC(NC(c2cc(Br)c[nH]2)=O)C1 68763,c1(C(=O)NCC(C)N(C(=O)CCc2ccc(N)c(F)c2)C)ccn2nnnc2c1 68764,C#CC(C(C)OC)NC(C1(C(C)C)CC1)=O.C12CC(C1)CNC2=O 68765,CC(CCCCC1CC1)(c1nnnn1CCC1CC1)NCCCS(=O)(=O)C(F)F 68766,C1(CCNC(COC)=O)CCCCC1OC1CN(C(=O)Cn2ccccc2=O)C1 68767,C1(C(C)C)CN(C)CCN1N1CCCCC1c1cn(CCN(C)C)nn1 68768,c1(C(N2CC3CC(C2)N3Cc2n[nH]cc2Cl)=O)ccc2nc(Br)sc2c1 68769,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)(NC(=O)CCS(N)(=O)=O)CC1 68770,Cc1cc(C)c(C=O)[nH]1.N12CCCC1CCC(=O)NCC2=O.C(C)(C)(C)O 68771,c1(C(N2CC(CC(C)NC(=O)CC3CCC3)C2)=O)ccn(CCO)c(=O)c1 68772,C1(O)(CCNC(c2c(COC)csc2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 68773,C(C)(C(CCc1ccccc1)NC(c1[nH]cc(C)c1C)=O)NC(CCSC)=O 68774,C(N=c1[nH]c(N2CCC(S(N)(=O)=O)CC2)nc2c1SCC2)C1(OCC)CCOC1 68775,N1(c2n(CC(C)C)c(-c3cc4c(s3)CCOC4)nn2)CC2OCCN(C)C2C1 68776,N1(C(C2(CNC(CSCCC#N)=O)CC23CCC3)=O)CC2C=CC1CC2 68777,N1(C(C2(COC)COC2)=O)CCC(C(=O)NCCCOC2CC2)CC1 68778,C(=O)(C#CC1CCOCC1)NCC1N(C(C(C)CSc2ccccc2)=O)CCC1 68779,C1(C(=O)NCCOCCC2(NC(CC3(C#N)CC3)=O)CC2)CC12CCCC2 68780,C(C)(CCC(=O)NC(CNC(=O)C(C)(C)c1cnc[nH]1)CO)OC 68781,C1(NC(C2C(CNC(CS(=O)(=O)NC)=O)C2)=O)CCC2CC2CC1 68782,N1(C(C(CC)N(C)C)=O)CCN(C)CC1CNC(c1ccc(CC2CC2)o1)=O 68783,n1(CC)nc2c(c1C(N1CC(NC(=O)C(O)C(C)C)C(C)C1)=O)CCCC2 68784,N1(C(C(C)=C(C)C)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C(C)C1 68785,CN1CC(C(=O)NCCNC(=O)C(C)(C)CF)CCC1C(F)(F)F 68786,C1(CC(N2CC(C)(NC(C(COC)C)=O)C2)=O)CCCS1(=O)=O 68787,C1(C)(C(=O)NC)CCN(C(=O)C(O)C(C)(C)C)CC1.C1(C)(CCC=O)CN(C=O)C1 68788,CC(C)C(C(=O)NCC(C)N(C(=O)C(F)C1CCOC1)C)n1ncc(N)n1 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68806,N#Cc1ccccc1-c1cccs1.N1(C(C2CC2)=O)CCC(F)(F)C1 68807,C(=O)(CCCN=C(NC1CCCC1(F)F)N1CC2CCN(C)C2C1)NC 68808,C(=O)(CCC1CCc2ccccc21)NC1C(CNC(=O)CCCCF)COC1 68809,C(CC(C)C(=O)NCC(c1ccc(-n2cc(NC(N)=O)nn2)cc1)SC)OC 68810,N1(C(CC=CCC)=O)CC2=C(C1)CN(C(c1cccc(CSC)c1)=O)C2 68811,c1(C(=O)NCC2C(NC(C3(OCC)CCC3)=O)CCC2)cccnc1S 68812,C(=O)(C(CC)C(C)C)N1CC(CNC(c2c(SC)cnn2C)=O)C(O)C1 68813,c1(CC)ccc(C(=O)NC2COCCC2NC(=O)Cc2ccc(C)cc2)c(O)c1 68814,c1(N2C(C)CC(CNC(CCOc3ccc(C)cc3)=O)C2)ncc(F)c(C)n1 68815,C12(C(N3CCC(C)(C)C3)=O)CCC(CN(C(=O)CC3CCCO3)C1)C2 68816,N1(C(CCCC#C)=O)Cc2ccccc2C(CNC(c2cnoc2C)=O)C1 68817,Cc1ccc(C(N2CCC(NC(=O)C(O)P(C)(C)=O)C(O)C2)=O)c2ncccc12 68818,N1(C(c2c(O)nc(CC)c(C)c2)=O)CC2(CCCC2NC(=O)C(CO)C(C)C)C1 68819,c1(C(=O)NCC(C)(Cn2cccn2)NC(C2C=CCC2)=O)cnnc(O)c1 68820,C1(NC(CN(C2CC2)CC)=O)CCC2CN(C(=O)COC(C)=O)CC12.C1(O)CCCCC1 68821,N1(C(C2CC(OCC)C2)=O)CC2(C1)SCCC2NC(c1cc2ncccc2o1)=O 68822,c1(N2CC(C#N)C(C(N)=O)C2)c(-c2ccccc2)[nH]c2ccccc12 68823,CC(C)C(F)C(=O)N(C(C)CNC(C1(Cc2nc[nH]n2)CCOCC1)=O)C 68824,CC1CCC(C(=O)NCC(=O)Nc2ccccn2)CN1C(C1C(C)(C)C1(C)C)=O 68825,C12(C(=O)NCC=C(C)C)CC(CO1)N(C(c1cccc[n+]1[O-])=O)C2 68826,c1(C(=O)NCCN(C(C23CCCCC2C3)=O)CC)c(O)nnc(C)c1C 68827,C1(NC(c2ccc(C(F)F)c(F)c2)=O)CC2CN(C(C3CC4CCCC34)=O)CC12 68828,C12(C)CC(C1)N(C)CCCCO2.C=C1C(C(=O)NCC)C1C(=O)NC 68829,c1(N(CC(F)(F)F)CC(C)OCC)c[nH]c2ncccc12.C(C)(C)(C)O 68830,C(C(C)C(C)C(=O)N1CC2C(CC(=O)NCc3cccc(F)c3O)C2C1)OC 68831,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CCNC(c2n[nH]c(C)n2)=O)C(F)(F)C1 68832,c1(CCSCC(=O)NCc2nnc(CC)n2N)nn(C)cc1[N+](=O)[O-] 68833,Cc1cc(C(=O)NCC2(CO)CN(C(=O)CCc3nnc(C)n3C)C2)c(C)cn1 68834,N1(C(C(C)CC2CCCC2)=O)CCC(CC(N)=O)(NC(c2cnn[nH]2)=O)CC1 68835,c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccc(-c2nc(=O)o[nH]2)cc1 68836,c1(C(=O)NCc2csc(Cl)n2)cc(C2=CCSC2)cc2cc[nH]c12 68837,Cc1ncc(C(=O)NCC2(NC(C3CN(C)C(=O)N3)=O)CC2)c(C2CC2)n1 68838,CCCCCCC(=O)NC(C)CCN(C(=O)C(C)OCC)C 68839,Cc1cncc(C(N2CCC(NC(C34CCCC3C4(F)F)=O)C(O)C2)=O)c1Cl 68840,C1(C(N2CCCC(CC)(NC(=O)C3=COCC3)C2)=O)CCCCCS1(=O)=O 68841,C1(CC)CN(C(c2cnsc2C)=O)CCC1NC(=O)C(C1CCOCC1)O 68842,N1(C(=O)NC(CC)C2CCC2)CC(C)(C)OC2COCC12 68843,N1(C(c2cnc(COC)s2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 68844,c1(NC(c2n(CCOCC)nnn2)c2scnc2Br)ccc2nc(C)ccc2c1 68845,c1(C(C(=O)NCCCSC)N(C(C)COC)C)cc2n(n1)CCC2 68846,c1(CC(=O)N(CCCN2CCC2C(=O)OCC)C)cc(Cl)ccc1Cl 68847,C1(C(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)(C)C)CCC2(CCC2)CO1 68848,C1(OCC(=O)NC(C2CN(C(C3C(C)C3C)=O)C2)C)CCCCCC1 68849,c1(OC)ccc(CCCNC(=O)CCNC(N2CC(CCO)(OC)C2)=O)cc1 68850,n1(CCOC2COCCO2)nc(-c2ccccn2)nc1NC(=O)COC1CCC1 68851,c1(C(N(C)C2CC2)=O)cccc(NC(=O)CC2OCCC2(C)C)n1 68852,c1(C(N(C2CN(C(=O)CC(F)(F)c3ccccc3)C2)C)=O)nccc2ccsc12 68853,CC1(C)CCC(C(=O)NC2CC(=O)NC2=O)CN1C(C1CCCCS1(=O)=O)=O 68854,C1(NC(C=CCN(C(=O)C(C)=O)C)=O)CC1C.C(CO)(C1CCC1)N 68855,C(C(CC(C)C)C(=O)N1CC(C(C)NC(=O)C(C)(C)C(C)O)C1)OC 68856,C1(NC(C2C(CC)CCO2)=O)CCCCC1NC(c1ccc(CN(C)C)cc1)=O 68857,C(=O)(C(C(C)CC)N(C)C)N1C(CN(C(COCCCC)=O)C)CCCC1 68858,C1(NC(COC(C)C)=O)CCC(C)(CNC(c2ccnc(C3CC3)c2)=O)C1 68859,C1(CCC)C(=O)NCC2(O)CN(C2)C(=O)C(C)OCC=CC(=O)N1.C(C)(C)(C)OC 68860,Cc1c(CCNC(C2(C)C=CCN2C(=O)C2=NOCC2)=O)cnn1C 68861,c1(C(N2CC(C)(NC(c3cccc(CC)c3)=O)C2)=O)ccc2cc(C)ccc2c1 68862,CC1CCN(C(=O)CC(=O)NC2CCC2)C1CNC(c1csc(CCN(C)C)n1)=O 68863,N1(C(C(CC)O)=O)CCC2(CCCCC2NC(c2ncc3c(F)cccn23)=O)C1 68864,N1(C(C(=O)N(C)CC2CCC2)=O)CC2COCC(O)CC2C1 68865,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCC(=O)NC(CCCC)CO)CC 68866,C1(COC)(CN(c2coc(C3CCCCC3)n2)C)CCN(C(=O)C(C)CCO)C1 68867,N1(C(CC(C)(C)C)C(=O)NCc2cccs2)CCn2c(Br)cnc2C1 68868,c1(C(N2CC(OCCNC(C3C(C=C)C3)=O)C2)=O)cccc(OCC2CC2)c1 68869,C(=O)(C1=C(CC)OCCC1)N1CC(NC(CC(=O)NCC#C)=O)CN(C)CC1 68870,C1(C(=O)NC(C2CCCC2)CC2(C#C)CC2)CCC(CNC(c2ccco2)=O)C1 68871,N1(C(Cn2c(C)ccc2C)=O)CCN2CCN(C(=O)C(O)C(C)(C)C)CC2C1 68872,C1(C(C2CCSC2)N(C(=O)C(=O)NC2CC2)C)CCCCO1 68873,Cc1nc2cc(NCc3ccc(-c4cnc(C(C)(C)C)nc4)s3)ccc2o1 68874,C1(OC)CN(C(=O)CC2(NC(C)=O)CC2)CC1C(N1CC(CC2CC2)C1)=O 68875,C1(NC(C2C(C)CCCC2)=O)CC2CCC1N(C(=O)CC(O)CN(C)C)C2 68876,c1(C(=O)NCCN(C(=O)CCCOc2ccccc2F)CC)cc(F)ccc1C 68877,c1(C(N2CCN(C(C3CCC(C)(C)CC3)=O)C3C2C3)=O)cccc2nn[nH]c12 68878,C=C(C)CCCC(=O)NCC(C)(C)OCC(=O)N(C)Cc1ccccc1F 68879,CCC(CC(=O)N(CCCC(=O)NCC1C=CCCC1)C)CC(C)C 68880,C=C(C)CC(C)C(=O)NCCc1ocnc1CNC(=O)CN1CCCCCC1=O 68881,C1(C(N2CC(C(C)NC(c3ccccc3Br)=O)C2)=O)CCc2ncncc2C1 68882,C1(C(=O)NCCC(CNC(C(C)=CC2CC2)=O)C)CC(=O)CCO1 68883,c1(OCC)ccc(C(=O)NCCN(CCOC)C(C2CC2F)=O)c2[nH]ccc12 68884,c12ccc(c(C)c1Cl)CS2.n1(CC)c(C)cc(-c2csc(-c3ncno3)n2)c1C 68885,CC(CC(C)(F)F)C(=O)N1CC(CNC(=O)CCC(F)(F)F)CC1(C)C 68886,C(=O)(CC(C)(F)F)N1CCC(n2cc(CNC(CN(c3ncccn3)C)=O)nn2)C1 68887,CC(=O)CCCC(C)C(=O)N1CC2CCCC2C1C(=O)NCCC(F)C1CCC1 68888,c1(C(N2C(C3CCN(C(c4cc(C)[nH]c4)=O)C3)CCC2)=O)cccc(C(F)F)c1 68889,N1(C(c2cc(C)[nH]c2C)=O)CCCC(NC(C2CCCC(C#N)C2)=O)CC1 68890,C(C)(CCN=c1[nH]c(Cl)ncc1C)NC(c1cccc(OC)c1[N+](=O)[O-])=O 68891,N1(C(COCCC#C)=O)CC=CCC1C(N1CCN(C2(C)CC2)CC1)=O 68892,c1(C(=O)NC(c2ccccn2)C(=O)OCC)ccc(C2CCC(=O)N2)cc1 68893,C(=O)(C(O)C(C)(C)C)NCC(c1cccc(CC)c1)NC(c1sccc1C#N)=O 68894,c1(CC(N2CC3C(NC(c4ncc(C)nc4)=O)(C3)C2)=O)ccnc(Cl)c1F 68895,C1(OCC(C)C)CCN(C(=O)C(C2CCCO2)NC(c2nccn2C)=O)C1 68896,C1(C(=O)NCC(C2CCC2)OCC)CCN(C(=O)CC(CC)C(F)F)CC1(C)C 68897,N1(C(C=CCOCCOC)=O)CCOC2(C1)CN(C(C1(C)CCCNS1(=O)=O)=O)C2 68898,N1(CCC#C)CCC(C(=O)ON2CCN(C(C3CCO3)=O)CC2)CC1 68899,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(NC(C2CC(C(=O)OC)C2)=O)C(CO)CC1 68900,C1(NC(C=CC2N(C(Cc3cc(CC)no3)=O)CCC2)=O)CCC2CC2CC1 68901,C1(NC(CCc2cc(C)ncc2)=O)CCCC12CN(C(c1coc(C)n1)=O)C2 68902,CC(C)C(C)C(=O)NCCC1CN(C(c2ccc(NC(N3CCC3)=O)o2)=O)C1 68903,CCC(C)(C)C(C#N)C(=O)N1CCCC1CCNC(C1(F)CCC1)=O 68904,C(=O)(C#CC1CCC1)NCC(C)C(=O)NCC1C2CCCC12 68905,CC1CC2(CCN(C(C(=O)NCCC#N)c3cnc[nH]3)CC2)CN1C(C1CCC1)=O 68906,n1(CC(=O)N(CCCCN(C(CCOCC)=O)C)C)nncc1-c1ccccc1 68907,c1(N2CCN(C(C(=O)N(CCCOC)CCO)=O)CC2)ccc(C)c(F)c1 68908,C1(C(N(C(C)C)CCN(C(=O)CC2OCCO2)C)=O)CCC2(CCCC2)C1 68909,N1(C(CC2C3CN(C(c4n(C=C)nnc4)=O)CC32)=O)CCCCC(C)C1 68910,C#CC1(OCC(=O)NCC(C)NC(=O)C(c2cnn(C)c2)=O)COC1 68911,C1(N(C)C(C23CCC2C3)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 68912,CCCCCC(O)CC(=O)N(C(CC(F)F)C(=O)NCC1=CCSC1)C.NC 68913,c1(NCC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCCSC(C)C2)c(Cl)c1 68914,C1(CC#C)(NC(=O)CCCNC(C)=O)CCN(C(=O)CCCOCCOC)C1 68915,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(C1NC(=O)CC1C(F)(F)F)=O)C2 68916,C(c1cnn(-c2ccccc2)c1)=CC(=O)NC1CN(C(C2N(CC)CC2)=O)C1 68917,C1(NC(=O)CCc2ncc[nH]2)CN(C(=O)CN2CCCCC2=O)CC1SC 68918,c1(CNC(CCc2cccc(N)c2)=O)cc2c(cc1O)OCO2 68919,N1(c2ccnc(SC)n2)CCN(C(c2cc3ccccc3[nH]2)=O)CCC1C 68920,Cc1ccc(C(=O)NCCCN(C(=O)COC2CCC2)C)c(N)c1 68921,CC(C)CC(C(=O)N(C1CCN(C(c2ccnnc2O)=O)C1)CC)c1ccccc1 68922,CC1CN(C(c2nc(Br)c[nH]2)=O)CCC1N(C(=O)Cc1cccc(F)c1)C 68923,N1(C(C(C(C)C)O)=O)CC2CCN(C(c3cc(C(F)(F)F)ccc3N)=O)C2C1 68924,N1(CCNC(c2c(C(CC)(C)C)ccc(F)c2)=O)CCCN(C(=O)C(F)(F)F)CC1 68925,CCCCC(O)CC(=O)N(c1cccc(Cl)c1)CCCNC(=O)CCCC#N 68926,C#CCC(C)(CC)C(=O)NC(CC(=O)N(C(C)CC)CCOC)C(F)(F)F 68927,C1(C(=O)NC(C#C)(C)C2CCCC2)CCCN1NC(=O)C1CC2(CC2)C1 68928,c1(CCC)ccccc1NC(C1CC(F)CN1C(=O)C(C1CCOCC1)C)=O 68929,CC1(CNC(c2ccc(F)c(O)c2)=O)CCN(C(C2SCCS2)=O)CC1 68930,c1(SCCN(C(c2ccncc2)CNC(=O)CC2CSC2)CC)ccccc1C 68931,c1(NCc2nccc(C)n2)nccc(=NCC2(CO)CC3C=CC2C3)[nH]1 68932,N1(C(C(C(C)C)n2cncn2)=O)CC2CCC1CN2C(=O)C1=COCCC1 68933,c1(CNC(C(N2C(C(N)=O)CC(O)C2)c2ccsc2I)=O)cccc([N+](=O)[O-])c1 68934,C1(CNC(C2CCC(COC)C2)=O)CN(C(c2ccnn2CCF)=O)CC1O 68935,C1(NC(c2cncc(N(C)C)c2)=O)CC2(C1)CN(C(c1cc(F)ccc1Cl)=O)C2 68936,c1(C(N2C3CC(CNC(CC(C)SC)=O)C2CC3)=O)coc2c(F)cc(Cl)cc12 68937,N1(C(C(C=C)NC(C)=O)=O)CCCC(CN(C)C(c2ccnnc2C)=O)C1 68938,CC(C)(CO)C(=O)NCCCN(C(=O)CCSC1CCCC1)CC1CCCC1 68939,N1(C(COCC)=O)CC=CC(NC(c2ccc(OCc3cccnc3)cc2)=O)C1 68940,O=C(CC(C(F)(F)F)n1ccnc1)NC1(CO)CN(C(=O)CSS(C)(=O)=O)C1 68941,C1(C(N2CCC(C3(C)N=N3)C2)C(=O)NCCCC)CCC(C(F)(F)F)CC1 68942,C1(C(=O)NC2CC(OCC(=O)NC3C(C)C3)C2)CCCC(=O)CC1 68943,CCCCC(CNC(c1nncs1)=O)NC(c1cc(CN2CCCC2)cn1C)=O 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68978,C(=O)(CC(=O)NCC(CO)NC(c1n[nH]cc1-c1ccccc1)=O)NCC 68979,N1(C(C2(C(=O)OC)CC2C)=O)CCN(C(C2CCN(CC3CC3)CC2)=O)CC1 68980,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(C)c1C(C)=O 68981,C(=O)(CCCC(C)(C)CC)N(C(=O)C(C)(C)Cc1ccccc1)C1CCC(CC)C1 68982,CCCCCCCN(C(=O)C(CC)N1CCCC1=O)C.N12CC(C1)C2 68983,C12(C(=O)NC(CC#C)C(N)=O)COCC1CN(C(c1c(Cl)ncn1C)=O)C2 68984,c1(NC(C2CCC(CC(=O)NC(c3nncn3C)C)C2)=O)ccc(CO)cn1 68985,N1(C(c2c(OC)scc2)=O)CCCC2CN(C(C34CC(C#N)(C3)C4)=O)CC12 68986,N1(C(c2ccc(CC)s2)=O)CCC(NC(=O)Cc2ccno2)C12CCC2 68987,C1(C(N(CCN(C)C)C)=O)C2CC(F)C(C2)N1C(C1C=CC(=O)N=N1)=O 68988,C(=O)(C(F)CC(C)(C)NC(=O)C1=CCCOCC1)N(C)Cc1cncs1 68989,c1(C(N2CC(CNC(C(CC)C)=O)C2)=O)cc(F)cc(Br)c1 68990,N1(C(c2ccc(OCC=C)c(OC)c2)=O)CC2(CC(N)C2)C1C(=O)O 68991,N1(C(c2cncc(COC)c2)=O)CCN(C(c2ccc(C)nc2)=O)CC1COC 68992,CCCC(C)N=c1cc(C)nc(N2CCN3C(=O)CCCC3C2)[nH]1 68993,N(C(=NCCCOCCC(C)(C)C)NCC1(C)CCS(=O)(=O)CC1)C(C=C)C 68994,O=C(CCCCn1ccnn1)C1CCCC(C(N2CC(c3nn[nH]n3)C2)=O)C1 68995,N1(C(C=CCOC)=O)C2CCC1C(NC(=O)Cc1csc(Br)n1)C2 68996,C=CCCC(O)CN(C(=O)CCC(C)NC(=O)C(CO)OC)C 68997,C=CCC(CC=C)C(=O)NC1(C(=O)NOCC(O)C(C)C)CCC(C)(C)C1 68998,N1(C(C2(CCC)CCNC2=O)=O)CCCCCC(NC(c2c[nH]ccc2=O)=O)C1 68999,c1(CC(=O)NC(C)CNC(C2CCOC2)=O)cc(-c2cccc(Cl)c2)n(C)n1 69000,c1(CNC(C(c2ccco2)NC(C23CC(CO)(C2)C3)=O)=O)ccc(O)cc1 69001,C(=O)(C(F)(F)C(F)(F)C(F)F)NC1(CNC(C2CC23CCOCC3)=O)CC1 69002,C12CCC3(CCC3)C1NC2=O.C1(C(C(=O)NCc2ccncc2)F)CCOCC1 69003,Cc1cc(=NC(=O)N(C2CC3(CCC3)C2)C)[nH]n1-c1ccccc1Cl 69004,O=C(N=c1[nH]nc(Cl)cc1Br)c1cc(Cl)ncc1NC(=O)Cc1ccc(Br)cc1I 69005,C1(NC(C(=O)NCC(C)N(N2CCCC2)C)=O)C[Si](C)(C)CC(O)C1 69006,N1(C(CCSCC(C)C)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69007,CCCCC(C)CCC(=O)NC(C)CNC(c1ccc(O)c(C)c1)=O 69008,C12(CCS(=O)(=O)C1)c1n(CC=C)c(nn1)N2C.C(CCOC)OC 69009,C(=O)(CC1COc2cc(O)ccc21)NCC(C(C)C)NC(c1ccc(C)nc1)=O 69010,C(=O)(C(C(C)(C)O)NC(C1CC12CCCCC2)=O)N(CC)Cc1ccoc1 69011,N1(C(C2C(C)OC(C)C2C)=O)CCC2CCC(C1)N2CCCc1nc(O)n[nH]1 69012,CCCC(C(=O)OC)C(=O)N1CC(C)CC1C(=O)NCc1ccccn1 69013,Cc1ccc(C(N2CCC(C)C2CNC(=O)CC2(C(F)(F)F)CC2)=O)c(N)c1C 69014,c1(C(=O)OCc2onc(C(C)(F)F)n2)cc2cc(Cl)ccc2[nH]1 69015,c1(NCC2CC(=C)C2)cc(=NC(C)c2ccn(C)n2)[nH]c(COC)n1 69016,Cc1cc(C(=O)N(C2CCCCC2N(C(=O)C2=C(Cl)CCC2)C)C)cc(O)n1 69017,N1(C(=O)Nc2c(C)onc2)CCCC(C(C)NC(=O)Cc2c[nH]nc2O)C1 69018,CC1CCOC1C(=O)NC1(C(=O)NCC2CC(Cl)(Cl)C2)CCC1 69019,c1(C(N2C(CNC(Cc3scc(C)c3)=O)CCCC2)=O)ccn2cccc2c1 69020,Cn1ccnc1CC(N1CCC(CNC(=O)CCOc2cccnc2)C1)=O 69021,C=C1CCN(C(=O)CCc2nc(O)n[nH]2)C(C(N2CC(O)(C(N)=O)C2)=O)C1 69022,C1(CC#C)(C(=O)NCCC(C)(C)NC(=O)C(CCCC)N(C)C)CCCCO1 69023,CCC(CNC(C1CC1(C)C(F)F)=O)(CC)C(=O)NCCS(=O)CC 69024,C(C(CC(C)C)NC(c1csc(F)c1)=O)NC(c1n(CCC)ccc1)=O 69025,N1(C(C2(CC)CCN(C(c3ccc4c(c3)OCC4)=O)C2)=O)CCC(C)C2(CCC2)C1 69026,c1(CN(CCCCOC2CC2)C)csc(-c2cnn(C)c2)n1 69027,CC1CN(C(C2(C)CC(C(F)(F)F)C2)=O)CCC1NC(c1cn(C)nn1)=O 69028,N12CCN(C3CCCCC13)C(=O)C1=CC=C(C=CO1)C2=O.Cc1nc(CO)co1.NCC 69029,c1(C(=O)NC(C(C)C)CCNC(=O)CC2C=CCCC2)nc2n(c1Cl)CCCC2 69030,N1(C(C2(NC(=O)CCNC(=O)CO)C(C)C2)=O)CCC(F)(F)C(O)C1 69031,N1(C(C2CC(C(=O)NC3(C(N)=O)CC3)C2)=O)CC2CCC2(CO)C1 69032,C1(O)(C(C)C)CCN(C(C23CC(NC(c4cc(C(C)C)no4)=O)(C2)C3)=O)C1 69033,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69034,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(C2CCC(=O)N2)=O)C1 69035,C1(CCOCC(=O)OC(C)(C)C)CCC(COC(C2(C(=O)OC)COC2)=O)CC1 69036,CC1CC(C(=O)Nc2c[nH]nc2Br)N(C(c2cncc(Br)c2)=O)C1 69037,c1(C(=O)NC(C)CCNC(N)=O)ccccc1NC(=O)CC(F)(F)F 69038,N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)C(C)(F)F)CC2C1 69039,c1(NC(c2cn(CCNC(C3CC3C3CC3)=O)nn2)=O)cccc(CC)c1 69040,c1(C(N(C)CC2CCN(C(c3c(CC)cns3)=O)C2)=O)c(C(F)(F)F)n[nH]c1C 69041,N1(C(=O)NC2CC(OC(C)(C)C)C2)CC2CC1CCC2OC1CC(=O)NC(=O)C1 69042,N1(C(Cc2c(C)ocn2)=O)C2CCCC1CN(C(C1CCCO1)=O)CC2 69043,N1(C(=O)NCC2CCO2)CCN(CC2CC2)CC1 69044,c1(NC(c2c(-c3cc(C)c(Br)cc3)cncc2)=O)nc(C)nc(Br)c1F 69045,c1(C2CC(Nc3ccc(CC(C)C(=O)O)cc3)C2)ccc2cccnc2c1 69046,N1(C(CCc2ccc(C)o2)=O)CCC2(CCN(C(=O)C(C)CN(C)C)C2)C1 69047,N1(C(C(=O)Nc2ccc(C(CC)C3CC3)c(F)c2)=O)CCCNC(=O)C1(C)C 69048,CC1Cc2cc(C(=O)NCC(C3CCOC3)NC(=O)CNS(C)(=O)=O)ccc2O1 69049,C1(n2cc(-c3nc(-c4ccc(C)s4)sc3)nn2)CCCN(C2CC2)C1 69050,N(C(=NCCCC1CCC1)N1CC=C(c2cccs2)CC1)CCOC 69051,CCC(CNC(=O)CCNC(c1cnco1)=O)OC 69052,C=CC1CN(C(=O)CC=CCNC(=O)CCOC(C)C)C1 69053,CCC(CC(=O)NCC1CCC12CN(C(c1ccc(C)nc1C)=O)C2)C(F)F 69054,c1(SC)cnc(N(C)C)nc1.c12n[nH]c(n1)CNC(=O)NC2 69055,S(=O)(=O)(c1c[nH]c(C(=O)NC2CN(C(c3cc(C)n(C)c3)=O)CC2O)c1)NC 69056,N1(C(CC=C)=O)CCCC(NC(c2nc(C)n(C3CC3)c2C)=O)C1C 69057,C(CCC(=O)NCCC1(NC(=O)CCF)CCCC1)=CC 69058,S(=O)(=O)(c1cnc(NC2CC3(CC3)CO2)c(Cl)c1)NCC(C(CC)CC)O 69059,N1(C(C(C2CC2)OC)=O)CC(CNC(=O)CSc2ccccn2)C2(CC2)C1 69060,CC1CCCCC1(CNC(C1(C)CC1(F)Cl)=O)NC(=O)C(N1CCC(O)CC1)C 69061,Cc1ccc(F)c(C(=O)NCc2cccc(CNC(=O)C(C)N3CCC3)c2)c1F 69062,C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)N(CCC)CC1CC1 69063,CC1CCC(NC(=O)Cn2cnc(=N)[nH]2)CN1C(=O)CC1(CO)CC1 69064,N1(C(c2cn(CCC)nc2C)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C(C)C1 69065,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69066,N1(C(C2(CNC(c3n(CC)nnc3)=O)CCCO2)=O)CCOC(C2(C)CC2)C1 69067,c1(C(=O)NC(C2N(C(c3ccc(COC)o3)=O)CCC2)C)cc(C)nc(C)c1 69068,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCOC2)cncc2c(F)cccc12 69069,c1(C(=O)NC2(C)CN(C(C(CCC)(C)C)=O)C2)n[nH]c2c(C)cccc12 69070,Cc1cccc(O)c1.N12CC(C(O)C1)NC(=O)CN(C)CC2=O.N(C)C 69071,C(=O)(CC1=CCCCC1)NCC(C)CNC(c1conc1C(F)(F)F)=O 69072,c1(C(=O)NC2CC(C(=O)NCC3CCCSC3)C2)ccn2ccccc12 69073,C1(C(N2CCOC(c3n[nH]c(CO)n3)C2)=O)CCOC2(CCCCC2)C1 69074,CCC(CC)C(C(=O)NC(CC(N)=O)C(=O)NCc1nnc(O)n1C)OC 69075,N1(C(CCNC(=O)OC(C)(C)C)=O)CC2CCC(NC(C3(CSC)CC3)=O)CC2C1 69076,C1(NC(=O)C(CC)N(C)C=O)CC2CCCC(C1)C2N.CCCCCCNC=O 69077,C(=O)(C(C)(C)C(O)C(C)C)NCC(C)=CC(=O)NCCC(CC)(CC)OC 69078,Cc1nc(=N)[nH]c(C)c1C(=O)N(C)CCNC(c1cc(F)ccc1C(F)F)=O 69079,C(=O)(CC(C)CC(=O)N1CCC(F)(C(=O)NCCC(=O)NO)C1)OC 69080,N#Cc1cnn(CC(=O)NC2CC(CNC(c3cccnc3Cl)=O)C2)c1 69081,Cc1nc2ccccn2c1C(=O)NC(CNC(C1CCCC1C)=O)C(C)(C)C 69082,C1(N(C(=O)Cc2cnc[nH]2)C)CCCCC1N(C)C(C1CCOC1)=O 69083,c1(CC)cc(N)c(C(=O)NCC2CCN(C(=O)CCC(CC)SC)C2)cc1F 69084,C1(CC(=O)NCCC(N2CC(C)(CSC)C2)=O)CCC(=O)CC1 69085,c1(CC)ncsc1C(=O)NCC1(CC(=O)NC(C)CCCO)CCCC1 69086,C(CC(C)(C)C(=O)NCCOCCN(C(=O)CC(C)(C)SC)C)OC 69087,S(=O)(=O)(c1cc(C)cnc1NCC1CSCCO1)N1CCN(C(CC)CO)CC1 69088,c1(OC)cc(C)sc1C(=O)NCCNC(c1cc(-c2ccc(F)cc2)n(C)n1)=O 69089,C1(CC)CCCN(C(C2(C)CCCN(C(C3CCC(C)(C)C3)=O)C2)=O)CC1 69090,c1(N2CCC(N(CC(C)C)C)C2)cc2nc(n1)CN2C.c1(SCC)cccnc1 69091,N1(C(C=CSC)=O)CCCC2(NC(c3ncn(C)n3)=O)CCCC12 69092,c1(OCC)cccc(CCN2CC(CN(C3CC4CC4C3)CC)C2)c1OC 69093,c1(NCC2CC(CC3CC3)C2)cc(OC)ncn1.C12(COC)CN(C1)C2=O 69094,c1(OC)nc(OC)nc(N(C2CCNCC2F)C(=O)CCn2nc(C)nc2C)n1 69095,C1(NC(CNC(N)=O)=O)CC2CN(C(=O)CSc3cccc(F)c3)CC12 69096,c1(CNC(C(C)CO)=O)cc2n(n1)CCN(C(c1cc3n(n1)CCCO3)=O)C2 69097,C12(C(=O)NC(C3CCCO3)C)CC(CO)(CN1C(c1ccncn1)=O)C2 69098,N1(S(CCC)(=O)=O)CCC(CO)(NC(c2ccc(C)cn2)=O)CC1 69099,N1(C=O)CC2CC1CN2C(c1ccc(C(C)(C)C)cc1)=O.C(=O)(C(C)OC)OC 69100,c1(CCC(=O)NC(C2(O)CCN(C(=O)Cc3cnoc3)C2)C)cc(F)cc(F)c1 69101,C1(C(=O)Nc2cnc(C)nc2)CCN(C(C2(C)CC3C=CC2C3)=O)C(C)(C)C1 69102,CC1CC(NC(=O)Cn2nnc(C(C)(C)C)n2)CN(C(c2ccoc2Cl)=O)C1 69103,Cc1cc(C(=O)N(C)C(c2cccc(C(F)(F)F)c2)C)nc(-c2cnccn2)n1 69104,n1(CCCSC)nnnc1C(c1n[nH]c(C)n1)NCCSC1CCOC1 69105,C(=O)(CC(O)CNC(=O)C(C)(CO)NC(=O)Cn1cccnc1=O)OC 69106,c1(SC)cccc(C(N2CCC(NC(c3occc3C)=O)C(F)C2)=O)c1[N+](=O)[O-] 69107,C1(NC(C=CCOC)=O)CN(C(C2CCN(c3ccccc3)C2)=O)C2CC12 69108,c1(C(N2CC3(CCN(C(c4cnc(C)s4)=O)C3)C2)=O)cccc2nc(O)oc12 69109,C1(c2nnnn2C2CCOCC2)(NC(c2nccn2C)CC)CCOC(CC)C1 69110,N1(C(CC2(CC=C)CCCC2)=O)CCC(C(=O)NC2C(C)C2(C)C)C(C)(C)C1 69111,c1(OCC)cnc(C)c(C#N)c1.c12cc(ccc1F)C(=O)OC2=O 69112,C1(CNC(Cc2n(C)cnn2)=O)COC(C)(C)CN1C(C1CCC2(CCC2)C1)=O 69113,c1(OC)ccc(OCC(N2CCC2CNC(=O)CC2COCC(C)O2)=O)cc1C 69114,c1(-c2ccc(C(=O)NC(C)CC#N)cc2F)cccc2ccsc12 69115,C(=O)(C(CC(C)C)ONC(c1cc(Cl)c[nH]1)=O)NC(C#C)CCC 69116,C(=O)(C(C)C(C)S(C)(=O)=O)Nc1ccc(NC(c2c(CC)onc2C)=O)cc1C 69117,CCCCCC(C)CC(=O)N1CC(NC(C2CC2(C)Br)=O)C1 69118,c1(OC)ccc(C(C)C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1F 69119,Cc1ccc(NC(C2CCC(NC(=O)C(C)C#N)C2)=O)c(C)n1 69120,c1(C2C(C(=O)NCC(CC=C)NC(c3ccc(O)nc3)=O)C2)c(C)cccc1C 69121,N1(C(Cc2cn(C)nc2)=O)CCn2c(CSc3ccc(Cl)nc3)nnc2C1 69122,C(c1ccc(C(N)=O)cc1)=CC(=O)NCC(C)N(C(C(C)C1CCC1)=O)C 69123,CCC(C)C(O)C(=O)NC1CCN(C(=O)CS(=O)(=O)N2CCC(C)CC2)C1C 69124,C1(O)(Cn2cc(C3(C(C)C)CCC3)nn2)CCCN(C(C2(Br)CC2)=O)CC1 69125,c1(NC(CCOCCN(C(CC(COC)C)=O)C)=O)ccc(C)c(F)c1 69126,N1(CCC(=O)NC2C(CNC(COCCCOC)=O)CCC2)CCC(F)C1 69127,c1(OC)c(C(=O)NCC(C)(CO)NC(c2cccc(N)c2)=O)ccnc1F 69128,C(CCCC(=O)NC12CCCC1(C(N)=O)C2)N(C(C(C)NC=O)=O)C 69129,C12(NC(C(CCCOC)NC(=O)CC3CCC(=O)N3)=O)CCC(O)(CC1)CC2 69130,c1(OCCC(N2CCC(C)(NC(C(CC)F)=O)C2)=O)c(C)cccc1C 69131,c1(C(C)=O)ccc(C(N2CC(CNC(c3ccncc3Cl)=O)C(O)C2)=O)c(O)n1 69132,N1(C(c2nn(CC)c(O)c2)=O)CC2CN(C(=O)CCC(=O)NC)CCC12 69133,C1(OC)CC(COCC(C(F)F)n2cccn2)N(C(=O)OC(C)(C)C)C1 69134,Cc1ncc2n1CC(C(N1CCC(CNC(=O)COCCCF)C1(C)C)=O)CC2 69135,Cc1oc(S(N)(=O)=O)cc1C(=O)NCC(C)N(C(=O)C(C)c1cncs1)C 69136,C=CCC(CNC(=O)C(C)OC)C(=O)NC(c1c[nH]ccc1=O)C 69137,c1(OC)ccc(OC)c(CNC(=O)NC2(OC)CCSCC2)c1 69138,CCCCC(F)C(=O)N1CCC(C(=O)NC2(n3cnnc3C3CC3)CC2)CC1 69139,C1(C(=O)NCC(C#C)OC)CCCCCN1C(c1nn(C)cc1C)=O 69140,c1(NC(CC)=O)ccc(CN2CCC(N(C)Cc3ccc(CC)o3)C2)cc1 69141,Cn1cccc(C(=O)NCC)c1=O.C12CCN(C1)CCN2C(C1(CCF)CCC1)=O 69142,N1(C(c2nnc(C)s2)C(=O)NCSc2ccccc2)CCN(S(=O)(=O)N(C)C)CC1 69143,C1(CNC(c2c(CC)nn[nH]2)=O)CCCCN1C(C1CCCCN1C(C)C)=O 69144,N1(C(c2ccc(C(C)=O)o2)=O)CC(CNC(=O)CC2CCCO2)OC2(CCC2)C1 69145,C(CC(CNC(c1cnn(C(C)C)c1)=O)NC(=O)CSCCC(C)C)OC 69146,N1(C(C(CC(N)=O)O)=O)CCCC2CN(C(c3scc4c3CCCC4)=O)CCC12 69147,C12(CNC(c3c(C)nco3)=O)CCC(CC1)N(C(c1ncccc1F)=O)C2 69148,CC1N(C(=O)CC2CN(C(=O)C(C3CCCCC3)F)CCC2C)CCC1(C)C 69149,c1(CC(=O)NCc2ccc(C(=O)OC)n2C)noc2ccc(O)cc12 69150,c1(NC(C2CC(C)OC2)=O)cnc2c(-c3ccccc3)cccc2c1Cl 69151,C1(CC(=O)NC(C2CC(F)(F)C2)C)CCCN1C(=O)C(C)(C)O 69152,N1(C(=O)CN(C)C(C)C)CCCC(C(C)(C)C(=O)NC(C=C)C2CC2)C1 69153,c1(CC(=O)NCC2(C(N)=O)CN(C(C(CO)OC)=O)C2)c(C)cc(C)cc1C 69154,c1(C(=O)NC2CC(CC(=O)N(CC)CC3(O)CCC3)C2)cc(C#N)oc1C 69155,N1(C(c2ncc(C)c(Cl)c2)=O)CC2CCN(C(C3CCCC3)=O)CC12 69156,c1(C(N2C(CNC(CC(=O)NCC)=O)C=CC2)=O)cccc2[nH]nc(O)c12 69157,C(=O)(C1=CC2(CCOC2)C1)N1CCCC(CNC(Cc2nc(CC)on2)=O)C1 69158,Cc1nc(C(=O)N(CC(C)NC(=O)CCN2CCNC(=O)C2)C)cc(O)n1 69159,c1(CN2C(CC(=O)Nc3cccnc3F)COCC2)cccc2ncccc12 69160,CC1CN(C(c2cc(CO)[nH]n2)=O)CC(C(=O)NCC2CC3CC3C2)O1 69161,c1(C(N2C(C(=O)Nc3cnc(OC)c(F)c3)CCC2C)=O)[nH]nc2ccncc12 69162,Cc1ccc(O)c(C(N2CCC(F)C(NC(c3ccc(Cl)nc3O)=O)C2)=O)n1 69163,C(=O)(C1=NNC(=O)CC1)N(C)CC1CN(C(c2c(C(C)C)c[nH]c2)=O)CC12CC2 69164,c1(CCC(=O)NC2C(CNC(c3csc(CO)n3)=O)CCC2)cccc(F)c1 69165,C1(C(=O)NC(C)C(N2CC3C(CC4NC(=O)NC4=O)C3C2)=O)C2C3CCC(C3)C12 69166,C(=O)(N=c1cc2ccccn2[nH]1)C1CCN(C(C(C)CN)=O)CCC1C 69167,N1(C(c2nn(C)cc2Br)C(=O)NCCC)CCC2(CCN(C)CC2)CC1 69168,c1(C(=O)NC2C=CCN(C(c3cc(C)[nH]n3)=O)C2)cn2c(n1)CCCC2C 69169,S(=O)(=O)(c1cc(Cl)ccc1F)N1CCN(C(c2cc(F)c(Cl)cc2Cl)=O)C2C1C2 69170,CC(O)CC(C)(C)CNC(C1CCN(C(c2cc[nH]c(=N)n2)=O)C1)=O 69171,C1(NC(C(F)=CC)=O)CCCC(CC)C1.c12ncc(s1)CCN(C)C2=O 69172,c1(C(=O)NCC(CNC(c2cccc(C)c2)=O)C)ccc2nnc(C3CC3)n2c1C 69173,c1(C(=O)NCCCN(C(CCN(CC)CC)=O)C2CC2)nccc2ccsc12 69174,C1(C(N(CC(C)C(=O)NCCc2cccc(O)n2)C)=O)CCOC(=O)CC1 69175,C1(N(C(C(CSC)C)=O)CCO)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1 69176,C1(C(=O)NCCN(C(C=CC(C)(C)SC)=O)C(C)C)C(F)(F)C12CCC2 69177,Cc1ccccc1.C12(CNC(CNC(N)=O)=O)CC(CN1C(C1CC1C(F)F)=O)C2 69178,Cc1c(CCC(N2CCCC(CN(C(=O)CCn3cnnn3)C)C2)=O)cnn1C 69179,C1(C)(NC(c2ccnc(C)n2)=O)CCN(C(c2cc(C(C)(C)C)ccn2)=O)CC1 69180,C(=O)(C(C)(C)C1=CCSCC1)NC(CCCC)CNC(c1cccnc1OC)=O 69181,CC(O)(CC(=O)N1CC=CC(NC(C2CC2c2ccc(NC)cc2)=O)C1)C(F)(F)F 69182,N1(C(=O)OC(C)(C)C)CC2CC(Nc3nccnc3Cl)C(C2)C1 69183,N1(C(c2scc(C)c2)=O)CCC(CNC(c2ccnc(C3CC3)c2)=O)C1(C)C 69184,C1(CNC(=O)Cc2ccns2)CCCN1S(=O)(=O)CCn1ccnn1 69185,CC(C)C(O)C(=O)N1CCCCC1C(=O)NOCc1nc[nH]n1 69186,C1(N(C(COCCOCCOC)=O)C)CCCCC1NC(c1cnn(C)c1N)=O 69187,C1(NC(=O)Cc2ccccc2OC(F)F)CC2CC(C1)N(Cc1ccccc1)C2 69188,C(=O)(C(=O)N=S(C)(C)=O)N1C(COC)CN(C(c2coc(C(F)F)c2)=O)CC1 69189,N1(CC)CCN(C(=O)CC2COCCN2C(=O)CCn2cc(C)cn2)CC1=O 69190,CC1CN(C(C2CC3(C2)CC(F)C3)=O)CC(C)N(C(c2cnc(S)n2C)=O)C1 69191,NC1(CNC(C2CCC(CNC(=O)CNC(=O)C3CC3)C2)=O)CCOC1 69192,C1(C(N(C2CCN(C(C3C=CCC3)=O)CC2)CCCC)=O)CC(O)CN1C(N)=O 69193,c1(C(=O)NC(CN(C(c2n(CC)ccn2)=O)C)(C)C)cc2ccc(Cl)cc2o1 69194,Cn1cc(C(=O)NCC(CNC(c2cnn(C3CCC3)c2)=O)CO)c(O)nc1=O 69195,N1(c2ncc(C(=O)OCC)cc2NC(=O)CC(C)F)CCC2CCC(OC)C1C2 69196,c1(C(=O)NCC2CN(C(c3ccnc(CO)c3)=O)CC2O)cnc2nccn2c1 69197,N1(C(C2C3N(C(c4c(C)ncs4)=O)C(CC3)C2)=O)CCc2c(C)cccc2C1 69198,CN1CC(O)CC1C(=O)NC1CCN(C(=O)C(C)(C)c2ccnn2C)C1 69199,C12(CC(=O)N(C)CC3(O)CN(C(c4cnn[nH]4)=O)C3)CC3CC(C1)CC(C)(C3)C2 69200,c1(SCC(=O)N(C2CCOC2)CCC#N)ccc(Cl)c(Cl)c1 69201,c1(C(N2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C(F)C2)=O)ccnc(C(F)(F)F)c1N 69202,Cc1nc2cc(C(=O)NCC3CCCN(C(=O)CC4(CO)CC4)CC3)cnc2s1 69203,c1(C(=O)Nc2cccc(NC(C)=O)c2C)cccc2cncc(C(C)(C)C)c12 69204,c1(C(=O)N(C2CC2)CC2(C(=O)NCC=C)CC2)ncc(F)cn1 69205,C=CC1OCCC1C(=O)NCC1(C(C)NC(C2CN(S(=O)(=O)CC)C2)=O)CC1 69206,CC1(C)CN(C(C2(F)CC2)=O)CC1NC(C1CCC=CCC1)=O 69207,CCC(C)C(C)C(=O)N(CCCNC(=O)CCc1scnc1C)C 69208,CN1N=CC(CC(=O)NCC2(CNC(C3CC(CF)C3)=O)CCCC2)C1=O 69209,CC1(C)CC(C)(CNC(c2ncc[nH]c2=O)=O)CN1C(c1cc(O)cc(Cl)c1)=O 69210,CC1(C)CCC(C)(CN2CCCC(NC(c3cnoc3C3CC3)=O)CC2)CC1 69211,C(CN=c1[nH]c(=N)[nH]c(=NCCN2CCCC(C)C2)[nH]1)c1ccn(N(C)CC)n1 69212,C1(CNC(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cc(Br)co2)=O)C(C)C1 69213,N1(C(Cc2ncn(C)c2)=O)CCC(CNC(C2(C3CC3)CC2)=O)C(O)C1 69214,C(=O)(N=c1cc(C)[nH][nH]1)C1CC(=C)CN1C(=O)OC(C)(C)C 69215,c1(C(CC2CCCO2)NCC)ccccc1C(F)(F)F 69216,c1(C(N2CCC(C(N3CC(CC#C)OCC3)=O)O2)=O)cc(F)c2ccccc2c1 69217,c1(C(N(C(CC)CNC(c2cnc(O)o2)=O)C)=O)cc(OC)ccc1C 69218,C1(NC(CCSCC(N)=O)=O)(CNC(=O)CCC2(C)CC2)CCOCC1 69219,C(=O)(C#CC(=O)N(C)C)NC1C(NC(C(C)CN(C)C)=O)CC1 69220,N12CCC3CN(CCC13)C2=O.C1(CC)CC1C 69221,C1(N(C(C(C)OC)=O)C(C)=O)CN(C(=O)CCOC(C)=O)CC1c1ccccc1 69222,c1(NC2CCN(C(C)C)C2=O)c(F)cc(Cl)cc1Cl 69223,C1(NC(C(C2CC3CCC2C3)C)=O)CCC2CC1CN2C(=O)CC1CCC(=O)C1 69224,c1(C(CC)NCCCc2cnc[nH]2)nnc2n1CCC2 69225,C(=O)(C1=NOC(C(N2CC(NCC(F)C(=O)N3CCCC3)C3(CC3)C2)=O)C1)OC 69226,C1(NC(C2(CNC(C=C(C)C3CC3)=O)CC2)=O)CCOCC1C 69227,c1(C(N2CCC(CN(C(=O)Cc3cnn(C)c3)C)C2)=O)ccc(N)c(F)c1F 69228,CC12CN(C(C3(CO)CC(F)(F)C3)=O)CC1CN(C(=O)CN1CCCNC1=O)C2 69229,N1(C(C2(C#N)C(C)C2)=O)Cc2occ(C(N3CC4(CCC(=O)O4)C3)=O)c2C1 69230,C(CN=c1[nH]cnc2ccsc12)C1CCC(NC(c2c(COC)noc2)=O)C1 69231,N1(c2ncc(C(=O)NC3CC3(F)F)cn2)CCN2CCCC2C1 69232,C(c1cn(C)cn1)=CC(=O)NC(C(C)NC(C1CC(CC(F)F)C1)=O)CO 69233,CC(C)C(CCNC(=O)C(C)(O)C1CC1)NC(=O)C(F)OC(F)(F)F 69234,N1(C(C2CCSC2(C)C)C(=O)N(CCOCC)CC)CCC2CCC(C1)N2C(C)=O 69235,c1(C(=O)NC2CC3CCC2(Br)N3)cc(Br)cc2nc(O)[nH]c12 69236,C1(NC(c2nc(C)sc2C)=O)CC2CC1N(C(c1cnn(C(C)C)c1F)=O)C2 69237,Cc1nc(C)n(CC(N2CCCCC2C(=O)NCC(C)(C)N(C)C)=O)n1 69238,N1(C(COCC=C)=O)CC(NC(C2CCOC(C)C2)=O)C(c2ccnn2C)C1 69239,C(CCCCCNC(=O)Cc1cnn(C)c1)N(C)C(c1cc(C(F)(F)F)n[nH]1)=O 69240,C1(C(=O)NCC2(F)CC(NC(C3(CCCC)CC3)=O)C2)COC2(CCC2)CO1 69241,C(CN=c1[nH]c(N2CCOC(C)(CO)C2)nc2c1CCCC2)C1CCN(C)CC1 69242,c1(C(C(C#C)C)=O)nc(C(=O)OC)c(C)o1 69243,N(C1CCc2cccnc21)c1cc(NCC2(CO)CCOC2)nc(C)n1 69244,N1(C(c2c(CC)ocn2)=O)CCC2(CCN(CCCc3ccc(O)cc3)CC2)C1 69245,C1(C(C(=O)NCc2ccc(CNC(=O)CO)s2)O)CCCCCC1 69246,CC1(CCNC(C2(C)CCCCC2)=O)CCN(C(C2(C)C=CCC2)=O)C1 69247,Cc1cc(Br)cc(S(=O)(=O)NCC2(C)CCCNC2)c1 69248,c1(C(c2n(CCOC)nnn2)NC(CCO)CC(C)C)cc(OC)ccc1Br 69249,c1(C(=O)NC2(C(F)(F)F)CCOC2)ccc(CN(C)CCO)cc1.C1C(C)(C)N1 69250,c1(C(=O)NC2(CC=C)CCOC2)cc(CNC(=O)CCCC2CCCC2)ccn1 69251,C1(C(=O)NCC(CNC(CSCC(=O)OC)=O)C)CC[Si](C)(C)C1 69252,C1(OCC)(CNC(=O)CC2COC(=O)N2)CN(C(=O)CN2CCSCC2)C1 69253,C1(NC(c2nn(CC)c(C)c2)=O)CN(C(c2csc(OC(C)=O)n2)=O)CC2CC12 69254,CCC(C)(CNC(C1CC1(F)Cl)=O)C(=O)N(CC(C)(C)OC)C 69255,N1(C(C(C2CC2COC)OCC)=O)CCC(CNC(=O)CCCNS(=O)(=O)CC)C1 69256,c1(OCC(=O)NCC(CC=C)NC(C2C3CC4C(C3=O)C24)=O)nc(O)nc(O)n1 69257,Cc1cccc2c1CC(C(=O)NCC1(C)CCCN1C(c1cnn(C3CC3)c1)=O)O2 69258,c1(CC)onc(C(=O)N(C2CCN(CC3CCSCC3)C2)CC)c1C 69259,C(=O)(C1C(=O)N2CCOC(C2)c2cn1nn2)OC.C1(C(=O)O)(OCC)CC=CC1 69260,C(=O)(CC(C)C(C)(C)NC(=O)CC(C)O)NC1C(C#C)CCC1 69261,C1(O)(CC(=O)NCC(=O)NCC(=O)NCCC2(C)CCOC2)CCCOC1 69262,Cc1cc(C(=O)NC(C)CN(C)C(c2cc(C(N)=O)cs2)=O)nn1C(C)(C)C 69263,C1(OC)CN(C(=O)C(F)n2ccnc2)CC1NC(c1cnn(C)n1)=O 69264,c1(C(=O)NC2CCCN(C(c3nccc(C)c3)=O)C2C)cc2cc(Cl)ccc2[nH]1 69265,Cc1cc(NCC2(NC(C3CC4CC(=O)C3C4)=O)CCCC2)nc(C2CC2)n1 69266,C1(F)(C(=O)NCC2(C)CC(NC(c3c(C)ncn3C)=O)C2)CCCCCC1 69267,C(=O)(CC(C)P(C)(C)=O)N1C(CNC(c2c(C)non2)=O)CC(O)C1 69268,c1(CCOC(NOCCC#N)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 69269,CC(C)(CCC(=O)NCC12CCC(CN(C(=O)CCCCCF)C1)C2)[N+](=O)[O-] 69270,N1(C(C2(OCC)CCOC2)=O)CCC(C2(NC(=O)Cn3ccc(CC)n3)CC2)C1 69271,CN1CCCC(C(=O)NCC2(NC(=O)CN(C)C(N)=O)CCC2)C1 69272,C1(CCNC(C(COC)C)=O)CSCCN1C(=O)C(C1(O)CCCC1)F 69273,C1(F)(C(N(CC(C)N(C(=O)CC2CCN(C)CC2)C)C)=O)CC=CCC1 69274,CC1(Cc2cn(Cc3ccc(C(N4CC5CC(C4)O5)=O)o3)nn2)CCOCC1 69275,n1(CC(N2CCCCC(NC(C3(O)CC(C)(C)C3)=O)C2)=O)cnc2ccccc12 69276,C(=O)(C(C(C)(C)C)c1ccccc1)N(C)CCNC(C1C(C#N)C1(C)C)=O 69277,c1(C(=O)NC2CC(C)CN(C(c3csc(C#N)c3)=O)C2)cnc2ccccn12 69278,C1(NC(c2n(C)nc(C3CCC3)c2)=O)CC2CN(C(=O)C#CC(C)(C)C)CC2C1 69279,C1(CNC(C(C2CCCC2)OCC)=O)CN(C)CCN1C(=O)C(C)Cn1cccn1 69280,C1(NC(C2(SC)CCC2)=O)CC2CN(C(c3cccc(C#N)c3)=O)CC2C1 69281,N1(C(c2n(CCCC)ncc2)=O)CCN(C(C2(C)CC3CC3C2)=O)CCC1C 69282,O=C(C(Cl)=CCl)NCCCC1CCCN1C(C1(c2ccncc2)CC1)=O 69283,C1(C(N(C)CC2(C)N=N2)=O)CCCN1C(=O)CCc1nc(O)n[nH]1 69284,C1(C(=O)NC2(COC)CCCC2)C2CCC(C2)N1C(C1C=CC=CC=C1)=O 69285,c1(C(N2C(CC(=O)Nc3ccc(N(C)C)nc3)CCCC2)=O)ncc(F)cc1N 69286,CC1(C)CN(C(=O)C(c2cccc(F)c2)(C)O)CC(CNC(=O)Cc2ccoc2)O1 69287,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(=O)C=Cc1ccc(Cl)cc1 69288,CCS(=O)(=O)CCN=C(NCCOCc1cccc(Cl)c1)NCC1CCOCC1 69289,CC1COCC1(c1nnnn1C)NCCC(=O)NCCCP(C)(C)=O 69290,C(CS(=O)(=O)CC(=O)NC1COCC1CN1CCOCC1)OC 69291,C(=O)(C(CO)N(C)C)NCC(C)CNC(=O)CCNC(c1ccsc1)=O 69292,C12(NC(CCCC=C)=O)CC(CNC(c3cc(C)n(C)n3)=O)(C1)OC2C 69293,C12(CNC(=O)CCc3cn(-c4ccc(F)cc4)nn3)COCC(CO)(C1)C2 69294,C(CC(C)(C)CNC(=O)Cn1ncc(Br)n1)NC(COC)=O.C1(C=O)CCCOC1 69295,c1(-c2cnc(NC(C)=O)c(Cl)c2)cnc2cc(-c3ccnn3C3CC3)ccn12 69296,C1(CC(=O)NCCCOC)C2CN(C(C3CCCOC3)=O)CC12 69297,C1(CC(=O)N(CCCN(C(Cc2cn(C(C)C)nc2)=O)C)C)CC2(CCC2)CO1 69298,C(c1ccc2[nH]ccc2c1)=CC(=O)NC1CN(C(C2C(C)C2)=O)C2(C1)CCC2 69299,Cn1cc(S(=O)(=O)NC2CCN(C(C3(c4ccc(F)cc4)CNC3)=O)CC2)cn1 69300,C1(C(C)C(=O)NC2(CNC(c3ccc(CC4CC4)s3)=O)CC2)CCCCCC1 69301,N1(C(c2cnn(CC)n2)=O)CC(NC(=O)C(C2CCCO2)OC)C(C(F)F)C1 69302,c12cccc(c1)NC(=O)NCCC(=O)NC2.c1(N2CCCCC2)cncc(F)c1 69303,N1(CC(=O)NCC2(CNC(=O)CCN3CCCCC3)CCC2)CCCC(O)C1 69304,C1(C)(C(=O)NCc2cccc(CNC(CC3CC(C)(C)C3)=O)c2)CCCNC1=O 69305,C1(CC(=O)NCCC2(OC)CCC2)CC(C)(C)CN1C(=O)C(F)F 69306,c1(CNC(C=C(C)C(C)C)=O)cccc(CNC(C2(C)CC3CC3C2)=O)c1 69307,CCCCCCC(O)CCC(=O)NC1CC2CC1CN(C(=O)C(C)(C)CC)C2 69308,c1(C(c2n(CC)nnn2)NCC(c2c(Cl)cccc2Cl)C)cnc2ccsc2c1 69309,c1(C(=O)NC2CC(CNC(c3cncc(C)c3)=O)C2)cc(Br)c(C)nc1N 69310,c1(NC(C2CC3(CCC3)C2)C)cnc2ccccc2n1 69311,c1(CC(N2CCC(CNC(Cc3nnc(C)s3)=O)C2)=O)ccc2nn(C)cc2c1 69312,N1(C(C)(C)CO)CCC(N=c2cccc(S(=O)(=O)NCC3(C)CCOC3)[nH]2)CC1 69313,N1(C(c2cnc(-c3cccs3)o2)=O)CCCC(Cn2cc(CCC3CC3)nn2)C1 69314,c1(C(=O)N(C)C)ccn2nccc2c1.C1(=O)CN(C(C)C)CCN1C 69315,c1(C(C)C)noc(CCC(=O)NCC2CC2CNC(=O)CN(C2CC2)CC)n1 69316,C#CCC(CC#C)C(=O)NC(C)(CNC(c1nc[nH]c2ncnc1-2)=O)CC 69317,N1(C(C(C)C2(O)CCC2)=O)CCC(C2CC2)(CNC(C2C=CCC2)=O)C1 69318,N1(CC)CC(CNC(=O)Cn2cc(CC(c3cccc(C)c3)O)nn2)NC1=O 69319,C1(CCOCC)CCCN(C(=O)NCCOc2cnn(C)c2)C1 69320,c1(C(=O)NC2CCCC(NC(c3c(C)[nH]nc3Br)=O)C2)ccc(O)c(Cl)c1 69321,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(C23CCC(CC2)OC3)=O)CC1C 69322,Cc1ccc(CC(=O)NCCC23CCC2CN(C(=O)CSC2CC2)C3)c(F)c1F 69323,CCC(C)CC(=O)NCCN(C(=O)CC(C)OC)C(C)C 69324,N1(C(c2oc(CC)c(C)c2)=O)CCC(C)(C)C(CNC(=O)CC2COCC2O)C1 69325,N1(C(CC2N(C)CCC2)=O)CCC(OCCNC(C2(CSC)CC2)=O)CC1 69326,C1(COC)(CO)CCN(C(c2cnn(C)c2)C(=O)NCC=C2CCSCC2)C1 69327,c1(C(=O)NC2CC(CCNC(CCC(CC)C)=O)C2)nc2nc(C)cc(C)n2n1 69328,CCC(C)(C)C(=O)NC(C1(CNC(=O)Cc2ccoc2C)CC1)C 69329,C1(C2CCC2)C(=O)NOCc2ncccc2O1.C(CO)OCC 69330,c1(CC(N2CCCCCC2CNC(=O)CC(F)(F)F)=O)ccc(Cl)c(F)c1 69331,C1(OC)(OC)COC(C(C(=O)NCCCC(C)C)N(C)CCn2cccn2)C1 69332,C(=O)(C1=CSCCO1)N1C(CCNC(=O)CCc2ccsc2)CSCC1 69333,C(=O)(CCS(C)(=O)=O)NC1CC(CNC(C(C)OCC2CCCCO2)=O)C1 69334,CC1(C)CN(C(c2ccsn2)=O)CCC1NC(c1cc2ccccn2n1)=O 69335,c1(C(=O)Nc2ccc(Cl)cc2Cl)ccc(S(N)(=O)=O)o1.CC1CN2CCN1C2=O 69336,S(=O)(=O)(c1cc(C(=O)NC2(CNC(c3cccn3C)=O)CCC2)co1)NC 69337,C(CN=c1cc(C(C)(C)C)nc(Cl)[nH]1)(C(C)(C)C)NC(C1C(COC)OCC1)=O 69338,C(=O)(C(C)(C)C(=O)NCC1(O)CCCN(C(c2coc(CC(C)C)n2)=O)C1)OC 69339,c1(C(=O)NC2C(OCC)CN(C(C(CC)COC)=O)C2)ccc2nc(C)oc2c1 69340,c1(-c2cn(CCC(=O)NCc3cc(Cl)ccn3)nn2)cc(F)cc(F)c1F 69341,C#CCC(C)(CC)C(=O)NCC(CCNC(c1c(C)[nH]c(C)c1C)=O)OC 69342,Cc1cccn2cc(C(=O)N(C3CCN(C(c4ccnn4C)=O)C3)C)nc12 69343,c1(CC(=O)NCCC(C)NC(C(C)SCC)=O)c(C)cc(OC)cc1Cl 69344,C1(NC(C2C(CNC(Cc3n(C)c(S)nn3)=O)OCC2)=O)CCC2CCC1C2 69345,c1(C(=O)NCCCCNC(c2nccc(C(C)(F)F)c2)=O)ccc2n[nH]cc2n1 69346,CCC(C(=O)NC1(CF)CN(C(C2CCSC2)=O)C1)C(C)(C)CC 69347,c1(C(N2C(C(C)NC(C(C)=CC)=O)CCC2)=O)ccc2nc(C)n(C)c(=O)c2c1 69348,c1(OC)ccc(N(C(=O)C(=O)N(CCCc2ccsc2)C)C)cc1OC 69349,C(C(=O)N(C)CC1CCN(C(=O)CC2(CC)CCCC2)C1)(C(C)C)SCC 69350,Cc1cnccc1N1CCN(Cc2cn(C3CCCCC3F)nn2)CC1 69351,N1(C(Cc2ncc(C)nc2)=O)CC(NC(c2sc(F)cc2C)=O)CCC1C 69352,CCC(CN(C)C)CC(=O)N(CCNC(C12COCC1C2(F)F)=O)CC 69353,CC1=NOC(C(=O)NCCC(C)NC(c2snnc2C2CC2)=O)C1 69354,CCCCC(CNC(=O)CC1CCN(CC)C1)NC(=O)C(C)(O)c1ccccc1 69355,C1(NC(Cn2nnc(C)n2)=O)C2CCC(C2)C1C(=O)N(C1CCN(C)C1)C 69356,C1(CCNC(=O)NC(C)C(c2ccncc2)C2CCCCC2)CCC(C)(C)O1 69357,C=CC(C)(O)CC(=O)N1CC(C(F)(F)F)CC1CNC(=O)CCC1CC1(Cl)Cl 69358,C1(CC(=O)N(C)CC=C2CCCC2)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 69359,C1(OC)CC2N(C1)C(=O)C1CC(C1)C(=O)NC(CO)C(C)NC2=O.S(C)(=O)(=O)SC 69360,CC1CC(NC(=O)Cc2ccc(Cl)cc2F)C(C)CN1C(c1ccc(F)o1)=O 69361,C1(NC(Cc2cnc(C)[nH]2)=O)CCCN(C(c2cncc(C(C)C)c2)=O)CCC1 69362,C1(CC(N2CC(c3ccccc3)(NC(C3CCC=CO3)=O)C2)=O)CCCCCC1 69363,CN1CCN(CCC(N2CC3C(NC(=O)COc4ccc(Cl)cc4)C3C2)=O)CC1 69364,C1(CC(=O)NCC(C)NC(=O)CS(=O)(=O)Nc2ccccn2)CC(=O)NC(=O)C1 69365,CC1(C)CCCN(C(c2c[nH]nc2F)=O)C1CNC(=O)Cc1nnc(O)s1 69366,c1(NC(=O)NC(C)CC2CCCCC2)ccc2c(c1)N(C)CCO2 69367,N1(C(C(C(C)C)S)=O)C2CC=C(C(=O)N3CCc4ncccc4C3)C1CC2 69368,O=S(=O)(c1csc(-c2ccc(F)cc2)n1)NCCSCc1ccccc1 69369,C(CCCCCC(=O)N1CC(CNC(=O)OC(C)(C)C)CC(F)C1)N(C)C 69370,O=C1CCC(C(=O)NC2CCCCC2NC(c2c[nH]nc2C(F)F)=O)=NN1 69371,C(=O)(CCC(C)S(C)(=O)=O)NCCCN(C(=O)CC(c1c(C)n[nH]c1C)C)CC 69372,Cn1cc([N+](=O)[O-])c(-c2nnc(-c3ccncc3)o2)n1 69373,c1(C(c2n(CCSC)nnn2)NCCOCc2cnsc2)ccc(C)c(F)c1F 69374,N1(c2ncc(C(=O)O)cn2)CCC2(CCN(S(=O)(=O)c3cncc(Br)c3)C2)C1 69375,N1(C(CCCC#C)=O)CCC2C1CCCN2C(c1cc2c[nH]nc2cc1C)=O 69376,c1(N(C(c2n(C(C)C)ncc2)=O)C)ccc(Br)c(N(C)C)c1 69377,C(=O)(C(=O)N=c1cc(C(C)=O)o[nH]1)NC(=O)Cc1ncoc1C(=O)OC 69378,N1(C(C2C(C)C2C)=O)CC2CCC1CN2C(C1CN(C(C)(C)C)CC1C)=O 69379,Cc1ccc2cc(C(=O)NCCC3CN(C(=O)C(N)=O)CC3C)[nH]c2c1 69380,C(=O)(CCCCCF)N(C(C(=O)NC1CCCN(CC)C1)C)C 69381,n1(C(C)C)nccc1CC(=O)NC1CNC(=O)C1 69382,CC1C=C(C(=O)NCC(c2ccccc2)NC(=O)C=Cc2ccc(F)cc2)CC1 69383,N1(C(c2c(C)cccc2)=O)CC(C)CN(C(=O)C2=CCCOC2)C(C)C1 69384,c12[nH]ncc1S(=O)(=O)N(CCO)C2=O.c1(SCC(=O)OC)cc(F)cc(Cl)c1 69385,c1(C(N2C(C)(CNC(C3(OC)CCSC3)=O)CCC2)=O)cnn2c1NCC(C)C2 69386,n1(CC=C)c(N2CCOC(c3oc(C)cc3C)C2)nnc1CF 69387,Cc1cc(NC(=O)CC2CCN(C(c3cn[nH]c3)=O)C2)cc(C#N)c1 69388,C(=O)(CCCC(C)(C)C)N(CC(C)(C)CN(C(=O)CCCOC1CCCC1)C)CC 69389,N1(C(C2N(C(c3c(COC)cc[nH]3)=O)CCOC2)=O)CCCN(C)CC1C 69390,c1(C(=O)NCCC2CCN(C(C3(O)CCC3)=O)CC2)c(Cl)nc2cc(Cl)ccn12 69391,C1(C(N)=O)CCN(CC(N2CCC2CNC(C2(O)CCOC2)=O)=O)CC1 69392,Cc1n[nH]c(C)c1CCC(=O)N(C(C)CNC(=O)CC1(CO)CC1)C 69393,C(CC(C(C)(C)C)NC(c1cccc[n+]1[O-])=O)N(C)C(c1cnc(Cl)cc1N)=O 69394,c1(SCC)ccc(C(=O)NC2CC2c2ccco2)cc1OC.C1(COC)CC1 69395,N1(C(=O)Cn2ncc3ccccc3c2=O)CC23CCCCC2(C(=O)OC3)C1 69396,C1(CC(=O)NCC(CC2CN(C(CP(C)(C)=O)=O)C2)(C)C)CCC2(CCC2)O1 69397,Cc1ncc2n1CCC(C(=O)NC1COCCN(C(=O)C(=O)NC3CC3)C1)C2=O 69398,CCC(C(=O)NC(CC1CCOCC1)C(=O)NC1CC(O)C(O)C1)C(C)(C)CC 69399,c1(C(N2CCC3(CCCC3=O)C2)C(=O)NCCCF)ccc2ncc(Br)n2c1 69400,N1(C(C(CCC)OC)=O)C2CCC1CC(CN(C)C(c1cc(C)nc(C)n1)=O)C2 69401,C(N=c1[nH]c(Cl)nc2c1CC(C)CC2)C1CN(C(c2ccc(C)[nH]2)=O)CC1C 69402,C1(N(C)C(c2cn(CCNC(c3cc(O)nn3C)=O)nn2)=O)CC(O)C1(C)C 69403,C(=O)(CS(F)(F)(F)(F)F)NC(C)C(C)NC(c1ncsc1C1CC1)=O 69404,CC1(C2CCCN(C(C3CC(NC(C45CCN(CC4)C5)=O)C3)=O)C2)CC1 69405,N1(C(C(C)(C)n2cnnn2)=O)CC(CNC(=O)CC2CC2C(N)=O)C(O)C1 69406,C1(NC(CCOCC)=O)CC1C1CCN(C(c2cn(C)nc2C)=O)CC1 69407,c1(C(=O)NCC2N(C(COC(CC)(C)C)=O)CC2)cncc(-n2ccnn2)c1 69408,CCCC(C(O)C(=O)NCc1ccc(F)nc1C)NC(c1cc(N)cc(F)c1)=O 69409,N1(C(C(C)=CC)=O)CC(NC(=O)CCOc2cccnc2)C2(CCOCC2)C1 69410,CC(C)CC(C)(CNC(c1cc(C(F)F)cc(F)c1)=O)NC(=O)C(F)=CCCF 69411,c1(C(COC)=O)nn(C)cc1C(=O)NC(=O)C(c1ccc(F)cn1)(F)F 69412,C1(NC(C2(C)CC(C)C2)=O)CCN(C(c2ccnc(F)c2)=O)CC1O 69413,CCC(CC)CCCC(=O)N(CC(N1CCc2c(ccn2C)C1)=O)C 69414,N1(C(Cc2c(OC)cccc2)=O)CC2OCC(CNC(C3CC(F)(F)C3)=O)C2C1 69415,c1(SCCN(C2(c3nnnn3C3(C)CC3)CSC(C)C2)CC)cnc(O)c(C)c1 69416,N1(C(C(CCC)C)=O)CCC(O)CC1c1ccccc1.c12ccc(cc1OCC)[nH]2 69417,N12CCCCC3(CCN(C3)CC1)C2.C1(C)(NC(CSC)=O)CCCNS1(=O)=O 69418,c1(C(N(C2CCN(C(=O)CC3CCOC3)C2)CCC)=O)cc(CC)ccn1 69419,N1(C(C(C2CCOC2)OC(C)=O)=O)CCCCC(CNC(=O)C=CC(C)C)C1 69420,c1(C(N2CCC(C)(C(=O)NC(c3cccs3)CC)C2)=O)ccc(C)c(C)n1 69421,C1(C(COC(C(C)c2ncco2)=O)C)CCCCC1 69422,C1(NC(c2ccc(CC)cn2)=O)CN(C(C2CCC(C(C)(C)C)O2)=O)CC12CC2 69423,c1(NC(c2c(CC)c(Br)ccc2)=O)cn2c(n1)CN(C(C)=O)CC2 69424,C(C)(CCC(C)C)(c1nnnn1C[SH](=O)=O)Nc1nc(C)c(C)s1.c1(CN)ccco1 69425,Cc1nn(CC(=O)N(C(C)CNC(=O)C(C)(C)Cc2cnn[nH]2)C)c(=O)o1 69426,CC1(C)C=C(c2ccc(C3(C(N4CC(NCc5n[nH]cc5Cl)C4)=O)CC3)cc2)C1 69427,N1(C(CSC(C)C)=O)CCC(CN(C(CNc2nnc(C)o2)=O)C)C1 69428,C1(NC(COCCOC)=O)CC(NC(c2cc(C)cc(F)c2)=O)C12CCC2 69429,c1(C(=O)NCCN(CC(C)O)C(C2CCC2)=O)cc2oc(Br)cc2s1 69430,C#CCCN=C(NCCc1ccc(Br)c(O)c1)NC1CC(=O)N(CC(C)CC)C1 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69587,N1(C(C2C(C)(C)CC2)=O)CC2CCCN(C(c3ccc(Cl)o3)=O)C2C1 69588,C1(NC(C2CN(C3CCOC3)C2)=O)CC2CC1N(C(c1csc(O)n1)=O)C2 69589,c1(C(c2cn(CCC3CC3)nn2)NCC(CC)NC(=O)NC)cccc(F)c1 69590,C=CCC(CC=C)C(=O)N1C2CCC1CC(CNC(=O)C(C)(C#N)CC)C2 69591,CCC(C(=O)NC(C)CCC(=O)NCCN(C1CC1)C(C)C)C(F)(F)F 69592,C1(OCCNC(=O)NC(C(C)NC(=O)CC(F)F)=O)CCOCC1.C(C)(C)(C)O 69593,CC(C(=O)NC(CC1CCC1)C(=O)N(C)Cc1cnco1)C(F)(F)F 69594,c12ccnc(c1)C(=O)NC2.N1(CC(N2CCC(C(C)(C)O)C2)=O)CCCCC1C 69595,N1(C(c2cc(C#N)c(F)cc2)=O)CCC2(C=C(C(=O)NCC3CC34CC4)C2)C1 69596,c1(NCc2nccc(C(F)(F)F)c2)nnc2ccc(Br)cn12 69597,N1(C(C2(C)CN(C(c3c(CC)n(C)nn3)=O)C2)=O)CCC2(CCC(O)C2)C1 69598,N(C1CN(C(=O)Cn2ccnn2)CCc2ccccc21)C(c1cnco1)=O 69599,n1(CCNC(C2(c3ccncc3)CC2)=O)cc(CCCCCC2CC2)nn1 69600,N(C1CCCc2cnccc21)C(C12COC(C)(C1)C2)C 69601,c1(C(=O)NCCC2CCCCN2C(=O)CCC2CC2CC2CC2)nnn2c1CCC2 69602,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1CC(O)(C(C)NC(=O)C#CC2CC2)C1 69603,c1(C)cncc(Cl)c1.c1(C(=O)NOCC2CCCC2)conc1CNC=O 69604,CCC(CCCC(=O)NCC1Cc2nccn2C1)NC(=O)CCC1CCC(C)O1 69605,c1(CNC(CNC(=O)OC(C)(C)C)=O)csc(CNC(C2CC2F)=O)n1 69606,CCCC(CC)C(=O)NC1CCC(NC(=O)CNC(=O)C=Cc2ccccc2)CC1 69607,c1(C(=O)NCCCN(C(C(n2ccc(C)n2)C)=O)C2CC2)cccc(C)c1C 69608,N1(C(CC(C)CN(C)C)=O)CCOC2(C1)CN(C(c1ccc(CO)nc1)=O)C2 69609,C(=O)(C(O)CC(F)(F)F)NC1C(NC(=O)CCCn2cc(C)cn2)CCOC1 69610,N1(C(c2c(C)onc2C(F)(F)F)=O)CCOC2(CCN(C(=O)CC#N)C2)C1 69611,CCS(=O)(=O)c1ccc(F)c(C(=O)NC2CN(C(=O)C#CC3CC3)CC2(C)C)c1 69612,C(=O)(C#CCC(C)C)NCCCN(C(=O)CCCOCCOC)CC 69613,C1(C(C)C)C(=O)N1.C1(NC(C2(COCC)CCCC2)=O)CCCCC1CN 69614,CC1CCN(C(=O)C2=NOCC2)C(C(=O)NCC(=O)NC2CCC2)C1 69615,N1(C(C(CCCC)F)=O)CCC2CN(CCC3CC3C(C)C)CC2CC1 69616,Cn1nccc1CNC(=O)CCC1(NC(=O)CCn2ccnn2)CCCC1 69617,C(C)(C)(CC(F)C(=O)N(CCN=[N+]=[N-])C)NC(CCC1CN(C)C1)=O 69618,c1(OC)ccccc1C(C)CC(=O)N1CCC(NC(=O)CSc2nnc(S)s2)C1 69619,c1(C(N(CCCNC(C2C(C)C2C)=O)C2CC2)=O)cccc2c1nnn2C 69620,CC1CN(C(C23CC(C2)OC3)=O)CCC1NC(=O)CCc1nc(O)n[nH]1 69621,c1(NC(c2nnc(C)s2)C)ccc(S(=O)(=O)NCC=CCl)cn1 69622,Cc1cc(N)cnc1C(=O)N(C1CCN(C(=O)Cc2cccc(C)c2F)C1)C 69623,CCCCCC(C)NCC(=O)NC1CCN(C(C)(C)C)C1=O 69624,N1(C(=O)Cc2cc[nH]c2)CCCC2(C1)CN(C(C13CC(F)(C1)C3)=O)CCO2 69625,c1(C(N2C(C)(CNC(CCSCCC)=O)CCC2)=O)coc(S(=O)(=O)NCC)c1 69626,c1(NC2(CNC(CCCS(N)(=O)=O)=O)CCOC2)cc2nn[nH]c2cc1[N+](=O)[O-] 69627,C(=O)(C(C)(O)CC(F)F)NCCCCCNC(c1ccc(CN(C)C)o1)=O 69628,c1(CC(=O)NC(CNC(C2CC(F)C2)=O)CO)coc(-c2ccccc2)n1 69629,O=C1Cc2cccc(C(=O)NC3CN(Cc4c(F)cc(I)cc4F)CC3O)c2N1 69630,C(=O)(N(CCC(=O)NCC1CN(C)CCN1C)OC)c1c(C)n[nH]c1 69631,N1(C(C2(OCC)CCC2)=O)C2CCC1C(CNC(=O)Cc1cccnc1Cl)C2 69632,N1(C(C(CN(C)C)O)=O)CCC(C(=O)NCC(O)C2(Cl)CC2)(CF)C1 69633,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 69634,c1(N2C(CC(C)=O)CN(C(c3ccc(CO)cc3)=O)CC2)ncc2cc(C)[nH]c2n1 69635,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 69636,CCC(C(=O)NCCOCCN(C(=O)CC1CCC(O)C1)C)C(C)C 69637,c1(C(=O)NC2(CC(=O)NCC3(SC)CCC3)CCC2)cnn(C=C)c1N 69638,C(=O)(C1=C(Cl)CCCC1)NC(C1CCN(C(=O)CC2CC(O)C2(C)C)CC1)C 69639,C1(O)(C(N2CCN(CCNC(=O)Cc3ccco3)CC2)=O)CC2CCC1C2 69640,N1(C(C(=O)NCCOC(C)C)=O)CC2CC(C1)N(C(C1(F)CC3(CCC3)C1)=O)C2 69641,N1(C(c2c(CC)n(C)nn2)=O)CCCC(C(=O)NCC(F)C2CCC2)C1C 69642,C(CC(C)C(=O)N1CCC(O)(CNC(c2nn(C)cc2SC)=O)C1)=CC 69643,N#Cc1ccccc1C=CC(=O)NC(C1CCOC1)CO 69644,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 69645,C1(C(C2CCOCC2)=O)CNc2ccccc2C1CNC(=O)CCCc1nc[nH]n1 69646,Cc1ccc(C(=O)NCC2C=CC(NC(C3CC(CC4CC4)C3)=O)C2)o1 69647,c1(CC(=O)N(CCN(C(=O)CCN2CCC(F)C2)C)C)ccccc1F 69648,C(=O)(C=CS(=O)(=O)CC)NCC(CC)NC(C1(C(F)F)CC(=C)C1)=O 69649,c1(C(N2C(C(=O)NC(CC(=O)OC)(C)C)CC2)=O)cc(C)nc(O)c1 69650,c1(SCCC)cccc(C(=O)NC(CNC(=O)C(c2cccs2)SC)CO)c1 69651,c1(C(N2CCOCC2c2ccncc2)=O)nc(C2=CCNCC2)cs1 69652,N1(C(C2(OC)CC2)=O)CCN2CCN(C(=O)CC3CCC(=O)N3C)CC2C1 69653,C1(CNC(C(CC)F)=O)CCC2CN(C(c3cc4n(n3)CC(F)C4)=O)CCC2C1 69654,N1(C(C)C)CC2CN(CC34CCCC3C4)CCC12 69655,C1(NC(c2c(CC)nco2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)CC1F 69656,c1(C(=O)NCC2CN(C(C=CC)=O)CC2O)nc(C(F)(F)F)n2ccccc12 69657,C1(COC)CC(C)(C)CN1C(C1CCCC(O)C1)C(=O)NCc1ccc(F)cc1 69658,C1(OC)=CC(C#N)=CC=NC(C2CC2)=N1.C12CC(F)(C1)CNCC1CC1C(=O)N2 69659,Cc1nnc(O)c(C(=O)NC(C)(CNC(=O)C2=NNC(C(F)(F)F)C2)C2CC2)c1C 69660,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(=O)CC2COC(=O)C2)C1(C)C 69661,c1(SCCC(=O)NCC(C(C)(C)C)NC(C2C(C)C2)=O)ccc(Cl)cc1F 69662,c1(CN2CCCC3(C2)n2cc(nn2)C(CC)NC3=O)cc(Br)c(F)cc1O.SC 69663,c1(CC)cc(=NC(=O)C2CCC(CC)N2C(=O)CC2CCCCC23CC3)[nH]n1C 69664,C1(C(=O)NCCC(=C)CNC(=O)C(C(C)C)SC)Cc2nncn2C1 69665,C12(C(=O)NC3(C4N(C(CC5(N(C)C)CCC5)=O)CCC4)CC3)CCN(CC1)C2 69666,c1(C(N(C2CCN(C(C3CC(=O)N3)=O)CC2)CC#C)=O)c[nH]c2cccc(F)c12 69667,c1(C(N(C(C)CNC(c2ccc(Cl)cc2Cl)=O)CC)=O)cccc2c1NCC2 69668,C(CN(Cc1ccc(C(F)(F)F)cc1)N1CCC1(O)CO)N(C)C 69669,C(C(=O)NC(C1CCOC1)CNC(=O)COC)(C1CC1)OCC 69670,c1(OC)ccc(C(=O)NCCn2cc(CNC3CCS(=O)(=O)C3)nn2)c(OC)c1 69671,N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(=O)CCC(C)=O)CC1C 69672,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCCC2)CCC(N=[N+]=[N-])CC1 69673,N1(C(C2CC=C(C)CC2)=O)CC2(C(N3CCCC3CN=[N+]=[N-])=O)CC1CO2 69674,C1(C(=O)NCCN2CCN(C(CNC(C)=O)=O)CC2)CC2(C1)CC(C#N)C2 69675,C1(CC)CN(C(=O)C=CC(=O)NCC)CCN1C(c1cc(C2CC2)ns1)=O 69676,C1(C(N(C)C)=O)C2CN(C(=O)C(F)CC3CCOC3)CC12.Cc1cc(C)on1 69677,C1(CNC(CSCC#C)=O)CN(C(C2CN(C(=O)OC)C2)=O)CCN1C 69678,CC1CCN(C(=O)C(=O)NC(C)(C)C(C)NC(=O)CCCc2ccsc2)CC1 69679,C(CCC(=O)OCCC1CCN(C(=O)OC(C)(C)C)C1)OCC 69680,C1(CCNC(C(c2cncnc2)C)=O)CCC(C(=O)NC(C2CCCC2)C)C1 69681,C1(C(=O)NCCN(C(C)C)C(c2ccoc2Br)=O)C(C(C)=O)C1[N+](=O)[O-] 69682,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 69683,c1(CCNC(C(=O)OC)Cc2ccc(C(F)(F)F)cc2)c(C)nn(C)c1C.C(C)(C)C 69684,CC(N=c1[nH]c2c(c(=NCCOc3ccccc3)[nH]1)CCCCC2)C1CCOC1 69685,C1(NC(c2c(CC)cccn2)=O)CN(C(c2cnsc2)=O)CCC12CCC2 69686,c1(C(C#N)C(=O)N2CCCC2c2ccccc2I)ccccc1N1CCCCC1=O 69687,C=CC(C)(O)C(=O)NCCCN(C)C(C1(c2cccs2)CC1)=O 69688,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 69689,N1(CC)CCN(c2nccc(-c3csc4ccccc34)n2)C2CCCCC2C1 69690,Cc1cc(C(=O)NCCn2c(C)ccc2C)c(Br)nc1C 69691,Cc1cc(C)c(C(=O)NCc2cc(C(=O)Nc3ccsc3C(C)C)n[nH]2)s1 69692,c1(C(N2C(C(NC(c3c(OC)c(=O)cco3)=O)CC)CC2)=O)c(C)ccc(C)c1C 69693,c1(C(=O)NC2CC(NC(=O)CCc3cccnc3Cl)C2)cccc2scnc12 69694,C1(NC(C(C)OCCN(C)C)=O)CC2CC(NC(c3n[nH]c(=N)s3)=O)C2C1 69695,C(=O)(CC(F)(F)F)NCC(=O)NC1C(NC(C(n2c(C)ccn2)C)=O)COC1 69696,C1(C(=O)NCCC(C)N(C(=O)CN=S(C)(C)=O)C)CNc2ccnn2C1 69697,C1(CC(=O)N(CC(C)N(C(=O)C(=O)Nc2ccccc2)C2CC2)C)COCCN1C 69698,CCCC(CC(=O)N(C1CCCC1)CC(N)=O)NC(=O)C(CC)N(C)C 69699,C(CCNC(=O)C(C)C#N)(C(=O)NCc1cncc(Cl)c1)OC 69700,C1(C)(C(N(C2(C)CC2)CC)=O)CC12CCN(C(C)C(c1cccc(Br)c1)=O)CC2 69701,C1(C(=O)NCc2cc(CC)[nH]n2)CC2(CCC2)CN1C(=O)Cc1ncccc1F 69702,N1(C(CCCCCC=C)=O)CCC2CN(C(c3cn(C)nc3CC)=O)CC2C1 69703,CCCCCCC(C(=O)NC1CCOC1=O)n1cc(CCSC)nn1 69704,c1(C(=O)NCC2(NC(C3CCC(O)C3)=O)CCOC2)cc(Cl)c(Br)[nH]1 69705,N1(C(C(=O)NC(CC)C)CC2CCCOC2)Cc2ccc(Br)cc2CC1C 69706,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 69707,C1(C2CC2)(CNC(CSC)=O)CCN(C(=O)C(C)(C)C(=O)OCC)C1.C(C)(C)(C)O 69708,c1(C(=O)NCCNC(c2c(OC)cc(Cl)cc2)=O)c(O)ncc2c1CCC2 69709,C1(CCN(C)C(c2ccc(F)cc2)=O)CCCCN1C(c1n[nH]cc1Cl)=O 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70064,C1(C(=O)NCC2CCC(NC(C3CC(=C)C3)=O)CC2)CN(CP(C)(C)=O)C1 70065,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(C2CCCCO2)=O)CC1CO 70066,c1(C(=O)NCC(C2(O)CCN(C(C3CCCCC3O)=O)C2)C)cccc(CO)c1 70067,CC(O)C(F)(F)C(=O)N1CCC(CNC(=O)CCNC(c2ccccc2F)=O)C1 70068,C1(C(=O)NCCN(C(c2cc(C)ncn2)=O)CC2CC2)CCS(=O)(C)(C)C1 70069,c1(C(N2C(C(C)NC(c3ccsc3)=O)CC(F)C2)=O)cn(C)cc1C(F)(F)F 70070,c1(C(C)NC(=O)NC(Cc2ccnn2C)C2CC2)ccc(F)c(F)c1 70071,Cc1cc(C(=O)NC2CCCC(NC(=O)CCNS(C)(=O)=O)C2)cc(C)c1 70072,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70073,c1(C(C)NC(=O)C(C2CC3(CCC3)C2)(F)F)ccc([N+](=O)[O-])c(O)c1 70074,Cc1c(Br)ccc(O)c1C(=O)NCC1CCCN1C(C1(C)C=CCC1)=O 70075,C1(CC)CC(C(=O)NCCN2CC=CCC2)CCN1C(C1CN(C)CCO1)=O 70076,O=C(C(O)Cc1ccsc1)NC1CC(F)(CNC(=O)CCc2cscn2)C1 70077,C1(C)(CNC(C2(OC)CC2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 70078,C(=O)(CCS(C)=O)N(C)CC1(O)CN(C(=O)C(C)(C)c2ccccn2)C1 70079,C1(NC(=O)CC2CCCC2)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70080,C1(C(N2CCCC2Cn2ccccc2=O)(C)C)CCN(CCn2ncc(Br)n2)CC1 70081,N1(C(CC2CCC(C(=O)OC)C2)=O)CCN(C(=O)CC(C)(C)C2CC2)C(CF)C1 70082,C1(CC#C)(C(=O)NCCNC(=O)CCOCC2CCC2)CCOC1 70083,C1(C2(C(=O)NCCCCNC(CC(C)NC(N)=O)=O)CC2)CCCCN1C.C(=O)N 70084,N1(C(Cc2n(C)ccn2)=O)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70085,C1(NC(CC(C)OC)=O)CCN(C(=O)CCF)C1(C)C 70086,CC(C)C(C)C(CNC(=O)CCc1cocn1)NC(=O)Cc1ccc(Cl)cc1F 70087,c1(C(N2CC3(C(C(=O)OCC)C3)C2)=O)cc(C)ccc1OCC(F)(F)F 70088,C1(CC(=O)NCCC(=O)NCCC)CC(NC(c2n[nH]cc2C(C)C)=O)C1(C)C 70089,c1(N2CCCC(SCC(N3CCS(=O)(=O)CC3)=O)C2)ncccc1[N+](=O)[O-] 70090,C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(C(C)C)=O 70091,c1(OC)cccnc1CN1CCC(C)(C(=O)NCC2CCO2)C1 70092,c1(C(=O)NCC2CC(NC(c3cnc(C(C)(C)C)s3)=O)C2)ccn2ccccc12 70093,N1(Cc2cn(CC(C(=O)OCC)C)nn2)CCC12CCSCC2 70094,c1(C(=O)NC(CSCC(=O)NCC)C(C)(C)C)ccc2cc(C(C)C)ccc2c1 70095,c1(CC)ccc(C)c(C(=O)NC2(CF)CCN(C(=O)C(C)C(C)(C)C)C2)c1 70096,c1(N(C(=O)CC2CCN(C(=O)Cn3cnnn3)CC2)C)ccccc1Cl 70097,C1(C(N2C(C(N(C)C)=O)CC2)=O)CCCC1CNC(=O)CC1(O)CCC1 70098,c1(C(=O)NC2CC(CNC(=O)CC3CC4COCC34)C2)cc2n(n1)CC(F)C2 70099,CC1CC(NC(c2cnc(C(F)(F)F)s2)=O)CCN1C(C1CC12CCCCC2)=O 70100,N1(C(c2c(C)n(C)cn2)=O)CC(C(=O)NCc2cnn(C)c2O)CC1(C)C 70101,C(C#Cc1cccnc1)NC(c1cccnc1CNC(C1CC2(CC2)CO1)=O)=O 70102,N1(C(C(=O)NCCN(C)C(C2CC(OC(C)(C)C)C2)=O)C)CCCC(O)C1 70103,c1(C(N2C(C(=O)NCC=C)CCC2)=O)cc(C)oc1CNC(=O)COC 70104,N=c1nc(CC(=O)NCC2CC(C(N3CC(n4cccn4)C3)=O)C2)[nH][nH]1 70105,C(C1=CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1)NC(CC1CCC(C)CC1)=O 70106,N1(C(C)=O)CCC(C(c2nc(-c3ccccc3)no2)NC(=O)COC)C1 70107,C1(C)(C(=O)NCCC2(NC(C3CCCN(C(C)=O)C3)=O)CCC2)CCC2CC2C1 70108,C1(C(=O)NCC(CC)(C)OC)CCN(C(C2CC=CCC2C)=O)C(C)(C)C1 70109,N1(CC(=O)NCC#CC(=O)NCC(n2cccn2)C)CCCCC1=O 70110,C1(CNC(c2c(C)nsc2)=O)CCCCN(C(=O)CCc2ccccc2)C1 70111,N(C1CCCc2cc(CNC(c3cnc(S)n3C)=O)ccc21)C(C(F)=C(C)C)=O 70112,Cc1ccc(CCCC(=O)NC(C)C(C)(C)NC(c2conc2C)=O)cc1 70113,c1(NC(c2c(C)c[nH]c2C)=O)ccc(C(=O)Nc2ccc(F)c(CO)c2)cc1F 70114,c1(OC)ccc(COCCC(C)C)cc1OC.N12CCCCC1CNC(=O)CC2 70115,c1(C(N(C2CCN(C(=O)CCCC#N)CC2)CC)=O)cc2ccsc2s1 70116,CCC(CC(=O)NC(C(=O)NC1CCSC1C)C(C)O)C(F)F 70117,C12(C(=O)NC3(CC(C)(C)O)CC3)CC(CN1C(C1C3CCC(F)C13)=O)C2 70118,C1(c2cn(C(COCC)C(=O)NC3(C4CC4)CCCC3)nn2)CCCC(C#N)C1 70119,N1(C(c2c(C(C)C)cco2)=O)CCCN(CCCCNC(C2CC(F)C2)=O)CC1 70120,Cc1c(CNCC2C3CN(C(=O)CC4CCCN(C)C4)CC23)cccc1O 70121,C#CCCCC(C)C(=O)N1CCOC(C(=O)NC2CCCC2N(C)C)C1 70122,C#CC1(NC(=O)CC2CCCN(C)C2)CCCN(C(=O)C(C)=C2CCC2)C1 70123,N1(C(=O)COC2CCOC2)CCCC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 70124,C1(NC(CN(C)S(N)=O)=O)CCCC12CN(C(=O)CCn1cc[nH]c(=O)c1=O)C2 70125,c1(C(N(C2C(CSC)CCC2)C)=O)cc(F)oc1C 70126,C(=O)(C(C)CC(C)C(C)=O)N1CCC(C)(CC(=O)NCC2N(CC)CCC2)C1 70127,C1(CNC(CC2CCC(C)O2)=O)CC2CCC1N(C(c1cc3n(c1)CCCC3)=O)C2 70128,c1(C(N(C(CNC(c2ccc(C)c(O)n2)=O)C2CC2)C)=O)ccc2[nH]ccc2n1 70129,N1(C(c2c(C)c[nH]c2CC(N)=O)=O)CCC2(CC1)OCC(C)(O)C(O)C2O 70130,c1(CN(C)C)ccc(C(=O)NCC2CCN2C(c2csc(Br)n2)=O)[nH]1 70131,C#CCC(C)C(=O)N1CCC(C(C)NC(c2ccc(C3(C)CCO3)cc2)=O)CC1 70132,C1(N(C(COCCOC)=O)C)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC1C 70133,N1(C(C2N(CCC)CCCC2)=O)CCC(F)(CNC(=O)CC(C)(C)O)CC1 70134,N1(Cc2cncc(OC)c2)CCC(C2CN(C(=O)C(C)CNC(C)=O)C2)CC1 70135,c1(C(N(C)CC2CN(C(c3ncccc3Br)=O)CCO2)=O)ccc(CO)c(Cl)c1 70136,C(C)(C)(C=CC(=O)NCCC1CC(C(N2CCC2)=O)C1)SC 70137,C(CCC(C)CCC(=O)O)SC(C(=O)Nc1c(OC)ccc(C)c1)C 70138,c1(C(=O)NC(CNC(C(C)c2ccsc2)=O)C(C)(C)C)cc2occc2s1 70139,C1(C(N2C(CCNC(c3n(C)cc(C#N)c3)=O)CCCC2)=O)CNC(=O)C(C)(C)C1 70140,C(C(=O)N1CC(CNC(C2(C(C)(C)O)CC2)=O)C1)(C(C)C)OCC 70141,c1(-c2nc(C(CC)C)nn2CC)cc2c(OC(c3cn(C)nn3)C)cccc2[nH]1 70142,C1(NC(c2c(CC)ocn2)=O)CN(C(=O)CSCC(C)C)C(C)(CC)C1 70143,C(CCCCC(=O)NCCN(C(C1CCC(F)CC1)=O)C1CC1)COCC 70144,Cc1nn(C)cc1CCC(N1CCN(C(=O)CN(C(=O)C(C)C)CC(C)C)CC1)=O 70145,CC(C)C(C(=O)NC1C=CCN(C(=O)CCSc2ccccn2)C1)NC(N)=O 70146,C#CC1(N2C(=O)C2)CCOC1.C(=O)(C(C)OCC1CCC1)NC(C)C 70147,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(O)C1CCC1 70148,N1(C(CC2C(=O)OCC2)=O)CCC12CN(C(C1CCCCCC1)=O)C2 70149,Cc1c(C(=O)NCC2COC(C)(C)CN2C(=O)C=CC2CCC2)nc2sccn12 70150,c1(COCCNC(C=C(C)CNC(C2C=CCS2)=O)=O)nc[nH]n1 70151,c1(NC(C(Cc2cn[nH]c2)NC(CC=CCCCCC)=O)=O)cccc(OC)c1 70152,N1(C(=O)NC(COc2c(C)cccc2)(C)C)Cc2cnc(N(C)C)nc2C1 70153,C1(C(=O)NCCOC2CCCCC2)CCN(C(c2cc(Br)ccc2F)=O)CC1(F)F 70154,c1(C(N2CC(C)CC(C)C2)C(=O)NCC2CC2)ccc(S(=O)(=O)C(F)F)cc1 70155,N1(SC)CC(C(N2CCCC(N(C(=O)C(C)Sc3ccncc3)C)C2)=O)CC1=O 70156,C(C)(CCS(C)(=O)=O)(c1n(CCSC)nnn1)NCC1(C)CSC1 70157,CC(C)CC(C)C(=O)N(C1CN(C(=O)CC2COCC2(C)C)C1)C 70158,C1(NC(C(c2cn(C)nc2)=O)=O)CC(NC(=O)CCN2CCCCC2)C12CCC2 70159,Cc1cc(C)c(C(N2CCN(C(=O)CC3COCCN3C)C(CO)C2)=O)c(C)c1 70160,c1(C(C)N(C(C2CC(NC(=O)OC(C)(C)C)C2)=O)CC2CC2)nc(Br)cs1 70161,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCCOC.c1(C(=O)N)ncoc1C1CC1 70162,c1(NC(C2N(C(=O)CS(N)(=O)=O)CCC(C)C2)=O)ccc2[nH]nc(Cl)c2c1 70163,c1(C(=O)NC2(C(=O)NCCc3ccncc3)C(C)C2)ccc(CO)o1 70164,C(CCN(C(=O)C(C)(C1CC1)OC)C)(C(C)(C)C)NC(C(CC)CC)=O 70165,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)ncn1)=O)C2 70166,C=CCC(F)(F)C(=O)NCC(F)CNC(c1ccc([N+](=O)[O-])o1)=O 70167,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)oc2c1 70168,Nc1ccc(C(N2CCOC(CNC(C3CCCS(=O)(=O)N3)=O)C2)=O)c(Cl)c1 70169,c1(CC)cccc(CNC(=O)CSCCNC(C2CCC(F)C2)=O)c1 70170,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70171,C1(CNC(CSCCOC)=O)CN(C(=O)C(N2CCN(C)CC2)C)CC1(F)F 70172,c1(NC(CCN(C(C(C)c2cccs2)=O)C)=O)ccc(C2CC2)nc1 70173,CCCC(O)C(=O)N1CCC(OCCNC(c2coc(C#N)c2)=O)C1 70174,c1(C(N(C(CC(=O)NC(C)C(C)(C)CO)(C)C)C)=O)cc(F)cnc1O 70175,c1(C(=O)NC2CCN(CCCOC)C2=O)noc2cc(Br)ccc12 70176,C(C(C)N=c1nc(OC)cc(OC)[nH]1)N(C(CCCCC(=O)NC)=O)C 70177,CC1CN(C(=O)C(=O)NC2CCCCC2)CC1C(=O)NOCC(F)(F)F 70178,C1(NC(c2ccn(CC)c2C)=O)CN(C(C23CCCC2C3)=O)C2(CCCCC2)C1 70179,C(CC(C(=O)NCC1CCCCO1)NC(=O)CC1CCC(=O)C1C)OC 70180,C(CCCCCNC(=O)CC1CCCC1)NC(c1cc(CCC)[nH]n1)=O 70181,C=C=C(C)CC(=O)NCCCC1CCCN1C(=O)Cc1nccn1C(F)F 70182,C(=O)(C1=CCCCO1)N(C1CCCN(C(C2C(C(=O)OCC)C2)=O)C1)C 70183,N1(C(CCN(CC(F)(F)F)C)=O)CCN(C(=O)C(N2CCCCCC2)C)C2CCC12 70184,C1(CC)(NC(=O)CC2CC(C)=NO2)CN(C(C2(C)CC2(F)Cl)=O)C1 70185,c1(OC)ccc(C(C)NC(=O)NC(C)Cc2ccc(F)cc2)cc1C 70186,N#CC1CN(C(CCCCC(=O)OC(F)F)C(=O)NCCCF)CC12CCC2 70187,C1(C=O)CCCC(O)CC1.C1(N(N2CC(C(O)C(=O)N)C2)C)CC(CO)C1 70188,CC(C)(CCCO)C(=O)NC1CC(NC(C2CS(=O)(=O)C2)=O)C1 70189,c1(C(=O)NCC2(NC(C3CCS(=O)(=O)CC3)=O)CCC2)[nH]c2ccccc2c1Cl 70190,CCCC(C(=O)NC(C1CN(C(c2coc(C#N)c2)=O)C1)C)S(N)(=O)=O 70191,c1(C(N2C(C(=O)OC)CCC2C(C)(C)C)C(=O)NCC(C)C)cc(Br)ccc1C 70192,c1(OC)cc(C)cnc1C(=O)NC(CNC(=O)CC1(n2cccn2)CC1)CO 70193,N1(C(c2n(C)ncn2)=O)CCC2CN(C(=O)CC3CSC3)CC2C1 70194,Cn1cnc2ccc(C(=O)NCC3CC4CC4N3C(C3CC3c3cccs3)=O)nc12 70195,Cn1ncc2nc[nH]c(=NC3CCCC(C(=O)NCc4ccc(O)nc4)C3)c12 70196,CP(C)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(c2ncccc2N)=O)cc1 70197,c1(C(=O)NC2CCCC(CC)C2)nc2cc(C)ccc2n1C 70198,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70199,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2ccoc2Cl)=O)C(C)(C)C1 70200,C(=O)(CC(C(=O)NC1CCCCC1NC(=O)Cn1nnnc1C)N(C)C)OC 70201,C1(C(N2C(C(N3CCC(O)(C4(C)CC4)C3)=O)CC(C)C2)=O)C2CCC(C2)C1C 70202,c1(C(=O)NC2CC(CCC(=O)NC3(CCCC)CC3)C2)cnc(C)n1C 70203,Cc1c[nH]c(NC(=O)CCc2cccc(C(=O)OC)c2)c1C.N12C(CCC1C)C2 70204,N1(C(C(=O)NC2C(NC(CCCC)=O)COC2)CC)C(=O)CCC1=O 70205,N1(C(CN2CCC2)=O)CC(C)CC(C)C1.c1(SCC(=O)NC)ccccc1C 70206,C=CCC(CNC(=O)C(C)(C)N(C)C)NC(=O)C(C)=C1CC1 70207,C1C(C)C(=O)N(C)CC(=O)N(CC)C(C)C(=O)N1.CCCCS 70208,c1(C(N(C2C(C)CCN(C(CCCC#CC)=O)C2)C)=O)cc(F)cc(Br)c1F 70209,C1(C(N(C)CCNC(=O)CSCc2ccsc2)=O)CC2(C1)CC(F)(F)C2 70210,c1(C2(CC(=O)NCC(CNC(C3C(COC)C3)=O)(C)OC)CC2)ccccc1F 70211,C(=O)(C(CNC(=O)CC1CC=CCC1)C(C)(C)C)NC(C1CCCCC1)C 70212,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70213,N1(CC(=O)NCC(CO)NC(C2(OCC)CC2)=O)CCS(=O)(=O)CC1 70214,N1(C(CC(CC)C)=O)CCC(C2CC2NC(c2cc(C)cc(Cl)c2)=O)CC1 70215,Cc1ccccc1C(F)C(=O)NC1CCN(C(c2cnccn2)=O)CC1 70216,c1(OC)cc(C)c(C(C)(C)CN(C(CCCSC)C(=O)OC)C)cc1OC 70217,N1(C(COC(C)=O)=O)CC2CCC(NC3CCC3)C2C1 70218,C(=O)(C1=CCCN(C(C2(COC)CCCO2)=O)C1)NC(CCCC)(C)C 70219,CCC(CC(=O)NCCCCn1cc(CC(O)C2CC2)nn1)CC(F)(F)F 70220,S(=O)(=O)(CC(=O)NC1C2CC1N(C(c1ncccc1CCOC)=O)C2)NCC 70221,N1(C(C2CC(OC)C2)=O)CC2CCCC(NC(c3cc(C(N)=O)ccn3)=O)(C2)C1 70222,C1(C(N2CC(C(N(CC(C3CCC3)OC)C)=O)OCC2)=O)CC(=O)NC1(C)C 70223,C(=O)(C(O)C(F)(F)F)NC(CN1CCN(C(c2n(CC)ncn2)=O)CC1)C 70224,c1(NCC(=O)NCc2ccncc2)ccnc(OC(F)F)c1 70225,c1(C(=O)NC2CCC(CNC(C(C)c3ccco3)=O)CC2)ccn2cnnc2c1 70226,C1(C(=O)NC2CON(CC)C2=O)CC(C)(C)CCN1C(C1CCC1C)=O 70227,C1(C(=O)OC)CN(C(C(=O)NCc2ccccc2)C2CCC2CO)C2(CCC2)C1 70228,c1(C(=O)NC2(C)CN(C(C3CCC(F)(F)CC3)=O)C2)cncc2c(O)nccc12 70229,c1(CC(N2CCC(C)(CNC(C3CCNC3=O)=O)C2)=O)ccc2c[nH]nc2c1 70230,N1(C(CC(C)CF)=O)CC2(C)CC1(C(=O)N(C)CC1(C)CCCC1)C2 70231,C(C(CC1CC1)C(=O)N1CCC1(C)CCO)NC(C1CC(N(C)C)C1)=O 70232,C=CCC(C)C(=O)NCCCCC1CN(C(=O)C2=CCOC2)C1 70233,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70234,c1(NC(C(CC=C)CNC(C2Cc3nccn3C2)=O)=O)cnc(C)c(C)c1C 70235,c1(CC(=O)NC2(C)CN(C(C(C3CC(F)(F)C3)C)=O)C2)ccccc1C1CC1 70236,C=CC(C)C=O.O(NC(=O)CN1CCC(CC(C)C)C1)CCO 70237,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70238,C1(C(N2CCN(CCCNC(=O)CC3CCCO3)CC2)=O)CC(=O)C12CCC2 70239,C12(C(N(CC(C)C(=O)NCCc3nc[nH]n3)C)=O)CCCC1C2(F)F 70240,CN1CCC(C)(C(=O)NCC2CCCCN2C(=O)C=Cc2cccc(F)c2)CC1 70241,c1(SCC(=O)N(CCC(C)NC(C(CCSC)O)=O)C)ncnc2[nH]cnc12 70242,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70243,c1(C(=O)N=c2ncs[nH]2)ccc2c(c1)oc1ccccc21 70244,c1(C(=O)NCC2CCN(C(CC=C)=O)C23CCC3)ccc2nc(N(C)C)sc2c1 70245,C1(CNC(CC2(C=C)CCC2)=O)CCN(C(c2ccc(N)c(O)c2)=O)C12CCC2 70246,CC1CN(C(c2cc(Br)n(C)c2)=O)CC1NC(C1CC12CCC2)=O 70247,C1(C(=O)NC(C)CCNC(c2conc2Cc2ccccc2)=O)CCCC(=O)O1 70248,C(=O)(C(F)(F)C1=CCOCC1)NCC1CN(C(C2C(C=C)OCC2)=O)CC1O 70249,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70250,C(c1ccc(F)cc1)=CC(=O)OC1(COc2ccc(F)c(F)c2)CC1 70251,C(C(CO)(CO)NC(=O)C=Cc1cn[nH]c1)N(C(=O)CCC1(C)CCC(=O)N1)C 70252,CC(C#N)C(=O)NC(CC1CCCC1)C(=O)NCC(O)C1(Cl)CC1 70253,C(=O)(CC(C)CC(C)C)NCC1(CCC=C)CN(C(C2CN(C)CCO2)=O)C1 70254,n1(CC(N2C(COC)CCC2)=O)cc2ncccc2n1 70255,c1(C(=O)NC(CC)CN(C)C)ccc(CCNC(=O)CC2CNC(=O)C2)cc1 70256,C1(c2cccc(NC(CC)C3CC3c3cn(C)nc3C)c2)CCC(F)(F)CC1 70257,C1(C(=O)NC(C2CCCN2C(C2CC(O)C2)=O)C)CCc2nnnn2C1 70258,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70259,C1(=O)CCCCC2CN1C2.CC1CCC(C(=O)NCc2ncoc2C(F)(F)F)O1 70260,c1(NC(C2N(C(CCS(C)(=O)=O)=O)CC=C2)=O)ccc2nc(Cl)sc2c1 70261,c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)(F)C2)nc2c(s1)CCCC2 70262,N1(CCNC(c2cnsn2)=O)CCN(C(C23CC(C(F)(F)F)(CO2)C3)=O)CC1 70263,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70264,c1(C(=O)NC2C(NC(CCC(C)CN(C)C)=O)COC2)cnc2c[nH]nc2c1 70265,Cn1nc(C(=O)NC2COCC2CNC(=O)CC2(C)CC2(F)F)c2ccccc12 70266,c1(C(=O)NCC2N(C(C3CC(CCC)C3)=O)CCCCC2)cccc2sncc12 70267,O(C1CCCc2ccccc21)CC(=O)NCC(CO)NC(C=C1CCC(C)C1)=O 70268,C1(CC)CN(C(c2cccc[n+]2[O-])=O)CCN1C(C1NC(=O)C2CCC12)=O 70269,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(N(C(=O)C=C(C)C2CC2)CC#C)CC1 70270,C1(C)(C(=O)NCC=CCC(=O)NCCCC(=O)NC)C=CCCC1 70271,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1C(NC(c2ccc(OC)nc2)=O)C1 70272,N1(CCCCN2C(CCOC)(C)C2=O)CCC2OCCN(C(=O)C3=C(Cl)CC3)C2C1 70273,C=C(Cl)C(C)(C)C(=O)NCC12CC1CN(C(c1ccccc1OC(F)F)=O)C2 70274,Fc1cncc(SCc2ccncc2)c1.c12nc(-c3ccnc(Cl)c3)nn1CC2 70275,C(=O)(CC(C)C(F)(F)F)NC(CC1CN(C(C=CC=CC)=O)C1)C 70276,CC(CC(=O)NCC(CC(=O)N1CC(N2CCCOCC2)C1)C1CCC1)C(F)F 70277,C(=O)(C#CC1CCCCC1)N1C(CNC(C2N(CC)CC2)=O)CC2(CC2)C1 70278,C1(C(=O)NCCNC(Cc2c(Br)cn(C)n2)=O)CC2C=CC1CC2 70279,N1(C(c2c(F)ccc(C)n2)=O)CC(C(N2CC(C(N)=O)C3(CC3)C2)=O)C2(CCC2)C1 70280,C1(CN(C(=O)CC2CC(C)(C)CO2)C)CC(C(F)(F)F)CN1C(C12CC(C)C1C2)=O 70281,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70282,c1(COC)cc(N2CCC(NC(C3C4CC5C(C4)C35)=O)C(F)C2)nc(SC)n1 70283,CC1(C)C2CCC(C(=O)NCC3(O)CCN(C(=O)CNC=O)C3)C1C2 70284,C1(CNC(c2c(CC)cco2)=O)COC(C)(C)CN1C(c1cc(N)nc(Cl)c1)=O 70285,c1(C(=O)NC(C(CO)NC(C(CC)NC(N)=O)=O)C)cnc(NC2CCC2)cn1 70286,c1(N(C)Cc2nc3ccc(Br)cc3s2)nc(Cl)nc2c1cnn2C 70287,N12CC(C(C)C1)NC(=O)c1cccc(c1)NC(C)C2=O.C(C(C)C)SC(C)C 70288,c1(C(=O)NCCOC2CCN(C(CC3C(C)C3)=O)C2)cc(C#N)ccc1F 70289,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70290,c1(N2CC(CNC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70291,C1(c2n(CCCSC)nnn2)(NC2(C(C)C)CCOC2C)CC2(C1)CC(C)(C#N)C2 70292,C1(CC)C(C(=O)N(C(C)CC(F)(F)F)CC)CCN1C(C1CC2C=CC1O2)=O 70293,CC1(C(=O)NC(C)(CNC(c2ncccc2C2CC2)=O)C2CC2)CCOCC1 70294,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70295,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncnc2C)=O)c(C)c1 70296,C(=O)(CCCC(=O)NCC(=O)NC1CCOC(c2ccncc2)C1)NC 70297,CN1CCC(C(=O)NC(C(=O)NCC2(C(C)(C)O)CC2)C2CCC2)C1=O 70298,c1(CNC(=O)CC(F)(F)F)ccccc1CN(C)C(C1C(C)CCC1)=O 70299,c1(CC)ccccc1CC(=O)NCC(C(C)C)NC(C1CCCC1F)=O 70300,N1(C(CNS(CC)(=O)=O)=O)CCC(CNC(c2cccnc2C)=O)CC1C 70301,C1(C)(CNC(C(CC)(C)C)=O)CN(C(C2CC(C)(C(=O)OC)C2)=O)C(C)(C)C1 70302,N1(C(C2CN(C)C(=O)CC2)=O)CCC(NC(=O)Cn2ccnn2)C12CCC2 70303,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70304,N1(C(=O)OC(C)(C)C)CC2(CCC2)CC1CNC(c1ccc2ncnn2c1)=O 70305,c1(C(=O)NCC(N2CCCC(C(=O)OC)C2)=O)cc(S(C)(=O)=O)cc(F)c1Cl 70306,CC1(C)CC(NC(=O)C=CC(=O)NCC2CC2)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70307,c1(CCC(=O)NC2CC(C(C)NC(=O)C(C)(C)n3cccn3)C2)ccc(Cl)s1 70308,C(=O)(CC(C)CNC(C1COCC(C)O1)=O)NCCc1cnc(C)[nH]1 70309,C1(CNC(=O)Cn2cc(Cl)cn2)CCC(CNC(=O)Nc2ccc(Cl)nc2)CC1 70310,C1(CNC(c2ccc(CC3CC3)s2)=O)CN(C(c2ccccn2)=O)CCO1 70311,O=C1CCc2nc(NC3CCCC(NCc4cc5ncccc5o4)C3)ccc21 70312,N(C1CCc2cccnc21)C(c1cc(-c2c(CN3CCCC3)cccc2F)[nH]n1)=O 70313,c1(C(N2CCC(C(=O)NCCCO)C(O)C2)=O)ccn2cncc2c1 70314,S(=O)(=O)(c1ccc(N(C)Cc2ccc(Cl)cc2)cc1Cl)NC(C)CCCO 70315,C1(C(=O)NC2(CCNC(c3c(C)nsc3)=O)CCC2)CC2CCC(C1)C2 70316,c1(C(N2CCCC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)cnc2n1CCCC2C 70317,c1(CCC(=O)NC(CNC(=O)Cc2cc[nH]n2)C2CC2)nc(C2CC2)no1 70318,C1(CCN(C(=O)Cc2ccc(C(F)F)cc2)C)CCCCN1C(=O)C=CCF 70319,C(=O)(CCCCCCNC(=O)C=CC)NCCC=CCC 70320,CCCC(C)CC(=O)NC(CNC(c1cc(C)cnc1Cl)=O)CC(C)C 70321,C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCCC1NC(=O)CCCCOC 70322,N#Cc1ccccc1NCC(N1CCN(C(c2cccnc2)=O)C(C(=O)O)C1)=O 70323,c1(C(N(C2CCN(C(=O)C(C)C#N)C2)CC)=O)cn(C)nn1 70324,C1(C2CC2)(C(=O)NCCC(=O)N(C)C)CN(C(=O)C(F)C2CCOC2)C1 70325,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(NC(=O)Cc2csc(Br)n2)C1 70326,c1(C(=O)NCC2OCCN(C(c3cc(CO)[nH]n3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 70327,C1(C2(NC(c3c(CC)nc[nH]3)=O)CC2)CCN(C(C2CC23CCOC3)=O)CC1 70328,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc(O)c2ccccc2c1 70329,C1(C(N(C2CCCCC2N(C(=O)C2=CSCCO2)C)C)=O)CCCCNC1=O 70330,c1(C(=O)NCC(CCCC)NC(=O)C2=C(C#N)CCC2)cnc2ncnn2c1C 70331,Cc1cccc2cc(NC(c3oc(CNC(=O)NCCCl)nc3C)=O)cnc12 70332,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70333,c1(C(=O)NCc2c(C(=O)OC)nn(C)c2)ccc2cccnc2c1F 70334,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70335,C1(CC#C)(C(=O)NC2CCOCC2C)CCN(C(c2csnn2)=O)C1 70336,CC1(C)CC(C(=O)NCC2CN(C(=O)C3CC3)CC23CC3)CCO1 70337,O(NC(=O)C(O)C1CN(C(C2(CC)CCC2)=O)C1)OCC#C 70338,C#CCCC(=O)NCCN(CC(=O)NCC(F)F)CCOCCOC 70339,C1(NC(C=C(NC(C)=O)C(N)=O)=O)CC2CCC(C1)N2C(c1ccccc1O)C 70340,C(=O)(C(CO)C(C)(C)C)N1CCC(C(N2CC(CC(=O)NC)C2)=O)(OC)C1 70341,c1(C(=O)NC(CC)CNC(=O)CCCCOC)ccnc2[nH]ncc12 70342,C1(NC(=O)CC(C2CC2)C2CC2)CCC2CN(C(=O)CC3CCOC3=O)C2C1 70343,c1(C(=O)NCC23C(CN(C(c4sc(C)c(O)n4)=O)C2)C3)ccc2nc(O)[nH]c2n1 70344,N1(C(C(C)=O)=O)C2CCC1CC(CNC(c1cc(Cl)ccc1OC(F)(F)F)=O)C2 70345,C1(N(C2CC(OC(=O)C(C)C)C2NCc2ccccc2)C)CN(CC)CCO1 70346,c1(C(N2CCCC(CNC(c3ccc(F)c(I)c3)=O)C2)=O)cc(F)cc(=O)n1O 70347,C12(c3scc(-c4n(CC)ncc4)n3)CCC(S)(CC1)CC2.N1(C=O)CCC(C)(O)C1 70348,CCCC(CCCNC(=O)Cc1sc(C)nc1C)NC(=O)C(C1CC1)OC 70349,c1(C(c2n(CCC)nnn2)N(CC(C(C)C)SC)CC)ccc(Cl)cc1 70350,c1(C(=O)NCCOCCN(C(C(CC#C)O)=O)C)cc2c(nn1)CCCO2 70351,Cc1cc(C(=O)NC2CCCCC2NC(C2(CO)CCOC2)=O)cc(C)c1Br 70352,Cn1cc(Br)c(C(=O)NC2CCCC(NC(c3ocnc3C(F)F)=O)C2)n1 70353,Cc1cc([N+](=O)[O-])nn1C(C)C(N1CC(C)NC(C)C1)=O 70354,C#CC1CC2(CC2)CN1C(=O)C(C(C)CC)N(C)C(c1oc(C)cc1C)=O 70355,c1(C(c2ccccc2Cl)C(=O)NCc2n(C(C)C)ccn2)ccc(Cl)nc1 70356,c1(C(N2C(C(=O)OC)CC(O)C2)=O)cc(C(F)F)ccc1OC 70357,c1(NC(c2noc(C3CCCN3)n2)=O)cc(C(=O)O)ccc1F 70358,C(=O)(C(O)CC(F)(F)F)NC1(CC(N2CCC(C(=O)OC)CC2)=O)CCC1 70359,N1(C(C(C)N(C(=O)CCS(N)(=O)=O)CC)=O)CCC(C)C(C)(C)C1 70360,C12(CCC1)C(=O)N2C.C1(C(=O)N(C(C)C)C2CC2)(SCCCCO)CC1 70361,C1(C(=O)NCC(CNC(c2cncnc2C)=O)OC)CCC(C)(C)O1 70362,C12CCC(CC1)CNC2=O.c1(SCc2cn(C(C)C(=O)O)nn2)ccc(F)cc1 70363,N1(N(CC#CC)C2CC2)CCC(C=O)C(O)C1.C(=O)C(CCC)N(C)C 70364,N1(C(C2(CC=C)CCN(C(c3ccsn3)=O)C2)=O)CCC12CCSCC2 70365,C(CCCCC(=O)N1CCC(F)(C(=O)NCc2ccc(C)cc2F)C1)OC 70366,C1(C(=O)NCCC2ON=C(CC)C2)CN(C(C2CCC3(CC2)CC3)=O)CC1(F)F 70367,C1(NC(c2cc(-c3ccco3)on2)=O)CCSC12CN(C(C1(O)CCSC1)=O)C2 70368,Cc1ccc(C(C)C(N2CCN(C(c3nnc(O)nc3O)=O)CC2)=O)cc1Cl 70369,CN1CC(=O)N(CC(=O)NC2CC(NC(=O)Cc3cn(C)cn3)C2)C1=O 70370,C1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)CCOCC12CCC2 70371,Cc1[nH]c(=NCC2CCN(C(C3CCc4cc(O)ccc4C3)=O)C2)ccc1C#N 70372,N1(C(c2c(C)n(C)nn2)=O)CC2CCC1C(CNC(c1c(O)cccc1Cl)=O)C2 70373,c1(N(CCOC)CCNC(C2(C3CCC3)CC2(F)F)=O)nc(C)nc2sccc12 70374,c1(C(C(=O)NCC2N(C(c3nccc(CC)c3)=O)CC2)SC)cc(Cl)cc(Cl)c1 70375,N1(C(C(=O)NCc2ccc(Nc3ncccn3)cc2)=O)CC2CCNCC12 70376,c1(C(N2CC(CCC)OC(C)C2)=O)nn(C)c(=O)c2ccccc12 70377,C(=O)(CC1=CCCCC1)N(c1nnc(N2CCC(CCO)CC2)s1)CCC 70378,Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)c3cnco3)C2)n(C2CC2)n1 70379,c12cccc(c1)C(=O)NC1CC(C)N(C1)C2=O.C1(C(=O)OCC)C(C#N)C1(C)C 70380,C(=O)(C1=CC(C)(C)C1)NCC1(CN(C)C(C2(Cl)CC2(F)F)=O)CC1 70381,c1(Cn2cc(C3C(C)CN(C(=O)C4=NOCC4)C3)nn2)cc(Cl)cc(Cl)c1Br 70382,C1(C(C)(C)C)C(=O)CC1C(=O)OCCN1CCC(CN=[N+]=[N-])C1 70383,C=Cc1cnn(C)c1C(=O)N(C)CCN(C)C(C1(O)CC1(C)C)=O 70384,c1(OC(C)C)cccc(NC(c2nnnn2CCn2cncn2)C2CC2(C)C)c1 70385,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70386,C(C1=CCSC1)(c1n(C)nnn1)N(C1CCCCC1O)CCP(C)(C)=O 70387,C1(N(C)C(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70388,C1(NC(CC2CN(C(C(CCCC)C)=O)C(C)(C)C2)=O)CCCCC12CCC2 70389,C1(CNC(c2scnc2Cl)=O)CN(C(c2cn[nH]c2)=O)C2(CCOCC2)C1 70390,N1(C(C(C)(C)OC(=O)NCC)=O)CCN(C(=O)C(C)c2cccs2)C(CCC)C1 70391,c1(C(=O)OCC(CC#C)OC)nc(C)ccc1Br 70392,c1(C(N2CCC(NC(c3c(NC)nccc3)=O)CC2C)=O)cc(C)cc2ccoc12 70393,c1(C(=O)NCCC(CNC(C2(CCC)CCC2)=O)O)cc(Cl)c2[nH]c(O)nc2c1 70394,c1(C(N(CCCNC(C2(C)C(C(=O)OC)CC2)=O)CCO)=O)cc(C)n(C(C)C)c1 70395,C1(C(N2C(CN(C)C)CCC2)=O)CCCCCN1C(c1nnc(S)n1C)=O 70396,C1C(C)(C)C(=O)N1.N1(C(C(C)NC(=O)OC)=O)CCC(NC(N)=O)CC1 70397,C(C(=O)N1CCOC(CC(N2CC(O)CC2CC)=O)C1)(C(C)C)SCC 70398,c1(CC)cccc(OCC(=O)NCCC(C)(CC)NC(C2CCC(C)O2)=O)c1 70399,c1(C(=O)OC)ccc(CN2CCC(C)CC2C(=O)OC)cc1C 70400,C(=O)(C(C(C)C)N(C)C)NCC1CCC(NC(C2(CSC)CCOC2)=O)C1 70401,c1(C(N2CCC(NC(CNC(CCC)=O)=O)C(C)C2)=O)cn2ccc(F)cc2n1 70402,C(=O)(CC(C)(C)CCC)NCC(CCCC)NC(C1(F)CCCCCC1)=O 70403,C(=O)(N=c1[nH]nc(Cl)s1)N1CCC(CN(CC)CC)C1c1ccccc1 70404,C1(C(C)NC(C2C(C=C)C2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)CC1 70405,C(CC(CC)(CC)NC(=O)C(CC(C)C)OC(=O)NC)NC(C(C)OCCCC)=O 70406,CN1CC(NC(c2cc(NC(=O)CN3CC4CCC3C4)ncc2)=O)CC12CCC2 70407,CCCCC(O)C(C)C(=O)NC(C(=O)N(C)Cc1nc(C)ns1)C1(C)CC1 70408,C#Cc1cc(C(N2CCC(F)C(NC(c3cc(Br)n(C)c3)=O)C2)=O)cc(N)c1 70409,N1(C(C(CCOC)OCCCC(C2(C)CC3CC3C2)=O)=O)CCC(F)(CN)CC1.OC 70410,c1(C(=O)OC)cccc(OC2CCCCC2)c1.c12cccc(c1)NC1CCSC21 70411,O=C(CCC[N+](=O)[O-])N1CCC2(C(=O)NCCc3cccc(F)c3)CC2C1 70412,c1(CC(C)(CO)NC(=O)C(N2CC(CCO)C3(CC3)C2)=O)ccc(C#N)cc1 70413,CC1CCC(CCC(N2CC(O)(CC(=O)NC34CC(C3)C4)C2)=O)O1 70414,N1(C(c2c(CC)con2)=O)CCCC(C)(C(=O)NC2CCCC2O)C1 70415,CCCCC(COCC)N=c1[nH]c(=NCC(N)=O)[nH]c2ccccc12 70416,c1(C(N2C(C)CC(NC(c3ccc(F)c(F)c3)=O)C2)=O)cnn2c1N(C)CC2 70417,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70418,C1(CNC(c2cnco2)=O)CC2(CCC2)CN1C(c1ncoc1C1CCC1)=O 70419,C(C1=NOC2OCCCC12)NCc1cc(C(=O)O)cc(Br)c1 70420,N1(C(CCc2ccn(C)n2)=O)CC(NC(C2(c3ccccn3)CC2)=O)CC(F)C1 70421,CC#CCCC(=O)NC1CCC(CCC(N2CCN(CCCO)CC2)=O)C1 70422,c1(N(C)C)ncc(C(C)(C)C)o1.C1(=O)C(F)(F)C(NC(N)=O)CN1 70423,C12CC(C1(C)C)C(=O)NC2.c1(C(n2cc(CN(C)C)nn2)C)ccc(Cl)cc1 70424,CCC(CC)C(F)C(=O)NCC1(NC(=O)C(OC)OC)CCCCC1 70425,C(CC1CC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)OC 70426,C=C(C)C(CC(=O)N1CCCCC1CNC(=O)CCc1nc(C)c(C)[nH]1)OCC 70427,C1(C(N2CC(CCNC(c3c(CC)con3)=O)C2)=O)CCCN(C)C1 70428,C1(CC(=O)NCC(C(C)C)(C)NC(=O)CN2CCC(=O)CC2)CCCCC1(F)F 70429,C1(C(N(CC=C)CCC)=O)C2CCC(C2)C1C.C12CCCCC1C(=O)N2 70430,c1(CC(=O)NC(CN(C)C(C2CC3OC(=O)OC3C2)=O)(C)C)nc([N+](=O)[O-])n[nH]1 70431,N1(N=S(C)(C)=O)CCCN(C(C2CC(Cl)C2)=O)CC1 70432,c1(NCCCCCCNC(C)=O)nc2c(cc1C#N)CCC(C)C2 70433,CC(C)CC(O)C(=O)NCC=C1CCN(C(C2(C3CCCCO3)CC2)=O)CC1 70434,c1(OC)ccc(NC(c2nnnn2C2CC(F)(F)C2)(C23CCCC2C3)C)c(F)c1 70435,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70436,CCC(C)C(O)C(=O)NC1(CF)CN(C(=O)Cc2conc2C)C1 70437,CN1C(=O)OCC1C(N1CC=CCC1C(=O)NCC(N1CC=CC1)=O)=O 70438,N#Cc1cnn(CCNC(C2CC3C=CC2C3)=O)c1NCc1ccnc(Cl)c1Cl 70439,Cc1cnn(C(C)C(=O)NC(c2cccnc2)C(=O)NCC2CCO2)c1 70440,N1(C(CC=C(C)C)=O)CCN(C(c2ccc(C(C)C)o2)=O)CC1c1cn[nH]c1 70441,C(CO)(CCCNC(=O)Cc1ccc(C2CC2)cc1)NC(C=CC(C)(C)SC)=O 70442,c1(N(c2nccc(C(C)C)n2)C(C2CCCNCC2)=O)ncc2ccccc2n1 70443,Cc1cc(C(N2CCC23CN(C(=O)CCC(C)(C)F)C3)=O)c(O)c(C)n1 70444,N12CCCC1C2=O.c1(C(=O)NCC)cccc(-n2ncc(C(=O)NCC)c2C)c1 70445,C(C(C(=O)N(CC1=CCSC1)C)N)SC(=O)CCCOCC 70446,c1(OC)cc(C)cnc1C(=O)NCC1C2CN(C(c3nn(C)cc3Cl)=O)CC12 70447,c1(CCC(=O)NCCC2(NC(C[SH2]C)=O)CCC2)ccc(=N)[nH]c1 70448,Cc1cc(C)n(CC(N2CCC(C)C(NC(C3CC(C)CO3)=O)C2)=O)c(=O)n1 70449,Cc1ncc(C(C)NC(C2(C)CC(NC(=O)CCCN(C)C(C)C)C2)=O)s1 70450,c1(C(=O)NCCC2CN(C(CC)=O)CC2C)cnc2n1CCCCC2 70451,CCC(C(=O)NC1CC(C)N(C(c2cc(C)n(C(F)F)n2)=O)C1)C(C)(C)CC 70452,c1(-n2ccc(C)n2)ccnc(C(=O)NCC2C=CCC2)n1 70453,c1(N2CC(C(C)C)NC(=O)C2)nc2cccc(F)c2c(=NCc2n[nH]c(=N)s2)[nH]1 70454,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)Cc2cc(C)on2)CCCO1 70455,C1(C)(C(=O)NCC(CNC(C2CCCC2(C)C)=O)OC)CCCN(C)C1 70456,N=c1[nH]c2ccc(C(N3CCCC(NC(=O)CC4CC=CCC4)C3)=O)cc2s1 70457,c1(-c2cn(C3CC(C(=O)NCC(=O)N(CCC)CCC)C3)nn2)ccc(C)cc1 70458,c1(C2(COC)CC2)ccccc1N(c1cc(CS(C)(=O)=O)on1)CC1CCCN1 70459,c1(CC(=O)N(CCNC(c2cn(C)cn2)=O)CC)cc2ccccc2c(C)c1Cl 70460,O=C(C(F)(F)CO)Cc1cn(CC(N2CC3CC3(C(F)(F)F)C2)=O)nn1 70461,CCCC(C)(C)C(=O)NC(C)C(C)NC(C1(c2ccc(OCC)cc2)CCC1)=O 70462,c1(C(=O)NC)cncc(C(=O)N(C)CCN(C(=O)CC2CCCC23CC3)C)c1.CO 70463,C(CC(=O)N1CCCC(O)C1)(C(C)CC)N(C)CCc1ccccc1 70464,C1(C(N2CCC(C(C)(C)C)C2)=O)COCCN1c1nnc(C(F)(F)F)s1 70465,C(C(=O)N(C)CC1CCSC1)(C(C)(C)C)NC(c1nc(C)c(C)s1)=O 70466,c1(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)c2c(nn1C)CCCC2 70467,c1(C(=O)NC2C3CN(C(C(C(C)(C)C)N(C)C)=O)CC32)ccc2oc(S)nc2c1 70468,c1(C(N2CCC(C)(CNC(=O)CC3CCC(=O)N3)C2)=O)cc2c(Cl)cccn2n1 70469,N1(C(C(C)OCC(C)C)=O)CC(C2CCCN(C(c3cc(C(C)C)[nH]n3)=O)C2)C1 70470,c1(C(=O)NCc2cc(C(=O)NCCC(COC)O)n(C)n2)ncc(F)cc1N 70471,CC1CC(CNC(=O)C=CC2CCCCCC2)CCN1C(c1nn(C)cc1Cl)=O 70472,c1(SCCCC)ccccc1-c1ccc(C(C)NCc2nc[nH]n2)s1 70473,CC1CN(C(C2CCN(C(=O)C3(COC)CCCO3)O2)=O)CC(C)C1O 70474,C(=O)(C#Cc1ccc(F)cc1F)N1C(C(=O)NCc2ccncc2)CCCC1 70475,Cc1ccc(CCC(=O)NC(C)(C)CNC(=O)CC2CN(C(C)=O)C2)s1 70476,C1(NCC(c2cccc(C)c2C)O)CCCCCC1(C)C 70477,C(=O)(C(O)CC(C)(C)C)NC(CNC(c1c(C)cc(OC)nc1)=O)CO 70478,c1(C(=O)NC2C(NC(CN(C(C)C)C)=O)CCC2)ncn2cc(Cl)ccc12 70479,c1(C(c2nnnn2C2CC2)NC(CC=C)C)ccc(Br)c(C(F)(F)F)c1 70480,N(C)(C(=NCC1CC2CC1C2)NCC(C)(C)C#N)C(COC)C 70481,C(CCCCCNC(c1nc(Cl)oc1C)=O)NC(CCCC)=O 70482,c1(C(N2CCN(C(C3C(=C)CC3)=O)C(C)CC2)=O)ccc2c(c1)C(C)CO2 70483,c1(C(=O)NCC(=O)OC)ccccc1CC(n1cccn1)=O.N1(C(=O)O)CCOCC1 70484,CC1SCCN(C(C2(C)CCN2C(=O)Cn2cccn2)=O)C1C 70485,N1(C(CC(=C)Br)=O)CCC2(CCN(C(c3cccc(C(C)C)n3)=O)C2)C1 70486,c1(C(N(C2CCN(C(COC(CC)C)=O)C2)CC)=O)cc(N(C)C)nc(Cl)c1 70487,n1(CC(=O)NCC(CC(F)(F)F)NC(CSCCCC)=O)cc(F)ccc1=O 70488,C1(C2CCC2)(NC(C(C2CCN(C(c3csc(F)c3)=O)C2)C)=O)CC1 70489,c1(C(=O)NCCN(CCC)C(=O)CN2CCNC(=O)C2)cnn2cccc2c1 70490,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)cccc(-n2ccnn2)c1 70491,CCCCC(C(=O)NCCOC1CCOC1)NC(=O)Cn1cc(C#N)cn1 70492,C1(C(=O)NC2(CCCNC(c3nnc(CC)s3)=O)CC2)COc2ccccc2C1 70493,C1(C#CC(=O)NCCn2cnc(C(=O)NC(C)(C)CC(C)C)c2)(CC)COC1 70494,C(=O)(C1CCOc2ccccc21)N1C2CN(C(c3nnc4ccccn34)=O)CC21 70495,C(=O)(CCC(=O)Nc1cn(-c2ccccc2)nn1)Nc1ccc(C(=O)OC)cc1 70496,C1(N(C(C(C)C)(C)C(=O)O)C(=O)CC2CSC2)CCC2CC=CCC1C2 70497,N1(C(CC=C)=O)CCC(Nc2ncc(Br)c(C)n2)C(CC)C1 70498,C1(C(CC)C)CCN(C(=O)COCCNC(C2(C)CSC2)=O)CC1 70499,N1(C(Cc2scc(C)c2)=O)CCC(C(N2C3CCC2CC3)=O)C12CC2 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70689,c1(C(=O)NC(CNC(COCCCC)=O)C(C)C)ccccc1C 70690,c1(OC(C(=O)NC2CC(NC(C(C(C)O)C)=O)CC2O)(C)C)ccc(Cl)c(F)c1 70691,Cc1ccc(OCC(C)NC(=O)NC2CCN(CCF)CC2)c(F)c1 70692,Nc1nc(Cl)ccc1C(=O)NC1CCCCN(C(=O)C(F)(F)c2cscn2)C1 70693,CCCC(CC)CC(=O)NCC1(C(C)(C)O)CN(C(c2cc(=O)cc[nH]2)=O)C1 70694,c12ccnc(c1)C(=O)N2C.c1(CNCc2cnc(Br)s2)ccccc1C(F)(F)F 70695,c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)C)ccnc(F)c1N 70696,Cc1csc(C(N2CCC2(C)CC(=O)N(C)CCO)=O)c1C 70697,C1(CNC(=O)CCC2(SC)CN(C(C3(C#N)CC=CC3)=O)C2)CCCCC1O 70698,c1(-c2c(C(n3cc(-c4ccc(=O)n(C)c4)nn3)C)c[nH]n2)c(Cl)cc(Cl)cc1Cl 70699,c1(CC)ccc(C(=O)NC(CN(C)C)C(N2CCC(C)(CCO)C2)=O)cn1 70700,C(=O)(C1COc2ccccc21)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 70701,n1(CC(=O)NCC2(F)CN(C(C(C)C(F)F)=O)C2)cnc2ccccc12 70702,C(=O)(CC1=CCCCC1)N1C(C(=O)Nc2cncc(OC)c2)CSCC1 70703,C(C(=O)NCCCN(C)C)N(CCC)C(C1CC1F)=O 70704,CCC(C)CC(C(=O)NCc1noc(C)n1)NC(=O)CSC1(C2CCC2)CC1 70705,c1(C(C(=O)NC2CC2)N(C)CCN(C)Cc2cccc(Cl)c2)ccc(OC)cn1 70706,N1(C(C(C)O)=O)CC2(CCOCC2)CC1CNC(=O)COCCN(C)C 70707,CCCCCCN(CC(=O)NCC(C)(CC)NC(c1coc(C(F)(F)F)c1)=O)C 70708,c1(C(=O)NC2C(C(N)=O)CCC2)ccc(Cl)nc1NCc1ccnc(O)c1 70709,O(C1CCCc2nc(C)ncc21)C(c1n(CCC)ccc1)=O 70710,C(=O)(C(O)C(F)(F)F)NCC(C)(C)OCCNC(C1CCCOCC1)=O 70711,c1(NC(CNC(CN(CCOCCOC)C)=O)=O)cccc(F)c1C 70712,CC1CCc2[nH]c(C(=O)N(C3CCCC3)CCCNC(=O)CC(C)(C)O)cc2C1 70713,N1(CC(N2CC(O)(CN(CCCCCC)C)C2)=O)CCCSCC1 70714,C1(C)(CNC(c2c(OC)nsc2)=O)CCN(C(=O)C(n2ccc(C)n2)C)C1 70715,C1(C#N)(C(=O)NC(C(=O)NC2CN(CC)C2)C2CCC2)CC2CC2C1 70716,n12c3c(cc(cc3)c1=O)CC2.N1(C(C(NOC)=O)=O)CCC(C)(N(CC)CC)C1 70717,c1(CC(C(=O)NCCC2CC2)N(CC(CC)(C)C)C)ccc(C)nc1Cl 70718,N1(C(C2(C)CN(C(c3cc4n(n3)CCO4)=O)C2)=O)CC2NC(=O)OC2C1 70719,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 70720,c1(C(=O)NC2CC(NC(=O)CC(F)(F)C(F)(F)F)C2)cc(Cl)cc2ccncc12 70721,c1(C(N(C)CCOCCNC(=O)CC2C=CS(=O)(=O)C2)=O)ccc2cncn2c1 70722,C1(NC(C(C=CC)O)=O)CCN(C(c2nccnc2C)=O)C12CC2 70723,c1(C(N2CCCC(C)(C(=O)OCC)C2)=O)cc(Br)c(C)cc1O 70724,C(C(C)(C)CC(=O)N1CC(CC(=O)NC(c2[nH]c(C)nc2C)C)C2(CC2)C1)OC 70725,c1(C(C(=O)NC2C(NC(c3cc(C)n(C4CC4)n3)=O)C2)(F)F)c(F)cccc1F 70726,N1(C(C2CC(C#N)(OC)C2)=O)CCOCCC1C(=O)NC1(CF)CC1 70727,S(=O)(=O)(c1ccc(NCC=CBr)c(F)c1)NCC1OCC(C)C1 70728,C(=O)(C#CC1CCCOC1)NC1CCCCN(C(CC(C)O)=O)C1 70729,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 70730,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 70731,C1(CCC(=O)NCC(C)OCOC)CN(C(C2(C)CC2)=O)CCO1 70732,C12(C(=O)NCC3C(NC(C4(C(C)C)CCCO4)=O)C3)CCC(CO)(CC1)CC2 70733,CC(C)(C)C(C(=O)N1CC(C#N)(CCF)C1)NC(c1cnsn1)=O 70734,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 70735,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 70736,CC(CCCNC(c1cccnn1)=O)NC(=O)CC1CC(C)(C)C1 70737,N1(C(CC(=C)C)=O)CCC2(CCCC2NC(=O)CCn2c(C)c(C)sc2=O)CC1 70738,C(=O)(CC(O)CC1CCCC1)NC(CNC(C(C)(C)NC(=O)OC(C)(C)C)=O)C 70739,N1(CCC)CCC(C(=O)N(CC(C)O)CCNC(=O)CCC2CCC2)CC1 70740,N1(C(C2C(CNC(C(C)NC(N)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 70741,c1(NC(=O)CC2COCCN2C(C2CCCO2)=O)ccc2ncccc2c1 70742,N1(C(Cc2n(C)ccn2)=O)CCCCN(C(c2cccc(NCC#N)c2)=O)C1 70743,N1(CC(=O)N(CC(O)C(C)(C)C)C)CCCC2(CCNC2=O)C1 70744,Cc1nnc2n1CCC(C(=O)NCC1CCN1C(=O)C=C1CCCCCC1(F)F)C2 70745,c1(N(CC(C)NC(C2CCS2(=O)=O)=O)C)ncc(O)cn1 70746,C1(OCCNC(=O)Cc2cncs2)CCN(C(C2COCOC2)=O)C1 70747,N1(C(C(CO)NC(C(C)C)=O)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 70748,C(=O)(C(C)Cc1cnc[nH]1)N(CCNC(=O)COC)CC 70749,C12(C(OC(F)F)=O)CCC(n3cc(-c4cncs4)nn3)C1C2.CC 70750,C(=O)(C(O)C(F)(F)F)N1CCC(N(C(C(CCO)N(C)C)=O)C(=O)C2CC2)CC1 70751,CCCCC(CNC(C1CN(C(=O)CN2CCCNC2=O)CC1OC)=O)CC 70752,N1(C(c2ccccc2)COC)CCC2(CCN(C(C3CCN(C)CC3)=O)C2)C1 70753,CCCC(CCC)CC(=O)NCC1CN(C(=O)COc2ccsc2)CC12CCC2 70754,c1(C(N(C2CCN(C(=O)CC(O)CC3CC3)C2)CC#C)=O)cccc(F)c1C 70755,CN1N=C(C(=O)NCC2COC(C)(C)CN2C(=O)C=C2CCC2)CCC1=O 70756,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 70757,C1(C(=O)NCC(C)NC(c2c(OC)cnc(Cl)c2)=O)CCOCC12CCC2 70758,c1(CNC(C(=O)NCc2c(Cl)ccc(C)c2)=O)cc2cccnn2n1 70759,N1(C(C2CC(SC)C2)=O)CC2OCCN(C(=O)CCC(=O)N(C)C)C2C1 70760,C1(C(N2CC(C#N)C(NC(c3csc(Br)n3)=O)C2)=O)CCc2ccccc2C1 70761,C1(O)(CCNC(c2cc(CC)nn2C)=O)CCN(C(C2(Br)CC2(C)C)=O)CC1 70762,c1(C(N2C3C(NC(C4CS(=O)(=O)C4)=O)CC(CC3)C2)=O)cccc2c1CCCC2 70763,C(=O)(C(C)(C)CCCNC(C1(C#N)CC1C)=O)N1CC(CCC#C)C1 70764,CC1CCCN(C(=O)C(=O)NC2CC(F)(CNC(C3CC(C(F)F)C3)=O)C2)C1 70765,CCC(C)(C(=O)N1CCC(OCCNC(c2cncc(C)n2)=O)CC1)C(N)=O 70766,Cc1cc(C(N2CCCC2CNC2CCC2NS(C)(=O)=O)=O)ncc1Cl 70767,c1(COCC(N2C(C(=O)NC3CC(Cl)=NO3)CCC2)=O)cc(Cl)cc(Cl)c1 70768,c1(C(N2CC(N3CCN(C(CC)=O)CC3)C2)=O)nccn2c(C)nnc12 70769,CCC(O)C(F)(F)C(=O)NCc1ncoc1CCCCNC(=O)CC1CC12CC2 70770,c1(OCC)ccc(C(=O)NCCCCNC(C2SCC=C2C)=O)cn1 70771,Cn1c(C(=O)Nc2cccc3c2ccn3C)cc2cc(Cl)ccc12 70772,N(C1CCCc2c[nH]nc21)C(C(CN(C)C)NC(c1ccc(CC)[nH]1)=O)=O 70773,Cc1ccc(Br)c(NC(=O)C2CC2)c1.C1C(=O)N1 70774,N1(C(c2ccc(Cl)cc2I)=O)CCN(Cc2cc(C3CC3)ccc2F)CC12CC2 70775,c1(C(=O)NCC2C(NC(COCCCOC)=O)C2)ccnc2c(Br)cccc12 70776,c1(NC(C2C(NCc3n(C)ncc3)C2)=O)cc(C(F)(F)F)ccc1C(F)(F)F 70777,c1(C(=O)NCC2OCCN(c3cc(OC)ncn3)C2)cc(O)nc(O)c1 70778,C1(COC(CNC(CCCc2[nH]c(=N)sc2)=O)=O)CCCC12NC(=O)NC2=O 70779,C(C)(C)(C(C)CC(=O)N1CCN2CCC1CC2)NC(CCSCCC)=O 70780,C=CCC(C(=O)N1CCCC1CSC1CCCC1)NC(=O)CC=CCC 70781,N1(Cc2cncc(C)c2)CCC(O)CC1C(=O)Nc1cccnc1CO 70782,C1(CC#C)(C(=O)NC(CC)CN(C)C(c2cnn(C(C)C)c2F)=O)CC=CCC1 70783,c1(C(=O)NCC2CN(C(c3c(C)nsc3C)=O)C2)cccn2ccnc12 70784,N1(C(c2c(C)nsc2)=O)CCC2CN(C(=O)C(O)CC3CCCCC3)CC12 70785,C1(NC(C2CCN(C(C)=O)C2)=O)CN(C(=O)COc2cccnc2)CC1C(F)F 70786,Cc1cc(C(N2CCSCC2C(=O)N=c2cc[nH][nH]2)=O)ccc1F 70787,c1(C(N2CCC(C)C(NC(c3nsnc3O)=O)C2)=O)ccc(C#N)c(Cl)c1 70788,C1(C2CCN(C(C3CC3F)=O)CC2)(NC(c2cnc(CC(C)C)[nH]2)=O)CC1 70789,N1(C(C=CC(C)C)=O)CC(O)(C(C)NC(=O)CNC(C2CCC2)=O)C1 70790,CCCCCC(CC)C(=O)N1CC(C)CC1C(=O)NOC1CCC1 70791,c1(C(N2CCC(OC(C(C)NC(CC)(C)C)=O)C2)=O)c[nH]c(C(=O)OC)c1C 70792,C(=O)(C1CSc2ccccc21)NC(CC)CN(C(=O)C(CCC)OC)C 70793,C1(C(N(CC(C)N(C(CN2CC(C)C2)=O)C)C)=O)CC(c2ccccn2)=NO1 70794,C#CC1(C(=O)NC2CC(C)(C)OC2=O)CCN(C(C2CCC(F)CC2)=O)C1 70795,N1(C(CC(C)N(C)C(c2csc(Cl)n2)=O)=O)CCC2(CCOCC2)C1 70796,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CC2)=O)o1 70797,C1(NC(CCc2n(C)ccn2)=O)CC12CCN(C(=O)CC1CC(F)(F)C1)C2 70798,c1(C(=O)NCCCC2OCCN(C(Cc3ccn(C)n3)=O)C2)cc(Cl)cc(Cl)n1 70799,N1(C(COC2CC(NC(c3cnn(COC)c3C)=O)C2)=O)CC(C)C(C)C1C 70800,c1(-c2c(C)nn(C)c2)cnc2[nH]cc(C(=O)NC(C3CCCOC3)C3CC3)c2c1 70801,CCC(C)C(O)C(=O)N1CCCC1C(C)NC(=O)C=CC=Cc1ccccc1 70802,C1(CCCNC(c2n(C)cnc2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)CC1 70803,Cc1ccc(C(=O)NCC2C3CN(C(=O)Cc4c(C)cnn4C)CC23)c(O)n1 70804,C12(C(N(C3CN(C(C4(O)CCC4)=O)CC34CC4)C)=O)CCC(C)(CC1)CO2 70805,c1(C(N2CC(CNC(CC3C(OC)CC3)=O)(OC)C2)=O)cnc2[nH]cc(C)c2c1 70806,C1(CNC(c2c(C)cc(C(F)(F)F)s2)=O)CCS(=O)(=O)C1(C)C 70807,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCO3)oc2cc1C 70808,C(=O)(C#CC1CCCCO1)O.CC1(C)CC(c2ccccc2F)N(C)C1 70809,c1(CCNC(N(CC=C)C2CC2)=O)ccc2c(C)[nH]nc2c1 70810,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 70811,C(c1ccncc1)=CC(=O)NC(C(=O)NC1C(CCOC)C1)C 70812,N1(CCNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2(C(F)F)CC2)CC1 70813,c1(CC)nc(C)ncc1C(=O)NCCN(C(c1ccc(C(C)CC)cc1)=O)CC 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70849,C(=O)(C(F)(F)c1cncs1)NCCN(C(=O)CSc1cnnn1C)CCOC 70850,C(CCN(C)C(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O 70851,c1(C(=O)NCCN2CCC(NC(C(CC)C)=O)CC2)ccc(Cl)c(Cl)c1F 70852,CN=C(NCCCCc1ccccc1)N1CCC(SC)CC1.N1CCCC1 70853,C1(NC(c2ccc(C3CCCC3)cc2)=O)CCCC(Nc2ncc(F)cn2)C1 70854,Cc1cc(C)c2nc(N3CCCC3CNC(c3cc(CO)nc(Cl)c3)=O)sc2c1 70855,Cn1c(C(F)(F)F)cnc1C(=O)OCC1CC2(C1)CC2F 70856,c1(-c2cn(C(C)C)nn2)ccc(C(=O)NCC23CC(C(=O)OCC)(C2)C3)c(N)c1 70857,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 70858,N#CCCC(=O)N1CCC(C(N2Cc3ccccc3C2)=O)O1 70859,N1(C(c2sc(C)c(O)n2)=O)CCCC2CN(C(=O)C3=CCC(C)(C)CC3)CC12 70860,C(=O)(CS(=O)CCC(F)(F)F)NCC1(O)CCN(C(C2(C)CCN(C)C2)=O)C1 70861,C#CCC(C)(C(=O)NCC(O)CCC=CC)NC(=O)C1=CC(C)(C)C1 70862,C1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CC2)CN(C)CCN1C 70863,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 70864,c1(CNC(=O)NC(C)C(=O)NC2CCCC2n2cccc2)ccc(Cl)c(Cl)c1 70865,N1(C(c2c(F)cccc2F)C(=O)NCC)CCNC(=O)CC1C 70866,c1(C(N2CC(C(C)NC(C(C)NC(=O)NC)=O)C2)=O)n[nH]c2c1CCCCC2 70867,c1(CC)nc(C)c(C(N2CC(CC(C)NC(C34COCC3C4)=O)C2)=O)s1 70868,N1(C(C(C2CC2)NC(c2c(C)cccc2)=O)=O)CCCN(C)C(=O)C1 70869,CC1CCSCCN1C(=O)C(N)Cc1cccc(-c2ccc(F)cc2)c1 70870,CC(CCC(C)(C)C)C(=O)N1CC(C)(CCC(N2CCN(CC(F)F)CC2)=O)C1 70871,C1(CC(=O)OCC)(NCc2sc3nccn3c2C)CCCS(=O)(=O)C1 70872,C1(CNC(c2ccn3c2CCC3)=O)CN(C(=O)COc2ccon2)CC12CCC2 70873,CC(C)CC(C(=O)N1CCOC(CCF)C1)NC(C1CC(C)OC1C)=O 70874,C(=O)(C1=CCOC1)N1CCCC(CCNC(C2CCSC2)=O)C1 70875,C1(NC(CCC(CC)NC(c2ncnc(C)c2C)=O)=O)C2CCC(C2)C1(C)C 70876,CC(CNC(=O)C(C1CCCCC1)O)(CO)NC(=O)CCC1CCC1 70877,CC(C)(C)CCCC(=O)NC1CCC(CNC(=O)COCc2cccc(Cl)c2)C1 70878,CCCC(F)C(=O)N1CCC(CC(=O)NC2CC2C(N)=O)CC1 70879,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cnc[nH]3)C1C2 70880,N1(C(c2c(CN(C)C)ccs2)=O)CCC(F)C(NC(c2c[nH]nc2F)=O)C1 70881,N1(C(=O)CCCc2cccs2)CCN(C(=O)CCc2ccncc2)C(C(F)F)C1 70882,c1(C(=O)NCC2C(C)CCN2C(c2cnco2)=O)cc(S(N)(=O)=O)ccn1 70883,C1(CC=C)(CNC(=O)C(C)OCCN(C)C)CN(C(=O)Cc2csnc2C)C1 70884,C1(CNC(C)=O)CC2(CCN(C(=O)CCc3c[nH]c4ccccc34)CC2)CO1 70885,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CN(C(C2CNC(=O)C2)=O)CC1F 70886,Cc1c(C(=O)NCC2CC(C)N(C(=O)Cc3cc[nH]n3)C2)cccc1C#N 70887,C1(NC(=O)COCCOCCO)CCCC(CNC(=O)CC2CCSCC2)C1 70888,c1(C(N2CCC(CN(CC(=O)NCCOC)C)C2)=O)ccc([N+](=O)[O-])o1 70889,c1(NC(C(CCOCC)NC(c2n(CC#C)ccc2)=O)=O)ccc(CO)cc1O 70890,c1(C(N2CCC2C(N2CCOCC2c2ccccc2)=O)=O)c(O)cccc1[N+](=O)[O-] 70891,c1(C(=O)NC(CC)CNC(c2cncc(O)c2)=O)ccc(Cl)c(O)c1 70892,c1(OC)nccc(C(=O)NC2CCC(NC(c3ccc(N)c(F)c3)=O)CC2)c1F 70893,C1(NC(C=CCC)=O)CC(C)CN(c2nccc(Oc3ccccc3)n2)C1 70894,O=C1CCCCCN1C(c1cn(CC2CCC2)nn1)C1CC1.C1CCOC1 70895,N1(C(c2c(CC)csc2)=O)CCCCC1CN(C(=O)CCCCOC)CC 70896,c1(CC)[nH]nc(C(=O)NC2C=CC(CNC(=O)CC(C)CC)C2)c1Br 70897,c1(OCC)cccc(OCC(C)NCCCC2CCS(=O)(=O)C2)c1 70898,CCCCCC(CC)C(=O)N1CC(F)(F)CC1(C)CNC(c1ccc(CC)s1)=O 70899,N1(Cc2cnc(OCC)nc2)C2CCC1CC(NC(=O)Cc1cccc(Cl)c1)C2 70900,Cc1ccc(O)c(CNC(=O)CCN(C(C2CC3CC3C2)=O)C2CC2)c1 70901,N1(C(COCC#C)=O)CCN(C(C2CCC(N(C)C)C2)=O)C(CO)C1 70902,N1(C(C(CCOC)C)=O)CCCCCC(NC(c2ccnn2C)=O)C1 70903,C1(O)(C(N2CC(N(C(=O)CC3CC(F)C3)C)C(O)C2)=O)CN2CCC1CC2 70904,N1(CCC)C2CCC1CC(N(C(CC)C(=O)OCC)C(=O)OC)C2 70905,c1(CC)cc(Br)ccc1NC(C1CC2CC2N1Cc1ncn(CC)n1)=O 70906,C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2coc(Br)n2)=O)CC1C 70907,N(C(=NCCCC1CCCCC1)NCC1CCOC1)CC1C(=O)NCCC1 70908,C#Cc1cn(C)nc1C(=O)NCC(CC)NC(c1ccc(N)cc1Cl)=O 70909,C1(CC)CCC(CC(N2CCC(N(C(=O)CCn3ccnc3C)CC)C2)=O)CC1 70910,C1(CNC(c2csnn2)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 70911,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 70912,c1(NC(C2N(C(C(C)N(CC)CC)=O)C(C3CC3)CC2)=O)ccc2nncn2c1 70913,c1(NC(C2COCC2(O)C(F)(F)F)=O)cncc(-c2nn[nH]n2)c1 70914,c1(C(N(C2CC(NC(=O)CP(C)(C)=O)C2)C)=O)ccc(-c2ncc[nH]2)cc1 70915,c1(C(=O)NC(CC)CN(C(=O)CC2CC2(C)C)C)cnc(-c2ccncc2)s1 70916,c1(C(N(C2CCCN(C(C3CC3c3ccccc3)=O)C2)CC)=O)ccc([N+](=O)[O-])[nH]1 70917,C(C1CCN(C(=O)C2=CCCCO2)CC1)=CC(N1C(COC)C=CC1)=O 70918,CCC(O)CC(=O)NCC=CC(N1CCOC(CC)C1)=O 70919,c1(CC)ccc(C(=O)OC)cc1C.C12(N)CC(C1)C(=O)O2 70920,c1(SNC(=O)NC(c2cc(Sc3ncccn3)on2)CC)cccc(C(C)=O)c1 70921,N1(C(CCOCCC)=O)CCN(C(=O)CCOc2ccc(SC)cc2)C(C)C1C 70922,N1(C(C(C)n2ccnc2)=O)CC2CCN(C(C34CCC(CO)(CC3)C4)=O)CC2C1 70923,c1(C(=O)NC(C2(O)CN(C(C(CC#C)C)=O)C2)C)ncnc2c1ccn2C1CC1 70924,c1(NCc2ccc(C(=O)NCC3CC(CF)C3)cn2)nc(Cl)ncc1Cl 70925,C(c1ncco1)=CC(=O)N(C1CN(C(=O)NC2CC2c2ccccc2)C1)C 70926,C1(COC)(CNC(C2CCCC(=O)N2)=O)CCN(C(=O)C#CC(C)C)C1 70927,C1(C(=O)NC)C2CS(=O)(=O)CC12.c1(NCC23CN(C2)C3=O)cncc(C2CC2)c1 70928,C12(C(=O)NC3CC(CNC(CNC(=O)NC)=O)C3)CCCN1CC(O)C2 70929,CS(=O)CC(=O)N(CCCN(C1CCCCC1)C(=O)Cc1cnccn1)C1CC1 70930,C1(C(=O)NCC2(C)CCN(C(CSCC)=O)C2)CCc2nc(C)nn2C1 70931,C(=O)(CC(CC)C(F)F)NC1C(CC)CN(C(=O)Cc2ccc(OCC)cc2)C1 70932,C1(C(C(=O)NCC(C(C)C)NC(C2(CO)COC2)=O)C)CCCC(F)(F)C1 70933,C1(CNC(=O)Nc2cccc(CN3CC(=O)NCC3)c2)CCN2CCCC2C1 70934,C12(CNC(N(C)Cc3cnn(C)c3)=O)CCCC1OCC2 70935,c1(C(=O)NC(C)CCNC(C2COCCO2)=O)ccc(Br)cc1[N+](=O)[O-] 70936,n1(CC)nc(C(=O)NC2CCCN(C(C3(CCOCCO)CCC3)=O)C2)cc1C 70937,c1(OCCC(=O)NCCN(C(C2C(C)(C(=O)OCC)C2)=O)C)ccc(F)c(F)c1 70938,C(=O)(CCP(C)(C)=O)NC(C(C)C)C(=O)NCCC1(C)CCCO1 70939,N1(C(C2C(C)CCCC2)=O)CCC(O)CC1C(=O)Nc1cc(F)ccn1 70940,CC1CCCN2C1CC2=O.C1(C)(C(=O)N(C)C)CN(C(=O)C(C2CCCCC2)F)C1 70941,C1(CNC(CC(C)NC(N)=O)=O)CCC2(CO1)CC(NC(c1cnc(O)o1)=O)C2 70942,C1(NC(C=NOC)=O)CN(C(=O)CC2(C3CC3)CC2)CCC1CO 70943,C1(C(N(C)Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)cc2)=O)CC1O 70944,c1(CCN)ccc(-n2cc(C3(C(=O)NC=O)CCOCC3)nn2)cc1 70945,c1(C(=O)OCCc2ccc(C#N)cc2)ccc(S(=O)(=O)CCS(C)(=O)=O)cc1 70946,c1(OCC)cc(C(=O)NCC(c2cccc(Cl)c2)NC(=O)C2=CCSC2)ccn1 70947,Cc1cc(C(N2CCCC2(C)CNC(=O)CC2CNC(=O)C2)=O)c2[nH]cnc2c1 70948,c1(CN2CCC(CC(=O)Nc3c(C)sc(C)c3C#N)C2)c(C)nn2ccccc12 70949,CC(C)(CS(C)(=O)=O)C(=O)NCC1(F)CC(CNC(=O)CN2CC=CC2)C1 70950,C=CC1CCCCN1C(C1(C)CCN(C(c2ccccc2C)=O)CC1)=O 70951,Cc1noc2ncc(C(=O)NC3CC(CNC(c4cccc[n+]4[O-])=O)C3)cc12 70952,C(=O)(C(C)(C)C(O)C(C)C)N(CC(=O)NC(C)CS(C)(=O)=O)CC 70953,c1(NC(c2nnnn2CC(F)F)(COC(C)=O)C)cc(C(C)(C)C)nn1C 70954,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 70955,Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CC(C)C2CCCC2)c(O)nn1 70956,CC1(C)CN(C(=O)CCCS(N)(=O)=O)CC(CNC(C2CC3(CSC3)C2)=O)O1 70957,CC1CCN(C(=O)CCc2cccnc2)CCN1C(=O)CC1(C#N)CC1 70958,N1(C(c2nc[nH]n2)C)CCc2cc(F)c(F)cc2C1 70959,c1(CNC(C2(NC(c3cn(CCC)nc3)=O)CC(C)C2)=O)c[nH]ccc1=O 70960,C=C1CCN(C(=O)CCCCOC)C(C(=O)N(C(CC)CO)C2CC2)C1 70961,C1(NC(=O)CC2CCCCC2)CN(C(=O)C(F)n2cccn2)C2CCCCC12 70962,C1(C(=O)NCCC2(CNC(c3c(C)scc3)=O)CC2)CCc2nncn2CC1 70963,c1(C(N2C(C(N3CCN(S(C)(=O)=O)CC3)=O)CC3CC32)=O)ccc(F)c(F)c1Cl 70964,N1(C(C)C)CCCC1CC(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 70965,N1(C(C(F)=C(C)C)=O)CCCOC(CNC(=O)CN2C(=O)CN(C)C2=O)C1 70966,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(Cl)(Cl)C2)=O)C1)=O 70967,N1(C(C(c2ccccn2)C)=O)CC2CCC1CN2C(=O)CSc1cccc(Cl)c1 70968,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cn(C)nn1 70969,C1(CCC(=O)Nc2cc(N)n(C)n2)CCCCN1CC1N(CCC)CCC1 70970,C(=O)(CC(C(F)(F)F)NC(C1CC2CC12)=O)NCCCCN(C)C 70971,N1(C(CC2ON=C(C)C2)=O)CCC(C(=O)NCCn2nnc(C3CC3)n2)C(C)(C)C1 70972,CC1CC(N(C(=O)CC2(N(C(=O)COCCCN=[N+]=[N-])C)CC2)C)CCO1 70973,N1(C(c2cc(Cl)cnc2O)=O)CC2(CCCN2C(c2cccc(Cl)c2Cl)=O)C1 70974,c1(CC(=O)N(C2CCC(CNC(=O)CN=S(C)(C)=O)C2)C)ccc2c(c1)CCC2 70975,C1(C(=O)NC(c2cc(F)cc(F)c2)CCOC)CCC(O)C(O)CC1 70976,N1(C(C(C)(C)C#N)=O)CCC2(CCC2NC(=O)Cn2cnnc2O)CC1 70977,C(=O)(C1CCCc2nncn21)NCC1CCCCN(C(CSCCC#N)=O)CC1 70978,C1(C(=O)NC2(CC)CCC2)COCCN(C(=O)CCc2nc[nH]n2)C1 70979,n1(CC)cnc2nc(N3CCC(C)(CO)C3)nc(N(CCS(C)(=O)=O)C)c12 70980,N1(C(C2CC(=C)C2)=O)CCC(C)C(NC(C23CC(CF)(CO2)C3)=O)C1 70981,Cc1cc(=NC2CCCc3ccc(C)cc32)[nH]c(=NCc2nncn2C2CC2)[nH]1 70982,N1(C(c2cn(CCC)nc2)=O)CC(NC(C2C3CCCC23)=O)C(n2cccn2)C1 70983,C1(NC(C2CC(=O)OC2)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 70984,N1(C(C2CC(SC)C2)=O)CCC(N(C(=O)C=CC(C)C)CCC)C1.C1(C)CC1 70985,c1(C(N2C(CN(C)C(C3CCCC3C3CC3)=O)CCC2)=O)cc(F)ccc1O 70986,CCN=C(NCc1cc(C2CC2)no1)NC1CC(O)C1c1ccc(Cl)cc1 70987,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(c1cncc(O)c1)=O)CC2 70988,C1(NC(CC2(CC=C)CCCC2)=O)CCC(C(=O)Nc2ncccn2)CC1 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71077,Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CCC1COC(C)(C)O1 71078,C12CCCC(CC1)NC2c1ccccc1.c1(O)ccnc(-c2ccccn2)c1.OC 71079,N1(CC)CC(NC(=O)CN2C(=O)CC(C)(C)C2=O)Nc2ccccc21 71080,C(=O)(N1CC(O)CCO1)c1cc(CNC(C(C(COC)C)C)=O)no1 71081,C1(C(N2C(C3CCN(C(c4c(C)con4)=O)CC3)C(C)(C)C2)=O)Cc2nccn2C1 71082,N1(C(C(C)OCCOC)=O)CCCC2(CC=CCC2)C1 71083,N1(C(=O)C=C(Br)Br)C2CCC1C(NC(C1(O)COC1)=O)C2 71084,C1(C)(NC(C(C)N(C(=O)CC2CCOC2)C2CC2)=O)CN2CCC1CC2 71085,c1(OCC(=O)N(C2CCCN(C(=O)C(C)OC)C2)CC)ccc(C(F)(F)F)cc1 71086,C(=O)(C1(C)OCCc2ccccc21)N(CCCNC(COCC(=O)OC)=O)C1CC1 71087,c1(C(=O)NCC(C)(O)CNC(=O)CCOC2CC2)cc2cc[nH]c(=O)c2o1 71088,N1(C(c2cc(CC)ncc2)=O)CC(C(N2CCCCC2CCO)=O)CC(C)C1 71089,Cc1cn(C)nc1C(=O)NCc1nc(C(=O)Nc2cncc(F)c2)c(C)o1 71090,N1(C(C(C)Cc2cnco2)=O)CCN(C(=O)CCc2nncs2)CC(O)C1 71091,C(=O)(C(C(CC)CC)OC(C)=O)NC(CC=C)C(=O)N1CC(CO)CC1CO 71092,C1(C)(CCCC(=O)NCC2(C)CC2)NC(=O)NC1=O.N1(C(C2CCC(C)O2)=O)CCCCC1 71093,N1(C(CC(CCSC)O)=O)CC2(C1)CN(C(c1nocc1C1CC1)=O)CC2CO 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71286,Cn1c(CC(N2CC(C)(NC(=O)C(C)(C)CF)C2)=O)cc2ccccc12 71287,N1(C(c2cc(C(C)C)ncc2)=O)CC2CN(S(=O)(=O)Cc3cccc(Cl)c3)CC12 71288,N1(C(C(CC=CCC)C)=O)CCC2CCCC12C(=O)NC(c1nc[nH]n1)C 71289,CCC(C)C(C(=O)NC1CCC(NC(c2ccccc2NCCO)=O)CC1)OC 71290,C=CCCCCCCCCC(=O)NCCC(=O)C(CCC)=CCC.C1CN(C)N1 71291,CC1CC(NC(C2CCCCN2S(C)(=O)=O)=O)CN(C(=O)CC2CCC2)C1 71292,C(C1CCOc2ccccc21)NC(NCC(O)C1CC1)=NCC1CCCCO1 71293,CC1CCCN(C(=O)C(CNC(c2cncn(C)c2=O)=O)N(C)C)CC1 71294,C=CCC(C)(C)CC(=O)N(CC(=O)NCCOC)C(C1(C)CC1)C 71295,c1(N2CCC(C)C(NC(C3CC4(CCCO4)C3)=O)C2)nc(Cl)nc2[nH]ccc12 71296,CCCCC(CC)C(=O)NCCN(C(c1nc(Cl)sc1C)=O)CC 71297,C1(CNC(C(CCC=C)(F)F)=O)CCC2(CCN(C(=O)C(F)C(C)(C)O)CC2)CO1 71298,N1(C(C2C(C)C2)=O)CCC(C(C)NC(C23CCN(CC2)C3)=O)CC1 71299,C1(CNC(c2c(C(=O)OC)csc2)=O)CN(C(=O)C(=O)NC2CC2)CCC1C 71300,N1(C(C2C(C=C)CC2)=O)CC(NC(c2cc(OC)ccn2)=O)CC12CCCCC2 71301,c1(C(N2CCC(NCC3(C4CC4)CC3)C2)=O)cccnc1F 71302,C1(CNC(COCCC)=O)CCCN(C(=O)CC2CCCS(=O)(=O)C2)CC1 71303,C(=O)(NOC1CSC1)C1(NC(=O)NCCC2CC=CC2)CC1 71304,CCCCCCCN(C(=O)C(CC1CCCCC1)NCc1ccccc1)C 71305,C1(C(N)=O)CN(C(C2C3CCCC23)=O)CCC1NC(c1conc1C(F)(F)F)=O 71306,CC(C)CN=C(NCC1CCCN1c1nc(Cl)cs1)NCC1CCOCC1(C)C 71307,C1(C(N2C(n3cc(-c4cncc(C)c4)nn3)CC2)=O)CCC(O)CN1C 71308,C(=O)(C1=CC2C=CC1C2)N1C(NCc2snc(CC)n2)CC1C.n12cc-1nn2 71309,N1(C(CN2CC(C)(C)C2)=O)CC2CC(C(N3CC4CC3CS4=O)=O)(C2)C1 71310,c1(C(N2CCC(CC=C)(NC(C3C=CCC3)=O)C2)=O)c(F)cc(F)c(N)c1F 71311,CC1CCC(CNC(=O)Cc2cc(C(F)(F)F)n[nH]2)N(C(c2ccc(Cl)cn2)=O)C1 71312,C(=O)(CC1OCCc2sccc21)N1CCCCC(NC(C2(C)CCCOC2)=O)C1 71313,c1(NC(CCC=CCC)(C)c2nnnn2C2COC2)cc(F)c(F)cc1OC 71314,c1(CC)cnc(C(=O)NCCN(C(=O)Cc2ccc(O)cc2)CC(C)O)cn1 71315,c1(C(N2CCCC(CC)(CO)C2)C(=O)NC2(C)CC2)cc(S(C)(=O)=O)c(C)o1 71316,C1(NC(c2ncc(OC)nc2)=O)CCCC2CN(c3nc4cccnc4s3)CC12 71317,C1(CNC(CC)=O)CCC(NC(c2ccc(-c3cnc[nH]3)cc2)=O)CC1 71318,O(C1CCc2c(Cl)ccnc21)C(=O)NCc1ccc(C#C)c(F)c1F 71319,C=CCCC(F)(F)C(=O)NC1CC(CCNC(C2(C)C=CCCC2)=O)C1 71320,CC(C)C(CCN(C)C(C1CC(C)OC1=O)=O)NC(=O)CCN1CCOCC1 71321,C=CCC(C)(C)CC(=O)NCCN(C)C.C12(C)CCN(C(=NCCCOCC)NC1)C2 71322,CC(CCC(C)(C)C)C(=O)NCC1=CCCN(C(c2ccc(Cl)cn2)=O)C1 71323,CCC(C)C(C(=O)N1CC(C2COCC2F)C1)c1ccccc1 71324,Cc1cc(=NCC2CCOC2)[nH]c(=NCc2cccc([N+](=O)[O-])c2C)[nH]1 71325,N1(C(Cc2ccnc(C)n2)=O)CC(C)(C)C(NC(=O)C(O)CC2CC2)C(C)(C)C1 71326,CC(C)C(C)COCCC(=O)NCCC1CN(C(=O)CC(C)F)C1 71327,Cc1nn(C(C)C)c(NCC(C)CNC(=O)C(C)(C)n2cncn2)c1[N+](=O)[O-] 71328,c1(C(N(C(CNC(c2c(C)cc(CC)o2)=O)C2CC2)C)=O)c(C)ccc(F)c1N 71329,Cc1ccc(CNC(C2CCOCC2NC(c2cc([N+](=O)[O-])n[nH]2)=O)=O)nc1C 71330,c1(CNC2CC(NC(COCCOC)=O)C2)ccc(Br)c(C#N)c1 71331,c1(COC2CC3CC(C(=O)OC)C3C2)oc2c(c1OC)CNCC2 71332,C(=O)(C(CC(F)F)N(C)C(C1CCC(=O)CC1)=O)NC1CN(C)CC1O 71333,c1(CC(=O)N(C2CCN(C(c3cc(N)ccc3Cl)=O)C2)C)cnc(O)nc1O 71334,C(=O)(C(CC1CCCC1)NC(=O)CCc1nccn1C)NC(C=C)CO 71335,c1(C(N2CC(N3CCN(C(c4ccc(C)o4)=O)CC3)C2)=O)cn2c(n1)CCC2 71336,C1(C(N(CCCO)C)=O)C2CCCC2CN1C(=O)CCOCCSC1CCCO1 71337,c1(OC)ccnc(C(=O)NCC2C3CN(C(c4nccnc4CO)=O)CC23)c1O 71338,N1(C(=O)Nc2ncccn2)CCC2CCN(C(=O)CN3CCC3)C2C1 71339,c1(CCC(=O)NC(c2cc(C)n(C)n2)C)ccc2c(c1)COCC2 71340,CC(C)C(C#N)C(=O)N1CCC(CCN(C(=O)C(C)N2CCC2)C)CC1 71341,Cc1ncc(C(N2CC3C(NC(c4cnc(-c5cccs5)o4)=O)C3C2)=O)cc1N 71342,C(F)(F)(C(F)(F)F)c1cc(C(N(C2CCN(CC(=O)NC(C)C)C2)CC)=O)no1 71343,CC1CCC2(CO1)CN(C(C1CCC1CNC(c1cn(C)nn1)=O)=O)C2 71344,C1(C(N(C(C)C)CCN(C)Cc2nc[nH]n2)=O)CCC(C)(C)O1 71345,C=CCC(CC)C(=O)NCC(CC)NC(c1ccccc1SCCC)=O 71346,C(=O)(C(O)C(F)(F)F)N1CCCC(C(C(=O)NCC(CC=C)CO)(C)C)C1 71347,c1(C(=O)NCC(C(C)C)NC(c2cc(OC(C)C)ncc2)=O)c(F)cccc1Cl 71348,c1(CC)ccccc1CC(=O)NC1CC12CC(NC(=O)Cc1ccc(C)o1)C2 71349,N1(C(C2CCN(C)C2)=O)CCC(N(C(c2ccc(F)cc2)=O)Cc2ccsc2)CC1 71350,C1(NC(=O)CCC2CCOC2)CN(C(=O)CCNC(=O)C=CCl)C2(CCC2)C1 71351,CC(C)CC(C)(CNC(C12CCC(C)(C1)OC2)=O)NC(c1cc[nH]n1)=O 71352,c1(C(COC)(C)NC(C)(C)C)nnnn1CCNC(C)=O 71353,c1(NCCC2N(C(C3CC(C#C)(O)C3)=O)CCCC2C)ncc(C)c(COC)n1 71354,c1(C(=O)NCCN(C(c2cc(COC)sc2)=O)C)ccc(C2(C)CC2)cc1 71355,c1(C(=O)NC(c2ccccc2)CNC(C2=CCCC2C)=O)nnc2ccccn12 71356,C1(CNC(c2coc3c2CCCC3)=O)CCN(C(=O)CC2OCCO2)C12CCC2 71357,CCC(C)CC(C(=O)N1CCCCCO1)OC(C(C)(C)C)=O 71358,C1(C)(C(=O)NC(C)Cn2cc(-c3ccnn3C)nn2)CCC(F)(F)C1 71359,C12(C(NCP(OCC)(C)=O)=O)CC(C)(CN1C(=O)CCCN(C)C(C)C)C2 71360,C1(CNC(c2ccccc2O)=O)CCN(C(=O)CCCOC2CCOCC2)C12CC2 71361,c1(N(CC(CC)C)C)cccc(S(=O)(=O)N2CCCOC(COC)C2)n1 71362,C(CC(C)C)(C(=O)NC1CN(C(c2c[nH]c(C#N)c2)=O)CC12CC2)NC(C)=O 71363,c1(CC)nccnc1C(=O)NCCCCCNC(=O)C(C1(O)CCOCC1)(F)F 71364,C=CC1CN(C(=O)CCCOc2cccc(C)c2)CC1NC(c1cc[nH]c1)=O 71365,CCCC(C(O)C(=O)NOCCC(C)O)NC(=O)COC 71366,c1(C(C(N2CC3C(NC(C4C(C)(C)CC4)=O)C3C2)=O)=O)cc(F)cc(Cl)c1 71367,C1(CNC(c2c(CCC)onc2C)=O)CCN(C(c2cc(Br)n[nH]2)=O)CC1C 71368,C(CCCC)(C(=O)NCC1CCCC1(C)C)NC(C=CCC)=O 71369,c1(NCC2(C)CCN(C(=O)CC(=O)NC3CC3)CC2)ncnc2cnccc12 71370,C(=O)(C(CC(C)C)n1ccc(C2CC2)n1)NC(CC)CNC(C1CC(F)(F)C1)=O 71371,c1(OC)ccc2ncc(C(N3CC(NC(c4[nH]nnc4C4CC4)=O)C3)=O)n2n1 71372,Cc1cnc(NC(C2C3CCC(C3)N2C(c2cc(I)ccc2Cl)=O)=O)cc1I 71373,c1(C(C(=O)NC)NC(c2ccc(O)c(OC)c2)=O)cccc(Cl)c1Cl 71374,c1(N2CCC(C)C(C)C2)nc(=NC2CCC(C(N)=O)C2)[nH]c2c1CCC2 71375,C1(C(=O)NC2CN(C(Cc3cc(COC)on3)=O)CC2F)CCCS(=O)(=O)C1 71376,c1(C(=O)NCC2(NC(C3CCC(F)(F)C3)=O)CC2)cc2cc(O)ccc2[nH]1 71377,C(C)(CNC(C1CCC(=O)N1C)=O)(C(C)C)NC(c1nc(CCCC)sc1)=O 71378,C1(NC(c2c(COC)cco2)=O)(CO)CCN(C(c2[nH]cc(C)c2C)=O)C1 71379,c1(CNC(COCC#C)=O)nc(C)c(C)o1.C12(CC(CO)C1)C(=O)N2 71380,CCC(CC)CC(F)C(=O)NC(C)(CNC(C1Cc2cscc2C1)=O)CO 71381,c1(Sc2cccc(NC(c3c(OCC)cccc3)=O)c2F)cc(Cl)c(C)cc1O 71382,C1(F)(C(=O)NCC(NOCC)=O)CCN(C(c2ccsn2)=O)C1 71383,C1(NC(C2(COC)CCC2)=O)CC2(CCC(NC(=O)C3=CCCCCC3)CC2)C1 71384,Cc1ncc(CC(=O)NCCOCC(=O)NCC2CCC(=O)N2)s1 71385,c1(C(=O)NC(=O)C(Cc2cn(-c3ncccn3)nn2)C2CC2)ccc2ncccn12 71386,CCCN(OOC)C(=O)C1CCCN(c2c[nH]ccc2=O)C1 71387,C(=O)(CC(C(F)F)NC(=O)Cc1ccnn1C)NC(c1cc[nH]n1)C 71388,N1(C(C(C)Sc2nncn2C)=O)CCOC(CC2CC2CNC(c2cncs2)=O)C1 71389,N1(C(COCC=C)=O)CC(C)N(C(c2cnc(OC)c(Cl)c2)=O)CC1C 71390,c1(C(=O)NC(C)CNC(=O)CC2CCCN2C)sc(F)cc1Br 71391,O=CN1CCCC1C(=O)NCc1nc(CNC(c2cnc(=N)[nH]c2)=O)cs1 71392,Cc1cnc2cc(C(=O)NC3CCCC(NC(=O)CC4(C)CCOC4)C3)nn2c1 71393,C1(C)(C(=O)NC(C2CCN(C(c3cc(N)cc(F)c3)=O)CC2)C)CCN(C)C1=O 71394,c1(CC(=O)NCCCN(C(=O)C(c2cnn(C)c2)C)C(C)C)cn(C)c(=O)cn1 71395,Cc1c(F)ccc(C(=O)NCCC(C)NC(C2C(C)(C)C2(C)C)=O)c1C#N 71396,C1(C(N(C2C3CN(C(c4ccc(C(F)(F)F)nc4)=O)CC23)C)=O)CC(=O)NC1=O 71397,C12(C)CCCN1C2=O.c1(C(N2CCC(CC(=O)OC)C2)=O)cnccc1Br 71398,c1(C(=O)NCC2(NC(C3Cc4n(cc(C)n4)C3)=O)CC2)cc2cc[nH]c(=O)c2s1 71399,N1(C(C(CC(C)C)OC)=O)CC2CC(N=c3nc(C)nc4[nH][nH]cc3-4)CC1C2 71400,C1(C(N2CCC(CSCC)C2)=O)(C(NC(=O)CCC2CCCO2)OC)CNC(=O)C1 71401,CCC(CC(=O)N(C)Cc1nncs1)N(C(=O)C=C1CCOCC1)C 71402,c1(N2CC(C)N(C(COC)=O)C(C)C2)nc(C(F)F)nc2ccccc12 71403,c1(C(C)NC(C2(CCNC(=O)CCC3CCCO3)CCC2)=O)ccc(F)cc1 71404,C=CCCCCCCC(=O)N1CCCC(NC(=O)Cc2cc(C3CC3)no2)C1 71405,c1(SCC)cc(C(=O)NCC2CCCCN2C(=O)C=Cc2cn(C)nn2)ccn1 71406,N1(C(=O)OC(C)(C)C)CCC(C)C1C(N1CCCC(c2noc(C)n2)C1)=O 71407,N1(C(C2C3CCCOC23)=O)CCOC(C2CN(C(C3CCO3)=O)C2)CC1 71408,CC1=C(C(=O)NC2CC2NC(C2(C)CC(C)C2)=O)CCC1 71409,N1(C(C2N(Cc3n(C)ncc3Br)C3C(C2)C3)=O)C2CCCC1COC2 71410,C1(NC(C(C)C)=O)CC2CN(C(c3[nH]nc(C(F)(F)F)c3C(C)C)=O)CC2C1 71411,c1(NC(C2CN(C(CCNC(=O)OCC)=O)CC2C)=O)ccn2cncc2c1 71412,Cc1nc(O)ccc1C(=O)NC1CC(C)N(C(=O)CN2CCCCC2=O)C1 71413,N1(C(C(C)n2cncn2)=O)CCC2(CCN(C(=O)CN3CCCC3=O)C2)C1 71414,N1(C(C2C(=C)CC2)=O)CCC2(CCC2NC(=O)Cc2ccc(Cl)cc2C)CC1 71415,c1(C(C(=O)NC2(C)CC2)N(C)Cc2n(CC)cnn2)nc2c(s1)CCCC2 71416,C1(O)(C(=O)NC(CNC(c2[nH]cc(CN(C)C)c2)=O)CO)CCCCCC1 71417,O=C1COc2ccc(CCN=c3nc(N4CCOCC4)cc(C(F)(F)F)[nH]3)cc2N1 71418,C1(NC(=O)CCSC2CN(C(=O)CCc3ccccn3)C2)CC2(CCC2)CO1 71419,c1(C(N(CC(C)NC(=O)COc2ccc(F)c(Cl)c2)C)=O)ccc2scnc2c1 71420,CC1(C)CN(C(C2(C)CC(C#N)C2)=O)CCC1NC(C1C2CCCCCC12)=O 71421,C1(C)(C(=O)NCC(CNC(C2C(C(C)C)CCC2)=O)O)Cc2ccccc2C1 71422,C1(C(=O)NC(c2ccc(C)cc2)C(F)(F)F)COC(C)(C)N1C(C(C)(C)C)=O 71423,N1(C(C(C)Oc2ccc(F)cc2)=O)CC2OCC(NC(=O)C(C)(C)OC3CC3)C2C1 71424,c1(C(N2CCCC(CC)C2)C(=O)NCCC2CC2)ccc2c(n1)CCCC2 71425,N1(C(CC)=O)CCCCCCC1C(=O)NC(c1ccccc1)C 71426,Cc1c(Cl)ccnc1C(=O)NC(c1ccc(F)cc1F)C1(N)CCC1 71427,C1(NC(c2cocn2)=O)(CO)CCCN(C(=O)C(c2ccc(Cl)cc2)CO)C1 71428,N1(C(c2c(OC)cccc2O)=O)CCC2(CCN(C(C3CC(CCO)C3)=O)C2)C1 71429,C1(C(=O)NCC(C)CNC(=O)CNc2ccc(C(N)=O)cc2)CCC(F)CC1 71430,CN1CCN(C(=O)C(C2(C)CC2)NC(C2COCCN2C=O)=O)CC1CO 71431,c1(C(c2ccccc2)NC(c2ccccc2C(F)F)(C)C)ccc(Cl)cc1 71432,N1(C(N2CCN(C(C)(C)C)CC2)=O)CCCC(C(=O)NC2(CC(=O)NCC)CC2)C1 71433,c1(CNC(C2CCN(NC(c3c(C)cc(O)cc3)=O)C2)=O)csc2sc(C)cc12 71434,C#CCC(CC#C)C(=O)NC(C)CN(C(=O)CCC(C)(C)OC)C 71435,c1(OC)ccc(F)cc1CCC(N1CC2(CCN2C(=O)C(O)CCSC)C1)=O 71436,Cc1cnc(C(=O)NCC2CC3CC3N2C(=O)C(C)n2cccc2)cc1C 71437,C(=O)(C1=NOC(CNC(C2(C#N)CC=CC2)=O)C1)NC(CSCC)CO 71438,Cc1cc(C#N)cnc1C(N1CCC(OCCNC(c2cscn2)=O)CC1)=O 71439,c1(C(=O)NC2CN(C(C3(C)CCCCC3)=O)CC(F)C2)ccc2c(n1)CCC2 71440,c1(C(=O)NCCS(CC)=O)ccc(CN2CCC(C)(C)C2)cc1C 71441,S(C(=S)N1CCCCC1)NC(NCC)=NCc1cc(F)ccc1OC.C1CC1 71442,C(=O)(C(=O)C(F)(F)F)NCCCC(C)NC(=O)CCOCCNC1CC1 71443,N1(CC)CCCC(C2CNC2)C1.Fc1cccc(C(C2CCCCC2)N)c1 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71797,C1(C(N2CCC(COCC)C2)=O)CC12CCN(C(C1(O)COC1)=O)CC2 71798,n1(CCC(=O)NC2CN(C(C3CC34CC4)=O)C2)c(=O)oc2cc(Cl)ccc12 71799,N1(C(Cc2c(C)nn(C)c2)=O)CC2(CC(NC(=O)COc3cnn(C)c3)CO2)C1 71800,C1(n2c(-c3c(SCC)cncc3)nc(-c3ccnn3C)n2)CC2CCC(C1)C2O 71801,C12(C(N3CCC(NC(CC)=O)C3)=O)CCCC1CCN2C(C1CC2CC(=O)C1O2)=O 71802,C1(CC)(NC(C2CC(C)CO2)=O)CCN(C(c2cc(CC(C)C)nn2C)=O)CC1 71803,c1(C(=O)NCCCN(C(=O)CC2CC2C)C(C)C)cnc2c(c1)NC(=O)CN2C 71804,c1(OC)cncnc1C(=O)NC1CC(O)(CNC(c2ccc(C3CC3)cc2)=O)C1 71805,N=c1nc(N2CCC(CF)CC2)[nH]c(=NC2CSCc3ccccc32)[nH]1 71806,C1(C2CCN(C(=O)CN(C)CCO)C2)(NC(C(C)OCCN(C)C)=O)CC1 71807,CCC(CCCC(F)(F)F)NC(=O)NC(c1ccc(C)cc1)CF 71808,c1(N2CC3C(O)C3C2)nc2c(c(=NC3CCc4ccc(F)cc4C3)[nH]1)CCC2 71809,CN=c1cc[nH]cc1S(=O)(=O)N1CCCC(C(=O)O)CC1.C1CCCSC1 71810,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCO)nn1)=O 71811,c1(-n2cc(C(N3CCCC3C(O)C(F)(F)F)C(=O)O)nn2)ccc(F)cc1Br 71812,Cc1ccc(CN(S(=O)(=O)C(F)(F)F)C2CCCC2)c(C)c1 71813,C(C(=O)N(CCCNC(C1(F)CCCC1)=O)Cc1ccccc1)(C(C)C)OC 71814,C=CCCCCCCCCC(C(=O)NCCCF)N1C2CCCC1CC(O)C2 71815,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 71816,CC(C)C(CC(=O)NCC1(NC(=O)Cn2ccccc2=O)CCOC1)C(C)C 71817,C(c1cccc(Cl)c1Cl)=CC(N1CCCC(NC(C(C)C(=O)N(C)C)=O)CCC1)=O 71818,C1(C(CO)NC(C(CC)OC)=O)CCN(C(C2CCCO2)=O)CC1 71819,CC1CN(C(C)C(=O)Nc2ccccc2C(N)=O)CCC1O 71820,c1(C(=O)NCC2(O)CN(C(C(C(=C)C)(C)C)=O)C2)cc(C)cc([N+](=O)[O-])c1N 71821,c1(CC)cccc(C(=O)NCC(C(=O)N2CCC2C(=O)NC)N(C)C)n1 71822,c1(CCNC(c2nnnn2-c2ccc(Br)cc2)C2CC(=C)C2)cc(C)oc1C 71823,c1(OCC(=O)NC2CCC(F)(CNC(C34CC(CCO3)C4)=O)C2)cccc(F)c1 71824,c1(C(=O)NC(C2CN(C(CCCOCC)=O)C2)C)cncc(C)c1C 71825,C1(C(=O)C2CC2)CC2(C1)CN(C(=O)C(F)Sc1c(OC(F)(F)F)nsc1)C2 71826,Cc1cccc(NC(=O)C(=O)Nc2ccc(-n3ccnc3C)nc2)c1C 71827,C(CCCCCN=c1[nH]c(Cl)ncc1F)NC(Cc1c(C)[nH]c2ccccc21)=O 71828,N1(c2c(C(=O)OC)cc(C)s2)CCC2(CC1)CC(CNC(=O)C(C)N(C)C)CO2 71829,CCCC(C(O)C(=O)N1CCCC1C1CC1)NC(=O)Cc1csc(C)c1 71830,C1(CC(=O)NC2C=CC(CNC(C(C=C)(C)C)=O)C2)CC(=O)NC(=O)C1 71831,C1(C(=O)NCC#CC)CCCCCCN1C(c1[nH]ccc1CC)=O 71832,N1(C(Cc2ncn(C)c2)=O)CC2(C1)CN(C(=O)C(O)CCc1ccccc1)C2 71833,c1(OC)ccc([N+](=O)[O-])c(NC2CC3CN(C(=O)C(C)S(N)(=O)=O)CC23)c1F 71834,C(Br)(C(=O)N(CC(O)CN(C(=O)C(=O)NCC1CC1)C)C)=C(C)C 71835,C(CCCOC)(C(=O)N1CC(O)CC1(C)CO)NC(c1ccc(CC)s1)=O 71836,N1(C(CCC)=O)CCCCC1C(N1CC(O)(CNC(=O)C=CCOC)C1)=O 71837,N12CCN(CC1)CCC(C)(C)C2.CC(Cn1cncn1)C(=O)NC(=O)C(Cl)=CCl 71838,n1(CCC(=O)NCCNCCC(C(C)C)OCC)cnc(C)cc1=O 71839,c1(C(=O)NC2C(C)(C)N(C(=O)CCC3CC3(F)F)CC2)n[nH]c2c1CCCC2 71840,C12(CNC(C(C3CCC3)OC)=O)CCC(CC1)N2C(=O)CSC(C)C 71841,c1(OCC)ccc(-c2nc(C3CCCN(c4cc[nH]n4)C3)n(C3CCC3)n2)cc1 71842,c1(C(=O)NC2CN(C(c3c(C(C)C)nns3)=O)CC2F)cccc2c1OCCO2 71843,C(CCCCC(=O)NC1CC2COCC12)N(C(=O)CCCCCF)C 71844,Cc1ccc(C(=O)N(C(CNC(=O)C(N2CCN(C)CC2)C)C2CC2)C)n1C 71845,CC1(CNC(=O)CCc2cnc(C3CC3)o2)CCCN1C(c1cc[n+]([O-])cc1)=O 71846,N1(C(CCN(C(c2cc(CC)oc2C)=O)CC2CC2)=O)CCN(C)C(=O)C1 71847,c1(CNC(c2c(C)con2)=O)ccc2c(c1)CCC2NC(=O)C(O)CCC(F)(F)F 71848,C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(=O)Cn2nc(C)n(C)c2=O)CC)CC1 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71866,C(=O)(C(C)C(F)(F)C(F)F)N1C2(CN(C(CN(C(C(C)C)=O)C)=O)C2)CC1 71867,CN1C(=O)Cc2ccc(C(=O)NCC(C)(C)NC(=O)C(C)(Cl)Cl)cc21 71868,C1(NC(c2c(C)cc(CNC(=O)CC3(O)CCOC3)o2)=O)CCn2nnnc2C1 71869,C1(C(=O)NC(C2CCCN2C(C2CC(F)(F)C2)=O)(C)C)CCCC2(C1)CC2(F)F 71870,N1(CC)N=C(C(=O)NC2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)CCC1=O 71871,c1(C(N(CCC(=O)NC2CCCOC2)CCO)=O)n[nH]c2c1CCC2 71872,C12(C(N3CCC(CCNC(Cc4nnc(C)o4)=O)C3)=O)CC3CC1C2C3 71873,N1(C(C(C2CCCC2)OCC)=O)CC(NC(=O)C=CC=C(Cl)Cl)C2(CC2)C1 71874,C1(NC(=O)CCN2CCCC2=O)CC2CCC(C1)N2C(=O)Cc1cc(F)ccc1Cl 71875,N1(C(c2cn(CC)nc2)=O)CCN(C(=O)CCc2cccc(Cl)c2)CCC1C 71876,C1(CC(=O)N(CC(C)NC(C2(F)CC2)=O)C)CCC2(CCC2)CO1 71877,C1(C(=O)NCCCC(C)NC(CCCCC#C)=O)CCC2(CCCC2)C1 71878,c1(C(=O)OC)nc(=NCC(C)CNC(=O)CCC(C)OC(C)=O)c(F)c(Cl)[nH]1 71879,C1(NC(C=CCOC)=O)CCC12CN(C(=O)CC1(O)CCCC1)C2 71880,c1(CN(C(=O)Cn2cc(-c3ccc(Br)cc3Cl)nn2)C)ccc2cccc(Br)c2n1 71881,N1(C(c2cnc(C#N)s2)=O)CCC2(CC1)CC2CNC(=O)CNC(=O)C1CC1 71882,c1(NCC2CCN(C(C(C)NC(c3ccco3)=O)=O)C2)ncc(F)cn1 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71901,c1(COC(C(C(=O)N(c2cccc(Cl)c2Cl)C)N)=O)cnnc(O)c1Cl 71902,CC1(CC(=O)NC2CCCC(NC(=O)C(C)(C)c3ccccc3)C2)CCCCC1 71903,C(=O)(C1OCCc2ccccc21)NCC1N(C(c2c(C)c[nH]n2)=O)CCC1(C)C 71904,c1(OC)ccc2c(c1)CC(C(=O)NCC(C(C)C)OC)O2 71905,C(C(=O)N(CC(C)SC)C)(C(C)C)N(C(CCOCC)=O)C 71906,c1(OC)ncnc(C(N2CCC(CCNC(=O)Cc3cnnn3C)C2)=O)c1F 71907,C1(NC(c2cnn(CC(F)F)c2)=O)CC(NC(=O)C2CC2)C12CCC2 71908,N1(C(=O)NC(C2(C)CCN2C(=O)OC(C)(C)C)C(C)C)CCC(CCO)CC1 71909,C(=O)(C(C(C)C)N1CCC1)NC(c1ccccc1)CNC(C(C)(C)OC)=O 71910,c1(C(N(C)CC2COCCN2C(=O)C(C)(C)CC#N)=O)cnn2c1N(C)CC2 71911,C1(C2CCN(C(C3CCCC(=O)CC3)=O)CC2)(NC(C(CC)NC(C)=O)=O)CC1 71912,c1(C(N2CCC(C)(C)C2C(=O)NC2CC2C2CCCC2)=O)c[nH]c2ncccc12 71913,c1(C(N(C2CN(C(C3ON=C(C)C3)=O)CC23CC3)C)=O)n[nH]c2c1CN(C)CC2 71914,C1(CC(=O)NS(=O)(=O)CCCl)OCC2CCN(C(c3cnc(F)cc3Cl)=O)CC12 71915,N1(C(C2CC(C#C)(O)C2)=O)CC(C)N(C(c2cnn(CC)c2C)=O)CC1C 71916,C(=O)(C(F)(CNC(C1CCCC1C(C)C)=O)C(C)C)NCCNC(=O)NC 71917,Cc1nc(CCC(=O)NCC(CNC(=O)CCC2CC(F)(F)C2)CO)cs1 71918,C#CCCC(N)C(=O)N1CCCC(C(=O)NCCCC2CCCC2)C1 71919,C1(CNC(c2c(C)ncs2)=O)CN(C(c2cc(C#N)c[nH]2)=O)CCC1C 71920,c1(C(=O)NC2(C)CCCN(C(C=C(C)C(F)F)=O)C2)cccn2c(C)nnc12 71921,C=CC1(C(=O)NCC(O)CC(F)(F)F)CCN(C(C2CCC(OC)CC2)=O)C1 71922,C(=O)(C1=CC2CCCCCCC12)NCC(CNC(c1nn(C)c(F)c1)=O)O 71923,C1(CC=C)(NC(C2(C)CC3CC3C2)=O)CCN(CC2(SCC)CC2)CC1 71924,CC(C)CC(C(=O)NC1CC(CN(C)C)C1)ONC(c1ccncc1F)=O 71925,C(=O)(CCC(C)(C)NC(=O)C(C1CCCCC1)O)NC(CC)CNC(C)=O 71926,c1(C(=O)NCC(C)N(C(=O)CN(C)S(N)(=O)=O)C)ccc2c(c1)OCCO2 71927,C#CC1(NC(C2CCCCN2C(=O)C(F)=CC2CC2)=O)CCC(C)(C)C1 71928,c1(C(=O)NC2C(CC(=O)NCC3OCCN(C)C3)CCCC2)cnc2n1CCC2 71929,CCC(C(=O)NCCOC(C)(C)CNC(c1ccc(F)cn1)=O)C(C)(F)F 71930,C#Cc1ccccc1CC(=O)NCC(N1CCC2(CSC2)C1)=O 71931,C1(C(C(N2CCCc3cnn(C)c32)C)=O)CC2(C1)CS(=O)(=O)C2 71932,N1(C(c2c(CC)nn[nH]2)=O)CC(C2CCCN(C(=O)C(C(C)C)C(C)C)C2)C1 71933,C12(CNC(C=Cc3cnc(C)s3)=O)CCC(CN(C(=O)Cc3cnccc3)C1)C2 71934,c1(CN2CCC(CC(=O)Nc3c(C(N)=O)occ3)C2)cc(O)ccc1F 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71953,c1(C(=O)OCCOc2c(OC)cccc2)cc(F)nc(F)c1F 71954,S(=O)(=O)(c1ccc2nc(Cl)cnc2c1)N1CCC(N(C(C2(CC)CC2)=O)C)C1 71955,c1(C(C(=O)NCCCF)N(C)Cc2cnc(CC)[nH]2)cnc(C)n1C 71956,c1(C(=O)NCCC(=C)CNC(c2oc(CC)nc2C)=O)cnc(N)c(N)c1 71957,c1(C(N2CC3C(NC(CC(C=C)CC)=O)C3C2)=O)ccc(=NCC2CC2)[nH]c1 71958,c1(C(N2CC(CN(C(CCOCC(C)C)=O)C)C2)=O)cc(C2CC2)cc(F)c1 71959,c1(COC)nc(C(=O)NCC(C2CC2)N(C(=O)C=NOC)C)co1 71960,N1(C(CCCOCCOCC)=O)CC2C(N(C(=O)C(C(C)C)SCC)C)C2C1 71961,C1(CN(C)C(C)C)CN(C(=O)CNC(C(COC)O)=O)CC2(CCC2)O1.C1C(=O)N1 71962,N1(C(C2CCCCO2)=O)CC2CCN(C(=O)COc3ccccc3Br)C2C1 71963,N1(CCC)CC2(C1)CN(Cc1cnc(NCC3(O)CCCC3)c(Cl)c1)C2 71964,C(CCC(C)CC(C(=O)Nc1cccc(Cl)c1)N1CCC(C(N)=O)C1C)=C(C)C 71965,CC(C)C(CC1CCCC1)C(=O)NCC1CCCN(C(c2cnc(C(C)C)o2)=O)C1 71966,CCCCCCC(C)CC(=O)N1CCN(C)C(CNC(c2cc(C)sc2N)=O)C1 71967,c1(C(N(CCCN(C)C)CCC)=O)ccn2ccccc12.C1(C)C(C)C(=O)N1 71968,C(C(CC(C)C)C(=O)NC1CC(O)C1CC(N1CCC(CCF)CC1)=O)OC 71969,C1(CCC(C)(C)NC(C)=O)CN(C(=O)CC2CC(OC)C2)CCO1.C1(C)C(=O)N1 71970,c1(CC(N)=O)cn(C(C2CC2)NC(=O)CC2CC2CC(CO)C2CC2)nn1 71971,c1(CNC(C(C2CN(C(CN(C3CC3)CC)=O)C2)OC)=O)cc(C)cnc1O 71972,C1(NC(CC=CCC)=O)CCC(C(N2CCC(F)CC2)=O)OC1 71973,c1(OC)ccc(CC(=O)NCC(CO)NC(C2CCC2OC)=O)cc1 71974,S(=O)(=O)(c1ccc(N2CCc3noc(N)c3C2)cc1Br)NC(CCC(=C)C)C 71975,C12(OC)CCCC(C(=O)NC(C)(CNC(=O)C3=C(Cl)CCC3)C3CCC3)(CC1)C2 71976,c1(C(=O)NC(C2CCN(C(=O)C=C3CCOCC3)CC2)C)cc(N(C)C)ccn1 71977,C1(N(C(=O)CC2(NC(C3C=CC3C(=O)N(C)C)=O)CCC2)C)CS(=O)(=O)C1 71978,C1(C2CCCN(C(=O)C3=CCCCC3)C2)(NC(=O)CC2COC(=O)C2)CC1 71979,c1(C(=O)NC(C(=O)NCCC(F)(F)CO)C2CCC2)cccc2nccn12 71980,C#Cc1ccc(C(=O)NCC(Cc2ccccc2)NC(=O)C(O)C2CCC2)cn1 71981,c1(CC)nn(C)c(CC(=O)NC2CC2NC(=O)COc2cncc(Cl)n2)c1Br 71982,CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCC1N(C(=O)CCN1CCOCC1)C 71983,C=CCC(C(=O)NCC1CCC(NC(=O)CCc2ccc(C#N)cc2)C1)C(C)C 71984,c1(C(=O)NC2(CN(C)C(C3(C)CC(C)(C)C3)=O)CC2)cccc(CS(N)(=O)=O)c1 71985,c1(CNC2C(C(=O)Nc3cc(C)c(I)cn3)CCC2)c[nH]c2ccc(Cl)cc12 71986,c1(C(=O)NC2CC(NCc3c(C)occ3)C2)ccc(-c2ccccc2)cc1 71987,c1(COC)ncccc1OCC.C12CC1C(=O)N(CC(=O)CC)CCCNC2=O 71988,C1(NC(COCCCOC)=O)CN(C(c2cc(C(C)C)nn2C)=O)C2CC12 71989,c1(NC(=O)NC(CC(=O)OCC)c2ccccc2)cccc(CC(C)C)c1 71990,CCCCC(O)CC(=O)NC1C2CCC(C2)C1C(=O)NCC(C)OCCO 71991,N1(C(c2cc(C)n(C)n2)=O)Cc2ccccc2C(CNC(C2C=CCC2)=O)C1 71992,CC1CCN(C(=O)COCCCOC)C(C(N)=O)C1.c1(C=O)cc[nH]n1 71993,c1(CN2CCCC(n3ccnc3-c3ccccc3)C2)cc2cccc(F)c2o1 71994,N12CC(C(C(C)C)C1)C2=O.Cc1cscc1CNC(=O)Cn1nnnc1C 71995,C1(C(=O)NC(C)CCCCNC(=O)CN2CC(C)(O)C2)(OC)CCC(C)(C)CC1 71996,c1(C(=O)NCC(CC(C)C)NC(C2(OC)CCCOC2)=O)cc(C)ccc1F 71997,CC1CN(C(c2sccc2CN(C)C)=O)CC1CCNC(c1snc(Cl)c1Cl)=O 71998,C1(OC)CCC2(CCN(C(c3coc(NC(C4CCCCC4CO)=O)n3)=O)C2)C1 71999,C1(NC(Cc2scc(C)c2)=O)CC=C(C(=O)NC2C(C)CCC2C)C1 72000,CC1(C#CC(=O)NC2CC2CNC(c2c(F)c(F)cc(F)c2F)=O)CCCO1 72001,c1(C(C)(C)C)ncc(C(=O)NCC2(O)CN(C(=O)CCCc3ccccc3)C2)s1 72002,C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(=O)CSCC(F)(F)F)C12CC2 72003,S(=O)(=O)(c1c[nH]ccc1=NCC1CN(C)CCN1C)N(CCC)CC1(C)CCCC1 72004,C(=O)(C(C)(C)C(=O)NC1CCC(CC(=O)NCCCc2ncnn2C)C1)N(C)C 72005,N1(C(CCCOC)=O)CCCC2(C1)C(NC(c1nc(C)ncc1Cl)=O)CCN2C 72006,C(=O)(CC(C)(C)O)NCCCC(C)NC(=O)C(F)(F)c1cncs1 72007,c1(C(N2C(CNC(CNC(C)=O)=O)CCC(C)(C)C2)=O)cnc2ncc(Cl)cn12 72008,Cc1cc(C(C)(C)C(=O)N2CC(C(C)NC(=O)C(C)(Cl)Cl)C2)cs1 72009,C1(NC(c2cc(C(C)(C)C)on2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1 72010,c1(C(=O)NCC(CNC(C(COC)(F)F)=O)CO)cc2nccnc2cc1F 72011,N1(C(c2c(CC)nc[nH]2)=O)CCC2CCN(C(=O)C#CC3CC3)CC2C1 72012,C1(NC(CN(CC)CC)=O)COCCC1NC(=O)C(CC)SC 72013,C1(C(=O)NCCC=CC(=O)NCCC(=O)NCC)C2CC3C(C2)C13 72014,c1(NC(C2C(C)(C)C(NC(=O)COCCNC(N)=O)C2)=O)cc(Cl)c(Cl)c(Cl)c1 72015,C1(NC(C(C2CCCC2)OC)=O)C2CCC1N(C(=O)Cc1cn(C)nc1C)C2 72016,C(=O)(CCS(N)(=O)=O)N1CC(C)(C(N2CCC(CC(C)(C)C)C2)=O)C1 72017,C(=O)(C1=COc2ccccc2O1)NC(C(C)NC(CC=CC=C)=O)C 72018,Cc1sc(C(=O)NCC2CC(NC(=O)CCc3ccccc3F)C2)nc1O 72019,CCC(O)C(=O)NC1(CCNC(=O)C(c2cncn2C)O)CCC1 72020,Cc1cc(=O)c(C(=O)NCC(n2cc(C3(C)CSC3)nn2)C)nn1-c1nccs1 72021,CC1CC(C(N2CC(CCNC(C3(C(N)=O)CC3)=O)C2)=O)CO1 72022,C(=O)(C(CC(F)F)c1ccccc1)Nc1cccc(NC(c2n(C)nnc2)=O)c1 72023,C(=O)(C1=CC(O)CCC1)NC(C)CCNC(c1c(Cl)csc1Cl)=O 72024,c1(C(C)N(C(C(=O)N(C)C)C2CCCC2)CCCO)ccc(Br)s1 72025,C1(NC(C(C)=CCN(CC)CC)=O)CC2CCC1N2C(c1cc(C)nnc1O)=O 72026,N(C(=NCC1COCCO1)NCc1nnnn1C)C(c1ccc(Cl)cc1)COC 72027,CCC(O)C(C)(C)C(=O)NC1CC(F)(F)CC1NC(C)=O.C1(N2C(=O)C2)CCCC1 72028,N1(OC(C2C(CCC)CCC2)=O)CCN(C(=O)CCc2ccc(C(=O)O)[nH]2)CC1 72029,CCCC(C(=O)NC1COC(CCC2CC2)C1)NC(=O)CC1CCOC1(C)C 72030,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC(C1)CN(C(C1CC(C)CO1)=O)C2 72031,N1(C(c2n(C(C)C)nc(C3CC3)c2)=O)C2CCC1CC(NC(=O)C(O)CF)C2 72032,N1(C(C(C)OCCCC)=O)CCN(C(C2CC3CCCC23)=O)C(C2CCC2)C1 72033,C1(C)(C(=O)NC2CN(C(COC3(C#C)COC3)=O)C(CO)C2)CC2(CCC2)C1 72034,CCCC(C(=O)N1CCCC(NC(=O)NCC2CCCCC23CCC3)C1)C(C)C 72035,C(CCCCCC(=O)NOCCCO)NC(C(C)(C)OCC)=O 72036,C(C(=O)NC(C(=O)N(C1CC=CC1)C)C1CCCC1)(C(C)C)OC 72037,c1(-c2cn(C)nc2)ccc2c(c1)COC2.n12[nH]c(cc1=O)-c1ccc(cc1)C2 72038,CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CCN1C(=O)Cc1ccccc1CC#N 72039,Cn1nc(C(=O)NC(CCF)C(=O)NCCOC2CCOC2)cc1CO 72040,N1(C(c2cccc(C)c2C)=O)CCC2CN(C(=O)CC(C)n3cccc3)CC12 72041,N1(C(CCC(CC)C)=O)CCOC2(CCN(C(=O)C(C)C3CCC3)CC2)C1 72042,C(=O)(C(CC)C(=O)OCC)N1CCC(C(C)(C)NC(c2n(CC#C)cnn2)=O)C1 72043,C(CCCCCNC(c1ccncc1Cl)=O)NC(C(C)ONC(=O)OC(C)(C)C)=O 72044,c1(SC)sccc1C(=O)NCC1CC1NC(c1cn(CC2CNC(=O)O2)nn1)=O 72045,N1(C(C(=O)NC(C(=O)OC)C)c2ccsc2)CC2C=CC2C1 72046,C=C1CCN2C(C1)C(=O)N(C)CC(O)C(=O)N1CCC(CC1)C2=O.OC 72047,C1(CNC(Cc2cc(C)nc(C)c2)=O)CC(C)(C)CCC1NC(=O)CCF 72048,N1(C(CC(C)N(C)C)=O)CCCC1(C)CNC(C1(C)CCOC1)=O 72049,N1(C(C2(OC)CCC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CC(F)F)C1 72050,c1(CN2C(C(=O)NCc3ccc(C#N)s3)CCC2)c(I)ccnc1Cl 72051,C1(NC(c2n(CC)ccn2)=O)CCN(C(c2cccc(C)c2)=O)CC(C)(C)C1 72052,S(=O)(=O)(c1cc(C(=O)O)c(Cl)cc1Cl)CN1CCC(C#C)CC1 72053,N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(=O)C=CCOC)C(c2cnn(C)c2)C1 72054,C1(C(=O)NCC(C)NC(=O)CCc2cccs2)CC1(C)C 72055,CCC(c1ccc(OC)cc1)=CC(=O)NC1CC1NC(c1c(C)noc1C)=O 72056,C=CCCC(C(=O)NCC1(O)CN(C(c2ccc(N)cc2Cl)=O)C1)c1ccccc1 72057,C1(C(=O)NCCc2nc(CC)[nH]n2)N(C(=O)C(O)CSC)CC12CCCC2 72058,N1(C(c2c(F)ncc(C)c2)=O)CC(N=c2[nH]nc(CCN(C)C)s2)CC(C)(C)C1 72059,C(=O)(CCC(CC)CCC)NCC1C2CN(C(CC3(C=C)CC3)=O)CC21 72060,c1(C(C(=O)O)NCC2(C)CCCS2)ccc(F)c(F)c1 72061,c1(C(N2CCC(OC)C2)C(=O)OC)nccn1CC(C)C 72062,c1(OC)ccc(COC(C23CC2CN(Cc2cccc(F)n2)C3)=O)nc1 72063,CC1(C)C(CO)CCN1C(=O)Nc1ncc(-c2ccccc2)c(=N)[nH]1 72064,N1(CCOCC)CCN(C(=O)CC2CCCN2C(=O)CCc2nc(C)no2)CC1 72065,c1(C(=O)NCCN2CCN(C(CN(C)S(N)(=O)=O)=O)CC2)cc2cccnc2[nH]1 72066,c1(OC)ccc(C(N2CCC(N(C(=O)C(O)P(C)(C)=O)C)C2)=O)c2ccoc12 72067,C(=O)(C1=CC(C)(CC)C1)N1C(COC)(CNC(=O)C(c2cccnc2)O)CCC1 72068,C(CN(c1cccc(Cl)c1)C)(CN=c1[nH]c(NCCOC)nc2c1SCC2)OCC 72069,N1(C(C2C(SCC)C2)=O)CCCCC1C(=O)NCC1(C(N)=O)CCCC1 72070,C1(C(C)C)C(NC(C2(C)CC2)=O)CCN1Cc1cnc[nH]1 72071,C1(CC=C)(NC(c2ccccc2)=O)CN(C(C2C(CC=C)CC2)=O)C1 72072,N1(C(CCCOC)=O)CCC2CCCC(C1)N2C(C1CCC2(CC2)C1)=O 72073,c1(OC(C)C(=O)NC2(C(=O)NC3CC(F)(NC(N)=O)C3)CC2)ccccc1 72074,c1(C(=O)NCCC2CCN(C(c3cc(N(C)C)ncc3)=O)C2)c(F)cncc1Cl 72075,c1(C(N2CCC(C)C(CO)C2)=O)cc(P(C)(C)=O)cs1 72076,N1(C(c2cc(CC(C)C)on2)=O)CCN(C)C(CNC(C2CCSC2)=O)C1 72077,C(=O)(CCCC(C)(C)C(=O)NCC=CCNC(=O)CSc1ccc(C)cc1)OC 72078,c1(C(N(C2CCCC(NC(C(F)=CC)=O)C2)C)=O)cnc(C)nc1C 72079,N1(C(c2cc[nH]c2C2CCC2)=O)CC2CCC1CN2C(c1snnc1C1CC1)=O 72080,c1(CCC)sc(C(=O)NC2CCC(NC(C3CCC(=O)N3)=O)C2)cc1COC 72081,c1(C(N(CCCNC(c2cc(CC)sn2)=O)C2CC2)=O)ccn2cnnc2c1 72082,c1(C(=O)OCC)cnc(=NCC2CC2CNC(=O)CCc2ccccc2F)[nH]c1 72083,CC1CC(C(=O)NC2(C(=O)N(CCCO)C)CC(O)C2)CCS1 72084,Cc1cc(C(=O)NC(CN(C)C)C(=O)NCCc2ccccc2O)c(C)n1C 72085,c1(OC(c2ccccc2Oc2ccc(Cl)c(I)c2)O)cccc2c(Cl)cc(Cl)nc12 72086,CC(CC(=O)NC(C)CC1CN(C(c2ccccc2)=O)C1)NC(=O)C1CC1 72087,c1(C(N2CC(CN(C)CCO)C2)=O)ccnc(CC2CCCN2C)n1 72088,N1(C(c2cc(CC)ncc2)=O)CC2(CCCC2NC(C2CC2F)=O)C1 72089,c1(CNC(C2CCN(C(CNC(=O)OC)=O)CC2)C2CC2)c(C)cccc1C 72090,C(=O)(CC(C)C(=O)N1CCC(C(C)C(=O)N(C2(CC)COC2)C)C1)OCC 72091,C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2cnnc(O)c2)=O)CC1C1CC1 72092,n1(CC(=O)NC(C(C)(C)C)CNC(=O)C(C)(C)c2cnco2)cc(F)ccc1=O 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72111,CCC(C)(COC)C(=O)NC1CCC(CCC(=O)NCC2(F)CC2)C1 72112,C(=O)(C1=NOC2(C1)CN(C(c1cc3ncccn3n1)=O)C2)OCC 72113,c1(CNC(c2ncccc2O)=O)ccc(OC(F)(F)F)cc1.C12(F)CN(C1)C2=O 72114,C1(C)(NC(C(CC2CC2)OC)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1 72115,c1(C(N2CCCC2C2(C(=O)NCCC3CCOC3)CC2)=O)nc2ncccn2n1 72116,C1(NC(c2nc(CNC(C(CC)CN(C)C)=O)oc2C)=O)CC(C)(OC)C1(C)C 72117,N1(C(c2ccccn2)CC)CCN(CC(=O)NCCn2nnnc2C)C(C(C)C)C1 72118,N1(C(c2n(CC#C)ccn2)C(=O)NC)CCNC(=O)C1C(C)C 72119,CC(C(=O)N(C1CCC(NC(c2cccc(O)c2F)=O)CC1)C)P(C)(C)=O 72120,N1(C(c2ncc(Br)s2)C(=O)NCC(=C)C)CCCC2(CCO2)CC1 72121,c1(CC(=O)NC2C(CSC3CC(F)(CF)C3)C2c2c[nH]cc2Br)ccccc1OC 72122,CC1CCCCC1C(=O)NCCC1CCCN(C(=O)CSCC2CCCO2)C1 72123,C1(OC(C)CC(=O)N(C)CC)CCC(NC(C2OCCC2C(C)C)=O)CC1 72124,C(CC(C(=O)NC1CN(C(C)(C)C)C1)NC(C1(SC)CCOCC1)=O)OC 72125,CC(CN=c1[nH]c2c(c(=NCC3CC4C=CC3C4)[nH]1)COC2)n1cccn1 72126,C1(NC(CC2CCC(C)C2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2(CC2)C1 72127,C(=O)(C(C)(CO)NC(c1ccncc1)=O)NCC(C)(C)OCC(F)(F)F 72128,C1(NC(CCN(CCC)C)=O)C2CCCN(C(C3CCSC3)=O)C2C1(C)C 72129,C1(NC(c2ccc(Cl)[nH]2)=O)CCC(CNC(c2ccnn2C2CCC2)=O)C1 72130,c1(C(=O)NCC23N(C(C4C(C)(C)CO4)=O)CC(C2)C3)ccc2ncnn2n1 72131,c1(CC(=O)NCC(CN(C(CCC2CCN(C)CC2)=O)C)O)cccc(F)c1Cl 72132,N1(C(CSCCOC)=O)CCC(NC(=O)CC2CCOC2)CC1C 72133,c1(C(N(C2CCN(C(=O)C(COC)COC)C2)CC)=O)nn(C)c(C)c1Cl 72134,c1(C(=O)OC)c(C)ccnc1NC(C1CCN(C(=O)C(C)CC2CCC2)C1)C 72135,S(=O)(=O)(c1ccccc1F)Nc1ccc(Cl)o1.C12CC1C(=O)NC2 72136,c1(CC(=O)N(C2C3CCC2CNC3)c2cccc(Cl)c2)cc(F)cc(F)c1F 72137,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(c2nccnc2C#N)CC12CCC2 72138,C1(CC(N2CC(OCCC(=O)NC(C(C)C)c3nc[nH]n3)C2)=O)NC(=O)NC1=O 72139,C(=O)(CCP(C)(C)=O)NC1CC(N(C)C(C2CN(S(=O)(=O)C(F)(F)F)C2)=O)CC1O 72140,c1(N2CC(F)C(F)C2)nc(=NC2CCC(CC(F)(F)F)C2)[nH]c2cccnc12 72141,n1(CCC)nnnc1C1(NCC(C2CC2)C2CC2)CC(C)C1 72142,N1(C(c2ccn(CC)n2)=O)C(C)CC2CN(C(c3c(C)coc3COC)=O)CC12 72143,Cc1cccc(C2CC2S(=O)(=O)NC2CC(CNC(=O)OC(C)(C)C)C2)c1 72144,N1(C(CCC)=O)CC2CC1CN2C(=O)CCN1CCCCC1C.C1CCCO1 72145,N1(C(C(=Cc2ccccn2)C)=O)CCC(CNC(C2CCOC2)=O)C(F)(F)CC1 72146,c1(C(=O)NCCCCCCNC(c2cc(Cl)nnc2O)=O)ccc2[nH]ccc2c1 72147,C(=O)(C#CC(C)C)NCC1(CC(=O)N(C(CC)CC)CC(C)C)CC1 72148,c1(C(N2C(C)CC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)cc(C)nc(Cl)c1N 72149,Cn1cc(Br)nc1CN1CCSCC1C(=O)Nc1ccsc1C#N 72150,C(=O)(C(CO)C(F)(F)F)N1CC(CNC(=O)C(F)n2cccn2)OCC1 72151,c1(N2CCC(C)(CC)C2)nc(=N)nc(N2CCC(CCOC)C2)[nH]1 72152,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C#C)(C(N2CCOC(CC(N)=O)C2)=O)C1 72153,N(C1CCc2ccc(Cl)cc21)S(CCCC)(=O)=O.c12cc(ncn1)N2 72154,c1(CNC(=O)NC(c2ccccc2Cl)CO)ccc([N+](=O)[O-])s1 72155,c1(CN2CCC(O)(CNC(c3c(C)cc(F)cc3)=O)CC2)cc(F)c(F)c(F)c1 72156,C1(CNC(CCC=C(C)C)=O)CN(C(=O)C(F)C(C)C)CC1C(F)(F)F 72157,c1(C(N2CC(NC(CCNC(N)=O)=O)C3(C2)CC3)=O)cccc2c[nH]nc12 72158,CC1(C)CN(CCO)CCN1C(c1ccnc(Cl)c1F)C(=O)NC1CC1 72159,C1(CN(C(=O)COC2CCOC2)C)CCN(C(=O)CCN2CCC(F)C2)CC1 72160,c1(C(N2CCCC(NC(c3cccc(Br)n3)=O)CC2)=O)c(Cl)cc(F)cc1Cl 72161,C1CCC(C)C(=O)N2CC(C2)O1.c1(CC)cc(OCCN(C)C)on1 72162,C1(NC(c2c(C)n(C(C)C)nc2)=O)CN(C(=O)C(C)C)CCC12CCC2 72163,N1(C(C(CC)C)=O)CC(C(=O)NC)C(n2cc(-c3cn(C)nc3C(N)=O)nn2)C1 72164,N1(C(=O)CC2CCCCO2)CCN(C(=O)CCCc2ccncc2)CC12CCC2 72165,C(=O)(C(C)(C)CCC(=O)OC(C)(C)C)NCCN(C(C(CC)CNC(=O)OC)=O)C 72166,c1(NCC2CC(NC(c3cc(C)n(C(C)C)c3C)=O)C2)ncc2ccnc-2[nH]1 72167,c1(C(=O)NCCN(CCCN(C)C)C(c2cc(F)n[nH]2)=O)c[nH]nc1S(N)(=O)=O 72168,N1(C(C(COC)N(C)C)=O)CC2CN(C(=O)CC(COC)C3CCC3)CC2C1 72169,c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)O)C)c[nH]c2c(Br)cccc12 72170,CCCCC(=O)NNC(=O)C(C)n1cc(N(C)C(c2ccccc2F)=O)nn1 72171,CC(CC(=O)N1CCCC1(C(N1CCCC1)=O)CO)C(F)(F)F.C1(O)CCC(C)(C)CC1 72172,C1(CNC(c2n(C)cnc2)=O)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC1(F)F 72173,CCN=c1[nH]c(C(=O)NCC(C2CC2)N(C)C(C)=O)cs1.c12nnnn1C2 72174,c1(CNC(CC=C)=O)ccnc(C(=O)NCC2C=CCCC2)c1 72175,CC1C(NC(c2nccc(C(F)(F)F)n2)=O)CCCN1C(C1CCCC12CCC2)=O 72176,C1(C(N(CCC)C)=O)CN(C(=O)CCSC(C)C)CC12CC2 72177,CC1CCC(NC(=O)CN2CC(=O)NC2=O)CN1CCCOCc1ccccc1 72178,C1(NC(Cc2cccc(C)c2)=O)CC(F)CN(C(c2cn(C(C)C)nc2C)=O)C1 72179,CCC1=NOC(C(=O)NCCCCNC(=O)C=CCn2cncn2)C1 72180,c1(CC)cc(Cl)cc2cc(C(=O)OCC3(CS(C)(=O)=O)CCOCC3)oc12 72181,c1(C(=O)NCC(C)CN(C(=O)CCCCC#N)C)ccc2c(c1)CCS2(=O)=O 72182,CC(CC(C)(C)NC(=O)Cc1cc[nH]c1)NC(C1C2CC3C(C2)C13)=O 72183,N1(C(CS(CC)=O)=O)CC2CC1CN(C(C1(c3cccc(OC)c3)CC1)=O)C2 72184,C1(CCNC(C(C=C)C)=O)CCN(C(C23CCOC(C)(C2)C3)=O)CCC1(F)F 72185,C1(CNC(c2scc(OC)c2)=O)CN(C(=O)CCCCF)CCC1C 72186,c1(C(=O)NCc2occ(C(=O)NCCCCCCC)c2)cn2c(n1)CCC2 72187,C1(C(=O)NC(CC(C)C)C)CCN(C(c2ccc(F)cc2)=O)C1(C)C 72188,C=CCCCCCC(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)s1)C 72189,N1(C(C(C)C)=O)CCC2CCN(C(c3cn(C)nc3-c3cccnc3)=O)C2C1 72190,C(=O)(C(C)(C)CC(=O)OC)NC(CC)CCC(=O)NCCc1cccnc1 72191,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(F)o2)=O)sc2ccccc2c1Cl 72192,CCC(C(=O)NCCCN(C(=O)CC1(CO)CC1)C)C(F)(F)F 72193,CC1OC(C)CC1C(N1CC(CC(C)NC(=O)CCC2CCOC2)C1)=O 72194,N1(c2cc(COC(C)C)ncn2)CCN(C(C2CCC(C(N)=O)O2)=O)CC1(C)C 72195,c1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CC)c[nH]c2cccc([N+](=O)[O-])c12 72196,CC(O)C1C(=O)NC2(C)CC(C2)NC(=O)C(=O)N1.C1(C(=O)NC)CC(O)C1 72197,C(=O)(C1CCCc2cncn21)NC(C)(CNC(C1CCCC1)=O)C1CC1 72198,C(CN=c1ccnc(N2CCC3(C)CCCC3C2)[nH]1)OC(C)C.C(C)NC=O 72199,N1(C(C2CCCC2Cc2ccccc2)C)CC(=O)Nc2ccccc21 72200,C1(C(=O)NCC2(C)CCN(C(C=CCOC)=O)CC2)COc2ccccc2O1 72201,N1(C(C(C)c2ccsn2)=O)CC2(CCN(C(c3ccc(=O)n(C)n3)=O)CC2)C1 72202,c1(CC)cc(F)c(C(=O)NCC2CC2NC(c2[nH]ccc2OC)=O)cc1F 72203,N1(C(c2n(C)cc(C#N)c2)=O)CCCC(C2CN(C(C3CC34CC(O)C4)=O)C2)C1 72204,C1(CN(C)C(C2(C3CCCN3C(C3CCC3)=O)CC2)=O)CCc2c[nH]nc2C1 72205,N1(C(C=Cc2scc(C)n2)=O)CCN(C(=O)CCC2CCOC2)CC2(CC2)C1 72206,N1(CCSC(C)(C)C)CC2CCCN(C(=O)COc3cccnc3)C2C1 72207,C(=O)(C(C(C)(C)C)C1CC1)N(C)CCn1cc(CCN2CCSCC2)nn1.N(C)C 72208,C1(NC(c2ncc(C)s2)=O)CCN(C(=O)C(C)(C)C)CC1 72209,c1(C(N2C3C(NC(C4(CN(C)C)CC4)=O)C(C3)C2)=O)cccc2occc12 72210,N(C(=NCC1CC(C)(C)C1)NCC1CC1)C(C)C1CC1.c12cn(C)nc1C2 72211,c1(-n2cc(C(=O)NC3CCC3CNC(C3CC3(F)F)=O)nc2)cccc(Cl)c1 72212,S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1C(CNC(c2ccc3nn[nH]c3n2)=O)CC1 72213,N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(C2CC(C)CC(C)C2)=O)C12CCCC2 72214,C(CCN(C)C)(C(=O)O)NC(C1N(C(C)=O)CC1)=O 72215,N1(C(C(C)Cc2cnc[nH]2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1C1CC1 72216,c1(C(=O)NCC2CCN(C(C(C)(C)C3CCOC3)=O)C2)cncc(P(C)(C)=O)c1 72217,CC1=NOC(C)(C(=O)NC2CCC(CCNC(=O)CCC=CBr)C2)C1 72218,c1(NC(=O)NCCc2cnc(C3C(C)C3)s2)cncc(Cl)n1 72219,C(C#CCNC(=O)Cc1cn[nH]c1)NC(COC1C(C(N)=O)C1)=O 72220,N1(C(C2CC(CNC(c3nnn(C)c3N)=O)OC2)=O)CCC(N=[N+]=[N-])C1 72221,C1(C2CN(C(c3cc4n(n3)CCO4)=O)C2)(NC(c2cc(OC)ncc2)=O)CC1 72222,C1(C(C)(C)CNC(=O)Cc2nnn(CCl)n2)CN(C(=O)CN2CC3CC3C2)CCO1 72223,N12CC(N(C(=O)C3CC3)C(C)(C)C1)C(=O)NC(CC#C)C2=O.OCC 72224,c1(-c2nc(C)sc2)ccc(NC(C)(C)CN2CCN(C(=O)C(Cl)=CCl)CC2)cc1 72225,N1(CCOCCOC)CC(NC(c2c(C(F)(F)F)n[nH]c2C)=O)CCC1C 72226,C1(C(=O)NC)C2CCN(C(=O)C(C)CCc3ccc(F)cc3)CC12 72227,C1(C(N2CC3C(NC(CCCCN(C(C)=O)C)=O)C3C2)=O)C(C)(C)OC1(C)C 72228,c1(C(=O)NCC(CNC(CSC(C)C)=O)(C)F)cc(F)cnc1O 72229,CC1OCCOC1C(=O)N(C1CCC(NC(=O)C(c2cncn2C)O)CC1)C 72230,C(C)(CCC(=O)N1CCCC1C(C)NC(C12CC(CCO1)C2)=O)OC 72231,N1(C(C2CC(Oc3ccccc3)C2)=O)CC2ON=C(C(F)F)C2C1 72232,CCC(C)C(C(=O)NCCCCCCNC(=O)CSC)NC(=O)CN(C)S(N)(=O)=O 72233,CCC(CC)(CO)C(=O)NCC1(O)CCCN(C(c2ccc(F)c(O)c2)=O)C1 72234,Cc1nccc(C(=O)NCc2ocnc2C(=O)NC(C)C(N)=O)c1N 72235,N1(C(C2(C)CC=CCC2)=O)CC2=C(C1)CN(C(=O)CCOCC1CC1)C2 72236,C(CC(C(=O)NC1(C)CC(O)C1)NC(=O)C(F)C(C)C)OC 72237,C1(NC(=O)NCc2ccc(OC)c(OCCO)c2)CCN2C(=O)NCC12 72238,c1(C(=O)NC2(CCO)CN(C(C=C(C)c3ccsc3)=O)C2)cc2scnc2[nH]1 72239,C1(C(=O)NC(C(=O)OCC)CC)C2CCC(C2)N1C(C1(C)CC1(C)C)=O 72240,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72241,CC1(C)OC1C(=O)NC(CCC1CC1)c1nn[nH]n1 72242,CS(=O)c1ccc(C(=O)NCCC2CCCN2C(=O)Cc2ccc(Cl)cn2)cc1 72243,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72244,CCC(CC(=O)N1CCC(NC(C23CC(CO)(C2)C3)=O)C1C)C1CCC1 72245,C1(N(CCCC)C)CCN(C(C2(C(=O)NC)CCC2)=O)CC1.C1(=O)CN1 72246,C(=O)(CCC1=CCCCC1)N1CCN(C(CCCC#CC)=O)CC1CC(F)(F)F 72247,c1(CC(=O)NCC(C)NC(=O)CCc2ccc(Cl)nc2)cccc(F)c1 72248,C1(NC(=O)CC2CCCCC2)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72249,c1(-n2cc(C(=O)NC(C(C)NC(CNC(=O)OCC)=O)C)nn2)ccccc1C 72250,C(c1cn(C2CCC(CCCNC(c3cncc(C(C)C)c3)=O)CC2)nn1)=CC 72251,C1(COC)CCC(C)N1C(C1CCCN1C(c1cc(O)nn1C)=O)=O 72252,N1(C(C(OC)OC)=O)CCCC(CCNC(=O)CCCc2cccc(Cl)c2)C1 72253,C1(NC(Cc2cccc(CC)c2)=O)CN(C(c2c[nH]c(=N)s2)=O)C2CCCCC12 72254,C(C1CCCCCC1)=CC(=O)N(CCCCN(C(C1CCC(OC)C1)=O)C)C 72255,N1(C(C(CC)OCc2ccccc2F)=O)CCC2(C1)CN(c1ccnc(CO)n1)C2 72256,C(=O)(CC(C)C(=O)OC)NCCC1(O)CCN(C(C2(OCC)CCOCC2)=O)C1 72257,C1(C2CN(C(=O)C(C)Cn3ccnc3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72258,C1(CNC(C(F)=CC)=O)CCN(C(=O)CNC(=O)CCC(C)C)C(C)C1 72259,c1(C(=O)NC2(CCCNC(CCC(=O)OCC)=O)CC2)cnc(C)cc1Cl 72260,Cc1nn(C)cc1S(=O)(=O)NC(=O)CN1CCN(Cc2cc(Br)ccn2)CC1=O 72261,C1(NC(c2c(C)sc(Br)c2)=O)CC2CC1CN2C(=O)C(N)=O 72262,Cc1ncnc(O)c1C(=O)NC1(CO)CN(C(C2CCC3(CCC3)O2)=O)C1 72263,C(CN=C(NCc1ccc(C(=O)OC)nc1)NCC)N1C(C)(COCC)COC1 72264,C(C)(C)(C(C)CC(=O)NC(C)Cc1nncn1C)NC(c1ccc(C)nc1O)=O 72265,c1(C(=O)NCC2CC(C(=O)NCC3(OC)CC=CC3)C2)nc(C)sc1C 72266,C(=O)(C(=O)N=S(C)(C)=O)N1CCN(C(c2c(C)cc(CC3CC3)o2)=O)CC1C(F)F 72267,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72268,N1(C(C(C=C)O)=O)CCC(F)(F)C(CNC(c2cc(-c3ccco3)n(C)n2)=O)C1 72269,c1(NC(c2n(CC)nnn2)c2cnc(-c3cccnc3)s2)cc(C)nc(C)c1 72270,C1(C(=O)NC(COC)C)CC2CN(C(c3ncn4ccccc34)=O)CC2C1 72271,C(C1CCCN1C(c1coc(SC)c1)=O)=CC(=O)N(C)Cc1ccco1 72272,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72273,S(=O)(=O)(C1(c2ccccc2F)CC1)NC(c1nc(CC)sc1)C 72274,Cc1c(C(=O)NCc2ncc(C(N3CC(C)(F)C3)=O)cn2)c[nH]c1C#N 72275,CCC(C)C(C(=O)N(CCC(=O)NCC(C)N(C)C)C)NC(N)=O 72276,c1(C(N2CCC(CNC(=O)CN3CCC(O)CC3)CC2)=O)cccc(Cl)c1Cl 72277,N1(C(C(C=C)OC)=O)CCN(C(c2cc(C(C)=O)on2)=O)CC1C 72278,N1(C(C(C)c2ccco2)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(C)CN(C)C2)C1 72279,c1(OCC)nc(Cl)cc(=NC(C)C2CCN(C(=O)CCS(C)=O)C2)[nH]1 72280,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CC)c2)C1 72281,C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)CC12CCC2 72282,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)Cn2ncc(O)nc2=O)C(O)C1 72283,C1(C(=O)NCC(C)C(=O)N(CC(O)CN(C)C)C)CNC(=O)CC1C 72284,c1(C(N2C3(CN(C(c4c(C)nn(C)c4)=O)C3)CC2)=O)ccc([N+](=O)[O-])c(F)c1 72285,n1(CCC(=O)NC2C=CCN(C(CSCC#C)=O)C2)nc(O)c2ccccc12 72286,C1(C(=O)NCC2(CCO)CCC2)CC2CCCC2N1C(=O)C1=COCCC1 72287,N1(C(CCC=C)=O)CCC(SC(=O)Nc2cncc(C3(C)N=N3)c2)CC1 72288,N1(C(c2cncc(C)c2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72289,C(=O)(CCCC(=O)NCC1CN(C(=O)CC2CCCCN2C(C)C)CCO1)OC 72290,N1(C(c2nc(C)n(-c3ccccc3)n2)=O)CC2CC1CN(C(C1(F)CC1)=O)C2 72291,C(=O)(CS(N)(=O)=O)NCCC1CC(C(N2C(C(C)(C)C)CC2)=O)C1 72292,N1(C(CC(C)C2CCCO2)=O)CCC(N(C(=O)Cc2cnn(C)c2)CC2CC2)CC1 72293,C(C(CC)(CC)C(N)=O)NC(C1C(CNC(CCC=C=C)=O)CCC1)=O 72294,N1(C(Cc2c(S(C)(=O)=O)cccc2)=O)CCCn2nc(C(=O)O)cc2C1 72295,c1(CC2COC3(CCNCC3)C2)cc(NNC(=O)OC)ncn1 72296,CCCC(CNC(=O)C=CC(F)(F)F)C(=O)N(CCCO)CCN(C)C 72297,n1(CCSCC)nc(-c2ncccn2)nc1CC1CC(OCC)C1 72298,CCC(C)C(=O)C(=O)NCCN(C(C1CCCC1C)=O)C1CC1 72299,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1coc(C3CCOCC3)n1)=O)C2 72300,Cc1cc(OCCC(=O)NCC(C2CCCC2)NC(=O)C(=O)C2CC2)cc(C)c1 72301,c1(C(=O)NC2C(NC(C3(C)CNC(=O)C3)=O)COCC2)ncc2ccccn12 72302,C(=O)(C1=CC(O)C(NC(c2ccoc2C2CC2)=O)C1)NC1(CO)CC(OC)C1 72303,c1(OC)ccc(NC(C2CCC(CNC(c3ccccc3Cl)=O)CC2)=O)cc1 72304,C1(C(N(C)CC2OCCN(C(CC(C)O)=O)C2)=O)CCCCN(C)C1=O 72305,C1(C(=O)NC(CNC(c2c(SC)csc2)=O)C2CC2)CCCCCCC1 72306,c1(NC2CC2)cc(Br)cnc1I.CC(O)C1(CO)CN1 72307,C1(NC(CC=C)=O)CC2(CCN(C(c3cc4sccc4cn3)=O)CC2)C1 72308,N1(C(C(C)=CC)=O)CCCC1CNC(c1nc[nH]n1)=O 72309,N1(C(C2(C)CNC(=O)C2)=O)CC(C2CN(C(c3nccc(Cl)c3F)=O)C2)C1 72310,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)N(C(C)C(C)(C)O)C 72311,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72312,C(=O)(CC(CC(C)C)NC(=O)CCn1cnc(=N)[nH]1)Nc1cn(CC)nc1 72313,N1(Cc2ccc(C(N)=O)nc2)CC(C2CC2)C(F)(CO)C1 72314,C1(C(N2CC(NC(c3c(C(C)C)cccc3)=O)C(O)C2)=O)CCN(C)S1(=O)=O 72315,C1(N(C(CSCCC)=O)C)CCCN(C(=O)CN2CCCC2CSC)CC1 72316,c1(C(=O)NC2(C3CCN(C(COC)C)C3)CC2)ccc2c(c1)NC(=O)CN2C 72317,C=C(C)C(C)(C)C(=O)NC1CCCC(CNC(c2ccc(C(=O)CC)cc2)=O)C1 72318,C1(CNC(C2C(C)=C2)=O)CN(C(C2(C)CC(F)C2)=O)CC12CCC2 72319,C1(NC(C2CC2F)=O)CCNCC12CC2.c1(-c2ccccc2)cccc(-n2cncn2)n1 72320,c1(CCC)nsc(N(CCCCN(C(=O)C(CC2CCOCC2)OC)C)C)n1 72321,Cc1cnc(C(=O)N(C2CC(NC(c3cnc(C)[nH]c3=N)=O)C2)C)c(C)c1 72322,C1(CC(=O)N(CCCCN(C(=O)Cc2cnco2)C)C)OCCC1(C)C 72323,S(=O)(=O)(c1cccc(C(=O)OC)c1)N(C(CC)C(C)O)Cc1ncccn1 72324,c1(C(=O)NC2CC3(CN(C(CC=CC)=O)C3)C2)cc([N+](=O)[O-])ccn1 72325,N1(C(c2n(C)nc(Br)c2)=O)CCOCC(NC(C2(F)CCCC2)=O)C1 72326,C1(CNC(COCc2nnc(C)s2)=O)CNC(=O)CN1C(C1CN(C)CCO1)=O 72327,CC(C)C(C)C(CNC(C12CC(C)(CO1)C2)=O)NC(=O)CCCc1cnn[nH]1 72328,C(=O)(C(C)(C(=O)OC)C(C)OC(=O)Cc1cn(C)nc1C(F)(F)F)OC 72329,c1(C(CC)OC(=O)C=Cc2cnc(-c3ccccc3Cl)s2)ccc(OC)c(OC)c1 72330,c1(CC(C)C)ccc2c(N)c(NC(c3cncc(-c4nncn4C)c3)=O)sc2n1 72331,N(C1COc2cc(F)cc(C)c21)C(=O)Nc1ccc(-c2nc(C)sc2)cc1N(C)C 72332,C=CCCC(C(=O)NC1CCCN(CC2CCC2)C1)CC 72333,N1(C(c2nc(C3(C)CC3)on2)=O)CCCC(n2cc(C(C)(C)F)nn2)CC1 72334,c1(C(C2(C)CSC2)NC(COC)(C)C2CCC2)nnnn1Cc1ccccc1 72335,CC1C(C)N(C(C23CC(CO)(C2)C3)=O)CCN1C(=O)Cc1cnn(C)c1 72336,C1(C#N)(C(N2C(CN(C(C(CSC)O)=O)C)CCC2)=O)CCCC1 72337,c1(C(N(C(C)CCNC(c2cnc(N)c(O)c2)=O)C)=O)cnn2ccccc12 72338,c1(C(=O)NC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72339,C(=O)(C(C)(C)CCC#N)NC(C1COCC1c1ccccc1)C 72340,c1(N2C(c3cc(C(CC)(C)C)no3)C2=O)ccc2c(c1)OCO2.C1(CO)CCC(C)C1 72341,C(=O)(C(O)CC[S+](C)C)NCCCCNC(C(C)OCC=C)=O 72342,C1(NC(c2n(C)nnc2)=O)CCCC(NC(C2CC=CCC2)=O)C1 72343,C(=O)(NN1CCCC1C(=O)NC1(C(C)(F)F)CC1)C1CC(N(C)C)C1 72344,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(C3CC(F)C3)=O)CC2)ccc1C 72345,c1(C(=O)NC2(CCNC(CCCOC)=O)CCOC2)ccnc(OC)c1 72346,N1(c2ccnc(C)n2)CCc2cc(-c3ccc([N+](=O)[O-])c(F)c3)ccc2C1 72347,c1(CCC(=O)NC2CCC(CNC(C3(C)CC3)=O)C2)cc(Cl)ccc1Cl 72348,n1(CCC(=O)NC(C(C)C)c2nc[nH]n2)cc(C(C)CC2CCC2)nn1 72349,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72350,Cc1ccc2ncc(C(N3CCCC(N(C)C(c4coc(C)n4)=O)C3)=O)n2c1 72351,c1(CC(=O)NCC2(O)CN(CC3CCCCO3)C2)cccc2c1oc1ccccc21 72352,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72353,C1(NC(c2ccc(OC)c(CO)c2)=O)CCCCCCC1NC(c1ccsc1C)=O 72354,CC12CN(C(c3ncc(Br)cn3)=O)CC1CN(C(c1ncc(Cl)cc1F)=O)C2 72355,c1(C(C)NC(=O)NCc2n[nH]c(O)n2)cccc(-c2cnn(C)c2)c1 72356,C1(NC(c2cc(OC)ns2)=O)CCCC(CC(=O)NCCF)C1 72357,c1(C(=O)NC(CCNC(C(CCCC)O)=O)C)cc(Cl)cc(F)c1N 72358,c1(CCCCC)cc(C(N2CC(CO)(NC(=O)C(C)CSC(F)(F)F)C2)=O)n[nH]1 72359,c1(C(N2C(C(C)NC(=O)CC3CC(F)C3)CCC2)=O)ncnc2c1OCCO2 72360,N1(C(c2cccc(NC)n2)=O)CCC2CC(CNC(=O)COC(F)F)CCC2C1 72361,C1(OC)CCN(C(c2ccc(C(=O)OC)[nH]2)=O)CC1F.C1(F)(F)C(=O)NC12CCC2 72362,c1(C(N(CCC(=O)NCCC(=C)C)CCCO)=O)cncc(S(C)(=O)=O)c1 72363,c1(C(=O)NCC2N(C(C3CCC(C)(C)CO3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] 72364,c1(SCCC(=O)NC2CC(CNC(C3CCC3c3nc[nH]n3)=O)C2)ccccc1 72365,CC(C)CCCCCC(=O)NCC1C2CC1N(C(c1coc(Cl)n1)=O)C2 72366,C(=O)(CCCCCCBr)N1CCC(F)(C(=O)Nc2ccc(SC)cc2)C1 72367,c12ccc(cc1F)-c1cn(nn1)CCC(=O)NC2.C1(CC)CC(N(C)C)CCO1 72368,c1(C(c2n(C(C(=O)OC)C)nnn2)NCc2c(C)nsc2C)c(Cl)nc(Cl)n1C 72369,c1(CC2(C(=O)NC3CC(F)(CNC(c4cocn4)=O)C3)CC2)ccccc1 72370,CC1CN(C(=O)CC(C)CN(C)C)CCCN1C(=O)CCn1cccc1 72371,c1(OC)cccc(Cl)c1CC(N1CCC(F)(CC2CCCO2)C1)=O 72372,N1(C(C2(CC=C)CCC2)=O)CCCC(CC(=O)NCC2(N)CC2)C1.N(C)(C)C 72373,C(C(COC)C(=O)NCCN(C)C(c1ccc(CC#N)cc1)=O)OC 72374,c1(C(c2nnnn2CC(F)F)N(C(=O)COC2CCC2)CC=C)ncc(C)s1 72375,c1(NCC2OCc3c(ccc(OC)c3)C2)nc2c(c(=NCCCP(C)(C)=O)[nH]1)COC2 72376,c1(OCC)cccc(C(N2CC(O)CC2C(N2CCNC(C(N)=O)C2)=O)=O)c1 72377,C1(NC(CSSC)=O)CCN(C(=O)Cc2csc(NC=O)n2)CCC1CO 72378,c1(C(C)NCc2nnn(-c3ccccc3)n2)cccnc1F 72379,c1(OCC)cccc(OCC(N2CC(C)(NC(C3(C)CC3Br)=O)C2)=O)c1 72380,c1(C(C)C)ncc(NC(=O)C(C)C(C)NC(=O)Cc2ccoc2)cn1 72381,c1(CC(=O)NCC2(F)CC(NC(CCCOCC)=O)C2)ccc(CC2CC2)cc1 72382,c1(CN2CCC(N(C)C(C3(c4ccncc4)CC3)=O)C2)cccc(I)c1F 72383,C(CC)(CCCC(=O)N1CCC(F)C1)NC(c1cn(CC=C)nn1)=O 72384,CCCCCC(C)CC(=O)N1CCC(N(C(=O)CCn2cccn2)CC)CC1 72385,C(=O)(CC(C)CC(C)(C)C)N1C(C(=O)NC(C)CO)CSC1 72386,C(=O)(CC(F)(F)Cl)NCC(C)(C)CNC(C1(C(=O)Nc2ccc(F)cc2)CCC1)=O 72387,CC1Cc2cc(C(=O)NC3COCC3NC(=O)Cn3cncn3)ccc2O1 72388,C#Cc1nccnc1NC(=O)NC1CCC(COCCC)CC1 72389,N1(C(c2c(CC)csc2)=O)CC(NC(c2cc(C)cc(C)n2)=O)CC(O)C1 72390,N1(C(COCCCC#C)=O)CC2CCC(CNC(=O)C(O)CC(C)C)(C2)C1 72391,CC(Cl)(Cl)C(=O)N1CC(C(N)=O)(CNC(c2ccc(C(N)=O)o2)=O)C1 72392,C1(CNC(C23N(C(c4cc(C)ncc4)=O)CC(C2)C3)=O)OC(=O)CC1(C)C 72393,c1(C(=O)NC2(c3cn(C)nn3)CCCC2)ccc(Br)cc1Cn1cccn1 72394,c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)ccn3)=O)C(C)C2)c(F)c1Cl 72395,C1(C(N2CCN3CCCC3C2)=O)C2CC(O)C(C2)N1C(=O)COCC1CC1 72396,N1(CCNC(C(c2cccc(Cl)c2)(C)C)=O)CCC(NC(c2ccncc2)=O)CC1 72397,N1(C(=O)NCc2cc(Cl)ccc2F)C2CCCC1CC(F)(F)C2 72398,c1(C(N2CC(C(=O)OC)C2)=O)cnc(CNC(=O)CC2CCC(=O)C2)nc1 72399,N1(C(C(C)C2CCOC2)=O)CCN(CC2CN(C(=O)COC3CC(F)(F)C3)C2)CC1 72400,c1(C(N2CCC(CCC(=O)NCc3cncc(Cl)c3)C2)=O)c[nH]nc1[N+](=O)[O-] 72401,CCCC(C(=O)NC1CCCC1F)NC(C1CC1C(C)(F)F)=O 72402,c1(OC)ccc(CC(N2CC(O)(C(C)NC(=O)C(c3cncnc3)C)C2)=O)cc1 72403,C1(C(=O)NCCCCN(C(=O)COCC(C)(C)C)C)CCCCN1S(C)(=O)=O 72404,c1(C(=O)NC2CCCC(CCNC(C(=O)NCC)=O)C2)c(C)cnnc1O 72405,c1(C(N2CCCC(C(C)NC(c3c(C)sc(Cl)n3)=O)C2)=O)ccc2n[nH]cc2n1 72406,C(=O)(CCCC(C)(C)C)N1CCC(n2cc(SC)nn2)C1.C1(C(=O)NC)CC1 72407,c1(CNC(=NCC=C)NCc2ccsc2)ccc(S(=O)(=O)N2CCCC2)cc1 72408,C1(CN(C(C2C(C)=C2)=O)C)CCCN1C(C1CCC(=O)N1)=O 72409,C12(CNC(C3CC4(CCC4)C3)=O)CCCC1CCN2C(c1cc2c(s1)CCC2)=O 72410,C(=O)(CC(C)(C)C1CC1)NCCCC(C)NC(=O)CC1C=NN(C)C1=O 72411,CC1CCCn2cc(C(N3CCCC4(NC(=O)CC5CC(F)C5)CC4C3)=O)nc21 72412,c1(C(N2CC3C(CNC(c4c(CC)onc4C)=O)(C3)C2)=O)ccc(F)cc1O 72413,C1(CC(F)(F)F)CCN(C2=NCC3(CC3)CN2)C1.C1(CC2CC2)CCCOC1 72414,c1(CC(=O)NCC2N(C(CC(C)O)=O)CC2)ncncc1Cl 72415,C1(OCC)CC(OOC(=O)C=CC2CCCC2)C1(C)C.c12cncc(c1)C2O 72416,C#CCCCC(C)C(=O)N1CCC2(CC2NC(=O)C(c2ccccc2F)C)C1 72417,C(C(F)(F)C(C)(C)O)NC(CC1(CNC(C(C)O)=O)CC1)=O 72418,CCC(C)CC(C(=O)NCCn1cccnc1=O)NC(=O)CCc1cncn1C 72419,CS(=O)(=O)c1ccc(C=CC(=O)NCC2COCCN2C(=O)Cc2ccsn2)o1 72420,Cc1ccc(C(N2CCCC(N(C)C(c3cc(N)ccc3C)=O)C2)=O)c(F)c1 72421,N1(CCC2CCC(CNC(C)=O)CC2)C2CCC1COC2 72422,C1(CNC(c2c(C)nco2)=O)C2CN(C(=O)Cc3coc(C(F)(F)F)c3)CC12 72423,N1(C(=O)C2=CCCCC2)CCC2CCCC12C(=O)NC1CCCC1(F)F 72424,C1(C(=O)NC(c2ccc(C)o2)COC)C(C2CC2)CCN1C(=O)CCCC(C)=O 72425,C(=O)(CC(CC1CC1)NC(=O)CC(O)CN(C)C)N1CC(N(C)CC)C1 72426,N1(C(c2cnc(OC)s2)=O)CC(C2CCN(C(=O)COc3ccccc3O)C2)C1 72427,N(C1CN(C)Cc2ccccc21)C(c1ccc(-n2cc(C(=O)NC)nn2)cc1)=O 72428,CC1(C)CCCC1C(=O)NCC(O)CNC(C1(c2cccc(F)c2)CC1)=O 72429,N1(C(C(C(C)C)O)=O)CC(NC(C23CC(c4ccccc4)(C2)C3)=O)CCC1C 72430,c1(C(N2C(C(=O)NCC3C(C(=O)OC)C3)CNC(=O)C2)=O)cccc2cncn12 72431,c1(C(N2C(C(C)NC(C(CC)OCC)=O)CCC2)=O)cc(O)c2sccc2c1 72432,O=C1CCC(CCC(=O)NCC(O)CNC(=O)CCc2nc(C3CC3)no2)=NN1 72433,C1(CNC(C(=O)Nc2cc(OC)ns2)=O)CCCN(S(C)(=O)=O)CCO1 72434,C1(OC)CC(NC(=O)CCn2ccnc2)CN(C(C2(C#N)CCCC2)=O)C1 72435,C1(NC(c2ncc(OCC)nc2)=O)CC2(CCN(C(C3CC3CC)=O)C2)C1 72436,c1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)cc(Br)cc(C)c1F 72437,C1(CC(N2CC=C(CNC(C3(CN(C)C)CC3)=O)CC2)=O)CCCC2(CC2)C1 72438,C12(NC(c3c(C)nncc3)=O)CCC(CN(C(=O)C(C)OCCN(C)C)C1)C2 72439,C1(C(N(CC(C)NC(c2cccc(C3(C#N)CC3)c2)=O)C)=O)CCCCC1(C)C 72440,C1(NC(COc2cccc(CC)c2)=O)CCN(C(=O)C(C)c2ccco2)CC1O 72441,N1(C(c2cc(N(CCC)C)ncc2)=O)CC(C(=O)NC)CC(F)(F)C1 72442,CCC(O)CCNC(=O)COc1ccsn1 72443,C1(NC(=O)CC2CCOC2=O)CC12CCN(C(=O)C1=C(Cl)CC1)C2 72444,N1(C(CCSC)=O)CCCC2(NC(c3coc(C#N)c3)=O)CC2C1 72445,c1(C(N2CCC(C)C2)=O)c(CNC(c2cc(Cl)cs2)=O)cnn1C 72446,c1(CC(=O)NC23CC(CNC(C4CCC(CC)C4)=O)(C2)C3)nnc2ccccn12 72447,c1(CNC2C(C)CN(C(c3cc(Cl)ncc3F)=O)C2)cccc(F)c1C#N 72448,C(C(C)N=c1[nH]c(Cl)nc2c1SCC2)(C1CC1)NC(c1n(CCC)ncc1)=O 72449,C1(C(=O)NC(c2ccccc2)CC2CC2)CCCCN1Cc1ccc(I)cc1 72450,C1(=O)C2=CCC(C2)N1.C(CC(COC)NC(=O)CC1OCCCO1)OC 72451,C(N1CCOc2ccccc21)n1ncc(-c2nc(C)sc2C)c1 72452,c1(C(=O)Nc2ncc[nH]2)cn2c(n1)CN(C(c1c(F)c(Cl)cc(Cl)c1F)=O)CC2 72453,c1(C(=O)NC(C2CCN(CCC3(C#N)CCCC3)C2)(C)C)ccc2cccnc2n1 72454,N1(CC(=O)N(C(C)CNC(C2CC23CCOC3)=O)C)CCS(=O)(=O)CC1 72455,N1(C(c2cnc(C)n2C)=O)CCN(C(=O)CC(O)C2CCCC2)CC1C1CCC1 72456,CCC(CC)C(C)C(=O)NC(CCOCCO)C(=O)Nc1ccc(F)cc1C 72457,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(C(F)(F)F)c2)S1(=O)=O 72458,c1(C(=O)NC(C)C(CO)NC(=O)CC(Cl)Cl)ncncc1Cl 72459,C(=O)(C1=C(c2cncs2)N(CCF)C(=O)NC1c1ccc(CC)cc1)OCC 72460,O=C1CCC(OCn2cc(C3CN(C(C4CC5(CC5)CO4)=O)C3)nn2)C(=O)N1 72461,N#CC1CCCC1Cc1nc(CO)n[nH]1.c12c(cnn1CC(=O)CC)C(=O)NC2 72462,C(CCCCC(=O)Nc1c(C)nccc1)NC(=O)C(C)N(C)C 72463,C1(NC(=O)C=CC2CCCO2)CCN(C(c2cc(Br)ccc2OC(F)F)=O)CC1F 72464,Cc1nc(SC(F)F)sc1C(=O)NCCC(C)NC(=O)CC(C)N(C)C 72465,CN1CCN(C)C(C(=O)N(C)CC2(O)CCN(C(=O)C=CC(N)=O)CC2)C1 72466,c1(SCC2(NCN(C)N=O)CCC2)ccc(-c2ccncc2)nc1 72467,c1(C2C(=O)O2)ccc2c(c1)OCCO2.c1(-c2ccc(COC)s2)c[nH]ccc1=O 72468,c1(OC(C(NOC(CCC)CC)=O)C)cnc(N)c([N+](=O)[O-])c1 72469,Cc1c(C(=O)NCC2(NC(C3C(Cl)(Cl)C34CC4)=O)CCOC2)sc2ccsc12 72470,C(=O)(CCS(=O)(=O)CC(C)C)NCC1N(C(c2cc(C(C)=O)sc2)=O)CC=C1 72471,N1(C(C2(C(=O)CC)CCCC2)=O)CCCC2(C1)CN1C(CCC1)C(=O)N2.C=CC 72472,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72473,C1(C(N2CCOCC(C(C)C)C2)=O)C(C2CC2)CCN1C(=O)CC1CCOC1=O 72474,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)CCCSC)CCO2 72475,N1(C(CCC=C)=O)CCC(C(=O)NC2CN(CCC)C2)=C(F)C1 72476,O=C1NCC2(CCN(C(C34CCCCC(C(=O)O)(C3)C4)=O)CC2)N1 72477,C(=O)(C#CC(C)(C)O)NCC(=O)NCC1CC(C[Si](C)(C)C)C1 72478,c1(N2CCN(C)CC2CNC(c2ccc(O)nc2)=O)nc2ncc(Cl)cc2o1 72479,c1(CC(=O)NC2C(CNC(C(CCC)C)=O)CCCC2)sc2ccccc2c1C 72480,c1(C(=O)NC(CC)CNC(=O)C(O)C2CCCC2)ccnc(N2CCCC2)n1 72481,N1(C(c2cnc(C)c(Cl)c2Cl)=O)CCn2cccc2C1c1ccccn1 72482,C1(CNC(C(C)OCC#C)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1(F)F 72483,C(C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnc[nH]1)(C(C)C)SC 72484,c1(SCC)cccc(C)c1C(=O)NCC1CC(NC(c2ccc(C#N)cc2)=O)C1 72485,C=C(CNC(=O)CC(C)CNC(C1CC1(C#N)CCC)=O)c1ccccc1F 72486,C(C(C)(O)C(=O)N1CCC1(C)CC(=O)NCc1nnnn1C)OC 72487,C1(C(=O)NC(c2ncc[nH]2)C)CCCCCN1C(C1CC2(CCC2=O)C1)=O 72488,C1(C(=O)NC2CC3(C(NC(CC4CC(=C)C4)=O)C3)C2)(COC)CC(C)(C)C1 72489,C1(CNC(C2CC(CC)C2)=O)CC(O)(CNC(=O)CSS(C)(=O)=O)C1 72490,C(=O)(C=CS(F)(F)(F)(F)F)NC(CNC(c1c(C)[nH]c(C)c1C)=O)CC(C)C 72491,C(C(CCNC(C1CC(CC2CC2)C1)=O)OC)OC.C12CC(C)N1C2=O 72492,Cn1ccc2ccc(C(=O)NCC3CN(C(C4(C)CCOC4)=O)CC3(C)C)cc12 72493,N1(C(C(C(=O)OC)C)=O)CCN(C(C2(O)COC2)=O)CC1c1cn[nH]c1 72494,N1(C(CCC)=O)CC(NC(c2cc(C)nc(N(C)C)n2)=O)CCC1C 72495,C(C(C)(CCO)NC(=O)CC1C2CN(C(c3ccoc3)=O)CC12)OC 72496,c1(C(N2C(CC3(C(=O)NCC)COC3)CC2)=O)ccc(OC)c(OC)c1Cl 72497,c1(C(N2CCC(CCNC(c3cnc(OC)nc3)=O)C2)=O)ccsc1S(C)(=O)=O 72498,C1(CC)(NC(=O)CCCc2ccncc2)CCN(C(=O)C(C)(C)C2CCC2)CC1 72499,c1(C(=O)NCc2cccc(-n3cc(CCO)nn3)c2)cc(O)ncc1Br 72500,C1(NC(C(CC)NC(N)=O)=O)CCN(C(c2ccc(N)c(F)n2)=O)C12CCC2 72501,C1(NC(c2sccc2F)=O)CCC(O)CN(C(=O)Cc2ccc(Br)cc2)C1 72502,c1(CC(=O)NC2CC(CNC(C3CC=CC3)=O)C2)ccc(OCC(F)F)cc1 72503,c1(N2CCN(C(c3cc(-c4ncc(Cl)s4)ccc3F)=O)CC2)cc2ncnn2cn1 72504,c1(C(N2C(C(C)NC(C3(SC)CCC3)=O)CCCC2)=O)nccc2ccn(C)c12 72505,C(=O)(C1CCc2c[nH]nc21)N1CC2C(CNC)C2C1.C1(C#N)(C=O)CC(F)(F)C1 72506,c1(C(=O)NCC2C(C)CCCN2C(C2CCS(=O)(=O)C2)=O)cnn2c1CCCC2 72507,c1(C(N2CCC(OC)(CNC(=O)CNC=O)C2)=O)c[nH]c2cc(F)ccc12 72508,C12(NC(c3c(N)c(F)ccc3)=O)CCCC1CN(C(=O)CCCC1CCCC1)C2 72509,c1(CNCC2(CNC(c3noc4c3CCC4)=O)CC2)c[nH]c2ncc(Cl)cc12 72510,c1(C(=O)NC2(CNC(c3cccc(C)n3)=O)CCCC2)cc(F)c(Cl)nc1Cl 72511,O=[N+]([O-])c1cc(NCCN2CCCC(C(F)F)C2)ccc1CN1CCC(O)C1 72512,C(=O)(NNC(=O)C(C)(C)CNC(C(O)CC1CC1)c1ccccc1)c1ccc(C)o1 72513,CS(=O)CCC(=O)N1CCC(CCN(C(c2ccc[nH]2)=O)C2CC2)CC1 72514,c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CCN=[N+]=[N-])CC)c[nH]c(=S)cn1 72515,c1(SC)ccccc1-n1nnnc1C(C1CC1)NC1(C(N)=O)CCC(C(C)(C)C)C1 72516,Cc1cc(C(N2CC(C)CC2C(=O)N(C(CO)CO)C)=O)nc(C)c1 72517,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(C1CN(S(C)(=O)=O)C1)C 72518,CC1(C)C(NC(c2cc[nH]n2)=O)CCN1C(=O)Cc1cccnc1Br 72519,N1(CC(=O)NC(C(=O)NCCC)C)CCC(COc2ccccc2)CCO1 72520,N1(C(COCC(=C)C)=O)CC2(CCN(C(=O)C(C3CCCO3)NC(C)=O)C2)C1 72521,N1(C(c2ncc(C)s2)C(=O)NCCCOC)CCc2c(nnn2C)C1 72522,CCC(CC)C(F)C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)C(C2CC2)C1 72523,C(=O)(CC(=O)NCCCN(C(=O)CC1(C)CC1(F)Cl)C)NCC#C 72524,N1(CCC(=O)N(C)CCNc2ccc(C3CC3(F)F)cc2)CCC(O)CC1 72525,C(=O)(C(O)C1=CCCCC1)CC(C)CNC(c1cccc(F)c1C#N)=O 72526,C1(NC(C2C(CCC)C2)=O)CCN(CCCNC(C2CCC3(CC3)C2)=O)CC1 72527,Cc1[nH]nc(C(N2CCC(O)(C(C)NC(=O)CCC3CC3)C2)=O)c1N 72528,N1(C(CC(c2c(C)nccc2)C)=O)CCN(C)CC1C(C)C 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72599,N1(C(C(C)(C)OCCC)=O)CCC(CNC(c2cnncc2O)=O)C1(C)C 72600,c1(C(N2C(CN(C(CCn3ncc(C)c3)=O)C)CCC2)=O)c(C)nsc1C 72601,C1(NC(C(C(C)C)NS(N)(=O)=O)=O)COCCN(C(c2c(Cl)cncc2Cl)=O)C1 72602,N1(C(CN(C)C2CC2)=O)CC(NC(C2CC(=O)N(C(C)(C)C)C2)=O)CC(C)(C)C1 72603,C(CC(O)C(=O)NC1CCN(CCO)CC1)N(C(=O)C(C)(C)C1CCC1)C 72604,c1(C(=O)NC2(CNC(C(CC)Br)=O)CCC2)cnc2sccn2c1=O 72605,C#Cc1ccc(C(=O)NCC2(C)CCN(C(=O)CC(C)CC)CC2)nc1 72606,S(=O)(=O)(C1CCN(C2CCOC(C)(C)C2)C1)NC 72607,C(C1CCCN1C)=CC(=O)NCCCN(C(C(C)=C1CC1)=O)C(C)C 72608,Cc1cccc(C(=O)NC(C)CC(C)NC(=O)CSCC(=O)NC(=O)CCF)c1 72609,c1(C(N2CC(CNC(C3CC(O)C3)=O)C3(CC3)C2)=O)cc(Cl)ccc1OC1CC1 72610,c1(CC(C(=O)NCC=CCNC(C2N(S(C)(=O)=O)CCC2)=O)O)ccc(Cl)cc1 72611,C1(CCNC(C2(F)C(C)C2)=O)CCN(C(c2ccns2)=O)CC1(F)F 72612,C1(O)(C(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)(F)F)CCOCC1 72613,Cc1cccc(C(CF)NC(c2cc(-c3ccncc3)[nH]n2)=O)c1 72614,c1(-c2cn(CCOC)nn2)csc2cncn12.C12CCN(C1)C(=O)N2 72615,c1(C(N2CC(NC(C(C)C3(O)CCC3)=O)C3(C2)CC3)=O)cc(F)cc(Br)c1N 72616,O=C(C1=CCCSC1)NCCN1CCN(C(=O)CSc2ccncc2)CC1 72617,C1(NC(=O)NCC(C(C)C)O)CC12CCN(C(=O)COc1cccnc1)CC2 72618,C1(NC(Cc2c(OC)cccc2)=O)CC2CC(NC(C3CC3C(C)C)=O)CC12 72619,N1(C(C=CC(C)NC(=O)CCc2nc[nH]n2)=O)CC2C=CCC(C2)C1 72620,c1(CN2C(C(N3CCC3CO)=O)CC3CC32)cc(F)c(O)c(F)c1 72621,N1(c2cc(C(C)=O)ncn2)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC2C1 72622,N1(C(C(C)OCCOC)=O)CC2OC(C)C2C1 72623,N1(C(C2CC2CC2CC2)=O)CC(n2cccc2)C1 72624,c1(COCC)ncc2c(n1)CCN(C(=O)NC(c1c(C)n[nH]c1C)NC)C2 72625,c1(C(=O)NC(CCC(C)C)C)cccc(N=c2cncc[nH]2)c1 72626,CC(C)(C#N)C(=O)NCC1CCC(NC(C2CC2C(F)(F)F)=O)C1 72627,CCCCCC(O)C(=O)N1CC2(C(N3CCC(O)C(C)(O)C3)=O)CCC1CC2 72628,CCC(CO)NCCNC(C1(Cl)CC1C(=O)O)=O 72629,c1(C(=O)NC(CNC(C=CCOC)=O)C(C)C)cnc(O)n(-c2ccccc2)c1=O 72630,N1(C(C=C(COC)C)=O)CC2CCCC2(C(=O)Nn2ccnn2)C1 72631,N1(C(c2n(C)c(C(N)=O)cn2)=O)CC23CCCCC2(C1)CN(C(C1CC1(C)C)=O)C3 72632,N1(C(c2cc(CNC(CCC=CC)=O)sc2)=O)CCC(O)(CC)CC1 72633,C1(C(=O)NCCN(C(=O)C(=O)NC)CC)CCN(c2ccccc2)C1 72634,Cc1cc(Cl)cc(C(=O)NC2C3CC2N(C(=O)COC(F)F)C3)c1O 72635,CCCCC(CNC(=O)Cc1csc(S)n1)NC(c1cc(O)no1)=O 72636,C=CCC(CC(F)F)C(=O)N1CC2CC(NC(c3cnccc3OC)=O)CC1C2 72637,N1(C(c2c(C)coc2C)=O)CCCC(C2CN(C(C3CC3(F)F)=O)C2)C1 72638,C1(COC)CN(C(C2CC(C#N)C2)=O)CCN1C(c1cc(C)ccc1Br)=O 72639,S(=O)(=O)(c1ccc(C2CC2)cc1Cl)N(CCCCC(C)(C)C)C1CCC(O)C1O 72640,C1(CNC(CCCCOC)=O)CC2CCC1N(C(c1nc(Cl)sc1Cl)=O)C2 72641,CC1CN(C(c2cc3n(n2)CCCC3)=O)CCN(C(=O)COC(C)(C)C)C1 72642,CCC(CNC(=O)C=Cc1ccsc1)(CC)NC(C1CC2CC2C1)=O 72643,c1(NC2CCCCN(CC)C2=O)nc(N2CCCN(C(C)C)CC2)nc2c1CCC2 72644,CC1CC(CCC(=O)NCc2ccccc2)C(C)N1C.c12ccccc1OCC2=O 72645,C1(COC(N2CCC(C(=O)OC)C2C)=O)CCCCCN1Cc1ccccc1 72646,c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)C)=O)c[nH]nc1Br 72647,c1(N(C)C)cc(S(=O)(=O)C(=O)NCC2(CN(C)C(C3CCC4CC34)=O)CC2)c[nH]1 72648,C1(C(=O)NCC(CCOC)NC(c2ccn(CC)c2C)=O)CCC2(CC1)CC2 72649,C=CCCCC(=O)NCC=CCC(=O)NC1CCC(C(N)=O)O1 72650,C1(NC(C)CS(C)=O)(CNC(=O)OC(C)(C)C)CC12CCC2 72651,N1(C(c2cccnc2N2CCN(C)CC2)C(=O)NCC)CCn2ncc(Cl)c2C1 72652,c1(C(=O)NCC(CN(C(=O)CSc2nccn2C)C)C)ccccc1C1CCC1 72653,Cc1nc(C(c2nnnn2C(C)(C)C)NCCN2CCOCC2)cs1 72654,c1(CN(C)C(c2nscc2Br)=O)ccccc1CNC(c1cnn[nH]1)=O 72655,n1(C(C)C)cc(C(N2CC3CC2C3CNC(=O)CS(=O)(=O)CC)=O)c(O)nc1=O 72656,c1(NC(c2cc(OC)c(OCCO)cc2)=O)ccc2oc(C)c(C)c2c1 72657,N1(C(CN(CCOC)C)=O)CCCC2(NC(C3(C(F)(F)F)CCCC3)=O)CC2C1 72658,C1(CN(C(=O)CSc2cnn(C)c2)CC)CCCCN1C(=O)C=Cc1ccco1 72659,N1(C(C2N(C(CC(COC)(C)C)=O)CC3(CC3)C2)=O)C2CCC1CC(O)C2 72660,N1(C(C(F)=CCC)=O)CC(CNC(C2CN(c3nncs3)C2)=O)C2(CCC2)C1 72661,Cn1ncc(C(=O)NCCC2(NC(C3C=CC=CC=C3)=O)CCC2)c1F 72662,C(=O)(CC(O)CNC(C1(C(C)C)CCCC1)=O)N1CCC(OC(C)C)C1 72663,Cn1c(=O)oc2c(C(=O)NC3CCN(C(=O)CCCC4CC4)CC3O)cccc12 72664,c1(C(c2nnnn2C)NCC#CC)ccnc2[nH]c(C(F)F)nc12 72665,C1(CNC(c2cc(C)nn2C)=O)CCN(C(=O)CC=C(Cl)Cl)CC1O 72666,N1(C(Cc2nc(CC)sc2)=O)CCOC(C)(CNC(c2cc(C)cs2)=O)C1 72667,c1(C(N2CCC2CNC(N)=O)C)cc(C(=O)NCc2cncn2C)no1 72668,Cc1ccc(O)c(CNC(C2(C)CCN(C(=O)Cc3cc(F)cc(Br)c3)C2)=O)c1 72669,c1(CC)[nH]c(Cl)nc(=NCC2CCCN(C(c3ccn4cncc4c3)=O)C2)c1C#N 72670,c1(C(=O)NC(C)CCNC(=O)Cc2ccccc2C(C)C)ccc(N=[N+]=[N-])cc1 72671,c12nc(O)c(cc1C)C(=O)OCC(C)C(=O)NC(C1CCCC1)C2.CC 72672,N1(C(C2CC2F)=O)CCC2OCCN(C(C3CC3c3ccc(F)cc3)=O)C2C1 72673,N1(CC)CCCC(C(N2CCC(C(=O)Nc3ccc(I)cc3)CC2)=O)C1 72674,N1(CC)CCNC(=O)C1CCO.C1C(C)CC(=O)N1.C12CC(C1)CC(=O)N2 72675,Cc1ccc(NC(=O)C(C)N(C)C2CC2)cc1I 72676,c1(C(CNC(CC)=O)C(=O)O)ccc(O)cc1 72677,c1(C(N2CC(O)(C(=O)NCCC(Cl)Cl)C2)=O)c[nH]c2nccc-2c1 72678,N1(Cc2c[nH]c3ccc(C#N)cc32)CCC2CCN(C(=O)OC(C)(C)C)CC2C1 72679,C1(CC)(CC)CC(NC(=O)CSc2cccnc2)CN1C(=O)C(F)C1CCCC1 72680,N(S(=O)(=O)N1CCC(C2COC(C)(C)O2)CC1)c1cccc(OC)c1 72681,CC1(C)CCCN(C(c2cc(C(N)=O)c[nH]2)=O)C1CNC(c1cc(O)ncn1)=O 72682,c1(OC)ccc(CC(=O)NC2CN(C(C3COC4CC3C4)=O)CC2OC)cc1O 72683,c1(OCCC)ccccc1C(N1CCC(C)(NC(c2ccc(=O)oc2)=O)C1)=O 72684,C(=O)(CC(=O)NCCOC(C)(C)CNC(=O)CCc1nccs1)N(C)C 72685,C1(C(=O)NC2CCCC(NC(CS(CC)(=O)=O)=O)C2)CCCC2(CCC2)C1 72686,c1(CC(N2CCCCC(NC(CC(CC=C)C)=O)C2)=O)cccc2ccccc12 72687,C1(C(N(C)Cc2cocn2)=O)CCCCN(C(=O)Cc2ccc(F)cn2)C1 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72705,c1(-n2c(C(=O)NC(C(=O)OCC)CC)ncc2)cccc(Cl)c1 72706,N1(C(COCCOCCN(C(=O)CC2OCCO2)C)=O)CCCC1CO 72707,N1(C(c2cn(CC(C)O)nn2)=O)CC2CCCC2(CO)C1 72708,N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(C3(O)CCSCC3)=O)CCC12 72709,c1(C(N(C(C)CNC(=O)CCc2cn[nH]c2)CC)=O)cc(Cl)n[nH]1 72710,c1(C(N2CCCC(NC(c3ncn(C)c(=O)c3)=O)CC2)=O)ccc2cnsc2c1 72711,C1(NC(C(CC(C)(C)C)F)=O)CC2CCC1CN(C(=O)CN1CCC(=O)CC1)C2 72712,C1(NC(CSC(C)C)=O)CCN(C(c2cc[nH]n2)=O)CC1C 72713,CC(CN=c1[nH]c(=NC2COC(C3CCC3)C2)[nH]c2c1CC(C)CC2)N(C)C 72714,Cc1cnc(N(C(c2cn(CC3CC3)nn2)(C)C)CC2C3CCCC23)cn1 72715,C1(CC(=O)NCC(=O)OC)CCC(NC(=O)CCc2cnoc2)CC1 72716,C1(CC(=O)NCC2CCCC23CC3)COCCN1CCN1CCCC1=O 72717,CC1CCC(NC(=O)C(c2ccccc2)O)CN1CCc1cccc(Cl)c1 72718,C1(CN(C)C(c2cc(F)n[nH]2)=O)CCCN1C(=O)CCc1nc[nH]n1 72719,c1(C(N(CC(C)NC(=O)CSCF)CC)=O)c(Br)ccc(F)c1N 72720,c1(OC)ccc(C(=O)NCC2CCC2NC(=O)CCc2cncnc2O)c(F)n1 72721,CC(C)CC(C)CC(=O)NCC1(F)CCC(NC(=O)C(c2ccc(F)cc2)=O)C1 72722,C1(C(=O)Nc2ccc(OC)c(C(F)(F)F)c2)CC12CCN(C(=O)C(F)F)CC2 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72740,c1(C(N2CCC(CNC(CSC)=O)C2(C)C)=O)ncn2c1CCCC2 72741,C1(NC(c2[nH]cc(C(N)=O)c2)=O)CCOC(C(=O)NCCC2CCCC2)C1 72742,c1(C(=O)NC(CC(C)NC(c2c(OC)c(Cl)sc2)=O)C)ccc(F)c2[nH]ccc12 72743,CC1CC(N(C2CCC2)N(CC(=O)N)C)CCO1.c1(C=O)cccc(C2CC2)c1 72744,CCCC(C)(O)C(=O)NC1CCCC(C(N2CCC(O)CC2C)=O)CC1 72745,N1CCCC(CO)(CNC(=O)COCC2CC2)C1.c1(OC)cccc(C=O)n1 72746,C1(C(=O)NC(CN(C(CN(C)CC)=O)CC)C)CC2OC(C)(C)OC2C1 72747,c1(CCC(=O)N2CC(NC(c3cnn(-c4nccs4)c3)=O)C2)cnc(O)[nH]1 72748,N1(C(C(C)Cn2cccn2)=O)CC(NC(c2c(Cl)cnn2-c2ccccc2)=O)C(O)C1 72749,c1(C(C2CC2)OC)nc(-c2cc(Br)oc2C)n(-c2ccccc2N(C)C)n1 72750,C1(C)(NC(c2ccc(Oc3ccc(Cl)cc3)nc2)=O)CCC12CCC2 72751,CC1(C(=O)NCC2CCC2NC(=O)CCCCN2CCCCC2)CCCCO1 72752,N1(Cc2ccn(C)c2)CCCCCC(C(=O)Nc2ccnc(CO)c2)C1 72753,c1(CCC)nc(CCc2cc(C)oc2C)n(-c2c(C)noc2C)n1 72754,C1(O)(CNC(C(CC)NC(C)=O)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1 72755,Cc1cccc(C(=O)N(CCC(C)NC(c2ccncc2Br)=O)C)c1N 72756,c1(C(N2CCCN(C(C3C4CC5C(C4)C35)=O)CC2)=O)coc2ccccc12 72757,c1(C(=O)NCc2cn(CC(=O)NC(C3CCCOC3)CC)nn2)cc(C)ncn1 72758,c1(C(=O)OC)cnc(N2CCCC2CCNC(=O)CSC2CCCCO2)nc1 72759,C(=O)(CCCS(N)(=O)=O)NCCC(C)N(C(Cn1nc(C)n(C)c1=O)=O)C 72760,c1(C(N2CCC(CNC(C(C)NC(C)=O)=O)C(C)C2)=O)cccc2c1CNC2=O 72761,N1(C(c2cn(CC=C)nn2)=O)CCCCCC(NC(C2(COC)CCCC2)=O)C1 72762,C1(NC(C(=O)NCCOCCOC)=O)CCC(C)N(C(=O)C(C#N)C2CC2)C1 72763,c1(CC(N2CCC(C(NC(=O)C(O)C3CCC3)C3CC3)C2)=O)ccc(Cl)c(F)c1 72764,C1(C(N2CC(CC(C)NC(C3CCCCC3O)=O)C2)=O)C2CC3CC(C2)CC1C3 72765,C1(NC(c2c(CCC)occ2)=O)CC(C)CN(C(c2ccn(CC)c2C)=O)C1 72766,N1(C(CN(C2CCCC2)C)=O)CC2CC(N(C(=O)C(=O)C(C)(C)C)C)C1C2 72767,CC(CNC(=O)Cn1cncn1)(C1CC1)NC(C1CCN1S(C)(=O)=O)=O 72768,c1(C(=O)OC(C2CCCC2)C)cc2ccc(Cl)nc2s1 72769,c1(N2CCC(N(C(=O)C(c3cnn(C)c3)O)C)C2)ncncc1Br 72770,c1(-c2nc(CCCC=C)n(CC(C)C)n2)ccc(OCCOC)c(Cl)c1 72771,CCC(CC)(CC)C(=O)N(C(COC(=N)O)C)N(c1ccc(S(N)(=O)=O)s1)C 72772,c1(OC)ccc(C(=O)COc2ccc(F)cc2)c(O)c1OC 72773,c1(C(N2CCC(CC=C)(NC(=O)CC3CCCCC3)C2)=O)nc(OC)ncc1OC 72774,c1(C(C)C)sc(Cl)nc1C(N1CC(N(C(=O)CCC2CCOCC2)C)C1)=O 72775,C(CNC(C1CC12CC2)=O)(CC(=O)NCCCF)N(C)C 72776,C1(C)(C(=O)NCC(C)(CNC(=O)C(C)=C(C)C)OC)CCC(C)C1 72777,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NCCC2CC2)CC1(C)C 72778,c1(C(=O)NC2C(NC(c3ccn(C)c(=O)c3)=O)CCCC2)c[nH]nc1S(N)(=O)=O 72779,N12CCCC(C1)C2=O.C1(CC)C(=O)N1C1CC1.C=O.N(C)(CCO)CCO 72780,c1(C(=O)NC(C)CCCNC(c2ccon2)=O)c(Cl)oc2ccccc12 72781,c1(OC)ncnc(C(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1F 72782,C(=O)(C(CO)C(C)(C)C)NCC1(C)OCCN(C(c2cnc(C(C)(F)F)[nH]2)=O)C1 72783,N1(C(c2c(SC)nn(C)c2)=O)CCC(C2CCC2)(C(=O)NCc2ccoc2)CC1 72784,N#CCCCCCC(=O)NCC1CN(C(=O)Cn2cc(C(C)O)nn2)CCCO1 72785,c1(C(=O)NC2CN(C(c3ccc(C)cn3)=O)CC2O)cc(C(F)(F)F)ccc1O 72786,CC1CCCC(O)(C(N2CCCC(CCCc3ccccc3)C2)=O)CC1 72787,c1(C(N2CC(CNC(c3n(CC=C)ccn3)=O)C2)=O)ccc(N)c(F)c1Br 72788,c1(OC(C(N2CC(NC(C(C=CC)O)=O)C2)=O)C)cc(Cl)cc(Cl)c1 72789,Cc1cccc(C(C)C(=O)NC(=O)OCC(=O)Nc2cnn(CC#N)c2)c1 72790,C(=O)(CCC(C)(C)[N+](=O)[O-])Nc1c(OC)nn(C)c1 72791,c1(NC(C2CC(O)(CNC(=O)Cc3cc(Br)co3)C2)=O)ccc(CO)cc1 72792,N1(C(=O)C(C2CCCCC2)O)CCN(C(c2ccn3c2CCC3)=O)C2(CC2)C1 72793,C#CC(CNC(=O)CCCNC(=O)CC1(C)CC1)C(C)C 72794,c1(C(=O)NC(CCCNC(CN(C(=O)OCC)C)=O)C)ncnc2cc[nH]c12 72795,C1(CCOC(N2CC(NC(C=C(C)C(C)C)=O)C2)=O)CCCCN1C(=O)COC 72796,C(=O)(C1CCCc2scnc21)NCC1N(C(c2c(C)[nH]c(=NCC)s2)=O)CCC1 72797,CC1COCC(C(=O)NC2CCC(C(N3CCC(C4(C)N=N4)C3)=O)CC2)O1 72798,CCCC(C)CCCC(=O)NCC1(F)CCCN(C(C2C=C(C)CS2)=O)CC1 72799,C(=O)(C(C#N)(CF)C(=O)O)NC(c1scc(C)n1)c1ccccc1 72800,c1(-c2ccn(C(C)C)n2)cc2cc[nH]c2cc1C(N1CC2CC2C1)=O 72801,C1(NC(C(C)=CC2CC2)=O)CCCC(NC(c2c(C)noc2C(F)(F)Cl)=O)C1 72802,C1(COC(=O)C#CCc2ccccc2)C(F)(F)C12CC2 72803,c1(NC(CC=C)C)[nH]c(=NCc2cnc[nH]2)nc2c1cnn2C 72804,C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(C)CC(NC(C=CC)=O)C1 72805,C1(C(N(CCF)CC)=O)CCC2(CC2)N1C(c1cc(C2CC2)ccn1)=O 72806,C(CC(CNC(c1cc(C)co1)=O)NC(=O)C=CC1CCCC1)OC 72807,CCCCC(C)(F)C(=O)N1CCCC(CN=c2cc(C(=O)OC)nc[nH]2)(O)C1 72808,C1(C(=O)NC2(CC=C)CC2)CN(C)CCN1C(=O)C(CCC)OCC 72809,C(=O)(C1=CC2(CCOC2)C1)NC(CCNC(c1c(C)nc(C(F)(F)F)s1)=O)(C)C 72810,c1(C(N(C)CC2CCCN(C(=O)CCC3CCC3)C2)=O)n[nH]cc1[N+](=O)[O-] 72811,C(=O)(C1=CS(=O)CCC1)NC12CC(NC(CC(=O)NCC#C)=O)(C1)C2 72812,CCC(C)C(C(=O)NCC(C)(C)CCOC)NC(c1ccccc1NC)=O 72813,c1(C(C)Nc2ccc(-c3nnnn3CC3CCCO3)nc2)cccc2c1CCC2 72814,N1(C(CC2(COC)CC2)=O)CCC(C2CCN(C(C3(F)CCCC3)=O)CC2)CC1 72815,N1(C(C(C)(C)SC)=O)CCCN(C(c2nccs2)=O)C(C)C1 72816,CCC(C(=O)NCC1(F)CCN(C(c2cc(OC)n[nH]2)=O)CC1)C(C)O 72817,C1(NC(=O)COCC2CCCO2)CCCCN1Cc1nc(C2CC2)no1 72818,CC(C)(C)CCCN=c1ccc(S(=O)(=O)NCCCCC2CCCC2)c[nH]1 72819,c1(C(N2CCC(C(N(CC=C)CC=C)=O)C2)=O)c(C)nc2ncnn2c1C 72820,CCC(C(=O)NCC(C(C)(C)C)NC(c1cc(Br)n(C)c1)=O)C(C)C 72821,c1(OC)cc(C(=O)NC(C2(O)CCN(C(=O)C(C)(C)CO)C2)C)cc(Cl)c1O 72822,C(=O)(C#CC(C)(C)C)NCC1(C(N2CCC(CCC#C)CC2)=O)CC1 72823,c1(C(N2C(C)CC(CNC(c3n[nH]c(C)c3N)=O)C2)=O)cnn2c1CCCC2 72824,C(C)(CNCCC(C)C)(CC(C)C)NC(=O)C(O)CC(N)=O 72825,C(=O)(CC(C)(C)CNC(C1CC(=C2CCC2)C1)=O)NCC1CN(C)C(=O)C1 72826,c1(OC)ccc(O)c(C(=O)NC2CCN(C(c3ccc(NC(C)C)cn3)=O)C2)c1 72827,N1(C(CN(C(=O)OC)C)=O)CCN(C(=O)Cn2cc(CC(C)O)nn2)CC1 72828,C(=O)(CCCCS(C)(=O)=O)NCC1CCCCN(C(C(c2ccc(C)s2)C)=O)C1 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73055,c1(C(=O)NC(C2CCCN(C(C3CC(=C)C3)=O)C2)C)cnc2cc[nH]c2c1 73056,c1(NC(c2ccc(CNC(C)=O)cc2)=O)ncc(I)nc1Cl.C12CCCC1NC2 73057,C1(C(N2CCSCC2)=O)C2CCCC2CN1C(c1cccnc1O)=O 73058,N1(C(C(C(CNC(CC2C(CC)CC2)=O)C)F)=O)CC2CCC1C(O)C2O 73059,N1(C(C=CCNC(C(CC)C)=O)=O)CCCOC(CO)C1.C1(=O)COCCN1 73060,C(C)(C(C(=O)N1CC=CC(O)C1)C(C)C)NC(C1(CC=C)CCC1)=O 73061,N1(C(c2c(C)nsc2)=O)CCC(O)CC1C(=O)NCC12CC(CN1C)C2 73062,C1(CC=C)(NC(C2(C(F)(F)F)CCCC2)=O)CCN(C(=O)C2=COCCC2)CC1 73063,C(=O)(CCCC(C)(F)F)NCCSC.C1(C)(c2n(CCOC)nnn2)CCCO1 73064,C#Cc1ccc(NCCCCCC)cc1.C12OCCCC1c1nc2no1 73065,N1(C(c2cc(F)cc(C)c2O)=O)CCCC2CN(C(=O)C(C)(O)C(C)C)CC12 73066,CN1CCN(C(C2CCSCC2)=O)CC1C(N1CC(O)C(C)(C)C1)=O 73067,c1(C(N2C(CNC(C(CC=C)(C)C)=O)CCC(C)C2)=O)cnc2ccoc2c1 73068,Cc1ccc(C(=O)NC(C)CN(C)C(C2(F)CCOCC2)=O)nc1O 73069,C1(CNC(CC(CCC)O)=O)CC2(CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)CO1 73070,C1(CNC(C23CC(NC(C45CC(C(=O)OC)(C4)C5)=O)(C2)C3)=O)CC12CCOC(C)C2 73071,c1(CNC(C2N(C(c3csc(C)c3C)=O)CC(F)C2)=O)ccc(C#N)cn1 73072,C1(C(N(C)C)=O)CCCCC1C(=O)NCC1(c2cnn(C)c2)CCCO1 73073,N1(C(Cn2cc(C(=O)OC)nn2)=O)CCC(CNC(=O)C(C)CCC2CC2)CC1 73074,N1(C(C=CSC)=O)CCC(NC(c2cc(=O)c(C)c[nH]2)=O)C(F)C1 73075,C1(C(N2CC(NC(c3c(C)[nH]c(C)c3C)=O)C2)=O)(OC)CCCC(C)(C)C1 73076,C(=O)(CCCCC(CC)CC)N1CC(N2CCN(C(=O)NC)CC2)C1.C1C(=O)N1 73077,C1(NC(c2cnn[nH]2)=O)CCC12CCN(C(C1(CF)CC1(F)F)=O)CC2 73078,C1(CC)CN(C(c2ccc(Cl)cc2)=O)CCC1NC(=O)C=CC1CCCO1 73079,c1(OC)cc(C(N2CCC(C(C)NC(c3ocnc3C3CC3)=O)C2)=O)n(C)n1 73080,C#Cc1cccc(NC(C2CCC(C)N(C(=O)Cc3ccncc3C)C2)=O)c1 73081,CC1CN(C(c2cccnc2C(F)(F)F)=O)CC1NC(=O)C(O)CC1CC1 73082,N(C(=S)N1CCN(S(=O)(=O)C(F)(F)F)CC1)C1C(=O)NCCC1 73083,c1(C(=O)NCC2C(NC(c3c(OC)cccc3F)=O)C2)ccc2nc(C)[nH]c2c1 73084,Cc1noc(C)c1CCN(CCC(=O)N(C)C)CCCOCC(C)(C)C 73085,c1(OC)ccn2ncc(C(=O)NCC3CN(C(=O)CCC(C)O)CCN3C)c2c1 73086,C#CCC(CC#C)C(=O)N1CC(OC)C(NC(=O)C(CC)CC)C1 73087,c1(C(=O)NC2CCN(Cc3cn(C(CC)C)nn3)C2)c(C)nnn1CC 73088,C1(OCC)C(C(=O)O)CC1N=c1[nH]c(-c2ccco2)nc(C)c1C 73089,Cc1nc2c([nH]1)CC(C(N1CC(C(C)NC(=O)Cn3nccn3)C1)=O)CC2 73090,c1(OC)cc(N2CCC(NC(c3cc4ccccc4[nH]3)=O)C2)ccc1[N+](=O)[O-] 73091,N1(C(C(C)Oc2cccnc2)=O)CCCC(N(C(C2CCC3(CC3)C2)=O)CC)CC1 73092,C#Cc1cnn(CC(=O)NCC(C)(C(C)C)NC(c2nc(Cl)cs2)=O)c1 73093,CC#CCC(C(=O)NCCN(N1CCCC1)C)NC(=O)C(C(C)(C)C)OC 73094,c1(N2CCC(C3(NC(C4CCC(OC)C4)=O)CC3)C2)nc2cccc(F)c2s1 73095,c1(C(N2CCOC(CNC(C3(F)CCCOC3)=O)C2)=O)cc(F)ccc1Br 73096,C1(CNC(CN(CCOC)C)=O)(CO)CCN(C(=O)Cc2c[nH]ccc2=O)CC1 73097,C12(C(=O)NC(CC(C)NC(c3coc(CC4CC4)n3)=O)C)CC(C)(CO1)C2 73098,C(C(=O)N1CC(O)C(O)CO1)SC(C)C(N1CC2(CCCC2)C(=O)N1)=O 73099,C12(C(=O)OC(C)(C)C)CN(C(N)=O)C1CN(C(C(c1cocn1)C)=O)C2 73100,CN1CC(O)CC1C(=O)NC1CN(C(=O)COCCF)CC1F 73101,c1(C2(C(=O)NNC(C3CC4(CCC4)CO3)=O)CC2)nccc2[nH]ccc12 73102,CC1CC(NC(c2cc(Cl)c(Cl)n2C)=O)CN(C(C2CC(=O)N(OC)C2)=O)C1 73103,C(=O)(C1=NOCC1)NC(C1CN(C(=O)CCNC(C2CCCC2)=O)C1)C 73104,C(=O)(C(O)C(F)(F)F)NC1(CO)CCN(C(=O)CCN2CCOCC2)C1 73105,C1(C(=O)NC2CCCN(C(c3ccc(F)nc3)=O)C2)CCc2nnnn2C1 73106,C1(C(=O)NCCCCCN(C(CC2(CSC)CC2)=O)C)CNc2ccccc2O1 73107,Cc1nc(NC2CCC(NC(=O)CC(C)n3ccnc3)CC2)cc(C#N)n1 73108,c1(C(=O)Nc2ncc(F)cn2)ccc(Cl)nc1NCc1ccc(O)cc1F 73109,Cc1cccnc1C=CC(N1CC(N(C)C(C2CCS(=O)CC2)=O)C1)=O 73110,C#Cc1ccc(F)c(F)c1NC(c1cncc(NC(=O)CN2C(=O)CNC2=O)c1)=O 73111,Cc1cccn2cc(C(=O)NC3CC(CCNC(=O)CSc4nncs4)C3)nc12 73112,c1(NC(c2sccc2C)CC)cc(C)nc2ccc(C)cc12 73113,c1(C(N2CC(C)(NC(C3(OC)CCCC3)=O)C2)=O)c(C)nn(C)c1Br 73114,c1(C(=O)NCC(C2CCCC2)NC(C(C)n2cccn2)=O)cc(Cl)cnn1 73115,c1(OC)cccc(F)c1C(N1CC(O)(C(C)NC(=O)CCCCC#N)C1)=O 73116,CC1(NC(=O)CCC2CCCO2)CCC(NC(c2ccnn2CC#N)=O)CC1 73117,C=CC(CC)CC(=O)N1CCCC1C(=O)NC(CCOC)C(C)C 73118,N1(C(C(C)CN(C(=O)CCC2CC2(C)C)C)=O)CCCC2(CC(O)C2)C1 73119,c1(CC(=O)NCC2C(NC(CCN(CCCCC)C)=O)C2)cncnc1 73120,CC(C)CCC(O)C(=O)NN1CCCC1C(=O)NC1(C)CCCC1C 73121,N1(C2(NC(=O)Nc3cnccc3C)CC2)CC(Cc2nc(C)on2)CC1=O 73122,C1(NC(C2(CC)CCOC2)=O)C2CC(NC(c3cn(C4CC4)nn3)=O)CC12 73123,C(=O)(CCC(C)(F)F)NC(C)CCCNC(C1CCN(C(N)=O)C1)=O 73124,C(C(CC(F)(F)F)NC(=O)C=CSc1nc[nH]n1)NC(C=C1CCC(C)C1)=O 73125,N1(C(COCCCC)=O)CC(CNC(=O)CCCN(C)C)C(C(F)(F)F)C1 73126,c1(C(=O)NC(C)CN(C)C(c2cc[nH]c2C2CC2)=O)csc2c1CCCC2 73127,N1(C(c2c(C)n(C)nc2)=O)CCC(C(=O)Nc2cccc(Cl)c2)C1(C)C 73128,C1(O)(CNC(C=C(C)C(C)C)=O)CC(CNC(C2CSCCS2)=O)C1 73129,C1(COC)CC(CNC(c2cn(C3COC3)nn2)=O)N(C(=O)C(C)C(C)O)C1 73130,N1(C(CCCCCCCCC=C)=O)CC(=O)NC2CN(C(=O)C(CC)CC)CCC12 73131,C1(C(=O)OCC)CCON1S(=O)(=O)NCCSCCC(C)(C)C 73132,C1(CNC(C2N=C(C)SC2)=O)CC(C)N(C(=O)CSC2CCS(=O)(=O)C2)C1 73133,c1(-c2cn(CCCNC(C(C3CCOCC3)C)=O)nn2)ccc(CO)nc1 73134,c1(OCCC)ccccc1C(=O)NC1CN(C(C2CCCN2C(C)=O)=O)CC1C 73135,c1(C(=O)NCC2CC(C)N(C(=O)C=CCn3cncn3)C2)csc(S(C)(=O)=O)c1 73136,N=c1[nH]cc(C(=O)NCC2(O)CN(C(=O)CCOCC3CCCO3)C2)s1 73137,N1(CCOC)CCN(C(C2CCCC(NC(=O)Cn3cnc(Br)c3)C2)=O)CC1 73138,C1(NC(C(N2CCCC(C)C2)=O)=O)CCC12CN(C(=O)CCc1ccncc1)C2 73139,N1(C(c2nn(C)nc2Br)C(=O)NCCOCC)CCN2C(=O)N(C)C(=O)C2C1 73140,C(N=c1cc(NCCC(F)CN=[N+]=[N-])nc[nH]1)C1N(CC)CCCC1 73141,c1(N(C(=O)NC(CCC)Cc2ccccc2)C2CC2)ccc2c(c1)OCO2 73142,CC1(C)CCC(CNC(c2ncc3ccccn23)=O)N(C(C2CNC(=O)C2)=O)C1 73143,CCC(C)(CO)C(=O)NC1COCC1n1cc(-c2ccnc(NC(C)=O)c2)nn1 73144,c1(-n2c(CCn3c(C)ccc3C)nc(C(OCC)C)n2)ccc2ncsc2c1 73145,N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)C1CNC(c1ccc(Cl)o1)=O 73146,C(=O)(CN=S(C)(C)=O)N1C(C)CC(NC(c2n(CC=C)ccc2)=O)C1 73147,c12ccc(c(Br)n1)c1nc(-c3cnn(C)c3)nn21.c1(C(C)C)ccccc1 73148,c1(C(=O)NCCC(C)NC(C=NOC)=O)cc[nH]c2nccc1-2 73149,C(CCCC(C)NC(=O)Cc1nc(C2CC2)oc1C)NC(C(COC)OC)=O 73150,c1(CNC(=O)Nc2cnn(C3CCCCC3)c2)c(Br)ccc2ncccc12 73151,N1(C(C(C)(C)c2ccccn2)=O)CC2COCC2C1.c1cc(O)ncn1 73152,C1(C(N2CC(CC(C)NC(=O)CCNC(N)=O)C2)=O)(OC)CCOCC1 73153,c1(NCN2C(CNC(C=CC=CC)=O)CCC2)ccc(C=CC(C)C)nc1 73154,N1(NCc2cn(-c3ccc(N(C)C)cc3)nn2)CCc2n[nH]cc2C1 73155,C(=O)(C1=CS(=O)(=O)CCC1)NC(C1(O)CCN(C(c2ccn(CCF)n2)=O)CC1)C 73156,N1(C(c2c(C)coc2)=O)CCN(C(=O)C(F)(F)Oc2ccccc2)C(C)C1 73157,c1(C(N2CC(C(C)NC(=O)CN3CCCCS3(=O)=O)C2)=O)ccn2ccccc12 73158,Cc1nc(-c2c[nH]cc2C(=O)NCCN(C)C(c2sccc2CC#N)=O)cs1 73159,N1(C(c2c(CC)cco2)=O)CCC(C)C1CNC(c1n[nH]c(C)c1Br)=O 73160,C1(CNC(COC(CC)C)=O)CCC(CC(=O)NC(C)CCCCO)CC1 73161,CC1CC(CNC(c2ccc(F)o2)=O)CN1C(=O)CCc1ccsc1 73162,C(c1c(C)coc1C)=C(C)CSc1cnn(NC(N2CCCCC2c2nnco2)=O)n1 73163,C1(CCNC(c2cc(CC)no2)=O)CC(F)(F)CN1C(C1CCC(COC)C1)=O 73164,C(=O)(C(C#N)=CC(C)C)N(CCC)CCNC(C1(CO)CCC1)=O 73165,C=CCCCCCCC(=O)NCC1(OC)CCN(C(c2cncc(C)c2C)=O)C1 73166,N1(C(C2C3CN(C(C4CC5(CC(C)C5)C4)=O)CC32)=O)CC(O)C(O)C12CCC2 73167,N1(C(C(Cc2cnn[nH]2)NC(CC(C)N(C)C)=O)=O)CCCCCCCCC1 73168,CC(C)CC(=O)N(C1CC(NC(=O)CC2CC(C(F)F)C2)C1)C 73169,Cn1cnc2sc(C(N3CC(F)(CNC(C4CC4F)=O)C3)=O)cc12 73170,C1(Cn2cc(C(CC)O)nn2)CC(O)CN1C(c1cocn1)=O 73171,O=C(C1=CCCOC1)NC1(CO)CCN(C(c2ccccc2)=O)C1 73172,Cc1cc(N2CC(C)(C)CC2(C)CNC(=O)CCC2CCCO2)ccc1[N+](=O)[O-] 73173,C(=O)(C(CC(F)F)NC(=O)C(F)n1cccn1)N(C)Cc1ccnn1C 73174,Cc1nc(C(=O)NCc2c[nH]nc2C(=O)NC2CCC2O)c(C)s1 73175,c12ccccc1O2.C1(c2ccccc2)(CNC(=O)NC2CC2)COCCO1 73176,C=CC(C)C(C)C(=O)NCC1(CNC(c2cncc(Cl)c2C)=O)CCC1 73177,CCCCCCC(C)C(=O)C1=NC2(CCC2)CCNSC=NN1 73178,C1(C(C2CCCC(=O)N2)N(C2(C(F)(F)F)CC2)CC)CCN(C(=O)CC(C)O)CC1 73179,C(=O)(C(C)(C(=O)N1CCC(CC(c2ccc(F)cc2C)=O)CC1)C(C)OC)OC 73180,CN1CCC(CC(=O)N(CC(O)C2CC2)C2CC2)C1=O.C1C(=O)N1 73181,Cc1ccc2oc(C(N3CCN(C(=O)Cc4ccsc4Cl)CC(O)C3)=O)cc2n1 73182,CCCC(C(=O)N(CCC(C)NC(=O)CC)C)C(C)C 73183,C1(C(=O)OC)CC(C)(C)CCO1.C12CCN(C1)C2=O 73184,CC1(NC(=O)CCc2ccncc2)CC(NC(c2cncnc2)=O)C1 73185,C1(NC(C(C2CCN(C(c3ccc(O)nc3)=O)CC2)C)=O)CC(O)C1(C)C 73186,C1(C)(C(=O)NCC(C)(C)NC(C2(C)CC3CCC2C3)=O)CC2CCC1C2 73187,CC1(C(=O)NCC2(C)CCN(C(=O)Cc3csc(Cl)n3)C2)COC(=O)OC1 73188,C1(CNC(c2c(C)coc2)=O)(CO)CCN(C(=O)CCc2cccc(C#N)c2)CC1 73189,c1(NCC(=O)NCCC(=O)O)ccc(I)c(Cl)c1.C1(N)CC1 73190,C(CCF)(C(=O)N1CC(C(C)(C)O)C1)NC(CN(CCC#C)C)=O 73191,c1(-c2c(C(=O)OCC3(CC(=O)OC)CC3)noc2)cccc(I)c1 73192,C1(CNC(C(N2CCOCC2)C)=O)CCN(C(=O)CSc2cccs2)CC1(F)F 73193,CC1OCCC1CNC(=O)Nc1csc(C(N2CCCC2)=O)n1 73194,N1(Cc2nc(N(c3ccccc3Cl)C(C)=O)sc2)CCOc2ccccc21 73195,c1(C(=O)NC23C(CN(C(C(CCSC)OC)=O)C2)C3)n[nH]c2c1CSCC2 73196,CCC(CO)(C(=O)NCC1CCN(C(=O)C(C)N2CC(C)C2)C1)OC 73197,C12(C(=O)NC3C(NC(CCc4cc(C)no4)=O)C3)CCC(CC1)C(C)(C)O2 73198,C1(NC(C(C)N2CCC2)=O)C2COCC1CN(C(c1cnn(C3CC3)c1Cl)=O)C2 73199,Cc1ccc(C)c(C(N2CCC(C)(CCNC(c3c(C)ccnc3O)=O)C2)=O)n1 73200,c1(C(=O)NC23CCN(C(CCC(=C)Cl)=O)CC2C3)cc2c(C)c(F)ccc2[nH]1 73201,C1(COC)CN(C(=O)C(C(C)C)OC)CCN1C(=O)Cc1ccccc1C 73202,c1(CN2CC(C(N3CCC34CCCC4)=O)OCC2)c(F)cc(Cl)cc1Br 73203,C(=O)(CCCN(C(=O)CN(C(=O)CC1C=CCCC1)C(C)C)C)NC 73204,C1(CCNC(C(c2cncnc2)C)=O)CN(C(C23CCCCC2C3)=O)CCCO1 73205,C(=O)(C(CC(N)=O)NC(=O)Cc1cnsc1)NC(C(C)C)C1CC1 73206,Cc1cc(F)ncc1COC(C1CC(C)CCC1C)=O 73207,CN(Cc1c[nH]c2ccccc12)N(C)C1CCCOC1 73208,N1(C(C(COC)C)=O)CCN(C)C(CNC(=O)C=Cc2cc(Br)cs2)C1 73209,c1(N(C(C2CCC(n3cc(C(C)(C)CC4CC4)nn3)CC2)=O)CCl)ccc(F)cc1Cl 73210,C12(C(N3CCCN(C(CCC(C)OCC)=O)CC3)=O)CCCCC1C2(F)F 73211,C1(CC)(CC)CN(C(=O)C(C)(CO)NC(C2CC2C(N)=O)=O)CCO1 73212,C(CCN(C)C(c1cnn(C2CC2)c1)=O)(C(C)C)NC(c1cn(CC)nn1)=O 73213,N1(C(C2C3CN(Cc4[nH]n(C)c(=O)n4)CC32)=O)CCC(F)(F)C(F)C1 73214,c1(N(C)C)ccc(C(=O)NC2COCC2NC(C2(C(F)(F)F)CC2)=O)nn1 73215,C1(C(N(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)=O)CC(=O)NC(=O)C1 73216,c1(CNC(C=CCNC(CNC(CCC)=O)=O)=O)nnc(O)n1C.OCC 73217,CC(CCCCNC(=O)CCCCN(C)C)NC(=O)C(C)Cn1cccn1 73218,C1(C(N2CC(CNC(CC(C=C)(C)O)=O)C(C)C2)=O)CN2CCN1C(C)C2 73219,c1(CC)c(C(=O)NCC2CC(F)CN2C(C2CCC(C)S2)=O)cccc1C 73220,CC1CC(C(=O)NCCCCNC(C2(c3ccccc3Cl)CCCC2)=O)CCO1 73221,C1CC(C)(C)C(=O)N1.C(CCF)N(C(C=CC(=O)OC)=O)CCO 73222,CN1CCN(C(c2cc(CCNC(c3cc(O)nn3C)=O)on2)=O)CC(O)C1 73223,C1(C(=O)NC2CC(C(=O)NCC(=O)NC3CCC3)C2)(CC)CCCC1O 73224,c1(C(N2CCC(NC(Cc3cccc(OC)n3)=O)CC2)=O)cc(C)c(O)nn1 73225,N1(C(C#CC2(C)CC2)=O)CCC2CN(C(=O)CCOc3ccc(Cl)nc3)CCC12 73226,c1(CC)c(NC(Cc2ccccc2)C2CC2)cnn1-c1cccc(Cl)c1 73227,c1(SC)ccc(-c2cn(-c3ccccc3C(C)NC(=O)CC(C)F)nn2)cc1 73228,c1(C(C)C)cccc(C(N2CCC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)=O)c1O 73229,N12CCC3OCCN(C3C1)C(=O)C2.N1(C(CC)(C)C)CCCN(C(=O)OC)CC1 73230,C(=O)(CC(C)(C)c1cccs1)NC1(CC)CN(C(=O)CNc2nccs2)C1 73231,C1(O)(CNC(C2CC2CF)=O)CCN(C(=O)CCC=CBr)CC1 73232,Cc1cc(C(N2CC3C(CNC(C4(C)CCN(C)C4=O)=O)C3C2)=O)cc(C)c1 73233,CC(=O)CCCC(C)C(=O)NC1(C(N2CCC2C2CCCCC2)=O)CC(F)(F)C1 73234,C1(C(N2CCC(N(C(C(C)O)=O)C)C2)=O)COCC1(C)C.C1(C)(C)CC=CC1 73235,c1(C(=O)NC2C3CCC2N(C(c2occc2F)=O)C3)cc2ccc(F)cc2o1 73236,Cc1cc(CC(=O)NCCC2(O)CN(C(=O)CCc3ccc(C)s3)C2)on1 73237,N1(C(C(c2ncc(C)s2)C)=O)CC(O)CC1CC1CCNCC1 73238,c1(C(N2C(CNC(CN(C(=O)OC)C)=O)CCC2)=O)cc(Cl)cc(F)c1F 73239,c1(C(N(C)CC2(O)CCN(C(C(CC=C)CC)=O)C2)=O)cc2ccccc2cn1 73240,C1(CC(=O)N(C(CC)CO)CC)CN(C(c2cnc(C)nc2)=O)CC12CC2 73241,C1(C(=O)NCCN(C(=O)CN(C)CCO)CCOC)CCCSC1 73242,c1(CN(c2c(C(N3CCC3c3ccccc3)=O)n[nH]c2)CCO)cnc2[nH]ncc2c1 73243,N1(C(C2(c3ccccc3)C(C)(C)C2)=O)CCN(C(C2CCCC2)=O)CC(O)C1 73244,c12cc(ns1)C(=O)N(C)C(C)C(=O)NC2C1CC1.c1(CC)ccccc1 73245,c1(CC(C(=O)NCCC2(O)CN(C(C3(OC)CC3)=O)C2)O)cc(Cl)sc1Cl 73246,C1(C(=O)NCCCN(C(c2cccc(C)c2O)=O)CC)CC12CCC(F)(F)CC2 73247,O=C1CC(C(=O)OC(C(=O)NCCC(F)(F)F)C(F)(F)F)C2(CCC2)C1 73248,c1(C(=O)NCC(CO)NC(c2ccc(CO)o2)=O)cc2ccc(Cl)cc2[nH]1 73249,C(=O)(C(C)C1CC1)NCCN(C(CC1C(C)C1)=O)C1CC1 73250,C1(C(N(CC(=O)OCC)CC)=O)CCC(CNC(=O)Cn2cc(C#N)cn2)CC1 73251,C1(C)(C(N2CCC(C(=O)OC)CC2)=O)CCN(C(c2csnc2OC)=O)CC1 73252,C(=O)(CCCCCCCC(=O)NC1(C)CN(C(C2CCC(C)(C)CC2)=O)C1)OC 73253,c1(CCSCCC(=O)N(C)CCNC(C2(SC3CCCO3)CC2)=O)cccs1 73254,C12(C(N(C)CC3N(C(=O)C(=O)NCC4CC4)CCC3)=O)CCOC1CCOC2 73255,N1(C(c2cn(C(C)(C)C)nc2)=O)CCOC2CN(C(=O)Nc3ccc(Br)cc3)CC12 73256,C1(NC(c2sccc2F)=O)CC12CCN(C(c1cncnc1C1CC1)=O)CC2 73257,C1(CNC(CNC(CC)=O)=O)CCCN(Cc2cc(F)cnc2Cl)C1C 73258,N#Cc1ccc(NC(=O)C(N2CC(O)C(C#N)C2)=O)nc1 73259,c1(C(N2CCC(C(c3ccccc3)C(=O)NC(CC)C)C2)=O)cc(O)cc(Br)c1 73260,CN1CC(O)CC1(C)C(=O)NCC1(CCNC(C2CNC(=O)C2)=O)CC1 73261,C#CCCC(O)C(=O)NC1CC(C)(NC(c2csc(CCOC)n2)=O)C1 73262,C1(OC)CC(F)CN(C(c2cnn(C3COC3)c2)C(=O)NC2CCOC2)C1 73263,CCCCC(CN1CCCC1)N=c1[nH]c(=N)[nH]c(=NCCc2ccoc2)[nH]1 73264,N1(C(Cc2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCc1ccc[nH]1)C2 73265,N1(C(C2C(CC)C2)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73266,CCC(C)C(C)N=c1[nH]c(=NCC2(c3cnccc3C)CCC2)[nH]c2c1COCC2 73267,C=CCC(F)(F)C(=O)NCCN(C(=O)CC(=O)N(CC)CC1CC1)C1CC1 73268,C(=O)(CS(=O)(=O)CCOC)N1CC(CC(=O)N(CCCOC)CCO)OCC1 73269,C1(CC(=O)OC)(CO)CCN(C(CCCC2(CO)CC2)=O)C1 73270,N1(C(C2C(C(C)=O)C2(C)C)=O)CCC(N(C(=O)C(=O)NC2CC2)C)C(C)C1 73271,c1(C(=O)NC(CCOC)CNC(=O)C(C)NS(C)(=O)=O)c[nH]c(=S)cn1 73272,c1(C(=O)OCCC)nc2ccccc2c(NC(c2c(F)cncc2Br)=O)c1C 73273,C1(C(=O)NC(CCC)C2CCCC2)C=CCN(C(=O)C(C2CC2)OC)C1 73274,N1(C(C(CC(=C)C)NC(=O)Cc2ccn(C)n2)=O)CCN2C(=O)OCC2C1 73275,c1(C(C(=O)OC)NCC(Cc2ccccc2)N(C)C)ccccc1Cl 73276,c1(OCC)ccc(Cl)nc1C(=O)NCC1CCN(C(=O)CNC=O)CC1C 73277,C=C1CC2(C1)CC(C(=O)NC1(CF)CCN(C(c3cc(N)cc(F)c3)=O)C1)C2 73278,C1(NC(c2ccc(C)cc2)=O)CCCC12CN(C(C1(C)CCC(=O)N1)=O)C2 73279,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)sc(C(F)(F)F)cc1C 73280,c1(CCC)cccc(-n2nc(CS(C)(=O)=O)nc2C(O)CC2CCOCC2)c1 73281,c1(CCC(=O)NC(CN(C(C(C)=CC)=O)C)(C)C)c(C)ncnc1O 73282,Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)Nc3nccc(Br)c3O)nc2)c1 73283,c1(-c2n(CC3N(C(=O)Nc4c(C)cccc4)CCCC3)ccc2)cc(F)c(F)cc1F 73284,Cc1ccc(C(O)C(N2CCC(NC(=O)CSCC(F)(F)F)C2C)=O)cc1 73285,c1(C(N2C(C)CC(NC(c3ncccc3F)=O)CC2)=O)ccc2nc(O)sc2c1 73286,c1(NC)ccccc1C(=O)NC(N1CCC(C(C2CCCCO2)(C)C)CC1)=O 73287,C1(C(CNC(C2CC(OC)(OC)C2)=O)C)CCN(C(=O)Cc2conc2C)CC1 73288,N1(C(C(C=C)(C)CC)=O)CCN(C(=O)C(O)COC)CC(C)(F)C1 73289,N1(C(c2c(CC)cccn2)=O)CCC(NC(=O)COCCC(C)C)C(C)C1 73290,Cc1[nH]cnc1C(N1CCCC1Cc1nc(C2CC2)cs1)C(=O)NC(C)C 73291,CCCCC(CNC(=O)CC(C)OC)NC(c1cncc(Cl)c1)=O 73292,C1(NC(C(CC=C)C)=O)CCN(C(=O)Cc2ccccc2Cl)C12CCC2 73293,n1(C(C)C)cc(CC(=O)NC(C2CCN(C(C3(N(C)C)CC3)=O)C2)C)cn1 73294,CCCCCC(C)(C)C(=O)NN1CCOCC(O)(CC(C)C)C1 73295,Cc1cc(C#N)ccc1S(=O)(=O)NCC1(S(C)=O)CC1 73296,N1(C(c2c(CNC(CC(C(CC)C)O)=O)cc[nH]2)=O)CC23CCC2(COC3)C1 73297,C(=O)(CC(C)CC)N(C1(C(=O)NC(CCC)C2CC2)CCC1)C1CC1 73298,c1(C(=O)NC2C(NC(=O)Cc3nc[nH]n3)COC2)cc(O)nc(O)n1 73299,C=CC(C)CCN=c1[nH]c(N2CCOC(C(=O)NC)C2)nc2c(F)cc(F)cc12 73300,c1(C(=O)NC2C(NC(c3cc[nH]n3)=O)CCC2)ccnc2ccncc12 73301,N1(c2ccc(S(=O)(=O)NC(CO)C=O)cn2)CCN2C(=O)CCC2C1.C1CC1 73302,C12(C(=O)NC(CNC(C3(NC(C)=O)CCC3)=O)Cc3ccccc3)CC(C)C1C2 73303,FC(F)=C1CCC(c2nnnn2CC(F)F)(NCC2CCC2CO)CC1 73304,c1(NC2C=C(C)CCC2)ccc(S(=O)(=O)NC2CCn3nnnc3C2)cc1Cl 73305,CC(C)(CCC(=O)N1C2CCC1CC(C(=O)NCc1cnccn1)C2)[N+](=O)[O-] 73306,CC(C)C(C#N)C(=O)NCCCC(=O)NCCC1CCC(C)O1 73307,C(=O)(C1Cc2ccc(F)cc21)NC(CNC(C1(CCOC)CCCC1)=O)C(C)C 73308,C1(O)(CN(C(c2nnc(C)s2)=O)C)CCN(C(=O)C2=CCCCO2)CC1 73309,C(CC(C)C)(C(=O)N1CC(C)CCC1CO)NC(C(C)NC(C)=O)=O 73310,C1(C(=O)NCC2(F)CN(C(c3ccc(C)c(F)c3F)=O)C2)COc2ccccc2O1 73311,c1(C(N2CCC(CC=C)(NC(=O)CCCSC)C2)=O)ncc2cc(Cl)ccn12 73312,CON(CCC(=O)N1CCCC1c1ccnc(F)c1F)C(=O)N(C)C 73313,Cc1nncnc1C(=O)NCC1CC(F)(CNC(C2CNC(=O)C2)=O)C1 73314,C(=O)(C(C)(C)C(C)C)NCC(C1(O)CCN(C(c2n[nH]c(C)c2Cl)=O)C1)C 73315,N1(C(c2ccc(Cl)c(Cl)c2)=O)CC2CC1CN(C(c1coc(CC3CC3)n1)=O)C2 73316,N1(C(CCC)=O)CCC(NC(c2ccnc(N3CCCC3)c2)=O)C(F)C1 73317,N1(c2nccc(CC)n2)CC2CN(C(c3cccc(OC)c3OC)=O)CC2C1 73318,c1(C(=O)NC(CCNC(C2C(c3n(C)cnn3)CC2)=O)(C)C)ncnc(O)c1F 73319,CCCCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCN=[N+]=[N-])C1 73320,c1(C(=O)NCCN2CCN(C(C(C)CC(N)=O)=O)CC2)cnn2c(N)ccnc12 73321,C1(NC(C2N(CC)CC2)=O)CC2CC(NC(=O)CCNC(=O)C(C)(C)C)CC12 73322,N1(C(c2c(CNC(C(C)C(F)F)=O)cco2)=O)CCC(CO)C12CCC2 73323,N1(CCNC(C(C)OCC2CCCO2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1 73324,N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)C(F)C(C)C)CC2)CC1C 73325,c1(C(N(C)CC2N(C(C(C(C)O)(F)F)=O)CCCC2)=O)coc2cc(O)ccc12 73326,c1(C(=O)NC23CC(NC(=O)Cc4ccc(F)cc4)(C2)C3)noc2ccc(O)cc12 73327,N1(C(c2snc(COC)n2)=O)CCC(c2nn[nH]n2)CC1 73328,C(C(C(=O)NC1CC=CCC1)C(C)C)NC(c1c(C)ccn1C)=O 73329,CS(=O)(=O)c1ccc(CS(=O)(=O)N2CC(NCc3c(O)cccc3Cl)C2)cc1 73330,CC12CCC(C(N3CCC(NC(C4CCC(CC#N)CC4)=O)C(F)C3)=O)(CO1)C2 73331,c1(-n2cc(C3C(C)(C)C(C(=O)NCCC(=O)O)C3)nn2)cnn2c1OCC2 73332,c1(CC)cccnc1C(=O)OC.N12CC(CC1C(=O)OC)OC(CSC)C2=O 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73666,c1(N2CC3(CCN(C(CC(=O)N(C)C)=O)C3)C2)nc(Cl)nc2[nH]cnc12 73667,c1(NC(C2C(NC(C3CCC(=C)CC3)=O)C2)=O)ccc2ncsc2c1Br 73668,C(Cn1ccnn1)(C(=O)NOCCC(F)F)NC(C(C(C)O)N(C)C)=O 73669,C1(NC(CC2N(C(C=C(CC)CC)=O)CC2)=O)CNC(=O)OC1 73670,C1(NC(=O)COC(C)=O)CN(C)C(C)(COC)C1.n12cc(nn1)C(=O)N1CC2C1 73671,Cc1ccc(F)cc1CC(N1CC=CC(NC(c2occc2CN(C)C)=O)C1)=O 73672,Cc1ccc(C=CC(N2CC(F)CC2CNC(C2(C)CC3CC3C2)=O)=O)o1 73673,C1(NC(c2sccc2Cn2ccccc2=O)=O)CNC(=O)OC1 73674,c1(CC)nc2ccc(Br)cn2c1C(N1CCC(CCNC(=O)C(C)CO)C1)=O 73675,c1(CC)cc(C(=O)NCC(C2CN(C(=O)C=CC3CC3)C2)F)cn(C)c1=O 73676,n1(CC(=O)NC2CCC(NC(c3nc(COC)sc3)=O)C2)cnc2sccc2c1=O 73677,C1(NC(COCC#C)=O)CCN(C(=O)C(c2ccc(C)cc2)OC)CC1F 73678,CC(=O)C(C)CC(C)C(=O)N1CC(OCCC(=O)Nc2cccn(C)c2=O)C1 73679,c1(C(=O)NCC(CC=C)NC(=O)C(F)=CCC)ccc(-c2coc(O)n2)cc1 73680,C1(C(=O)NCCC(=O)NC)C2CCC(C2)N1CCC1CCOCC1 73681,c1(CC(=O)NC2CCC(N(C(=O)CCF)C)CC2)c[nH]c2ccc(Cl)cc12 73682,C1(CC(=O)N(CC=C)CCO)CCN(C(c2ccn(C(C)C)n2)=O)CC1 73683,Cc1nc(C(C)C)[nH]c(=NC2CCCC23CN(C(=O)Cc2ccccc2F)C3)c1Br 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73703,C(=O)(C(O)CC(C)(C)C)NCCCN(C(C(=O)NCCCC)C)C1CC1 73704,Nc1ccc(C(N2CCCC(CNC(=O)C(c3ccc(F)cc3)(F)F)C2)=O)nc1 73705,S(=O)(=O)(CCCS(=O)(=O)N(C1CN(C)C1)C)NC 73706,CC(C(=O)NC1CCN(C(=O)CNC(c2ccc(Cl)cc2)=O)C1)C(C)(F)F 73707,C1(CNC(C=C(CC)CC)=O)(NC(=O)CCc2ccc(Cl)c(Cl)c2)CCCCC1C 73708,CCCC(C)(C)CC(=O)N1CCOC(C(=O)NC(C)(COC)CCO)CC1 73709,c1(C(C(=O)N(c2ccn(C)c2)CC)N(C(c2ccccc2)CCO)C)coc(C)c1 73710,c1(NC(C(N2CCCC(CCC)CC2)c2ncccc2Cl)=O)cc(C)c(C)cc1C 73711,c1(C2C(C(=O)NCC3(F)CN(C(CCOC)=O)C3)C2)cccc(OC(F)(F)F)c1 73712,N1(C(C2C(CNC(=O)COc3cccnc3)OCC2)=O)CC2CCC2C1 73713,C(=O)(C1=CCC(NC(=O)C(O)CC(C)C)C1)NCC(CSC)(C)O 73714,c1(C(N2CC(CNC(C(CC)OCC)=O)(COC)C2)=O)c[nH]c2cccc(Cl)c12 73715,N1(C(C(CC)(C)O)=O)CC2CCC2(CC(=O)NCc2ccnnc2)C1 73716,CC1CN(C(C2(C)CC2)=O)CC(C)N1C(c1cccc(Oc2ccncc2)c1)=O 73717,C(C)(C)(CC(=O)NC1CCC(C(=O)NCCN2CC=CCC2)C1)OC 73718,C1(CCC(=O)OC)CN(C(c2ccc(C)nc2)=O)CCN1C(=O)C#CC1CCC1 73719,c1(CN(C(CC2(N(C(C(C3CC3)OC)=O)C)CC2)=O)C)ccccn1 73720,C(C(CC(=O)NCC1(C#N)CC1)C1CCC1)NC(c1c(C)[nH]cc1)=O 73721,c1(C(C)OC(C)=O)nc(CC(C)C)nn1-c1cccc(Br)c1 73722,C(=O)(CS(=O)(=O)NC(C)(C)Cc1ccccc1O)NC1COCC1O 73723,C1(C(=O)NC(C)CCNC(C2(C)CCC2)=O)C2CC1N(C(=O)OC(C)(C)C)C2 73724,c1(C(=O)NCC#CCNC(C(C(C)(C)C)N(C)C)=O)cc(N)cc2c1CCCC2 73725,C1(OC)(CC(C(=O)NC(C)C(C)(C)NC(c2ccc[nH]2)=O)=O)CCC(C)(C)CC1 73726,N1(C(Cc2ccc(COC)cc2)=O)CC2CC(C1)C2NC(=O)CC1(C)CCOC1 73727,C(N=c1[nH]cnc2c1COC2)C1N(C(=O)CC(F)(F)F)CCCC1 73728,c1(NC(C2(COC)CCCN2C(=O)CC2CC2OC)=O)ccc2cccnc2c1 73729,C1(CNC(COc2c(C)cccc2)=O)N(C(=O)C(C)NC(N)=O)CCC1(C)C 73730,N1(C(CC(C)(C)C2CC2)=O)CC2CCC(NC(C3COCCN3C(N)=O)=O)(C2)C1 73731,C1(N(C)C)CCC(NC(C2N(C(=O)C(N3CCCCC3)=O)CC2(C)C)=O)CC1 73732,C(=O)(C)NC1(C(C)(C)N(CC(C)N(C(C)=O)C)C)CC1 73733,C(=O)(C1=NNC(=O)CC1)NCC(C)(Cn1cccn1)NC(C=NOC)=O 73734,C1(C(N2CC3(N(C(CC4C(C)(C)CC4)=O)CC3)C2)=O)CCCCC(F)(F)C1 73735,N1(C(C2(CNC(=O)CC3(O)CCCC3)CC2)=O)CC2CC2C2CC12 73736,C(=O)(C(C)(C)C(=O)NC(C)C(C)CO)OC.n12cc(nn1)CN1CC2C1 73737,C1(CC(N2CCC(CCC(=O)NCCC(C)(C)C)C2)=O)CC2(C1)CC21CC1 73738,c1(NC(C(C(C)NC(C2C3CCC(F)(F)C23)=O)(C)C)=O)ccc2ccoc2c1 73739,CCCCC(C(=O)N(CC(C(C)C)OC)C)NC(=O)Cc1coc(C)n1 73740,c1(N(C)Cc2ccsc2)cc(N2CCC(CC3CC3)C2c2ccccc2)ncn1 73741,Cc1nc(C(=O)NCC(C2CCC2)NC(=O)C(=Cc2c[nH]cn2)F)nn1C 73742,C1(C(=O)NCc2cc(C)ncc2)CC(C)(C)CCN1C(=O)C1=CCCOCC1 73743,N1(C(COC2(C)CCCC2)=O)CC(NC(c2cc(O)nc(O)n2)=O)CC(F)C1 73744,N1(C(C(C)(C)C#N)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 73745,C(CC(C)(O)C(=O)NC(C1CCCC(O)C1O)=O)n1cc(C(C2CCOC2)C)nn1 73746,CC1CCCn2c(C(N3CCCCCC3CNC(=O)COC(C)C)=O)cnc21 73747,C(CCC(C)C)(C(=O)NCCC(C)(C)C)NC(c1c(C)cccn1)=O 73748,c1(C2C(C(=O)NCC(CC)(C)NC(=O)CCC(C)=O)C2)cc(F)cc(F)c1 73749,Cc1nc(NC(=O)C(N2CCOC(CS(C)(=N)=O)C2)=O)ccc1CO 73750,n1(-c2cn(C)nc2)nc(-c2cccc(N)n2)nc1-c1cnn(C(C)(C)C)c1I 73751,c1(C(=O)NCC(CC)NC(C2(C)CC(C(C)C)=NO2)=O)[nH]c2cc(C)ccc2c1C 73752,N1(C(=O)CCC2CCC2)CCC(N(C(=O)CC2CC2)Cc2ncccn2)C1 73753,C=CCCCC(C(=O)N(c1nc[nH]n1)C)NC(=O)CC(=O)NC(C)CSC 73754,C1(C(N2C(C)CC2C(=O)NCC2(CN(C)C)CC2)=O)CN(C)CCO1 73755,C1(C(=O)NC23C(CN(C(c4n(CC)nc(C)c4)=O)C2)C3)CC2(C1)CC1(CCC1)C2 73756,c1(C(=O)NCCC2(O)CN(C(c3ccsn3)=O)C2)cc(Br)ccc1Cl 73757,c1(CN2C(C(=O)Nc3c(C(C)=O)cccc3C)CC2)cn2nc(C)sc2n1 73758,CCCCC(CC(=O)NCC1(CO)CCOC1)NC(=O)C=CC(=O)OCC 73759,S(=O)(=O)(c1ncnn1C)NC12CC(CN(C)C)(C1)OC21COC1 73760,C1(NC(C(C)(CO)OC)=O)CCC2CCN(C(c3cn4ccccc4n3)=O)C1C2 73761,CCC(C)(C(=O)N1CCC(C(C(C)C)NC(C2CC(F)(F)C2)=O)CC1)OC 73762,N1(C(C(=Cc2ccco2)C)=O)CCCC(O)(CNC(=O)CNC=O)C1 73763,C(=O)(C(O)C(C)N(C)C)NC1(COC)CN(C(=O)C(c2ccc(Cl)cc2)=O)C1 73764,N1(C(c2cc(C(=O)OC)cn2C)C(=O)NCC(C)C)CC2(C1)CC2(F)F 73765,C1(C)(CNC(C(C)OCC)=O)CN(CCc2ccc(Cl)cc2)CCO1 73766,Cc1ccc(F)c(CC(=O)NC2CCN(C(=O)C(C)CC(N)=O)CC2O)c1 73767,N1(C(CC2ON=C(CC)C2)=O)CCC2CN(C(c3cncnc3C(C)C)=O)CC2C1 73768,C(C(CC)(CC)CO)NC(C1N(C(C(CC)COC)=O)CCCC1)=O 73769,CN1CCN(C(c2cncnc2)=O)C(C(=O)NCCCOCC2CC2)C1 73770,c1(CC(=O)N(CCC(=O)NCCC(CC)O)CCO)ccc(F)nc1 73771,N1CCN(C(=O)C(C)S(C)(=O)=O)CC1C.c1(-c2cn(COC)nn2)c(O)oc2c1CCC2 73772,O(P(C)(=O)CN1CCCC2(C1)OCCO2)CC1N(CC)CCC1 73773,c1(C(=O)OC)cc(NC2CC(C(F)F)C2)cc(Br)c1 73774,N1(C(Cn2c(C)nnn2)=O)CCCC12CCC(NC(=O)C(CO)N(C)C)CC2 73775,CN1CC2CCN(C(=O)C(CCC3CC3)NC(=O)CCC3(C)N=N3)CC2C1 73776,Cc1cn(C)cc1C(=O)NC1CC(CNC(=O)CC2(C)CCCO2)C1 73777,c1(OC)cc(OC)cc(CC(=O)NCCCC(C)NC(C2CCCNC2=O)=O)c1 73778,c1(CCN(C2CCN(C(C(C)OCC)=O)C2)C)nccc(C(F)F)n1 73779,N1(C(c2c(C)ccc(C)c2)=O)CCc2ccc(OC(F)F)cc2C1 73780,c1(C(=O)NC(CN(C(=O)C(C)c2ccsc2)CC)C)snc(O)c1Cl 73781,c1(SCC(=O)NC2CC2NC(c2ccoc2C2CC2)=O)cccc(Cl)c1 73782,c1(CC)nc(O)c(C(N2CCC(NC(=O)C(C)OCCN(C)C)C2)=O)cc1C 73783,C1(C(=O)OC)CN(C(c2ccc(Oc3ccc(NC(C)=O)cn3)cc2)=O)CC1C 73784,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCOCC1CNC(=O)C(=O)Nc1ncc[nH]1 73785,C=C(C)C(C)(C)C(=O)N1CCC(O)(CNC(=O)CNC(C2CCCC2)=O)CC1 73786,c1(CC(=O)Nc2ccc(NC(c3cocn3)=O)cn2)c(F)cccc1F 73787,C(=O)(CC1C(=O)Nc2ccccc21)NCC1(F)CN(C(CC2CN(C)C2)=O)C1 73788,C1(NC(c2c(SCC)cncc2)=O)CCN(C(=O)CNC(=O)C2CC2)CC(O)C1 73789,C1(O)(CC(=O)NCC(C)NC(C2(C(=O)N(C)C)CC2)=O)CCOCC1 73790,c1(OC)cc(C)c(S(=O)(=O)N(c2nnc3n2CCS3)C)s1 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73930,CC1(C#N)CCC(C(=O)OCC2CCCCC2c2ccccc2)CC1 73931,C1(C(=O)NCC(CN(C)C(C2CCN(C)C2=O)=O)O)CCC(=C(F)F)CC1 73932,c1(C(N2C(CNC(C(CC=CC)C)=O)CCCCC2)=O)cc2c(nn1)CCCC2 73933,CC#CCC(C)N=c1nc2c(ncn2C)c(NCC(n2cccn2)C)[nH]1 73934,C1(CNC(CCc2cnc(C)s2)=O)CN(C(c2cc3c(s2)CCC3)=O)C(C)(C)C1 73935,C1(c2ccc(C)c(F)c2)CC12CCN(n1nnnc1-c1cnc(C)c(C)c1C)CC2 73936,CC1OCCC1CN(C(=O)Cn1nnc(C2CCCCC2)n1)C 73937,C#CCC(CC#C)C(=O)NCC12CC1CN(C(=O)CN(C)C(C)C)C2 73938,C1(CNC(c2c(C(C)C)onc2)=O)CCN(C(c2ccoc2C(C)C)=O)CC1C 73939,c1(C2C(NC(c3cn(C4CC4)nn3)=O)C2)ccc(Br)cc1 73940,C1(C(N(C(C2CCCC2)C)CC)=O)CCN(C(=O)C=C2CCC2)C(C)C1 73941,C(C(C)CC(=O)N(CCC(=O)NCC1(C)CCCS1)CCCO)OC 73942,C1(NC(C2CC(=O)NC2)=O)CCCC12CCN(CCCc1csc(O)n1)CC2 73943,C(=O)(C(C)C1=CCCC1)NCCCN(C(C1CCc2nncn2C1)=O)CC 73944,C=C(C)CCC(=O)N1CC(CNC(=O)C(C)Sc2ccccc2)C(C)C1 73945,C1(O)(CNC(C(c2cccnc2)C)=O)CCN(C(=O)C=Cc2ccnn2C)C1 73946,n1(CC)cc(C(=O)NC2CC(F)(CNC(=O)C(CO)NC(N)=O)C2)cn1 73947,c1(OC)ccc2c(C(N3CCCC(c4cncn4C)C3)=O)ccnc2c1 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74125,C(=O)(CC(O)C(=O)NC(C)CNC(c1ccc(-c2cnn(C)c2)cc1)=O)OCC 74126,c1(C(C)C)nc(C(=O)NCC(O)CNC(=O)CSc2nnnn2C)cs1 74127,c1(C(=O)NCCC2(OC)CN(C(C3CC3C)=O)C2)cnn(C)c1C 74128,N1(CCc2cc(OC)cc(Cl)c2)CCC(=O)N(CC2CCC3(C2)OCCO3)C1=O 74129,C1(C(N2CC(CC(C)NC(C(C(C)C)NC(C)=O)=O)C2)=O)CCCC(C)(C)C1 74130,C1(C(=O)NC2CC(CCNC(CCC=C=C)=O)C2)Cc2ccccc2O1 74131,c1(CCCNC(=O)OC(C)(C)C)cn(CC(=O)NCc2ccoc2C(=O)O)nn1 74132,Cc1cc(Br)cc(C)c1-n1cc(C)nn1.C(=O)(C(F)C1CC1)NC1CC(C(C)(C)C)C1 74133,CC1CCC(O)(CNC(C23CC(CN2C(=O)Cc2cncnc2)C3)=O)C1 74134,C12(NC(C3C(COC)C3)=O)CC(C1)N(C(c1ccccc1NC)=O)C2 74135,c12cc(ccc1F)C(=O)O2.C1(NC(CC2(OC)CCC2)=O)CCC(F)(F)CC1 74136,N1(CCCN2CC(C)OCC2)C(=O)C2COC3(CCC3)CN2C1=O 74137,C=C=CCCNC(=O)C(C1CCOC1)NC(=O)CN(C)CCOC 74138,c1(N(C)C)nccc(OCCN(C(c2ccc(CC=C)cc2)=O)CC)c1C 74139,c1(C(=O)O)cnn(CCCCC=C)c1.C(=O)(C(F)(F)Cl)NCCS 74140,C1(C(NOCCCOCC)=O)(NC(c2ccc(C(C)=O)[nH]2)=O)CCCC1C 74141,c1(OC)cccc(S(=O)CC(=O)N2CCC(NC(c3coc(O)n3)=O)CC2C)c1 74142,C1(NC(CC(C=C)C)=O)CC2(CCN(C(=O)CCn3nc(C)cc3C)C2)C1 74143,c1(C(=O)NC2C(OC)CN(C(CCCOCCC)=O)C2)cnn2ccn(C)c12 74144,CCCCCC(O)C(=O)N1CCC(C(F)(F)F)CC1CNC(=O)COCC(C)C 74145,N1(C2CC(CC)C(=O)O2)CCOCCC1C(=O)N(CCN(C)C)C(C)C 74146,C1(O)(SCC(c2n(C(COC)C)nnn2)Oc2ccccc2)CCCCCC1 74147,N1(C(c2c(C)snn2)=O)CC2CCC1C(NC(c1n[nH]cc1[N+](=O)[O-])=O)C2 74148,C(CC(C(=O)NC(C1CCCN1C(=O)Cc1sccc1Cl)C)OC)OC 74149,N1(C(CSCCOCC)=O)CCOC2(CCN(C(=O)NCC)C2)C1 74150,CC1(C(N2CCC(O)(CCNC(=O)CCn3cc(Cl)cn3)C2)=O)CCC2CC2C1 74151,C(C(N=[N+]=[N-])C(=O)NCC1(NC(=O)CCP(C)(C)=O)CC1)OCC 74152,C1(NC(C(C(C)C)SC)=O)CC2CCC1CN(C(C1(O)CCCCCC1)=O)C2 74153,C(=O)(C#CC1(CC)COC1)N1CCC(N(CC#C)C(c2cncc(F)c2)=O)C1 74154,Cc1nsc(N)c1C(=O)NC1CC(F)(CNC(C2CC2C(F)(F)F)=O)C1 74155,C1(C(C#C)C)CCN(C(=O)NCCNC(=O)CC2CCCN2C(C)=O)CC1 74156,C1(C2CCN(C(C3CCN(c4nccs4)CC3)=O)C2)(NC(C2CCSC2)=O)CC1 74157,Cc1cc(C(N2CCCC(CNC(c3nncn3C)=O)CC2)=O)cnc1O 74158,CC(C)C(C(=O)NC1COCC1NC(C1CC(O)(C(F)(F)F)C1)=O)C(C)C 74159,C(C(O)CC(=O)N1CC(N(C)CC)C1)NC(CSCC=C)=O 74160,C(=O)(C1=CC2C=CC1C2)N1CC(NC(c2cc(C)oc2)=O)C(C(N)=O)CC1 74161,Cc1noc(Cl)c1CCC(=O)NC(C12CC(C1)C2)CNC(=O)C(=O)N(C)C 74162,c1(OC)cc(-c2nnc(C3(OC)CCCC3)o2)cc(OC)c1OC 74163,c1(CNC(c2cccc(Cl)c2)c2cncs2)csc2ccccc12 74164,C=C(Cl)C(C)(C)C(=O)OCC.c1(C=O)ccc(Cl)cc1.C1(=O)CO1 74165,n1(CCC(=O)N(c2ccccc2)C2CCN(C3CCCCCC3)C2)ccccc1=O 74166,CC#CCCC(=O)NCC=CCNC(=O)C(CC)C1CCCCC1 74167,N1(C(Cc2c(C)cc(C)s2)=O)CCC(NC(=O)C(C)NC=O)C(C)(C)C1 74168,N1(C(Cc2nc(C)c(C)s2)=O)CCC2CN(C(C3CC(F)(F)CS3)=O)CC2C1 74169,CC(=O)CCCC(=O)NCC(N1CCN(C(c2cc(C)cnn2)=O)CC1)C(F)F 74170,c1(N2CCc3c(OC)cccc3C2)nc(C)c2cc(Br)ccc2n1 74171,C(=O)(C#CC1CCOC1)NC(CCCC)CNC(c1ccc(OC2CC2)nc1)=O 74172,c1(C(=O)NC2(CC=C)CN(C(C3(CC(C)C)COC3)=O)C2)c(Cl)cnn1C 74173,C(=O)(C1CCc2c[nH]nc21)N1CC(c2cncnc2)(C(=O)OC)C1 74174,CC1CCN(C(=O)CC2CC(=O)NC2=O)CC1N(C)C(c1c[nH]c(=O)cn1)=O 74175,n1(CC(=O)NC2(CO)CCN(C(=O)C(c3ccc(F)cc3)F)C2)ccccc1=O 74176,C(=O)(CCCCCF)NCCOCCCN(C(c1cccc(CC(C)C)c1)=O)C 74177,Cc1cc(C(=O)NCC2C3CC2N(C(c2conc2C2CC2)=O)C3)cc(=O)n1C 74178,CCC(CNC(c1[nH]ccc1C)=O)(CC)C(=O)NC1CC(N(C)C(C)=O)C1 74179,c1(C(=O)NC(C2CCCO2)CC)cncc(CNC(=O)C(C)c2ccco2)c1 74180,C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2C)C1C 74181,Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CCN(CC(C2COC2)=O)CC1)=O 74182,N12CCC(CC1)NC2=O.c1(N(C)C)nnc(SC(C)(C)C)s1 74183,N1(CC)CCCCC1C(N1CC(O)CC1CNC(c1ccsc1C(F)F)=O)=O 74184,C(CC(C)C)(C(=O)N(C(C)CN(C)C(c1ccncc1C)=O)C)OC 74185,CC(C)(C)CS(=O)(=O)NCCCC1(O)CC2CCC1C2 74186,C1(CCOC)(NC(c2cn(CCCC)nn2)=O)CCN(C(C2CC(=O)CO2)=O)C1 74187,N1(C(CCC)=O)CCn2ncc(CN(C)C(c3cccc(Cl)c3F)=O)c2C1 74188,Cc1cccc2c1CCN2C(=O)CC(C)CC(C)C.C1(C2CNC2)(n2ccnn2)CC1 74189,c1(C(=O)NCCC2(O)CN(C(C=CCCC)=O)C2)cccc(OCC2CC2)c1 74190,c1(C(=O)NCC2CC(C)N(C(c3cc(C(C)(C)C)on3)=O)C2)cnc(F)c(F)c1 74191,C(c1ccccc1)=CC(=O)N(C(CNC(C1(C2CCCO2)CC1)=O)C1CC1)C 74192,Cc1ccc(C=CC(=O)NCC2(NC(C3CCN(C)C3)=O)CCC2)nc1 74193,N1(C(C=CCC)=O)CC(C)(C)C(NC(c2cc(CO)[nH]n2)=O)C(C)(C)C1 74194,c1(C(N(CC)CC2CCCCN2C(=O)CCC(C)C)=O)ccc(C)c(F)c1N 74195,Cc1cc(C(=O)NC2COCCC2NC(=O)CC2(O)CCOC2)oc1Br 74196,CCCCC(O)C(C)C(=O)NC(C(=O)NC1CC(C)(C)OC1(C)C)c1cccs1 74197,c1(OCC(N2CC(C)(C)OC(CNC(=O)C(C)(F)F)C2)=O)cccc2cccnc12 74198,c1(OC)cc(CNC2CCCN(c3cccc(F)c3)C2)ccc1OC(C)C 74199,N1(C(C(COC)NC(=O)C(O)CN(C)C)=O)CCC(C)(C)C1 74200,c1(OCC)ccc(C=CC(N2CC(CNC(C3CC(O)C3)=O)CC2C)=O)cc1OC 74201,c1(C(=O)NC2CN(C(c3c(C)ncs3)=O)C2)cccc(Cl)c1F 74202,C1(CC(C)NC(C2CCC(=O)O2)=O)CCN(C(C2C3COCC23)=O)CC1 74203,C(=O)(C(C)C(O)C(C)C)N(CCNC(COc1c(C)cccc1)=O)C 74204,N1(C(=O)Cc2cnsc2)CCN(C(C2CC(=C(F)F)C2)=O)CC1c1ccccc1 74205,C1(CN(C)C(C2(C)C=CCC2)=O)CCN(C(c2ncoc2C(F)(F)F)=O)CC1 74206,c1(C(N2CCC(N(C(CC(CC)SC)=O)CC)C2)=O)ccc(C)nc1C1CC1 74207,N1(C(c2c(C)nc(O)[nH]2)=O)CC2CCC1CC2NC(C1CCCO1)=O 74208,S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NCCNC(CCCC(N)=O)=O 74209,C1(NC(CCSC)=O)CCCN(C(c2sc(-c3ccsc3)nc2C)=O)CC1F 74210,C(c1ccc(O)c(OC)c1)=CC(=O)NCC(CNC(C1C(CC)C1)=O)C 74211,N1(C(C23C(C)OC(C)(C2)C3)=O)CCC2CN(C(=O)CCc3cncc(F)c3)CC2C1 74212,N1(C(C(C)O)=O)CCN(Cc2cc(Cl)ccc2Br)CC1C(F)(F)F 74213,N1(C(c2ccnn2CCF)=O)CCN2C(=O)C(OC3(CC(=O)OC)CC3)CC2C1 74214,Cn1c(C(=O)NC2CCC(CCNC(c3c[nH]c(=N)s3)=O)C2)cc(Cl)c1Cl 74215,N1(C(C2CC(C)CC(C)(C)C2)=O)CCCC2(C1)CN(C(c1cncs1)=O)CCO2 74216,c1(NCC2N(C(c3ccc(CCCC)cc3)=O)CC2)ccc(OC)cc1O 74217,CN1CC(O)CCC1C(=O)NCc1cnn(C)c1C(=O)NC12CC(C1)C2 74218,C(=O)(CCN(OC)C(=O)c1cn(C)nc1C#N)NC(CC(CC)C)C 74219,c1(CC)cnc(O)c(C(N2CC=CC(NC(=O)CCCc3nc(C)no3)C2)=O)c1 74220,c1(C(=O)NCC2N(C(C=NOC)=O)CCCC2)cncc2n[nH]cc12 74221,O=S(=O)(c1cc(F)cc(F)c1)NCCNc1nc2c(s1)CCCC2 74222,c1(C(=O)NC2N(C(N)=O)C3C(C2)C3)ccc(=O)n(CCNC(=O)CCCCO)c1 74223,c1(C(=O)NC2CN(C(C(C)C#N)=O)CC2C(F)F)ccc2nn[nH]c2c1 74224,c1(N2CC(C(C)NC(c3c(C)nc(C)s3)=O)C2)cc2c(cn1)C(=O)CCC2 74225,N1(CCC#C)CCN(C(=O)C(C(C)C)NC(=O)C(CSC)OC)CC1 74226,C1(C)CN(C(=O)NCC2OCCN(C(C)C)C2)CCC12CCC2.C(C)(C)(C)O 74227,N1(C(C2(C)C(C)CN(C(=O)C(=O)N=S(C)(C)=O)C2)=O)CC2(CCCC2)CC1C 74228,C12(CNC(C)=O)CC(CN(C)C)(CN1C(=O)CN(C)S(N)(=O)=O)C2 74229,c1(C(=O)NCC(C2CCCC2)NC(c2ccoc2Cl)=O)ccc2oc(O)nc2c1 74230,C1(C(C(=O)N(CC(=O)N(C)CC2CC(SC)C2)C(C)C)F)CCOCC1 74231,c1(C(N2CC3CN(C(CC(C=C)(C)C)=O)CC3C2)=O)nc(SC)n2ccccc12 74232,CC1CC(NC(=O)C(F)n2cccn2)CN1C(c1cncn1-c1ccccc1)=O 74233,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)CN(C(=O)CCCn1cccn1)C 74234,C(=O)(C1OCCc2c(O)cccc21)NC(C)(C)CCCNC(c1csnn1)=O 74235,c1(C(=O)NCCOCCCNC(C(CC)(C)C)=O)cn2c(n1)C(C)CCC2 74236,C1(C2CN(C(C3(OC)CCCC3)=O)C2)(NC(C(C2CCOCC2)OC)=O)CC1 74237,C(=O)(CC(C(F)F)c1ccccc1F)NCCN(C(CC(C)SC)=O)CC1CC1 74238,c1(C(N(CCNC(C2CC2C(F)F)=O)CC)=O)c(CO)c(C)nc2ccccc12 74239,C1(O)(CC(=O)N(CC(CC)NC(=O)Cc2csc(SCC(C)C)n2)C)CCOC1 74240,Cc1ccnc(O)c1C(N1CC2C(C(=O)N(C(C)C(C)C)C3CC3)C2C1)=O 74241,c1(C(N2CC(NC(c3n(C)nc(C(C)(C)C)c3)=O)C2)=O)cc2cc(F)ccc2s1 74242,c1(C(N(CC(C)N(C(c2cc(OCC)ns2)=O)C)C)=O)nc(O)nc(O)c1N 74243,N(C1CC2CCC(C)(C)c3cccc1c32)C=O.c1(OC(CC)CNCC)cccnc1 74244,c1(OC)ccc2cc(C(N3CCC(NC(c4oc(C)nc4C)=O)C3)=O)ncc2c1 74245,c1(CNC(CC(COC)NC(c2n[nH]cc2Cl)=O)=O)c(C)cccc1C 74246,CC(C)(CCCNC(C1CCOC1)=O)NC(=O)CSc1cccc(F)c1 74247,c1(C(N2CCN(C(CSCC)=O)CC2COC)=O)cn2nc(C)sc2n1 74248,c1(CN(C)C(=O)NC2CCOC2c2ccccc2)cccc2cccnc12 74249,C1(CC)COCCN(C(C2COCCC2NC(=O)COCCC(C)C)=O)C1 74250,C(=O)(C1=CC(C)(C)C1)N1CCC(NC(c2cn(CCC)nc2)=O)(COC)C1 74251,c1(NCC(CC)CO)ccc(S(=O)(=O)NCC2(C3CC3)CN(C)CCO2)c(Br)c1 74252,C1(C(=O)OC)(NCC(O)COc2ccc(F)cc2)CCOC(C)(C)C1 74253,CC1Cn2nccc2CN1C(=O)C1=CCCN(C(=O)COCCCF)C1 74254,N1(C(C(C)OCC=C)=O)CC(O)CC1CNC(=O)C1=C(Cl)CC1 74255,c1(CC(N2C(CNC(C3C(C(C)C)C3)=O)CC2)=O)cnc2ccccc2c1 74256,C1(N(C)C(c2ccc(Cl)s2)=O)CCCN(C(=O)CC23COC(CF)(C2)C3)CC1 74257,Cc1cc(CN2CCC(CC(=O)Nc3cnsn3)C2)c(C)n1Cc1ccccc1 74258,C(=O)(C(CNC(C1(Sc2cccnc2)CC1)=O)OC)NC(C#C)(C)C 74259,c1(CC)cccc2[nH]c(C(N3CCN(C(=O)CCOC(C)C)C4CC34)=O)cc12 74260,C1(F)(CN=[N+]=[N-])CN(CC2CCCO2)CC1C1CC1.c12ccc(cc1)NC2.OC 74261,c1(C(=O)NCCC(C)NC(=O)CCF)c(F)ccc(Br)c1N 74262,CC1CCN(C(C2CC2c2ccccc2)=O)C1CNC(=O)CCC1CCCC1 74263,CC1C(NC(c2cccc(Cl)n2)=O)CCN1C(=O)CC1(C)CCCO1 74264,CC(Cn1cccn1)C(=O)NCC1(C(=O)NCC(C)N(C)C)CCCO1 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74734,C(CCC(C(=O)N(C(C)CO)C)NC(=O)CC1CCCC(=O)N1)OC 74735,C1(NC(c2c(C)cn(C)c2)=O)C(C)CCN(c2ncc(Br)cn2)C1C 74736,N1(C(c2cc(C)cc(F)c2)=O)CCCN(C(C2C(C)C2C)=O)CC1C(C)C 74737,C1(NC(CC(COC)C)=O)(CO)CCCN(C(c2ccnn2C2CCCC2)=O)C1 74738,C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2cc3ccccc3o2)=O)C1 74739,N1(C(C2CC(=C)C2)=O)CCN(C(c2ncn3ccccc23)=O)CC2(CC2)C1 74740,C(C(COC1(O)CC(OC)C1)C(=O)N1CCC(C(C)(C)C)C1)OCC 74741,N1(C(C(C=C)OC)=O)CC2(CC(C(=O)N(C)CC3(COC)CCC3)CO2)C1 74742,c1(C(=O)NCC(CNC(=O)C2=NOCC2)O)cnc2[nH]c(O)nc2c1 74743,C1(C(=O)NC(CN(C(=O)CCN2CCOCC2=O)CC)C)CCC(O)CN1C 74744,N1(C(C2C(C)(C)C2C(F)F)=O)CCC(C)CC1.C(O)(C(F)(F)F)C1(C=O)CCC1 74745,C1(N=c2nc(C3CC3)[nH]s2)(CNC(C(C(C)O)C)=O)CCCCC1C 74746,C1(OC)CN2CC1C2=O.C1(NC(c2nc(Cl)cs2)=O)CCN(C)C1 74747,C1(CC(N2CCN(C(C)C(N3CC(F)(CN)C3)=O)CC2)=O)CCCC(F)(F)C1 74748,N1(C(CN(CC)CC)=O)CC2CCCC2(NC(=O)C(c2ccc(C)cc2)C)C1 74749,C1(=O)C2CC(=O)c3cccc(c32)O1.C(C)(CC(=O)OC(C)(C)C)N(CCC)C 74750,Cc1ncc(C(=O)NCC2(CN(C)C(c3cc(C)ns3)=O)CC2)s1 74751,C(=O)(C#CC1CCC1)NCCCC(C)NC(C1CC(c2ccccc2)O1)=O 74752,c1(CC(=O)NC2CCCC(CNC(C)=O)C2)ccc(F)cc1[N+](=O)[O-] 74753,N1(C(CN(CCOC)C)=O)CCCC(C(N2CC(C)SC(C)C2)=O)(CC)C1 74754,N1(C(c2ccc(F)s2)C(=O)NCC)CCc2c(cc(F)c(F)c2F)C1 74755,c1(N2CCN(Cc3sc(Br)c(C)c3C)CC2)ccn2ncnc2c1 74756,Cc1ccc(C#N)c(N2CC(O)(CN(C)C(C3CCS(=O)(=O)N3C)=O)C2)n1 74757,c1(C(N(CCCCCCNC(C2CCC(=C)CC2)=O)C)=O)cc2ccsc2n1C 74758,C12(C(=O)NCCCN(C)C(c3cccs3)C)C(NC=O)C3CC1C2C3.C(C)(C)(C)O 74759,Cc1c(C(=O)NCC2CN(C(c3occ4c3CCC4)=O)CC2C)cncc1Cl 74760,c1(C(=O)NCC(CN(C(c2c(C)n(C)cn2)=O)C)O)cc(C(F)(F)F)ccc1F 74761,c1(C(C)SCC)nc(-c2ccn(C(C)CC)n2)n(C2CCC2)n1 74762,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 74763,C1(S(C)=O)(C(=O)OC)CCN(C(c2nnc3n2CCCC3)=O)CC1 74764,Cn1c(=O)n(CCC(=O)NC2CCCCN(C(=O)CC#N)C2)c2ccccc12 74765,C(CNC(=O)CC1CCCN(C(=O)OC)C1)(CC(C)C)NC(C=CCCC)=O 74766,c1(CC(=O)NC2CC(NC(c3ccncc3Cl)=O)C(O)C2)cccc(Cl)c1F 74767,c1(COC)nc(Cl)cc(=NC2CC3CCC2N(C(C2(OC)CCSC2)=O)C3)[nH]1 74768,C1(NC(C(CC)=CC)=O)CCCN(C(=O)CCCC(C)N(C)C)C1C 74769,O=C(C1CCc2ccccc21)NC(CO)C(C)NC(C1CCCS1(=O)=O)=O 74770,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC2)=O)ccsc1S(N)(=O)=O 74771,N1(C(C23C(CN(C(c4cn5ccccc5n4)=O)C2)C3)=O)CCCC(F)C(F)(F)C1 74772,c12cc(COC)cc(c1Cl)N(CCN)C2=O.N1CC2CCC1C2.C(=O)(CCO)CC 74773,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)Cn1ccc(C)n1 74774,C1(NC(c2ccc(CC)cc2)=O)CCN(C(=O)C(C)C(C)C)C12CCC2 74775,C1(OC)CN(C(=O)CC2CCCOCC2)CC1NC(=O)CSc1ccccc1O 74776,CCC(C(=O)NC(C1CN(C(=O)CN(S(C)(=O)=O)C)C1)C)n1nccc1C 74777,N1(C(C(C)N(C(C)=O)C)=O)CCC(NC(=O)CC(C)(C)O)C1Cc1ccccc1 74778,c1(C(N2CCC(NC(C=CS(CC)(=O)=O)=O)C(F)C2)=O)cc(F)c(C#N)c(F)c1 74779,C=C(Cl)C(C)(C)C(=O)NCC1CC(NC(=O)Cc2cnc(C3CC3)s2)C1 74780,c1(C(=O)NC2CN(C(CCOC)=O)C3C2C3)ccc2ncn(C)c(=O)c2c1 74781,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 74782,C1(CN(C(COCC(=C)C)=O)C)CN(C(c2cnc(N(C)C)s2)=O)CCO1 74783,N1(C(c2ccnc3[nH]nnc23)=O)CCC2CCC(C1)N2C(C1CC=CCC1)=O 74784,N1(CC(=O)N(c2cccnc2)CC2OCC(N)C2)CCCc2occc2C1 74785,C(C(C)N=c1[nH]c(Cl)c(C(F)(F)F)c(Cl)n1)(c1ccccc1)NC(CC=CC)=O 74786,n1(C(CC)C)ncc(C(=O)NC2C3CC(NC(c4ncccc4O)=O)CC23)c1C 74787,C1(NC(c2ccc(-n3cccc3)nc2)=O)(CO)CCN(C(c2ccno2)=O)CC1 74788,C(=O)(CC(F)(F)C(F)F)N1C(CN(C(=O)CN2CCNC2=O)C)CCC1 74789,C1(C(=O)NC(C)Cc2nc[nH]n2)(CNC(c2nonc2N)=O)CCCCC1 74790,C(=O)(CC(C(F)F)n1ccnc1)NC1(C)CC(NC(=O)C(C2CCCCC2)O)C1 74791,n1(CCC(=O)NCC(CC)NC(c2cncc(C(C)C)c2)=O)nc(C)cc1C 74792,C(c1ccc(OCCO)cc1)=CC(=O)NC(n1ccnc1)C 74793,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(c2ccon2)=O)CC1(C)C 74794,C1(NC(C(C)OC(=O)OCC)=O)CC12CCN(C(=O)CCC1CCOC1)C2 74795,N1(C(C(C)Cn2ccnc2)=O)CC(C)(C)CC(C)(C)C1 74796,C1(F)(C(=O)NCC(c2ccccc2)NC(CC(C)OC)=O)CCS(=O)(=O)C1 74797,C1(CNC(CCC#C)=O)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 74798,N1(C(C)C)CC(C(=O)NCCCCCCNC(=O)C2=CCC2)CC1=O 74799,CCCC(C(C)(C)C)NC(=O)CC1(NC(C2CCC(=O)N(C)C2)=O)CCCCC1 74800,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CCO)C3)=O)CC2)CCC1=O 74801,C1(C(=O)NC2C(NC(C3CC4CCC3C4)=O)CCC2)CCC(F)(F)CC1 74802,c1(N(C2(CC#N)CCCC2)CCO)ncc(Cl)cc1[N+](=O)[O-].N12CCCC1CC2=O 74803,N1(C(C(C=C)OC)=O)CC(O)CC1C(=O)NCCOC1CCOC1 74804,N1(C(C(Br)=C(C)C)=O)CC(C)CC1CNCC(OCCO)OC 74805,c1(CNC(C=C(C#N)C(=O)N2CC(N3CC4CC4C3)C2)=O)c[nH]c(=S)cn1 74806,C=CCC(CC(=O)NC(C)C(C)(C)OC)NC(=O)C(C)OC1CCCC1 74807,C(=O)(CC(c1ccccc1)N(C)C)N(C)CCOCCN(C)C(C1CCCS1)=O 74808,c1(C(=O)NC2CCN(C(C(C)NS(CC)(=O)=O)=O)C2)cc(N)ccc1O 74809,c1(C(N(CC(=O)N(C)Cc2cncn2C)C2CCC2)=O)cc(F)cnc1O 74810,Cc1cnc(C)c(NC(=O)Cc2ccccc2NCc2cnn(C)c2)n1 74811,c1(C(=O)NCC23CN(C(C4(F)C(C)C4)=O)C(CC2)C3)cccc2c1CC(=O)N2 74812,C(=O)(CC1=NNC(=O)C1)NC1C(OC)CN(C(c2cscc2C(F)(F)F)=O)CC1 74813,C1(C(C(=O)NCCCC)N(C2CCCO2)C)C2CCOCC12 74814,N1(C(C=CCCC)=O)CC(O)CC1C(=O)NCC1(C(F)(F)F)CC1 74815,C(C(C)(C)S(C)(=O)=O)SCCNc1ccc(C)cc1 74816,CC(C)(C#Cc1cn(-c2ccnc(Cl)c2)nn1)NC(c1nsc2ccccc12)=O 74817,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(c2ccc(F)cn2)=O)C(c2ncc[nH]2)C1 74818,C12CCN(CC1)CCN2C(=O)CO.C(CCC(=O)Nc1ccccn1)=C(C)Cl 74819,c1(C(=O)NCC23CC2CN(C(=O)C(=Cc2c[nH]cn2)F)C3)nsc2ccccc12 74820,C1(F)(CNC(C(CC(C)C)N(C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 74821,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 74822,c1(NC(C2CCCN(C(c3nc(Cl)cn3C)=O)C2)C)[nH]c(=O)n(C)c(=O)c1C#N 74823,c1(OC)cccc(Sc2ccn(C(F)(F)C(F)c3cn(CCC#N)nn3)c2)c1 74824,c1(C(=O)NCC2CC(CC)CN2C(c2cc(=O)n(C)cn2)=O)ccc(F)c(O)c1 74825,N1(C(c2nccc(OC)c2)=O)CCC(NC(c2c[nH]c(C(N)=O)c2)=O)C(C)C1 74826,Cn1cc(C(C(=O)NCCC(C)(C)O)NC(=O)CNC(N)=O)nn1 74827,c1(NCC)cc(Cl)ccc1C(N1CCCC(NC(=O)C(C)C#N)C1)=O 74828,N1(C(CC2C(C)C2)=O)CCOC2(CCN(C(c3cc4cnccc4[nH]3)=O)CC2)C1 74829,CCC(CC)C(C)NC(c1ccoc1CNC(C1OC2CCC1C2)=O)=O 74830,Cn1ncc(C(N2CCC(O)(CNC(=O)CCCC(C)(C)C)C2)=O)c1S(C)(=O)=O 74831,c1(C(=O)NC2CC(CCNC(CC(C=C)C)=O)C2)cccc2oc(=N)[nH]c12 74832,c1(C2N(C(C3C(NC(CC(C)O)=O)CCC3)=O)CC2)ccc(F)cc1 74833,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 74834,C1(NC(C2C(C(=O)OC)C2(C)C)=O)CCC(C)N(C(c2ccc(F)c(F)c2)=O)C1 74835,C1(NC(c2cccc(CC)c2)=O)CCN(C(C2(CF)CCOCC2)=O)C(C)C1 74836,c12cc(ncn1)C(=O)N1CCOCC1CC(=O)NC2(C)C.c1(SC)cnc[nH]1 74837,C(C(C)C(C)C(=O)NCC1(NC(=O)CCCc2ccc(C)s2)CCOCC1)OC 74838,C1(CNC(CCC(=C)Cl)=O)CC12CCN(C(c1ccc(=NC)[nH]c1)=O)CC2 74839,c1(C(=O)NCCC(=C)CNC(C2OCC3CCCC2C3)=O)c(C)cc(C)nc1O 74840,c1(OC)cc(N)cc(C(=O)NC23CC(CNC(=O)C(C)(C)C)(C2)OC3C)c1OC 74841,O=C(C#CC1CC1)NCCOC1CCN(C(C23CCC(CO2)C3)=O)C1 74842,N1(C(C2CC(CC)(CC)C2)=O)CC(C(N2CCCC2CNC(C)=O)=O)CC1(C)C 74843,c1(C(=O)NCC(C)N(C)C(c2ncncc2Cl)=O)c[nH]cc(Cl)c1=O 74844,CC1CC(=O)NCC1C(N1CCCC1(C)CNC(C1CC(O)C1)=O)=O 74845,c1(OCC)ccc(Br)nc1NC(=O)CC1CC(C)N(C(C)C)C1 74846,Cc1cnoc1C(=O)N(C(C)CNC(=O)CC1(N2CCOCC2)CC1)CC 74847,C#CCCCCC(=O)NCc1cnn(C)c1C(N1CCCC1CC(C)O)=O 74848,CCCCCCCCC(=O)N(C1CCCN(C(=O)CC2CCCCC2O)C1)C 74849,CCCC(CCC)C(=O)NCC(O)CN(C(=O)CCOCC(F)(F)F)C 74850,C1(C(N2C(C)CCC2C(=O)Nc2ccc(F)nc2)=O)CC2CCCC2C1 74851,c1(C(=O)NCC(C)NC(c2ncn(CC)n2)=O)ccc(C)n1C 74852,c1(CC)ccsc1C(=O)N(C1CCN(C(=O)CCC=C(C)C)C1)CCOC 74853,C12(CC(=O)N(C3CC3)Cc3c(C)noc3)CCC1CNC2 74854,CC1CC(CNC(=O)CC2CCCCC2O)N(C(=O)C(c2ccc(Cl)cc2)O)C1 74855,c1(N(C)C(=O)C2CC2)ccc(C(=O)NCC(N2CCCCC2C)(C)C)cn1 74856,C(C(=O)NNC(=O)c1ccc(Br)cc1)(OC(F)(F)F)OC 74857,Cc1cc(C(=O)NC2CC(CCNC(C3(c4ccno4)CC3)=O)C2)cn1C 74858,C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(c2c(C)cc(F)s2)=O)CC1O 74859,N1(C(CSC)=O)CCN(C2CCC(NC(=O)Cc3cnns3)C2)CC1 74860,c1(C(N2CC(NC(C=CC(C)(C)C)=O)C(F)C2)=O)cc(C(F)(F)F)ccc1Cl 74861,N1(C(C2CN(c3cc(OC)ncn3)C2)=O)CC(C)C(C)C1C 74862,c1(OC(C)(C)C)ccc(C(=O)NC2CC(NC(C3C(C)C3C)=O)C(O)C2)cc1 74863,CC(C(=O)N1CCN(C2CCN(c3cncc(Cl)n3)CC2)C(=O)C1)S(C)(=O)=O 74864,C1(C(=O)NCC(COC)NC(c2ccsc2Cl)=O)(OCC)CCSCC1 74865,C1(F)(CNC(CC2(OC)CN(C(=O)Cc3cc(C)on3)C2)=O)CCN(C)C1 74866,Cc1cc2[nH]c(C(=O)NC3CC4(CCN(C(=O)C(=O)NC5CC5)C4)C3)cc2o1 74867,N1(C2(CC(=O)N(C(C)(C)C)CC3CC3)CCC2)CC(O)C(C)(C)C1 74868,C(C)(C)(CC(=O)NC(CCN(C(=O)C(c1ccncc1)OC)C)C(C)C)OC 74869,c1(C(=O)NC(c2cnn(C)c2)C(=O)N(CC(C)OC)C)cc(OC)n(C)n1 74870,N1(C(CCNC(C2=C(C)CC2)=O)=O)CCN2C(=O)CCC2C1 74871,CC1CCN(C(c2ccc3c[nH]nc3n2)=O)C(C)C1NC(=O)C1=COCCO1 74872,C1(NC(c2cc(C)nc(C)n2)=O)CC2CCC(C1)N2C(=O)C(O)C1CC1 74873,c1(C(=O)NC2CCC(F)(CNC(C)=O)C2)ccc(Nc2ccncc2)cc1Cl 74874,c1(OC)cccc2[nH]c(C(=O)NC(C)CNC(c3c(C(F)(F)F)ncn3O)=O)cc12 74875,C(=O)(C(F)(F)C(C)(C)O)NC(C1CCCCC1)CNC(c1cnc(CC)[nH]1)=O 74876,CCC(O)C(F)(F)C(=O)NC(C1CCCC1)CNC(C1CCNC1=O)=O 74877,N1(C(CC=C)=O)CCC2(CO)CN(C(c3coc4cc(F)cc(F)c34)=O)CC2C1 74878,Cc1cc(C)c(C(=O)NCCN(C(=O)CC2CC2C)C)c(C)c1 74879,N1(C(C(CCN(C)C)NC(=O)CCn2ccnc2)=O)CCC(F)(F)C(F)C1 74880,C#Cc1ccc(OCC(=O)NC2CCOCC2NC(=O)CN2CCOCC2)cc1 74881,O=C(C1CC=Cc2ccccc21)NC1CN2CCCC2CN1C(=O)C1=NOCC1 74882,CN=c1nc(N(C)Cc2ccc(S(C)=O)cc2)[nH]c(=NC(C)c2ncnn2C)[nH]1 74883,C1(NC(=O)CCCF)CC2CC1N(C(c1ccncc1C(F)(F)F)=O)C2 74884,C1(COC)CN(C(C2CC2(C)C)=O)CCN1C(c1ccn(CC(F)(F)F)n1)=O 74885,C(=O)(CC1=CCCCC1)N1CC(C=C)C(NC(C2CN(C)CC(C)O2)=O)C1 74886,c1(C(=O)NC2(CF)CCN(C(C(C(=O)OCC)(C)F)=O)C2)cnc2[nH]cncc1-2 74887,C1(C)(COC)COCCN1c1nnc(-c2nncs2)n1CCC1NC(=O)NC1=O 74888,Cc1ccc(C(=O)NCC2(NC(C3CCOC3c3cnn(C)c3)=O)CC2)c(N)c1 74889,N1(Cc2cc(C)ncc2)CCc2cccc(C(N3CCNC(=O)CC3C)=O)c2C1 74890,C1(C)(COC)CCN1C(=O)CCC1CC(NC(=O)CC2(C)OCCO2)C1 74891,C1(C(N(CCCN(C(Cc2cc(C)on2)=O)C)C)=O)CC1C1CC1C 74892,N1(C(c2c(CNC(C3(OC)CCOC3)=O)occ2)=O)CC(C)C12CCOCC2 74893,Cc1ccc(Cl)cc1-c1cn(C2CC(NC(c3csc(F)c3)=O)C2)nn1 74894,CC1(C)CCCCC1C(=O)NC1C=CC(C(=O)NCC2CC(O)C(O)C2)C1 74895,N1(C(c2cc(C)on2)=O)CCC(F)(C(=O)NC(C)CC2CCCOC2)CC1 74896,N1(C(C(CCC)(C)C)=O)CCCC(C2CN(C(=O)Cc3ccc(F)c(Cl)c3)C2)C1 74897,N1(C(C2(S(N)(=O)=O)CC2)=O)CCC2(C1)CN(C(=O)CC1COC3(CCC3)CO1)C2 74898,C1(CC(=O)NCC(CC)NC(c2cc(F)ccc2NC)=O)CC(C)(C)OC1=O 74899,C(C(C)(C)CC(=O)NCC(C1CC1)NC(C1CC(C)(C)CO1)=O)N(C)C 74900,c1(C(=O)NC2CC(NC(C34CCC(CC3)OC4)=O)C2)cc2cc(Cl)ccc2o1 74901,C1(O)(CCNC(C2(OCC)CCC2)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1 74902,N1(C(CCC(=O)N(CCC)CCC)=O)CC2CN(C(=O)CC(C)C)CC(C1)O2 74903,c1(C(N2CC(CC)C(NC(c3cscn3)=O)CC2)=O)cc2nccc(Cl)c2s1 74904,C1(C(N(CC(CCC)C)C)=O)CCC2(CC2)N1C(C1CCCO1)=O 74905,c1(SC)ncccc1C(N1CCCC1C(C)NC(c1ccnnc1)=O)=O 74906,N1(CCN(c2c(C)cnnc2)c2ncc(Br)cn2)CCc2cccc(C(F)(F)F)c2C1 74907,c1(CC)cc(C(N2CCOCC2CNC(C2CC(=O)N2)=O)=O)ccc1Cl 74908,CC1CC(CCN2CCCC2Cc2ccccc2)CCO1 74909,CCCCC(O)CC(=O)NCC1(CNC(=O)CCOc2ccc(C)cc2)CCC1 74910,C1(C)(C(=O)NC(C)Cn2cnccc2=O)CCN(C(=O)C=Cc2ccc[nH]2)CC1 74911,c1(C(N2CCN(C(C3CCC(=C)CC3)=O)C(CC)C2)=O)c(Cl)ccc(OC)c1N 74912,Cc1cc(=NCC(COCCO)C(C)C)[nH]cc1S(=O)(=O)NCc1nnc(CO)s1 74913,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 74914,C1(C(=O)NCC(C)NC(=O)CCC(=O)c2ccc(Cl)cc2)CCC2CCC1O2 74915,C1(OC)CC(N(C)C(c2ccc(-c3ccsc3)nc2)=O)C12CCCCC2 74916,N12C3CCC1N=C1N=CNN3C=C(Br)C=C1c1nc2nc(OC(C)C)c1SCC 74917,Cc1cc(NC2CCN(C(c3cc(Cl)nc(C4CC4)n3)=O)CC2)nc(C2CC2)n1 74918,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)SCC2CCCO2)CCCC1 74919,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)CC2CC(C)(C)C2)C1(C)C 74920,c1(C(N(CCCNC(C)(C)C)CC)=O)ccc(SC)cc1 74921,C12(COC)CCC(C(=O)N(C)Cc3csc(=N)[nH]3)CC(CN1)C2 74922,N1(C(CCN2CCC(C)CC2)=O)CC(NC(C2CCOC2)=O)C2(CC2)C1 74923,C1(CC(=O)N(CC(CNC(C2(CCC)CC2)=O)C)CC)COC2(CCC2)CO1 74924,C1(NC(C(n2cc(CC(C)(O)c3cccs3)nn2)C)=O)CNC(C#N)C1 74925,CC1CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(c2ncccc2F)=O)C1 74926,c1(C(N2CCCC2C2CCCCC2)C(=O)NC)cc(OC2CCOC2)n(C)n1 74927,N1(C(CCC2CC(NC(c3occ(C(N)=O)c3)=O)C2)=O)CC(O)CC12CCC2 74928,N1(C(c2nc(OC)c(F)cn2)=O)CCC2OCCN(C(=O)C(C)C)C2C1 74929,CC1CCCCC1(CNC(=O)CNC(c1cnn(C)c1)=O)NC(=O)C(F)=C(C)C.C(C)(C)=C 74930,c1(C(N2CC(NC(C3CC3Cl)=O)C2)=O)ccc(Br)c(Cl)c1Cl 74931,C1(N(C(=O)CSc2ccoc2)CC)CCN(C(C2CC(C)(F)C2)=O)C1 74932,Cn1ncc(=NC(=O)C2CN(Cc3ccc4nccn4c3)CCC2O)[nH]1 74933,N1(C(c2n[nH]c(CCOC)c2Cl)=O)CCOCC(C(=O)NCC(=O)OC)C1 74934,C12(CNC(c3cn(CCOC)nc3)=O)CC1CN(C(c1ccn(CCF)n1)=O)C2 74935,C(=O)(CCC(C)(F)F)NC(c1ccc(F)cc1)CNC(CN(C1CCC(=O)NC1)C)=O 74936,C(CCO)(C(=O)N1CC(O)C(O)C1)CN(C(=O)C(O)CC1CCCC1)CCO 74937,CC1=C(C(=O)N2CCCC(C)(C(=O)N(c3ccc(C)n3C)CCC#N)C2)CCO1 74938,Cc1ccn(CC(N2CC(CNC(C3CC3c3cccs3)=O)CC2C)=O)c(=O)c1 74939,C1(NC(CNC(C(CN(C)C)OC)=O)=O)CC2C=CCC(C1)C2 74940,C1(C(=O)N)CC(=O)N(CCC2(NC(=O)COCc3ccncc3)CCC2)C1 74941,Cc1c(F)ccc(Cl)c1C(N1CC2CC(NC(=O)C#CC3CC3)CC2C1)=O 74942,Cc1c(CC(=O)N(C)CCNC(c2cn(C)c(C)n2)=O)cccc1Br 74943,N1(C(c2nc(C(C)N)oc2)=O)CCC2(CC1)CN(C(=O)C=CCF)C2 74944,N#Cc1ccc(NC(c2n[nH]cc2NC(c2c(Cl)cc(O)cc2Cl)=O)=O)cc1Br 74945,C1(C(=O)NCC(N2CC(OC(c3cc(C(=O)OC)n[nH]3)=O)C2)=O)CCC(O)CN1C 74946,C(=O)(CC(C)C1CCCO1)NC1(C(N(CCF)CC)=O)CCC1 74947,C(=O)(C(=O)N=S(C)(C)=O)NC1CC(NC(C(C)CF)=O)C1 74948,Cn1nc(O)cc1C(=O)NCC1CC1CNC(c1nnsc1N)=O 74949,C12(NC(C=CSC)=O)CCCCCC1N(C(c1cc(F)c(N)cc1F)=O)CC2 74950,CCCC(CC)C(=O)N1CC=CC(NC(=O)Cc2cc(OC)cc(Cl)c2)C1 74951,N1(C(C2CC(CCC)C2)=O)CCC(CN(C)C(c2ncn(C)n2)=O)CC1 74952,c1(CNC(C(C)N(C)C(C2(C#N)CCCO2)=O)=O)ccccc1CO 74953,C#CC1CN(C(=O)C(C2CCC2)NC(=O)CCN2CCOCC2)CCO1 74954,c1(CNC(C(C)NC(CC)=O)=O)nc2c(s1)CCN(C(C1CCC13CCC3)=O)C2 74955,N1(C(C(C)OCCOC)=O)CCC2(CCCN(C(=O)CCCN(C3CC3)CC)C2)CC1 74956,c1(C(=O)OC)cccc2c(=O)c(C)c(CO)[nH]c12.C12CCCN(C1)Cc1cn2nn1 74957,Cc1ccc(C(=O)NCC2CCN(C(c3cc[n+]([O-])cc3)=O)C2)cc1O 74958,C1(C)(C(=O)NCC(C)CCCF)CCCN(C(=O)COCC2CCC2)C1 74959,c1(CNCc2n(CC(C)C)ncc2)cc(F)c(Cl)cc1F 74960,c1(NC(C(C)(C)C2CCN(C(=O)CC3(C)CCC3)C2)=O)ccc2nccn2c1 74961,C(C)(C(=O)NCC1CC1CNC(=O)CN(S(C)(=O)=O)C)OCC=C 74962,C1(NC(C(C2CC2)OCC)=O)CN(C(=O)Cc2ccc3c(c2)CC3)CCC1(F)F 74963,C1(C(=O)Nc2c(C)nsc2)CCC=CC1N.c1(C(=O)NC)cnn(C)c1C 74964,c1(N2CCN(CC)CC2)ncc(C(=O)OC(c2noc(CO)n2)C)cc1Cl 74965,N1(C(C(C2CC2)OCC)=O)CCC(F)(F)C(CNC(=O)CCNC(=O)CO)C1 74966,C(CNC(=O)C=C1CC1)(CO)NC(C=CC(C)C)=O 74967,C1(NC(c2cncc(Cl)c2Cl)=O)CN(C(C2(F)CCCCC2)=O)C2(CCCC2)C1 74968,C12CC3CCC(C1)N3C(=O)C13C(OC(C)(C1)C3)C(=O)OC2=O.C(C)(C)(C)N(C)C 74969,C1(CNC(CCc2onc(C)n2)=O)CN(C)CCN1C(C1CCC(=O)N1C(C)C)=O 74970,C1(O)(CNC(C2=CC(C)(CC)C2)=O)CCCN(C(c2cc(F)ccc2F)=O)CC1 74971,C(=O)(C1CCCc2nncn21)NCC(C(C)(C)C)NC(c1cc(Br)no1)=O 74972,Cc1cnc(NC(C2CC2C(=O)Nc2cccc(I)n2)=O)c(C)c1 74973,CC1CC(NC(=O)CCC2(C)CC2)CN(C(C2CC2C2(C)COC2)=O)C1 74974,C1(C(=O)OC)CCCC(C(=O)NCCCC(C)CO)C1 74975,c1(CC(=O)NCC(C)NC(c2cc(C3CC3)[nH]n2)=O)ccc(Cl)cc1.C(C)(C)(C)O 74976,C(=O)(C1CCCc2nncn21)NCC1CN(C(c2[nH]cc(CC)c2)=O)CC1C 74977,C1(CC(=O)NCC2CCC(NC(C=C(CCN(C)C)Cl)=O)C2)CCCN(C)C1 74978,c1(CC(=O)N(C)SC)cc(F)c(F)cc1F.C12(CCC1)C(=O)NCC1(CC1)N2 74979,C(=O)(C1=C(c2cc(F)cc(F)c2)N(C)C(=S)NC1c1ncc(Br)c(C(=O)OC)n1)OC 74980,N1(C(C(=O)NC(C)CCCNC(C2CCCO2)=O)C)CCCCCC1 74981,C1(NC(C(C)N(C(CCN(C)CC)=O)C)=O)CC2CCCC2C1 74982,c1(OC)ccnc(F)c1C(=O)NC1CN(C(c2csc(CO)n2)=O)CC1C 74983,C1(COC)(NC(C2CC23CCC3)=O)CCN(C(C2(C)CCCCO2)=O)CC1 74984,C(CC(C)C(=O)N(C)CC1CCCN1C(c1cc(-c2cccnc2)[nH]n1)=O)OC 74985,Cc1cccc(C(N2CCC2CNC(C2(C)CC(=O)N(C)C2)=O)=O)c1O 74986,c1(C(N(C2CCCC2)CCNC(CC(C)SC)=O)=O)c(NC(C)=O)cccc1F 74987,c1(N(C2CN(C(=O)NCCCOC(F)F)C2)C(C)C)c(OC)cccc1F 74988,CN1CCCC12CCN(Cc1nc(Cl)c(Cl)s1)C2 74989,N1(C(CCOCCNCCCO)=O)C(C(=O)OCC)CCC1C(C)C 74990,C1CC(F)(F)Cn2cc(nn2)C1.n1(C(=O)OCCSCCO)cc(COC)nn1 74991,C1(CC(=O)O)NCC2CCN(C(=O)CC=C(Cl)Cl)CC12.COCC 74992,N1(C(C2C(C)CC2)=O)CCN(c2ccc(CNC(=O)CC3CSC3)cc2)CC1 74993,C(=O)(CS(=O)(=O)CCOC)NC1C(NS(CCCC)(=O)=O)CCN(C(COC)=O)C1 74994,c1(C(=O)NCC(=O)NC2(CCNC=O)CC2)cnc(-c2ccoc2)s1.C1CCC1 74995,CC1(C(N2CC3C(NC(c4ccc(-c5ccco5)nn4)=O)C3C2)=O)CC2CC2C1 74996,S(=O)(=O)(CCNC(=O)C(=O)N(C1CCCSC1)CC1CC1)NC 74997,C1(CNC(c2n(CC#C)ccc2)=O)CCCCN(c2ccc(C#N)cn2)C1 74998,C(CC(C(C)(C)C)NC(C12CCC(C1)OC2)=O)N(C(c1c(CC)nns1)=O)C 74999,C1(SC)CC(CC(=O)N(C(C)C(=O)NCCCC2CCOC2)C2CC2)C1 75000,c1(CC(=O)NCCCN(CCC)C(C2CCOC2=O)=O)cnn(C(C)(C)C)c1 75001,N1(C(CS(CC)(=O)=O)=O)CC2COCC2(C(=O)NOCc2ccccn2)C1 75002,c1(C(=O)NCc2ccc(C(=O)NCCc3ccncn3)cn2)c[nH]c(=S)cn1 75003,CC(C)CC(C)N(C(=O)CC1(NC(=O)CCn2cncn2)CC1)CCO 75004,C1(CC)CN(C(=O)C(C)(C)COC)CCC1NC(c1ccnc(C(C)C)n1)=O 75005,Cc1cn(C(C)C)nc1CC(=O)OC(c1ccncc1Cl)C 75006,N1(C(CN(CCOC)C)=O)CCC(CC(C)NC(=O)CC(CC)C2CC2)CC1 75007,c1(CN(CC(F)(F)F)CC)ccncc1C(N1CC(O)CC1C)=O 75008,c1(N(C2CC=CC(C(=O)O)C2)CC)ccc(C2CCCO2)cc1 75009,Cc1ncc(CC(=O)N(CCCNC(=O)C(n2ccnc2C(C)C)C)C)[nH]1 75010,CCCCC(F)C(=O)N1CCC(NC(=O)CC(O)C2CCCC2)C12CC2 75011,C1(C(N(OCC(=O)OCC)C)=O)CC12CC(NC(=O)Cn1ccccc1=O)C2 75012,c1(C(N2CCOCC2c2ccc(Br)cc2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 75013,S(=O)(=O)(c1ccc(=NC2CS(=O)(=O)CC2O)[nH]c1)N(C)CCC1CCCCC1 75014,c12ncncc1OCCN(CCO)C2=O.c1(OCC)ccsn1 75015,c1(N(CC(=C)C)C)nc(=NC)[nH]c(=NCc2nc(C(F)(F)F)n[nH]2)[nH]1 75016,N1(C(C(CC)OCC)=O)CCc2c(CNC(C3(O)CCCC3)=O)cccc2C1 75017,C1(NC(c2cnn3c2OCC3)=O)CC2CCC1(NC(c1ccccc1F)=O)C2 75018,O=[N+]([O-])c1ccn(CSc2ccc(C(=O)NOCCF)cc2)n1 75019,Cc1ccc(CC(=O)NC(CC(N2CC(CS(C)(=O)=O)C2)=O)=O)cc1O 75020,c1(C(N(C2CCN(C(C=CC=CC)=O)C2)C)=O)ccc(C#N)n1C 75021,C1(Oc2c(C(=O)OCC)cnc(C)c2)CCOC2(CCS(=O)(=O)C2)C1 75022,CN1CCOCC1C(=O)NC1(CCC(=O)N(C2(C)CCC2)C)CCC1 75023,C1(N(C)C(C2CCC(N(S(C)(=O)=O)CCO)C2)=O)CCN(C(C23CC(F)(C2)C3)=O)CC1 75024,c1(CC(=O)NC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)(C)C)ccc(=N)[nH]c1 75025,C(C(CC)(CC)C(=O)NC)NC(CC1CC(OCCn2cc(CC)nn2)C1)=O 75026,N1(C(C(CNC(C=C(CC)C)=O)N(C)C)=O)CCS(=O)C(C)C1 75027,c1(CC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)CN(C)C)CC2)c1 75028,Cc1ccc(C(N)=O)cc1C(=O)NCCC(C)NC(=O)CC(c1cc(Cl)sc1Cl)O 75029,c1(C(N(CCCCN(C(C(CCCC)O)=O)C)C)=O)cnc2c(cnn2C)c1N 75030,N1(C(CCCN(C(C(CC)C)=O)CCOC)=O)CCS(=O)CC1C 75031,C(N=c1[nH]c(N2CCC(N(C)C)C2)nc2cc[nH]c12)c1c(SC)n(C)nc1 75032,N1(C(C(CC)CCOC)=O)CCC2(C1)CN(C(=O)C(C)(O)CCN(C)C)C2 75033,C1(NC(c2cn(C)nc2)=O)CC2(C1)CN(C(=O)Cc1cn3ccsc3n1)C2 75034,CCC(CC)(C(=O)NC1CC(C(N2CCC2(C)CC)=O)C12CCC2)OC 75035,C1(CNC(C(C)NC(=O)NC)=O)C(C(=O)Nc2ccc(C(C)F)cc2)CCN1C 75036,c1(C(=O)NC2(C)CN(C(CC(=O)NCC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C 75037,C(=O)(C(C#N)C(C)C)NCC(C(=O)N1CCC(SC)C1)O 75038,c1(C(=O)OC)cccc(F)c1NC(C1CCC(Nc2ncc(Br)cn2)C1)=O 75039,CCCC(C(=O)NC12CCCN(C(c3cccc(O)c3)=O)C1C2)S(N)(=O)=O 75040,N1(C(C(C)OCC=C)=O)CCC2(CC1)CN(C(c1cc(Cl)ccn1)=O)C2C(C)C 75041,C1(O)(C(C)NC(CNC(CCC)=O)=O)CCN(C(=O)CC2CCCOC2)C1 75042,C1(NC(=O)CSC2CC2)CCN(C(=O)C(O)CC(F)(F)F)CC12CCC2 75043,C1(NC(C(CCC)=CCC)=O)CCC2CC1CN2C(c1ncccc1OC)=O 75044,Cc1nn(C)cc1C(O)C(=O)NC1CC(CNC(C2CCCC(C(N)=O)C2)=O)C1 75045,C#CC1(O)CCN(C(C2CCN2C(=O)Cc2ncc(NCC)c(Cl)n2)=O)CC1 75046,Cc1cc(C(=O)N(CCCOCCN(C(=O)CC2CC2(C)C)C)C)nnc1O 75047,C#CCC(C)C(=O)NC1CCCC(NC(=O)C=Cc2cnccn2)C1 75048,c1(OC)cc(C(=O)NCCCCC(C)NC(=O)C(C)NC(=O)C2CC2)ccn1 75049,CC(CN=c1[nH]c(=NCc2cccc(Cl)c2)[nH]c2cnccc12)S(C)(=O)=O 75050,C1(n2cc(CCC)nn2)CCC(NCCCCCF)CC1.C(C)(CCC=O)SC 75051,Nc1nccnc1C(N1CCCC(CNC(c2csc(-c3cn[nH]c3)n2)=O)C1)=O 75052,c1(C(=O)NC2COCC2NC(=O)Cc2csnn2)cc2c(Cl)cccn2n1 75053,C1(NC(Cc2cn(CC)nn2)=O)C=CCN(C(C2(CC3CC3)CC2)=O)C1 75054,C(=O)(C(C)(C)CCOC)NC1COCCC1N(C(=O)CCCOC(C)C)CC 75055,C1(C(=O)NC2(CNC(CCC(=O)N(C)C)=O)COC2)CCc2cc(Br)ccc2O1 75056,c1(OC)n[nH]cc1C(=O)NCC1(O)CN(C(=O)C(F)CC2CCCCC2)C1 75057,c1(CN(C)C(c2cn(CCNC(C3(C)CC(=O)C3)=O)cn2)=O)ccn(C)n1 75058,C12(NC(CC3CC(SC)C3)=O)CCN(C(c3nc(C)ccc3F)=O)CC1C2 75059,c1(C(=O)NCCC2CN(C(c3ccccc3)=O)CC(C)O2)cccc2nncn12 75060,CCCC(C)N=c1nc(N2CCC3CCCCC3CC2)c2c(F)cccc2[nH]1 75061,Cc1ccc(-n2cccn2)c(-c2csc(C(=O)NCc3sccc3Cl)n2)c1 75062,C1(C)(CNC(C(CCC)C)=O)CC(F)(F)CN1C(=O)C(CC)Nc1ccccc1 75063,c1(C(N2CC(NC(c3n(CCCC)ncc3)=O)C(C)C2)=O)nn(C)c(=O)cc1C 75064,Cc1ccccc1CN(C(=O)C(O)CCNC(=O)C=CCCC(C)C)C 75065,C(N=c1ccnc(NCC2C3CCCOC23)[nH]1)c1n(C)ncn1 75066,C#Cc1ccc(NC(C2CCN(C(=O)c3ccccc3C)O2)=O)c(C)c1 75067,c1(C(=O)NCC(C)CNC(=O)Cc2nccn2C(C)(C)C)cccn2ccnc12 75068,N1(CC(=O)NCC(=O)NC(C2CCOC2)C#C)CC(C(F)(F)F)CCC1=O 75069,C1(C#N)(C(=O)NC(C)CNC(=O)CCC(=O)c2ccc[nH]2)CC2(CC2)C1 75070,c1(-c2ccc(C)o2)ccc(S(=O)(=O)N2CCCC2C(O)Cc2ccccc2)cc1 75071,N1(C(c2ncc(C(=O)OC)nc2)=O)CCC2(C1)CN(Cc1ccc(Cl)cc1F)C2 75072,c1(C(=O)OC)ccc(Br)cc1Nc1ccnc(-c2ccoc2)c1 75073,CCC(CN=c1[nH]c(=NCCCOCC(F)(F)F)[nH]c2cc[nH]c12)C(N)=O 75074,n1(COC)ccc(C(=O)NCC(C(C)C)NC(C2CCCN2C(=O)OC(C)C)=O)n1 75075,c1(C(=O)NCC=CCC(=O)N(CCC)Cc2ccnn2C)cccc(F)c1C 75076,N1(C(c2cncc(Br)c2)=O)CC(O)C(O)CC12CCOCC2.n1(O)cccn1 75077,N1(C(CC(CCC)CC)=O)CCOC2(CCCN(C(=O)Cn3cnnn3)C2)C1 75078,c1(C(C(=O)NCc2ccccc2)c2cccs2)cccc(F)c1.C12CCCN1C2=O 75079,C1(NC(C(C)OC2CCCC2)=O)CN(C(=O)CC2CCC(N(C)C)CC2)CC1O 75080,S(=O)(=O)(CC(=O)N1CC(CCNC(C2CCCN2C2CCCC2)=O)(OC)C1)NC 75081,N1(C(C(C2CCC2)NC(c2cc(C)nn2C)=O)=O)CC2CC2C2CC12 75082,CC(CC(C)(C)C)C(=O)NC(COC(C)C)C(=O)N(C)CC1CCOC1 75083,c1(C(=O)NC2C(N=[N+]=[N-])CN(C(=O)CCNC(N)=O)C2)cncc2cnccc12 75084,Cc1nc(O)c(C(=O)NC(C)CCCCNC(=O)Cc2cccnc2O)nc1C 75085,N#CC1CCCC(CC(=O)NCCCCC(CO)NC(c2ccc(CO)o2)=O)C1 75086,c1(C(=O)NC2C(NC(C=CCOC)=O)CCCC2)ccc(N)cc1C 75087,N1(C(=O)NCc2cccc(NC(C3CCCC3)=O)c2)CCOC2CS(=O)(=O)CC12 75088,N(C1COCc2ccccc21)C(Cc1c(NC(C(C(C)(C)C)O)=O)cccc1)=O 75089,c1(C(=O)NC2CN(C(CN(CCC)C)=O)C(C)C2)ccc2c(c1)S(=O)(=O)NC2 75090,N(C1CCCc2cc(C3CC3)ccc21)C(COC)=O.C12CCC(CC1)CNC2=O 75091,S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3COC(C4CC4)C3)=O)C2)=O)c1)NCC 75092,n1(CC(=O)N(CCNC(=O)C(F)(F)COC)CC)nc(C)c2cccnc12 75093,N1(C(C)=O)CCC(C)(NC(C2(C)CCN(C(=O)CCN3CCNC(=O)C3)C2)=O)C1 75094,c1(C(=O)NCC(C)N(C)C(c2cccc(N)c2N)=O)cc2sccc2cn1 75095,c1(C(=O)NC2CC(CNC(c3c(C)nccc3)=O)C2)cn2ncccc2n1 75096,C1(CN(C2CCCN(C(c3ncccc3F)=O)C2)C)CN(C(=O)N)CCO1 75097,c1(CC)cc(C(N2C3CCC2(CNC(=O)C(C)C(C)C)CC3)=O)cn(C)c1=O 75098,c1(C(N2CC(O)(CNC(C(CC)C#N)=O)C2)=O)cn(C)c2ccccc12 75099,N1(C(c2c(OCC)nccc2)=O)CC2(CCCN(C(=O)CN(C)C3CC3)C2)C1 75100,N1(C(CCCOCC)=O)CCC2CC12C(N1CC(c2nn[nH]n2)C1)=O 75101,C(=O)(C(CO)C(C)(C)C)N1CC(NC(C(C)(C)SC)=O)(CO)C1 75102,C1(CC(N2CC3C(CNC(CCC(C)OC)=O)C3C2)=O)CN2CCN1CC2 75103,c1(CC)nccnc1C(=O)NC1CC(C(=O)NC(c2ncccn2)C)C1(C)C 75104,C1(C2CCN(C(c3ccccc3Cl)=O)C2)(NC(=O)Cc2ccno2)CC1 75105,C1(C(N2CCN(CCNC(CC3(C)CCC3)=O)CC2)=O)CCCS(=O)(=O)N1 75106,Cc1nc(NC(=O)CCC2CCCN2c2nnco2)cnc1Br 75107,C1(C(=O)NCC2CCCN2C(=O)CNC=O)C2CN(c3nnc(C4CC4)s3)CC12 75108,c1(C(N(C(CNC(c2nocc2CN(C)C)=O)C2CC2)C)=O)cncn(C)c1=O 75109,CC(C)(C(=O)NCC12CC(C(N)=O)(C1)C2)C1CCCO1.C12CC(C1)C(=O)N2 75110,c1(C(=O)NC2C(NC(c3cc[nH]c3)=O)CC2)cc(CC2CCC2)on1 75111,N1(C(CCC2(CCC#C)N=N2)=O)CCN(CCNC(=O)C(C)C#N)CC1 75112,CC(C(=O)N1CC(O)(CN(C)C(C2CCCC(C)C2)=O)C1)C(F)F 75113,CC1CN(C(=O)CCN(C)C)CCC1N(C)C(C1CCCO1)=O 75114,C(N=c1ccnc(N2CC=C(Br)CC2)[nH]1)c1nn(CC)c(C2CC2)c1 75115,CC1CC(=O)NC1C(N1CC(CO)(NC(=O)C(C)NC=O)C1)=O 75116,C(=O)(C1CCCc2ncc(C)n21)NC1(CC)CN(C(c2cc(C)sc2C)=O)C1 75117,C12(C(=O)NC3(CN(C)C)CC3)CC(CO1)N(C(=O)Cc1ccncc1F)C2 75118,CS(=O)(=O)c1cnc(NC2CCN(C(=O)NCc3coc(C(F)F)n3)C2)c(Cl)c1 75119,Cc1cccc(S(=O)(=O)F)c1NC(C1CC(F)CN1C(=O)C(C)(C)C)=O 75120,Cc1cc(C(N2CC3(C2)CN(C(c2cc(CO)n(C)n2)=O)C3)=O)cc(O)n1 75121,N1(C(C2CCC(CC)O2)=O)CCC(C(C)NC(C2CSCC(=O)N2)=O)CC1 75122,c1(OC)cc(CCC(=O)NC23CC(C2)N(C(C2CCC4(CC4)C2)=O)C3)ccc1Cl 75123,C(CC(C)C)(C(=O)NC(C)CCN(C)C)NC(CC=CCCCCC)=O 75124,Cc1cccc(C)c1C(=O)NC1CCCN(C(c2cnc(C3CCC3)s2)=O)CC1 75125,C1(C(F)F)(NC(C(C2CC2)OC)=O)CC(NC(=O)CC2CCCOC2)C1 75126,CCCCCCCCC(=O)N1CC(O)(C(C)NC(=O)CCCOCCN(C)C)C1 75127,CC1(C)CCC(C)(NC(C2CCCN(C(c3[nH]nnc3C3CC3)=O)CC2)=O)C1 75128,c1(C(=O)NCC2(NC(C(F)OC)=O)CC(OC)C2)cccc(Cl)c1N 75129,c1(C(=O)NCC(=C)CCNC(C2(NC(C)=O)CCCC2)=O)ccc(F)c(C#N)c1 75130,c1ccc(C(=O)NNC(=O)NCC)cc1O.c1nc(CCN2CCCCC2)no1 75131,c1(CC(N2CCC(CCC(=O)NC3CC(CC)C3)C2)=O)coc2ccccc12 75132,C(=O)(CC(C)CC(F)(F)F)NC1COCCN(C(c2c(OC)ncc(F)c2)=O)C1 75133,C1(NC(C=C(C)C)=O)CC(C)CN(C(c2cc(C)cc(O)n2)=O)C1 75134,C(CC(C(=O)N1CCC(O)(C(C)CNC(=O)CSCC(N)=O)C1)N(C)C)SC 75135,c1(OC)c[nH]c(C(N2CCC(NC(c3nc(Cl)sc3C(C)C)=O)C2)=O)cc1=O 75136,N1(C(C(F)=CCC)=O)CCC(CNC(c2ccoc2)=O)C(CC)C1 75137,c1(CC)nc(=N)[nH]cc1C(N1CCC(CF)(NC(c2cnns2)=O)C1)=O 75138,C1(C)(C(=O)NCCCCNC(CCN(CCCOC)C)=O)CC(C(F)(F)F)C1 75139,C(=O)(CC(CCCC)NC(c1ccoc1CC)=O)N(CC(=C)Br)C 75140,N1(C(C(C)n2cncn2)=O)CC2CCN(C(C3CCCCC3(C)C)=O)CC2C1 75141,C(=O)(C(F)(F)C(O)C1CC1)NC(C1(O)CCN(C(C2CCC3(CC3)C2)=O)C1)C 75142,C(=O)(C(C)(CC)C(N)=O)N1CCCC(CNC(C2(CCCC)CCC2)=O)(CO)C1 75143,C1(NC(C2CN(CC(C)C)C2)=O)(CF)CCN(C(=O)CCc2ccoc2)C1 75144,CC1(C)CN(C(=O)Cc2csc(Cl)c2)CC1NC(=O)CC1CCOC1=O 75145,C1(NC(CCNS(C)(=O)=O)=O)CCC2(CC1)CC(NC(=O)C=CC1CC1)C2 75146,C1(CC)C(C)CCCN1C(c1cnc(C)cn1)=O.C(C(C)(C)n1cccn1)OCC 75147,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CCC2)C(NC(=O)C(C)Cc2ccco2)C1 75148,N1(C(c2oc(C)c(Br)c2)=O)CCC(NC(C2CC3CCC3C2)=O)C12CCC2 75149,c1(OC)cncc(C(N2CCC(C(N3CCC(F)(CO)C3)=O)(OC)C2)=O)c1 75150,CC1CCN(C(c2cscc2C(N)=O)=O)CC1NC(c1ccoc1)=O 75151,N1(C(c2nc(C)n(C)n2)=O)CCCN(C(=O)C(C)C(F)(F)C(F)F)C(C(C)C)C1 75152,Nc1cc(Cl)nc(C(N2CC(NC(=O)CN3CCC(O)CC3)C2)=O)c1Cl 75153,c1(CC)cc[nH]c1C(=O)NC(CN(C(=O)CC1(C)CC1(Cl)Cl)CCOC)CC 75154,CC1CC(NC(c2cc(=O)cc(Cl)[nH]2)=O)CN(C(=O)COCC2CCCCC2)C1 75155,Cc1cc2ncc(C(=O)NC3CCCC3NC(c3ncccc3F)=O)c(C)n2n1 75156,c1(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CC2)cnc2ncccc2c1 75157,N1(C(C(CC2CCOCC2)NC(CCC=C(C)C)=O)=O)Cc2ncsc2C1 75158,C1(CC)CN(Cc2cc(O)ccc2Cl)c2ccccc2O1 75159,N1(C(CC(C)(C)F)=O)CCCC(O)(CNC(c2ccc(C(C)(F)F)cn2)=O)CC1 75160,N1(CCCCOC(C)C)CCc2ccccc2C1CNC(=O)CN(S(C)(=O)=O)C 75161,N1(C(C2(CCC)CC2)=O)CCCC(CCNC(=O)Cc2ccc(C)cc2)C1 75162,CN1CCN(CCc2nc(-c3cc[nH]n3)n(CC3CCCC3(F)F)n2)CC1 75163,c1(C(=O)NC2(C3N(C(C(C)OCC)=O)CCC3)CC2)ccc(CC)c(O)c1 75164,n1(C(N(C(C)C)CCNC(=O)C2CC2)=O)cc(-c2ccccc2)nn1.C(=O)(C)O 75165,N1(C(CC(C)F)=O)CCC(C)(CCNC(c2c[nH]nc2F)=O)CC1 75166,C1(C(N(C2CCCN(C(=O)COC(C)=O)C2)CC)=O)CCc2nc(=N)[nH]cc2C1 75167,N1(C(=O)CCN(c2ccccc2)CC)CC2CC1CCC2NC(=O)CCC1CCC1 75168,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75169,C1(C(N2CCC(NC(C(CC)(C)C)=O)C2)=O)(Cc2cccc(Cl)c2)CC2(CCC2)C1 75170,c1(C(=O)NCCNC(=O)C(O)C2CC2)ccn(-c2ccncc2)n1 75171,c1(N(C(CNC(C(C)CC(F)(F)F)=O)C)C)nc2c(cc1C#N)CCC2(C)C 75172,N1(C(CCC(C)SC)=O)CC(CNC(=O)CCN2CCCC2=O)CC(C)C1 75173,CC1CCC(C)(C)N1C(C1CC(OC)C1)=O.C12(CCC1)C(=O)NC2 75174,C(=O)(CC1=NNC(=O)C1)N1C(CNC(C(C)Cc2cnn(C)c2)=O)CC1 75175,N1(C(c2c(CC)non2)=O)CCOC(C(=O)NC2(C)CCC2)C1 75176,CC(C)CC(CNC(=O)CCc1cccnc1)NC(c1cccc(C(N)=O)c1)=O 75177,CC(C)CCN=C(NCc1ccc(N(C)C)nc1)NCC1(C)CC1(Cl)Cl.C(=O)N 75178,c1(C(N2CC3(CCN(C(C4(OCC)CCC4)=O)C3)C2)=O)nc2nccc(C)n2n1 75179,C(CN=c1cc(-c2cccs2)nc[nH]1)OCCN(C(=O)CN1C(=O)CCC1=O)C 75180,c1(OC)cc(NC(=O)CC23CCCC2C3)nc(N2CCCCC2CCSC)n1 75181,Cc1cc(NCCc2cnsc2)nc(=NCC(C)(C)CCN2CCCC2)[nH]1 75182,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75183,N1(C=O)CCC23CCCCC2(C1)C3(F)F.O=C(NNc1ccccc1C(F)(F)F)OC 75184,c1(NC(N(C2CCCCO2)CC#C)=O)ccc(S(=O)(=O)CC)cc1 75185,C12C3CC3CN1C2=O.C(C)(CCCSC)NC(COCCCOC)=O 75186,C1(NC(C(COC)C)=O)CCC12CCN(C(=O)CC1Cc3ccccc3O1)CC2 75187,CC(CS(C)(=O)=O)C(=O)N(C)CC1CCCN(C(c2csnn2)=O)C1 75188,C1(CNC(CCCN(C)C)=O)CN(C(c2cc(O)nc(O)n2)=O)C2CCCC2O1 75189,Nc1cnc(C(=O)NCC(C2CC2)NC(C23CCC(CO2)C3)=O)c(Cl)c1 75190,C(=O)(CC(C)C(C)(C)C)N1CC(C(C)NC(=O)Cn2cnnn2)C1 75191,CC1CN(C(=O)C(C)CNC(=O)Cc2cnsc2)CC(C)(C)C1 75192,C1(NC(COCC)=O)CC2(C1)CN(C(=O)CSc1ccc(Br)cc1)C2 75193,c1(C(=O)NCC2N(C(C=Cc3cccc(C)c3)=O)CCC2)cc2c[nH]cnc-2n1 75194,Cc1cccc(C(CNC(=O)CCCn2ccnc2C)NC(C2CCO2)=O)c1 75195,C(=O)(CC(O)CC(C)C)NC1C(SC)CN(C(=O)CCCC(F)F)C1 75196,c1(CC(C)C(=O)NCC(C)(O)CNC(=O)Cc2nc[nH]n2)ccccc1F 75197,C12(CNC(C(C)(C)SC)=O)CC(CCO1)N(C(=O)Cn1cnnc1O)C2 75198,C1(CC(=O)NCC=CCNC(c2cnn(-c3ccccc3)n2)=O)C=CCCC1 75199,C(c1cccs1)=C(C)C(=O)N(CCCCN(C(=O)Cc1nnc(O)s1)C)C 75200,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75201,Nc1nc(C(=O)NCC2CC2CNC(c2cc(Cl)ns2)=O)ccc1[N+](=O)[O-] 75202,N1(C(C=C(C)c2cccs2)=O)CC(NC(=O)CN(C)C2CC2)CC12CCOC2 75203,Cc1nnc2n1CCC(C(=O)NCC(O)CNC(c1nnn3c1CCC3)=O)C2 75204,N1(C(C2CC(CCC)C2)=O)CCCC(NC(=O)C(c2cccc(OC)c2)O)CC1 75205,C1(NC(C2(CC)CN(C(=O)Cc3ncccc3F)C2)=O)CC2(CCCCO2)C1 75206,c1(OC)cc(=O)n(C)cc1C(=O)NCC1(F)CN(C(C2CC3CCC(C2)C3)=O)C1 75207,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75208,N1(C(CC2N(C)CCCC2)=O)CC2CCCC1C2CNC(=O)CCCC1CCC1 75209,N1(C(CSCC#C)=O)CCC(CNC(c2cc(C(F)F)nn2C)=O)C(O)C1 75210,C1(NC(CCc2ncn(C)c2)=O)CC2CCC1(NC(c1occ3c1CCC3)=O)C2 75211,C1(C(=O)NC(C2CN(C(=O)C(n3ccc(C4CC4)n3)C)C2)C)CCCC1(F)F 75212,c1(CC(=O)NC2C(CNC(C3ON=C(CC)C3)=O)CCC2)ncnc2sccc12 75213,CCCC(C)(C)CC(=O)NC1CC(O)(CNC(=O)C=Cc2ncc[nH]2)C1 75214,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(NC(c2ccnnc2)=O)CC2(CC2)C1 75215,N(C1CCc2ccccc21)C(CC(C)CNC(c1nsnc1O)=O)=O 75216,C1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)(C)C)CCc2n[nH]c(C)c2C1 75217,CS(=O)(=O)C1CC(N(C(=O)C(F)CC2CNC2)CCO)C1 75218,c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1cnc(Cl)[nH]1)=O 75219,C1(CNC(C2C(C)CCC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75220,c1(C(N2CC(N=[N+]=[N-])C2)=O)coc2c1CN(C(=O)CO)C2.C(CCN=[N+]=[N-])CCO 75221,c1(N2CCC(CC(C)F)CC2)nc(N2CCN(C3CCC3)CC2)c2c(n1)CCS2 75222,C(=O)(C(C)(C)COC)NCC12CC(NC(CC)=O)(C1)C2 75223,C1(NC(c2cnn(CCO)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1.CCO 75224,C1(NC(C(C)Oc2cccnc2)=O)CCCCCN(C(=O)CN2CCOC2=O)C1 75225,N1(C(C2CCCN(C)C2)=O)CCC2(C=C(C(=O)NC(c3cscn3)CO)C2)C1 75226,Cc1cn2nc(C(N3CC(NC(c4n[nH]c(C)c4C)=O)C3)=O)cc2c(=O)[nH]1 75227,N1(C(CC2N(CC)CCC2)=O)CCN(C(c2nnsc2C)=O)CC1CCO 75228,CC(C(F)F)N(C(=O)CC=CCN(C(=O)COCC(F)F)C(C)C)C 75229,c1(C(C(=O)OC)NC(C2CCC(C)(C)CC2)=O)ccc(Cl)c(OC)c1F 75230,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75231,Cc1sc(Cl)nc1C(N1CCC(C)(CCNC(c2coc(C3CCC3)n2)=O)C1)=O 75232,C(CN=c1ncc(F)c[nH]1)NC(c1cccnc1C(F)(F)F)=O 75233,c1(C(=O)NCC2C(C)CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)ccnc2ncnn12 75234,Cc1cncc(C=CC(=O)NCC=CCNC(=O)CC2(CO)CCS(=O)(=O)C2)c1 75235,CC(C)C(O)CC(=O)NCCCC1CCCN1c1cc(C2CC2)ncn1 75236,C1(C(=O)NC(C)CC(C)O)(CC)CCCN1C(c1cnc(OC)s1)=O 75237,c1(N(C(CS(C)(=O)=O)=O)CC2CCCNC2)ncnc2[nH]cnc12 75238,C(N=C(NCC(C1CC1)C1CC1)NC1CCOc2ccc(Cl)cc21)C1C(C)C1 75239,C1(NC(CSC)=O)CCCCC1NC(C1C(CO)CCO1)=O 75240,C12(NC(C3N(C(C(C)CO)=O)CCC3)=O)CCCN(CC1)C2 75241,C1(C(C(=O)NC(C(=O)N(CCC)CCC)c2ccco2)C)CCCCC1 75242,N1(C(c2n(CC=C)ccc2)=O)CCN(C(=O)CC2CCC(C)(C)C2)C(C)C1 75243,N1(c2c(OC)c(C)ncn2)C2CCC1CC(NC(c1cnoc1C1CCC1)=O)C2 75244,c1(C(N(CCN(C(=O)CC(C)C2CCCO2)C(C)C)C)=O)nc2cnccc2s1 75245,c1(C(N(C)CC2N(C(C3CN(CC)C(=O)C3)=O)CCC2)=O)ccc(Cl)nc1OC 75246,C1(C(=O)NC(C)(C)C(C)NC(=O)C(C)N(C)CC)(COCC)CCOCC1 75247,C(=O)(C1SCCc2sccc21)N(CC(C)(C)CNC(=O)CCc1nccs1)C 75248,c1(C(=O)NCC(CNC(c2cccc3c2CCC3)=O)O)ccc2nc(O)[nH]c2n1 75249,C1(C)(CNC(CC(C)CN(C)C)=O)CN(C(=O)CSc2ccccc2F)CCO1 75250,C=CCCCCC(=O)NC(N1CC(N(C(=O)CN2CCC(C)C2)C)C1)=O 75251,C1(NC(N2CCN(C)CC2)CC)CCN(C(=O)CCCc2sccc2C)C1CC 75252,c1(CN2C(CC(=O)OC)CCC2)ccc2ncsc2c1 75253,C(=O)(CC(C)C(F)(F)F)N(CCCNC(=O)C(CC(C)C)c1ccccc1)CC 75254,C1(C(=O)OCC)CCCN(C(=O)CCN(C(C2CCC2(F)F)=O)C2CC2)C1 75255,c1(C(=O)NC2C(NC(CC(C)C(F)F)=O)CCCC2)cc2cc(O)ccc2[nH]1 75256,C1(C)(C(N2CCCC(C(C)NC(C3CC4(CCC4)C3)=O)C2)=O)CCN(C)C1=O 75257,N1(C(=O)Cc2cnns2)CCN(C(C2(O)CCCCCC2)=O)C(CO)C1 75258,c1(CN2CCC(CC(=O)NCc3ccc(Br)c(O)c3)C2)cc2cccnc2[nH]1 75259,C(N=c1[nH]c(N2CCSCC2)nc2c1CCCCC2)c1ccc2c(c1)CO2 75260,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(F)F)nc2c1SCC2)OC 75261,C1(F)(CNC(=O)CCc2ccncc2)CCC(CNC(=O)CC2(F)CCC2)C1 75262,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(=O)COC3CCCC3)C2C1 75263,C1(SCC(N2CCCC(c3cn(-c4c(C)ccs4)nn3)C2)=O)CCCCC1(F)F 75264,N1(C(c2c(C)nsc2)=O)CCCC(CO)(NC(=O)C(N2C(=O)CCC2=O)C)C1 75265,c1(C(=O)NCC2(NC(=O)CC3CC(O)C3)CCC2)ccc(Cl)cc1O 75266,C12(n3cc(C(N4C(C)CN(C(=O)C=CBr)CC4)=O)nn3)CCN(C1)S(=O)(=O)C2 75267,c1(C(=O)NCCC2CC(NC(=O)CC3=CCCC3)C2)c(F)cccc1[N+](=O)[O-] 75268,c1(C(=O)NCCN(C(C2CCCCC2C(N)=O)=O)CC)ccc(OC)nc1Br 75269,C(=O)(C(F)CC(C)(C)C)c1nn(C)c(=O)c(O)c1 75270,N1(C(C(c2ccnn2C)NC(C(CC)O)=O)=O)CCCC(C2CC2)CC1 75271,C=C(C)CC(=O)N(CCC(C)NC(C1CC(OC(F)(F)F)C1)=O)C 75272,C(CC(CNC(c1cnc[nH]1)=O)NC(c1ccoc1)=O)OC 75273,C1(C(=O)NC(C)(CNC(=O)C(C2CCCCC2)O)CO)CCCCS1(=O)=O 75274,Cn1ncc(CCC(=O)NCC2CC(CNC(c3cnn[nH]3)=O)CO2)n1 75275,N12CC3COCC3(C1)C(=O)NCC1(CCC1)C2=O.C1(OC)(COC)CCC(C)C1 75276,c1(CC)c(C(=O)NCCCN(C(=O)C(C)Sc2cccc(F)c2)C)ccn1C 75277,C(=O)(C1=CC2CCC(C1)C2)N1CCCN(C(C2C(C(C)(C)C)C(=O)C2)=O)CC1 75278,c1(C(=O)NC2(C)CN(C(c3n(CC)ccn3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 75279,C1(OC)CC2N(C1)C2=O.c1(C(=O)NC)cn(C2CC2)nc1C.C1(C(=O)N)CCSCC1 75280,C1(OC)CN(C(=O)C(C)(C)N(C)C)C(C)(CNC(c2onc(C)c2C)=O)C1 75281,CN1CCN(C(c2ccccc2C(C)(C)C)=O)C(CNC(c2ccccc2)=O)C1 75282,c1(NC(C(CO)NC(c2cnc(OC)nc2)=O)=O)ccc(C#N)cc1O 75283,S(=O)(=O)(c1nc(N2CCC=C(Br)C2)ccc1Br)N1CCC(COCC)C1 75284,c1(C(N2CC(CNC(C3CN(C4CCC4)C3)=O)C(O)C2)=O)ccc2nccnc2c1 75285,c1(C(N2C3CN(C(C(F)OC)=O)CC2CC3)=O)c([N+](=O)[O-])c(C)nn1C 75286,c1(OCC)nc(Cl)ccc1N(CC(F)F)Cc1ccn(C)c1 75287,CC(C)CC(CNC(=O)CC1(CO)CC1)NC(=O)CC1CCOCC1 75288,C(CN=c1nc(N2CCN(CC(C)F)CC2)c2nn[nH]c2[nH]1)c1nnc(C)s1 75289,c1(C(C(=O)OC(=O)CC2CNC(=O)O2)NC(=O)C(CO)N(C)C)cccnc1 75290,c1(C(N(CCC(C)NC(c2ccc(CCC)s2)=O)C)=O)ccn(C)c1C1CCC1 75291,C(=O)(C1=NN(C(C)C)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75292,C(=O)(C(C)(C)CF)NCC1(NC(c2c(CC)onc2)=O)CCOC1 75293,CCC(C)(CCC(C)C)C(=O)N1CC(O)CC1C(=O)NCc1cccc(Cl)n1 75294,N1(C(C2(CN(C)C)CC2)=O)CC(CNC(=O)CC2CCCO2)OC(C)(C)C1 75295,c1(C(N2CCCC(F)(CNC(C(C)O)=O)C2)=O)cccc([N+](=O)[O-])c1N1CCCC1 75296,C1(CC=C)(C(=O)NCC2(CCO)CCCO2)CCCN1C(=O)C(C)CC#N 75297,c1(NC2(CCCO)CC2)nc2cccnc2c(=NC(C)C2CCCO2)[nH]1 75298,Cc1cc(C(=O)NC2C3CC(NC(=O)C(C)Cc4cnn[nH]4)CC23)nc(C)c1 75299,N1(C(C2CCC(C)C2)=O)CCN(C(C2CCCCN2C(N)=O)=O)CC1CCO 75300,C12CCOC(C1)CCC(=O)N2.C1(CNC2C(C(=O)OC)C2(C)C)CCCC1C 75301,N1(C(c2noc(CCCC)n2)=O)CCC(F)C(F)C1 75302,N12CC(CCC1C)C2=O.c1(C(=O)OC)sccc1CNC(=O)COC 75303,C1(C(C)NC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2cnn[nH]2)=O)CCO1 75304,c1(C(N2CCCC(CNC(=O)OCC)C2)=O)cccc2c1CCC(=O)N2 75305,S(=O)(=O)(c1cnc(N(C)CC2(CC)CCC2)cc1C)NCCOc1cncc(Cl)c1 75306,N1(C(=O)CC2(O)CN(C(=O)C(F)(F)F)C2)CC2CCN(C(=O)C3=CCCO3)C2C1 75307,C(=O)(C#CC1(C)CC1)NC(CNC(CCC(=O)NCC)=O)CO 75308,c1(CC(=O)N(CCCN(C(C(C(C)C)(C)C)=O)C)C)ncn2c1COCC2 75309,c12noc(n1)CN=C(NC(c1nc(C)cs1)C)N2.C1(COC)CCCC1 75310,C1(O)(CNC(c2ccc(C(N)=O)cc2)=O)CCCN(C(C2(Cl)CC2)=O)C1 75311,C(CCCCCC(=O)N1CCC(C(C)O)C1)NC(c1ccc(CC)o1)=O 75312,N1(C(c2cncc(CNC(C3C(C)OCCC3)=O)c2)=O)CC2(CCCC2)C1 75313,C1(CNC(C2C(CC)C2)=O)CC2CCC(C1)N2C(c1sccc1-n1cccc1)=O 75314,Cc1ccc(CC(N2CCCC(C(=O)NC3(C)CC(C(F)(F)F)C3)C2)=O)c(Cl)n1 75315,C(=O)(C(C)CCCC)NC(C1OCCN(C(CCC(=C)Br)=O)C1)C 75316,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(CCn2c(C)csc2=O)=O)C1 75317,c1(C(N2CCC3(NC(c4cc(C)cc(F)c4)=O)C(C2)C3)=O)ccc2nc[nH]c2c1 75318,c1(OC(CNCCO)OC)ccccc1.C1CCS1 75319,Cn1cnc2c(C(N3CC(NC(c4cc(Cl)cnn4)=O)CC3CO)=O)ccnc12 75320,N1(C(c2c(CC)occ2)=O)CCCC(CCNC(=O)CS(=O)(=O)C2CC2)CC1 75321,Cc1c(NCCCCCC2CCCC2)ncnc1N1CC(OC(F)F)C1 75322,C1(CNC(c2cccc(C)c2)=O)N(C(=O)Cc2n[nH]c(C)n2)CCC1(C)C 75323,c1(C(=O)NC(CC)CNC(c2cc(CO)[nH]n2)=O)cnccc1C1OCCO1 75324,Cc1ccn(C(C)CC(=O)N(CC(C)NC(C2CCCSS2)=O)C)n1 75325,N1(C(C(C)OC2CCOCC2)=O)CC2CC1CCN2C(=O)C1=COCCC1 75326,c1(OCC)ncccc1C(=O)Nc1cccc(NC(C2CC(C)(F)C2)=O)c1 75327,Cc1ccc(CC(NCC(O)Cc2ccc(Cl)s2)Oc2cccnc2)cc1 75328,c1(CNC(=O)Nc2cc(C(=O)OC)c(O)cc2)c(C)nc(C)nc1C 75329,Fc1ccc(F)c(CNc2ccc(N3CCCC(C(F)(F)F)C3)cc2)c1Br 75330,Cc1cccc(C(=O)CCC(=O)N2CCC(NC(C3CC3F)=O)C2C)c1 75331,c1(NC(CNCc2cnc(C)s2)=O)cccnc1I 75332,C1(OC)CCCC1C(=O)N(CC(F)(F)COC)C 75333,c1(N(c2n(CCCCC)c(-c3scnc3C)nn2)C)ccc(OCC)c(Cl)c1 75334,CCCC(CC)CCC(=O)N1CCOC(CN(C)C(c2ccnn2C)=O)C1 75335,N1(C(C2C(C)C2)=O)CC2CC1C2C(c1ccccn1)NC(=O)CSc1ccccc1 75336,C1(C(N2CC(NC(=O)C(F)Cl)C(F)CC2)=O)CCc2ccccc2C1O 75337,C1(NC(c2n(CC)ccn2)=O)COC2(CNC(C3(C(F)F)CCCC3)=O)CC1C2 75338,C1(CN(C(=O)CC2CCCSC2)C)CCN(C(c2nnsc2N)=O)CC1 75339,C1(C(=O)NCC(C(C)(C)C)OC)CCCCCCN1C(=O)C=CC1CCCC1 75340,c1(OC)cc(Cl)c(C(N2CC3CN(C(C4CCCCO4)=O)CC3C2)=O)cc1C 75341,c1(C2C(CC(=O)NC)C2)ccccc1NCC(C)(C)n1cccn1.C(C)(C)O 75342,N1(C(CS(=O)(=O)NC)=O)CCN(C(C2CC(=O)C23CCCC3)=O)CC(C)C1 75343,c1(NC)ccccc1C(N(CC(C)NC(C)(C)C(C)NC(=O)C(=O)N(C)C)C)=O 75344,N1(C(c2ccc(C)cc2O)=O)CC(F)(F)CC1(C)CNC(=O)C(C)C(C)(C)C 75345,Cc1ccccc1C(C)CC(=O)NC1CN(C(=O)C=Cc2csc(Br)c2)C1 75346,C(CC1=CCCCC1)C(n1cc(CC(C)(C)C)nn1)C1CCCN1C.[SH](C)(=O)=O 75347,c1(C(C)C)cc(C(=O)N(C)CCn2cc(-c3cc[nH]c3C3CC3)nn2)n[nH]1 75348,c1(NCCSC2C(NC(=O)Cc3ccns3)CCCC2)ncnc2c1CCC2 75349,c1(C(=O)NCC23C(CN(C(C(C)NC(N)=O)=O)C2)C3)cn(C)c(=O)n1C 75350,C1(CC(=O)N(CCN(C(=O)CC(C)n2cccc2)CC)CC)CCCC(F)(F)C1 75351,Cc1c(C(N2CC(C3(NC(=O)CSCCN(C)C)CC3)C2)=O)cncc1Cl 75352,N1(C(COCC#C)=O)CCC2OCCN(C(c3cc(C)cnc3C)=O)C2C1 75353,C(CCOCCO)(C(=O)OCC1CN(C)CC1C)NC(C(=O)NCC)=O 75354,N1(C(CCCCNC(N)=O)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 75355,CC(CF)CC(=O)N1CCC(N(C)C(c2ccc(CCN(C)C)cc2)=O)C1 75356,Cc1nc(C)n(CC(N2CCC(C(=O)N(C3CCC3)C3CC3)C2C(C)C)=O)n1 75357,C1(CC)CCCN(Cc2ncc(NC(=O)OC(C)(C)C)s2)C1C 75358,C1(C(N2CCC(NC(C3CN(C4CCOC4)C3)=O)(CO)C2)=O)CN2CCC1CC2 75359,C1(CNC(C=CC)=O)(OC)CCN(C(=O)CCOC(=O)Nc2ccccc2)C1 75360,C1(C(N2CC(CC(C)C)OCC2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)C1 75361,c1(C(=O)NCC(C)N(C(=O)C=CC)CC)[nH]nnc1C1CC1.c1(S)ccnn1C 75362,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCN(C(=O)CCCOC(C)C)C(CO)C1 75363,N1(CC(=O)NCC2CCC(NC(c3cnc(C(F)F)s3)=O)C2)CCCOC1=O 75364,C#CCC(CC(=O)NCCC1CCCO1)NC(C1(C)C=CCCC1)=O 75365,Cc1n[nH]c2cnc(C(=O)NCC(C)NC(C3(O)CCCCC3)=O)cc12 75366,S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)NC(C(=O)Nc1c(C(N)=O)noc1)=O 75367,Cc1cc(Br)c(F)cc1NC(C1CC1C(N1CC2C(C1)C2(C)C)=O)=O 75368,C1(C(=O)NC2(C)CCN(C(Cc3cc(OC)ns3)=O)C2)CCC(C2CC2)CC1 75369,c1(C(=O)NCCCC(C)NC(C2CCCO2)=O)ccc(C(=O)N(C)C2CC2)cc1 75370,Cc1ccc(C(=O)NC2CCC2NC(=O)Cc2cccc(C(F)(F)F)n2)cc1 75371,c1(C(=O)NCC(C)NC(C=CC(C)(C)SC)=O)cc(C2CC2)n(C)n1 75372,n1(CCOC(C)Cc2ccccc2)cc(-c2cccs2)nn1.C1(=O)CN1 75373,CC1CCCC(C(=O)NCCCCN(C)C(c2ccc(SC(F)F)cc2)=O)C1 75374,N1(C(CC)=O)CC2CCC1CN2C(=O)CCc1cc(F)c(F)c(F)c1 75375,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75376,C=CC(C)(C)C(=O)N(C(C)CNC(C1CC1C#N)=O)CC 75377,c1(C(=O)NC(CCCNC(c2nn(CC)c(=O)cc2)=O)C)cc[nH]c2nccc1-2 75378,C1(NC(CCC2C(C)(C)C2)=O)CCC(C(=O)NCCN=[N+]=[N-])CC1 75379,C1(C(=O)NCC2N(C(C(C)OC3CCCC3)=O)CC2)CCCN1C 75380,c1(C(N2CCC(NC(C(F)=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75381,c1(C(N(CCC)CCNC(C2(C)CCCC2)=O)=O)ccc(SCC#N)cc1 75382,Cc1cccc(C(N2CCN(C(=O)C(c3ccccc3)O)CC2)=O)c1C#N 75383,N1(C(C(C(C)C)SCC)=O)CC(C)(CNC(=O)COCCCF)CC1(C)C 75384,C1(C)(C(N(C2CCCC2)CC(N2CC(OCC(C)C)C2)=O)=O)CCCNC1=O 75385,N1(C(C2C(C)CC2)=O)CCN(C(C2CC(O)(c3ccccn3)C2)=O)CC1C(F)F 75386,C(=O)(CC(COC)NC(C1(C)CC1(F)F)=O)N(CC(O)CF)CC 75387,CC1(NC(C2CCO2)=O)CCN(C(c2c[nH]nc2-c2ccco2)=O)CC1 75388,S(=O)(=O)(c1ccc(CN2CC3(CCC3)C2c2ccccn2)cc1)NC(C)C 75389,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(COC(C)=O)=O 75390,C1(C(=O)NCC2(CNC(c3cnoc3)=O)CC2)CCCN1c1ccccc1 75391,Cc1cc(C(=O)NCCSCC(=O)NCCCOC(F)(F)F)c(C)[nH]1 75392,CC(C)(CCCN=c1nc[nH]s1)NC(C1CCC2CC2CC1)=O 75393,N1(C(c2cccc(CC)c2)=O)CCCN(C(=O)C=Cc2cncc(F)c2)C(C)C1 75394,C1(NC(c2c(CC)cccc2)=O)CN(C(=O)CC(C)CCC)CC12CC2 75395,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75396,c1(C(N(C(=O)Nc2c(C)nn(C(C)C)c2)C)C)ccc(Cl)c(C(F)(F)F)c1 75397,Cc1n[nH]c(C)c1CC(C)C(=O)NC1CC(C)(CNC(c2ncn(C)n2)=O)C1 75398,C1(C(N(C(C)C(=O)NCC2CCC=CCC2)CCC)=O)CC2(CCC2O)C1 75399,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cnnc3C2)cc(Cl)c(O)cc1C 75400,C1(O)(CCNC(C2(F)C(C)C2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75401,c1(C(N2CCN(C(CCC=C)=O)CC2C)=O)ccc2ccccc2c1Br 75402,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75403,Cc1csc(C(=O)NCC(CO)NC(C2(n3cc(Cl)cn3)CC2)=O)c1 75404,N1(C(c2c(C)nns2)=O)CC(NC(C2CSCN2C(C2CCC2)=O)=O)C2CC2C1 75405,c1(C(N(CC(CNC(c2nn(CC)c(C)c2)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 75406,c1(C(N2CCC(CC)C2CNC(C2CCN(C)C2=O)=O)=O)cc2cnn(C)c2s1 75407,C1(C(N(CC(C2(O)CN(C(C34CC5CC3C4C5)=O)C2)(C)C)C)=O)CCC(C)(C)C1 75408,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)CCc1ccon1)C2 75409,c1(C(=O)NC(C(C)NC(c2c(Cl)ccc(C)c2)=O)C)cccc2cnnc(O)c12 75410,c1(CCC(N2CCN(C(C3C(=C)C3)=O)CC2CCO)=O)c(C)oc2ccccc12 75411,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CC(F)(F)F)[nH]n2)=O)cc2n(n1)CCO2 75412,C(=O)(C1CCc2nccn21)N1CCC2C(C(=O)NC3(CC=C)CCOCC3)C21 75413,c1(C(N2C3C(NC(Cn4c(C)cnn4)=O)C(C3)C2)=O)cc(C)c(F)cc1F 75414,C1(C(=O)NC2(CC(=O)OC)CCOCC2)CN(C(=O)C(COC)OC)C(C)(C)C1 75415,c1(C(=O)NCC2CCN(C(=O)CSc3ccccc3Br)C2)cnn2c1CCC2 75416,c1(C(N2CC(F)CC(NC(CSCC=C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75417,C(=O)(C(O)C1=CCCCC1)N(C1CCN(C(CCCCNC(C)=O)=O)CC12CC2)C 75418,c1(CNC(=O)NCc2ccn(CC(C)C)n2)c(F)cc(I)cc1F 75419,N1(C(c2oc(CC)c(C)c2)=O)CCC2(CC1)CC2CNC(c1cscc1OC)=O 75420,N1(C(C=CC=CC)=O)C2CCC1CN(C(=O)Cc1ccsc1C)CC2 75421,c1(NC(C(C(C)C)CNC(C2CCC(=O)N2)=O)=O)ccc2c(c1)COC2 75422,C1(C(N(C2CCC2)C(C)C)=O)CC(C)N1C(=O)CCc1cncnc1 75423,C1(CCNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]nc1Br)=O 75424,C(c1cccc(F)c1F)=CC(=O)NC(C1(O)CCN(c2nnco2)C1)C 75425,C(=O)(CCCCC(C)C)NCC(C)(C1CC1)NC(COc1cccc(CC)c1)=O 75426,c1(OC)cccc(CN2CCC(C(=O)NCc3ccsc3)CC2)c1Br 75427,c1(C(c2n(CC=C)nnn2)NCc2ncc(Br)s2)cc(C)c(OC)c(C)c1 75428,CC12CCC(C(=O)NCCC3(O)CN(C(=O)CC4CCCC45CC5)C3)(CC1)C2 75429,C(CCC(C)C)(C(=O)NC1CCC2CC1CO2)NC(C(C(CC)C)=O)=O 75430,CC1CC(NC(=O)Cc2cnoc2)CCN1C(C1OCCO1)=O 75431,CC(CNC(C1C(C)C1C)=O)C(=O)NCC(c1ccsc1)O 75432,CCC(C(=O)OC)C(=O)N1CCC(NC(=O)CCc2nnc(C(C)C)o2)CC1 75433,N1(C(CC2CC(C)N(C(=O)CN(c3ccccc3)C)C2)=O)CC(=O)N(C)C(=O)C1 75434,c1(C(=O)NC23N(C(=O)CC45COCC(C4)C5)CC(C)(C2)C3)ccc2n[nH]cc2c1 75435,C(=O)(CC1=CCCC1)N1C(C)CC(NC(=O)Cc2ccc(Cl)cn2)C1 75436,c1(NC(=O)NC(c2csc(Cc3c(C)cccc3C)n2)=O)cc(Cl)c(F)cc1I 75437,CC1(C)CC(CNC(c2cn3cnnc3cn2)=O)CN(C(=O)COC2CC2)C1 75438,c1(C(=O)NCCC(C)N(C(=O)C(F)C(F)(F)F)C)cccc2cnccc12 75439,c1(C(N2CCC(CC(=O)Nc3nccc(Br)c3O)C2)=O)cc(F)c(F)cc1O 75440,N1(C(C=CCCC)=O)CC(O)CC1CC(=O)NCC1CC1c1ccccc1 75441,CC1CC(NC(C23CCCC(C2)OC3)=O)CCN1C(=O)COCc1cccnc1 75442,CCC(C)C(O)C(C)C(=O)NC(C1CN(C(c2cccc(C(=O)OC)n2)=O)C1)C 75443,c1(C(=O)NCCN(C(C2CC(=O)N(C)C2)=O)CC)cnc2c(C)cccn2c1=O 75444,N1(C(c2ccc(Cl)nc2C)C(=O)NC)CCC2CCCC(C2)C1 75445,c1(NC2CC(O)(CNC(c3ccc(COC)o3)=O)C2)snc(C)c1C#N 75446,c1(C(N2C(CCNC(C(=O)NC(C)C)=O)CSCC2)=O)ccc2c(c1)OCO2 75447,C1(Cn2c(-c3c(C)c(-c4ccc(O)cc4F)cnn3)ncc2)COc2ccccc2O1 75448,N1(C(c2cncc(Br)c2)C(=O)NCC=C)CC(C)(C)c2ccccc21 75449,CC1C(NC2CC3(CCN3)C2)CCCC1NCCCC(C)(C)C 75450,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCCO2)=O)CCNC(=O)CC1C 75451,c1(C(=O)NCc2c(C(=O)Nc3c(C)nn(C4CC4)c3)con2)ccc(Cl)c(N)c1 75452,c1(NC(C2CN(S(=O)(=O)CCBr)CCO2)=O)c(F)cccc1I 75453,CC1COCCN1C(C1CCCN1C(=O)Cc1ccccc1Cl)=O 75454,CC1=CCSC1C(=O)NC(c1cnn(C)c1)C(=O)NC1CCC(O)C1 75455,C#Cc1cc(C(N2CC(CCO)(NC(=O)C3=C(C)CCCC3)C2)=O)cc(N)c1 75456,C1(NC(C(C(C)C)N(C)C)=O)CC2CC1CC2n1cc(-c2ccccc2)nn1 75457,c1(NC)cnccc1C(=O)NCC1CCCN(C(C2C(C(=O)NC)C2)=O)C1.N(C)C 75458,c1(OC)cc(C(=O)NCC2(O)CC(NC(C3(COC)CCOC3)=O)C2)cc(Cl)c1 75459,c1(C(=O)NC(C)C(C)NC(=O)CCNC(c2ccco2)=O)cc(Cl)ccc1N 75460,N1(C(CN(C2CCSC2)C)=O)CC2CCN(C(c3c(F)ccc(O)c3F)=O)CC2C1 75461,C12(C(=O)NC3CCC(CNC(c4ccc(OCC)s4)=O)C3)CCOCC1C2 75462,c1(C(C(=O)NCC(C)NC(=O)C=Cc2ccoc2)O)ccc(Cl)c(Br)c1 75463,C=CCCCCCNC(=O)C(C)(C)C1CCN(C(=O)C(C)Cn2ccnc2)C1 75464,c1(C(=O)NC2CC3CC(C2)N(C(C2(CO)CC2)=O)C3)cc(Cl)c2[nH]c(O)nc2c1 75465,c1(C(=O)NC2CC(C)N(C(c3ncccn3)=O)CC2)ccc2c(c1)nc(O)n2C 75466,c1(CC(=O)OC)ccccc1CN1CCOCC1CNC(c1cncn1C)=O 75467,N1(C(CSCCCC)=O)CCCCC1C1CCCN1CC(=O)Nc1ccccc1 75468,C(=O)(CC1=CCCCC1)NC1CC(CNC(CC(C)C2CCCO2)=O)C1 75469,CCCCCN(CCC(=O)NCCCO)C.C1(C=O)CN(CCOCC)C1 75470,CC1CCc2[nH]c(=NCC(F)F)nc(N3CCCN(CC(F)(F)F)CC3)c2C1 75471,C(CC(=O)N1CC2(CC2)CC1CNC(=O)Cc1ccno1)(C(C)C)OCC 75472,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75473,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75474,C1(C(=O)NCCN(C(c2cnc(C)cc2Cl)=O)CC)CCC2(CCOCC2)O1 75475,N1(C(C2C(C)CCC2)=O)CCC(CNC(C2CCCCN2C)=O)CC1 75476,c1(CN2CCCC(CC(N3CCN(C4COC4)CC3)=O)C2)c[nH]c2ccccc12 75477,N1(C(C=C(C)C2CC2)=O)CCC2C(C1)NC(=O)CN2C(C1CCOC1C(C)C)=O 75478,C#Cc1ccc(C(N2CCCC(CCNC(C3(CCO)CC3)=O)CC2)=O)nc1 75479,c1(CC)ncc(C(=O)NCc2nc(C)cc(C)n2)c(C)n1.C(CCNC(=O)CN)O 75480,c1(C(N(C(CNC(C(CC=C)CC)=O)C)C)=O)cnc2cc(O)ccc2c1 75481,C(=O)(CCCC1NC(=O)NC1=O)N(C1CC1(C)C)CCOC 75482,C1(NC(=O)C=CCF)CC2CN(C(=O)CCc3ncc[nH]3)CCN2C1=O 75483,N1(C(CSC(C)C)=O)CCCC2C(CCCN2C(C2CC(CF)C2)=O)C1 75484,C(=O)(CCC(C)OC)NCC(=C)CCNC(c1c[nH]c(C(=O)OC)c1)=O 75485,c1(C(=O)NC2C(NC(C3C(C)(C)C3)=O)COCC2)cn2c(n1)SCC2 75486,C1(C)(CC)CC(NC(=O)CCCN2CCCCC2)CN1C(c1n[nH]cc1Cl)=O 75487,Cn1ncc(C(N2CC(NC(=O)CCc3nncs3)C(F)C2)=O)c1C(C)(F)F 75488,C(=O)(C(C)(C(C)C)OC(c1cc(Cl)cc(C(F)(F)F)n1)=O)OCC 75489,C1(CC(=O)N(C)CC2CCC(NC(c3cncs3)=O)CC2)CC2(CCC2)CO1 75490,N1(C(CCOc2c(C)cccc2)=O)CC2CC1CCN2C(C12CC(C1)C2)=O 75491,CCC(CC)C(=O)NCC#CC(=O)NOC1CCCC1 75492,c1(C(=O)NCC2CCN(C(=O)CSC(F)(F)F)C2)c[nH]c2cccnc12 75493,Cc1cc(OC(=O)CC2CCN(CC(F)(F)F)C2)ccc1CN 75494,c1(OC)noc(C)c1C(=O)NCC(C(C)C)NC(C12CC=CC(C1)O2)=O 75495,N1(C(C(CC)(C)OC)=O)CCC(C)(C)C(NC(C2C(C)(C)OC2(C)C)=O)C1 75496,C(=O)(C#CC(C)C)NCCC(=C)CNC(=O)C(C)(C)NC(c1ccc(SC)s1)=O 75497,C(=O)(N=c1cc[nH]c(CCO)c1)C1N(Cc2cc(C)[nH]n2)CCC1O 75498,C#Cc1ccc(C(=O)NC(C(=O)NOCC(C)(C)CO)C2CCC2)cc1 75499,C#CCC(C)C(=O)Nc1ccc(C2CCN(C(=O)CC3(CO)CC3)C2)cc1 75500,c1(COC)cc(C(=O)NCc2nc(CNC(=O)CC(C)F)cs2)cs1 75501,C12(c3onc(C(N4C(CS(N)(=O)=O)CCCC4)=O)n3)CCC(CC1)CC2 75502,C1(NC(CCC=C)=O)CCCCC1NC(C1C(F)(F)C12CC2)=O 75503,N#CCCCCCC(=O)NCc1cc(C(N2CCSC3CCCC23)=O)cs1 75504,c1(C(N2CCCC(C)C2CNC(=O)CC2C=CCCC2)=O)cc2cccnn2c1 75505,C1(OC)CCN(C(=O)CC(C(C)C)NC(C2CCCN2C2CC2)=O)CC1(C)C 75506,c1(C(C(N2C(C)CC(NC(c3cnc(Cl)s3)=O)C2)=O)=O)c[nH]c2ccc(F)cc12 75507,c1(CNCC2N(C(C(c3ccccc3)N(C)C)=O)CC2)ccncc1Br 75508,Cn1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)c(C2CCCCC2)n1 75509,C12(CC)CN(C(c3cc(C)nc(O)c3)=O)C(CNC(=O)Cc3nonc3C)(C1)C2 75510,N1(C(C2CC(C)C2)=O)CCN(C(=O)Nc2ncnc3ccccc23)C2(CCC2)C1 75511,c1(C(=O)NCC(CN(C)C(C2CCSCC2)=O)O)ccc2c(O)nnc(O)c2c1 75512,Cc1nccnc1C(=O)NCC1CC(CNC(c2csnn2)=O)C1 75513,C12(C(N(C3CCCN(C(C45CC(C)(C4)C5)=O)CC3)C)=O)CCCCC1C2(F)F 75514,CC(C)(C)CC(F)C(=O)NN1CCCC(O)C1.c12c[nH]nc1C(=O)NC2 75515,C=Cn1nccc1C(N1CC(F)CC1CNC(c1ccccc1)=O)=O 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75602,c1(SC)sccc1C(=O)NC1CC1NC(=O)CC1CCCOC1 75603,N1(C(c2cc(C)c(C)[nH]2)=O)CCC(NC(=O)CCOC(C)CC(C)C)C(F)C1 75604,CC1CN(C2CC2)CCN1C(=O)C(c1ccc(C2CC2)cc1)O 75605,N1(C(c2cnc(CC)nc2)=O)CCC(NC(C2CC2c2ccccc2)=O)C12CC2 75606,c1(C(N2CCC(Oc3ccccc3C(N)=O)CC2)C)cn2c(n1)COCC2 75607,c1(C(C)N)ccc(C(N2CC(NC(c3ccc(F)nc3)=O)C2)=O)cc1F 75608,Cn1cc(NC(C2CCCCN2C(=O)Cn2cccnc2=O)=O)c(Cl)n1 75609,c1(OC)ccc2[nH]c(=NCC(C)NC(c3cc4c(C)sc(C)c4s3)=O)sc2n1 75610,N1(C(C2CCCC(CC)C2)=O)CC2CCCC(C1)N2Cc1c(C)cccc1O 75611,Cc1csc(=O)n1CC(=O)NC1(CF)CCN(C(C23CC(O)C2C3)=O)C1 75612,N1(CC)CCC(NC(C2CC(NC(=O)C(=O)NCC3CC3)C2)=O)C1 75613,C12(C(=O)NCCCN(C(COCC#C)=O)C)CCC1CCN2 75614,c1(C(=O)OC)coc(NC(C)C(C2CCCCC2)NC(=O)C=Cc2cn[nH]c2)n1 75615,c1(CC)ccccc1C(N1CC2C(NC(c3cc(C4CC4)nn3CC)=O)C2C1)=O 75616,[N-]=[N+]=Nc1ccc(NC(c2cncc(CNC(C3CC(O)C3)=O)c2)=O)cc1 75617,C1(NC(C2CC(N(C)CC)C2)=O)CCC2CN(C(=O)CCC3CCC3)CC2C1 75618,C1(NC(CCC(=C)C)=O)CCN(C(C2CCC(=O)C2)=O)CC(O)C1 75619,c1(C(C)NC(CNC(CCC)=O)=O)ccc2c(c1)CN(C(C1(F)CC=CC1)=O)C2 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75952,Cc1cc(F)ccc1CNC(=O)CC1CCCC1NC(C1C2COCC12)=O 75953,N1(C(C=CC)=O)CCOC(CNC(c2cc(-c3c(C)cccc3C)[nH]n2)=O)CC1 75954,c1(CC)ccc(-c2noc(C(N3CCC(C)C3c3cccc(F)c3)=O)n2)cc1 75955,C1(C(=O)N)CN(CC2(N(C)CC)CN(C(=O)C(O)C3CC3)C2)CCO1.CSC 75956,Cc1ccccc1C=CC(=O)NCC12CC(NC(=O)CC3CCC4CC34)(C1)C2 75957,N#Cc1cccc([N+](=O)[O-])c1NC(=O)NC1CC1.N12CC(CC(F)C1)C2=O 75958,Cc1csc(C=CC(=O)NC2CC2CNC(=O)CSc2nncn2C)n1 75959,CC(CS(C)=O)N=c1ccc(Br)c(S(=O)(=O)NCC(c2c(F)cccc2F)(C)C)[nH]1 75960,N1(C(CCCC=C)=O)CCC2C(C1)CN2C(c1c(F)cnn1C(C)C)=O 75961,C1(C)(C(N2CC(CNC(c3ccc(OC)o3)=O)C(F)(F)C2)=O)CCC(C)C1(C)C 75962,c12nnc(N3CCCC3)n1CCCNC(=O)C(C)S2.C(C(F)(F)F)OCC 75963,C=C1CCN(C(=O)CC(CC)CC)C(C(=O)NC(C)C)C1 75964,C(CCC(CC)CC)NC(C1C(CC)CCN1C(=O)CN(C(=O)COC)C)=O 75965,C(=O)(CC(C)(C)CC(F)F)N1CCC(N(C(C(C)SC)=O)C)C2(C1)CC2 75966,N1(C(c2cn(CC)nc2)=O)CCc2ccc(CCC(C)N(C)C)cc21 75967,c1(CC)cccc(NC(=O)CCCCCNC(=O)CN2CSCC2=O)c1C 75968,c1(C(N(C2CCCN(C(C3CCCN3C3CC3)=O)C2)C)=O)ccccc1F 75969,c1(NC)cc(Cl)c(S(=O)(=O)N2CCCC(c3ccccc3)(CO)C2)cc1[N+](=O)[O-] 75970,c1(CN2C(C(=O)Nc3ccc(OC)cc3OCC)CC2)cnn2cccnc12 75971,c1(C(=O)NCCNS(CC)(=O)=O)[nH]ccc1CNC(c1cnco1)=O 75972,C(=O)(C1=CCN(C(=O)Cn2ccccc2=O)C1)NCCN(c1ccsc1)C 75973,C(CCCC(=O)N(C1CCNC1=O)C)N(C(C(C)=CCC)=O)C 75974,c1(C(N2CCC(CNC(CN(C)C(=O)OC(C)(C)C)=O)C2)=O)nccc(Cl)c1C 75975,S(=O)(=O)(c1cc(C)cnc1NCCOCCO)NCCC(CC)O 75976,C1(NC(C2(OC)CCN(C(=O)C(F)(F)C(C)(C)O)C2)=O)CCn2ncnc2C1 75977,c1(SC)ccc(S(C)(=O)=NC(=O)C(=O)NCC(N)C2(Cl)CC2)cc1 75978,Cc1nn(C)cc1S(=O)(=O)N1CC2C(C1)N2S(=O)(=O)c1ccccc1F 75979,N1(CC)CC2CCC(C1)C2Nc1ncnc2occc12 75980,C#CCCCCCC(=O)NCCOC1CCN(C(=O)C(C)C2CC2)CC1 75981,c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2cnc[nH]2)CO)c(C)n1 75982,c1(C(=O)NC(CNC(Cc2c(C)nsc2)=O)C2CC2)cccc(-n2cccn2)c1 75983,C1(NC(C(CC)C(C)C)=O)C2CC3CN(C(C4CN(C)CC(C)O4)=O)C1C3C2 75984,c1(OCC(=O)NC2CCCC(NC(Cc3nnc(C)s3)=O)C2)c(C)occc1=O 75985,c1(C(N2CC=C(CNC(=O)C(O)O)CC2)=O)cccc2c1CNC2=O 75986,Cc1[nH]c(C)c(C(=O)NC2CCC(N(C)C(c3ccc(CO)cc3F)=O)C2)c1C 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76178,C=CCC(CC(=O)N(C1CC2CC2C1)C)NC(=O)C(O)C1CCCC1 76179,C1(NC(c2c(SC)csc2)=O)C2CC(NC(=O)CS(C)(=O)=O)CC12 76180,N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3sccc3C(F)F)=O)CC2C1 76181,C1(NC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2CCSCC2)C2CCCCC12 76182,c1(C(N2CC(NC(C#CC(C)(C)C)=O)CC2(C)C)=O)cc2ccc(F)cc2s1 76183,c1(C(=O)NC2CN(C(c3ccc(C)c(N)c3)=O)C(C)C2)ccc2[nH]nc(Cl)c2c1 76184,N1(Cc2ccc(C)nc2)CCC(O)C(C(N2CCCC2)=O)C1.c12ccc-1o2 76185,C=CC(C)(CCOC)C(=O)N1CCOC(C(C)NC(C2CC(O)(C#N)C2)=O)C1 76186,C1(CC(=O)NCc2c(CC)scc2)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 76187,c1(C(N2CC(NC(C(C3CCCOC3)OC)=O)(CO)C2)=O)ccc(N(C)C)cn1 76188,C12(NC(C=CC=CC)=O)CC(C1)N(C(C1CC(=O)N(C3CCC3)C1)=O)C2 76189,C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(Cc1ncc(C)s1)=O)C 76190,N1(C(c2n(C)nc(C)c2Cl)=O)CC2CCOC2(CNC(c2c(C)ncnc2O)=O)C1 76191,C1(NC(CC(C)OC)=O)CN(C(c2ccc(C)c(F)c2)=O)C2(CCCC2)C1 76192,C1(O)(C(N2CCC(N(CC#C)C(c3cc(C(N)=O)c[nH]3)=O)C2)=O)CCC(C)CC1 76193,N1(C(C2CCN(CC(C)C)CC2)=O)CC(O)(C2(CNC(=O)C(C)CC(N)=O)CC2)C1 76194,C1(NC(CC(C)(C)C)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(N)c1)=O 76195,C(CCCCCNC(=O)C(C)(C)CNC(C1C=CCCC1)=O)OC 76196,Cn1c(C(N2CC3CC(NC(C4CCC(F)C4)=O)CC2C3)=O)cnc1[N+](=O)[O-] 76197,O=C(C#CC1CCOC1)NCCSCC(O)C(=O)N1CCC1c1ccccc1Br 76198,c1(-n2c(CCCOC)nc(C3CCOC3)n2)cc(Cl)nc(Cl)c1 76199,c1(NC(C(=O)N(C)Cc2nc(Cl)ccc2Br)=O)cccc(F)c1Cl 76200,c1(C(N2CCC(C)(NC(c3cc(C(C)C)no3)=O)CC2)=O)cc(O)cc(F)c1F 76201,CC1CC(C(=O)NCC2CC3CC(=O)C2O3)CCN1C(=O)COCC(F)F 76202,C1(N(C(=O)Cc2cnccn2)C)CC2CCC(C1)N2C(=O)Cc1nn(C)cc1Cl 76203,N1(CC)CCCC(CNC(C2CC(C)N2C(c2cn(CCO)nn2)=O)=O)C1 76204,C1(CC(=O)NC2CCCN(C(C=CSC)=O)C2C)CCCCC12OCCO2 76205,C1(C(N2CC(CC(N)=O)C2)=O)CCC2(CN(C(=O)NC3(Br)CC3)C2)O1 76206,N1(C(c2c(C)nsc2C)=O)CC2(CNC(c3snnc3C3CC3)=O)CCC1C2 76207,c1(OC(N2C(CC)(CNC(C3(COC)CC3)=O)CCC2)=O)c(C)cccc1Cl 76208,Cc1nn(C)cc1C(N1CC2C(NC(C3(C)CC3(Cl)Cl)=O)C2C1)=O 76209,C1(CNC(=O)CSCc2ncoc2-c2ccon2)CCN(C(c2cscn2)=O)C1 76210,c1(C(=O)NCCNC)ccc(-c2ccc(CC(C)C)nc2)c2cc[nH]c12 76211,c1(C(=O)NC(C(C)C)CCNC(=O)CCc2ccco2)cccc2nc(O)[nH]c12 76212,n1(CC)ncc(C(N2CC(CNC(C3(O)CCSC3)=O)C(C)C2)=O)c1C1CC1 76213,CCCC(CC)C(=O)N1CCCCC1CNC(=O)CC1CCC(=O)N1C 76214,c1(CC(=O)NC2C(n3cc(-c4cnc(CC)s4)nn3)CCC2)ccc(OC)c(F)c1 76215,C#Cc1ccc(C(=O)NC2CCCC2(C)NC(=O)CCCC2CC2C)c(F)c1Cl 76216,C1(NC(=O)CCCc2ccncc2)CC2CCC1N2C(c1cc2sccc2[nH]1)=O 76217,CC(Cc1cccs1)CC(=O)NCC(C1CCCCO1)(C)C 76218,c1(C(N(CCCN(C(=O)CCC(F)F)C)C)=O)cnc2ccoc2c1 76219,C1(CNC(C(C)c2ccco2)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)CC12 76220,c1(C(=O)OC)cc(C)c(C(N2CCCCC2C2CCN(C(=O)CC(C)F)CC2)=O)o1 76221,c1(C(N(C)C(C2C3CCC(F)C23)=O)=O)ccc(O)c(=O)cc1 76222,C1(COC)CCN(C(=O)C(=O)NCC(C(F)F)c2ccccc2)CC1 76223,c1(C(N2CCC(c3cccc(OC)c3C(F)F)CC2)=O)nc2cc(Br)cnc2[nH]1 76224,C1(C(=O)NCC(C)(C2CCC2)NC(C(=O)N(CC)CC)=O)CC2(CCO1)CC2 76225,ClCCCN=C(NN1CCC(O)C1)NC1CCCCC1.C1(C)CCCO1 76226,C(CC(CO)SC)N(C(=O)Cc1cn[nH]c1)C1CC1.C12CC(C1)NC2=O 76227,N1(C(CSCC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOC2)CCF)C1 76228,Cc1cn2cc(C(=O)NC(C)CNC(C3CCCNS3(=O)=O)=O)ccc2n1 76229,C1(CNC(C(C)NC(CNC(CN(CCC)C)=O)=O)=O)COCC1(C)C 76230,Cc1cn2c(C(N3CC4(C3)CN(C(C3(C)CCC3(F)F)=O)C4)=O)c(C)nc2s1 76231,CCCC(C(=O)NC(C)CC(F)(F)F)N(C)C.c12cc[nH]c1C(=O)NC2 76232,N1(C(C2CCN(C)C2)=O)CCc2nn(C)c(C(=O)Nc3nccc(F)c3F)c2C1 76233,C#CCC(O)C(=O)NCC1(CN(C)C(c2cscc2Cl)=O)CC1 76234,c1(CC(=O)OCC)sc(NC(c2occc2Br)c2ccccc2)nc1C 76235,N1(C(c2c(C)nc(CC)o2)=O)CCCC(C)(NC(=O)CC2(OC)CCCC2)C1 76236,Cc1cc(CCC(=O)NC2CC(CCNC(=O)C(F)C(F)(F)F)C2)ccc1Cl 76237,c1(OC)cnc(C(=O)NCC=CCNC(C2CC(=O)CCO2)=O)cn1 76238,CC1CN(C(=O)CC2CN(C(=O)OC(C)(C)C)C2)CC(C(=O)Nc2cn(C)cn2)O1 76239,N1(C(C(F)=CC)=O)CCCC(O)(CN(C(=O)C(C)(C)CC)C)C1 76240,C(=O)(CC(C(F)F)NC(c1cccc[n+]1[O-])=O)N(C)Cc1ncnn1C 76241,c1(C(C(=O)NCCCC)N(C2CCCCC2)CCF)cc(C)ncn1 76242,C1(NC(c2cc(C)nc(C)n2)=O)CCC12CCCN(C(=O)C=C(C1CC1)C1CC1)C2 76243,c1(C(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2F)cccc2c1C(F)(F)CC2 76244,C(Cc1ccccc1OC)(C(=O)Nn1cnnc1)c1ccc(S(CC)(=O)=O)cc1 76245,C(=O)(CCCN(C)N=O)N(C(C)CCNC(=O)C(C)CSC(F)(F)F)C 76246,N1(C(c2[nH]cc(CC)n2)=O)CCCC(O)(CNC(=O)CCNC(=O)COC)C1 76247,C1(NC(=O)CC2CCCC(F)(F)C2)CC2CN(C(c3nccc(C(F)F)n3)=O)CC12 76248,C1(c2cn(C)nc2)CS(=O)(=O)CCN1C(C12CCC(C(N)=O)(CC1)C2)=O 76249,Cc1cc(CCC(=O)NC2CN(Cc3c(C)cccc3F)CC2F)cc(C)c1 76250,N1(C(CC2N(C)CCC2)=O)CC2(CCCC2NC(c2cn3ncccc3n2)=O)C1 76251,c12cc(ccc1F)C(=O)NC(C)C(C)(C)NC(=O)CNC2=O.C(C)(C)(C)S.CC 76252,C(=O)(CS(=O)(=O)C(C)C)NCC(CNC(C1C(C)=CCS1)=O)(C)C 76253,CCCCCCCc1cn(CC2C(CNC(=O)CC3CC(SC)C3)C2(F)F)nn1 76254,N1(C(CCCC#C)=O)CCN(C(=O)CCc2csc(Br)c2)CC1CC 76255,Cc1cc(NCC2CCC2(F)F)ncc1S(=O)(=O)NC(CC1CC1)C1CC1 76256,c1(CC)cc(CN2CCC(C(=O)NC3CCCN(C(C)=O)C3)CC2)ccc1F 76257,C1(C(N(C)Cc2cnc(C)s2)=O)CC2CC3(CC2C1)OCCO3 76258,C1(=CCNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCF)CC1 76259,C12(C(N(C)CC)=O)CCCC1N(C(C1C3CCC(C3)C1C)=O)CC2 76260,n1(CC(=O)NCCNC(c2cnccn2)=O)ncc2cc(Br)cnc2c1=O 76261,C(=O)(CC(C(F)F)NC(=O)CC1(NC(C)=O)CC1)NCC(=C)C(F)(F)F 76262,Cc1c(C(=O)NC(C)CCN(C)C(C2CCCCC2O)=O)cnn1CC(F)F 76263,C1(NC(COC)=O)CC2C1CCN2C(=O)CC1CCOC(C)(C)C1 76264,c1(-c2ccc(CNC(C3CCC(C4CCC4)N3CC)=O)o2)cccc2c1CCC2 76265,C1(C(C)C)(CO)CCN(C(C2CC(C)N(C(=O)COC(C)(C)C)C2)=O)C1 76266,C1(CNC(C2C(C)C2)=O)CCC(NC(=O)C(F)(F)C2CCOCC2)CC1 76267,C(=O)(C1c2ccccc2C2CC1C2)NCC1(C)CC(NC(C=CC=CC)=O)C1 76268,Cc1ccc(-c2csc(C(=O)Nc3ccnc(OC(F)(F)F)c3)c2)c(F)c1 76269,c1(N(CCCSc2ccccc2)C(c2cc(C(F)F)on2)=O)ccc(Cl)c(F)c1 76270,c1(N(C(COCC)C)C)nc(N2CCC(Cc3nncs3)CC2)c2c(n1)CSC2 76271,CC(O)C(C)(C)C(=O)N1CCN(C(=O)CC(O)Cc2ccccc2)CC1 76272,CC1(CNC(c2cc3occc3s2)=O)CCCN(C(C2C(F)(F)C23CC3)=O)C1 76273,c1(C(=O)OC)cc(Cl)cnc1N1CCC(C2NC(=O)NC2=O)C1 76274,c1(OC)cc(N(C)C)ccc1C(=O)NCC(C)(C(C)C)NC(=O)CC1(C#N)CC1 76275,c1(CCC(C)NC(c2n(CCCOC)nnn2)c2cnc(C)o2)ccc(F)cc1 76276,N1(C(C2CC3CC3N2C(=O)CC2CC2)=O)CCC2(CCOC2=O)CC1 76277,C1(NC(CC2(NC(C)=O)CC2)=O)CC12CCN(C(=O)C(c1ccccc1)O)C2 76278,C(=O)(CC(COC)NC(c1c[nH][nH]c1=N)=O)N(C)Cc1c(CC)noc1 76279,C1(C2CC2)(C(N2C(C)(C)CC(O)C2)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)C1 76280,c1(OC)ccc(C(=O)N(C2CN(C(=O)CN(C)C)C2)C)c2[nH]ncc12 76281,c1(CC(=O)NCC(CNC(=O)CC2CCOC2)OC)ccc(C)c(Cl)c1 76282,N1(C(CC2C=CC(N)C2)=O)CCc2c(F)ccc(I)c2C1 76283,c1(CCOC)cn(CCC(N2CCCC2CC(O)CO)=O)nn1 76284,N1(C(=O)Cn2ccnn2)CC(CNC(C2(O)CCC2)=O)C1 76285,N1(C(=O)NC2C(N3CCN(C)CC3)CCC2)CCOC(C)(C)C1C 76286,n1(CC)ncc([N+](=O)[O-])c1C(N1CC2(CC2NC(C2CC(C)C2)=O)C1)=O 76287,CC1(C)CN(C(=O)C=Cc2ccc[nH]2)C1C1CC1.C12CC(C1)CNC2=O 76288,C(=O)(CCN(OC)C(=O)C1CC1CC1CC1)OC.c12ncn(C)c1-c1cn(nn1)C2 76289,C12(C(=O)NCCNC(CC)=O)CC1CCN2C(=O)CCc1cc(C)no1 76290,c1(C(=O)NC2CCC(NC(c3cc(C(C)=O)sc3)=O)C2)ccc2c(c1)ncn2C 76291,N1(C(C(C)SCC)=O)CC2CCC1C2NC(c1nccnc1-n1ccnc1)=O 76292,c1(OC)ccnc(C(N2CCC(OCCNC(=O)C3=NOC(C)C3)C2)=O)c1F 76293,C(C(CC1CCC1)C(=O)N(C1CCC1)C1CC1)NC(=O)COCC1CC1 76294,c1(CC(C(=O)N(C)CC2(CF)CCOCC2)C)ccc(F)cc1 76295,c1(N2C(CC)CN(C(=O)Cc3cccc(SC)c3)CC2)ncc(C#N)cc1Cl 76296,C1(CN(C(CC2(COC)CC2)=O)C)C2CN(C(=O)CSc3ccccc3F)CC12 76297,c1(N(C)C(N2CCCC(c3noc(=O)n3C)C2)=O)cccc(C2CCC2)c1 76298,Cc1ccc2c(c1)CCN2C(=O)Nc1ccc(OC(F)F)cc1 76299,c1(NC(c2n(CCCC)nnn2)C2(C)CCCO2)ccc(F)c(C(N)=O)c1 76300,Cc1ncoc1C(=O)NCC1CCCC1NC(=O)C(C)C1CCCC1 76301,C=CCCN=C(NCC1CCC(C(N)=O)O1)NC1CCN(SC)C(C)(C)C1 76302,Cc1ccc2cc(C(N3CCN(C(c4cnc(O)n(C)c4=O)=O)CC3C)=O)[nH]c2c1 76303,C1(N(C(=O)COCc2nc[nH]n2)CCC)CN(C(=O)C(CC)OC)CCC1O 76304,C1(C(N2C(CN(C(C(CC)C)=O)CC)CCC2)=O)CC(=O)N(C2CC2)C1 76305,C1(CNC(C)CC2CC2)CCCC2(CCN(C(=O)OC(C)(C)C)CC2)O1 76306,C1(C(=O)NC2(C3CN(C(C4(CCCC)CC4)=O)C3)CC2)CCCC(C)(C)CC1 76307,C1(C(=O)NCC(C)C(=O)NCc2ccoc2)C(C)(C)C1(C)C 76308,C12CN(CCO1)C(=O)CNC2C.c1(CNC(COC(CC)C)=O)cc(C)on1 76309,c1(CNC(C(COC(C)C)NC(=O)C=CC(F)(F)F)=O)ccc(F)cc1F 76310,c12ccc(cc1)C(Cc1nn[nH]n1)O2.C1(C#N)(OC)CCCC1 76311,c1(CC)cc(C(=O)NC(c2ccccc2F)CNC(c2cc(Cl)no2)=O)n(C)n1 76312,C#Cc1ccc(NC(=O)C(F)C(C)CNC(c2cc[nH]n2)=O)cc1 76313,c1(C(N2CC(OCCN(C)C(C3(C)CCC3)=O)C2)=O)cc(Cl)ccn1 76314,c1(C(C(=O)Nc2ccc(Cl)cc2F)N(C(C)C)C(C)C)ccc2occc2n1 76315,N12CC3C(C3C1)OCC2=O.C(=O)(C(C)CC#C)NCCOCCOCC#C 76316,C1(C(=O)NCC2CN(C(C(c3cccc(OC)c3)C)=O)C2)CCc2nc[nH]c2C1 76317,c1(C(c2n(CC(=C)C)nnn2)NCC(N2CCCCC2)=O)ccnc(C)c1 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76685,n1(CC)nc2c(c1C(N1CCCCC(NC(C3CCC(C)O3)=O)C1)=O)CCCC2 76686,CC(C)(F)CCC(=O)NCC(CNC(c1ccnc(C(N)=O)n1)=O)CO 76687,c1(C(=O)NC23CN(C(Cc4c(C)n[nH]c4C)=O)C(C2)C3)c2c(nn1C)CCC2 76688,C1(CN2C(C)CN(C(=O)N(C)C)CCC2)COc2ccccc2O1 76689,CCN=c1ccc(C(=O)NCC(C)NC(=O)CCc2nnc(C)n2C)c[nH]1 76690,c1(CC)[nH]c(=N)sc1C(N1CC(O)CC1CNC(C1CC1C(C)C)=O)=O 76691,Cc1cccc(C(=O)NCC2CCC(NC(=O)C(C)(F)F)CC2)c1Cl 76692,C1(NC(c2ncn(CC)n2)=O)CC2CCC1(NC(c1ccc(Cl)c(O)c1)=O)C2 76693,C1(C(N2C(CNC(c3ccn(CCC)n3)=O)CCC2)=O)CCCN(C(=O)NC)C1 76694,c1(NCC(CC)N(C)CC)ncccc1S(=O)(=O)N1CCCCCCC1 76695,N1(C(C(N2CC(C)C2)C)=O)C(C(=O)NCC2CC23CCCCC3)CC2CCCC12 76696,Cc1cc(C(=O)NCC(C)NC(C2(C(C)C)CC2)=O)nc(C2CCC2)n1 76697,N1(C(CSCC(N)=O)=O)CCC2CCC(NC(c3ccc(C(F)F)c(Cl)c3)=O)C12 76698,c1(C(=O)NCC2(C(N3CCC3)=O)CN(c3ncc(C)cn3)C2)cccc2ccnn12 76699,C1(CNC(COCCC=C)=O)(CNC(=O)C(C(C)C)Nc2ccoc2)CC12CCC2 76700,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)NC(C(c1c(OC)cccc1)C)=O 76701,N(C1CCCc2c1ccn2C)C(C(C)n1ccnc1)=O 76702,C(=O)(C(C)CCCOC)N1CC2C(N(C(c3ccn(CCC)c3C)=O)CC)C2C1 76703,C(=O)(CCCCCCOC)NC(C(C(C)NC(CN(C(CCC)C)C)=O)(C)C)=O 76704,N1(CCNC(C(C)OC)=O)CCCN(C(c2sc(Br)nc2C)=O)CC1 76705,C#CCCCC(=O)N1CC(OCCC(=O)NC(C)C(C)CO)C1 76706,CC1(C)C=C(C(=O)N2CCC(C)(NC(=O)Cn3ncccc3=O)C2)C1 76707,C1(O)(C(=O)NC(CC)CNC(=O)C2=CCOC2)CCc2ccccc2C1 76708,N1(C(c2nc(-c3cccnc3)no2)C)CCC(O)C1NC(=O)NC(C1CCC1)C 76709,N1(C(C=CC(=O)N(C)C)=O)CC2(CC2)CC1CNC(C12CCC1C2)=O 76710,C1(NC(COC2(C)CCC2)=O)CC2CC1CN(C(c1cncs1)=O)C2 76711,CC1CC=C(C(=O)N2CC3(CC(NC(c4ccccc4OCCF)=O)C3)C2)CC1 76712,Cc1cc(C(N2CCCC2CC(=O)N(CC(C)(C)N(C)C)C)=O)co1 76713,C#Cc1cncc(C(=O)NC(C)CNC(C2(C)CCCCO2)=O)c1 76714,C=CCCC(F)(F)C(=O)NC1(COC)CCCN(C(=O)C(CC)C(C)C)C1 76715,c1(C(N2CC(NC(c3nc(NC(C)=O)sc3)=O)C(C)C2)=O)cc(S(C)(=O)=O)co1 76716,c1(OC)ccc(C2CCN(C(c3c(C)n[nH]c3C)C(=O)NC(C)C)C2)cc1 76717,N1(C(CCN(CC=C)C(C2CC3CC3C2)=O)=O)CCCC(C)(C)CC1 76718,CC(CC(C)(C)C)C(=O)NC1CN(C(c2cnc(S)n2C)=O)C(C)(C)C1 76719,N1(C(CCCCOCCC=C)=O)CCC(NC(C2(CN(C)C)CC2)=O)CC1C 76720,C=CCCC(C)C(C)N1CCN(CC(=O)NCC)C(C)C1.C1(C2CC2)CCO1 76721,N1(C(c2cc(C#N)[nH]c2)=O)CCC(CNC(=O)CC2CCCC2O)C(F)(F)C1 76722,C1(N2CCN(C=O)CC2)COCC12OCCO2.n12cc(nn1)C2 76723,c1(C(N2CC(NC(CCC)=O)C(C)(C)C2)=O)ccnc2[nH]ncc12 76724,N1(C(C=C(CC)C)=O)CCC(C2CCN(C(=O)CCn3nc(C)cc3C)C2)C1 76725,c1(C(COC(C2C(C(=O)OCC)CC2)=O)F)ccc(F)cc1F 76726,N1(C(C2(SCC)CC2)=O)CC2(CCN(C(c3cc4ncc(Br)cn4n3)=O)CC2)C1 76727,CC1(C)CCC(C)(C(=O)NC(C)(CNC(c2cncc3c2CCC3)=O)C2CC2)CC1 76728,c1(OCCC(=O)NCCC2C(C)CN(C(=O)CCF)C2)ccc(Cl)c(F)c1O 76729,C1(NC(CNC(C)=O)=O)CC2C1CCN2C(c1cnn(C)c1Cl)=O 76730,N1(C(CN(C)CC)=O)CC(C)CN(C(=O)Cc2ccc(O)c(Cl)c2)C(C)C1 76731,N1(C(CNC(CCCCC)=O)=O)CCN(C(C2CCCCN2C)=O)CC1C(F)F 76732,c1(C(=O)NCC2N(C(C(COCC)C)=O)CC2)cnn2ccsc12 76733,N1(C(C2N(C)C(=O)CC2)=O)CCCN(C(=O)CCCCC#N)CC1C(C)(C)C 76734,c1(C(=O)NCC(C(C)C)NC(c2cccc3nn[nH]c23)=O)ccnc2[nH]ncc12 76735,C1(C(n2cc(-c3ncccc3Br)nn2)COC)CCC(F)(F)C1 76736,C(=O)(C(C)(C)CCCC=C)NC(C(N1C(C#C)CC1)=O)COC 76737,C1(NC(c2cnc(OCC)s2)=O)CCCC(NC(=O)CCc2cnccn2)C1 76738,Cc1c(F)ccc(C(=O)NC2(CNC(C3CCCCO3)=O)CCOC2)c1O 76739,CCC(C)CCCC(=O)N1CCC(NC(=O)CSCc2cccnc2)C1C 76740,N1(C(c2ccnn2C)C(C)C)CCC(N=c2cc[nH]cc2)C(C)C1 76741,N1(C(CCN(c2cncnc2)C(c2c(Cl)cn(C)n2)=O)=O)CC23CCC2(COC3)C1 76742,c1(OCC(=O)NCC2CN(C(C=C(C)C(C)C)=O)C2)cccc(C#N)c1 76743,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 76744,C1(CNC(C2CN(CCOC)C(=O)C2)=O)(CO)CCN(C(=O)CSC(F)F)CC1 76745,C=CC(C)C(C)C(=O)N1CC(O)(CNC(c2ccc(C(=O)N(CC)CC)nc2)=O)C1 76746,C1(NC(CCCSC)=O)COCCN(C(C2CC3C=CC2CC3)=O)C1 76747,C1(C)(CC2CC2)COCCN(C(=O)CNC(Cc2cc(COCC)nn2C)=O)C1 76748,CCC(CC)CC(F)C(=O)NC1CC=C(C(=O)N(C2CCNC2=O)C)C1 76749,C1(CNC(COCCC)=O)CN(C(=O)C=Cc2cccc(O)c2)CC(C)(C)O1 76750,C(=O)(CCC(=O)C(C)(C)C)N(CC(=O)NCC1CNC(=O)C1)CCS.CO 76751,c1(NCc2ccc(OC(C)C(=O)O)cc2)cc(Br)c2ccccc2c1 76752,C(=O)(C(C(=O)NC1CCCN(C(=O)CCN2CCCCC2)CC1)C(C)C)OCC 76753,C1(O)(CNC(C2(CSC)CCC2)=O)CCCN(C(=O)C(=O)NCC(F)F)CC1 76754,N1(CC(C)(C2CC2)OCCOC)CCCC(C)C1C 76755,C1(CCNC(C(C)C2CC2)=O)CCN(C(C2COCCN2CC(F)(F)F)=O)CC1 76756,CC(C)C(F)(F)CC(=O)NC(C1CN(C(C2CCCC(F)C2)=O)C1)C 76757,CC(C(C)C(=O)N1CCCC(CCF)C1)NC(C=CC(=O)OC(C)(C)C)=O 76758,Cc1ccc(C(=O)NCC2(F)CC(CNC(=O)COCc3ncnn3C)C2)cc1 76759,Cn1[nH]c(C(=O)NCCCNC2CCN(CCC3CC=CCC3)CC2)nc1=O 76760,c1(C(C(=O)NCC)N(C)Cc2nc3ccc(Br)cc3o2)cnc2ccc(Cl)cn12 76761,c1(C(=O)NC2CCCC2CNC(C2CCC3CC3CC2)=O)c[nH]c2cccc(F)c12 76762,c1(-n2cc(C3CCN(C(C4C(C#N)CC4)=O)C3)nn2)nc(O)cc(O)n1 76763,c1(N(C2CC2)C)cccc(C(N2CCC(N(C)C(c3[nH]c(C)nc3C)=O)CC2)=O)c1 76764,c1(OC)ccc(CNC(=O)CN(c2ncc(F)cn2)c2ccccc2)cc1 76765,c1(C(N2CCN(C(c3cc(CCO)on3)=O)C3CC23)=O)cc2c(cn1)OCCO2 76766,C1(NC(=O)CCC2CC2(F)F)CN(C(C23CCCC2C3)=O)CC2(CCC2)C1 76767,N1(C(C(CC)CCOC)=O)CC2(CCCN(C(=O)C(F)CC(CC)CC)C2)C1 76768,C1(NC(C(C)N(C)Cc2ccccc2)=O)CCC(NC(c2sccc2F)=O)CC1 76769,C1(F)(C(N2CC(F)(CNC(c3cc(C)[nH]c3)=O)C2)=O)CCN(C)CC1 76770,c1(C(=O)NC2CC3CCC2(NC(=O)C(O)C(F)(F)F)C3)[nH]nc([N+](=O)[O-])c1Cl 76771,c1(C(N2CC(N(C(C=C(C)c3ccco3)=O)C)C2)=O)cnc2ccccc2c1C 76772,c1(CC(=O)Nc2cnn(CC(F)(F)F)c2)nc(C2CC2COC2CCC2)cs1 76773,N1(C(=O)CCSC(F)(F)F)CCC2CN(C(C3CC3C3CC3)=O)CC2C1 76774,c1(CC)ccc(C(=O)OC2CCOC2)c(C)c1.C12CCN(C1(C)C)C(=O)NC2=O 76775,c1(N2CCCC(CNC(c3nc(NC(N)=O)sc3)=O)C2)ncc([N+](=O)[O-])cc1F 76776,CC1CN(CC(=O)NC2CCCOC2)CC(C)CN1C(C1C2CCCC12)COC 76777,Cc1cccc2cc(C(N3CCCC(CO)(NC(=O)CC4(CO)CC4)C3)=O)sc12 76778,c1(C(=O)NCC(CNC(C(C)c2ccco2)=O)O)ccn(C)c1 76779,N1(C(C(C)NC(=O)C(N)=O)=O)CCN(C)C(CO)C1 76780,N1(C(=O)CNc2ccccn2)CCC2(CCN(C(=O)C(F)CC3CCCCC3)C2)C1 76781,c1(N(C)C)ccc2c(N3CCN(c4cccc(Cl)n4)CC3)nc(Cl)nc2c1 76782,c1(C(N2CC(C(=O)NC(Cn3ncc(C)c3)C)C(F)C2)=O)cc(C)nnc1C 76783,C1(C(=O)NCC2CCN(C)C2)(OC)CCN(C(c2cc(C3CC3)no2)=O)CC1 76784,c1(C(=O)NC2C(NC(C3C(CC)C3)=O)COC2)cc(C)c(OC)c(C)c1 76785,CCCC(C)(C)C(=O)NC(c1ccccc1)CNC(=O)C(C)S(C)(=O)=O 76786,Cc1nc(CNC(=O)CCc2csnn2)oc1C(=O)N(C)Cc1ccccc1 76787,N1(C(C(C)NC(COCC#C)=O)=O)CC(N(C)C)C(SC)C1 76788,c1(C(N2C(CNC(c3ccccc3)=O)C=CC2)=O)cc2cc(Br)ccc2o1 76789,C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CSc2ccccc2)C1(C)C 76790,N1(C(C(C)OCC#C)=O)CC2(CC(CC(N3CC4(CC=CC4)C3)=O)C2)C1 76791,O(C=CC(=O)N1CCC(C2(NC(=O)CSC(C)C#N)CC2)C1)CC 76792,N1(C(C2NC(=O)OC2)=O)CC2CCCC(NC(c3cc4ncccc4s3)=O)C2C1 76793,c1(-n2c(-c3ccc(C(F)(F)F)cc3)nc(C)n2)ccc(-n2cnnc2)cc1[N+](=O)[O-] 76794,c1(C(=O)NCC(=O)Nc2cccc(C(O)C(F)(F)F)c2)c[nH]c2ncc(F)cc12 76795,C1(CNC(c2c[nH]c(=S)cn2)=O)CCN(C(=O)C=Cc2ccoc2)CC1C1CC1 76796,c1(OCCC)ccccc1CNC1CCC(NC(c2cnn[nH]2)=O)CC1 76797,N1(C(CCN(C)C)=O)CC2CC1N2.C1(C#N)(CC(N2CCCC2)=O)CCC1 76798,N1(C(CC(COC)(C)O)=O)CC(C2CCN(C(C3(CCF)CC3)=O)CC2)C1 76799,Cc1c(C)n(C)c2ccc(C(=O)NC3CCOCC3NC(C3CC(O)C3)=O)cc12 76800,C=CC1OCCCC1C(=O)N(C)CCOCCN(C)C(c1nncn1C1CC1)=O 76801,c1(OC(C)C(=O)N(CC(O)CNC(=O)CN2CCNC2=O)C)ccccc1Cl 76802,N1(CC(=O)NCC2CC(C3CCC3)C2)CCc2sccc2C1 76803,C1(C(C)NC(CC(=O)NCC#C)=O)CCCN(C(=O)Cc2cn(C)nc2Cl)C1 76804,C1(NC(c2ccc(C)o2)=O)(CNC(C2CCOCC2)=O)CC(F)(F)C1 76805,C1(COC)CN(C(c2ccc(Cl)nc2)=O)CCN1C(=O)CCCc1cccc(Cl)n1 76806,c1(CCCC)ccc(C(C)N(C(=O)C(C)OC(=O)CC2CCC2)CCO)cc1 76807,C1(NC(CCSCCCC)=O)CCN(C(=O)CNC(=O)NC)CCC1(F)F 76808,c1(-c2ccc(CN3CC(Nc4cc(C)[nH]n4)C(O)C3)cc2)cc(F)cc(F)c1C 76809,C=CCC(C)C(C)(c1nnnn1CCCC)NCC1(CO)CCOCC1 76810,CC(C)(C)C(CNC(=O)CCCN1CCCC1)C(=O)NCCC1=CCCCC1 76811,N1(C(c2c(C)cccc2)=O)CCN(C(c2ocnc2C(F)(F)F)=O)CC12CCC2 76812,C(=O)(CC(CC1CCCCC1)NC(=O)CNc1ncccn1)OC 76813,C1(F)(C(N2CC(OCCOC)C2)=O)CCCN(C(=O)CC2CCCSC2)C1 76814,Cc1cc(C(=O)NC2CN(C(=O)CCc3ccco3)CC2F)cc(Br)c1 76815,N1(C(C(CCC)C(C)C)=O)CCN(C(=O)CC2CCCCC2F)CC(C)(C)C1 76816,S(=O)(=O)(c1cccc(N2CCOC3(CCC3)CC2)n1)NC1CC(C)OC1=O 76817,N1(C(CCn2cc(C)nc2)=O)CCc2cnn(-c3ccc(C#N)cc3)c2C1.C(=O)(CN)N 76818,N1(C(C(CCC)C)C(=O)NCC)CCc2c(-c3ccc(N)cc3)cccc2C1 76819,c1(C(C)OC(=O)C(N)C2(C)CC2)cnnn1-c1ccccc1 76820,C1(C(=O)NCC2CN(C(CCN(C(C)=O)C)=O)C2)CCCC(C(F)(F)F)O1 76821,C(=O)(CCC(C)OC)N1CC(CC(C(=O)NCC(C=C)(C)O)F)C1 76822,c1(OCC(=O)NCC(C2CCN(C(CC=C)=O)CC2)(C)O)ncc(CC)cc1Cl 76823,N1(C(COCCCCOC)=O)CCC(C(CO)NC(C2(C)CC3CC3C2)=O)CC1 76824,c1(C(C)=O)nc(C(=O)NC2CC(CCNC(c3cnn(C(C)C)n3)=O)C2)cs1 76825,c1(CN2CCC(N(C(C)C)C(c3ccc(CO)cn3)=O)C2)ccc(C#N)c(Cl)c1 76826,N1(C(CN2CCN(C)CC2)=O)CC2CCC(C1)C2CNC(=O)Cc1ncccn1 76827,CC#CCCC(=O)NCC1(F)CC(CNC(c2c(Cc3ccc[nH]3)noc2C)=O)C1 76828,c1(OC)cc(C(=O)NCC2CCC2NC(=O)C(C)SC)cnc1OC 76829,C12(NC(c3ccc(CCC)[nH]3)=O)CC1CN(C(=O)C(CC)n1cccn1)C2 76830,C1(CNC(c2c(OC)cccn2)c2nnnn2C2CCC2)CC2CCC(C1)O2 76831,c1(C(=O)NC(CC)CN(C)C(C2(C(N)=O)CC2)=O)cn(C)c(=O)c2cncn12 76832,c1(OC)ncc(C)cc1NC(=O)CC(C1CC1)NC(=O)CC(C)C(C)C 76833,C1(C(=O)NCC(COC(C)C)O)CC(NC(=O)Cc2cccnc2O)CCO1 76834,c1(SC(=O)C(c2nnc(Cc3onc(C(=O)OC)n3)s2)C)ccc2c(c1)CCC2 76835,N1(C(COCC)=O)CC2COCC(C1)C2NC(=O)CCC1CCC(=O)N1 76836,c1(OC)ccc(C(=O)NC2CCC(C(=O)NC3(C)CCC(C)C3)C2)nc1 76837,C1(CC(=O)NCC2C(CNC(C3C(CC(C)C)C3)=O)C2)CC=CCC1 76838,N1(C(C2(C#C)CC2)=O)CC2(CCN(C(C3C4CCC3(c3ccc(F)cc3)C4)=O)C2)C1 76839,C=Cc1ccc(C(N2CC(O)CC2C(=O)Nc2cnc(C)c(CC)c2)=O)cc1 76840,c1(CC)ccc(C)cc1C(=O)NCC(CNC(c1cc(C)on1)=O)S(C)(=O)=O 76841,c1(C(N(CC(=O)NC2CCC(C#N)C2)C2CC2)=O)coc2c1COC2 76842,c1(NC(C(C)N(C(=O)COCCCN=[N+]=[N-])C)=O)cncc(Cl)c1 76843,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccnc1C)NCC(CC)(C)OC 76844,c1(NC(c2cccc(C(=O)NC3CC3)c2F)=O)cccc2nsnc12 76845,N1(C(C(C)CCN(C)C)=O)CCC2(CCC(N(C)C(c3nccn3C)=O)CC2)C1 76846,c1(C(C(=O)NCCC)N(CC(O)CCO)CC)cc2c(cc1OC)CCC2 76847,C1(NC(C(c2n(C)ccc2)=O)=O)CCN(C(=O)CCCC2CC2)CC12CCC2 76848,N1(C(C2C(CNC(C3CC34CCOC4)=O)CCO2)=O)CCN2C(=O)CCC2C1 76849,c1(C(=O)NCCC2(O)CCCN(C(C3(C(N)=O)CC3)=O)C2)cc(S(C)(=O)=O)co1 76850,C1(OCCC(C(=O)N(CCOC)Cc2cn(C(C)(C)C)nn2)C)CCOC(C)(C)C1 76851,N#Cc1c[nH]c(=NC23CCCC2CN(C(C2CCN2C2CC2)=O)C3)c2ccccc12 76852,C1(c2n(CCCCCC)nnn2)(NCC)CC2CSCC2C1.C(=O)(C1CC1)OC 76853,c1(C(=O)NC2CCCN(C(=O)CO)C2)cnc2[nH]nc(O)c2c1 76854,CC1(C)C(NC(=O)CC2(C)CC2(Cl)Cl)CCN1C(=O)COc1ccsn1 76855,C12(NC(c3c(OC)c(=O)cco3)=O)CCCC1CN(C(c1cc(=O)n(C)o1)=O)C2 76856,CCC(C)C(=O)C(=O)N1CCC(F)(C(=O)N(C)Cc2ccncc2C)CC1 76857,N1(C(C(C2(Cl)C(OC)C2)=O)=O)CCOC(c2cn(-c3cccc(C)n3)nn2)C1 76858,C12(NC(C(C)C(C)(C)C)=O)CCCC1(F)CN(C(c1sccc1CC#N)=O)C2 76859,C1(CC(=O)NCC(CC)N(C(CCN(CCC)C)=O)C)CC(O)C1(C)C 76860,C1(C)(C(=O)OC)CN(C(=O)C(C2CC(F)(F)C2)O)C1.c12cc([nH]n1)CNC2=O 76861,CC(C)C(C)CC(=O)N(C1CC(C(=O)NC(C)CS(C)(=O)=O)C1)C 76862,O=S1(=O)CC2CN(c3ncccc3S(=O)(=O)NCC3CC3C3CCCCC3)CCN2C1 76863,c1(C(C2(CN3CCN(C(F)(F)CO)CC3)CC2)=O)csc2cc(Cl)ccc12 76864,CCCC(C(=O)N(CC(C)(C)NC(C1CC(SC)C1)=O)C)OCC 76865,c1(NC(=O)NCCc2ccc(CC)cc2)ccc(Br)c(Br)c1 76866,N1(C(=O)NC2CC(F)(C(N)=O)C2)CCC(C(O)CO)CC1.c1(C2C(C)C2)ccco1 76867,c1(Oc2scc(CC3C4CN(C(=O)OC(C)(C)C)C3C4)n2)cccc(Cl)c1Cl 76868,c1(CN2CCC(N(C(c3cccc(C)c3)=O)C)C2)c(F)cccc1Cl 76869,N1(C(CCC=CC)=O)CCCC(NC(=O)COCC2CCOC2)C1C 76870,CS(=O)(=O)c1cnc(CCNC(=O)NC2COCC2N)nc1 76871,CC1CCC(C)C1NC(C1C=CC(NC(c2cc(C#N)c[nH]2)=O)C1)=O 76872,c1(C(N2CC(CNC(Cc3cnc(C)s3)=O)CC2(C)C)=O)cc2scc(C)c2[nH]1 76873,c1(OCC(=O)NCC(C)N(C(C#CC(C)C)=O)C)cc(Br)ccc1F 76874,C(=O)(CC(C)(C)C(=O)OC)N1CC(CC(=O)NCCCCCCC#C)(OC)C1 76875,C(=O)(CC(COC)NC(C1(C)CNC(=O)N1)=O)NCC1CCC(C)C1 76876,C(=O)(C(C)CC(C)(C)C)NCC1(C(N2CCC(SCC)CC2)=O)CCOC1 76877,c1(C(N2CCN(C(C3N(C(C)C)CCCC3)=O)C(C)C2)=O)ccccc1N=[N+]=[N-] 76878,C1(CC=C)(C(=O)NC2CCCC2CNC(=O)CCSc2n[nH]c(=N)s2)CCCC1 76879,Cc1onc(C(N2CCCC2c2ncc(-c3cnccc3Cl)[nH]2)=O)c1Br 76880,c1(C(=O)NCCCC2N(C(C#CC(C)C)=O)CCC2)nccc2c(Cl)cccc12 76881,c1(C(=O)NC(C(C)NC(c2cccc(CO)c2)=O)C)ccc(O)c(N)n1 76882,C(=O)(CCCCCC(C)O)NCC1CC(NC(c2cc(C)c(C)[nH]2)=O)C12CCC2 76883,N1(C(C(CC)Cl)=O)CC(O)C(O)C(O)C12CCN(C(=O)OC(C)(C)C)CC2 76884,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(C)s2)cc(OC(C)C)cc(F)c1 76885,C(=O)(C(C1CC1)N(C)CC1SCCS1)NCC=C 76886,C1(NC(C(C=CC)O)=O)CCCC(C(F)(F)F)C1.n12cc(nn1)CCNCC2 76887,C(CNC(=O)C(C)Cc1ccccn1)(CC(F)(F)F)NC(C=C(C)C(F)F)=O 76888,Cc1ccc(Br)c(C(=O)N(C2CCN(Cc3c(C)cccc3O)C2)C)c1 76889,c1(NC(c2c(CNC(c3cnsc3)=O)ccs2)=O)cnc2ccnn2c1 76890,C(=O)(C(C1=CCSC1)N1CCc2n[nH]cc2C1)NCCSC 76891,c1(C(C)C)ccc(C(=O)N(C(C)CNC(=O)CN2CCCS2(=O)=O)C)cn1 76892,c1(CN2C(C(N(CC(F)(F)F)CC)=O)CC2)ccc2cnccc2n1 76893,C(=O)(C(F)CCC(C)(C)C)N(C(C)C(N1CCC(CO)C(C)(C)C1)=O)CC 76894,S(=O)(=O)(c1nc(=N)[nH]c(=N)[nH]1)N1CCN(C(C)C)CC1.c12ccc(c(C#N)c1)[nH]2 76895,CC(CC(C)(C)O)c1nc(-c2ccccc2C(c2cccnc2)N(C)C)no1 76896,C(CCCCC(=O)NC1CCCCCC1C(=O)NCCCOC(=N)O)OCC 76897,C(=O)(C1=CC2CC=CCC12)N1CCC(C2CN(C(c3c(C)[nH]c(=NCC)s3)=O)C2)CC1 76898,Cc1c(C(=O)NC2CN(C(C34CCCN3CCC4)=O)CC23CC3)cccc1Cl 76899,CCC(CC(F)F)C(=O)N1CCC(NC(=O)CC2CC3(CCC3)CO2)C12CCC2 76900,N1(c2c(C)c(N3CC4C(C3)C4(F)F)ncn2)CCC2(CC1)OCC(C)(C)CO2 76901,Cc1cc(C(N2CC(F)CC2CN(C)C(C2CN3CCN2CC3)=O)=O)cnc1C 76902,C#Cc1ccc(C(=O)N(CCCNC(c2cc(C)n(CCO)n2)=O)CC)c(C)c1 76903,CN1CCC2(C1)C(=O)N2.C(=O)(C#CC1CC1)Nc1ccccc1OCF 76904,N1(C(COCCOC)=O)CCCC(C2CCCN(c3nnc(C#N)s3)C2)C1 76905,c1(SCC(C(=O)NC(CC2C(CC)C2)=O)N(C)C)cccc2c1NC(=O)CO2.C 76906,C(=O)(C(C)(O)C(F)(F)F)N1CCC(OCCNC(c2c(O)ncc(SCC)c2)=O)C1 76907,C1(NC(c2ccc(SC)s2)=O)CN(C(C2CC2C2CC2)=O)CC(F)(F)C1 76908,CCCC(CC(=O)NCCC(C(C)C)OC)NC(=O)CC1COCCO1 76909,C1(CNC(C(C(C)C)N2CCCCC2)=O)CCN(C(=O)CCC(F)F)C1(C)C 76910,Cc1cc(C)c(C(=O)NC2CCCN(Cc3cccc(Br)c3Cl)C2C)c(Cl)n1 76911,N1(C(C2(CCC)CCC2)=O)CC2(NC(=O)CC(C)F)CCC1C2 76912,c1(NCC(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cccc(Cl)c1 76913,c1(CCC(=O)NC(CC)CNC(=O)C(C2CCC2)OC)ccccc1C 76914,n1(CC)cc(-c2cccc(CS(C)(=O)=O)c2)c(C(=O)NC(CO)CCSC)n1 76915,C1(CC(=O)NC(c2cc(F)cnc2Cl)C)CCCCC1(F)F 76916,N1(C(CCc2c(C)n[nH]c2C)=O)CCC2(CCCN2C(=O)CC2CSCCS2)C1 76917,CCCCCCC(C)C(=O)NC(CN(C(=O)C(CC)n1cncn1)C)CC 76918,N1(C(C(CCC#C)O)=O)C2CCC1CC(C(=O)NCCOc1cc(Br)no1)C2 76919,C1(CC)CCN(C(=O)C(C)Cc2ccccn2)C1CNC(=O)Cc1cccnc1 76920,CCC(CC(F)(F)F)C(=O)NC1CC(NC(=O)CC(CN(C)C)C(F)(F)F)C1 76921,CS(=O)(=O)C1(C(=O)NC2CN(C(=O)CCOC3CCC3)C2)CCOCC1 76922,CC(C)(C)C(CNC(=O)CCCNS(C)(=O)=O)NC(c1cnccn1)=O 76923,CN1CCOC(C(=O)NC2CCN(C(=O)CC3CCC(C)(C)O3)C2)C1=O 76924,N1(CCNC(CCCOC)=O)CCC(NC(=O)C(C)Sc2ccccc2F)CC1 76925,c1(NSCc2snc(-c3cccc(C)c3)n2)nc(=NCC(C)C(C)C)[nH]c2ccsc12 76926,N1(C(=O)CCn2cnnn2)CCCC(n2cc(COc3ncccc3Cl)nn2)C1 76927,CCS(=O)CC(=O)Nc1coc(C2COCCN2C)n1 76928,C1(CNC(C2(CCNC(CC3C(CC)C3)=O)CCOCC2)=O)CC2(C1)CC(O)C2 76929,C1(CCOC)(NC(=O)CC2CC(C)C2)CCN(C(=O)CC2CCC(=O)O2)C1 76930,n1(CC)ncc(NC(C2CCN(C(=O)C(C(C)C)SC)CC2)=O)c1C 76931,c1(OC)cc(C(=O)NCc2cccc(NCC3CSC3)c2)cc(C)n1 76932,N#CC1CN(C(c2cccc3c2OCO3)=O)CCN1C(c1ccccc1)=O 76933,C(C(C)(Cn1cc(C)nn1)CC(=O)O)OC.C1(CC(=O)N)CCCCC1(F)F 76934,CCCC(C)(O)CC(=O)N1CCC(NC(c2cnc(S)nc2)=O)C(C)C1 76935,N1(C(C(c2cccc(Cl)c2)OC)=O)CC2CC(NC(=O)CC3CC(OC)C3)C2C1 76936,c1(C(=O)NCCNC(CC(C)c2ccco2)=O)ccnc(-c2ccco2)c1 76937,N1(c2c(CC)cnc(Cl)n2)CCC(C2CC2)C1CNC(=O)C(C)N1CC(C)C1 76938,N1(C(c2c(NC)snc2C)=O)CCN(C(=O)C(C)N(C)C)C(C(F)F)C1 76939,C(=O)(CCCCN(C)C(C)C)N(C1CN(C(c2c(C)nns2)=O)C1)C 76940,C(=O)(C(CCO)N(C)C)NCCC(=C)CNC(=O)CCCOc1ccccc1 76941,c1(C(N2CC3(N(C(c4c(C)cc(F)cc4)=O)CC3)C2)=O)ccc(C)c(C)c1Cl 76942,c1(CC(=O)N(CC(CC)NC(=O)C(C)(C)N(C)C)C)ccc(Cl)cc1C 76943,CN1C(=O)NCC1C(=O)NC1CCCN(C(=O)C(F)n2ccnc2)C1 76944,C(=O)(CC(C)CCCCC)N(C1CCN(C(c2cc(C)sn2)=O)C1)CC#C 76945,N1(C(C2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(C(C)C)c(F)c1)=O 76946,C(=O)(C(O)C(C)(C)CC)NC(CCC)C(=O)N1CCC2CC12 76947,CN1CCC(C(=O)N(CC(F)C(=O)N2CC(COC3CC4CCC3C4)C2)C)C1=O 76948,C1(CC(=O)NCCN(C(=O)C=C(C)C(F)F)CCOC)CNC(=O)C1 76949,O(P(C)(=O)CNC(=O)CC1(C)CCN1C(C1C2COCC12)=O)CC 76950,c1(C(=O)NCC2CC(NC(c3c(OC)ccnc3)=O)C2)ccc(F)c(O)c1 76951,c1(NC(=O)NCC23C(CN(C(C4C(COC)CC4)=O)C2)C3)cccc([N+](=O)[O-])c1 76952,CC(CNC(=O)C(CC1CC1)NC(=O)Cn1ncnn1)C(C)(C)C 76953,C1(C(C)NC(CCC)=O)CCCCN1C(C12CC(OC(C)=O)(C1)C2)=O.C(C)(C)(C)O 76954,c1(OCC)ccc(-n2nc(C(F)F)nc2-c2nnc(-c3ccccc3)o2)cc1 76955,c1(CC(=O)OCc2n(C)nnc2Br)cccc([N+](=O)[O-])c1C 76956,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCC2)ccn(C)c1C 76957,c1(CC)nnc(O)c(C(=O)NCC23CC2CN(S(=O)(=O)CCCCl)C3)c1CC 76958,c1(NCC)scnc1C(=O)NCC1CCN(C(=O)CN2CC3CC3C2)C1 76959,C(=O)(C(C)(C)COCc1ccccc1)NC(C)(C)CC=C(CCC)C.C1CC(=O)N1 76960,N1(C(C2(CC=C)CC2)=O)CCN(C2CCN(C(=O)CNS(N)(=O)=O)C2)CC1 76961,C1(CCOC)(NC(C2CCCN2C2CC2)=O)CCN(C(c2nc(O)sc2C)=O)C1 76962,C1(N(C(=O)CCCF)CC)CCCN(C(c2cn(C(C)C)nc2Br)=O)C1 76963,C1(C(=O)NC)CCN(C(=O)CCN(C(=O)CN2CCCC2C)C(C)C)C1 76964,c1(CCCC)cc(C(=O)NCC2CC(O)CN2C(c2ccc(Cl)cn2)=O)c(C)o1 76965,N1(C(c2c(OC)nsc2)=O)CCCCCC(NC(=O)CN2CCC(F)(F)C2)C1 76966,C1(NC(c2n(CCC)nnn2)C2(C)CC2(C)C)CC(=O)N(CC)C1 76967,c1(C(=O)NCCOCCN(C(C2C(CC)OCC2)=O)C)ccn2cc(C)nc2c1 76968,c1(OC)ccccc1C(=O)NCC1(CCNC(C2(CO)CCCO2)=O)CC1 76969,CC(N=c1nc2scnc2c(NCCS(=O)(=O)C(F)F)[nH]1)c1cncc(Cl)c1 76970,c1(CC(=O)NC(C)C2=CCNCC2)cccc(P(C)(C)=O)c1 76971,C(=O)(CCCC(C)(C)C#N)N1C2(CNC(C(CC)O)=O)CC(C1)C2 76972,C(C1(C)OCCc2ccccc21)NC(C1CN(C)CCO1)C 76973,N1(C(=O)N(c2ccccc2F)c2cncs2)CCCC(Nc2ccccn2)C1 76974,c1(C(C)=O)ccc(Cl)c(N(C(=O)CN2CCCC(OC(C)C)C2)C)c1 76975,N1(C(COCC(C)(C)C)=O)CCN(C(c2ccc(CCO)cc2)=O)CC(C)(F)C1 76976,CC(C)CCC(C(=O)NCCC(C)N1CCC1)NC(=O)CC1CCCOCC1 76977,C(=O)(C1=CC2C=CC(C1)C2)N1CC(C(=O)NC2CC23CCCCC3)C(C2CC2)C1 76978,c1(C(NOCCC(C)=O)=O)ccc(-c2cn(CCCCCO)nn2)o1.C(=O)(C(C)C)OC 76979,c1(C(C)=O)cc(C(N2CCOC(CCCNC(=O)C3=COCC3)C2)=O)cc(C)c1 76980,S(=O)(=O)(c1ccc2nc(N3CC4CC=CCC4C3)sc2c1)N1CC2C(C)(CC2)C1 76981,N1(C(C2C(NC(c3c(C)n(C)nn3)=O)C2(C)C)=O)CCOCC(O)C1 76982,Cc1c(N)ccc(C(N2CCC(C)C(NC(C3CCCC3(F)F)=O)C2)=O)c1C 76983,Cc1nc(C(=O)NCC(N2CCN(C(=O)C(C(C)C)N(C)C)CC2)=O)ccc1C#N 76984,C1(CCC(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)CC(C)(C)CO1 76985,N1(C(CC(CC)SC)=O)CCCCC(C2CN(C(=O)C=Cc3ncc[nH]3)C2)C1 76986,CC1(C)CC(NC(C2(C)CCCN2C(N)=O)=O)c2cc(C(F)(F)F)ccc2O1 76987,c1(C(=O)NCC2C(CNC(c3nc(SC)sc3)=O)CC2)cc(C)n(C)n1 76988,CCCC(CC(=O)NCc1c[nH]nc1C1CCC1)NC(=O)OC(C)(C)C 76989,c1(C(=O)NCC2(C)CCN(C(C(CC)SC)=O)C2)ccc2c(c1)C=CCC2 76990,N1(C(c2c(OC)ccs2)=O)CCC(CC(C)NC(=O)C(C)(C)CC)CC1 76991,c1(C(=O)NC(C(C)C)CNC(c2ccc(C3(C)CC3)cc2)=O)ccc([N+](=O)[O-])[nH]1 76992,c1(OC)ccccc1C(N1CCC=C(F)C1)C(=O)NCCCOCC1CC1 76993,C12(NC(CCN(C(C=C(COC)C)=O)C)=O)CCC(C1)OC2C 76994,C1(NC(C(CC)C(C)C)=O)C2CCCN(C(c3cc(Cl)nnc3O)=O)C2C1(C)C 76995,CC(O)C(C)(C)C(=O)N1CC2CC1(C(=O)NCCCn1cncn1)C2 76996,c1(CC)ccc(C(=O)NC2(CNC(C3NC(=O)C4CC34)=O)CCC2)cc1F 76997,C1(CNC(c2ccc(CCC)cc2)=O)CCC(C)CN1C(=O)CCc1nncs1 76998,C=CC(C)(O)CC(=O)N(CCC(=O)N1CCC(O)C1CC)OC 76999,c1(C(=O)NCC2CCC(NC(C3CC=CC3)=O)CC2)c[nH]c2nc(Br)ccc12 77000,c1(C(N2C(C)CCC(NC(c3csc4cncn34)=O)C2)=O)cc([N+](=O)[O-])ccn1 77001,c1(C(=O)NCC2CN(C(=O)CCc3cccs3)CC23CC3)cnc2[nH]cnc2c1 77002,C(=O)(C(O)CC(N)=O)N(CCCC(=O)NC(CC)Cn1cncn1)C 77003,C1(NC(C2(COC)CCCCC2)=O)CCC12CCCO2 77004,c1(C(=O)OC)coc(CNC(=O)C=CC(=O)NC2CC2)n1 77005,CCCS(=O)(=O)N1CCCC1C(=O)NC12CC(CNC(=O)C(C)C)(C1)C2 77006,c1(CNC(C2(CC)CCCO2)=O)nc(CNC(c2cncnc2)=O)cc(O)n1 77007,CC(C)C(F)C(=O)NC1COCC1C(N1CCN(c2nncs2)CC1)=O 77008,C1(C(N(CCC(=O)NCCCCOC)C2CC2)=O)CCC(=O)CC1C 77009,N1(C(CNC(=O)OC)=O)CCC(C2CC2)C1CNC(c1n[nH]c2c1CCOC2)=O 77010,C1(C)(CC(=O)NCCCOC)CN(C(=O)COC2CCC2)C1 77011,n1(CC(C)C)nccc1C(C(=O)NCC(F)F)N(C)CCC1CCC1 77012,c1(C(=O)NC(CC)CNC(c2cc(O)cc(Cl)c2)=O)nc2sccn2c1C 77013,N1(C(c2cc(COCC)oc2C)=O)CC2(CC2)CC1CNC(C1(C)CC(F)C1)=O 77014,N1(C(C(C=C)O)=O)CCC2CCCN(C(=O)C=CCOc3ccc(F)cc3)C2C1 77015,CC1CC(=O)NC(C(=O)NCC(O)CNC(=O)C(=O)NCCC(N)=O)C1 77016,c1(CNC(=O)CC2CCCO2)cccnc1CNC(C1CCC(F)(F)C1)=O 77017,CCCC(CNC(C1CC(CC2CC2)C1)=O)C(=O)NC1CCCCC1C#N 77018,CCC(C)(C)C(O)C(=O)NCC1CN(C(=O)COC2(C)CCOCC2)CC1(C)C 77019,CN1CCn2nc(CNC3CCc4ccc(C(F)(F)F)cc43)cc2S1(=O)=O 77020,c1(C(=O)NCC(CC)NC(=O)C(C)N2CCC2)ncc(Br)cc1F 77021,N1(c2nc(=N)[nH]c(N3CCCC(F)C3)n2)CCOC2(CCCOC2)C1 77022,c1(C(N2CC(CNC(C(COC)O)=O)C3(C2)CCC3)=O)cc2c(nc1N)CCC2 77023,c1(CC(=O)NC)ccc(-n2cc(C(C)NC(=O)CCC3OCCO3)nn2)c(C)c1 77024,Cc1n[nH]c(=N)n1-c1cccc(C(=O)NC(c2ncon2)Cc2ccccc2)c1 77025,C(CCC(=O)NC(C)CN(C(=O)C(C)CSC)C)OCCC 77026,CCCCC(CNC(=O)CCC(C)=O)NC(c1csc(C)c1C1CC1)=O 77027,c1(NCCc2ncc(CC)cn2)nc2ccccn2c1[N+](=O)[O-] 77028,N=c1nc(C2CCCC2)[nH]c(=NC2CCN(C(c3cc(C(F)F)[nH]n3)=O)CC2)[nH]1 77029,C1(C)(C(=O)NC2(CC(=O)N(C3CCC(F)(F)C3)C)CCC2)CCC2CC2C1 77030,C1(C(=O)NCCn2cc(CNC(C(C(C)C)C)=O)nn2)CCCCNC1=O 77031,Cc1cc(Cl)cc(Cl)c1OCC(N1CCC(CCNC(C2CC(C)CO2)=O)C1)=O 77032,C1(C)(CNC(C2C(OC)CC2)=O)CCN(C(c2cc(N)c(O)c(F)c2)=O)CC1 77033,C(=O)(CCCNC(C1CC1C)=O)N(C)CC1(CNCC(c2ncc[nH]2)C)CC1 77034,c1(C(N(CC(C)NC(c2ccc(C(C)(F)F)cc2)=O)C)=O)ccc(N)c(O)c1 77035,c1(N(C)C)ccc(CN2CCOC(C(=O)Nc3nncn3C)C2)c(F)c1 77036,CCC(CC)C(c1nnnn1CCCF)Nc1cnccc1C 77037,N1(C(C(=O)NC2C(C(=O)OC)CN(C(C)=O)C2)=O)CCCCC(C)C1 77038,Cc1cc(C(N2CC(NC(c3cc(Cl)ccc3N)=O)CC(F)C2)=O)c(Cl)cn1 77039,CCCC(C(=O)N1CCC(OCC(=O)NCCC2CC(C)(C)C2)C1)NC(C)=O.C 77040,C1(NC(C(c2cccnc2)OC)=O)(CO)CN(C(=O)CC2C=CCC2)C1 77041,C(=O)(C(Cn1cncn1)N(CCc1ccco1)CC1OCCCOC1OC)OC 77042,C1(OC)CCCC1C(=O)N(CCN(C)Cc1ccco1)C 77043,c1(N(C(=O)C(=O)Nc2cnn(CSc3ccccc3)c2)CC2CCC2)cccnc1 77044,C1(CC=C)(C(=O)NC(CCO)C2CCCC2)CN(C(=O)CCc2ccc[nH]2)C1 77045,c1(OCC)cc(C(=O)NC2(CNC(C3CCC3(C)C)=O)CC2)on1 77046,c1(C(N2C(Cn3cc(CC(C(=O)OC)OC)nn3)CCC2)=O)ccccc1C(N)=O 77047,N1(C(C(F)=CCC)=O)CCC2CN(C(c3cn(CC)nn3)C3CCC3)CC2CC1 77048,CC(C(F)F)=CC(N1CCC1CNC(=O)COCCOCCO)=O 77049,c1(CNC(c2cnn(C)c2C)c2n(C(CC)C)nnn2)cc(F)ncc1C 77050,C(=O)(C(C)S(C)(=O)=O)N(CC(C)NC(C=C(CCC)C)=O)C 77051,c1(OC)ccc(CC(=O)N(C)CC2CCCN2Cc2ccccc2)cc1O 77052,CN1CCN(C(=O)CC2CNC(=O)O2)CC1C(=O)NCC1(C)NC(=O)NC1=O 77053,c1(OCCC(=O)N(C(C)CCNC(=O)CC2CCCN2C)C)ccccc1F 77054,N1(C(C=CC)=O)CCC(C)(C)C(CNC(C2CCOC2)=O)C1 77055,c1(CNCc2c(OCC)scc2)sc(-c2cccc(F)c2)nc1C 77056,C(=O)(CCC(=O)N(CCC(C)NC(C1CCCN1C1CC1)=O)C)NCCC 77057,C1(CC#C)(C(=O)NCCCN(C(=O)Cn2cc(Cl)c(C)n2)C)CC=CCC1 77058,c1(C(=O)NCC2(CCNC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)cc(C#N)c[nH]1 77059,c1(C(=O)NC2C(NC(C3CCC(C)(C)O3)=O)CCC2)cc(N)c(Cl)cn1 77060,C(=O)(CC(C)(C)CNC(=O)C(CC(C)C)OC)NC1(C(=O)NC)CCOCC1 77061,c1(C(C(=O)N(CCCCCNC(C(C)OCC)=O)C)O)cccc(Cl)c1 77062,CC1C(NC(C2CCCCCC2)=O)CCN1C(=O)C(c1cccc(Cl)c1)C 77063,N1(C(CS(C)(=O)=O)=O)CCC2(CC1)CCN(C(C1CC13CCOCC3)=O)C2 77064,N1(C(CCOCC(=O)NC(C(F)(F)F)C2CC2)=O)CCC(c2cnn[nH]2)C1 77065,N1(C(CCC(=O)OCC)=O)CCC(C)C(CNC(=O)Cc2cc(C)ccc2F)C1 77066,N1(C(=O)OC(C)(C)C)CC2CC1(CC(=O)NCCc1cnc(O)nc1O)CO2 77067,c1(C(N(C)CC2N(C(C(CN(C)C)O)=O)CCC2)=O)ccsc1C#N 77068,c1(C(N(CCOCCNC(C2(C)C(CC)CCC2)=O)C)=O)c(C)nc(C)n1O 77069,C1(CNC(C(C)SC)=O)N(C(=O)CCn2cccn2)CCC1(C)C 77070,c1(CCN2C(CC(=O)NC(COC)C(C)C)CCC2)ccc(OCl)c(O)c1 77071,c1(C(=O)NCC(CN(C(C2CC2F)=O)CC)(C)C)ncccc1Br 77072,C1(NC(CN(C)C(N)=O)=O)(CNC(=O)CC2CCCOCC2)CC(F)(F)C1 77073,c1(C(C(C)NCC(c2ccc(F)cc2)CO)C)cc(F)cc(F)c1 77074,C1(CNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C 77075,Cc1ccc(O)c(CC(=O)NCCC2(C(=O)NC(C)CC(C)C(F)F)CCC2)c1 77076,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cccc(C#N)c2)=O)CC1 77077,N1(C(c2c(C)n(C(C)C)nn2)=O)CC(CNC(=O)C#CC2CC2)CC(C)(C)C1 77078,C1(NC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cc2cccc(C)c2C)C(C)C1 77079,c1(CC)cc2n(n1)CCN(C(=O)C(C(C)C)OCC(C)C)C2 77080,NS(=O)(=O)CCCCCCC(=O)N1CC(C2CN(C(C3C4CC5C(C4)C35)=O)C2)C1 77081,Cc1nn(C(C)C)cc1C(=O)NC(C)(CNC(=O)C(C)C(C)O)C(C)C 77082,c1(C(N2CCC(CCNC(C3=CCCC3C)=O)C2)=O)ccc(Cl)c(Cl)c1N 77083,n1(CC(=O)NCC2(C(N(C(C(C)SC)C)C)=O)CCCC2)cccnc1=O 77084,C1(CN(C(=O)Cc2cn(C)nc2Cl)C)CCN(C(=O)CCN2CCCCC2)CC1 77085,c1(N2C(C)CNCCC2)nc(=O)c2c(Br)c[nH]c2[nH]1.C(=O)CCC(F)(F)F 77086,C(=O)(CCC(=O)NC1COCC1NC(c1cnc(C(N)=O)s1)=O)N(C(C)C)C 77087,C1(CNC(CSCC#C)=O)CN(C(c2cccc(F)c2CC)=O)CCC1(C)C 77088,c1(N2CCC(N(CCCO)CC)CC2)ncnc(C)c1F 77089,N1(C(CN2CCCC(CC)C2)=O)CC=C(CNC(c2ccsc2)=O)CC1 77090,CCC(CNC(c1ncccc1F)=O)(CC)C(=O)NC1CC1C1CCC1 77091,N1(C(C=CC)=O)CCOC2(CCC(NC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)C1 77092,CC1CN(CCCNC(=O)CCCn2cc(CNC3(C)C=CCC3)nn2)CC(C)O1 77093,C1(CC)CN(C(c2cn(C(C)C)nn2)=O)CCC1NC(C1(C)CCN(C)C1=O)=O 77094,C(=O)(CS(=O)CCC(F)(F)F)NC1C(CNC(C=Cc2n(C)cnc2)=O)CC1 77095,c1(C(C)=O)cccc(C(N2CC3(NC(=O)CC4(O)CCOCC4)CC2C3)=O)c1 77096,c1(NC(C2C(OC)(OC)CC2)=O)cncc(-n2nnnc2C)c1.C(C)(C)O 77097,N1(C(C2CCC(C(=O)OC)C2)=O)CC(C(=O)NC(C)CC(C)C(F)F)CC1(C)C 77098,C1(C(N(CC(C)(C)NC(C2(CCCC)CC2)=O)C)=O)CC(=O)NC(C)C1 77099,c1(OC)ccc(OCC(C)OC2CCCCC(=O)N2)cc1[N+](=O)[O-] 77100,C(=O)(C1CCCn2c(Br)cnc21)NC1CC(NC(c2ccc(C#N)[nH]2)=O)C1 77101,Cc1cc(N2CCN(C(C3CCCC4(CCC4)O3)=O)CCC2C)n2ncc(C)c2n1 77102,C1(O)(C(C)NC(=O)CNC(=O)C(C)(C)n2cc(Cl)cn2)CCN(C(=O)C2CC2)C1 77103,N1(C(C(C2CC(NC(CCN(C)C)=O)C2)F)=O)C2CCC1CC(CO)C2 77104,C1(OC)CC(NC(c2sccc2SC)=O)C12CCN(C(=O)C1=CCCCC1)CC2 77105,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77106,C(=O)(C(O)COCc1ccccc1)N(CCC)CCNC(=O)CNC=O 77107,c1(OCC)ccccc1C(C(=O)NCCN(C(C1(F)CC1)=O)C(C)C)OC 77108,O=C(CCCCCCNC(c1cc2ccoc2cn1)=O)NCc1cnn[nH]1 77109,C1(N(C(=O)Cn2ccsc2=N)C)CCCN(C(=O)CC2CCCCCO2)CC1 77110,C1(N(C)C)CCCN(C(C2CC(O)CN2C(c2ncncc2N)=O)=O)CC1 77111,c1(SC)nc(O)nc(C)c1C(=O)NC(C1CCCCN1C(=O)C(C)C(C)(C)C)C 77112,C1(C(N(CCNC(C(C(C)c2ccccc2)O)=O)C(C)C)=O)CC2C=CC1CC2 77113,Cc1ccc(C(=O)NC(C)(C)CC2CCN(C(C3(O)CC3(C)C)=O)CC2)nc1 77114,n1(CC)cnc2[nH]c(=NCC3CCCC3O)nc(N3CCCC(COC)C3)c12 77115,N1(C(c2ncc(Cl)s2)=O)CCOC(NC(C2(C)CC2)=O)C1.C1(C)CCS(=O)(=O)C1 77116,C1(NC(c2ccc(C(C)C)cn2)=O)CCC(C)N(C(C2CCOC2C)=O)C1 77117,C1(N(C(n2ncc(C)c2)=O)CCF)CCCN(C(c2scnc2C(C)C)=O)C1 77118,N1(C(C2CC(CC)C2)=O)CC2CCCN2CC1COC.C1C(=O)N1C1CC1 77119,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77120,c1(-n2cc(CNC(CCc3nc(C)sc3)=O)nn2)cccc(C(N2CCCC2)=O)c1 77121,c1(NC(CC)=O)cccc(CNC(C2C=CCN2C(c2ccoc2I)=O)=O)c1 77122,c1(OC)cc(Cl)cc(Cl)c1NC(c1c(NC(c2cnc(C)s2)=O)cccc1F)=O 77123,N1(C(CSCC#C)=O)CCN(C(=O)C=C2CCC(C)CC2)C(CC(F)F)C1 77124,c1(C(=O)NC2(CNC(C3N(N=O)CCC3)=O)CC2)cc(O)ccc1F 77125,CCCC1C(O)C(=O)N2CCCCC2C(=O)N1.C(=O)(CC(C)(C)CCOC)N.OC 77126,C#CCC(C(=O)NOCC1CC1)NC(C1CC12CCC2)=O 77127,c1(C(=O)NCC(CN(C)C(c2cnn(C3CCCCC3)c2)=O)O)cccc(O)c1 77128,C1(NC(c2cnc(CCCC)s2)=O)C2CCN(C(=O)CC(=O)OCC)CCC12 77129,C12(CCNC(CCCC=C)=O)CCC(CC1)N(C(c1ncn3c1CCC3)=O)C2 77130,c1(C(=O)NCC2C=CCN2C(=O)CC2CC2)c[nH]c2ccc([N+](=O)[O-])cc12 77131,N1(C(C=Cc2c(C)ncs2)=O)CCCC2(CCCN2C(=O)CC(C)O)C1 77132,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77133,C#CC1(OCCNC(=O)C(C2CCN(C(=O)C(O)C3CC3)C2)C)COC1 77134,C(N=c1cccc(S(=O)(=O)NC2COCC2CO)[nH]1)C1CC(C)(C)C1 77135,C=CC1(C(=O)NCCCCCCF)CCN(C(=O)CC(CC)CC)C1 77136,c1(C(CO)NC(c2cc(Cn3cc(Br)cn3)no2)=O)ccccc1Br 77137,c1(C(=O)NC2CN(C(C3(CCC=C)CC3)=O)C2)cc(S(N)(=O)=O)c(F)c(F)c1F 77138,C(=O)(C1=CS(=O)CCC1)NC1CC(N(C)C(C2CC2c2ccccc2)=O)C1 77139,c1(CCC(=O)N(CC(O)CN(C(=O)C=CBr)C)C)c[nH]c2ccccc12 77140,N12CCN(CC1)c1ccc(cc1)C2=O.C1(SC)(CNC(C2CCSC2)=O)CCC1 77141,c1(OC2(CNc3c(COC)n(C(CC)CC)nc3)CC(C)C2)ccc(F)cc1F 77142,N1(C(c2ncn(C)c2)C(=O)NCc2cccs2)CCCC(N=[N+]=[N-])CC1 77143,N1(C(C2CCCCO2)=O)CC2CC(C(=O)NOCC3CCCC3)(C2)C1 77144,C1(CCNC(c2sc(CC)c(N)c2)c2nnnn2C)CCS(=O)(=O)CC1 77145,C1(C(=O)NCC(C)(C)C2CCC2)C=CCN1C(=O)COCCN(C)C 77146,C1(CNC(c2n(CC)ncc2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77147,c1(CN(C)C(C2CC(C)(NC(=O)OC(C)(C)C)C2)=O)ccc(OC)nc1 77148,C(=O)(C(C)N=[N+]=[N-])NCCNC(C1CN(C(c2ccc(C)s2)=O)C1)=O 77149,CC(C)(C)C(CNC(=O)Cn1cc(C#N)cn1)NC(C1COCCN1CC#N)=O 77150,Cc1cc(C(O)CNC(=O)Nc2cccc(C(=O)N(C)C)c2)ccc1F 77151,CN1CC(C(N2CC(F)(CNC(c3csc(C(N)=O)n3)=O)C2)=O)CC1=O 77152,C1(CC(N2CCC(C(C)O)CC2)C(=O)NCCOCC)Cc2ccccc2O1 77153,N(C1CCCc2c(C(=O)O)cccc21)C1CCC(C(=O)O)CC1 77154,C1(CNC(=O)CC2CC2)CCC2CN(C(C3CS(=O)C3)=O)CC12 77155,c1(C(N2CCC(NC(c3ccc(OC)s3)=O)(CF)C2)=O)cc2sc(C)nc2[nH]1 77156,C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)C)=O)CC(F)(F)C1(F)F 77157,Cc1ccc(OCC(=O)N(CCNC(C2(C(C)C)CNC(=O)C2)=O)C2CC2)cc1 77158,C(N=c1cc[nH]cc1)NS(=O)(=O)Cc1ccc(C(F)F)cc1 77159,c1(C(=O)NC(c2cccnc2)C(=O)NCc2[nH]nc(C(C)C)n2)ncncc1Cl 77160,C1(CNC(C(N2CCC(O)CC2)(C)C)=O)CCCCC1NC(=O)CCC1CCOC1 77161,Cc1cc2c(C(N3CC(NC(C4CC4(C)C)=O)C4(CCCC4)C3)=O)nccn2n1 77162,N1(C(CCS(C)(=O)=O)=O)CC(C)(CNC(c2csc(-c3ncc[nH]3)n2)=O)CC1(C)C 77163,N1(C(=O)NC(c2ccc(C(C)C)cc2)C)CCCC(C#N)(C(=O)OC(C)(C)C)C1 77164,C(=O)(C#CC1(C)CC1)NC(CC)CN(C(=O)CSCC1CCCO1)C 77165,CCCC(O)CC(=O)NC1CC2CC1N(C(=O)CC(COC)COC)C2 77166,C12(NC(CCc3onc(CSC)n3)=O)CCN(C(=O)C(C)(C)F)CC1C2 77167,CC1CN2CC(C)CN1C(=O)Cc1cccc2c1CCN 77168,c1(C(=O)NCCCN(C(=O)CNC(=O)C(F)(F)F)C2CC2)nnc2n1CCCCC2 77169,Cn1nc2c(c1C(=O)NC(C)(CNC(C1CC(O)(C#N)C1)=O)C1CC1)CCC2 77170,C1(C(C)C)CN(C(c2cnc(-c3ccco3)s2)=O)CCN1C(C1CNC(=O)N1)=O 77171,c1(CCCC(N2CCC(O)(CNC(CN3C(C)CC3)=O)C2)=O)ccc2c(c1)OCO2 77172,C1(CC=C)(C(=O)N(CC(C)(C)C)C)CCN(C(C2CC(CC)=NO2)=O)C1 77173,C1(NC(C(c2cncnc2)OC)=O)CCC(NC(C2CC(C)(F)C2)=O)CC1 77174,c1(NCc2nnc(SC)s2)cc2c(I)cnn2cn1 77175,C(=O)(C(F)(F)CC(C)C)NC(CN(C(c1cnc2ccnn2c1)=O)CC)C 77176,O=C(CCC(F)(F)F)NCC1C(C(N2CCC2)=O)CC(O)C(O)C1 77177,N1(C(CCc2ccc(C)s2)=O)CCC(C)C(NC(C2CCCNS2(=O)=O)=O)C1 77178,N#CC1(C(N2CC3CC3(CNC(=O)CCc3cnc(O)[nH]3)C2)=O)CC12CCC2 77179,c1(C(=O)OC)cc(C(=O)NC(CNC(=O)CSc2nccn2C)CC)ns1 77180,c1(OC)ccc(F)c(C(N2CCC(N(C(=O)CC3CC4CC4C3)C)C2)=O)c1 77181,CC1=C(CNC(=O)C(C2CCN(C(=O)CC3CCC(=O)C3)CC2)C)CCC1 77182,c1(C(=O)NCCN(C(C(CC)C#N)=O)C2CC2)cc(C)ccc1O 77183,c1(C(=O)NC2CC(CNC(C(C)Cn3ccnc3)=O)C2)cc(N=S(C)(C)=O)ccn1 77184,C=CC(CC)CC(=O)N1CCOCC1CN(C)C(c1cn(C(F)F)cn1)=O 77185,CC1(CNC(=O)CC2CC(O)CN2C(=O)COC2CC=CC2)CCCCCC1 77186,C1(N(C(c2cn(CC(CC)O)nn2)=O)C)CN(C(C2CC23CC3)=O)CC12CC2 77187,c1(C(=O)NC(C)CCCNC(=O)CSCCc2ccnc(Cl)c2)cccc(F)c1 77188,CC(C)C(O)CCNC(=O)C(CCF)NC(=O)COC1CCC1 77189,c1(C(=O)OCC)c(C)cc(C)nc1NC1CCN(CCCOC)C1 77190,C1(CC(=O)N(C)CC2CCN(C(=O)CS(N)(=O)=O)C2)CCC2(CCC2)O1 77191,CC1CC(NC(=O)Cc2ccco2)CN1C(=O)CC1CCCC(O)C1 77192,c1(N2CCN(C(N3CC(C)C(C(=O)NC4CC4)C3)=O)CC2)ccc(F)cc1F 77193,C12CCN(CC1)C(C)c1cc(on1)C(=O)N2C.C1(CC(C)C)(COC)CC1 77194,Cc1cc(C)c(C)c(C(=O)NCC2CCN(C(c3cnoc3CO)=O)C23CC3)c1C 77195,c1(C(=O)NCC2N(C(CC3(C=C)CCC3)=O)CC2)cccc(C)c1CC 77196,C12CC13C(O)C(CC3)N2.C(CN(C)C)(CC(C)C)NC(C(=O)OCC)=O 77197,C(=O)(CN=c1cc[nH]cc1)N1CC2C(NC(=O)CC3(O)CC3)(C2)C1 77198,c12cc(Br)cnc1S2.c1(C(C2CCCO2)(C)N(C)C)nnnn1C 77199,N1(C(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(=O)C3CC3)CC1C2 77200,N1(C(CN(CCN(C)C)C)=O)Cc2ccccc2C1C(=O)NCC=CCO 77201,c1(CC)cc(C(=O)NC2CCN(C(=O)C(CC)CC)C2c2ccccc2)c(C)o1 77202,C1(CC(=O)NCC2(OC)CN(C(=O)CCNC(N)=O)C2)CCCC(C#N)C1 77203,C(=O)(C1=CCC2CCC1N2C(=O)C(C)(C)CC)NCC(C=C)O 77204,CC(=O)CCC(C(=O)O)NS(=O)(=O)Cc1ccc(OCCN(C)C)cc1 77205,C(CC(C(=O)NC(C)C(C)N1CCCC1)NC(=O)CSC(F)F)SC 77206,C1(C)(CNC(c2cnn(CC)c2C)=O)CCCN(C(c2c(C#N)cnn2C)=O)C1 77207,Cn1nnc(CNC(=O)C(C)(C)C#N)c1C(=O)NOCCCF 77208,N1(C(CCc2n(C)cnn2)=O)CCOC2(CCN(C(=O)C=CCO)C2)C1 77209,c1(CC(=O)NCC(CC)NC(CC(C=C)C)=O)nn(C)c(=O)c2ccccc12 77210,c1(CC(=O)NCCO)csc(-c2ccncc2)n1 77211,N1(CC)CCC(C(=O)NC2CCCC(CNC(=O)C(COC)CC)C2)CC1 77212,CCC(C(=O)NC(C)Cc1ccco1)N(C(=O)CC1CCCN1C)C 77213,c1(CCC)ccc(C(N2CCCC2C2(CNC(=O)C(Cl)=CCl)CC2)=O)cc1 77214,c1(CN2CCC(C(N(C)Cc3ccccc3)=O)(C(=O)O)C2)cc(Br)cc(F)c1O 77215,CC1CN(C(c2c(F)ccc(F)c2F)C(=O)NCCCF)CCN(C)C1 77216,NC(CCC(=O)N1CCN(Cc2ccoc2)CC1)C(=O)O 77217,C1(CCC(=O)NC2(CCC)CCC2)CCCCN1C(=O)Cn1ncnn1 77218,C12SC3C=CC1CC3CN(CCCC)C(=O)NCC(C)NC2=O 77219,C1(C(C)NC(c2conc2CNC(C2(n3cnnn3)CC2)=O)=O)CC2CCC1C2 77220,N1(C(CCCCCNC(c2n[nH]c(CC)c2C)=O)=O)Cc2ccncc2C1 77221,c1(OCC(C)(C)CN2CCC3(C=CCO3)C2)nc2ccc(F)cc2s1 77222,N#Cc1ccncc1NC(=O)Cc1ccccc1NC(c1ncccc1Br)=O 77223,c1(C(=O)NC2C(C)CCN(C(c3scc(C)c3C)=O)C2)cnc(O)c([N+](=O)[O-])c1 77224,c1(CC(N2CC(Cn3cc(C(C)(C)C4CC4)nn3)C2)=O)ccccc1Br 77225,c1(CN(CCNC(C(n2cc(C(=O)O)nn2)C)=O)C)ccccc1 77226,C(CCCCCNC(C1COCC1(C)C)=O)N(C(=O)CCCN1CCCCC1)C 77227,C1(C(N(CC(C)(F)F)C)=O)CCN(C(=O)C2CCCO2)O1 77228,C#Cc1cncc(CNC(c2ncc(OC)cc2F)=O)c1 77229,C(c1cscn1)=CC(=O)NCCC1CC(NC(c2coc(-c3cccs3)n2)=O)C1 77230,C(=O)(C1=CCN(C(=O)CN2C(=O)CCCC2=O)CC1)Nc1c(CC)cccn1 77231,N1(C(CN2CC(C)OC(C)C2)=O)CC2CCC(CN3CCCCC3)(C2)C1 77232,C1(C)(C(N(CCCN(C(C(CC)C#N)=O)C)C)=O)CC2(CCC2)C1 77233,c1(C(=O)NCCC2CCCN2C(=O)CCC=CBr)cnc2c(=O)[nH]ccc2c1 77234,CC(C(=O)NC1(CNC(c2cn(CC(N)=O)nn2)=O)CCOCC1)S(N)(=O)=O 77235,C1(C)(C(N(CC(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)=O)CCOC1 77236,CC1CN(C(NOCCNC(=O)COc2ccn(C)n2)=O)CC1C 77237,c1(C(=O)NC2(CC)CN(C(=O)Cc3c(C)noc3C)C2)cc2c(s1)CN(C)CC2 77238,c1(CN(CCOC)C)cc(C)c2nc(C)nn2c1.c12cn(nn1)CC2 77239,c1(C(N(C2CCCN(C(C3(C)CC(F)C3)=O)CC2)C)=O)cn2cnnc2cn1 77240,Cc1cc(=NC(=O)C(=O)NC2CC3CN(C(=O)Cc4cc(C)[nH]n4)CC23)[nH]o1 77241,Cc1cc(=NCc2nc3ncccn3n2)[nH]c(N(C)Cc2cc(C)nn2C)n1 77242,C(C)(CC(=O)O)(c1n(CCOC)nnn1)NCCCC1OCCC1C 77243,C1(C)(NC(Cn2c(C)ccn2)=O)CCCN(C(=O)C2=COCCO2)C1 77244,Cc1ccc2c(c1)C(C(=O)N1CCN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC1CO)C2 77245,c1(NC(C2C(c3c(OC)nccc3)C2)=O)ncc(Br)cc1I 77246,N1(C(CC2(C)CC2)=O)CCC(C(F)(F)F)CC1CNC(=O)Cn1cccnc1=O 77247,N1(C(=O)NCCCCC)CCC2CCN(C(=O)CC(O)CCOC(C)(C)C)CC12 77248,N(C1CC2(CCCC2)Oc2ccccc21)C(=O)CCc1c(C(F)(F)F)cccc1Cl 77249,c1(C(=O)NC(CN(C(CCC(=O)N(CC)CC)=O)C)C)cnn2c1CCCC2 77250,c1(SC)nc(N2CC3CCN(C(=O)Cc4cscn4)C3C2)nc2ccccc12 77251,C1(CNC(c2cnc(OCC)c(Cl)c2)=O)(CC(C)C(=O)NC)CCCCC1C1CC1 77252,C1(C(=O)Nc2cccc(C(C)(C)C)c2O)C(C#N)CC12CCC2 77253,N12CC(C)(CC1(C)C)NC(=O)C1C(C1)C2.c1(NC(C)C2CC2)ccc(Cl)c(Cl)c1 77254,N1(C(C2C(C(C)C)C2)=O)CC2(CCCC2)C1C(N1CCC2C(C1)C2(F)F)=O 77255,C(C(C)(C)CCNC(c1ccn(CC(F)F)n1)=O)NC(Cc1c(C)ncs1)=O 77256,c1(OC(C)C)cccc(C(=O)NCCN(C)C(c2cc(C(C)(C)C)on2)=O)n1 77257,N1(C(C(=O)NC)C2CC(OC)C2)CCCC(C2CN(C(=O)OC(C)(C)C)CCO2)C1 77258,c1(CC(=O)Oc2c(SCC(=O)OC)c[nH]n2)cncc(C)c1 77259,CCCC(C)C(=O)NCc1cc(C(=O)NC(C2CCOC2)CO)ccn1 77260,C12(CC(N3CCCC(OC(C)C)C3)=O)CCC1CN(C(C1(O)CCOCC1)=O)C2 77261,CC(C)C(C(=O)NCCCn1cc(CC2(O)CCC2)nn1)n1cnnn1 77262,C(C(CNC(c1n[nH]c2c1CCC2)=O)S(C)(=O)=O)NC(C1OCC(C)(C)C1)=O 77263,N1(C(Cc2cn(C)nn2)=O)CCC2(NC(=O)CC(F)(F)C(F)(F)F)CCCCC12 77264,N1(C(c2occ(C(N)=O)c2)=O)CCC(C2CCN(C(=O)C(C)N3CCC3)CC2)C1 77265,C12(C(=O)NC(C3CCN(C(C4CCOCC4)=O)CC3)C)CCOC(C)(C1)C2 77266,c1(N2CCC(OCC(N)=O)C2)nc(N2CCC(n3cncn3)C2)c2[nH]ccc2n1 77267,C(=O)(C(C)CCC(C)(C)C)N1CCCC(N(C(c2cn(CC)nn2)=O)CC)CC1 77268,c1(NCC2(NC(=O)CC3(c4ccc(Cl)cc4)CC3)CC2)ccc2nccc(I)c2c1 77269,C1(C)(CNC(C(CCC)C)=O)CCCN(C(=O)C(CC)n2nccc2C)C1 77270,c1(CNS(CC)(=O)=O)nnc(C)s1.C1(C2CNCC(=O)N2)CCCCC1.C1C(=O)N1 77271,c1(C(N2C(CNC(CCOC(C)C)=O)CC(O)C2)=O)nccn2ccnc12 77272,n1(CC)ncc2c(C(N3CC(c4ccccc4NC(=O)NC)(O)C3)=O)ccnc12 77273,c1(C(C(=O)NC(CN(C(C(C)C#N)=O)C)C)C)cn(C)nc1C(F)F 77274,Cc1ccc(C(=O)NC2C=CCN(C(=O)CCOCC3CC3)C2)c(F)c1 77275,N1(C(c2cc(OC)n[nH]2)=O)CC(C(N2CCCC2C2(COC)CC2)=O)OC(C)C1 77276,CC(C)(F)C(C)(F)C(=O)NCC1(O)CC(CNC(c2cc(O)nc(Cl)c2)=O)C1 77277,c1(CCC)n[nH]cc1C(=O)NC(COC)C(=O)N(CCC(C)(C)O)C 77278,n1(CC(=O)NCC(CNC(C=C(C)C)=O)CO)c(-c2cccs2)nnc1S 77279,c1(C(=O)NC2C(OC)CN(C(=O)C(O)CN(C)C)C2)ccc(C)c(F)c1 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77315,N(C(=NCCCCC)N1CCc2c(cc(F)c(F)c2F)C1)C(C#C)(C)C.C1C(=O)N1 77316,CCCCC(C(=O)N1CCC(CN(C(=O)CCCC(C)C)C)C1)NC(N)=O 77317,N1(C(C(C)c2ccsc2)=O)CCCC12CCN(C(=O)CC(C)(C)N(C)C)CC2 77318,n12nc(C)c(c1C)C(=O)NCC1CCN1OC2.c1(C=O)ncccc1F.CC 77319,c1(C(=O)OC)cn(C)nc1C(N1CC(NC(=O)CNc2ccco2)C(F)C1)=O 77320,CCC(C)CCC(=O)NCCC(C)NC(c1ccc([N+](=O)[O-])s1)=O 77321,c1(CC(=O)NCC(C2CC2)NC(=O)CCn2ccnc2)ccc(Cl)nc1F 77322,c1(C(=O)NC(CC=C)CNC(=O)C(C(C)O)N(C)C)ccnc2[nH]c(C)nc12 77323,Cc1cc(C(=O)NCC(CNC(=O)CC#N)CO)n(C(C)(C)C)n1 77324,n1(CCC)ccnc1CN(CC(N1C(C(=O)NCC(=O)NC)CSC1)=O)C(C)C 77325,c1(C(=O)NCCC2CCN(C(CSCC=C)=O)CC2)csc2nnsc12 77326,c1(OCCNCCOCCOC(C(=O)OC)C)ccccc1 77327,n1(CCC)ccnc1CCC(=O)N(CC#N)CCc1ccsc1 77328,CCC(C)CC(C)NC(c1nnnn1C(C)(C)CC)C1(C(F)(F)F)CC1 77329,C1(NC(C(=O)NCC)=O)CCN(C2CCCCC2NC(C2(COC)CC2)=O)CC1 77330,CCCCC(O)C(=O)NCCC1CCCN(C(c2ccc(C)c(OC)c2)=O)CC1 77331,N1(C(C=CCN(C(CC2CC(CC)C2)=O)C)=O)CCCCC(C)(F)C1 77332,CCS(=O)(=O)CCn1nc(-c2cnn(CC)c2)nc1-c1cnc(OC(C)C)cn1 77333,c1(C(=O)NC2(CCNC(c3n(C(CC)C)ncc3)=O)CC2)cnc(C)c(N)c1 77334,c1(CNC2C(NC(c3ccc(Oc4ccccc4)o3)=O)C2)cccc(CO)n1 77335,N1(C(C(C)Oc2ccccn2)=O)CCC2CC1CN(c1ncnc3occc13)C2 77336,c1(-c2onc(CNC(=O)NC3CCCC=C3Br)n2)cccc(F)c1 77337,N1(C(C(C2CC2)OC)=O)CCN(C(c2cnn(Cc3ccco3)c2)=O)CC(O)C1 77338,C1(CNC(c2n(C)c(S)nn2)=O)CCN(C(=O)CC23CCC(CC2)C3)C12CCC2 77339,n1(CC)c(=O)n(CC(=O)NC(CNC(C2CCC2)=O)CC(C)C)c2ccccc12 77340,CC1CN(C(=O)CCC2CC2(Cl)Cl)CC2(CCN(C(C3CCCN3C)=O)CC2)O1 77341,c1(N(C)CCN(C2N(C(C(CC#C)O)=O)CCCC2)C)cc(C)nc(C)c1 77342,N1(C(c2c(C)nsc2)=O)CCCCC1CCCNC(C1CCS1)=O 77343,S(=O)(=O)(c1nc(C)cs1)Nc1cc(OC)c(OC(F)F)cc1 77344,N1(C(CC2(CC)CCC2)=O)CCCC2CCN(C(=O)CC3(C)N=N3)CC12 77345,N1(C(=O)Nc2csc(Cl)n2)CC(C(=O)NOC2CCSCC2)C2(CC2)C1 77346,N(C1COc2cc(Br)cnc21)C(N=S(c1c(C(C)C)nn(C)c1)(C)=O)=O 77347,C(CC(C(=O)NC1CCNC(=O)C1)NC(=O)CCc1ccoc1)N(C)C 77348,c1(C(C)C)c(C(=O)N(CC(C)NC(=O)CC2COC(=O)N2)C)cnc2ncnn12 77349,Cc1cc(CC(N2CC(NC(=O)C(=O)Nc3ncc[nH]3)CC(O)C2)=O)ccc1Cl 77350,CC1(C)CC(C(=O)NCCC2(O)CCN(C(c3c[nH]ccc3=O)=O)C2)=NO1 77351,CCCC(CCC)C(=O)N1CCOCC1CNC(=O)CN(C)CCOC 77352,C(=O)(C(C)Cc1cnn(C)c1)N(C1CCN(C(c2cc(Cl)ns2)=O)C1)CC 77353,C1(c2cn(C(CNC(C(C=C)(C)CC)=O)C)nn2)(OC)CC2(CCOCC2)C1 77354,C(C)(CCN=c1[nH]cnc2ccc(C(F)(F)F)cc12)NC(c1cc(C)nc(Cl)c1)=O 77355,c1(C(=O)NCC(=C)CCNC(=O)CSc2ccncc2)[nH]nc(CC)c1Cl 77356,C(C(C)(C)C(=O)N1CCCC1)N(C(C=C1CCC(C)C1)=O)C 77357,N1(C(C(C2CCN(C(CC3C(C)OCC3)=O)CC2)C)=O)CC2CCC2(C)C1 77358,C(c1csc(C)n1)=CC(=O)N(C(CN(C(C1CCN(C(C)=O)C1)=O)C)C)C 77359,Cc1[nH]c(=N)sc1C(N1CCCC(CN(C(=O)CC2C=NN(C)C2=O)C)C1)=O 77360,N1(C(C2(C)N(C(C3C(OC)CCC3)=O)CC=C2)=O)CCC(C)(COC)CC1 77361,N1(C(Cc2c(C)cnn2C)=O)CC2CC3CC2C1C3NC(c1cnc(S)n1C)=O 77362,Cc1ncc(C(=O)NCc2nc(C3CC3)no2)o1.C12(CCC1)C(=O)N2 77363,N1(C(C2(C(=O)NCC(C)CC(C)C)CCC2)=O)CC(C=O)CCC1(C)C.CN 77364,c1(CN(C(=O)C(C)(C2CCC2)NC(c2cn(C)nn2)=O)C)cccc(O)c1 77365,c1(CC)nnc2n1CCCC2C(=O)N1CCN(C(c2cccn2C)=O)C(CO)C1 77366,C1(n2cc(-c3cccc(C)c3)nn2)CON(C(=O)C23CC2C3C(F)(F)F)C1 77367,c1(C(C)C)ncc(C(=O)NC2(C)CC(NC(=O)C3CC3)C2)s1.C1(C)C(=O)N1 77368,C(=O)(N1CCC(C(N2C3CCC2CC3)=O)O1)c1cc(CC)ncn1 77369,C1(C(=O)NC2(CC#C)CC2)CC12CCN(C(C1(n3ccnc3)CCCC1)=O)C2 77370,c1(C(C(=O)NC2CCN(C(c3c(NCC)scn3)=O)C2C)O)ccc(Cl)cc1F 77371,CC(CCC(F)(F)F)NC(C1C2CCC1(c1ccco1)C2)=O 77372,C1(NC(CCCSC)=O)(CO)CCN(C(=O)CC2CC(F)C2)CC1 77373,Cc1nc(O)c(CNC(=NCCN2CC3CC3C2)NCC(F)F)cc1Br 77374,N1(C(C=C(CC)C)=O)CCC2(CCC(NC(c3cc(O)ncn3)=O)CC2)CC1 77375,C1(CC(C(=O)NC(C)CC)N(C)CC2(OC)CCCC2)COC(C)(C)O1 77376,c1(C(=O)OC)ccc(Br)c(C(=O)NC2(C)CN(C(=O)C(C)C(C)O)C2)c1 77377,C1(C(N2CC(C)N(C(c3sccc3F)=O)CC2)=O)CC(C)(C)SC(C)(C)C1 77378,c1(C(N2CCC(NC(C3(C)CC3(Cl)Cl)=O)C(F)C2)=O)cnc2[nH]cncc1-2 77379,N1(CC)CC(CSc2cc(-c3ccn(C)n3)on2)CC12CCC2 77380,Cc1cc2ncc(C(N3CCC(NC(C4CSCC(=O)N4)=O)C(F)C3)=O)cn2n1 77381,c1(C(=O)NCc2cc(F)ccc2F)ccc2occc2n1.C12CN(CC1O)C2=O 77382,c1(C(=O)OCCCC(C)(C)O)cc2nc(Cl)ccc2s1 77383,N1(C(C2(C)CCCN2C(C23CCCC2C3(F)F)=O)=O)CCC2(CC1)CSC2 77384,C(=O)(C(O)CCCNC(=O)CCc1cccnc1)NC(CCC)c1nn[nH]n1 77385,C=C=CC(C)C(=O)N1CC(C)C1C(=O)Nc1cnc(N(C)C)nc1 77386,C1(C(=O)NC(C(C)C)CCN(C(=O)Cc2cnnn2C)C)OCCN(C)C1=O 77387,C1(CNC(c2csc(C)c2C)=O)CN(C(C2CCOC(C)C2)=O)CC(C)(C)C1 77388,C1(NC(CCC=C)=O)CC(O)CN(C(C2(c3ccc(OC)c(C)c3)CC2)=O)C1 77389,c1(C(=O)NCCCNC(CNS(CCOCC#C)(=O)=O)=O)ccc(C)cc1SC 77390,c1(C(=O)NC(C2N(C(c3cnc(C(=O)OC)s3)=O)CCC2)C)c(Cl)c(C)nn1C 77391,c1(C(=O)NC(CCCNC(COC(CC)(C)C)=O)C)nccc(Br)c1O 77392,c1(OC)cc(C(N2CCCC(C)C2CCNC(=O)CC(F)F)=O)c(N)c(C)c1 77393,c1(C(N2C(C(CNC(CCC#C)=O)(C)C)CCC2)=O)cccnc1O 77394,N1(C(C2(COCC)CC2)=O)CCC(C)(CNC(C2CCC(C)O2)=O)CC1 77395,N1(C(Cn2ncc(CC)c2)=O)CC=C(CNC(C2CCN(C(C)=O)CC2)=O)CC1 77396,C1(C(=O)NCC2N(C(C3CC(C)(CC)C3)=O)CC(O)C2)C2CC3CC(C2)CC1C3 77397,C(=O)(C(F)(F)CC(=O)NCC1CC(NC(C2CC(C)(C)O2)=O)C1)OC 77398,C1(C(=O)OCC)(NC(C2CCC2)=O)CN(N2CCC(c3ccn(C)n3)C2)C1 77399,Cc1[nH]nc(C(=O)NC2CCC(F)(CNC(c3cccn3C)=O)C2)c1Br 77400,c1(CNC(C2(C)C(C)C2)=O)cccc2c1CN(C(c1cc(Br)sn1)=O)C2 77401,c1(NC(CC2CC(CC)C2)=O)ccc(Cl)cc1N=[N+]=[N-] 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77540,c1(NCC(F)(F)Br)cc(=NC2CCCc3sccc32)[nH]c(COC)n1 77541,C1(CNC(C(C)OCC)=O)(Cn2cc(C3(O)CCOC3)nn2)CC12CCC2 77542,C1(NC(C)=O)CC(C)CN(C(=O)CC(C)F)C1 77543,c1(OC)c(C(N2CC3C(C2)N3C(=O)Cc2ccccc2I)=O)cccc1F 77544,S(=O)(=O)(c1ccc(=NCC(C)COCC(c2ccccc2)O)[nH]c1)NC 77545,C(=O)(C1=CCCC(C)(C)C1)NC(c1ccc(F)cc1)CNC(C1CC(C)C1)=O 77546,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1COC1)=O)C2 77547,N1(C(C2(CC)CC2)=O)CCC(O)C(C(N2CC3CCCC2C3)=O)C1 77548,CC1CCC(NC(=O)CCC(=O)c2ccc[nH]2)CN1C(c1cc(F)ccc1O)=O 77549,c1(OC)ccc(CC(=O)NC(C)C(C)NC(c2csnn2)=O)c(Cl)c1 77550,N1(C(CSCC)=O)CCc2sccc2C1CNC(=O)C(C)(O)COC 77551,C(C1=CCCOC1)N(C)C(C1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)=O 77552,N1(C(C2N(CC)CCC2)=O)CCC2CCCC12C(=O)NCCNS(N)(=O)=O 77553,C(CCN(C(=O)Cn1nnc(C2CC2)n1)C)(C(C)C)NC(c1n(CC)nnc1)=O 77554,C(C)(C)(CC(F)C(=O)NCc1nc[nH]n1)N(C(=O)COC(C)(C)C)C 77555,N1(C(C2(SC)CC2)=O)CC2CCC1CN2C(C1(CO)CC1)=O 77556,c1(C(c2ccccc2)OC)nnc2c(N3CCC(O)(C(F)(F)F)C3)nccn12 77557,c1(OC(C(C)NC(=O)C(=O)NCCN2CCCC(C)C2)C)cc(Cl)cc(Cl)c1 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77646,C1(C(=O)NC(c2cc(SC)on2)C)C(C)CC2(CC2)C1.C1(C)C(=O)N1 77647,N1(C(CCCCC)=O)CCN(C(c2ccn(CCC)n2)=O)C(C)C1C 77648,C#Cc1ccc(CC(N2CCC(O)C(C(=O)NC(CO)CCCC)C2)=O)cc1 77649,CCN=C(NCc1noc(C2CCC2)n1)NC1CC1C(F)F 77650,C1(C(C)NC(=O)C=Cc2cocn2)CCN(C(C2(C)CCOC2)=O)CC1 77651,C(=O)(C1=CC(O)CCC1)NCC1(C)CCN(C(c2cncc(Br)c2)=O)CC1 77652,C(=O)(C(F)C(C)C(F)(F)F)NC1(C)CN(C(CCOc2cccc(C)c2C)=O)C1 77653,C1(N(C(CN2C(C)CC2)=O)CCF)CCCN(C(=O)COCC(C)(C)C)C1 77654,C(=O)(C(C)C(C)O)NCCC(C)(C)NC(C(c1cnn(C)c1)C)=O 77655,C1(C(=O)NC(c2cn(Cc3ccccn3)nn2)(C)C)CCC2CC12 77656,CN1CC(CC(=O)NOc2ccc(C(F)(F)F)c(Cl)c2)CCC1C(F)(F)F 77657,N1(C(c2cnn(CC)n2)=O)CCN(C(=O)CCN2CCC(F)C2)CC1.C1(=O)CN1 77658,C(=O)(C1=C(C)OCC1)NCC(C)=CC(=O)NCC1(C)CC(C(=O)OC(C)(C)C)C1 77659,C=CCCCC1C(=O)NC(CCC)CCC(=O)N1.C(=O)(C(F)(F)C=C)NC 77660,C(=O)(CC1CCCO1)NC1(CCNC(CCC(=O)NCC)=O)CC1.C1CCCCO1 77661,C12(NC(C=CC)=O)CCC(F)(F)CC1CN(C(=O)CC1CNC(=O)C1)C2 77662,C1(O)(NC(C2COCCN(C(=O)CC3COCCO3)C2)=O)CCCN(CCF)C1 77663,N1(C(C(C)(C)CCl)=O)CCCC(C(=O)NC2CCCNC2=O)CC1 77664,c1(C(N2CCC(O)(C(CNC(C(CC)CC)=O)C)C2)=O)cc(F)c(CC)cc1F 77665,C1(NC(c2coc(Cl)c2)=O)C2CC3CN(C(c4ccc5n[nH]cc5c4)=O)C1C3C2 77666,CCC(CC(=O)NC(c1ccc(CNC(c2n[nH]cc2F)=O)cc1)C)C(C)C 77667,c1(NC(=O)CCCSc2ccc3c(c2)OCO3)nc(C(F)(F)F)[nH]c2ncnc1-2 77668,c1(N2CCC(c3c(OC)ccnc3)C2)ncccc1S(=O)(=O)NC1C=CCC1 77669,C#Cc1cn(C)nc1C(=O)NC(C1CN(C(C2CS(=O)(=O)C2)=O)C1)C 77670,CC1CC(CC(=O)NCC(c2cc(C(F)F)no2)=O)C(C)O1 77671,C12(CC(=O)NCCC(CC)C)CCC1CN(C(c1cc(CO)on1)=O)C2 77672,N1(C(C2Cc3ccccc3C2)=O)CC2(CCCCN2C(C2CCCSS2)=O)C1 77673,c1(NC(c2n(CC)nnn2)C2CC(NC)C2)cccc(-n2ncnn2)c1 77674,N1(C(c2c(C)nco2)=O)CCC2CCCC12C(N1CCCC(CF)C1)=O 77675,CCC(C)CCCCC(=O)N(C(C)C(=O)NCCN1CC2CC2C1)C1CC1 77676,c1(C(=O)NC2(C)CN(C(C3N(CC(C)C)CCC3)=O)C2)cc2ncccn2n1 77677,C(=O)(C(C(C)C1CC1)N1CCN(c2ncc(F)cn2)CC1)NCCOC 77678,N1(C(c2c(C)cccc2)=O)C2CCC1C(CNC(C1CN(C)CCO1)=O)C2 77679,N1(C(c2c(C)scn2)=O)CC(NC(c2ccnc(N3CCCC3)c2)=O)CCC1C 77680,C(=O)(CC(CC1CC1)NC(c1c[nH]c(=O)cn1)=O)N1C(CC(N)=O)CCC1 77681,C1(NC(CN(CCCCCC)C)=O)(CNC(c2ccsc2Cl)=O)CCCCCC1 77682,C=CCC(CC=C)C(=O)NCc1cc(C(=O)NC2CCCCCC2C)co1 77683,C(=O)(C(C)(C)C1CCCCO1)N1CC(C(C)NC(=O)Cn2nnc(C3CC3)n2)C1 77684,C(C)(C)(CC(F)(F)F)NC(C(C)CNC(=O)C=Cc1cccnc1)=O 77685,c1(C(=O)NCC2CC(NC(CC3C(OCC)C3)=O)C2)[nH]c(C)c(C(=O)OC)c1C 77686,c1(C(=O)NCC2(NC(c3c(N)cccn3)=O)CCCCC2)cnc2ccnn2c1 77687,c1(CCC(=O)NCC2C(NC(C=CS(C)=O)=O)CCCC2)cccc([N+](=O)[O-])c1 77688,C1(N(c2n(CC)c(CC(c3ccc(Cl)s3)(F)F)nn2)C)COc2ccccc21 77689,c1(C(=O)NCCC(C(C)C)N(C(C(=O)NCC)=O)C)ccc(C2CC2)c(F)c1 77690,c1(C(N2C(C)(CNC(C3(SC)CC3)=O)CCC2)=O)cccc2c1nc(O)n2C 77691,C(CNC(=O)CCC1(C)N=N1)(CC(=O)N(C1CC1)Cc1ncc[nH]1)OC 77692,C1(CCNC(=O)CCc2ccccc2)CCCCN1C(C1CC=CCO1)=O 77693,c1(C(N2CC(NC(=O)C3CC3)C(c3ccccc3)CC2)=O)c(F)c(F)nc(F)c1F 77694,c1(C(=O)NC(C(C)NC(=O)CCCC2CC2)CO)cc(S(C)(=O)=O)ccc1N 77695,c1(C(=O)NC(c2cn(CCCC)nn2)C)c(C)nn2ccccc12 77696,CCCCCS(=O)(=O)CC(=O)OCc1cc(Br)cnc1I 77697,Cc1cc(CC(N2CCC(CCC(=O)NCCn3ccnn3)C2)=O)no1 77698,N1(C(c2cn(CCC)nn2)=O)CCC(CO)(CNC(C2C(F)(F)C23CC3)=O)C1 77699,c1(C(=O)NCCCN(C(C(C)O)=O)C2CC2)c[nH]nc1-c1cccs1 77700,c1(-c2c(C(C)Nc3cncc(C(F)(F)F)c3)c[nH]n2)ccc(C#N)cc1 77701,c1(CNC(c2cnc(Cl)cc2Cl)c2n(CC(=C)C)nnn2)ccc(F)c(C)c1C 77702,C(=O)(CCCCCC(C)(C)C)NC(C(C)NC(=O)CCCC1CCOCC1)C 77703,c1(-c2ccc(C(=O)NCCCCN(C(C)=O)C)nn2)cn(C)c2cc(Cl)ccc12 77704,c1(C(=O)NC(CNC(C(=O)NC(C)(C)C)=O)CO)cccc(OC(F)F)c1 77705,C1(NC(CN2CC(C)(C)C2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 77706,C(=O)(N=c1cc(C)n(C2CC2)[nH]1)C1OCCC(NC(c2cc(C)nc(Cl)c2)=O)C1 77707,C12(CNC(C(C)(C3CC3)OC)=O)CCC(NC(=O)CCC(C)C)(CO1)C2 77708,c1(C(N2CC(C)(NC(C=CSC)=O)C2)=O)ccnc(S(N)(=O)=O)c1 77709,c1(OC)ccn2cc(C(=O)NCC3(C)CCN(C(C4CC4F)=O)C3)nc2c1 77710,c1(C(=O)NCC(C)(CO)NC(c2ncn(CC)c2)=O)cc(C)c(F)cc1O 77711,C1(OC)(CNC(c2nc(Cl)cs2)=O)CCN(C(C2CCC(C)C2)=O)CC1 77712,N1(C(C(C)(C)CCCF)=O)CCC(C(=O)NCC(C)(O)C(F)F)=C(F)C1 77713,N1(C(C=C(CC)CC)=O)CCC2C(C1)CN2C(c1cc(C)cc(OC)c1N)=O 77714,C1(C(=O)NC2(CNC(C34CC(F)C3C4)=O)CCCC2)CC2(CCCCC2)C1 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77927,c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)cc(F)ccc1F 77928,c12cncc(c1)C(=O)N2.c1(CC(=O)N(CCN)CC2C(C)C2)ccccc1F 77929,C(=O)(C1=CNC2=NCCCC2=C1)NCCOCCCNC(CCSCC)=O 77930,CC1CCC(SCCc2ccccc2)CN1 77931,N1(C(c2coc(O)n2)=O)CC2CC(C1)N(C(c1cc(Cl)nc(Cl)c1)=O)C2 77932,C1(N(C(C(c2ccc(C)cc2)F)=O)C)CCN(C(C(=O)OC(C)(C)C)=O)CC1C 77933,C1(CNC(C(COC)(C)O)=O)CC2CCC1N(C(c1cnn3c1OCC3)=O)C2 77934,c1(C(c2ccccc2C(C)C)OC(C(C)OCCOC)=O)cccc(C#N)c1 77935,C(=O)(C(F)(F)C(C)(C)O)NCC(=C)CCNC(=O)Cc1ccccc1 77936,N1(C(c2c(OC)csc2)=O)CCC2(NC(=O)CCCCC(C)C)CCCCCC12 77937,C1(NC(CCN(CC#C)C(c2cc(C(C)=O)[nH]n2)=O)=O)C=CCCCC1 77938,Cn1cc(C(C2CC(CF)C2)NC(=O)CCCn2cc(CCCCO)nn2)cn1 77939,C1(COCC)CCN(C(=O)CC(OCC)NCC(N)=O)C1.C1CO1 77940,c1(C(=O)NC2C(NC(c3sccc3C3CC3)=O)CC2)cn2c(n1)CCC2 77941,C#Cc1ccc(C(=O)NCC(C)(C)C(=O)NC2CCN(CCOC)C2)cc1 77942,c1(C(=O)NCC2(C)CCN(C(c3c(C(C)C)cco3)=O)C2)ccc(N)c(Cl)c1O 77943,C(=O)(C(F)(CNC(=O)C(C)NC=O)C(C)C)NC1C(C)(CC)C(O)C1 77944,N1(C(CCC2CC(NC(=O)C=CC3CCOC3)C2)=O)CC2CCC(C1)O2 77945,C1(C(N(CC(=O)NCC(C2CC(C)(C)C2)O)C2CC2)=O)CCNC(=O)C1 77946,c1(CC(N2CC(NC(CCSC)=O)C3C2C3)=O)csc2cccc(F)c12 77947,CC(C)CCCC(C)CNC(=O)C(F)CC1CN(C(C2CC2(F)Cl)=O)C1 77948,c1(OC)cccc(CNC(=O)OC(C)(C)C)c1C.C12CCCN(C1)C(=O)C(=O)N2 77949,C(=O)(C#CC1CCCOC1)NC1(CNC(C(COC)CC(C)C)=O)CC1 77950,c1(NC(c2c(C)n(C3CC3)nc2)=O)ccc(C(C)C)cc1O.N12CCSCC1C2=O 77951,C(=O)(CC(C)CC(=O)N(C(CC(F)F)C(=O)NCC1=C(C)CCC1)C)OC 77952,N1(C(c2ccc(CC)o2)=O)CCC2C1CCCN2C(=O)CCOCCCCOC 77953,C12(CNC(=O)C(N3CCC(c4cccc(Br)c4)CC3)=O)CCNC1CNC2 77954,CC1CC(=O)NCCN1C(c1c[nH]nc1-c1ccc(Cl)s1)=O 77955,N1(C(=O)NC2C(C)NC(=O)CC2)CC2CCCC(C1)N2C(=O)OC(C)(C)C 77956,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)(C)CO)cc(C(F)(F)F)ccc1F 77957,C1(N(C)C(c2cnnn2C)=O)CC2CCC(C1)N2C(C1CC1F)=O 77958,C1(C(=O)NCCNC(CCCCC#N)=O)CC12CCC1(CC1)CC2 77959,S(=O)(=O)(CCC(=O)NCCn1cc(-c2ccc(C(=O)O)nc2)nn1)N(C)C 77960,C1(CC(=O)N(c2ccc(-c3cccnc3)s2)CCC)CC(CC)=NN1C 77961,CCC(C)CC(C(=O)NCC=CCOC)NC(=O)Cc1cn2ccccc2n1 77962,C1(NC(c2cc(OC)ncn2)=O)CCCN(C(=O)OC(C)(C)C)C1C 77963,c1(NC(C2(F)CCCN(C(CS(N)(=O)=O)=O)C2)=O)ccc2nncn2c1 77964,C(=O)(CC(C)CC(=O)NCC(=O)NCC(C)(C)NC1CCCC(C)(C)C1)OC 77965,N1(C(C(CC)NC(=O)CC2CCOCC2)=O)CCC(OOC(F)F)CC1 77966,C(=O)(C(CC(C)C)n1cc(-c2cc(C)ccc2O)nn1)OC.[nH]1ccnc1 77967,N1(C(CCc2ncc(C)[nH]2)=O)CCC2CN(C(=O)C#CC3(C)CCCO3)CC2C1 77968,N1(C(C=CC=CC)=O)CCOC2CN(C(c3cc(C)c(Cl)s3)=O)CC12 77969,c1(C(=O)OC)cc(OCC(=O)OCC(C2CCCC2O)C2CC2)c2c(c1)CCC2 77970,CC1CCC(NC(c2coc(O)n2)=O)CN1C(c1cc(Br)n(C)c1)=O 77971,c1(CC(CN(C(=O)NC(CC)C(F)F)C)=O)ccc(F)c(F)c1 77972,N1(C(c2nc(CC)oc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 77973,N1(C(C2(COC)CC2)=O)CC(OC)C(NC(c2cc(OC)ns2)=O)C1 77974,c1(C(CC)C)nc(NC2(CO)CCCN(C(c3sccc3OC)=O)C2)cc(C)n1 77975,c1(OC)cc(C(N2CCCC(SC)CC2)C(=O)NC2CCC2)ccc1S(C)(=O)=O 77976,C1(N(C(=O)CC2(CO)CCCCC2)CC#C)CCCN(C(=O)CC(O)CC)C1 77977,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CCN(C)C)CCC2)=O)C1 77978,C1(N(C)C)(CNC(C2COCC2CNC(C2CC(F)C2)=O)=O)CCOC1 77979,CC1CCN(C(c2ccns2)=O)CC1CNc1occ(C(=O)OCC(F)(F)F)n1 77980,CC(C)CCCC(C)C(=O)N(C1(N(C(C2CC2Cl)=O)C(C)C)CCC1)CCO 77981,c1(NC(C(C)C)CNC(C2CCCCC2CO)=O)cc(C(F)F)ncn1 77982,c1(C(N2C(CNC(c3csc(C(C)=O)c3)=O)CC(OC)C2)=O)cc2cnccc2o1 77983,c1(CC)cc(C(=O)NCc2nc(C3CCCN(CCOC)C3)no2)ccn1 77984,C(=O)(C1=CCCC1C)N(C(C)C)CCNC(c1ccc(C2CC2)o1)=O 77985,Cc1cc(C)c(CN(c2cccc(F)c2)C(C2CCC2)=O)s1 77986,CC1CN(C(=O)CCOC2COC2)CC(C)N(C(=O)C(c2ccc(Cl)s2)O)C1 77987,c1(CC)cc(C(=O)NCC2C3CN(c4ncc(C(C)(C)O)cn4)CC23)ccn1 77988,n1(CC(=O)NC)cc(C)c(NC(=O)CCCC2(N)CCC2)n1 77989,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)C(C)(C)c2cnsc2)CC1C)=O 77990,N1(CC(=O)Nc2c(C)nsc2)CCCN(Cc2ccc(C(=O)O)cc2)CC1 77991,Cc1nn(CC(F)F)cc1C(=O)NCCC1CCCN1C(C1CSCCS1)=O 77992,c1(C(=O)NCC2(O)CCC(C)CC2)cc2c(ccn2C)s1 77993,C(CC(=O)N1CC2CC1CN2C(N)=O)(C(F)(F)F)NC(CCCc1[nH]c(=N)sc1)=O 77994,CCC(O)C(C)C(=O)NC1CCCN(C(C2CN(C(C)C)C2)=O)CC1 77995,C1(CN(CCCNC(C(C)SC)=O)C(=O)Cc2ccnn2C)CCC(F)(F)C1 77996,N1(c2nnc(CCC)s2)CCc2cc(O)ccc2C1 77997,N1(C(C(CC)N(C)C)=O)CC2(CCOCC2)CC1CNC(C1(C(=O)NC)CC1)=O 77998,CN1CCC(NC(c2c[nH]nc2CCNC(=O)C(O)P(C)(C)=O)=O)C(C#N)C1 77999,C(=O)(C1CCCS1(=O)=O)N(C1CCCC1)CCNC(C(c1cnn(C)c1)OCC)=O 78000,C1(F)(CNC(c2n(CC(C)C)ncc2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1 78001,N1(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC(S(=O)(=O)NCC(=O)O)C1 78002,c1(C(=O)OC(C2CC2Cc2c(OC(C)C)cccc2)=O)c(Cl)cccc1[N+](=O)[O-] 78003,N(C(=NCC(C)(C)OCC(F)(F)F)NC1CCCS(=O)(=O)C1)C(C)C 78004,N1(C(=O)OC(C)(C)C)CCC(O)C(O)C1OC(c1cc(-c2ccco2)on1)=O 78005,CN1N=C(C(=O)NCCC2CC(NC(C3CCCCS3(=O)=O)=O)C2)CCC1=O 78006,N#Cc1ccc(C(=O)NCCN2CCN(C(c3cnsn3)=O)CC2)cc1C(F)(F)F 78007,C(=O)(C1=CC(C)C1)N(CC(CC)NC(=O)C(C1CC1)SC)C 78008,N1(CCN2c3cccc(c3)C3N(CCCC3)CC2=O)CCOCC1C.C(=O)O.CO 78009,c1(CC2(C(=O)NCC3(NC(C4(C)CCC4)=O)CCC3)CC2)cccc(F)c1 78010,c1(C(=O)OCC)ccc(OC)cc1NC(C1COCCN1)=O 78011,c1(-c2cn(CC3CCN(C(C4(Cl)CCC4)=O)C3)nn2)cccc(F)c1 78012,C123CC1CN(C2)C3.N1(CC(=O)NCc2ncoc2CCSC)CC(=O)NC1=O 78013,c1(C(C)=O)ncc(C(=O)NC(c2cnc[nH]2)C)s1 78014,N1(C(=O)OC(C)(C)C)CCC(NCC2(CO)CC3(CCC3)C2)C(O)C1 78015,CC1OCCN(C(C2CC3(CCC3)C2)=O)C1C(=O)NC1CC(O)C1O 78016,c1(NC(Nc2cc(C(=O)OCC)n3c2COCC3)=S)ccc2occ(C)c2c1 78017,N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(c3cn[nH]c3)=O)CC(C2)C1 78018,C(=O)(C(C1(C)CC1)NC(=O)C(F)OC(F)(F)F)NCC(C1CCC1)OCC 78019,N1(C(c2ccc(C#N)s2)C(=O)Nc2c(C)cc(F)cc2)C2CCC1CC(CO)C2 78020,CCCCC(CNC(=O)C(C)Cc1cnco1)NC(c1cc(C)nn1C(F)F)=O 78021,Cc1ncncc1C(=O)NCC1CN(C(=O)CCC2CCCO2)CC1C 78022,c1(OC)cc(C(=O)NC2(C3CN(C(=O)CC4CCCC4C)C3)CC2)cc(OC)c1C 78023,N1(C(C=C(CC)CC)=O)CCC2(CCCC2NC(C2CCS2(=O)=O)=O)CC1 78024,C1(CC=C)(NC(=O)COCC(C)C)CCCN(C(c2coc(C#N)c2)=O)C1 78025,c1(C(=O)NC(c2ccccc2)C(=O)N(C)Cc2ccnn2C)ccc(C#N)cn1 78026,CN1CC(C(N2CCCCC2C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)NC1=O 78027,C1(C(=O)NC(c2nocc2C(=O)N(C2CC2)CC2CCCC2)C)CC=CCC1 78028,c1(CC(N2CC3C(CNC(C(CC4CC4)OC)=O)C3C2)=O)c(C)cccc1Cl 78029,Cc1nn(C)c(C(=O)NC2CC2)c1C(C1(F)CCOCC1)N.c1(S)ccc(Cl)cc1Cl.N 78030,C1(O)(C(N2C3CC(NC(C(c4scc(C)n4)C)=O)C3CC2)=O)Cc2ccccc2C1 78031,c1(C(=O)NC(CNC(C2CCC(=C)CC2)=O)CO)cc(C(F)(F)F)ccc1F 78032,c1(OC)cc(C)cc(C(N2CC(NC(=O)Cc3ccnn3C)C3CC23)=O)c1O 78033,c1(SC)ncc(C)c(N2CC3(CC3C(N3CCCC3CN(C)C)=O)C2)n1 78034,c1(C(=O)NC2(N)CCOC2)cc(Cl)c2cccc(Br)c2n1 78035,C1(C)(NC(C(C2CCCCC2)C)=O)CCCN(C(=O)CN(c2ccccc2)C)C1 78036,C1(CNC(c2ccn(CC)n2)=O)CC2(CCC2)CN1C(=O)Cc1ccsc1 78037,C(c1csc(C(F)(F)F)c1)=CC(N1CCC(CCNC(CCC#C)=O)C1)=O 78038,C1(CNC(c2c(C)snn2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C(O)C1 78039,N1(Cc2cn(CCC3(C)CC3(F)F)nn2)C(=O)COCC1=O 78040,C1(C(=O)NC2CCN(CCNC(c3c(C)n[nH]c3)=O)CC2)CC(C)CC(C)C1 78041,C1Cc2ccccc2O1.c12ccc(cc1)C(=O)NC1(c3cn-2nn3)CC1.COC 78042,N1(C(c2cnc(-c3cccc(C#N)c3)s2)=O)CCC2(CC(=O)NC2=O)C1 78043,CC1(C)CCN(C(=O)COCc2nccs2)CC1C(=O)NCCCc1ncco1 78044,C(N=c1[nH]c(C)c([N+](=O)[O-])cc1Cl)C1CC(NC(c2c(SC)cccc2)=O)C1 78045,N1(C(C(C)NC(c2ccc(F)cc2)=O)=O)CCCC(CNC(C2CCCC2)=O)C1 78046,C1(CN(CCN=C(NS(C)(=O)=O)NCC2CC2)C)CCC2C(CC1)C2(F)F 78047,C(CC(C(C)C)NC(=O)CONC(=O)Cc1ccccc1Br)OC 78048,C1(CNC(Cn2ncc(C)c2)=O)CC2(CO1)CN(C(=O)C(N1CCCCC1)C)C2 78049,CC1CN(C(=O)C=CCO)CC(C)N(C(c2ccc(-c3cnc[nH]3)cc2)=O)C1 78050,C(CC(C)C(=O)NC1(CCNC(=O)CCCC2CC2)CCCC1)OC 78051,N1(C(CC=C=C)=O)CC(C(=O)NOC(c2ccncc2)C)CC12CCC2 78052,CC(N=[N+]=[N-])C(=O)NC1(CCCNC(C2CCS2(=O)=O)=O)CC1 78053,Cc1cc(C(=O)NCC2COCC2NC(c2cnn(C)c2Cl)=O)[nH]c1C#N 78054,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CC2(CCN(C(c3cc[nH]n3)=O)C2)C1 78055,C1(N(C(c2cccs2)=O)CC)CCCN(C(=O)CSc2ccccc2)C1 78056,C(=O)(C(C)(C)CCCSc1c(C)cccc1Cl)NCc1c[nH]c(=N)o1 78057,c1(C(=O)NC2C(NC(=O)C=Cc3ccco3)CCC2)ccnnc1Cl 78058,N1(C(C2N(C(C(CC3CC3)OC)=O)C3(CC2)CC3)=O)C2CCC1CN(C)CC2 78059,C(CCCCC(=O)NC(C1(O)CN(C(C2CC2C#N)=O)C1)C)OCC 78060,c1(C(=O)NC2CCCC(NC(C3(OC)CCSCC3)=O)C2)ccc(C)cc1F 78061,c1(C2(C)CCO2)ccc(NC(C2CCC(Nc3ncc(I)cn3)CC2)=O)cc1 78062,c1(NC(C(c2ccccc2)C)=O)cccc(NCC(F)(F)F)c1 78063,c1(C(=O)NCC2(F)CC(NC(CCCCOC)=O)C2)cc2n[nH]cc2cc1C 78064,C(=O)(C(O)CCCC)N1C(C(=O)NC2(CC=C)CCCCC2)C2CC2C1 78065,c1(C(=O)NCC2CC(OC)CN2C(c2cc(C)no2)=O)ccc(C#N)cc1O 78066,N1(C(=O)Nc2ccc(SCC(=O)NC)cc2)CCCCCC2(CCCCC2)C1 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78084,C1(C(N2CC(NC(C3OC4CCC3CC4)=O)(CO)C2)=O)CC2CCC1CC2 78085,CC1(CO)CCCC1NC(C1CCOCC1NC(C1CC2C=CC1C2)=O)=O 78086,N1(C(=O)Cc2ccc(Cl)cn2)CC2CCCN(C(C3COC4COCC34)=O)C2C1 78087,c1(CC)nc(N2CCC(N(C(=O)C(O)CC(C)C)CC)C2)c2ccsc2n1 78088,C1(F)(C(N(C(CC(CC)C)C)C)=O)CCCN(C(c2cnsc2C)=O)C1 78089,C(=O)(CCCCC(C)(C)C)N1C(C(C)NC(c2cc(OC)no2)=O)CCCC1 78090,C(=O)(C1CCc2snnc21)N1CCC(N(C(C2CCC(=C)CC2)=O)C)C(C)C1 78091,c1(C(=O)NCC(C)N(C)C(C2OCCO2)=O)ccnc2ncsc12 78092,c1(CC)nnc2n1CCCC2CCC(=O)Nc1ccc(OC)cc1F 78093,C1(CC(=O)NCC(C)(C2CC2)NC(C=CSC)=O)CCCCN1C(=O)OC(C)(C)C 78094,c1(C(N2C3(CNC(CCSC)=O)CCC2CC3)=O)cccc2c1OC(C)C(=O)N2 78095,Cc1ccc(C(N2CC=CC(NC(C3(F)CC3c3ccccc3)=O)C2)=O)nc1C 78096,N1(C(c2ccc(CC)cc2O)=O)CCN(C(=O)CC2CCCC2)C(C)C1C 78097,C1(CC(C)(O)SCC(=O)OC)CCCN(C(=O)C(F)(F)c2csc(C(F)(F)F)n2)C1 78098,N1(C(C=CC)=O)CCCC2(C1)C(NC(c1cn(C)nc1SCC)=O)CCN2C 78099,N#Cc1ccc(OCC(=O)NCC2CC2C(F)(F)F)cc1 78100,N1(C(C(C(C)C)NC(=O)OCC)=O)CCN(C(=O)C(C)CF)CCC1C 78101,Cc1cc(C(=O)NC2CCCN(C(=O)CSC3CC3)CC2)ccc1[N+](=O)[O-] 78102,c1(C(=O)NC2CCC(CNC(c3c(CC)non3)=O)C2)ccc2ccc(F)cc2n1 78103,C1(C(=O)NCC2CC(CNC(COC3(C)CCC3)=O)OC2)CN2CCN1C(C)C2 78104,C1(C(=O)NCCNC(C(CC)C)=O)(NC(C)CN(C)C)CCC(C)(C)C1 78105,c1(CC)ccc(C)c(C(N2CCC(C)C2CNC(=O)CCCc2cncs2)=O)c1 78106,C1(C)(CNC(C(C2CN(C(=O)CC3(C)CCOC3)C2)OC)=O)CCCC1 78107,c1(C(=O)NCCCC(C)NC(C2CC3(CC(=C)C3)C2)=O)ccc2sc(=N)[nH]c2c1 78108,C1(C(=O)OC)CCC(C(=O)NCCC2COCCN2C(c2cn(C)cn2)=O)CC1 78109,C(CCCC(C)NC(=O)CC1CC2CC2C1)NC(Cn1c(C(C)C)nnn1)=O 78110,c1(C(N(C2CCCC(NC(c3occc3F)=O)C2)C)=O)ccc(F)cn1 78111,Cc1nc(CNC(=O)C(O)CNC(C2CC(C3CC3)C2)=O)sc1C 78112,C1(CNC(C(C)NC(N)=O)=O)C(C(N2CCC(C(F)F)C2)=O)C1(C)C 78113,Cc1cc2ncc(C(=O)NC3CC3CNC(c3ccc(Br)c(F)c3)=O)cn2n1 78114,CC(CC(=O)N1CC(NC(c2cc(F)cc(Br)c2)=O)C(O)C1)C(F)F 78115,N1(c2snc(CCC)n2)CC(CNC(=O)C(N2CCSCC2)C)OC(C)(C)C1 78116,N1(C(c2nc(OC)c(C)s2)=O)C2CCC1CN(C(=O)CN(C)C(C)C)CC2 78117,C1(NC(C(C)Oc2ccccc2)=O)CC2CCC1N2C(C1CNC(=O)C1)=O 78118,CCC(C)(COC)C(=O)N1CCC(CNC(c2cnn(C3CCC3)c2)=O)C1 78119,CCC(CC(C)C)C(=O)N1CC(O)(CNC(c2nc(Cl)sc2Cl)=O)C1 78120,c1(C(N2CCCC(C3CC(C(=O)O)N3)C2)=O)cccc(-c2ccc[nH]2)c1 78121,c1(CC)cc(C(N2CCC(N(C(=O)CN(CC)CC)C)C2)=O)oc1CC 78122,C(=O)(CCC1=CCCCC1)NCCCCCNC(c1nc(N)c(Br)cc1)=O 78123,CC1=NOC(CCNC(=O)C(C2(C)CC2)NC(=O)CC2(C)CC2)C1 78124,c1(C(N(CCN(C(=O)Cc2cccnc2Cl)C)C)=O)ccc([N+](=O)[O-])cc1O 78125,C1(C)(NC(c2cnc(C)[nH]c2=N)=O)Cc2ccccc2C1.c12nc(cs1)C(=O)NC2 78126,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78127,C12(NC(=O)OC(C)(C)C)CCCC1CCN2C(c1ccc(F)c(N)c1)=O 78128,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78129,C1(NC(CCCOC(C)(C)C)=O)CC(C(N2CCC23CC(O)C3)=O)C12CCC2 78130,C(C(CN=c1[nH]cnc(Cl)c1OC)CC(C)C)NC(c1ccc(OCC)cc1)=O 78131,C(C(O)C(=O)NCC1(O)CC(NC(=O)C(c2ccccc2)(F)F)C1)SC 78132,C(CCC(=O)NC1CC1)(C(C)C)NC(C=CC(=O)N(C)C)=O.C1(C)C(=O)N1 78133,N1(C(=O)CCc2cscn2)CCOC2(CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 78134,c1(NCCN(C(=O)CCCN2CCCCC2)C(C)=O)ncc([N+](=O)[O-])cc1C 78135,C1(C(CC)O)CN(CC(=O)NCCP(C)(C)=O)CCO1 78136,CC1C(NC2(c3nnnn3C3CCOC3)CCC(Br)C2)C(CO)C1(C)C 78137,c1(CC(=O)NC2CC(C(=O)NCCn3c(C)nnc3)OCC2)c(F)cccc1F 78138,C1(O)(CNC(C(CC)C(C)C)=O)CCCN(C(=O)C=C(C)C(C)(C)C)CC1 78139,c1(C(C(N2C(Cn3cc(CCS(C)(=O)=O)nn3)C=CC2)=O)=O)ccc(F)c(F)c1 78140,c1(C(=O)NCC(C)NC(c2cc(C(C)(C)C)no2)=O)cn(CCC2CC2)nn1 78141,Cc1cc(C(N2CC(CNC(C3COC(=O)C3)=O)CC(C)C2)=O)ncc1F 78142,N1(C(c2c(C)noc2C)=O)CC2CC1CN2C(=O)CSCC(F)F 78143,C(C)(C(C)NC(n1cc(C(c2ccccc2)C2CC2)nn1)=O)(C1CC1)OC 78144,N1(C(c2c(C)cccc2Cl)=O)CC2(CCCC2NC(C2CCC3CC3CC2)=O)C1 78145,c1(COC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)c3ncco3)C2)=O)s1 78146,CCC(CC1CCCN1Cc1cnc(C)s1)CO 78147,CC1(C)CC(NC(c2cccc(O)n2)=O)CN1C(C1CCN(S(C)(=O)=O)C1)=O 78148,N1(C(CCN(C)C(C2CCC(N(C)C)CC2)=O)=O)CC(S(N)(=O)=O)C1 78149,c1(C(=O)NC(CC)CC(=O)NCC(F)Cl)ccnc(C)c1C 78150,c1(C(C)(F)F)ccc(C(=O)NC2CCC2NC(C2C=CCC2)=O)cn1 78151,Cc1ccc(CCCNC(c2nnnn2C2CCOC2)C2CCC2)cc1Cl 78152,c1(NC(C2OCCN(C(=O)OC(C)(C)C)C2)=O)nc2c(cc1Cl)C(=O)NC2 78153,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)C2=C(C)CC2)CC12CCC2 78154,c1(C(C)C)nc(C(=O)NC(C)C=CC(=O)NCC=CC2CC2)co1 78155,C1(CC(=O)N(C2CCN(C(=O)C(C)COCC)C2)CC#C)CCCOC1 78156,C=CCCCCC(=O)NCC1(C)CCCC1NC(c1ccc(C(C)(C)C)cc1)=O 78157,C1(CC(=O)N(C(C)(C)C)C(N(CCC)C2CC2)=O)CCCCC1.C1C(=O)NC2(CC2)C1.O 78158,N1(C(COCC)=O)CCCN(C(c2ccc(Br)nc2F)=O)C(C)C1 78159,c1(OC)ccn2c(C(=O)N(CCCNC(c3nn(C)cc3Cl)=O)C(C)C)cnc2c1 78160,CN=C(NCCc1cc(C2(C)CC2)n[nH]1)NC(C)C.C1C(=O)N1 78161,N1(C(C2(CC)CC2(F)F)=O)CC2C(CNC(=O)CC3CCCC3)C2C1 78162,C1(C(=O)NCCC2C(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)CN2CCCN1CC2 78163,C(=O)(C(COC)CC(C)C)NC1CCC(CC)CC1.C12(CCCO1)C(=O)N(C)C2 78164,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(F)F)C1 78165,C1(N(C)C(c2cccc(Cl)c2)=O)CC2CCC(C1)N2C(c1cnon1)=O 78166,C(=O)(CC(O)C(=O)NC1COCCN(C(c2ccnc(OC)n2)=O)C1)OCC 78167,S(=O)(=O)(c1cccc(C)c1C#N)N(CCC)CC1CCN(C(C)=O)C1 78168,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78169,C(=O)(CCCCCCCCCCO)N(CC(CC)NC(C1(F)CCCCC1)=O)C 78170,Cc1ccccc1C=CC(N1CCC1C(=O)NCC12CCN(CC1)C2)=O 78171,c1(CC)cccc(C(=O)NC2(C)CCC(NC(C3CC(F)(F)C3)=O)CC2)c1O 78172,c12cc(oc1C)C(=O)NC2c1n(CCCC)nnn1.C1(CC#N)COC(=O)C1 78173,N1(C(CCCCNC(CCOCCOC)=O)=O)CCCC2CNC(=O)C12 78174,n1(CC)cnc2c(NCCCOCC(F)F)[nH]c(=NCC(N)=O)nc12 78175,C1(N(C(=O)CN(S(C)(=O)=O)C)C)CCCN(Cc2nc(CC3CC3)no2)CC1 78176,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78177,O=C(CCCC1(NC(C23CC(F)(C2)C3)=O)CCC1)N1CCC(C2CCCCC2)C1 78178,C1(C(=O)NC2(CC)CN(C(=O)CNC(=O)C3CC3)C2)CCNC(=O)C1 78179,c1(NC(C2CCCC(NC(c3cc[nH]n3)=O)C2)=O)ncc([N+](=O)[O-])cc1I 78180,n1(CC(=O)N(C2CN(C(c3cnn(C(F)F)c3)=O)CC2F)C)nc(Cl)ccc1=O 78181,N1(C(C(C)c2ccsn2)=O)CCC(F)(CNC(c2cc(Cl)cc(Cl)c2)=O)CC1 78182,N1(CC)CC2=C(C1=O)C(c1ccc(F)c(F)c1)NC(=O)N2Cc1ccc(Cl)cc1 78183,c1(C(=O)NC(C)CCNC(=O)CC(C)(C)C)c(O)cnc2cc(F)ccc12 78184,C1(CC(=O)NCC(C)OCCO)(OC)CN(C(=O)CCn2ccnn2)C1 78185,N1(C(C2C(C)CC2)=O)CC2(NC(c3conc3C3CCCO3)=O)CCC1CC2 78186,C1(CNC(COCCC=C)=O)CCC2CN(C(c3nc(O)c(C)s3)=O)CCC2C1 78187,C1(C(N2C(CNC(C(C)CC3CCC3)=O)CC2)=O)CC12CCC1(CC2)OCCO1 78188,C(c1cn(C)c2ccccc12)=CC(=O)NCC1CN(C(COC(C)C)=O)CC1C 78189,C(=O)(C(C)NC(C1CCC1NC(=O)CCn1cncn1)=O)OC(C)C 78190,c1(C(=O)NCC(CN(C(c2n(C(C)C)ccc2)=O)C)O)[nH]ncc1C#N 78191,CCCCS(=O)(=O)NCC(=O)NC1CCCCC1CNC(=O)CCCC#N 78192,c1(-n2ncc(C(=O)NCCCN(C(C(C)n3ccnc3)=O)C)c2)ccccc1F 78193,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78194,C=CCCN=C(NCC1CC(=O)N1)NC1CCC(C(C)(C)C)CC1 78195,c1(C(=O)NC2(CNC(C(C)SC(C)C)=O)CCCC2)c(F)cncc1Cl 78196,N1(C(Cc2ccc(OC)nc2)=O)CCC2C(C1)NC(=O)CN2C(C1CC1F)=O 78197,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CCC(CCCO)C3)=O)c2C1 78198,Cc1cc(C)n(CCCC(=O)N2CC(O)(CCNC(C3CCC3C(F)F)=O)C2)n1 78199,Cc1ccc(CNC(=O)C(=O)NC2CN(C)CCO2)cc1CN(C)C 78200,c1(C(C(=O)NC2C(OC)CN(C(C3CN(C)C3)=O)C2)O)ccc(Cl)cc1Cl 78201,Cc1nc2ccc(S(=O)(=O)NC3CCC4CCCCC4C3)cc2o1 78202,Nc1ccc(Br)c(F)c1C(=O)OCC(c1ccccc1)C1CC1 78203,N1(C(c2cn(CC)nn2)=O)CC2CCC2(CNC(c2occc2C)=O)C1 78204,c1(CCC(=O)NCC2N(C(C(CC)C(C)C)=O)CC2)ccccc1[N+](=O)[O-] 78205,C1(CNC(C(CCC)(C)C)=O)CN(C(c2cn(C)c(=O)cn2)=O)CCC1(C)C 78206,C1(=CC(=O)NCC2COCC2NC(C2CCOC2)=O)C2CC3CC(C2)CC1C3 78207,N1(C(c2scc(C)c2C)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78208,C(CCCCCC(=O)N1CC2CCC2(CC(=O)NC(C)(C)CF)C1)SC 78209,C(=O)(CC(C)(C)C(F)F)NC1(CC(=O)NC(CCC)C(=O)N(C)C)CCC1 78210,c1(C(=O)NC(CCCC)CNC(=O)CCCC(C)C)n[nH]c2c1CCCCC2 78211,Cc1cc(C(=O)NCC(C)(C2CC2)NC(c2ccn(C)n2)=O)sc1C 78212,C(N=c1[nH]c(=NC2CC2CO)c2ccccc2[nH]1)c1cnc(C(C)C)[nH]1 78213,c1(OC)ccc(OCC(N2CC(NC3(O)CCCCCC3)CC2C)=O)cc1C 78214,C12(N=C3NN=C(S3)C1)CCCC2.c1(C(C)(C)C)ccc(C(=O)NN2CCC2)[nH]1 78215,C(=O)(N=c1cc(Cl)nc(Cl)[nH]1)c1n(C)cc(NC(c2ccc(OC)cc2Br)=O)n1 78216,N1(C(CC2(OCC)CC2)=O)CCCC1C(C)(C)C(=O)NC1CC(F)C1 78217,c1(C(N2CCC(O)(CCNC(=O)CSC3CCCOC3)C2)=O)ccc(CO)cc1 78218,C1(C(=O)NCC2CN(C(CSCCOC)=O)C2)CCc2cncn2C1 78219,N1(C(COCC(C)C)=O)CC2C3CCC(C2C1)N(C(c1ncccc1F)=O)C3 78220,c1(NC(=O)NC)cccc(C(=O)NCC(O)CN(C)C(c2nn(C)cc2Cl)=O)c1 78221,C1(C(=O)Nc2snc3cc(Br)c(Cl)cc23)CCc2nnc(O)cc2C1 78222,c1(C(C)C)ccc(SCC(=O)NCC(C)NC(=O)CS(=O)(=O)N(C)C)cc1 78223,Cc1nnc2n1CCC2(C)C(=O)N1CCC(C)(NC(C2COCCN2C)=O)C1 78224,CCCC(C)C(=O)N1CC=CC1(C(=O)NCCC1C=CCC1)COC 78225,C(=O)(C1=NOC2COCC12)NC(CCC(=O)NC1(C#C)CCC(C)CC1)C 78226,Cc1nn(C)c(C)c1CCC(N1CC(NCc2cc(C(C)(C)C)n[nH]2)C(C)C1)=O 78227,N#CC1CCCCC1NC(C1CCN(C(=O)CCCC(N)=O)CC1O)=O 78228,c1(N(C)C)cc(N2CC(C(=O)N=S(C)(C)=O)C2)nc(Cc2ccccc2)n1 78229,CC1CC=C(C(=O)NCC2CC(CNC(c3cccc4nccn34)=O)CO2)CC1 78230,C1(C)(Cn2cc(-c3n(C)nnc3)nn2)CCN(C(c2csc(C#N)c2)=O)CC1 78231,CC1(C)CC=C(C(=O)NCCOCC(=O)Nc2cc(CO)ccn2)CC1 78232,c1(OC)cc(C)ccc1C(=O)NCCC(C)NC(=O)C(C)C=Cc1ccccc1 78233,CC1=C(C(=O)NCC2(NC(C3CCCN3C3CCCC3)=O)CCOCC2)CCC1 78234,CC1CCC(C(N2CCCC2CNC(=O)CCc2nc[nH]n2)=O)C1 78235,c1(C(CC(=O)O)OC)cccc(-c2csc(C3NCCN(CC(=O)NC)C3)n2)c1 78236,N1(C(C)C)CC2CC1CN2C(=O)C(F)CC1CN(C2CCCS2)C1 78237,C=CC1(CC(=O)NC(C)C(C)NC(=O)CC2CSC2)CCCCC1 78238,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)C(C)C1 78239,N1(C(C(C)(C)OCCC)=O)CCC2CN(C(=O)NC3CCC=CCOC3)CC2CC1 78240,N1(C(c2c(C)cc(C)o2)=O)CCC(C)(C)C(CO)C1.C1C(C)(C)OCC(=O)N1C 78241,C1(NC(c2nc(OCC)oc2)=O)(CO)CCN(C(c2ncccc2F)=O)C1 78242,c1(C(C(=O)OC)NC(C2(F)CCOC2C)=O)c(C)nn(-c2ccccc2)c1C 78243,Cn1cnc(CNC(=O)C(Cn2cccn2)NC(=O)COCC(F)(F)F)n1 78244,CCC(C(=O)N1CC(CC(C)NC(=O)CC2CCOC2)C1)OC 78245,N1(c2nc(-c3ccc(C)o3)[nH]n2)CCN(c2ccc(-c3nn[nH]n3)cn2)CC1 78246,CC1(C)COCCC1C(C1CC1)NC(c1ccccc1-c1nc[nH]n1)=O 78247,C(CCC(F)(F)F)NCc1scc(C(C)(F)F)n1 78248,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)C(=O)NCC1C=CCOC1 78249,c1(C(=O)NC(C)CCNC(c2cc3ccnn3cn2)=O)c(F)c(F)cc(F)c1F 78250,c1(-n2c(CN)nc(-c3cc(Cc4ccccc4)ccn3)n2)cccc2nc[nH]c12 78251,C(=O)(CC(C)(C)C=CC(=O)OCC)N(CC(C=C)O)C 78252,C1(C(N2CC(C(=O)NCc3cc(=O)cc(Cl)[nH]3)OCC2)=O)CC2(CCC2O)C1 78253,CC(CCCC(=O)NCC#CC#CCO)NC(C1CCCN1C1CC1)=O 78254,c1(CC2N(C(c3sccc3Cl)C(=O)N)CCC2)ccc(OC(F)F)cc1 78255,c1(C(N(CCC)CCNC(C2CCC3CC3CC2)=O)=O)ccc2n[nH]cc2c1F 78256,c1(CC(=O)NC(CC)CN(C(=O)CCCF)CC)ccc(C)c(F)c1 78257,C#CCCCCCCCC(=O)NCC1(NC(=O)CNC(=O)NC(C)C)CC1 78258,CCCCCCCC(=O)NC(CNC(C1CC1C(=O)OC)=O)CC 78259,C1(CNC(COC2(C)CN(C(CCCOC)=O)C2)=O)CCCS1(=O)=O 78260,c1(C(=O)NC(C2CCCCO2)C)ccn(CCNC(=O)CCCc2ncco2)c1 78261,C1(CC(N2C(CCCOCC)CCC2)=O)CCC2(CCC2)O1 78262,N1(C(CCCc2cc(C)no2)=O)CC(NC(=O)CC2CC2(Cl)Cl)CC(F)C1 78263,C(=O)(CCS(N)(=O)=O)NCC(c1ccccc1)N(C(C(CC)OC)=O)C 78264,c1(CC(=O)NC2C(CNC(CSCCOC)=O)CCC2)c(C)cc(C)nc1O 78265,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78266,C1(NC(CNC(C2C(C)C2)=O)=O)CC2CCC1(C(=O)NCC1(F)CCC1)C2 78267,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78268,C1(C(=O)NCC2C(NC(COCC)=O)C2)CCCN1C=O 78269,C1(OC)CC2N(C1)C2=O.C(Cc1ccccc1)(C(F)F)NC(=O)OC(C)C 78270,N1(C(Cc2c(C)ocn2)=O)CCOC(CNC(=O)CC2CCCC(=O)N2)C1 78271,Cc1ccc(F)c(C(=O)NCCC2(O)CCN(C(=O)CCC3(O)CCC3)C2)c1F 78272,C1(C)(C(N(CCCO)C)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 78273,C12(NC(CCC)=O)CCCC1CN(C(c1sc(C(C)C)nc1C)=O)C2 78274,C1(OCCONC(C2CCN(C(c3ccc(O)cc3)=O)C2)=O)CCC2(CCC2)C1 78275,c1(C(N2CC(CC)N(C(C3CC4CC4C3)=O)CC2)=O)ccc2nccn2n1 78276,C1(C(N2CC(C(C)NC(c3ccc(F)s3)=O)C2)=O)CSc2ccccc2O1 78277,N1(C(c2cnc(C(C)OCC)s2)=O)CC2C(NC(C3CCCC(CF)C3)=O)C2C1 78278,CCC(CC)(C(C)C)NC(=O)C(O)CCNC(=O)CC1CC1.C1(C2CC2)CC1 78279,c1(C(C(=O)N(CCCNC(=O)CC2(C)CCCCC2)C)O)ccc(F)cc1 78280,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(c1cnoc1C)=O)C3 78281,N1(C(c2nccc(CC)c2)=O)CCN(C(=O)CC2CN(C)C2)CC1CC(C)(C)C 78282,c1(CN(C(C)C(N)=O)C(=O)CCc2ccccc2)cc(F)nc(F)c1 78283,C1(CN)CC2(CC(C(=O)O)C2)C1.C12CCN(C1)CC1(CC1)C(=O)N2C 78284,c1(C(=O)NC(C)(C)CNC(C2(C)CCCOC2)=O)cc2c(nn1)CCCC2 78285,N1(C(C2C(C)CCC2)COC(F)(F)F)CCC(O)C(N=[N+]=[N-])C1 78286,c1(C(=O)NCC(CNC(C(C)Sc2nncn2C)=O)F)nnc(O)cc1O 78287,c1(OCCOCCNC(C=CC(=O)OCC)=O)cccc([N+](=O)[O-])c1C 78288,c1(NC(=O)NCC2C(C)C2(F)F)ccnc2c(Br)cccc12 78289,C1(Oc2cccc(OC)n2)CCN(C(=O)C2CC2)CC12CCC2.C(C)(C)(C)OC(=O)NC 78290,c1(C(N2CC(CC(C)NC(=O)C(F)(F)c3cnn(C)c3)C2)=O)cc2n(n1)CCCO2 78291,N#CC1NC(=O)CCN(CC2(c3ccccc3OC(F)(F)F)COC2)C1=O 78292,Cc1onc(C2CCCCC2)c1C(=O)NC(CNC(=O)CC(F)(F)F)C1CCC1 78293,Cc1ccc(F)c(C(=O)NCC2(C)CC(NC(c3cnc4n3CCS4)=O)C2)c1F 78294,N1(C(=O)OC(C)(C)C)CC(OC(C2CC2C(=O)OC(C)(C)C)=O)C(C)(C)C1 78295,CC(C)(CC=CC(=O)NC1CCCC1C)NC(=O)CC1CCSC1 78296,c1(C(N2C(C(C)C)CN(C(=O)C=CCO)CC2)=O)cccc2cc(Cl)ccc12 78297,C1(CC)CNC(=O)CN1C(C1(NC(C2CCCCNC2=O)=O)CCCC1)=O 78298,C1(CCCC)CN(C(c2ccc(C(N)=O)o2)=O)CCN1C(c1ccc(O)c(C)c1)=O 78299,c1(C(N(CCN(C(=O)C(C2CC(F)(F)C2)O)C(C)C)C)=O)ccn(C)c(=O)c1O 78300,c1(C(N(C)CC2CCN(C(=O)CCCCc3ccccc3)C2)=O)cnc(S)n1C 78301,N#CC1(C(=O)NC2CC2NC(=O)CSc2ccccc2F)CCCCC2CC12 78302,CCCC(O)C(=O)N(C)CC1CN(C(c2sc(COC)nc2C)=O)CCO1 78303,C1(C(=O)NC2CC3CN(C(=O)CC(=O)NC4CC4)CC23)(OC)CCCCCC1 78304,c1(C(=O)NCCCCNC(C2(C#C)CCOCC2)=O)ccsc1S(N)(=O)=O 78305,CC(CNC(C1(C(C)(C)O)CC1)=O)CC(=O)Nc1cccc(O)c1 78306,CN=c1[nH]c(=NCc2cncc(C)c2)[nH]c(=NC2CCN(c3cc(C)nn3C)C2)[nH]1 78307,Cc1cnc(C(=O)NCCC2CCN(C(C3(c4ccncc4F)CC3)=O)C2)cn1 78308,C(C(F)(F)C(=O)NC(c1scc(N(C)C)n1)C)n1c(CO)nnn1 78309,N1(C(c2ccccc2[N+](=O)[O-])=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC2C1 78310,C1(CNC(C(C)=O)=O)CCC(C)(C)CN1C(c1sc(C)nc1C)=O 78311,C1(NC(C(C=CC)O)=O)CCCN(C(CO)C(C)C)C1 78312,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2snnc2C)=O)Cc2ccccc2C1 78313,C12(C(N3CCC(OCCNC(CCCOCC)=O)C3)=O)CCCC1CC(=O)CC2 78314,c1(CNC(C2CC(CC(=O)NC3CC(Cl)(Cl)C3)C2)=O)cc(F)c(F)cc1O 78315,c1(OCCNC(N(C2CC(C)(C)C2)C)=O)ccc(S(N)(=O)=O)cc1F 78316,c1(CNC(CN(CC)CC)=O)ccc(SC)c(OC)c1 78317,CC1CCN(C(c2ccoc2Cl)=O)CC1NC(c1cnc(-c2ccccc2)o1)=O 78318,N1(C(C(C=C)C)=O)CCC2(C=C(C(=O)N3CCOCC3C3CC3)C2)C1 78319,c1(C2(C(N3CCC(N(C)C(c4nccnc4N)=O)C3)=O)CCC2)ccc(F)c(Cl)c1 78320,C(CC(C)(C)CNC(=O)C(=O)NCc1ncc(C)o1)OC 78321,C(=O)(CC(C)C(C)(C)NC(C1CCCC1n1cccc1)=O)OC 78322,CC1CC2(CCCC2)CN1C(C1CCC(C2CC2)N1C(C1CCCN1C1CC1)=O)=O 78323,CC1CC(NC(=O)CCc2ccsc2Br)CCS1(=O)=O 78324,N1(C(C(CC)CN(C)C)=O)CCN(C(=O)COc2ccc(Cl)c(Cl)c2)CC1C 78325,C(CS(=O)(=O)Cc1cn(C2COCC2OC(C)C)nn1)NC(c1c(C)noc1)=O 78326,C(C(C)C(F)C(=O)NCC1C2CCCCC12)NC(c1c(C)cnn1C)=O 78327,C(=O)(C(C)(C)NC(=O)C=Cc1ccco1)NC(C)CC1CCCO1 78328,c1(OCCC)ccccc1C(=N)NOCC1CC12CCOCC2 78329,C(=O)(CCCCC(C)=O)N1C(C)CC(CC(N2CC(CC#CC)C2)=O)C1 78330,N1(C(C2(C(=O)NCC=C(C)c3ccco3)CC2)=O)CCCC(N=[N+]=[N-])C1 78331,c1(OCCCOCCC(=O)NCC(CNCCCOC)OC)c(C)cc(Cl)cc1C 78332,C(CCC(=O)N1CC(CC2CCCC2)C1)N(C(C(C)=C(CC)C)=O)C 78333,CC1CN(C(c2occc2Br)=O)CC(C)C1NC(=O)Cn1nnnc1C1CC1 78334,c1(N(C)C)ccc(C(=O)NCC2CCCN2C(c2snnc2C2CC2)=O)nc1 78335,Cc1nccn1CCCC(=O)N(C)CCN(C)C(c1cc(C(F)(F)F)n[nH]1)=O 78336,c1(C(=O)NCC(C)C)cc(OC(c2ccccc2)C(=O)O)ccn1 78337,CCC(C)C(=O)NCC(=O)N(CCNC(c1cc(C)no1)=O)CC1CCCC1 78338,N1(C(c2c(CC)c[nH]n2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC1CCCOC1 78339,Cc1cc(NC(C2CC23CN(C(c2cc4sccc4[nH]2)=O)C3)=O)ccc1Cl 78340,N1(CCC#C)CCN(C(=O)C(C)(C)NC(=O)C=Cc2ccsc2)CC1 78341,N1(CC(=O)NC(C2(O)CCN(C(c3cn(CCO)nn3)=O)C2)C)CCNC(=O)C1 78342,c1(N(C)Cc2ccnc(C)n2)nc(N2CCn3nnnc3C2)c2c(n1)CSC2 78343,C1(C(N(C(CC(=O)OC)c2ccccc2)C)=O)CCN(CP(C)(C)=O)CC1 78344,N1(C(c2c(Cl)ncc(N)c2)=O)CC2CCCC1(CNC(=O)CCC(F)F)C2 78345,C1(F)(C(N2CCC(N(C)C)C2)=O)CCN(S(=O)(=O)Cc2ccc(Cl)cc2)CC1 78346,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78347,Cc1cnc(CN(C(C2CN(C(=O)CN3CSCC3=O)C2)=O)C(C)C)[nH]1 78348,Cc1cc(C(=O)NCCN(C)C(c2cc(Br)c(C)o2)=O)c(Br)c(C)c1 78349,c1(C(=O)NC2CC3CN(C(CCOCCC)=O)C2C3)nc2cc(O)ccc2[nH]1 78350,C1(N(C(=O)CN2CCOCC2)C)CN(Cc2cnc(Cl)s2)CC1(C)C 78351,N1(C(C2C(C=C)OCCC2)=O)CC2OCCN(C(c3cnc(CC)o3)=O)C2C1 78352,Cc1csc2cc(C(=O)NCC(C)N(C(=O)Cc3csc4nc(C)cn34)C)[nH]c12 78353,CC1(C)C(NC(=O)Cn2cnccc2=O)CCN1C(=O)Cc1cccnc1N 78354,c1(C(=O)NCCOC2CCN(C(ON=CCC)=O)C2)ccc2c(c1)CC(C)O2 78355,C#Cc1ccc(OCC(=O)NCC2(NC(=O)C=Cc3ncccc3C)CC2)cc1 78356,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78357,c1(C(=O)NCC(C(C)C)NC(c2c(OC)cc[nH]2)=O)ncc(N)cc1C 78358,c1(OCC)cc(CNC(=O)CC(c2cccs2)C2CC2)ccc1OC(F)F 78359,C1(O)(CNC(CCSCCC)=O)CCN(C(C2(NC(C)=O)CCC2)C)C1 78360,C(=O)(CCCC(F)(F)F)NCCNC(CN(CCN(C(C)C)CCOC)CC)=O 78361,N1(C(c2cnc(CC(C)=O)s2)=O)CCC(NC(C2CCC(=O)NC2)=O)CC1C 78362,CCC(O)C(C)C(=O)N1CCC(O)(C(C(=O)NC2CCCCC2)c2cnsc2)CC1 78363,c1(C(N(C(C)CNC(=O)Cn2[nH]cnc2=N)C)=O)ccnc(Cl)c1Cl 78364,c1(C(=O)OC)cc(=NC(=O)C(C)C(C)NC(=O)C(C)CCOC)[nH]n1C 78365,CC1(C)C2CCC(C(=O)NC3C4CN(C(=O)Cc5cccnc5O)CC34)C1C2 78366,C1(CC=C)CN(N2CCCC3(CCC(F)(F)C3)C2)CCN1C(=O)OC(C)(C)C 78367,N1(C(c2ccc(CNC(C(C(CC)C)N(C)CC)=O)o2)=O)CCCC2(CC1)CC2 78368,C(=O)(CCCCC(F)(F)F)NCCCN(C)C(c1nnc2n1CCCC2)=O 78369,CC1CCCCC1(CNC(C1C2(CC2)C12CC2)=O)NC(=O)CN1CCSCC1 78370,C1(CNC(c2ocnc2C2CC2)=O)COCCN(C(=O)Cc2cn[nH]c2)C1 78371,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2nc(C)cn2c1 78372,CC1=CCC(C(=O)NCC(C)(C)NC(C2CCCN(C(=O)OC(C)C)C2)=O)CC1 78373,N1(C(C2N(Cc3cnc(C)nc3)CC3(CC3)C2)=O)Cc2ccc(Cl)nc2C1 78374,N1(C(c2ccc(NC(C)=O)cc2)=O)CC2CN(C(=O)Cc3ccsc3)CC2C1 78375,C1(c2n(CCCN(C(=O)OCCOCC(C)(C)C)C)nnn2)(SC)CCN(C)CC1 78376,c1(C(n2cc(C(C)NC(=O)CCc3ccsc3)nn2)C)cccc(Cl)c1Cl 78377,C(=O)(C(CNC(c1ccc(OC)o1)=O)CC(C)C)N(CCOC)C(C)C1CC1 78378,Cc1c(N)cc(C(=O)NCC2CCN2C(=O)C(C)CC(C)(F)F)cc1N 78379,Cc1cc(NCc2ncc(-c3ccccc3)[nH]2)sc1C(N1CCCCC1)=O 78380,C1(NC(C(CC)c2cccnc2)=O)CN(C(=O)COCC(=O)NC)CCC1F 78381,C(=O)(C(O)CCN(C)C)NC(C1CCCCC1)C(=O)NC(C)COC(F)(F)F 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78471,C(C(C)(C)C1=CCCC1)NCC(NOCc1scc(C(=O)OCC)n1)=O 78472,N1(C(Cn2ncc(C)c2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 78473,c1(C(=O)OC)ccc2[nH]c(=NCC3CCC(NC(=O)CCCN(C)C)C3)sc2c1 78474,C1(CC)(CC)CC(NC(c2ncncc2Cl)=O)CN1C(=O)C(F)F 78475,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 78476,n1(CC(=O)NCC2CN(C(c3cc(C)ncc3)=O)CC2C)nnc2ccccc12 78477,C(=O)(C1=CCCOC1)NC1C(OC)CCCC1.c12ccccc1NC(=O)C21CC1 78478,CC(=O)CCCC(C)C(=O)NC1(C(N2CC(C)C2)=O)CC(O)C1 78479,c1(C(=O)N(C(CNC(C(C)NC(=O)OC)=O)CO)CCO)ccc(OC(F)F)cc1 78480,N1(C(CS)=O)CC(NC(=O)CCOCC(F)(F)F)CC1CO.Cn1cnnc1C1CC1 78481,c1(CN(C(C(C2CCCC2)NC(C2CC(=C)C2)=O)=O)C)cccnn1 78482,C1(C(C(=O)NCC(C)N(C)C)(C)C)CCCN(C(=O)CC(=O)NC2CC2)C1 78483,C1(CNC(c2cn(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=Cc1ccc[nH]1)C2 78484,CC1CCc2ncc(C(=O)NC3CCN(C(C4CCCSS4)=O)CC3C)n2C1 78485,N1(C(C(C(C)C)OCC)=O)Cc2occ(C(=O)NC(C)C(O)C(F)F)c2C1 78486,C=CCC(CNC(=O)C(O)c1ccco1)C(=O)NCCC(C)C 78487,C1(NC(c2c(CNC(CCC(C)N(C)C)=O)n[nH]c2)=O)CCC(O)C(O)C1 78488,C1(C(=O)NC(C(=O)OC)Cc2cn(CC(C)(C)C)nn2)CCn2cncc2C1 78489,Cc1cnccc1C(C)C(=O)NC1COCCC1NC(c1ncn(C)c1C)=O 78490,C1(NC(CS(CC)(=O)=O)=O)CN(C(=O)Cc2conc2C)Cc2ccnn2C1 78491,c1(OC)ccc2c(N3CCCN(C(c4cc(C)ccc4Cl)=O)CC3)ncnc2c1 78492,CC1(C(N2CCC(N(CCO)C(C3(CF)CCOCC3)=O)C2)=O)CCCCO1 78493,c1(C(N2CCC(C)(C(=O)NCC3CSC3)C2)=O)cc(F)cc(F)c1 78494,CC1(C)OCCC1(O)C(=O)NC(C(=O)NCc1ccn(C2CC2)n1)C1(C)CC1 78495,c1(C(=O)OCCCOCCOC)c(Br)c(SC)nn1C 78496,c1(CC)c(C(=O)N(C2CCCN(C(=O)CC(CC)OC)CC2)CC)cccc1F 78497,C(=O)(C#CC1CCC1)Nc1c(N(C)C)nn(C)c1.c1(C2C(=O)O2)ccccc1 78498,N1(CC(C)(C)N(C)C(=O)OCC(C)(C)C)CCN(C(=O)C(C)(F)C2CC2)CC1 78499,CN1CCN(CC(=O)NCC(O)CCC2CC2)CC1.N12CCOC(C1)C2=O 78500,c1(OC)cnc(C(=O)NCC(C)NC(c2ccc(C)c(C)c2)=O)c(OC)n1 78501,C(=O)(CC(C)(C)CN(C)C)NCC1(OC)CN(C(=O)CC2CCOC2=O)C1 78502,C=CCCCC(=O)NC(C1CCCCC1)C(C)NC(=O)CC1CC1 78503,N1(C(c2cc(C)no2)=O)CC2(CC2)CC1CNC(=O)CC1CC(C)C1 78504,C1(N(C(c2c(C(C)C)c[nH]n2)=O)C)CCN(C(c2cn(C)cn2)=O)CC12CC2 78505,CS(=O)(=O)c1ccc(F)c(C(N2CCCN(C(=O)C3=CCCCO3)CCC2)=O)c1 78506,C1(C)(NC(C2CC(SC)C2)=O)CCCN(C(c2ccc(F)cc2SC)=O)C1 78507,c1(C(=O)NC2C(NC(=O)CCSc3ccnc(O)c3)C2)c(F)ccc2[nH]ccc12 78508,CN1CCOC(C(=O)NCC2CN(C(=O)CCc3ncc[nH]3)CC2(F)F)C1=O 78509,c1(CC(=O)NC2CN(C(=O)CC3CCCCC3O)C2)ccc(O)cc1Cl 78510,C1(C)(CNC(CC2C(C(=O)OC)CC2)=O)CCCN(C(C2C3CCCC23)=O)C1 78511,c1(C(N)Cc2noc(Cc3ccc(Br)cc3)n2)c(Br)ccc(F)c1F 78512,CC1(CNC(=O)CCNC(C2(C)CCC(=O)NC2)=O)CC2(CCC2)C1 78513,c1(SC)ncc(C(F)(F)F)c(CN2CCC(CNc3ccc(F)cn3)C(C)C2)n1 78514,N1(C(CC2(C=C)CC2)=O)CCCC(NC(C2CCSCC2)=O)C(F)C1 78515,C(C(=O)N1CCC(C)(NC(c2cncc(OC)n2)=O)C1)(c1ccccc1)=CC 78516,Nc1cc(Cl)ncc1C(=O)NC1CC2(C1)CN(C(C1CC(O)CN1C(N)=O)=O)C2 78517,C1(CN(C(=O)CCN2CCCC2)C)COCCN1C(c1nc(Cl)c(Cl)s1)=O 78518,CC(CS(C)(=O)=O)C(=O)NC1CC(CCNC(c2ccc(C3CCOC3)s2)=O)C1 78519,Cc1[nH]nc(C(N2CCC2CC(=O)NC2(CC3CC3)CC2)=O)c1C 78520,c1(C(N2CC(C)(NC(C(C)NS(C)(=O)=O)=O)C2)=O)ccnc(C(C)(C)C)n1 78521,O=C(C1=CS(=O)CCC1)N1CCC(F)(Cc2cn(-c3cncc(F)c3)nn2)CC1 78522,N1(CC(=O)N(C(c2ccccc2)CNC(CCOC)=O)C)CCCCC1=O 78523,CC1(O)CCN(C(=O)CCC2CCCCN2C(=O)CCNC(=O)CO)CC1O 78524,C1(CNC(C(CC)C#N)=O)CC2CCCC2N1C(c1ccccc1F)=O 78525,C1(C#N)(C(=O)OCC)CCN(CC(CO)C(C)(C)C)CC1 78526,c1(OC)cc(N)c(Cl)cc1C(=O)NCCC(C)(C)NC(c1ccon1)=O 78527,N1(C(C2N(CC)CCC2)=O)CCC(O)CC1C(=O)NC1C2C=CC(C2)C1CO 78528,CNS(=O)(=O)CC(C)N(C)Cc1cccc(Cl)c1Br 78529,C(=O)(C1=CCCCCC1)NC(C(=O)NCC(C)O)CN(C)C 78530,C1(C)(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CC2)=O)CCCCCC1 78531,C(c1ccco1)=C(C(=O)NCC(C)O)C.c1(NC(N2C(=O)CC2)=O)cc(Cl)ns1 78532,Cc1cc(C(N2CCC(CNC(c3ccc(CC(C)C)s3)=O)C2)=O)cc(O)c1 78533,c1(C(=O)NC2C=CC(CC(=O)NCCCCN(C)C)C2)cc(O)cc(F)c1 78534,C1(C=C)(NC(CN(C(=O)CCN2CCOC2=O)CC#C)=O)CCCCC1 78535,N1(C(=O)NCCn2c(CC)ncc2)CC(c2cccc(Br)c2)C1(C)C 78536,C1(NC(=O)CCc2cccnc2F)CN(C(C23CC(F)C2C3)=O)CC12CCC2 78537,N1(C(CC2(C)CCCC2)=O)CCOCC(NC(=O)CCC2CCC2)C1 78538,C1(C(c2ccccc2)NC(c2c(NC(C)=O)cccc2)=O)CCCN(CCO)CC1 78539,C#CC1(C(N2CCC(OC3CCC3)C2)=O)CCN(C(C2CN(CC)C2)=O)C1 78540,Cc1onc(Br)c1C(N1CCC(C(C)NC(c2cccnc2O)=O)C1)=O 78541,CC(C)C(F)(F)CC(=O)OC(C)(C)C.C12CCC(C1)OC(=O)CCOC(=O)N2 78542,c1(OC)ccc(C(=O)N(C2CN(C(c3c(C)cccc3Cl)=O)CC2F)C)c(F)n1 78543,C(CC(O)CCO)C=O.C12C(O)CCN1C(=O)CONC2=O 78544,c1(NCC(CC)N(C(c2cc(Cl)cc(Cl)c2)CC)C)ncnc(COC)c1C 78545,C1(C(=O)NOCC2CC=CCC2)CC2(CCC2)C1NC(c1nn(CC)nc1C)=O 78546,CC(C)C(CNC(C1CCC2(CC1)CC2)=O)C(=O)NCC(C)Cc1cn[nH]c1 78547,CCCN=C(NCCN1CCCCCC1)N1CCN(c2ccccc2Cl)C(=O)C1 78548,CC(C)(C(C#N)NC(=O)C(=O)NCCC1CCS(=O)(=O)C1)c1ccccc1 78549,c1(C(=O)NC(C(C)NC(C(C)SC)=O)CO)ccc(N(C)C)c([N+](=O)[O-])c1 78550,c1(OC)cccc(CNC(C2CCN(Cc3ccn(C)c3)C2)=O)c1O 78551,n1(CC(=O)NCC2C(NC(CC(=O)NCC#C)=O)CCC2)nc(C)ccc1=O 78552,C(=O)(C1=CCCCC1)NCC(CN(C)C(C1(CC)CCC1)=O)O.CO 78553,C1(C(N(C2CC(NC(CC(=O)OCC)=O)C2)C)=O)CN2CCN1CC2C 78554,N1(C(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)N(C)C 78555,C1(C(C)C)CN(C(=O)CCCc2nncn2C)CCN1C(=O)C(=O)C(C)(C)C 78556,CC(CN(C(=O)CC(=O)NC1CC1)C)C(=O)NCCC(C)C1CCCC1 78557,CCC(C)(O)C(=O)NN1CCCC1NC(C1CCCC1NC(=O)C1CC1)=O 78558,N1(C(CCc2ccc(CC)cc2)=O)CC(C(=O)Nc2cc(CC)on2)C(C)(C)C1 78559,C(=O)(CC(C)n1cccn1)NCC(C)NC(COCCSC)=O 78560,c1(C(=O)NC(C)CN(C(=O)C(C)(O)C(F)(F)F)C)cc2cccc(Cl)c2s1 78561,c1(N(C)C)ncccc1C(=O)NCC(c1cccc(Cl)c1)NC(C1(O)CC1)=O 78562,CC(CNC(C12CC1CCN2C(C1CC1C(C)(C)C)=O)=O)C(F)(F)F 78563,N1(C(c2c(C)onc2)=O)CCC2(CCC2)C(NC(C2(CC3CC3)CCCC2)=O)C1 78564,C1(NC(=O)CSc2nncs2)CC2CC1N(C(c1ccc(O)nc1Cl)=O)C2 78565,CC1(C)CCCN(C(=O)CCc2cnco2)C1C(=O)NCC1CC1[N+](=O)[O-] 78566,c1(C(=O)NCC(C)CN(C)C(c2ccc(CO)c(F)c2)=O)cc2cn[nH]c2cn1 78567,C(CCC(O)C(=O)Nc1cccc(F)c1C)NC(c1cncc(C(=O)OC)c1)=O 78568,C1(C#N)(C(N2C(C)CC(NC(C3CC4CC4C3)=O)C2)=O)CCCCC1 78569,C(C(CNC(C1(CO)CCCO1)=O)C(F)(F)F)NC(C=C1CCN(C)CC1)=O 78570,c1(C(=O)NCCC(=C)CNC(c2sc(C)nc2CC)=O)cccc(C(=O)NC)c1 78571,C1(C)(CNC(c2cccc(OC)n2)=O)CCCN(C(=O)CONC(=O)OC(C)(C)C)C1 78572,N1(C(c2n(CC)ncc2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)CC1(C)C 78573,N1(C(c2nc(C)sc2)=O)CC2CCCC2(NC(=O)CN2CCC(=O)NC2=O)C1 78574,N1(C(Cc2c(C)ncs2)=O)CCC(C(N2CCN(C)CC2C)=O)C12CCC2 78575,N1(C(C)C)CC(NC(=O)N(CCN2CCN(C)CC2)Cc2ccccc2)CC1=O 78576,CCCC(CC(=O)NC(C)(CO)CCF)NC(C1OCCCC1(C)C)=O 78577,Cc1c(C(=O)NC(C)(CNC(=O)C(C2CCOCC2)C)CO)cnc2ncnn12 78578,C1(CC(=O)NC2CN(C(c3c(C)oc(C(C)C)c3)=O)C(C)C2)CCCC(C#N)C1 78579,C(CC(C(=O)NC1CCN(C(N)=O)C1)NC(c1occc1C)=O)N(C)C 78580,Cc1cc(C(=O)NC2C3CC2N(C(c2ccc(Cl)nc2N)=O)C3)c2occc2c1 78581,C(=O)(CC1OC(=O)c2ccccc21)NC1CC1c1c(C)ccc(F)c1.C1(=O)CO1 78582,CC(C)C(O)C(=O)NCC1CN(C(c2ccnc(-c3ccccc3)n2)=O)C1 78583,C(=O)(CC(COC)NC(=O)C1=C(C)CC1)NCC(COC)(C)C 78584,c1(CC(C(=O)O)NC(=O)NC2CCCC(C(N(C)C)=O)C2)cccc(Cl)c1F 78585,C1(NC(c2n(CC)cc(Cl)c2)=O)CCC(O)CN(C(=O)C=C(C)C(C)C)C1 78586,C1(C(N(C(c2ncc(C)s2)=O)C)C)CN(C)CCO1.n12cc(nn1)CNC(=O)C2 78587,C1(C(=O)NC(CNC(c2cnc(NC(C)=O)o2)=O)CC)CC12CCCCC2 78588,CON1CCC(C(=O)NCC2(O)CCCN(C(=O)CC3CCC3(C)C)C2)CC1 78589,N1(C(c2c(C)ncs2)=O)CCOCCC1C(=O)N(C1CCCCC1(C)C)C 78590,C(C(CNC(c1ncnc(C)c1C)=O)C(F)(F)F)NC(C=C(CC)C)=O 78591,N1(C(Cc2cccc(CC)c2)=O)CCN(C(=O)C(C)CF)CC(C)(C)C1 78592,c12ccc(cc1Cl)-c1nnc(o1)C(CC(C)C)C(=O)N2.c1cnn(CCF)c1 78593,Cc1cc(Br)ccc1C(N1CCC(CN(C)C(c2cccc(Cl)c2F)=O)CC1)=O 78594,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CC2)cnc2ccccc2n1 78595,CC1(C)CC2CN(C(=O)CC3CCCN3C(C3CC3F)=O)CC12 78596,C1(C(=O)NCC(=C)CCNC(=O)C(C)Sc2ccco2)(N(C)C)CCCCC1 78597,C=CCC(CNC(C1(CC)CCOC1)=O)C(=O)NC(C)(C)CNC(C)=O 78598,c1(C(N2CCC(CCCCNC(C3CC(=C)C3)=O)CC2)=O)cc(N)c(Cl)c(O)c1 78599,c1(C(=O)NC2C(NC(C3N(C(CC)=O)CCCC3)=O)CC2)cc(N)ccc1Cl 78600,CC(=O)CCCCC(=O)N1CCC(C(=O)NCc2ncccc2F)(CF)C1 78601,N1(C(CNS(N)(=O)=O)=O)CCCC2(CCCN2C(C2C3CCCOC23)=O)C1 78602,C(N=c1[nH]c2ccc(Cl)cc2s1)C1C(C)CN(C(C2(C)CNC(=O)C2)=O)CC1 78603,c1(CC(=O)NCC23CCN(C(CC=C)=O)CC2C3)cn2cc(Cl)cc(Cl)c2n1 78604,c1(CC)ccc(C)cc1NC1(c2nnnn2CCCOC)CC2(CSC2)C1 78605,CCCCCCCCC(=O)NC1CCN(C(c2ccc(N)c(O)c2)=O)C1 78606,CCC(C)(CC)C(=O)NCCCN(CCCNC(C1CCC(=O)NC1)=O)C 78607,CC1(C)COCC1CC(=O)NCC1(NC(c2ccc(C(=O)NC)cc2)=O)CCC1 78608,C=CCC(CC=C)C(=O)NCC1CC2COCC2N1C(c1cc(C#N)on1)=O 78609,CC(C)(CC(=O)NC12CN(C(=O)C=CCNC(N)=O)C(CO)(C1)C2)CC(F)F 78610,N1(C(CCCC(=O)NC(C)C)=O)CCC2(CC1)CC2CNC(=O)C(F)C(C)(C)O 78611,c1(C(=O)NC2CCN(C(COC(CC)C)=O)C2)nc(S(N)(=O)=O)c2ccccn12 78612,CN1CCN(C(=O)Cc2csnn2)C(CNC(c2cc3[nH]ccc3s2)=O)C1 78613,c1(OC)cccc(Cl)c1CN1CC(CO)(NC(c2cccnc2C(F)(F)F)=O)C1 78614,CC1=C(C(=O)N2CCCC2CCNC(C23CC(C)(C2)OC3(C)C)=O)CCS1(=O)=O 78615,C1(NC(c2c(C(C)C)scn2)=O)CCCC12CN(C(c1cnoc1C1CC1)=O)C2 78616,C(CCSC)(C(=O)NCCC1(NC(=O)COCP(C)(C)=O)CC1)OC 78617,Cc1cc(Br)c(-c2nnc(NC(=O)C(F)(F)F)o2)c(Br)c1 78618,C1(NC(C(C)S(C)(=O)=O)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)CN(C)C1CC1)C2 78619,c1(C(=O)NCC2C(O)C(O)CN2C(=O)C=CCO)cc2c(nc1O)CCSC2 78620,CC(CC(F)(F)F)C(=O)NCCOCC(C)(C)NC(c1cc2ccccn2n1)=O 78621,c1(N(CCN(C(c2ccc(C)nc2C)=O)C(C)C)C)ncnc2sc(C)nc12 78622,N1(C(CCc2onc(CCC)n2)=O)CC2CCC(CNC(C3(CF)CC3)=O)(C2)C1 78623,c1(N2CCC(COC)(NC(=O)Cn3cccn3)CC2)nccc(S(C)(=O)=O)n1 78624,n1(CC(=O)N(C2CCN(C(=O)C(c3csc(C)n3)=O)C2)CCC)c(C)csc1=O 78625,CON=Cc1ccc(C(=O)NCCCn2cc(C(O)C(C)(C)C)nn2)cc1 78626,N1(C(C(C)NC(C(n2c(C)ncc2)C)=O)=O)CCc2ccc(C#N)cc2C1 78627,N1(C(C(=O)NCCCSC)C)CCCC(c2nn(C(C)C)cn2)C1 78628,C1(COC)CCC(CC(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)OC)CC1 78629,C(C(CC)(CC)C(=O)NCc1cc(C(C)C)no1)NC(C1C(CC)CCCC1)=O 78630,c1(C(N(C)CCN(C(=O)CC(O)CN(C)C)C)=O)ccc(N)c(Cl)n1 78631,C12CN(CC13CCC3)C(=O)C1CCC1(NC(C(CC)CC)=O)NC2=O.OC 78632,N1(C(C23CN(C(=O)CC4CC5CC5C4)C(CC2)CC3)=O)CCN2C(=O)NCC2C1 78633,c1(NC(c2c(C(C)C)noc2)=O)nc2ccccc2s1.C1(=O)CCO1 78634,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(C1CCCO1)=O)C2 78635,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CCCCC3)(C1)C2)OC 78636,C(=O)(CCCCCCN=[N+]=[N-])N1CCCC(C)(NC(c2c(C)[nH]sc2=O)=O)C1 78637,CC1CN(C(=O)C(c2cccc(F)c2)N(C)C)CCN1C(=O)C(C)(C)C#N 78638,Cc1nc(O)c(C(N2CC(NC(=O)CCC(C)(C)F)C2)=O)cc1Br 78639,C(=O)(C(O)C(F)(F)F)NCCOCCCN(C(=O)CCc1ccccc1Cl)C 78640,C(CCC)(C(O)C(=O)NOCCOC)CCCSC.CCCCCC(C)C(=O)N 78641,N1(C(c2ccc(F)cc2)=O)CC=C(C(=O)N2CCCC(C(F)F)C2)CC1 78642,CC(C)(C)C(CNC(c1cccc2nccn12)=O)C(=O)N1CC(S(C)(=N)=O)C1 78643,N1(S(CCCOC)(=O)=O)CC(NC(=O)C(C)(C)c2cscn2)CCC1C 78644,c1(N2CCC(C)C(Nc3cc4c(s3)CCC4)C2)ncnc2cc(F)c(F)cc12 78645,C1(C)(C(N2CC(COC)(CNC(C3CCCO3)=O)C2)=O)CC2CC2C1 78646,N1(CC)CCCC(C(N2CCCC2C(C)(C)NC(=O)CC(C)(F)F)=O)C1 78647,CCC(CCCC(=O)N1CCCC1SC1CC1)NC(c1csc(C(C)(F)F)n1)=O 78648,C(=O)(CC(C(N)=O)NC(=O)C1CC1)N(CCCNC(=O)CCC1CC1)CC 78649,c1(C(=O)NCC(O)CCNC(C2COCCC2(F)F)=O)ccc2ccnn2c1 78650,N1(C(COCCC#C)=O)CCC2CN(C(=O)CC3CC4C=CC3CC4)CCC2C1 78651,N1(C(c2c(C)cc(F)cc2)=O)CC(C2CN(C(C3(O)COC3)=O)C2)C1 78652,C(=O)(C(c1cccs1)NC(C1CCCS1)=O)NCCOCC(=O)OC 78653,c1(CN2CCN(C(c3c(C)nsc3)=O)C(C)C2)ccccc1[N+](=O)[O-] 78654,c1(SC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 78655,CC(C)C(CNC(C1CCN1C)=O)C(=O)N1CCC1c1ccccc1 78656,O=S(=O)(c1cccc(O)n1)N1CCN(c2ccc(F)cn2)CC1 78657,Cc1ocnc1CC(N1CC(CNC(=O)C=CC2CCCO2)C1)=O 78658,C1(NC(CCCCOCC)=O)CC2CCC1N(C(=O)CSc1nc(C)no1)C2 78659,CCC(CC)C(=O)NC(C(C)c1ccccc1)C(=O)NCCNC(N)=O 78660,c1(C(=O)NC2C(C)CCN(C(=O)C=CBr)C2)nccc2ncccc12 78661,N1(C(CC=C)=O)CCC(O)(C(C)NC(=O)CCCc2ccccc2)C1 78662,C(=O)(C1SCCc2sccc21)N1CC(C)C(C)(CNC(c2n[nH]cc2Cl)=O)C1 78663,c1(C2CCN(C(C(C)NC3CCCC3)=O)C2)ccc(Cl)c(F)c1 78664,C(=O)(CCCCCC(C)O)NC1C2CN(C(c3nn(CC)c(C4CC4)c3)=O)C1C2 78665,c1(C(=O)NCC(C)(CC)NC(C(C=CC)O)=O)ccc2c[nH]nc2c1 78666,Cc1occc1C1(C(=O)N(CCCNC(C2CCC3CC23)=O)C(C)C)CC1 78667,c1(CC(C(=O)O)NC(C2CCC(C(C)(C)C)C2)=O)c(F)cccc1Cl 78668,C(=O)(CC1=CCCCC1)N1CC2(CN(C(C(CC)OC3CCOCC3)=O)C2)C1 78669,N1(C(CC(C)SC)=O)CCOCC(NC(=O)C(Oc2cccc(Cl)c2)OC)C1 78670,c1(CC)cc(C(=O)NC2CC(CNC(C3CC(OC)C3)=O)C2)nn1C 78671,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(C(C)C)c1C 78672,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 78673,c1(OCC)cccc2c1CN(C(=NCCF)NCCC1CN(C)CCO1)CC2 78674,Cc1ccc(S(=O)(=O)NC2CCCN3CCCC23)cc1[N+](=O)[O-] 78675,C(C(=O)NN1CCCNC1=O)S.N12CCN(CC1)C(=O)NOC1CC2C1.CO 78676,N1(C(C2CC(C)(F)C2)=O)CCN(C(=O)C=CCO)CC2CCCCC12 78677,C1(NC(c2cnc3[nH]nnc3c2)=O)CCN(C(=O)CN2CCCCC2)CCC1CO 78678,C1(C(=O)NC(C)CNC(c2nocc2Cl)=O)CCC(N2C(=O)CCC2=O)CC1 78679,N1(C(c2c(OC(C)C)cncc2)=O)CC2CC(NC(=O)C=C3CCC3)CC1C2 78680,CC(C)CCCC(=O)N1CC2(CNC(=O)C=CSCc3ccco3)CC1CO2 78681,N1(C(C(C2CC2)OC)=O)CC=CCC1C(=O)NCCCNC(N)=O 78682,c1(C(N(C(C(N2CC(CCC)C2)=O)C2CC2)C)=O)cc(C)cc(O)c1 78683,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 78684,c1(N(CCN(C(C)C)C)C)ccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)c(Br)c1 78685,C1(C(=O)NC2CCN(C(CSCCC(C)C)=O)C2C)CCC2CC1CO2 78686,N1(C(C(C)C#N)=O)CCN(C(=O)CSC(F)(F)F)CC1c1cc(F)cc(F)c1 78687,C1(NC(C#CC(C)(C)C)=O)CC2(CCN(C(=O)CSc3ccccc3Cl)C2)C1 78688,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)N(C1CSC1)C 78689,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 78690,C1(CC#C)(C(=O)NCCCOCCNC(=O)CCC2CCCN2C)CCOC1 78691,c1(CCC)cccc(C(=O)N(C)CC2CCN(C(C34CC(C)C3C4)=O)C2)c1 78692,N1(C(CCCOC)C(=O)NCc2ccco2)CCn2nc(CO)cc2C1 78693,c1(C(=O)N)cc(Br)ccc1N.CCC(O)C(=O)NCCC(C)C(C)=O 78694,c1(Cc2ncn(C(C)(C)Cc3ccc(Cl)cn3)c2)ccccc1Cl 78695,N1(C(CCn2c(C)ncc2)=O)CCCCCCC1C(=O)N(C)CC1CCOC1C 78696,N1(C(C2C(OCC)C2)=O)CCC(C)(C(=O)NC(CO)C2CCC2)CC1 78697,c1(OCC)cnc(C(N2CCC(CNC(C3COC4(CCC4)C3)=O)C2)=O)c(Cl)c1 78698,C1(NC(C(C)(c2ccccc2)NC(C)=O)=O)CC(F)(F)C1(C)C 78699,C1(C(N(CC(O)CNC(c2cscc2Cl)=O)C)=O)Cc2nccnc2C1 78700,C1(CCC(=O)NCC(C)NC(C2C=CCC2)=O)CCCCC1 78701,c1(C(=O)NCCOCCCNC(c2cnns2)=O)ccc(C(F)(F)F)cc1Cl 78702,N1(C(c2cc(C)sn2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C2CCCCC12 78703,C(=O)(CC(C(F)(F)F)NC(=O)C(CC1CCC1)OC)NCC(CC)(C)C 78704,C12(CCc3cn(C4CCC(N(N5CCCC5)C)C4)nn3)COC(C)(C1)C2 78705,C(C1=CCN(C(=O)Cc2ccc(O)cn2)CC1)NC(c1c(C(C)C)n(C)nc1)=O 78706,CC1CCCN(C(=O)CCCCC#N)C1CNC(c1cc[nH]c1)=O 78707,n1(CC(CC)O)cc(C(=O)NCC#CCNC(=O)C(C2CCCC2)OC)nn1 78708,c1(C(=O)NCCC(O)CNC(C2C3CCC2(c2cnco2)C3)=O)cccc(Cl)c1F 78709,CC(C)CCCCCC(=O)NCC(C)CNC(=O)C=CC1CCOC1 78710,CCC(C)(C)C(O)C(=O)N(C1CCN(C(C2(O)CCC(C)CC2)=O)CC1)CCO 78711,C1(NC(c2cc(F)ccc2F)=O)CCC2(CC2)N1C(=O)Cn1cccn1 78712,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 78713,N1(C(=O)CCCCCl)CCC2(CCCC2N2CCCC(c3ccccc3)C2)CC1 78714,CC1CCN(C(=O)CC2CCOC2=O)CC1N(C(=O)C[SH](c1ccccc1)OC)C 78715,C1(CCC)(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CCN(C(c2ocnc2C)=O)CC1 78716,C(c1ccccn1)=C(C)C(=O)NCC(C1CCCC1)NC(C1(C#N)CC=CC1)=O 78717,C(CO)(CCCCNC(=O)C(F)CC1CCCC1)NC(C(c1ccccc1)C)=O 78718,C(c1cccnc1)=C1CCN(C(CN(CCCC=C)C=O)=O)CC1 78719,CC1COC(CO)CN1C(=O)CCN(C(=O)CCC1(C)CC1)C1CC1 78720,C1(C)(NC(c2c(COC)cccn2)=O)CCCN(C(C2CC3CC3C2)=O)C1 78721,Cc1ccc(NC(=O)CO)cc1O.C(CCCN)NC(=O)C=CC(=O)N(C)C 78722,c1(C(=O)OC)coc(=NCC2(N)CS(=O)(=O)C2)[nH]1 78723,C1(OC)CN(C(c2ccn(C3CC3)c2C)=O)C(C)(CNC(=O)Cn2ccnn2)C1 78724,c1(C(N(CC(C)C(=O)NC2CCN(CCF)C2)C)=O)cnn(C)c1Cl 78725,c1(N(C)CC2CN(C(=O)C(C)(O)C3CCC3)C2)cnn(C2CCC2)c1 78726,n1(CCOC)cccc1-c1cncc(NC(=O)CCc2cccc(C)c2)c1 78727,c1(C(=O)NCC2C(CNC(CN(CCOC)C)=O)C2)ccc(O)nn1 78728,c1(OC)ccc(NC(c2ccn(CCNC(c3ncn(C)c3C)=O)c2)=O)cc1 78729,Cc1nc[nH]c1C(=O)NC1(C(=O)NCCN(C)Cc2ccccc2)CC(CO)C1 78730,c1(CCC(=O)NC(CNC(C(C(CC)O)(F)F)=O)C)ccc2cccnc2c1 78731,c1(C(=O)NCCC2CC(NC(C(C)N(C(C)=O)C)=O)C2)nnn2c1CCCC2 78732,C(=O)(C1=COCCC1)N1CCC(F)(CNC(C2(S(C)(=O)=O)CC2)=O)C1 78733,C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N(C(c1ccnc(Br)c1)=O)C2 78734,N12CC3(CCC3)CC1CN1CCOCC(C1)C2=O.C1(C(=O)OC)C2CC3C(C2)C13 78735,C(=O)(CCCCCC(=O)NCC(C)NC(=O)C(C(C)C)c1ccc(F)cc1)OC 78736,N1(C(c2c(CC)nn(C)c2)=O)CC2CC3CC2C1C3NC(c1snc(O)c1Cl)=O 78737,N1(C(CC=C=C)=O)CCC2CN(C(=O)CCSc3ccc(Cl)cc3)CCC2C1 78738,c1(C(N2CC(CCCCNC(C(CCOC)OC)=O)C2)=O)ccc(Cl)c(F)c1 78739,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CCC)=O 78740,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 78741,CC(CCC(=O)N(C1(CC(=O)NCC2CC2)CCC1)C1CCC1)N(C)C1CC1 78742,C(N=c1[nH]c(=NCc2ncc(Br)s2)[nH]c2c1CCCC2)c1ncc(C)cn1 78743,N1(Cc2c(NC(C(CC)N(C)C)=O)cccc2Cl)C(=O)c2ccccc2C1=O 78744,C1(N(C(CCSCCC)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 78745,N1(C(C2CC3(CCC3)C2)C(=O)NCCOCC)CC2CCCCC2(C(=O)OC)C1 78746,C12(NC(Cc3ccn(C)n3)=O)CCCC1N(C(c1cc(F)cnc1O)=O)CCC2 78747,C1(COC)(CNC(=O)CN2CCCCC2=O)CCN(C(=O)Cc2[nH]cnc2C)C1 78748,N1(C(c2cc(CCCO)on2)=O)CC2=C(C1)CN(C(C1(CO)CC3CC3C1)=O)C2 78749,CCCC(C)CC(=O)NC(C1CCN(C(c2c[nH]c(C(=O)OC)c2)=O)CC1)C 78750,c1(C(N2CCN(C(C3CCSC3)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 78751,N1(C(C2CN(CCC)C(=O)C2)=O)C2CCCC1CC(NC(C1(C(C)C)CC1)=O)C2 78752,Cn1c(Cn2ccc3c(NC(=O)CSC4CC4)cccc23)nc2ccccc12 78753,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)NC(C)(C)C)CC2C)=O)cc1C 78754,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(C1COCC(C)O1)=O)OC 78755,C1(NC(c2cccc(CSC)c2)=O)CN(C(c2n[nH]c(C)c2F)=O)CCC12CCC2 78756,c1(CNC(C(C)N(C(CCC(C)C)=O)CCO)=O)cncc(C#N)c1 78757,c1(C(=O)N(CC(CC)NC(c2c(CC)nc(C)o2)=O)CC)cc(NC)nc(Cl)c1 78758,C1(C)(CNC(C(C)=CC2CC2)=O)CCN(C(=O)C=C2CC2)C1 78759,c1(C(N2CCC(C(C)NC(c3c(CCC)nco3)=O)C2)=O)c(C)nnn1CC 78760,N1(C(c2ccc(OC)nc2)=O)CCC2(NC(=O)CNC(N)=O)CC2C1 78761,C1(C)(C(=O)NCC(C(=O)Nc2cnc(C)nc2)N(C)C)CCCN(C)C1 78762,CC(CS(C)=O)C(=O)NC1COCCN(C(c2c[nH]cc2-c2ccccc2)=O)C1 78763,N1(C(C(C2(O)CCC2)NC(CC(=O)NCC)=O)=O)CC(C#N)C2(CCC2)C1 78764,C1(NC(C(c2cccc(F)c2)C)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1 78765,C1(CC(=O)N(CCC(=O)NC(C)C2CC2)C2CC2)COCC1O 78766,N1(C(CCC(C)SC)=O)CCCC(NC(=O)C=Cc2cnn(C)c2)CC1 78767,C1(CC)(CC)CC(NC(C2CCCC2CNC(=O)CC(=O)OC)=O)C1 78768,c1(NC(c2cccc(OCC=C)c2)=O)cccc2c1NC(C)CC(=O)N2 78769,c1(CNC2CC(NC(c3c(N)ccc(C(F)(F)F)c3)=O)C2)ccc2ncnn2c1 78770,C1(NC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CC1c1cccc(F)c1 78771,Cn1cc(S(=O)(=O)NC2CC(CO)(CO)C3CC23)nn1 78772,c1(C(=O)NC(CC)CNC(=O)COCCC(C)C)ccc(O)nc1Cl 78773,C(CNC(=O)CC(C)Cn1cccn1)(C(C)(C)C)NC(C[SH](CC=C)C)=O 78774,N1(C(CC2CCN(C)CC2)=O)CC2CC(C(=O)N(C)OCc3ccccc3)(C2)C1 78775,N1(C(C2C(c3c(C)n(C)nc3)C2)=O)CC(NC(=O)C(C)C(C)C)CC(F)C1 78776,CON1CCC(C(=O)NC2(CNC(=O)CC3CCCCC3O)CCC2)CC1 78777,CC1CC(=O)CCC1C(=O)NOC(C[N+](=O)[O-])NC(N1CC(C(=O)OC2CC2)C1)=O 78778,N1(C(C2C(C)(C)COC2)=O)CC2(C1)CN(C(=O)CNC=O)Cc1ccccc1O2 78779,N1(C(C(CCC)Cl)=O)C2CCC(C2)C1C(N1CCC(C)(CO)C1)=O 78780,C(=O)(C(C(C)C)OC)NCC(CC)(C)NC(=O)CSCCN(C)C 78781,C1(NC(CC(C)C(F)F)=O)CC2CC(C1)N(C(c1ccc(N)c(F)c1)=O)C2 78782,C(=O)(C#CC(=O)N(C)C)NC1CC(NC(c2c(SC)occ2)=O)C1 78783,Cc1ncnc(O)c1C(=O)NC(C1(O)CCN(C(=O)C(C)(C)CF)CC1)C 78784,c12cn(nn1)CCNC2=O.c1(C(=O)OC(C)(C)C)csc(Cl)c1 78785,CC1(CC(N2CC3CC3C2C(=O)NCC2C3COCC23)=O)CCCCC1 78786,Cc1nc(C)n(O)c1C(=O)NC(C)(CNC(=O)Cn1ccc([N+](=O)[O-])n1)C(C)C 78787,N1(C(C=C(C)CN2CCCC2=O)=O)C2CCC1CN(C(c1cncn1C)=O)CC2 78788,C1(C(=O)NCC2(F)CCN(C(C(C=C)O)=O)C2)(OC)CCCCCC1 78789,C(=O)(CCC(F)(F)F)N1C(C)(CC(=O)NC(C(=O)OCC)C)CC1 78790,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCCC2(NC(C3CCC3)=O)CC2C1 78791,C1(NC(C2CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)CCc1ccc(Cl)c(F)c1)C2 78792,CC1(C(=O)NCC2CCC(NC(=O)CC(=O)NCC3CC3)CC2)CC2C=CC1C2 78793,c1(C(=O)NCC2C(NC(COCCC)=O)CCC2)ccn2c1CCCC2 78794,C12(CNC(C(C=C)(C)C)=O)COCCN1C(=O)CN(C(C1(CC)COC1)=O)C2 78795,c1(OCCCC)ccc(C(=O)NCC(C2CC2)NC(C2CC(C)(C)C2)=O)c(Cl)c1 78796,c1(C2C(C(N(CCC(=O)NC(c3nc[nH]n3)C)C3CC3)=O)C2)ccccn1 78797,C1(C(=O)NCc2ccc(F)cn2)CC(O)CN1C(C1CC=CCO1)=O 78798,c1(C(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)OC)c(F)cccc1F 78799,CCC(C)(C)CCCC(=O)NCC1=CCN(C(=O)CSCC(F)F)CC1 78800,c1(OC)cc(C(=O)NC2CCC2NC(=O)Cn2ncnn2)sn1 78801,Cc1cc(SC(C)(C)C)cc(O)c1F.n12cc(nn1)CC(C)C(=O)NCC2 78802,CC#CCCCC(=O)N1CCC(O)(C(C)NC(=O)Cc2ccc(Cl)cc2)CC1 78803,Cc1nn(C)c(N2CCN(C)CC2)c1CNC(C1CC12CC2(F)F)=O 78804,C(=O)(C(O)CC(F)(F)F)N(C(CC)Cc1ccccc1)CC 78805,c1(C(=O)NC(C(C)NC(C(C)OCCCC)=O)CO)nc(C2CC2)ncc1Cl 78806,C1(C(=O)NC(C2(O)CN(C(=O)C(O)Cc3cnc[nH]3)C2)C)C2CC(=O)CC12 78807,C1(C(N(CCCNC(=O)C2=CCCCC2)C2CC2)=O)CCCC2CCCN12 78808,c1(SC)cc(C(=O)NC2CCCCC2NC(c2n[nH]c(C)c2Cl)=O)c(C)o1 78809,C1(COC)CN(C(=O)CCc2ccsc2)CCN1C(C1COC(=O)N1)=O 78810,N1(C(c2n(CC)nnc2)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC12CCOC2 78811,N1(C(c2ccc(C)cc2)=O)CCCC(C)(C)C1CNC(c1c[nH]c(C#N)c1)=O 78812,c1(C(=O)NC2(CNC(c3cnc[nH]3)=O)C(C)CCCC2)ccc2nn(C)cc2c1 78813,c1(CCC(N2CCC(OCCNC(=O)Cc3nncs3)C2)=O)ccc(Cl)c(Cl)c1 78814,c1(C(C)C(=O)NC2C3CC(NC(=O)C(C)O)CC23)n[nH]c2c1CCCC2 78815,C12(NC(C3C4(CC(NC(Cc5c(C)nn(C)c5)=O)C4)C3)=O)CC1COC2(C)C 78816,c1(C(=O)OC)cccc(C(N(CCCCNC(=O)C(=O)NC2CC2)C)=O)n1 78817,Cc1c(C(=O)NC2CC(OC(C)(C)C)C2)ccn1CCO.c1(N)ccn(C(F)(F)F)n1 78818,c1(NC(CCCCCn2cc(C3COCC3O)nn2)=O)ccc2c(c1)OCCO2 78819,c1(COC)cc(C(=O)N(C2(CN3CCNCC3)CC2)C)nn1CCO 78820,c1(CC)c(C(=O)NCC2C3CN(C(=O)CCSC(F)(F)F)CC23)oc2ccccc12 78821,C1(NC(C(=O)NCC)=O)(CNC(=O)CC2CC(OC)C2)CCCCC1C 78822,C1(NC(c2cc(Cl)cc(F)c2F)=O)CN(C(C2(O)CCOC2)=O)CC2(CC2)C1 78823,c1(C(=O)NCC2CC(NC(C3N(CC)CCCC3)=O)C2)ccnc2c1nnn2C 78824,N1(C(c2c(C3(C)CC3)noc2)=O)CC2(CCC(CNC(=O)CCCCC(N)=O)O2)C1 78825,N1(C(C(CC)COC)=O)Cc2ccc(C(C)NC(C3CCCCCC3)=O)cc2C1 78826,c1(C(=O)NCC2C3CN(C(C(CC(N)=O)O)=O)CC32)cccc2nc(O)[nH]c12 78827,Cc1ccc(O)cc1CNC(C1CCC(C(N2CCCC(C)C2C)=O)CC1)=O 78828,N1(C(C2C(CC)OCC2)=O)C2CCCC1CC(CNC(C1(Cl)CC1)=O)C2 78829,C1(O)(CN(C(c2c(C)oc(C3CCC3)n2)=O)C)CCCN(C(=O)CCC2CC2)C1 78830,C(C)(C)(CC(=O)NC1CCCN(C(C2COCC2c2ccc(F)cc2)=O)C1)OC 78831,N1(C(C(CNC)c2ccccc2)=O)CCCC(N(C(c2c[nH]nc2C)=O)CC)C1 78832,C1(NC(CC=CCC)=O)CCC2(CCCN(C(c3cnc4n3CCC4)=O)C2)C1 78833,c1(CCC(=O)NCCC2(CCNC(C(C)N(CC)CC)=O)CC2)cccnc1F 78834,c1(CN2CC(NC(c3cncc(C)c3)=O)CC(F)(F)C2)ncc(Br)cc1[N+](=O)[O-] 78835,C12(NC(C(C)CN(C)C)=O)CCCC1(F)CN(C(c1ccc3c(c1)OCC3)=O)C2 78836,c1(C(=O)NC2(C3CN(C(CC(C)F)=O)C3)CC2)cccn2cnnc12 78837,C#CC1(C(=O)N(C)CC2(C)CCCO2)CN(C(=O)C(O)CN(C)C)C1 78838,O=C1CC2(CCN(C(C3CN(C(=O)CCSc4ccccn4)CCS3)=O)CC2)C1 78839,CN1C(=O)CN(C(C2CCCCN(C(c3cc(C#N)ccc3N)=O)C2)=O)CC1=O 78840,N1(C(C2N(C)CC2)=O)CCC(C(=O)NOCCN2CCCC2)C1(C)C 78841,N1(C(C(C=C)C)=O)CC2(C=C(C(=O)Nc3cccc(SC)c3)CO2)C1 78842,C1(COC)(NC(c2c[nH]c(Br)c2)=O)CN(C(=O)C(c2ccccc2)F)C1 78843,CC(C)(C(=O)NCC1(O)CCN(C(c2ccccc2O)=O)CC1)C(N)=O 78844,c1(CC(=O)NC2CN(C(C=CC)=O)C2)c(C)nc(-c2ccccc2)nc1O 78845,N(C)(S(=O)(=O)N(C)C)CC(=O)NCCCCC1CCCN(C(C(C)C2CC2)=O)C1 78846,C(CC(C)C)(C(=O)NC1CC(C)N(C(=O)C(C2CCCCC2)O)C1)OC 78847,C(=O)(CCC(C)NC(c1cnnn1CC)=O)NCCOCC=C 78848,CC1OCCC1CNC(=O)N(C1(CO)CC1c1ccccc1)C 78849,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(=O)COCC1CCC1 78850,C1(CC)C(NC(=O)Cc2ccccc2O)CCCN1C(=O)Cc1cccs1 78851,c1(SCC(N2CCCC2Cn2cc(C(=O)O)cn2)=O)ccccc1Cl 78852,c1(CCC(N2CCC(O)(CCNC(C(CC)(C)O)=O)C2)=O)c(Cl)cncc1Cl 78853,C1(OCC(=O)N(C2CCN(C(=O)COCc3nccn3C)C2)CC)CCOCC1 78854,C1(C(=O)NCCC(C)NC(c2cccc(C(N)=O)n2)=O)CC2C(C1)C2(C)C 78855,c1(CN2CCCC(N3CCC(N(C)C)C3)CC2)nc(=N)c(C#N)c[nH]1 78856,C1(CC(=O)NCC(C)NC(c2ccccc2-c2cccs2)=O)CC2(C1)CC21CC1 78857,C12(C(=O)OC)CC(NC(=O)C(F)(F)F)(CN1C(=O)CNC1(CCF)CC1)C2 78858,CC1=C(C(=O)NCCc2nn(C)cc2Cl)C(C)(C)CCC1 78859,c1(OC(C(=O)NCC(C(C)C)NC(c2cn(CC=C)nc2)=O)C)cccc(F)c1 78860,N1(C(CCNC(=O)C=CCl)=O)CCC2(CC(NC(C3CCCCC3(F)F)=O)C2)C1 78861,C(=O)(CCC(C)(C)F)NC(C1CCN(C(=O)Cc2ccn(C)n2)C1)C 78862,N(C(=NCCCN1CCOCC1)NCc1cc(C2CC2)on1)CC1CCCC(O)C1 78863,c1(NC(c2ccc3nc[nH]c3c2)=O)ncnc2cccc(F)c12 78864,C(N=c1[nH]c(=NCCc2ncc[nH]2)[nH]c2c1CCCC2)c1c2cccc(F)c2sc1 78865,C=CCC(C(=O)NC(CCC)C(O)C(=O)N(CCCO)CCO)C(C)C 78866,c1(-c2ccc(CN3C(C(=O)OC)CC(O)C3)s2)cccn(CO)c1=O 78867,C(N=c1ccnc(NCC(C)C(F)(F)F)[nH]1)C1(C=C)CCOCC1 78868,C1(NC(C(CC)C(C)C)=O)CCOC2(CCC2)C1 78869,N1(C(CC(C)n2cccn2)=O)CCCC(CCC(=O)NCCOc2ccco2)C1 78870,c1(C(N(CCC(C)(C)NC(C(CC)C(C)C)=O)C)=O)c[nH]c2cc(OC)ccc12 78871,N1(C(C2(c3cc(C)no3)CCC2)=O)C(CNC(=O)C(C)NC(N)=O)CC2COCC12 78872,C1(C(=O)NC(c2ccc(O)cc2)C)CCN(C(=O)c2cc(O)cc(=O)o2)O1 78873,C1(C2CN(C(=O)CCCCOC)C2)(NC(c2ccc(CC)o2)=O)CC1 78874,C1(C(=O)NCC2CCN2C(=O)CCc2cc(F)ccc2F)Cc2cccnc2C1 78875,N1(C(CC2ON=C(C)C2)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(F)C1 78876,CC1CN(C(c2cc(CCO)on2)=O)CCC1NC(c1csc(C(C)N)n1)=O 78877,CCN=c1cc(C(N2CCC3(NC(c4nc(OC)c(C)s4)=O)CC3C2)=O)cc[nH]1 78878,c1(C(N2C(CNC(Cc3c(CC)cccc3)=O)CC2)=O)cnc2c(c1)COCC2 78879,C1(OCC)(CNCC2(CF)CCC2)CCOCC1 78880,CC(CSC#N)C(=O)NCC1C(CNC(=O)C(F)CC2CCOC2)C1(F)F 78881,Cc1cnccc1C(C)NC(C1(C(C)NC(=O)CC(C)n2cccn2)CC1)=O 78882,CC(CC(C)(F)F)C(=O)N(C1CCCCCC1)CCNC(c1nnn(C)c1N)=O 78883,C1(C(N2CCCC(C(=O)NCC3N(CC)CCC3)C2)=O)CCCCC(C)O1 78884,S(=O)(=O)(C1CC2(CC2CC(=O)O)C1)N(C(CCC)=O)CC1CC1 78885,C=C(C)CCC(=O)N1CCC(CNC(c2c[nH]nc2-c2cccnc2)=O)C1 78886,c1(C(=O)O)cc(CN2CCC(n3cc(CO)nn3)C2)c[nH]1 78887,c1(C(=O)NC2CCCC(NC(c3c(CC)c[nH]c3)=O)C2)nncc2c1CCCC2 78888,N1(c2cnc(-c3c(C)cccc3)s2)CCC2(CC1)CC2C(=O)N(C)C 78889,c1(OC)cc(CO)ccc1C(=O)NC1C2CC1N(C(=O)C(=Cc1ccco1)C)C2 78890,Cc1cc(N2CC(NC(C3CCC(=O)N3C(C)C)=O)CCC2C)ccc1Cl 78891,N1(C(C2CCN(C)C2)=O)CCC(C)(NC(=O)CSC(F)F)C1 78892,c1(C(=O)OC)cc(C(=O)NC(CNC(C2CNC(=O)N2)=O)C(C)C)c(C)o1 78893,Cc1cc(=O)n(C)cc1C(=O)NCC1(F)CCCN(C(=O)CC2C=CCCC2)C1 78894,N1(C(CN(c2ncccc2Cl)C(C)=O)=O)CCCC(C)(C(=O)O)C1 78895,N1(C(C(CC)=CC)=O)CCC2(CCCCN(C(=O)CCc3ccc(O)nc3)C2)C1 78896,c1(OC)ccc(C(N2CCOC(CN(C(=O)C(n3ccc(C)n3)C)C)C2)=O)nc1 78897,C1(CNC(C2(C(C)(C)C)CCCC2)=O)CCCCN1C(c1nn[nH]c1Cl)=O 78898,C1(C(=O)NCCCNC(CCCCNC(C)=O)=O)CCC2CC2CC1 78899,c1(N2CCCC(N(SC(F)(F)F)C)C2)nc2cc[nH]c2c(=NCC2CCCO2)[nH]1 78900,N1(C(C=CCC)=O)C2CCCC1CC(NC(=O)C=C1CCC(C)CC1)C2 78901,c1(C(=O)OCC)c(NCC2CC(C3CC3)C2)cc(C(=O)O)cc1I 78902,C(C1CN(C(=O)COC2(C)CCOCC2)Cc2ccccc21)NC(C(C)(C)CF)=O 78903,C1(CC(=O)NC2CCCCC2NC(C2(SC)CC2)=O)(C(=O)NC)CCOCC1 78904,c1(OC(C)=O)ccc(C=O)cc1C(=O)OC(C)=O.c1(SC)ccc(NC(C)(C)C)s1 78905,C1(CC=C)(C(N2CC(NC(=O)C(=O)NC3CC3)C2)=O)CC=CC1 78906,Cc1cnc(C)c(C(=O)NCC2CCCN2C(C2CCC(C(N)=O)O2)=O)c1 78907,C(=O)(C(O)C(C)(C)CC)NC(CNC(c1cc(C(C)(F)F)n[nH]1)=O)C1CC1 78908,CCC(O)C(C)(C)C(=O)N1CCC(C(F)C(=O)N(C2CC3(CCC3)C2)C)C1 78909,Cc1cccc(CC(N2CCC(C)(c3cn(CC4CCOC4)nn3)C2)=O)n1 78910,c1(CC(N2CC3C(CNC(C4C(C)C4)=O)C3C2)=O)cc2ccccc2s1 78911,C(=O)(C(F)(F)C(F)(F)F)N1CCN(C(C2CCN(CC(C)C)C(=O)C2)=O)CC1 78912,c1(NC(C(C)C)CNC(C2CCCNS2(=O)=O)=O)ncnn2cccc12 78913,Cn1cc(NC(=O)Cn2cc(Cl)ccc2=O)ccc1=O 78914,C1(NC(C(COCC)C)=O)C2CC3C1C3C2C(=O)NC1CCC(SC)C1 78915,C(=O)(CCCCC(=O)Nc1ccccc1)NC(N1CC(CNc2nccn2C)C1)C 78916,C(CC(=O)N=c1cc2ccccn2[nH]1)NC(C1(F)C(C)OCC1)=O 78917,Cc1ccc2c(C(=O)NC(C3(O)CN(C(c4scc(C)c4Cl)=O)C3)C)n[nH]c2c1 78918,CC(CCF)NC(=O)CN(C(=O)CC1CCSC1)CC1CC1 78919,c1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)C#N)C2)cccc2ccncc12 78920,C#CCC(O)C(=O)NCCC(O)CNC(=O)Cc1ccc(OCC(N)=O)cc1 78921,c1(CCC(=O)N(CCCN(C(C=CSC)=O)C)C)ccc([N+](=O)[O-])cc1 78922,C(=O)(C1CCCc2nc[nH]c21)NC1C(NC(=O)Cc2cscn2)CCC1 78923,Cc1nn2cccnc2c1C(=O)NCCCCNC(=O)COC1CCCCC1C 78924,Cn1ncc(C(=O)NCC2(NC(C3CCC(F)CC3)=O)CCC2)c1Cl 78925,C(=O)(C(C)CCC(C)(C)C)NC1C(OC)CN(C(=O)Cc2csc(Cl)n2)C1 78926,N1(C(c2c(C)cnn2C)C(=O)NC2CCC2)CCC(C(F)(F)F)C(F)C1 78927,C=CCN=C(NCc1cc(Cc2ccccc2)no1)NC1CC(C)N(CC)C1 78928,Cc1cncc(CCC(=O)N(C(C)CN(C(=O)Cn2nnc(C3CC3)n2)C)C)c1 78929,C1(C(=O)OC)Cc2c(Br)cccc2CN1C(=O)NCC(=O)CC1CC1 78930,Cc1cc(CCC(=O)NC(C)C(C)NC(=O)CCc2cscn2)n[nH]1 78931,S(=O)(=O)(c1cc(C(N2CCCN(C(=O)C=CCF)C(C)C2)=O)cc(C)c1C)NC 78932,CCCCC(O)C(=O)NCC(CC(F)(F)F)NC(c1cc(Cl)ccc1CC)=O 78933,C1(C(=O)NCC2N(C(C(C)=CC3CC3)=O)CCC2C)CC(C)(C)CCO1 78934,c1(C(=O)NC2CCC(NC(C3CCC(C)C3)=O)CC2)cnn2c1N(C)CC2 78935,C12(NC(=O)CSC3CC3)CN(C(c3cc[nH]c3)=O)CC1CS(=O)(=O)C2 78936,C(=O)(CC(O)CCCC)NCC1N(C)CCN(C(C=CC)=O)C1 78937,c1(C(N(C2CN(C(c3cc4occc4[nH]3)=O)CC2O)C)=O)cn2ccccc2n1 78938,C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NCCc2ncn(C)n2)CC(C)(C)C1 78939,C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(CC)C1CC1 78940,c1(CC(C(=O)NCC(CC(C)O)C)(C)C)ccnc2ccccc12 78941,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C 78942,C1(CC)CN(C(C2CCOC2c2cnn(C)c2)=O)CCN1C(=O)C=CBr 78943,C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NC2(c3c(C)cccc3)CC2)CCCC1 78944,C=CC1CN(C(c2cn(C)ccc2=O)=O)CC1NC(c1conc1C(C)C)=O 78945,c1(CC(=O)NC2CCCCN(C(=O)C=C(Cl)Cl)C2)noc2ccc(F)cc12 78946,C1(C(=O)NC2CC(CNC(c3ccccc3C(N)=O)=O)C2)(OC)CCCC(C)C1 78947,N1(C(Cc2c(C)nsc2)=O)CC2CCCC1C2CNC(C1CC1Br)=O 78948,C1(NC(c2c(C)c[nH]n2)=O)C2CC3CN(C(c4cnc5sc(C)cn45)=O)C1C3C2 78949,N1(C(CC2CC(CC)OCC2)=O)CCCN(C(c2cnsn2)=O)CCC1 78950,C(C1c2ccsc2CCN1C(=O)C(O)CC1CCCCC1)NC(CCC=C=C)=O 78951,c1(OC)ccc(S(=O)(=O)N(C)C)cc1NC(c1csc(C(C)C)n1)C(=O)O 78952,Cc1cc(C(=O)NC23CC2CN(C(c2coc(CC4CC4)n2)=O)C3)nc(Cl)c1 78953,C1(CC(C)C)CN(C(C2(CCNC(=O)CC3COCCN3C)CC2)=O)CCO1 78954,N1(C(c2cc(C)c(F)cc2)=O)CCC(CCNC(=O)CC2C=CCC2)C(F)(F)C1 78955,CC1(CNC(C2CCCC(c3ccccc3)O2)=O)CCCN1C(=O)CS(N)(=O)=O 78956,Cn1nnc2cc(C(=O)NC3(C)CC(NC(=O)C(CO)OC(N)=O)C3)ccc12 78957,C1(NC(Cc2nnc(C)s2)=O)CCN(C(c2c[nH]c(=N)s2)=O)CC1CN(C)C 78958,C(=O)(CC1CCc2ccccc21)OC.C12(CC3CNCCO3)CCCN1CCC2 78959,C1(CN(C2CCCOC2)C(c2n(C)c(-c3ccco3)nn2)=O)CN2CCN1CC2 78960,C(C(=O)NCCN(C(=O)Cc1ccnc(Br)c1)C)(C(C)(C)C)N(C)C 78961,c1(OCC(=O)NC(C)(C)CNC(=O)C(C)(C)CCC#N)ccc2ccoc2c1 78962,CCC(CCC(=O)NCC1CC(CC(=O)NCCC2OCCC2(C)C)C1)OC 78963,c12n[nH]c3c(cccc13)C(=O)NC2.C1(C)(SC)CCC(N)C1.C(=O)O 78964,c1(N2CCCC(C=C)C2)nc2ccc(S(=O)(=O)NC3CC3CCC)cc2s1 78965,C1(COC)CCCCC1C(=O)NC1(CC(=O)NCc2ccc[n+]([O-])c2)CCCC1 78966,N1(C(c2ccc(C)cc2F)=O)CC2CCC(CNC(C3C4CC5C(C4)C35)=O)(C2)C1 78967,c1(C(N2CCN(C(C(C)OC)=O)CC23CC3)=O)cc2c(O)ccc(F)c2[nH]1 78968,c1(NCc2ccc(C)nc2C#N)c(I)cc2ccccc2c1C 78969,c1(-c2ccc(OC)cc2)n[nH]c(=NC2CCC2C)c2ccccc12 78970,C1(C(=O)NCC2(F)CCN(C(C=C(C)Cl)=O)CC2)CC(C)(C)OC(C)(C)C1 78971,C1(C(N2CCC(NC(=O)Cn3nnc(C4CC4)n3)CC2)=O)OC2CCC1CC2 78972,c1(C(N(C)CC2CCCN(C(CCN(C(C)=O)C)=O)C2)=O)ccn2ccnc2n1 78973,N1C(=NCc2ccc(NS(C)(=O)=O)cc2)NC(C)C2CCOC1C2.C(CO)SC 78974,c1(C(=O)NC2CC(CCNC(C(CCOC)OC)=O)C2)ccnc(C)c1N 78975,c1(C(N2C(COCC)CCCC2)C(=O)NCCCSC)cc2c(cn1)OCCO2 78976,Cn1cc(C(=O)NC2COCC2NS(C)(=O)=O)c(NC(=O)Cc2ccc(Cl)s2)n1 78977,N1(C(C=COCC)=O)CC(C)CCC1CNC(c1ccc(N(C)C)cc1)=O 78978,Cc1cc(C(=O)N(CCC(=O)NC(C2CCC(C)(C)O2)C)C(C)C)cn1C 78979,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1cscn1)C2 78980,Cc1cc(=NC(CCO)C2CCSCC2)[nH]c(=NCc2cccc(CO)c2)[nH]1 78981,C1(NC(CNC(CC)=O)=O)(CF)CCN(C(=O)C=C2CCC2)C1 78982,c1(C(=O)NCC2C(NC(c3c(SC)ccs3)=O)COC2)ccc(F)c(C)c1C 78983,C=CC(C)(CC)C(=O)NC(C)CC(=O)Nc1cnc(N(C)C)nc1 78984,N1(C(c2cn(CCC)nc2)=O)CCC2(C)CN(C(=O)CC3CNC(=O)C3)CC12 78985,C1(C(=O)OCC)CCCCC1NC(=O)CC1(C)CN(Cc2ccsc2Cl)C1 78986,Cc1c(CNC(=O)C(=O)NC2CCN(Cc3ccccc3)C2)cccc1O 78987,c1(C(=O)NCCCNC(C(CC2CCCCC2)OC)=O)c([N+](=O)[O-])c(C)nn1C 78988,n1(CCOC)nc(-c2ncccc2OCC(F)(F)F)nc1C(C)C(C)F 78989,c1(CC)cccc(CC)c1C(=O)NC1CCN(Cc2cnc(Cl)s2)CC1F 78990,c1(C(N2CCC(CC=C)(NC(=O)CSC3CCCCO3)C2)=O)c(F)cncc1Cl 78991,c1(C(=O)NC2C(CC)N(C(c3nccnc3N)=O)CC2)cc(=O)cc(Cl)[nH]1 78992,C=C(C)CCCC(=O)NCC1CCCN1C(=O)CN1CCOCC1 78993,N1(C(C2N(CC)CC2)=O)CC(CO)C2(C1)CN(C(=O)C(O)Cc1ccccn1)C2 78994,N1(C(C=C2CCC(C)C2)=O)CC2CC(NC(c3ccnc4[nH]ncc34)=O)CC1C2 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79169,Cc1ncc(Cl)cc1C(=O)N(C)CCN(C)C(c1cccc(F)c1F)=O 79170,c1(C(=O)NC2CC(C)(C(=O)NCC)C2)cc(OC)ccn1 79171,N1(C(C(C)C)=O)CCOC(CN(C)C(c2ncsc2Br)=O)C1 79172,C1(CC(=O)N(c2ccn(CCF)n2)CC)(CC=O)CCCN1C(=O)C(C)C 79173,CC1=C(C(=O)N2CCC(NC(=O)CN3CCNC(=O)C3)C23CC3)CCO1 79174,c1(C(C)C)ccc(O)c(C(=O)NCCCNC(c2cc(F)ccc2Cl)=O)c1 79175,CC1(CNC(c2ccsc2Cl)=O)CCN(C(c2cnc(Br)s2)=O)C1 79176,C1(OC)CN2CCC2(C(N2CC(CN(C)C(C3CCCCN3C)=O)C2)=O)C1 79177,N1(C(=O)CCc2ccc(Cl)cc2)CCC2C1CCCN2C(=O)CC1CCCC1 79178,Cc1cccc(C)c1C(C1CC1)NC(=O)C=CC(C)(C)NC(=O)CC(C)(C)C#N 79179,N1(C(C(C(C)(C)C)NC(c2c(C)c(F)ccc2)=O)=O)CCC2CCCCC12 79180,C(=O)(C(C(C)(C)C)NC(=O)C(C)=C(C)C)N1CCC(CC)CC1 79181,N1(C(C=CCCC)=O)CCC2CCN(C(=O)CCc3cnc[nH]3)C2C1 79182,C12CC(C13CCC3)NC2=O.c1(C(N(C)CCN(C)C)=O)n[nH]c2c1COC2 79183,c1(NC(C2CCCN2C(c2cnc3ccc(Br)cn23)=O)=O)cc([N+](=O)[O-])cnc1Cl 79184,c1(CC)ncc(C(=O)NCCC2CCCCN2C(C2CN(C)CCO2)=O)c(O)n1 79185,C1(NC(C(CCC)(C)C)=O)CN(C(=O)Cc2cnc(C)o2)C2(CCCCC2)C1 79186,C1(NC(C2(C)COC2)=O)CN(Cc2ccc(-c3ccccc3)cc2)CC1F 79187,C1(C(N(C2CCCC2)CCCC)=O)CCC(C(C)C)N1C(=O)CNC=O 79188,C(=O)(CCC(C)(C)OC(C(CC#C)CCC)=O)NCCN(C)CCC 79189,c1(C(=O)NCCCCCCN(C(C(CC)N(C)C)=O)C)cc(OC)nc(Cl)c1 79190,N1(C(CCC=CC)=O)CC2(CCOCC2)CC1CNC(c1cc2occc2[nH]1)=O 79191,C1(N(C)C(=O)C2CC2)CN(C(=O)C=CC(=O)NCC2CC2)C2(CCCC2)C1 79192,C(C)(C)(C(C)(C)O)N(C(C(CC)N(C)C(C1CCCO1)=O)=O)C1CC1 79193,N1(C(C2(COC)CCOCC2)=O)CCOC(C)(CNC(=O)Cc2cc(C)no2)C1 79194,Cc1cc(C)nc(CCN2CCC(C)C(C(=O)ON3CC(C)CC(O)C3)C2)n1 79195,c1(C(=O)NC(CC(C)NC(CNC(C(CC)C)=O)=O)C)sc(CC2CC2)nc1C 79196,N1(C(COCCC(C)C)=O)CC=CC1CNC(c1cnn(C)c1)=O 79197,c1(C(=O)NC2CCCN(C(C(C=C=C)C)=O)C2)ccc2c(c1)NC(=O)CC2 79198,N1(C(c2c(C)nc(CO)s2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 79199,c1(OC)cc(C(=O)NC2CC2CNC(c2c[nH]c(=N)s2)=O)cc([N+](=O)[O-])c1C 79200,c1(CNC(=O)C(c2c(C)[nH]c(-c3ccccc3)c2C)ON)ccc2cccc(Br)c2n1 79201,C1(NC(CCN(CC)CC)=O)COC2CN(C(c3cccc4nc[nH]c34)=O)CC12 79202,c1(C(=O)NCC(C)NC(c2ccc(O)c(F)c2)=O)c([N+](=O)[O-])cnn1CC(F)F 79203,C1(CC)C(NC(c2cccn(C)c2=O)=O)CCCN1C(c1cccc(CO)c1)=O 79204,C1(NC(CCC(=O)NC)=O)CCCC2CN(C(=O)C=Cc3ncccc3C)CC12 79205,N1(C(C#CC(C)(C)C)=O)CCOC2(CCCN(C(C3(C)CCCC3(F)F)=O)C2)C1 79206,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC2C(NC(c3cc(COC)on3)=O)C2C1 79207,c1(OCC)cccc(C(=O)NC2(C)CCN(C(c3cnoc3C3CC3)=O)C2)c1 79208,CC(C)C(N=[N+]=[N-])C(=O)NC1CC(=O)NC1c1nccn1C 79209,c1(OC)ccc(C(N2CCCC2C2CCN(C(C3(N(C)C)CC3)=O)C2)=O)c(Cl)c1 79210,c1(C(=O)OC)cncc(C(N2CCN(C(C3CCCNCC3)=O)CC2)=O)n1 79211,C1(C(N2CCC(C(CNC(CN(C)CC)=O)(C)O)CC2)=O)CCn2ccnc2C1 79212,CCC(CCN1CCCC1=O)N1CCCC1 79213,C1(NC(c2cc(C)sn2)=O)CN(C(c2ccc(N)cc2O)=O)CCC1C 79214,C1(NC(C2(COCC)CC2)=O)CCOCC1NC(c1ccc(Cl)o1)=O 79215,N1(C(c2onc(CC)c2C)=O)CCC2CCC(C1)N2C(=O)CC1=CSCCC1OC 79216,CCCCC(O)C(=O)NCC(C(=O)NCC1CCCN1C)C(C)C 79217,N1(CC(C)CNC(=O)CCCn2cc(C3CC3)nn2)CCCC(C(=O)O)(CO)C1 79218,N12CC3COCCC3(C1)NC(=O)C1CN(CCC2=O)C1.N(C)(C)CC 79219,Cc1ccc(C(=O)NCCC(C)N(C)C(C2CCS(=O)(=O)N2)=O)c(Cl)c1 79220,c1(N(C)CC2CC23CCC(O)CC3)nc(=NCc2ncccc2Cl)[nH]c2c1COC2 79221,CCCCCC(O)C(=O)N1CCN(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CC(C)C1 79222,c1(N)cccc(S(C)=O)c1.c1(-c2n(CCCC)nnn2)cc(C)c(O)cc1C 79223,S(=O)(=O)(c1cc(F)cc(Br)c1)N1C(C)CC(F)(F)C1.c12cc(ncn1)N2 79224,O(C1CCCc2ccccc21)CC(N1CC(NC(=O)C=CCO)C(C(F)(F)F)C1)=O 79225,c1(C(=O)NCC#CCNC(C(C)=C(CC)C)=O)ccc(NC(=O)NC)cc1Cl 79226,C12C(C3CC3)CCN1C2=O.C1(NC(CN(c2ccccc2)C)=O)C(C)(C)C1(C)C 79227,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CC#C)CCOC)CCF 79228,c1(C(C(C)NC(=O)CCc2ccon2)NC(c2coc(Cl)c2)=O)ccccc1F 79229,C1(NC(CCNC(=O)NC)=O)CN(C(=O)CC2CCC(C)(C)C2)C2CCCCC12 79230,C1(CCNC(C2C(c3ccccc3)(C)C2)=O)CSCCN1C(C1CC(F)(CO)C1)=O 79231,C(N=c1[nH]c2c(c(=NCc3cccc(C(F)F)c3)[nH]1)CCC2)c1c(CC)nns1 79232,C(CCN=c1[nH]c2c(c(=NCCOCCCF)[nH]1)CSC2)c1n[nH]c(=N)s1 79233,C#CC1(C(N2CCN(C)C(C)C2)=O)CCN(C(=O)OC(C)(C)C)C1 79234,C1(NC(CN(c2ccncc2)C)=O)CN(C(C2CCOC2C2CC2)=O)CC12CC2 79235,CCC(CC)C(F)C(=O)NCC1C=CC(NC(c2sccc2C#N)=O)C1 79236,C1(C(C2CC2)NC(COCC(C)C)=O)CN(C(C)=O)C1 79237,CCC(CNC(=O)C(O)CCCNC(C1CCC(=O)CC1)=O)(CC)C(N)=O 79238,CCCCC(CC(=O)N1CCC(F)C(F)C1)NC(C1CC2(CCC2O)C1)=O 79239,c1(C(N(C)CC2(CNC(=O)Cn3ncccc3=O)CC2)=O)cc2scnc2[nH]1 79240,c1(C(N(C(C)C)CCNC(c2cnn(C3CC3)c2Cl)=O)=O)cc(F)c(F)cc1Cl 79241,C1(C(C)NC(C)C(=O)NCCCC)CCCCN1C(=O)Cc1cccc(OC)c1 79242,C1(NC(c2cn(CCC3CC3)nn2)=O)COCCN(C(=O)CC23CCCC2C3)C1 79243,C(=O)(CC(F)(F)F)NC(C)C(=O)NC(C)CN(C)C(C1CC1(F)F)=O 79244,CN1CCC(CC(=O)N2CCC(c3ccc4c(c3)CCC4=O)C2)c2ccccc21 79245,c1(CN(C(=O)CC2CCCC2O)CCNC(c2cnn(CC)n2)=O)ccc(F)cc1 79246,C1(F)(CNC(c2cnc(S)[nH]2)=O)CCC(CNC(=O)C(O)C2CCC2)CC1 79247,C(CCF)(C(=O)N(C(CO)C1CC1)C)NC(C1CCC(C)O1)=O 79248,c1(OC)cc(N)c(C(N2CCCC(CNC(C3C(C)C3C)=O)C2)=O)c(F)c1 79249,c1(NC(C)C)ccc(C(=O)NCC2(NC(C3C(C)CC3C)=O)CCC2)cc1 79250,c1(C(=O)NC(C2CCCC2)CNC(CCSCC(N)=O)=O)cc2cccnc2[nH]1 79251,C1(C(N2CCC(N(C)C)C2OC(=O)NC(C)(C)C)=O)CCCC2(CCCOC2)O1 79252,C(c1ccc(C(F)F)o1)=CC(=O)NCCC(C)NC(c1cc(Cl)c[nH]1)=O 79253,C1(NC(c2sc(C)c(O)n2)=O)CCOC2(CCN(C(=O)CC(C)(C)F)CC2)C1 79254,C=CCCC(C(=O)N(C)Cc1nnc(C)o1)NC(c1cnncc1OC)=O 79255,c1(CNC(C2CCSC2)=O)ccc2c(c1)CN(C(C1CCCC(CF)C1)=O)C2 79256,C=CCC(C(=O)NC1(CNC(c2cccn3ccnc23)=O)CCC1)C(C)C 79257,C(=O)(CCc1csnn1)NCCCN(C(=O)Cc1nncs1)CCOC 79258,c1(CC(C(=O)NC(c2ccc(F)cc2)CC)N)c[nH]c2cc(Cl)ccc12 79259,O=C1NC2(CCN(C(=O)CC3CCN(n4ccccc4=O)C3)CC2)CO1 79260,c1(C(c2n(C)nnn2)NCC2CC(F)C2)cncc(C(C)(C)C)c1 79261,c1(C(=O)NCC2C(N(C)C)CN(C(C3N(CC)CC3)=O)C2)c(OC)cccc1O 79262,N12CC(C1)C2=O.N12CC(C1)CC2=O.C1(N(CC=C)CCC)(C(=O)OCC)COC1 79263,C(C(CC(=O)NC1CCC(=O)NC1)NC(c1cncc(F)c1)=O)OC 79264,N(C1CN(C(=O)CC2CC3CC3C2)CCc2ccccc21)C(C(C)=C(CC)C)=O 79265,c1(C(N2CCC(c3noc(C4CCC4)n3)CC2)=O)ccc(C2CC2)cc1C1CC1 79266,c1(C(=O)NCCCN(C(C(CC)SC)=O)CC)cccc2ncoc12 79267,C12(NC(CCOCC#C)=O)CCCC1N(C(c1cc(SC)ccc1C)=O)CCC2 79268,C1(CC(=O)NCC(=O)NCC(=O)NC(C(C)C)C2CC2)COCC1O 79269,c1(N(C(C(C)CN(C)C)=O)C2CC2)cn(C)nc1-c1ccoc1 79270,c1(SCCC(=O)N(C2CN(C(C3CC(CCCCC)C3)=O)C2)C)nccn1C 79271,C1(COC)(N(C(=O)C(O)CC2=CC=C(CC)C2)c2ccccc2)CCN(C(=O)CS(N)(=O)=O)C1 79272,C1(CNC(C2CC2CCOCC)=O)CC(C)C(O)C1.n1(CC)cc(CC(=O)OC)cn1 79273,C1(OC)(CNC(=O)CC2CCC3CC23)CCN(C(=O)Cc2cccc(O)c2)C1 79274,CCC(C)C(C)NC(=O)C(C1CCCCC1)NC(=O)CC1OCCO1 79275,c1(OC)cnc(C(=O)NCCC2(OC)CN(C(C3C4CCC(=O)C34)=O)C2)c(F)c1 79276,C1(NC(c2[nH]cc(CC(C)C)c2)=O)C2CC1N(C(C13CC(C#N)(C1)C3)=O)C2 79277,C(=O)(C(C)CC(C)(C)C)NC12C(NC(C(C(CC)O)(C)C)=O)CC(CC1)C2 79278,c1(CNCCC2C(c3ccc(C(=O)OC)cc3)C2)ccc(F)cc1Cl 79279,N1(C(c2ccc(C)nn2)=O)CC(C)(C)CC1CNC(=O)CC1CCCC12CC2 79280,C1(C(=O)NCC(=O)N(C)Cc2cn(C3CCC3)nn2)CCC2(CCC2)O1 79281,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79282,C1(NC(C(C)(C)C23CC(C2)C3)=O)CCCCN(C(=O)Cc2cccnc2Cl)C1 79283,Cc1ccncc1CN(C)C(c1nc(CNC(c2cc(C)c(C)o2)=O)oc1C)=O 79284,N1(C(N(CCCC)C(C)CC)=O)CCC(CCN(C)C)C(F)(F)CC1 79285,c1(CN2C(=O)CN(CCCc3ccn(C)n3)C2=O)ccc(Cl)c(C)c1Cl 79286,C(=O)(C1=Cc2ccccc2C1)N(CCOCCCN(C(CCC(C)SC)=O)C)C 79287,c1(OC)ccc(Cl)c2[nH]c(C(=O)NC3(CCNC(C4CNC(=O)N4)=O)CC3)cc12 79288,Cc1n[nH]cc1C(=O)NC(C)CCN(C(=O)CC1(O)CCOC1)C 79289,C1(CC(=O)N(C2CCN(C(C(COC)(C)C)=O)C2)C)CC2CCC(C1)N2C 79290,c1(CC(N2C(C(=O)NCC3(CO)CC3)CCCC2)=O)cc(F)ccc1[N+](=O)[O-] 79291,c1(C(=O)NC(C)CNC(c2ccc(C(=O)N(C)C)nc2)=O)cccc2nsnc12 79292,c1(-c2cc(C(=O)NC(c3ccccc3N(C)C)C)no2)ccc(Br)cc1[N+](=O)[O-] 79293,C1(NC(C(C)(C)n2cc(Cl)cn2)=O)CCC(O)CN(C(C2CC2F)=O)C1 79294,C1(C(=O)NC23CCC(C(N)=O)(CC2)C3)CC2(CCC2)CN1C(=O)CC(F)(F)F 79295,C(=O)(C(C(=O)NCC1(F)CC(NC(=O)CCCCC(C)=O)C1)C(C)(C)C)OCC 79296,Cc1cccc2[nH]cc(CCC(=O)NCC(CC(C)C)NC(c3ccns3)=O)c12 79297,c1(C(N2CC(NC(Cc3cc(OC)no3)=O)(CO)C2)=O)c(C)ncn1O 79298,c1(CC)nc(C(=O)N(C2CCCC2)CC(=O)NCc2cc(=O)cc[nH]2)c(C)o1 79299,c1(COC)cc(C(N2CC(C)C2c2cccnc2)=O)co1 79300,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2cc(C)on2)=O)C2(CCC2)C1 79301,C1(NC(CCOCCOC)=O)CS(=O)(=O)CC1NC(c1cc(OC)ns1)=O 79302,C(=O)(CCC(C)(C)F)NCC(C)N(C(c1ccc(OC2CCCC2)cc1)=O)CC 79303,N1(C(=O)CN2CCNC2=O)CC2(CC(C(N3CCC(C(=O)O)C3)=O)C2)C1 79304,c1(C(N(CC(C)(C)CNC(c2cncn2C)=O)CC)=O)ccc2nc(S)oc2c1 79305,C1(C(N(C(CNC(=O)C2=CC(C)(C)C2)C2CC2)C)=O)CCCN2CCCCC12 79306,Cc1cc(N2CC(CNc3ccnc(N4CCN(C)CC4)n3)C2)cc(O)c1 79307,c1(C(N2CC(NC(C3C=CCCC3)=O)C(C(F)F)C2)=O)n[nH]c2ccccc12 79308,CCC(CC(=O)N1CC(C(N2CC3(C2)CN(C(C)C)C3)=O)C(F)(F)C1)C(F)F 79309,N1(C(CCC#CC)=O)CCC(C2CCN(C(=O)Cc3cc(C)cc(C)c3)C2)CC1 79310,N1(CCC)CC(C(=O)N(CCCCN(C(=O)CC2CC2(Cl)Cl)C)C)CC1=O 79311,c1(C(=O)NC2(CCNC(c3nc(C(N)=O)sc3)=O)CC2)ccnc(OC(F)F)c1 79312,N12CCN(CC1NCc1ccncc1Cl)C2=O.Cn1cc(-c2cccs2)cn1 79313,C1(CNC(C2C(C)CN(C(=O)C=CCN(C)C)C2)=O)CCCC(C)(C)C1 79314,N(C(=NCCCCl)NCc1ccc(OC)cc1OC)C(CC)CO 79315,C1(NC(Cc2nc(C(C)C)sc2)=O)CN(C(c2ccc(C(F)F)cc2)=O)CC1C 79316,n1(CCCNC(=NC)N(C)CCNCC(F)(F)F)ccc(=NC(=O)OCC)[nH]1 79317,c1(-c2c(C(N(C(C)CNC(=O)C(C)OC)CC)=O)scc2)ccc(Cl)cc1 79318,N#Cc1ccc(NC(=O)CSCc2cc(-c3ccc(Br)cc3)n[nH]2)cc1 79319,C=C(C)C1CN(C(=O)C(=O)NCCCNC(=O)C(C)OCCOC)CCO1.C(C)=O 79320,N1(C(c2c(C)c[nH]c2)=O)CCC2(CC1)COC(C)C2N(CC(C)(C)F)C 79321,c1(N2CCC(CCNC)CC2)ccn2nccc2n1 79322,c1(OC)cnncc1C(=O)N(C)CC1CCN(C(C2CCNC2=O)=O)C1 79323,C1(C(=O)NCc2noc(-c3ccccc3Br)n2)CNCCS1(=O)=O 79324,c1(SC)ccc(C)c(NC(=O)C(N2CCN(C3(O)CCS(=O)(=O)C3)CC2)=O)c1 79325,C1(CNC(c2cccc(OC)n2)=O)CCN(C(=O)C(C)(F)F)CC1O 79326,CCCCCCCCCC(O)CC(=O)N1CC(CNCc2ccc(O)c(O)c2)C1 79327,CC1(CNC(c2csc(Cl)n2)=O)CCN(C(C2CC=CCC2C(F)(F)F)=O)CC1 79328,C1(C(N2C(CC(=O)NCc3cnc(CC)s3)CCCC2)=O)C2C3CCC(C3)C12 79329,CN1CCN(C(C2CC2C(F)(F)F)=O)C(CNC(=O)Cc2cccc(Cl)c2F)C1 79330,c1(C(=O)NC(N)=O)cc2oc(Br)cc2s1.n1(CCC)cc(CCO)nn1 79331,c1(-c2ncc(C(=O)NCC(CO)NC(c3cccs3)=O)s2)ccccc1Cl 79332,C(=O)(CCCSC1CC1)N(C(C)(C)CNC(=O)COCCF)C 79333,c1(C(N(CCCNC(C(=CC2CCC(C)CC2)C)=O)C)=O)ccc(Cl)c2occc12 79334,C(=O)(C(C)(C)C1=CCN(C(=O)C(C)N=[N+]=[N-])C1)N1C(CCC)CCC1 79335,N1(C(CC(C)C2CC2)=O)C2CCC1CC(N(C(=O)C(C)(C)C1CCC1)C)C2 79336,N1(C(C2CC3CC2C3)=O)CCN(C(C23CC(C2)C3)=O)C2CCCC12 79337,CC1CCCCC1(CNC(C1C2CC(=O)CC12)=O)NC(C1CCOCC1)=O 79338,C1(NC(c2cc(C)cc(Cl)c2)=O)CS(=O)(=O)C2CN(C(C3CSCCS3)=O)CC12 79339,N1(C(CCSC)=O)CCC(C2(CNC(c3cc4ccc(F)cc4[nH]3)=O)CC2)CC1 79340,c1(CCNC(C(C)(C)C)c2nnnn2Cc2ccccc2)ccc(F)cc1Cl 79341,Cc1cnc(NC(=O)CC2CN(C(=O)CC(C)C)CCO2)c(C)c1 79342,C1(C(=O)NCC(CC)(CC)NC(c2ccc(C)c(C)n2)=O)(CC)CCC(O)CC1 79343,CC1CN(C(CC2CCC(F)CC2)C(=O)NCCC2(C)CC2)Cc2c[nH]nc21 79344,N12CCN(CCC1C)C(=O)CN1CCCCC1C2=O.C1(OC)CCCCC1C 79345,c1(OCC(=O)N(CCCC(=O)N(CC(C)N(CCCF)CC)C)C)ccc(F)cc1 79346,C(=O)(C(c1ccoc1)NC(=O)CSC)NCC1(OCC)CC1 79347,C1(O)(CCNC(c2cccc(CS(C)=O)c2)=O)CCN(C(C2CCCC2)=O)CC1 79348,CCCC(C(=O)NCc1ncccc1C(=O)N(c1cnn(C)c1)CC)NC(N)=O 79349,C(=O)(CC(C(F)(F)F)NC(C12CCC(CC1)C2)=O)N(c1cnc(C2CC2)nc1)C 79350,N1(C(CCN(CC#C)C(c2ccn(CC)c2C)=O)=O)CCOC2COCC12 79351,Cc1ncc(Cl)c(-c2nc(-c3cncn3C)no2)n1 79352,C1(C(=O)NCC(CNC(C(N(C)C)C2CC2)=O)O)CC(c2ccccc2)(CO)C1 79353,N1(C(c2cc(C(N)=O)cs2)C(=O)NCC)CCN(Cc2cccnc2)CC1C 79354,c1(OC2CCC(F)(C(N3CC(NC(=O)OCC)C3)=O)C2)cccc2c1cnn2C 79355,N1(C(C(CCOC)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 79356,N1(C(C2(C)CSC2)=O)CCC(CNC(C2(C)CCC(=O)NC2)=O)C(F)(F)C1 79357,C1(C(=O)N(C)Cc2[nH]nnc2C)CCN(C(=O)C2(C(=O)OC)CCC2)O1 79358,C12(NC(CN(CC)CC)=O)CC(C)(C1)OC21CN(C(c2cc(C)c(C)cc2C)=O)C1 79359,C1(CC(=O)NC2CCCC(CNc3cc(OC)ncn3)C2)C(=O)N(C)N=C1C 79360,C1(C)(CC(=O)NCCC=CC)CCN1C(c1cnc(N)s1)=O 79361,CCCC(C(=O)NC1(c2ccsc2)CC1)NC(c1cscc1OC)=O 79362,C1(C(C)NC(c2cc(C)on2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 79363,c1(CNC(C=CC2N(C(C(CC)CN(C)C)=O)CCC2)=O)ccc(F)cc1F 79364,C1(NC(CNC(=O)NC)=O)CCOC12CCN(C(c1cc[nH]c1)=O)CC2 79365,Cn1cccc1-c1cn(CCCC(=O)NCC(O)Cn2cccn2)nn1 79366,Cc1nnc2cc(C(=O)NCC3CC(NC(C4(NC5CC5)CCC4)=O)C3)ncn12 79367,N1(C(c2c(C)coc2)=O)CCC(C(=O)NC2CN(C3CCC3)C2)CC1C1CC1 79368,CCC(F)(F)C(C)(C)C(=O)N1CC2CCC1CN(Cc1[nH]nc(C(F)(F)F)c1C)C2 79369,N1(C(C2CCN(C)CC2)=O)CCC2C1CCCN2C(c1ccn(C(F)(F)F)n1)=O 79370,C12(C(=O)O)COCC1CN(Cc1csc(-c3cccc(Cl)c3)n1)C2 79371,c1(CCN(C(C(=O)N(CCN=[N+]=[N-])CC)=O)CCCCC)cc(C)nn1CC 79372,c1(C(=O)NCCCC(=O)NC(CC(=O)OCC)C)cccc(C)c1O 79373,c1(C(N2CCC(C(C)(C)C)(CNC(C3(OC)CC3)=O)C2)=O)cc(C)nc(C)c1 79374,CON(C)CCCNC(C1C=CCCN1C(C1(C=C)CCC1)=O)=O 79375,C(CCCCC(=O)NC(C)C(C(C)C)NC(C1CCSCC1)=O)OC 79376,O=C(CC1COCc2ccccc21)NCCC1CCN(C(=O)Cn2cnnc2)C1 79377,C(CCOC(C)=O)(C(C)C)NC(C1(N(C(CCC)=O)C)CC1)=O 79378,c1(C=O)c(C)nc(C)n1O.N12CC(C(C)(C)O)(C1)CNC(=O)C1C(C1)C2=O.CO 79379,c1(C(N2CC(CNC(C(n3cc(Cl)cn3)C)=O)C2)=O)c[nH]cc1C(F)(F)F 79380,C1(C)(C(=O)Nc2ccc(COC)c(F)c2)CCCN(C(=O)OC(C)(C)C)CC1 79381,C1(CN(CCOc2cccc(NC(C(CC)OC)=O)n2)C)CCC=CCCC1 79382,C1(CNC(C(C)OCCC=C)=O)CN(C(C2CCCCN2N=O)=O)CCC1(F)F 79383,C1(C(=O)NC(CC)(C)CNC(=O)CCOCC2CCC2)CCCC(C(=O)OC)C1 79384,N(C1CCCc2n[nH]cc21)C(c1cc(CNC(C(C(C)C)NC(C)=O)=O)sc1)=O 79385,C=C(C)CCCN=c1c(Br)ccc(S(=O)(=O)N2CCC3CCCCC23)[nH]1 79386,C1(C(=O)NC2COCC2n2cc(-c3ccsc3)nn2)CCC(=C(F)F)CC1 79387,C1(NC(C2C(CNC(c3c(CC)oc(C)c3)=O)CCC2)=O)CC2CC1C(O)C2O 79388,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)cc1O)=O)CC2 79389,N1(C(C=CC2N(C)CCC2)=O)CCN(C(c2cc[nH]c2)=O)CC1CF 79390,C1(CC(=O)N(CCC(=O)N(C)Cc2ncc[nH]2)CCO)CC1C1CC1 79391,C1(NC(C(C)C#N)=O)CN(C(c2cn(C)nc2Br)=O)CCC12CCC2 79392,CC1CN(C(c2cn(C)c(=O)n2C)=O)CCC1NC(C1(CO)CCCC1)=O 79393,C1(SC)(CNC(=O)CC2CN(C(=O)CSc3nc[nH]n3)C2)CCC1 79394,CCC(O)C(C)C(=O)N(C1CCN(C(=O)CC2C(CC)C2(F)F)CC1)CCOCC 79395,C1(NC(C2CC2C2CCC2)=O)CC2CC1CC2C(=O)NC(CC1CCCC1)CO 79396,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79397,C1(NC(C(CC=CC)C)=O)CC12CCN(C(c1cc(C#N)cn1C)=O)CC2 79398,c1(CCC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)C)C2)s1 79399,C(=O)(C#CC1CCOC1)N1CC(NC(c2c(C)nc(-c3cnn(C)c3)s2)=O)C1 79400,C12(NC(COCC(C)(C)C)=O)CCCCCC1N(C(C1(N(C)C)CC1)=O)CC2 79401,c1(OC)ccc(F)c(C(=O)N(CCNC(c2nc(Br)cnc2N)=O)C(C)C)c1 79402,c1(C(=O)NCC(C)N(C(c2ccc(N)c(O)c2)=O)CC)ccc2c(C)[nH]nc2c1 79403,C1(C(N2C(CCNC(Cc3cncc(C)c3)=O)CSCC2)=O)C2CCC(F)(F)C12 79404,c1(C(N2CC(O)(C(C)NC(C3CC(N(C)C)CCO3)=O)C2)=O)cc(O)cc(Br)c1 79405,CC1COCC2(CCN(CC3(C#N)CCOCC3)CC2)O1 79406,c1(COC)cc2c(cn1)NC2=O.C1(COC)(CO)CN(C(=O)CC2OCCO2)C1 79407,C1(CCC=C)(C(=O)NCC(C)OC(F)F)CN(C(=O)C(C)C2CCOC2)C1 79408,C1(CC(N2CC(O)(CN(C(=O)C(C)(C)C3CCOC3)C)C2)=O)OC(C)(C)OC1=O 79409,C(=O)(C(C)C(O)CC(C)C)NC1CC(CNC(C2(CCCC)CC2)=O)C1 79410,C(=O)(C(CC(C)C)CC(C)C)NC1CC2CN(C(CC(C)SC)=O)C1C2 79411,C1(CC)CN(C(c2ccc(CC3CC3)nc2)=O)CCN1C(=O)CC1(C)CCC1 79412,C1(CC=C)(NC(=O)C=CCN(C)C)CCCN(C(c2cc(CN(C)C)[nH]n2)=O)C1 79413,n1(CC(C)C)ccc(C(=O)NCCN(CC(=O)NC2CCSC2)C(C)C)n1 79414,C1(CCC)COCCN1C(=O)C(C)C(C)NC(=O)C=C(C)C 79415,C1(NC(C2CC(=O)NC2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CC12CCCC2 79416,C1(C(C)C)CN(C(=O)COC(C2CCN(C)CC2)=O)CC(c2ccccc2)O1 79417,C1(C(N(CC(=O)NCCNC(c2ncccn2)=O)C)=O)COC(=O)N1C 79418,C1(NC(=O)NCC(C2CCCO2)O)CC12CCS(=O)(=O)CC2 79419,N1(C(C(C)N2CCC2)=O)CCCC12CCN(CC1(OC)CC1)C2 79420,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1cccs1)C2 79421,c1(CCNC(=O)NC(CC=C)CC=C)noc2c1CCC2 79422,c1(NCCCCNC(=O)CCCc2cccs2)nccc(-c2ccnn2C)n1 79423,N1(C(CC(CCC)C)=O)CCN(C(c2cccc(=O)n2C)=O)C(C)CC1C 79424,C1(CCNC(C2CCC(CC)O2)=O)COCCN1C(c1cccc(C(F)F)c1)=O 79425,c1(C(=O)NC(CCC)C2CCC2)cc2[nH]nnc2cc1OC 79426,C1(N(C(=O)NC)CC2C(CCC)C2)CC(=O)CN1C(c1ccccc1OC)=O 79427,N1(C(=O)C2CC2)CCCC(F)(SCc2ccc(C(C)NC(=O)CCS(C)=O)s2)C1 79428,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(=O)CC2OCCO2)C1 79429,N1(S(CCC)(=O)=O)CC2CN(C(c3cc4n(n3)CCC4)=O)CC2C1 79430,C(=O)(C1=C(C)Oc2ccccc2C1)NCC(CCCC)NC(c1ncc(C)s1)=O 79431,C1(C(=O)OCCOC)CCN(S(=O)(=O)Cc2nc(-c3ccccc3Cl)no2)CC1 79432,CN=c1ccc(C(=O)N(C(C)CNC(c2csc(C3CCCO3)n2)=O)C)c[nH]1 79433,C(=O)(C(C)S(=O)(=O)NS(=O)(=O)Cc1cc(C(F)(F)F)oc1C)OC 79434,NS(=O)(=O)c1cccc(CC(=O)Nc2ccc3nc(Cl)sc3c2)c1 79435,N(C(=NCCCOC)N(C)Cc1cc(C)c(C)s1)CC(c1cccc(Cl)c1)OC 79436,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79437,CCS(=O)(=O)CC(=O)Nc1cccc(NC(=O)NC2CCN(C3CC3)C2)c1 79438,Cc1cnc(N(C2CC2)CCNC(=O)C(C)Cn2cccn2)nc1S(C)(=O)=O 79439,c1(C(N2CC(NC(=O)CC3CCOC3)C(F)C2)=O)ccnc(Cl)c1Cl 79440,c1(C(=O)NCC2CC2NC(c2ccccc2C)=O)cc(OC(F)F)ccc1Cl 79441,C(=O)(C1=CCCCC1)N1CCC(c2cn(Cc3cnc(OC)nc3)nn2)C1 79442,c1(C(=O)NCCC(C)NC(CCc2c(C)cccc2)=O)c(C)cc(O)nc1C 79443,N1(C(C(C2(C)CC2)NC(C2CC2(F)Cl)=O)=O)CCC(CO)C(C)C1 79444,C1(C(=O)NCCOCCOC)CCCC1CNC(C1CSCCO1)=O 79445,C1(C(N2C(CNC(c3cc(Cl)ccc3F)=O)C=CC2)=O)Cc2ccccc2N1 79446,c1(C(N2C(C(=O)NC3C(CC=C)COC3)C3CC3C2)=O)ccc(C#N)cn1 79447,C12(CNC(Cc3cccc(C)c3F)=O)CCCC(CN1C(=O)C(F)F)C2 79448,C(=O)(C(F)CCC(C)C)N1CCN(C(CCCC#C)=O)C(CCO)C1 79449,C=CC1(C(=O)NC(C2CC=CCC2)C(=O)N(C)Cc2n[nH]c(C)n2)CCCC1 79450,C1(C(=O)Nc2cc(C)sn2)CCCN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CC1 79451,c1(C(=O)NCC(C2CC2)NC(C(C(=O)Nc2nccs2)C)=O)ccc2nccn2n1 79452,c1(C(=O)NCCCN(C(C2CCC(C)CC2)=O)CCO)c[nH]c2c(C#N)cccc12 79453,N(C1CCCc2c(C)cccc21)C(c1n(CC=C)nnn1)c1cn(CC)nn1 79454,c1(C(=O)NC2C(C)CN(C(C3CCCO3)=O)C2)cc2cccc(Br)c2[nH]1 79455,C1(C)(CC)C=C(C(=O)NC(C)CC2CN(C(=O)C(O)CC3CCCC3)C2)C1 79456,C1(OC)CC(C(=O)NC2CCCC2)N(C(c2cnc(C)s2)C(=O)OC(C)(C)C)C1 79457,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 79458,C(CC1=CCN(C(C2CC23CC(C)(C)C3)=O)CC1)NC(CCCC(=C)C)=O 79459,N1(C(C(C)CC(F)F)=O)C2CCC1CN(C(=O)C(C)(C)C1CCCO1)C2 79460,c1(-c2cccc(C(C)O)c2)ccc2cc(C(=O)NCC3COC(C)(C)O3)[nH]c2c1 79461,c1(C(=O)NCC2N(C(C3CCCC(OC)C3)=O)CCC2C)cccn(C)c1=O 79462,CCC(CC)C(C(=O)N1CCCC1CN(C(=O)CCCN1CCCC1)C)OC 79463,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(N(C(=O)CCCc2cccnc2)C)C1 79464,n1(CC(=O)NC(CCC)C2CCC2)cc(C(N)=O)nn1 79465,c1(CC2C(C(N(CC(=O)NC3(c4cc[nH]n4)CC3)C)=O)CCC2)cccc(F)c1F 79466,c1(OC)ccncc1C(=O)NC1CC(C)(CNC(=O)CC(C)(C)NC(C)=O)C1 79467,C1(C(C(C)NC(c2cnsc2)=O)NC(=O)COCCN(C)C)CCCCC1 79468,C(C(CO)(CO)NC(=O)CN(C)C1CC1)N(C(c1nc(CC(C)C)sc1)=O)C 79469,C12(C(=O)NCC3C4CN(C(c5nncs5)=O)CC43)CC3CC(C1)CC(F)(C3)C2 79470,N1(C(C=CC(C)(C)C2CC2)=O)CCC(C(=O)N2CC(SC(F)F)C2)=C(F)C1 79471,N1(C(c2c(CC)noc2)=O)CC2CCC2(CNC(=O)C(CCC)N(C)C)C1 79472,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 79473,C(=O)(CC(C)CCCC)NC(C1(C(=O)NCCC#C)CC1)C 79474,C1(OCC)CC(C)CN1C(=O)C(=O)NOC 79475,Nc1cc2[nH]cnc2cc1C(=O)NCC1CC1NC(=O)Cc1csc2cncn12 79476,C(C(O)CC(=O)NCCC1OCCC1(C)C)NC(CCCOCCC)=O 79477,C(=O)(C(C)(C)C(F)(F)F)N1CCCCC(CNC(C(C)OC2CCCC2)=O)C1 79478,C1(NC(CSCC)=O)CN(C(c2ccn(C3CC3)n2)=O)CCC12CCOCC2 79479,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 79480,N1(C(c2c(CC)con2)=O)CC(CC(=O)NCc2nc(CC)no2)CC12CCC2 79481,C12(NC(=O)CO)CCCC1N(C(c1cnc(-c3cccnc3)s1)=O)CCC2 79482,C(=O)(C1CCc2cc(Br)ccc21)N1CCN(C2CCCN(C)C2)CC1 79483,C1(CNC(c2ccc(CSCC)o2)=O)CCCN(C(=O)CN2CCOCC2)CC1 79484,c1(NC(C2(C(CCC)c3cncs3)CC2)=O)ccc(=N)[nH]n1 79485,c1(CC(c2n(CC=C)nnn2)NCc2csc(C)c2C)cccc(F)c1 79486,Cc1cc(C(=O)NCCC(O)CNC(c2nncs2)=O)ccc1O 79487,C(C(=O)NN1CCCC1C(N1C(C)CC1(C)C)=O)c1c(C)n[nH]c1 79488,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 79489,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 79490,C1(NC(C2(O)Cc3ccccc3C2)=O)CC2CCC1N(C(C1CC1(Cl)Cl)=O)C2 79491,c1(NCC(=O)NC2C(NC(c3c(C(C)C)noc3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 79492,Cc1cc(CC(=O)N(CCC(C)NC(=O)Cc2ccc[n+]([O-])c2)C)ccc1F 79493,N1(C(C(CC=CC)C)=O)CCCC(C)(NC(C2CC3C=CC2C3)=O)C1 79494,c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)CC(F)F)cc1F 79495,N1(C(c2ccn3ccccc23)=O)CCCC2(CCCN2C(=O)C(F)=CCCF)C1 79496,C1(NC(C2CC=C(C)CC2)=O)CCN(C(c2ccn(CCO)c2C)=O)C(C)C1 79497,c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 79498,N1(C(C(CC)n2cncn2)=O)CC(F)CC1CNC(=O)COc1cccc(C)c1 79499,CC(C)C(C)(C)C(=O)NCCCNC(C1(C(F)(F)F)CC(O)C1)=O 79500,c1(Cc2cn(CC(C(=O)N3C(C(=O)NC(C)C)CC3)O)nn2)ccccc1F 79501,CC1CCN(C(C2CC(=O)N(O)C2)=O)CCN1C(c1cc(-c2ccoc2)[nH]n1)=O 79502,c1(S)nc2ccccc2[nH]1.C1(NC(C(C)CCN)=O)CCN(CC2CCC(=O)O2)C1 79503,c1(C(=O)NCCN(C(CCc2onc(C(C)OC)n2)=O)C)cnncc1O 79504,C1(C(=O)NCC(CNC(c2ccn(CCN(C)C)n2)=O)O)CC2C=CCC(C1)C2 79505,Cn1nc(Br)c2c(NC3CC(=C4CC4)C3)ncnc12 79506,c1(C(=O)NCC(C(C)C)NC(C2(CC(C)C)CCC2)=O)ncccc1C(C)(C)C 79507,N1(C(C=NOC)=O)CCC2(CCN(C(c3c(C)noc3C(F)(F)Cl)=O)C2)C1 79508,N1(C(CCCc2onc(C)n2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 79509,c1(CC(=O)OC)ccc(Cn2cncn2)c(-c2ccccc2)c1 79510,n1(CC(C)C)c(N)c(N(C(C)C)Cc2ccc3nonc3c2)c(O)nc1=O 79511,c1(C(=O)NCc2cc(C)c(C(=O)NC(C)CS(N)(=O)=O)o2)cc2ccncc2[nH]1 79512,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CN(C(c1ncccc1Br)=O)C2 79513,c1(OCC(=O)NCCC2N(C(CC(C=C)(C)O)=O)CCC2)cccc([N+](=O)[O-])c1 79514,C1(C(=O)NCCOC2CN(C(c3nc[nH]n3)=O)C2)CC2COCC(C1)C2=O 79515,C1(C(N2CC(SC)C(NC(=O)COCCN(C)C)C2)=O)CC2C(C1)C2(C)C 79516,O=S(=O)(c1ccc(N2CCCCCCC2)c(Br)c1)NCC12CCCC1C2 79517,c1(CCCC(N2C(C3(NC(C(CC)F)=O)CC3)CCC2)=O)ccc(F)c(F)c1 79518,Cc1cc(C(N2CC(NC(c3cnco3)=O)C3(CC3)C2)=O)nc(O)n1 79519,N1(C(C2N(C)C(=O)C(F)C2)=O)CCS(=O)(=O)CC1c1ccc(C)o1 79520,c12ccccc1C1(CC1)C(c1ncc(Br)cn1)N2.c1(CC)n[nH]cc1C(=O)O 79521,C1(NC(C2CCC(C)O2)=O)CCCCC1NC(c1ccc(Cl)s1)=O 79522,Cc1nc2ncnn2c(C)c1C(=O)NC1CC2CC1N(C(C1CCCNCC1)=O)C2 79523,C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(C1CCN(C)C(=O)C1)=O 79524,N1(c2nc(C(=O)OC)c(C)s2)CCC(C)(NC(=O)CN(C)C(C)C)CC1 79525,c1(-c2c(Br)cnc(N3C(C)COC(CO)C3)n2)nc2ccccc2n1C 79526,CCN=C(NCc1ccc(C#N)cc1Br)N1CCCC1 79527,CCCCC(CC)C(=O)NCCc1cnc(COc2ccccc2)s1 79528,C1(NC(CN2CCN(C(C(C)CO)=O)CC2)=O)CCCC2(CCC2)C1 79529,N1(C(c2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)CC1CNC(=O)C1 79530,O=NN1CCCC1C(=O)NCC1CCN(C(C2CC=CCC2)=O)CC1 79531,n1(CC)nc(C)c(C(N2CCCC(N(C(=O)CC3(C#N)CCC3)C)CC2)=O)c1Cl 79532,c1(N2CCC(O)(C(F)F)C2)nccc(=NCC2CC2)[nH]1.c1(C2(CN)CC2)ccccc1 79533,c1(C(=O)NCC(CO)NC(C(CC)OC)=O)ccc(N2CCOCC2)cc1 79534,Cc1c(C(=O)NCC2CC2)c(-c2ccccc2)nn1CC(F)(F)F.C(C)(C=O)O 79535,C#Cc1ccc(C(=O)NCC23CC(CN2C(=O)CSc2ccccc2F)C3)nc1 79536,N1(C(C2CC(=O)NC2)=O)CCCC(C2(NC(c3c(F)cc(F)cc3Cl)=O)CC2)C1 79537,CC1CC(C(=O)NC(C)(C)Cc2ccccc2)C(=O)N1Cc1ccccc1 79538,n1(C(C)C)cc(C(=O)NC(C)(CNC(C2CC=CC2)=O)C(C)C)c(Br)n1 79539,c1(C(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 79540,c1(-c2nc(C(=O)NC(c3cccc(Br)c3)C(C)C)on2)cccc(OCCF)c1 79541,CC(C)S(=O)(=O)c1ccc(-c2cc(NC(c3cc(F)ccc3O)=O)ccn2)cc1 79542,Cc1ccc(CC(C)C)c(C(N2CC(C(=O)O)C(C(F)F)C2)=O)c1 79543,CCC(C)C(O)C(=O)N(CC(CC)NC(c1cc(-c2ccccc2)oc1C)=O)CC 79544,CCC(C)(C(=O)NCC1CN(C(c2ccn(C)c(=O)c2)=O)C1)C(N)=O 79545,c1(-c2cn(CC(=O)NC(Cc3cccc(F)c3)CO)nn2)cccn2ccnc12 79546,Cc1cnc(C(=O)N(CCCCCNC(C2CC(=O)C2(C)C)=O)C)c(F)c1 79547,N1(C(c2ccc(SC)s2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)n2)CC1 79548,CCC(CC(F)F)C(=O)N(CCCNC(=O)CCc1cccc(F)c1Cl)C 79549,c1(C(=O)NCCOCCN(C(C2CC(C)OC2)=O)C)cccc2ccn(C)c12 79550,CC(CC(=O)N1CC(C)(NC(c2ccn(CCF)n2)=O)C1)c1ccccc1 79551,N12CCC(CC1C)OC2=O.Cc1ccc(C(C)C)cc1.N12CCC(C1)OCC2=O 79552,c1(C(N(C2CCC(NC(C3(N(C)C)CC3)=O)C2)C)=O)nc(C(F)(F)F)cn1C 79553,c1(-c2cn(C(CC)C)nn2)cnn(CC(=O)NCCSc2cccnc2)c1SC 79554,c1(COC)nc(C(=O)N(C(C)CCNC(C2CC23CCC3)=O)C)co1 79555,c1(C(C)NC(CC2(NC(Cn3c(C)nnn3)=O)CCC2)=O)cc(Cl)ccc1F 79556,C(CN1C(=O)Cc2cc(CN3CCNC(=O)C3)ccc21)OC(C)C 79557,C#Cc1cncc(C(N2CCC(NC(C3COCCN3CC)=O)C2)=O)c1 79558,N1(C(CSCCC)=O)CC(NC(c2cc(C)c(C)cn2)=O)CC1(C)CC 79559,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CC)CNC(=O)CN2CCC(C)CC2)C1 79560,C(CCCCCC(=O)NCC1CC(C)N(C(c2ncc(F)cn2)=O)C1)SC 79561,c1(C(=O)NC2CC3CC2CN(C(C2CC2F)=O)C3)cc2n(n1)CCCCO2 79562,C1(N(C)C)CCN(C(=NCc2ccc(Cn3ccnc3)s2)NC(C2CCCO2)=O)C1 79563,c1(CC(=O)NCCC(C(=O)NC(C)C(=O)NC2CC2)OC)ccccc1C#N 79564,C1(NC(C2(C(=O)OC)C=CCC2)=O)CCN(C2CC2NC(N)=O)CC1 79565,C(CCCC(=O)NCCC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)OCCC=C 79566,O=C(C#CC1CCCOC1)NC1(CNC(c2ccnc(S)c2)=O)CCOC1 79567,c1(NCCCc2ccccn2)cc(N2CC3C(C2)C3(F)F)ncn1 79568,CN1CCN(c2ccc(C(N3CCC(NC(C)=O)C3)C(=O)NC3CC3)cn2)CC1 79569,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C)CC2F)=O)C1 79570,S(=O)(=O)(c1ccc(NCC(O)CC2CC2)nc1)N1C(C)CCc2ccccc2C1 79571,c1(NC(C(CCC)C#N)=O)cnn2c(Br)cccc12.c12nc(sc1C)NC2=O 79572,C1(N(C(CC(c2ccc(F)cc2)C)=O)C)CCCCC1N(C(=O)C(N)=O)C 79573,C1(N(C(C(COC)N(C)C)=O)C)CCN(C(=O)CNC(c2ccco2)=O)C12CC2 79574,c1(NC(C2(C)N(C(C3N(C(C)=O)CCCC3)=O)CC2)=O)ncc(Cl)cc1[N+](=O)[O-] 79575,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 79576,C1(C(=O)NC2CN(C(C(C)NS(CC)(=O)=O)=O)C2)(OC)CC(C(F)F)C1 79577,c1(NCC2CCCCN(C(C3CC(=O)N3)=O)C2)nc(Cl)nc2sccc12 79578,Cc1c(N(CCC(C)C)C)ncnc1N1CCC(F)(SCC2CCC2)C1 79579,c1(NC2C(C)CN(C(=O)C(CO)NC(N)=O)CC2)cc2nn[nH]c2cc1[N+](=O)[O-] 79580,c1(C(=O)NC2CCCC(NC(CC(C=C)(C)C)=O)C2)cc2ccccc2nc1C 79581,c1(C(=O)NCC2N(C(CCCC=C)=O)CCCC2)cc2ccc(OC)cc2[nH]1 79582,O(C=C(C#N)C(=O)NCC1CC1NC(c1ccc(=O)n(CCO)c1)=O)CC 79583,C1(NC(C2C(C(C)C)C2)=O)CCCN(C(c2cncn(C)c2=O)=O)CC1 79584,C1(NC(=O)CCc2ccccn2)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO 79585,c1(C(=O)NCCN(C(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 79586,c1(C(C)OC)ncc(C(=O)NCCN(C)C(C2CC2C2CC2)=O)s1 79587,c1(NC(CC(c2cccc(Cl)c2)C)=O)cc(Cl)cc2sc(Br)nc12 79588,C1(C(C)C)C(NC(=O)CCC2CCOC2)CCN1C(=O)CCCN(C)C 79589,c1(CC)oc2ccccc2c1CNN1CCN(CCCO)CC1C 79590,n1(C(C)C)ccnc1C(=O)N(C1(CC(=O)NC2CC(C)(C)C2)CCC1)C1CC1 79591,N1(C(c2c(C)nc[nH]2)=O)CC(NC(C2(C(=O)NC3CC3)CC2)=O)C2(CCOCC2)C1 79592,C1(C(N2CC(NC(c3ccnc(S)c3)=O)C2)=O)CCC2CCC1O2 79593,N1(C(C(C(C)C)OCC)=O)CCCCCC1CNC(c1c[nH]c(Br)c1)=O 79594,C1(NC(CCN(C(C)C)C(c2cncnc2O)=O)=O)CCC(C2CC2)C1 79595,C(C)(C)(CNC(=O)C(C1(C)CC1)NC(=O)C(C)C1CCCO1)OC(C)C 79596,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 79597,N1(C(CC2(COC)CC2)=O)CCOC2CN(C(C3CCSCC3)=O)CC12 79598,N1(C(C2(OC)CCC2)=O)C(CNC(c2cnn(C)c2Cl)=O)CC2COCC12 79599,c1(C(N2C(CCNC(CSCCN(C)C)=O)CSCC2)=O)cnc2ccoc2c1 79600,c1(C(=O)OC)sc(NCC2CCCCC2NC(c2nccn2C)=O)c(C#N)c1C 79601,CC(C)CCC(=O)C(=O)NC(Cc1cc[nH]n1)C(=O)NCC1CC1(F)F 79602,C1(OC)CC(C)CN(C(=O)C(CCC2CCC2)NC(C2CCC(O)CC2)=O)C1 79603,C=CC(C)(CC)C(=O)NCC1CCN(C(c2nc(O)c(C)s2)=O)C(C)C1 79604,C12(C(=O)OC)CCC(CN3CCC(CNC(=O)C(C)C4CC4)C3)(CC1)CC2 79605,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 79606,C#CCCC(O)C(=O)N1CCOC(CN(C)C(c2ccc(-c3cccs3)o2)=O)C1 79607,Cc1c[nH]c(-c2ncccn2)nc1=NCC1(C#N)CCC1 79608,C(=O)(CC(CC)c1ccccc1)N(CC(CC)NC(C1(S)CCC1)=O)C.CCC 79609,CCCCCCC(C)CC(=O)NCCN(C)C(C1(O)CCCC(C)(C)CC1)=O 79610,N1(C(CC2(COC)CCCC2)=O)CCC(C)(NC(=O)C=CCN2CCCC2)C1 79611,CC(C(C)C(=O)Nc1cc(C(F)F)no1)NC(C1(C(F)(F)F)CC1)=O 79612,Cc1ccc(NC(C2CC2N2CCOCC2)=O)c(C(F)(F)F)c1F 79613,C(CCOCCO)(C(=O)N(C(C)CO)C)NC(Cc1c(C)scc1)=O 79614,CCCN=C(NCc1nnnn1C1CCC1)NCc1ccn(-c2ccccc2)n1 79615,C1(C(=O)NCC2(C(=O)O)CC(=C)C2)CCCCC1NC(=O)COCCCCCC 79616,c1(CCC(=O)NC2C(NC(C(C(C)C)N(C)C)=O)C2)ccc(F)cc1Cl 79617,N1(C(CN2C(COC)C(C)CC2)=O)CCC2(CCC(O)C2)C1 79618,n1(CC)cccc(CN2CCOC(c3ccccc3Cl)C2)c1=O 79619,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 79620,CC1(CC(=O)NCC=CCNC(=O)CCCNC(N)=O)CC1(Cl)Cl 79621,N1(C(C2CC(N(C)CC)C2)=O)CCCOC(CCNC(=O)CCCCC2CC2)C1 79622,N1(C(=O)OC(C)(C)C)Cc2ccnn2CC(C(=O)OCC2CC2C(C)(C)C)C1 79623,c1(NCC(=O)NCC2CC(NC(C(CO)NC(C(C)C)=O)=O)C2)ccc(F)cc1O 79624,N1(C(COC)=O)CC(CNC(c2cc(Cl)c3c(c2)OCCO3)=O)C2(CCOCC2)C1 79625,C1(C)(C(=O)OCC)CCN(C(c2sncc2C)C(=O)NCCSC)C1 79626,N1(C(Cc2c(C)nn(CCOC)c2C)=O)CCOC2(CCOC2C)C1 79627,C12(CCC(CO)CC1)C(=O)N2.C(CCC(=O)N1CC(COC2CCCC2)C1)SC 79628,Cn1nc(C(F)F)cc1NC(=O)NCCn1cnc(C(F)F)n1 79629,C(=O)(C(C)(C)CCNC(=O)CCC=CC(C)C)N1CCC(CC)(COC)C1 79630,C(=O)(C1=CCCN(C(=O)CCn2cnnn2)C1)N1CC(C)S(=O)CC1 79631,c1(NC(C2N(Cc3ccc(OCC)cc3O)CCOC2)=O)nc(Cl)c(C)c(Cl)n1 79632,C1(CC(=O)NC2CC3(C(NC(C4CN(C)C4)=O)C3)C2)Cc2ccccc2NC1=O 79633,Cc1ccc(CC(N2CCC(=CCNC(=O)CC3CC(F)C3)CC2)=O)nc1 79634,Cc1cc(C(N2CC(N(c3ncc4[nH]ccc4n3)C)C2)=O)ncc1[N+](=O)[O-] 79635,CC1CCN(C(=O)C(C)CC(N)=O)C(CNC(=O)Cc2cccc(O)c2)C1 79636,N1(C(C(C)C2CC2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 79637,C1(CC(C)C)CCN(C(=NCCNS(C)(=O)=O)NC(C)CNc2ccccc2)C1 79638,n1(C(C(=O)NC2CCN(C(CCCC)=O)CC2)C)nc([N+](=O)[O-])cc1C 79639,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 79640,C1(C(N2CC(C(=O)NCCCCC)C2)=O)CCCC(CC)C1 79641,N#Cc1ccc(N)c(C(N2CCC(F)(NC(c3ccc4nncn4c3)=O)C2)=O)c1 79642,C1(NC(C(C)NC(N)=O)=O)CC2CC1CC2C(N1CC(O)(C(N)=O)C1)=O 79643,Cc1cc(-n2ccnc2SC(C)C(=O)NCC(C)NC(=O)C(C)(F)F)ccc1Cl 79644,C1(C(=O)Nc2ccc(C3CCN(C(C=COCC)=O)CC3)cc2)CCCC(C#N)C1 79645,C(=O)(C(CC1CC1)NC(c1ccncn1)=O)NC(C(=O)OCC)(C)C 79646,C1(O)(CNC(CCC(C)OCC)=O)CCCN(C(=O)CCCC2CCC2)C1 79647,N1(C(CC(=O)N(C)C)=O)CCCC1C1CCCN1C(C1CC2(C1)CC(F)(F)C2)=O 79648,N1(C(C=Cc2n(CC)ccn2)=O)CCN(C(c2ccc(S(C)(=O)=O)o2)=O)CCC1C 79649,N1(C(c2cnn(CC(F)F)c2C)C(=O)NCCOC)CCC(OC)C(C)C1 79650,c1(C(N2CCC(N(C(=O)CCC3CCOC3)C)C2)=O)cnc(N)c(N)c1 79651,N12CC3(CC1C3)C2=O.C1(OC(C)=O)CC1NC(=O)COC1CCC1.C(N)=O 79652,C(CCC(C)C)(C(=O)NC1CCCC1(C)CN(C)C)NC(c1ccc(C)n1C)=O 79653,c1(C(=O)NC2C3CN(C(=O)CCC4CCCC4)CC23)ccn2ncnc2c1 79654,CC(CNC(=O)CNC(=O)NC1CC1)N=c1ccnc(C2CCCC2)[nH]1 79655,N1(C(COC)=O)CCC(NC(=O)C(C)Cc2ccco2)C(F)(F)CC1 79656,N(C1CC2(CN(C(=O)Cc3cccnc3)C2)n2ccnc21)C(C(CC)(C)C)=O 79657,c1(NC(c2c(C)cco2)=O)cccc(C(=O)NN2CC(C)C(O)C2)c1 79658,c1(NC(C(CC2CC2)NC(C2C(C=C)OCCC2)=O)=O)cccc2cnccc12 79659,c1(C(=O)NC2C(n3cc(CN(C)C)nn3)COC2)cc(Cl)ncc1Br 79660,C(=O)(NN=c1cc[nH]cc1[N+](=O)[O-])C1(Sc2onc(C)n2)CC1 79661,c1(C2CCN(S(C)(=O)=O)C2)cccc(OC(F)(F)F)c1.N12CCCC1(C)C2=O 79662,C1(C(=O)NC(CC#C)(C)C)(CC)CCCN1C(=O)CC(CC)SC 79663,CN(C)NC(=O)CCC(=O)NCC(CC1CCCC1)C(=O)N1CCC(C)(F)C1 79664,C1(NC(=O)C(=O)NC(C)(COCC2CC2)CNCC)CCCCC1CC 79665,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 79666,c1(CNCC2C3CN(C(C(C)OCC4CC4)=O)CC32)nnn2ccccc12 79667,C1(C(=O)NCCCCOC)CCOCC1NC(=O)C(C)(F)F 79668,N1(C(CC=C(C)C)=O)CCC(CNC(=O)C=Cc2cscn2)CC1C 79669,Cc1ccc(C)n1CC(N1CCOC(CNC(C2(C3CC3)CC2)=O)C1)=O 79670,CCCC(F)C(=O)NCCC1CCN(C(c2ccc(C)cn2)=O)CC1 79671,n1(CC(=C)C)nnnc1C(c1ncnn1C)NCC1CC2(CC2)C1 79672,S(=O)(=O)(c1ccc(C(=O)NCC(C)CNC(C2CCC(OC)CC2)=O)o1)NC 79673,Cc1ccc(NC(=O)CN(c2ncc(F)cc2C)CCN2CCCCC2)c(Cl)c1 79674,N1(C(c2cncc(OC(C)C)c2)=O)CC(C)(C)CCC1CNC(C1CCSC1)=O 79675,N1(C(COC2CN(C(C(CC#C)O)=O)C2)=O)CCOCC(O)C1 79676,N1(C(CC(c2cccc(Cl)c2)C)=O)C2CCC(C2)C1c1ccccc1 79677,c1(C2N(C(c3cc(C(C)C)no3)C(=O)NCCCCC)CC2)ccccc1F 79678,O=C(C1CCCc2n[nH]cc21)NC1(CF)CCN(C(=O)C(F)(F)C2(O)CCC2)C1 79679,c1(C(=O)NC(CCCC)CNC(=O)C(N2CCCCC2)C)cncc2nc[nH]c12 79680,NS(=O)(=O)c1n[nH]cc1C(N1CC2(CCC2NC(=O)CCCn2ccnc2)C1)=O 79681,Cc1cnc2cc(C(N3CCOCC3CNC(=O)CCc3cnoc3)=O)ccn12 79682,C(=O)(C1=CC2(CN(C(=O)C(C(CC)CC)OC)C2)OC1)N1C(C#C)CCCC1 79683,C(=O)(C(CNC(=O)CNC(=O)C(C)(C)C)C(C)C)Nc1c(CC)noc1C 79684,C1(N(C(c2cc(COC)[nH]n2)=O)CC)CCCN(C(=O)COCCC(C)C)C1 79685,c1(C(CC)(C)NC(C2CN(C(=O)NCCC3(C)CCCO3)C2)=O)cn(CC)nn1 79686,Cc1cc(C#N)c(O)nc1C(=O)NCC1CC2CCCCC2N1 79687,C12(n3c(=O)c3=O)CCCN1CCC2.N1(CC)CCC(O)CC1.CCC1CSC(=S)N1 79688,c1(C2OCCN(C(C(=O)NCCCCCC)C3CC3)C2)ccc2ccccc2c1 79689,C1(C(=O)NC)CCC2(CCN(C(C3CC(F)(F)C3)=O)CC2)O1 79690,Cc1cccc(Oc2ccc(C(=O)NC(=O)NC(c3cccnc3)C)cc2)c1 79691,c1(C(=O)NCCCCCCn2cc(C(C(C)C)O)nn2)cccc2cn(C)nc12 79692,CC1(C)OCCC1C(=O)NC1CCC(NC(=O)C(C2CCCC2)C2CCCC2)CC1 79693,C(CC(C(=O)NCC1CSC1)NC(=O)Cn1ncnn1)OC 79694,c1(C(C)C)ccc(F)c(C(N2CC(NC(c3ccnc(C(C)C)n3)=O)C2)=O)c1 79695,C(=O)(C1=CC2(CCN(C(=O)C(C)(C)OC)C2)C1)NCC1CCN(CC)C1 79696,C(=O)(CC(CC)C(F)F)NC(CC#CC)C(=O)NCc1cnc(C)c(C)c1 79697,C1(C2CC2)C(=O)N1C.C12(CCC1)CC2.C(=O)(CCC1CCC1)C(C1CC1)CC1CCC1 79698,C=CC(C)(C)CC(=O)NC(C1CCCCN1C(c1ncccc1NC(C)=O)=O)C 79699,c1(C(=O)NCC23OCCC(NC(C(C)SCC)=O)(C2)C3)cncc2c[nH]nc12 79700,c1(C(=O)NC2C(NC(C3(C)CC3(F)F)=O)C2)cc(N=S(C)(C)=O)ccn1 79701,N1(C(C2CC(OC)C2)=O)CC2CC1CN2C(C1CC=C(C)CC1)=O 79702,N1(C(C(C(C)C)SC)=O)CCCC2(C1)CN(C(c1cccc(O)c1F)=O)CCO2 79703,C123CCC(CC1)(CC2)CNC3=O.CC(O)C(C)(C)C(=O)N(CCN(C)C)C1CC1 79704,CC1(CNC(c2cc(N)ccn2)=O)CCCN(C(=O)C=CCF)C1 79705,CC1(C)CN(C(C23CC(F)(C2)C3)=O)C(CNC(c2n[nH]c3c2CC2CC32)=O)CO1 79706,c1(C(=O)NCC(C)(C2CC2)NC(=O)CCCC#N)cc2cncn2c(O)n1 79707,c1(C(N(CCC)CCNC(=O)CC(C)(C)C#N)=O)cc2nc[nH]c2cc1F 79708,c1(C(N2CC(c3cn(C(CC=C)CC)nn3)(O)C2)=O)nccc(C(=O)O)n1 79709,C1(NC(CC(CC)C)=O)CCOC12CCN(C(=O)C(C)OC)CC2 79710,C1(C(=O)NC(C2(O)CN(C(=O)CN(S(C)(=O)=O)C)C2)C)CC1[N+](=O)[O-] 79711,c1(CN(C(NNC(c2cccc(OC)c2)=O)=O)C)ccc(S(C)(=O)=O)cc1 79712,c1(CCCCOC(C2CC(C(OC)OC)C2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 79713,C1(C(=O)NCCCN(C(c2cncc(N(C)C)n2)=O)CC)CCCCC1C1CC1 79714,N1(C(CCC(C)(C)OC)=O)CCC(C(=O)NC(CC)C(C)CN(C)C)CC1(C)C 79715,Cc1nc(NC(C2CNCCN2Cc2ccc(CO)c(F)c2)=O)ccc1C(F)(F)F 79716,C(=O)(C(C(C)CC)NC(N)=O)N(CCN(C(CC(=C)Br)=O)C)CC 79717,Cc1ccc(O)c(C(=O)N(C(C)CNC(=O)C=Cc2cccnc2)C)c1 79718,c1(OCC)ccc(C(=O)NCC2CC(NC(C3CC3c3ccsc3)=O)CCO2)cc1 79719,C1(CNC(c2c(C)nco2)=O)COCCN(C(c2cc(Br)n(C)n2)=O)C1 79720,C(=O)(C1CCc2cc(C)ccc21)N1CC(CNC(C=CC=CC)=O)(COC)C1 79721,C(CC(=O)NOCCC(C)C1CC1)C1CC(NC(C2(C(=O)OC)CC(F)C2)=O)C1 79722,c1(C(N(CCOCCCN(C)C(c2cncn2C)=O)C)=O)c[nH]ccc1=N 79723,O(NC(=O)C(O)Cc1ccccc1)CC(=O)N(C1CCCCC1)C 79724,c1(C(N2CC(NC(CCC(=O)NC)=O)C(F)CC2)=O)cc(C)cc(OC)c1C 79725,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 79726,c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CCCSS3)=O)C2)C)cn1 79727,c1(C(=O)NCC(C2CCC2)NC(C2CC3CC2CC3O)=O)ccn2ncccc12 79728,Cc1nc(N2CCCCC(CNC(=O)CC(C)C)C2)c2c[nH]nc2n1 79729,CC(N=c1cc[nH]cc1S(=O)(=O)NC(c1c(F)ccc(Cl)c1F)C)C1CC1(C)C 79730,c1(C(=O)NCC2C(CNC(C3(SCC)CC3)=O)C2)c(C)cc(Br)cc1C 79731,CCCC(C(=O)OC)NC(=O)C(C1CCC1)NC(c1cnccn1)=O 79732,C(C(N=[N+]=[N-])C(=O)N(CCCCCCOC(C)=O)C)OCC.C12CCCN1C2=O 79733,N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCC(CC)CC2)=O)CC12CCC2 79734,N1(N2C(C(C)C)SCC2C(=O)O)CCC(N)c2c(Br)cccc21 79735,CC(C)C(CC1CCCC1)C(=O)NCC1CCCN1C(=O)CCc1ccc(O)cc1 79736,N1(C(C(C)(C)CCl)=O)CC2(CCC(N3CCc4ccc(Cl)nc4C3)CC2)C1 79737,c1(SCC(=O)Nc2n(C)ccc2)ccc2nccnc2c1.c12noc(n1)C2 79738,C1(NC(c2ccc(CCCCC)o2)=O)CCSC12CN(C(C1CCCN1CC)=O)C2 79739,C(c1ccc([N+](=O)[O-])s1)=CC(N1CC=CC(NC(C(n2ncc(C)c2)C)=O)C1)=O 79740,N1(C(C2CCC2)=O)CC2CCC(C1)N2C(c1cccc(N2CCCC2=O)c1)=O 79741,CC1CCN(C(c2cnn(C)c2Cl)=O)CC1NC(=O)CCCc1ccsc1 79742,C1(COC(=O)Cc2cccnc2O)CC2CC1CC2O 79743,n1(CC)ncc(C(=O)NC(C2CC=CCC2)C(=O)N(C2CC(F)(F)C2)CC)c1C 79744,c1(C(=O)NCc2cc(C(=O)NCC3CC3(Cl)Cl)no2)n[nH]c(C2CC2)n1 79745,N1(C(CC2(OC)CCCC2)=O)CCC(NC(=O)Cc2cncn2C2CC2)C1C 79746,c1(C(=O)NC2CCCCN(C(C(CC)C#N)=O)C2)cc2cc(OC)ccc2cn1 79747,n1(C(C)C(N2CC=CC(NC(=O)CC3CC3(Cl)Cl)C2)=O)cnc2ccccc12 79748,c1(C(N2CCCC(O)(CNC(C(C)CF)=O)C2)=O)ccc2cnccc2n1 79749,C1(C(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)CC12CCS(=O)(=O)CC2 79750,c1(N2CC(NC(C(c3ccc(Cl)cc3)C)=O)C(C#N)C2)ncnc2cnccc12 79751,N1(C(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)CSC(C)C)C2)C1 79752,c1(C(CCC)C)nc(-c2cc[nH]c2)n(-c2ccn(C(C)C)n2)n1 79753,c1(C(N2CCC(C(CNC(CCCC=C)=O)(C)O)CC2)=O)ccnc2[nH]cnc12 79754,C1(CC)(NC(=O)NC(c2ccc(F)c(F)c2F)C)COC(C)(C)OC1 79755,N1(C(Cc2cnc(C)s2)=O)CCC(CNC(c2c[nH]nc2C)=O)C(C)C1 79756,C1(C(N2CCC3(CCC3O)C2)=O)CCC2(CCNCC2)CO1 79757,c1(C(NC(=NC)NCCc2cncc(C)c2)C)nc2c(s1)CCCC2 79758,c1(NC(CC2CC(COC)N(C(=O)C(C)C(=O)OCC)C2)=O)coc2c1CCCC2 79759,C(=O)(C1Cc2ccccc21)N(CCCCNC(=O)Cc1csnn1)C(C)C 79760,N1(CC(=O)NC2(CC(=O)NCC3(CCOC)CCC3)CCC2)CC2CCC1C2 79761,c1(NC(C2CCCN(Cc3ccccn3)C2)=O)ccc(O)cc1O 79762,C1(COC)(NC(=O)CC(C)(C)C2CC2)CCN(C(=O)C2=NOC(C)C2)CC1 79763,CCCCCC(O)CC(=O)NCC12CC(CN1C(=O)C(C1CC1)SC)C2 79764,C12(C(=O)NC3CCN(C(CNC(C(CC)C)=O)=O)C3C)CCC(O)(CC1)CC2 79765,c1(C(N2CCCC(F)(C(=O)NCCC(O)C3CCC3)C2)=O)cc2occc2[nH]1 79766,CC(C)(C)C=CC(=O)NC1(CCNC(=O)C(=O)NCCOCCF)CC1 79767,c1(C(=O)NCCCC(C)NC(C2(CCOC)CCC2)=O)cnc(O)c(OC)c1 79768,S(=O)(=O)(c1ccc(Cl)s1)N1CCN(C(=O)NCc2ccn(CC3CCCO3)n2)CC1 79769,C1(NC(C(CSC)O)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC(O)C1 79770,C=CCC(CC=C)C(=O)N1CCC(F)(F)C(CNC(c2cncn2C2CC2)=O)C1 79771,c1(C(N2C(CC(C)O)CCCC2)=O)cccc2c1COC2 79772,c1(NC(C(=O)NC(C)CNC(=O)COc2ccc(Cl)cc2)=O)cc(F)c(N)cc1F 79773,C1(CC)CCCC1(C)C(=O)NC1CN(C(c2cccc(OC3CCC3)c2)=O)C1 79774,CCCCS(=O)(=O)CC(=O)NC1(CC)CCN(C(=O)C(C)=C2CCCC2)CC1 79775,c1(C(N2CCC(CNC(CCc3n(C)ccn3)=O)C2)=O)ncccc1F 79776,c1(C(N2CCC(C)(NC(C(C)C)=O)C2)=O)cnc(O)c2ccccc12 79777,c1(C(CC)NCc2nc(CNC(=O)OC(C)(C)C)ns2)nnnn1C 79778,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(=O)CC3(C=C)CCOCC3)C2C1 79779,C1(CNC(CC(CNC(c2n[nH]cc2Cl)=O)C2CCC2)=O)CC2CCCC2C1 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80078,N(C1CCCc2nc(C)nc(O)c21)C(C(=O)N(CC(C)OCC)C)=O 80079,CCC(CCCC(=O)NCc1nc(C)c(C)[nH]1)NC(C1(C2(C)CC2)CC1)=O 80080,N1(C(C2(CCC)CCC2)=O)CCC(NC(=O)C(CC)n2nccc2C)C1 80081,c1(C(CC)NC(=O)CC2CN(C(=O)C=Cc3ccccn3)C2)ccc(C)c(C)c1 80082,C1(C(=O)NC23CC(NC(C(C)C4CCCO4)=O)(C2)C3)CCCCN(C)C1=O 80083,C(CC1OCCc2ccccc21)NC(C(N1CCc2cc(F)ccc2C1)C)=O 80084,C(=O)(CC(C)(C)C#N)NCCCC(C)(C)NC(C1(CCCC)CCC1)=O 80085,C1(NC(=O)CCOC2CN(C(C3(CO)CCCCC3)=O)C2)CCN2CCCC2C1 80086,c1(C(N2CC(CCC)N(C(=O)CC=C(C)C)CC2)=O)n[nH]c2c1CCSC2 80087,C1(N(C(=O)Cc2ccsc2)C)CCCN(C(=O)CCn2cccnc2=O)CC1 80088,CS(=O)(=O)c1nc(Cl)cc(=NC(=O)C23CCC(CC2)C3n2ccnc2)[nH]1 80089,C(CCCCC(=O)NCc1cncc(C)c1)NC(C(C)=CC1CC1)=O 80090,N1(C(C(C(C)C)O)=O)CCC(C(=O)NC2CCN(C3CC3)C2=O)C(C)(C)C1 80091,c1(C(=O)NC(CC)CN(C)C(C2(C)CNC(=O)C2)=O)cc(F)cc(F)c1 80092,Cc1ccc2nc(C(N3CCC4CN(C(c5ncn(C)n5)=O)CCC34)=O)cn2c1 80093,c1(C(=O)NC(C(C)NC(c2cc(C)[nH]n2)=O)C(C)C)cc2ccc(Cl)cc2o1 80094,N1(C(c2c(C)nn(CC)c2C)=O)CC(C)N(C(c2cncc(OC)n2)=O)CC1C 80095,c1(CC)oc(C)cc1C(=O)NCCC1(CNC(c2cn(C)cn2)=O)CC1 80096,CCC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)CC1 80097,CN1CCN(C(=O)CCCCC2CC2)CC1CNC(c1cc(C(F)F)nn1C)=O 80098,N1(C(CN2CC(CC)C2)=O)CC(C)N(C(=O)C(c2cncn2C)O)CC1C 80099,CCCC(C)C(=O)N1CCN(CCCN)CC1.C(=O)(CC(C)c1ccco1)C(=O)COC 80100,C(=O)(CC1=CCOCC1)NC1C2CC(NC(CN(C(C)=O)C)=O)CC21 80101,CCC(CC(=O)N1CC(C(C)NC(=O)C(C2CCCCC2)O)C1)SC 80102,c12ncc(cn1)C(N1CCC(C(N)=O)CC1)C(=O)N2.C1(CC)CC1 80103,c1(C(=O)NC(c2c(C)cccc2)CNC(=O)C(C)(F)F)[nH]c2ccc(F)cc2c1C 80104,c1(CC)cc(C(=O)NC2(COC)CCN(C(=O)CCC3CCOC3)C2)cc(C)c1 80105,CCCCCC(O)C(=O)N1CCC(N2CCN(C(=O)C(C)(C)C#N)CC2)C1 80106,C1(CCOC)(NC(=O)COC2CC2(C)C)CCN(C(=O)C(C)C2CCOC2)CC1 80107,c1(SCc2nc(CCNC(=O)Oc3ccccc3)on2)ccnc(C2CC2)n1 80108,N1(C(c2c(C)n(C)nc2)=O)CCC(C)N(C(C2CC3CCC2CC3)=O)CC1 80109,c1(NC(COCCCC#C)=O)cn(C)c(C(=O)NC2(OCC)CCSC2)n1 80110,c1(NC(C2C3(CCN(C(C(C)(C)Br)=O)C3)C2)=O)ccn2cnnc2c1 80111,c1(NC2CCN(CC)CC2)ccc(S(=O)(=O)NCC2CSC2)cc1Br 80112,C1(C(=O)NCc2ccc(C(N3C(C(C)(C)OC)CCC3)=O)o2)CSCC(=O)N1 80113,CCCCC(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CN(C)C(C)C 80114,N1(C(CCc2scc(C)n2)=O)CCC(C(C)NC(=O)C(F)(F)C2CCCC2)CC1 80115,C12(C(N(CC(COC)O)C)=O)CCC(CC1)N(C(c1nc(O)sc1C)=O)C2 80116,C1(NC(C(COC)NC(=O)Cc2cc(C)n(C)n2)=O)CC2C(O)C(O)CC12 80117,c1(C(N2CCN(C(C3CCC(=O)NC3)=O)CC2CO)=O)noc2ccc(Cl)cc12 80118,Cc1nc(CO)ncc1NC(C1(CCNC(C2(C)COC(=O)N2)=O)CC1)=O 80119,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(c2ccncc2N)=O)CCCO1 80120,Cn1nnc2cc(C(=O)NCCC(O)CNC(c3cc(C4(C)CC4)n[nH]3)=O)sc12 80121,N1(C(C(C)O)=O)CCC(CO)C(NC(=O)Cc2c(Cl)cnn2C)C1 80122,c1(C(N2CCC(N(C(CC)=O)CC)C2)C(=O)NC(C)(C)CC)nn(C)c(C)c1Cl 80123,Cc1ncc(C(=O)NC(C(=O)N(C2CCNC2=O)C)c2ccoc2)o1 80124,Cc1cc(F)cc(F)c1CN1CC2CN(C(=O)CCc3ccc(O)cc3Br)CC12 80125,C1(C(=O)OCC)CCCCCCN1C(c1c(N)cccc1F)=O 80126,N1(C(C2CC(C)CC(C)C2)=O)CCCN(C(=O)CCSc2ccccn2)CC1C 80127,c1(CC)cc(C(=O)NC2(CNC(=O)C=NO)CC2)ncn1.c12ccc(cc1)[nH]2 80128,C(=O)(C(C)(C)CCSC)N1C(C(N(CC(=O)OC)CC(C)C)=O)CC(F)C1 80129,C(C)(C(=O)N1CCCC(N(C)C(c2cnc3sccn23)=O)C1)(C(C)C)OC 80130,C1(C(N2CCC(C(N3C(COC)CC3)=O)C2)=O)CC12CCCCC2 80131,CC1CCN(C(C2CCCCCN2C)=O)C(C(=O)N(C)Cc2ncnn2C)C1 80132,C1(NC(c2ccc(SCC)nc2)=O)Cc2ccccc2C1NC(=O)C(O)O 80133,C12(CC(=O)NC3(CN(C)C)CC3)CCC1CN(C(c1ccc(O)cn1)=O)C2 80134,N1(C(C#CC(C)(C)C)=O)CCCCC12CN(C(=O)C(=C1CCCCC1)F)C2 80135,c1(CC(=O)N(CC(C)NC(C(C)OCC)=O)C)c(F)cccc1Cl 80136,N1(C(Cc2c(C)noc2)=O)CCN(C(=O)C2=NOCC2)CC1CF 80137,C1(OC)CN(C(=O)C=CSc2nc[nH]n2)CC1NC(=O)Cc1ccc(F)nc1 80138,c1(OCCN(C(CC(=O)OCC)=O)C)ccc2c(c1)OCCC2 80139,CCC(C)CCN=c1ccc(S(=O)(=O)N2CCC(Cl)=C(Cl)C2)c[nH]1 80140,c1(C(=O)NCC#CCNC(C(CSC)OC)=O)cccc2c1OCCO2 80141,c1(C(=O)NCC2OCC(C(N(C(C)C)CC)=O)C2)ccc2cc[nH]c2c1 80142,C1(C(=O)NCC2CN(C(c3ccnc(CC(C)C)n3)=O)C2)CC2CCC1C21CC1 80143,C(=O)(C(O)(Cc1ccccc1)C(F)(F)F)N(CCNC(C=CC(CC)=CC)=O)CC 80144,c1(CN(C=O)Cc2nnnn2C)c(OCC2C(C)COCC2)cccc1Cl 80145,N1(C(CNC(=O)CNC(c2ccnn2CCF)=O)=O)CCc2n[nH]cc2C1 80146,C(c1nnc(C(C)C)o1)=CC(=O)N(CCN(C(C)=O)CC)CC 80147,Cc1cc(C(N2CCC(C(C)(C)C(=O)NCCN(C)C)C2)=O)c(C)cn1 80148,C1(C(N(C)Cc2c(C)nsc2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 80149,CC#CCCC(=O)N1CCC(NC(c2cc(C(C)=O)cs2)=O)C1C1CC1 80150,C(C(N=[N+]=[N-])C(=O)NCC(C(C)C)NC(c1ccncc1O)=O)OCC 80151,c1(NC(C2(C)CCN2C(=O)Cn2cccn2)=O)cc(Cl)ccc1I 80152,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CCN(C(c3nc4ccccn4n3)=O)C2)C1 80153,C(C)(C)(C(C)(C)CO)N(CC(=O)NCC)C(c1nc(CCC)oc1)=O 80154,c1(CNC(CCCC)(C)c2nnnn2C2CC(F)(F)C2)ccc(O)c(Br)c1 80155,c1(CCNC(=O)Nc2ccnc(N3CCOCC3)c2)ccc(F)c(F)c1 80156,Cn1cnc(C(=O)NC(C)(C)CCCNC(=O)CC2CC3CCC2C3)cc1=O 80157,C1(CNC(C2C(C(=O)NCC#C)C2)=O)CCN(C(C2CCOC2CC)=O)C1(C)C 80158,c1(CCNC(C2CCCOC2)C)ccccc1 80159,c1(C2(C(=O)NCC(CN(C)C(c3sccc3F)=O)(C)C)CC2)ccnc(Cl)c1 80160,C1(N(C(C(C(CC)O)C)=O)C)CC2CCC(C1)N2C(c1ncc[nH]c1=O)=O 80161,C(=O)(C1=CCC(NC(=O)C(C)NC(C)=O)C1)N(C(C(=O)NC)C)C 80162,C1(C#N)(C(=O)NCCN(CCCCCC)C(C2CCO2)=O)CCOC1 80163,C1(CNC(C(c2cn(C)nc2)(F)F)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C1(C)C 80164,c1(C(CC)NC(=O)NC23CC(C(N(C)C)=O)(C2)C3)nc(Cl)sc1Cl 80165,N1(C(c2cn(C)nc2)=O)CCC2CCN(C(C34COCC3C4)=O)CC12 80166,CC1CC(CNC(C2CC2F)=O)CN(C(=O)C=C(C2CC2)C2CC2)C1 80167,C1(NC(c2cccc(CC)n2)=O)CCCCCC1C(=O)NOCC(C)O 80168,CC(C)CC(C(=O)NCCCC1CCCCC1)ONC(c1cscn1)=O 80169,c12cc(ncc1Cl)OCCN2C.CCC(C)(C)C(=O)N1CCC(NCC)C1 80170,c1(C(C)(C)NC(c2c(CC)ncs2)=O)cccc(Br)c1O.C12CCCN1C2=O 80171,c1(N2CC(C)N(C)C(C)C2)nc(N2CCC(COC(F)F)CC2)nc2c1CCCC2 80172,c1(C(N(C2CCN(C(=O)COC(c3nccn3C)C)C2)C)=O)cc2occc2[nH]1 80173,c1(N(C)C)ccnc(CC(=O)NC(CNC(=O)COC2CCCC2)CO)n1 80174,c1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC2O)nc(Cl)ccc1OC(C)C 80175,C(CC(F)F)(C(=O)N1CC(CS(C)=O)C1)NC(C(CC)OCC)=O 80176,c1(COC)ncc(C(=O)NCC(CO)NC(C23CC(CCO2)C3)=O)c(O)n1 80177,C1(OCC)CCCCC1C(=O)NC(C)C(=O)NCc1c(C)noc1C 80178,c1(C(=O)NCC2(F)CCC(NC(c3c(C)cno3)=O)C2)cn(C)c(=O)nc1O 80179,C12(C(N3C(C)CN(C(c4ncc(F)cn4)=O)CC3)=O)CCC(C)(CC1)CO2 80180,c1(-c2cncc(OC)n2)ccc(F)c(C(=O)NC(c2ccno2)C)c1 80181,C1(NC(c2cnc(Cl)s2)=O)CCCCCC1C(N1CC(Cc2ccoc2)C1)=O 80182,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC(C)CN2CCOCC2)C1 80183,C1(CNC(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(C23CCCC2C3)=O)C1 80184,n1(C(C)C)ncc2c(N3CC(F)C(F)C3)[nH]c(=NCC3C=CCCCC3)nc12 80185,c1(C(=O)NCCC2CCN(C(C(C)N(C(C)=O)C)=O)C2)onc2c1CCCC2 80186,C1(C(=O)NCC(CNC(C(CC)SC)=O)O)Cc2ccccc2N(C)C1=O 80187,N1(C(CN(C(CCSCC(C)C)=O)CC2CC2)=O)CC(C2CCCC2)C1 80188,C1(C(=O)NCCC2CN(C(c3ncc[nH]3)=O)C2)CCc2nnnn2C1 80189,Cc1ccc(CC(=O)NC(CNC(c2scnc2C(F)F)=O)CC(C)C)cc1O 80190,CC1CC(=O)NCC1C(=O)NC(C)(C)CNC(C1CCC(C(N)=O)C1)=O 80191,c1(C(N(CCCNC(=O)CC2CCOC2)CC)=O)ccc(-n2ccnc2)cc1 80192,c1(NC(CC2(C)CN(C(CC(C)C)=O)C2)=O)c(F)ccc(Br)c1F 80193,C#CC(CNC(C1CN(C(=O)C(C)(C)C)CCN1)=O)CC(C)(C)C 80194,c1(CC(=O)NCCC(=C)CNC(C2CCCNC(=O)C2)=O)ccc2c(c1)OCO2 80195,C(CCC(C)C)(C(=O)NCc1nc(=O)o[nH]1)NC(C(C1CC1)OCC)=O 80196,c1(C(=O)OC(c2ccccc2)C(=O)OCC)ccnc2[nH]cnc12 80197,CC1OCCCC1C(=O)NC12CC(C(=O)NCC3CC(O)C3)(C1)C2 80198,N1(C(CCN(C(=O)C(C)SCC(C)C)CCOC)=O)CCCCCCC1 80199,C(=O)(CC(C(C)C)NC1CCC(=O)NC1)OCC 80200,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)OCCNC(C2CC23CCOC3)=O)c1 80201,C1(C(N(CC(C)NC(=O)C(C)(C)COC)CC)=O)CCC(=O)CC1(C)C 80202,c1(C(N(CCCCCCC=C)C)=O)ccc(O)c([N+](=O)[O-])c1 80203,Cc1cc(C)cc(C=CC(N2CC3(CCCC3NC(=O)C(F)C3CCC3)C2)=O)c1 80204,C1(CC(=O)NCCN(C(=O)CCC(F)(F)F)C(C)C)CC2(CCCC2)CO1 80205,C1(C(=O)NCC(=O)N(CC(C)(C)C)C(C)C)CN(C(=O)OC(C)(C)C)CCC1C 80206,Cc1cc(NC(C2(C)COC(=O)C2)=O)ccc1NC(=O)C(=Cc1cccc(F)c1)F 80207,N1(C(C(C(C)C)C#N)=O)C(C)CC2CN(C(c3sccc3OC(F)F)=O)CC12 80208,N1(C(COCC)=O)CC2CC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 80209,Cc1ccc(OC(C)C)cc1C.N12CCC(CC1)OC2=O.C12CC1C(=O)N2 80210,c1(C(=O)NCC(C2CCC2)N(C(C(C)N(C(C)=O)C)=O)C)ccc(CO)s1 80211,C1(CC(=O)NC2(CCC)CCC2)CCCN(C(C2C3CN(C)CC23)=O)CC1 80212,N1(C(n2cc(-c3cnn(CC4CC4)c3C)nn2)=O)CC=CC1(CO)CC1(C(C)(F)F)CC1 80213,c1(OC)cccc2c1C(C(=O)N1CCCC1CN(C)C(C1(CF)CC1)=O)CC2 80214,Cc1nn(C)c(C)c1C1CC1NC(C1(C(F)(F)F)CCOC1)=O 80215,CC1(C)C2CCC1(C(N1CCCC(CC(=O)N(CC3CC3)CC3CC3)C1)=O)C2 80216,CC(C(C)(C)C(=O)NCCCN(C)C)NC(=O)Cc1ccco1 80217,c1(C(N2CC(CCNC(CNC(C)=O)=O)C2)=O)ccc2c(c1)C(=O)NC2 80218,CCCCC(CNC(c1n[nH]c(C)n1)=O)NC(c1cnccc1Br)=O 80219,CC1CCCCC1(C)C(=O)N(CCC(=O)Nc1cc(Cl)ncc1Cl)CCO 80220,N1(C(=O)CCN2CCOCC2)CC2CS(=O)(=O)CC2(NC(c2cn[nH]c2)=O)C1 80221,C12(C(N(CC(C)CNC(C3CC(C)(O)C3)=O)C)=O)CC(CO)(C1)OC2C 80222,C1(C(=O)NC(CC#C)CO)CC(NC(c2cccc(F)c2)=O)C1(C)C 80223,N1(C(=O)OCC)CSCC1C(=O)NCC(C)CO.C1CC(=O)N1 80224,C=CCCCCC(=O)N1CC(CO)(NC(c2nc(C)n(C3CC3)c2C)=O)C1 80225,C(=O)(CCCCCCCC1CC1)N(C1CCCN(C(C(CC)=CC)=O)C1)CC 80226,C1(CC=C)(NC(=O)Cc2ccnn2C)CCN(C(=O)CCc2ccoc2)C1 80227,C(C)(CCC=C(F)CNC(=O)NCCC1CC1)=CC 80228,S(=O)(=O)(c1cc2c(cc1OC)CCC2)NC(c1cnc(SC)s1)C 80229,c1(CNC(C(C2(C)CC2)NC(C2C3CCCC(=O)C23)=O)=O)ccc(F)c(O)c1 80230,Cc1c(OCCC(N2CCN(c3ccccc3C(F)F)CC2)=O)cccc1F 80231,N1(C(C(CCN)c2ccccn2)=O)CCOC2CS(=O)(=O)CC12 80232,N1(C2CCN(C(C(C)(C)NC(C3CCOC3C3CC3)=O)=O)C2)CCCOCC1 80233,Cc1cccc(C(N2CCCC(NC(C3CCC(CO)CC3)=O)C2)=O)c1Br 80234,C1(N(C)C)CC(CC(=O)NCCOCCNC(=O)C(F)n2cccn2)C1 80235,S(=O)(=O)(c1ccc(OC)cc1C)NC(C1(CO)CN(C(C(CCC)O)=O)C1)=O 80236,C1(CNC(CN(C(C)=O)C)=O)(CNC(C2C(C)(C)C2(C)C)=O)CCOCC1 80237,c1(C(C)=O)ccc(N2CCCC2)cc1.c12ccc(o1)NC(=O)CC1CN(C1)C2=O 80238,C(c1nnc(C(C)C)o1)=CC(=O)NCC(C1CCCC1)NC(C)=O 80239,C1(C(N(CC)Cc2nc[nH]n2)=O)CC12CCN(C(=O)C=Cc1cncs1)C2 80240,Cc1ccc(C(=O)NC2CCCC(NC(=O)CCC3CCOC3)C2)nc1O 80241,N12CC(NC(C3(C)CCC(C)C3)=O)C(C1)CNC(=O)C1(CCC1)CC2=O.CCO 80242,C(=O)(C(CC(F)F)c1ccccc1)NC(C)(C)CNC(C1SCCS1)=O 80243,N1(C(C(C(C)C)OC)=O)CCC(C2CN(C(c3cc(OC)ns3)=O)C2)CC1 80244,CCCC(C)(CC)C(=O)NC1CC(N(C)C(c2cc3occc3s2)=O)C1 80245,c1(OC)cccc(C(C(=O)NCC2CC2)N(C)Cc2ccsc2)c1Br 80246,C#CC1CN(C(=O)CCSCC)CCN1C(C1CCOC(=O)N1)=O 80247,c1(C(N(C)CC2(NC(C3CN(C(C)=O)C3)=O)CC2)=O)csc([N+](=O)[O-])c1 80248,C(=O)(C(F)CC1CCCC1)NCC(C)N(C(=O)CC1CCCCO1)C 80249,C1(c2nn[nH]n2)(NCc2c(CSC(C)(C)C)ccs2)CC2(CCC2)C1 80250,c1(NC(C(=O)NCC(CC)(CC)CO)=O)ccc2c(c1)CNC2 80251,c1(CCC(=O)NC(C2CCN(C(Cc3nnc(C)o3)=O)C2)C)ccc(C#N)cc1 80252,Cc1cc(C(=O)NC2CCC(CNC(=O)COC(C)(C)C)CC2)cc(F)c1C 80253,CN=O.C1CCN(CC2CC2)CCN1C(C1CCC1)=O 80254,C1(C(N(CC(C)NC(c2c(CCC)nco2)=O)CC)=O)CCCCC1O 80255,C12(NC(Cc3scc(C)c3)=O)CCCC(NC(=O)CC(C)(C)O)(C1)C2 80256,c1(C(C)NC(=O)COC2CCCCO2)cnc(OC)c(Br)c1.c1(S)ccccc1Br 80257,C1(C(N)=O)CCCCC1C(=O)NC(CNC(=O)COc1cccc(Cl)c1)CO 80258,c1(C(N(CCOC)CC2CC2)=O)cc2c(s1)CC(C)(C)C2 80259,C=C(C)CCCC(=O)N1CC(c2ccccc2)(CNC(=O)CC2CNC(=O)O2)C1 80260,N1(C(COCc2cc(C)on2)=O)CCSCC1C(=O)Nc1cc(C(C)C)no1 80261,Cc1csc2nc(CC(=O)NC3(C)CN(C(=O)NC4COC5COCC45)C3)cn12 80262,C(CN=c1[nH]c(=NCc2cccnc2C)[nH]c2c1COCC2)OCC 80263,c1(C(=O)NC(C)C(=O)N(C2CN(C(N)=O)C2)C)cnc(CCn2cccn2)o1 80264,c1(C(=O)NCC(C)=CC(=O)NCCc2c(C)noc2C)ccc(F)c2c1CCC2 80265,C1(CNC(c2cc(C)[nH]n2)=O)CCC(C)CN1C(c1cncc(NC(C)C)c1)=O 80266,C(C(C)(C)C(=O)NCC1(F)CCN(C(=O)C(CN(C)C)c2ccccc2)C1)OC 80267,c1(C(=O)NCC2CN(c3nccc(SC)n3)C(C)C2)cccc2cccnc12 80268,c1(NC(C2CCCCC2)C(=O)NCCNC(COCC(=O)OC)=O)nc(C)cs1 80269,c1(C(N2C(CC(=O)N(C)CC3CCC3)CCC2)=O)ccc2ncnn2c1 80270,Cn1nc(C(F)(F)F)cc1C(=O)NC(C)(CNC(C1(CO)CC1(F)F)=O)CO 80271,C1(C(N(CCCNC(C2CCN(C)C2=O)=O)CCC)=O)CCN(C)C1C 80272,c1(C(N2CCN(C(c3cc(OC)ncn3)=O)CC2)=O)ccc(N(C)C)cc1OC 80273,c1(C(C(=O)Nc2cnn(C(C)C)c2)NC(C(COC)OC)=O)ccccc1F 80274,C1(C(=O)NC(CC=C)C)CN(C(c2cc(C)c(N)cn2)=O)C(C)(C)C1 80275,c1(CNC(=O)Nc2ccc(N3CC(C)OC(C)C3)nc2)cn2c(Br)cccc2n1 80276,CC1CC(CNC(=O)C(F)(F)c2cscn2)CN1C(=O)COc1ccc(F)cc1 80277,C1(OC)CCCN(C(C2CC(C)N2C(c2cc(OC)no2)=O)=O)C1 80278,c1(C(=O)NCCc2nc(C)sc2)c(N)sc2c1CCN(C(=O)OC(C)(C)C)C2 80279,c1(C(N2C(C)CC(NC(C(C)OCCC=C)=O)C2)=O)cnc2c(cnn2C)c1 80280,C(=O)(CC(C)C(F)(F)F)N1CC(OCC)C(NC(c2ccc(F)cc2OC)=O)C1 80281,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(CCNC(=O)Cc2cc[nH]c2)C1 80282,C1(C#N)(C(=O)NC(C(=O)OCC)C2CCCO2)CCCC1 80283,N1(C(CCNC(Cc2c(C)con2)=O)=O)CCS(=O)CC1C 80284,CC1(NC(c2coc(CC3CC3)n2)=O)CCN(c2nnco2)C1 80285,C(=O)(C1=CCC(C)(C)CC1)N1CCC(NC(Cc2ccc(CC)cc2)=O)C1C 80286,Cc1cncc2cc(C(N3CC(N(C(=O)C(O)C4CC4)C)C4(CC4)C3)=O)sc12 80287,Cc1ccccc1CC(=O)NCC1(NC(c2cc(-c3ccccn3)ns2)=O)CC1 80288,C1(C(N2CCCCC2Cc2cn(CCCCO)nn2)=O)(CN(C)C)CCCCO1 80289,c1(C(=O)NCC(N2CCC(CNC(C3(C)CC3(F)Cl)=O)C2)=O)cccc(O)c1 80290,N1(c2nc(C3CN(c4c(CC)cccc4)C(=O)C3)n(C)n2)CCC2(CCCO2)C1 80291,C1(C(=O)OC)N(C(=O)C(CN(C)C)NC(C2(C(C)(F)F)CC2)=O)CC1(C)C 80292,C(CC(C)C(=O)NCC1(NC(=O)C(N2CCCCC2=O)C)CC(F)(F)C1)OC 80293,C(=O)(CC1=CCCC1)NCCN(C(=O)CCc1ccc(Br)nc1)CC(C)O 80294,C1(NC(C=C(C)Cl)=O)CC2CCC1N2C(=O)CCCN1CCOCC1 80295,N1(C(CCN(C)CCO)=O)CC(NC(c2cn(C(F)(F)CO)nn2)=O)C(O)C1 80296,C1(NC(=O)CCC2CCCC2)CCN(C(=O)C2=CCOC2)CC1O 80297,N1(C(CCn2c(C)nc(C)n2)=O)CCCC(C)(CNC(C2CC3(C2)CC3F)=O)C1 80298,C1(CNC(C2(CCCC)CCC2)=O)COCCN1C(=O)CCC1CCCCO1 80299,C1(CNC(=O)OCC)CCCC1(CC(C(=O)OC(C)(C)C)c1ccccc1)OC 80300,Cc1nc(C(=O)NCCC2(NC(=O)CSCC(F)(F)F)CCC2)cn(C)c1=O 80301,C(CCC(C(=O)NC1(CCF)CC1)NC(=O)CC1CCC(C)CC1)OC 80302,N1(C(C2(CC=C)CC2)=O)CC2CC1CN(C(=O)C(COC(C)(C)C)NC(C)=O)C2 80303,Cc1cc(C(N2CC3(CCC3NC(C3C=CCC3)=O)C2)=O)ncc1C#N 80304,CC(C)(C)C(O)C(=O)N1C2CCC1C(NC(c1cnc(S)nc1)=O)C2 80305,O=C1COCC2(CN(C(=O)CC3CC4(CC4)CN3C(c3cc(Cl)ccn3)=O)C2)N1 80306,C1(NC(C2C(C)C2)=O)CC2(C1)CN(C(c1cnn(-c3ccccc3F)c1N)=O)C2 80307,n1(C(C)C)cnc(CNC(=O)COCCNC(C2CCCC2O)=O)c1 80308,C(=O)(C(O)CC(F)(F)F)NC1(CO)CCN(C(CCCc2ccc(C)s2)=O)C1 80309,C#Cc1cccc(NS(=O)(=O)CC2CCCC(CC(=O)OC(C)(C)C)C2)c1 80310,c1(C(=O)NC(C)CNC)cccc(N(C)C(C2C3CNC(=O)C23)=O)c1.C(N)(=O)N 80311,c1(NC(c2nccc(-c3ccc(C)nc3)c2)=O)cc(S(C)(=O)=O)ccc1C 80312,C1(C(=O)OCC)COCCN1C(C1(C)CCN1C(C1CC=CCC1C(F)(F)F)=O)=O 80313,C1(NC(C2(COC)CCCN2C(=O)C(O)CCN(C)C)=O)CC=C(C(C)C)CC1 80314,C1(NC(C2C(CNC(C3(CC(C)C)CC3)=O)CC2)=O)CN2CCC1CC2 80315,N1(C(C(CNC(CSCC)=O)CC2CC2)=O)CC(C)CC(O)C1.C1(C)CC1 80316,N1(C(C(C)c2cc[nH]n2)=O)CC2CCN(C(c3nnn4ccccc34)=O)C2C1 80317,c1(C(=O)NC2CCC(N(C(C3(C#C)CCCC3)=O)C)CC2)cnc(O)c(Cl)c1 80318,C1(C(=O)NCc2oc(C(=O)NC(COC)C)c(C)n2)CCCC(=O)N1C 80319,C(=O)(CC(C)CC(C)(C)C)NC1OCCN(C(CN2CC(C)(OC)C2)=O)C1 80320,C1(OC)CC(C(=O)NC2CC2(C)C)N(C(=O)Cn2c(O)nnc2O)C1 80321,N1(C(CCC(=O)N(C)C)=O)CCCC(C)(CNC(=O)CC(O)CN(C)C)C1 80322,c1(C(=O)NC(C(C)C)CNC(=O)Cc2cccnc2)cc2cccc(O)c2n1C 80323,N(C1CCc2cc(-c3ccc(F)c4c3OCC4)ccc21)C(C(CC)Cl)=O 80324,c1(OC)cc(C(=O)N(C(C)CCNC(=O)C(c2ccccc2)F)C)c(F)c(Cl)c1 80325,c1(C(N2C(CNC(CCc3ccn(C)n3)=O)CC2)=O)nnn2c1COCC2 80326,C1(O)(CC(=O)NC(C2CCCN(C(c3scc(C)c3)=O)C2)C)CCCN(C)C1 80327,C=C(Cl)CC(C(=O)N1CC(F)(F)CC1C)NC(C1CCC(CC)C1)=O 80328,C1(C(=O)NCC2(C)CC(NC(=O)C(c3ccccc3)O)C2)CC2CCC1C2 80329,C1(C(N2C(CCNC(C3N(C(C)=O)CCC3)=O)CSCC2)=O)CC2CC1C1CC21 80330,C1(C(=O)NCC2CC(NC(CS(=O)(=O)NC)=O)C2)CCCC2C1C2(F)F 80331,O(N1CCC(CC(=O)N(CC(O)CN(C(=O)Cc2nc[nH]n2)C)C)CC1)CC 80332,C1(N(C(=O)C=CC2CCCN2C(=O)NC(C)(C)C)C)CCc2c[nH]nc2C1 80333,c1(C(=O)NC2CC2NC(c2nn[nH]c2Cl)=O)cc(F)cc(Br)c1 80334,O=C(CCC(F)(F)C(F)(F)F)NC1CCCCC1C(N1CCC(O)C1)=O 80335,C1(CNC(C(C)=C(CC)C)=O)COC(C)(C)CN1C(C1CCCCC1)=O 80336,C1(C(N2CC(NC(COC)=O)C2)=O)CCN(C(=O)CCC(C)(C)N(C)C)C(C)C1 80337,N(C(=NCCC1COC(C)(C)C1)NCC(C)(C)OCCN(C)C)C(C)C 80338,Cc1nc(O)ccc1C(=O)N(C1CCCN(C(=O)COCP(C)(C)=O)CC1)C 80339,Cc1ccc(CC(CNCCC(=O)OCc2ccc(C(=O)N(C)C)o2)(C)C)cc1 80340,C(=O)(C1Cc2ccccc21)N1CC(NC(c2coc3c2COC3)=O)C(O)C1 80341,C(N=C(NCc1ccccc1)N1CCC2CCOCC2C1)c1cnco1 80342,CC(CCC(=O)NC1CN(C(C2CC2Br)=O)C1)N(C)C 80343,CC1(CNC(=O)CCOC2CCOC2)CCN(C(=O)C(F)n2ccnc2)CC1 80344,C1(C(=O)N(C2CCCCC2)CCO)CCCC(NC(c2cn[nH]c2)=O)C1 80345,CC(O)CCCCCC(=O)NC(C)CCNC(c1c(F)cc(C(F)(F)F)cc1F)=O 80346,C1(C(N(C2CCN(C(CC)=O)C2)C)=O)CN(C(C2CN(CC)C2)=O)CCO1 80347,C(=O)(CC(C(F)(F)F)NC(c1cc(C2CC2)ccc1F)=O)N(C(C)C)C 80348,C12(NC(c3occ(C(=O)OC)c3)=O)CCCN(C(C3CC(=O)N3)=O)CC1C2 80349,c1(C(N(CC(C)NC(c2cccc(SCCC)c2)=O)C)=O)cnn2c1CCCC2 80350,N1(C(C(=O)OC(c2ccc(C)cc2)C)C)C(C)CCCC1C 80351,S(=O)(=O)(c1cccc(-c2cccs2)c1)N1C(CN(C)C)CCCC1 80352,C1(CCNC(c2nn(CC)c(C3CC3)c2)=O)CCCN(C(=O)C(N)=O)CC1 80353,c1(NCC2CCN(C(CC#C)=O)C2)ccc2c(n1)CCC2=O 80354,C1(CC=C)(NC(c2cnc(C)o2)=O)CCCN(c2cc(C)nc(SC)n2)C1 80355,N1(C(C=C(C)C(C)C)=O)CC(CO)C2(C1)CN(C(C1(CO)CCOC1)=O)C2 80356,CCC(CCCC(=O)N1CCCC1CN(C)C)NC(C1CC(O)C(F)C1)=O 80357,Cc1oc(C2CC2)nc1CNC1CCOC1C(C)(C)C 80358,C1(CCNC(C(C2CC2)OCC)=O)COCCN1C(=O)C(F)(F)CO 80359,C(=O)(C(CC)C(=O)N1CC=C(CNC(=O)CN2CCCC2CO)CC1)OC 80360,N1(C(c2nnn(CC)c2C)=O)CCC(C(F)(F)F)C(NC(=O)C(C)C2CC2)C1 80361,C1(C(N2CC(SC)C(NC(=O)COC(C)C)C2)=O)Cc2cscc2C1 80362,c1(C(=O)NC(CNC(c2c(CCC)nco2)=O)CCC)cc(N(C)C)ccn1 80363,N1(C(CCOCCC(=O)SC)=O)CCC(C(N(CCOCCSCC)C)=O)CC1 80364,CCC(F)(F)Cn1cc(-c2conc2CC(=O)NC2CCCCO2)nn1.CCC 80365,N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ncccc2F)=O)C(c2ccnn2C)C1 80366,c1(C(N(C)C)C)ccc(Br)c(C(=O)N=C2CCON2)c1N 80367,C1(NC(C(c2cccnc2)N(C(=O)Cc2csnc2C)C)=O)CCC(C(N)=O)C1 80368,Cc1nn(C2CCC2)cc1C(N1CCCC(NC(=O)Cc2cc(Cl)n(C)n2)C1)=O 80369,Cc1cccc(C)c1C(N1CC(NC(c2cc3sccc3[nH]2)=O)C2(CC2)C1)=O 80370,C1(NC(C2(COC)CCCC2)=O)CC(C)CN(C(=O)CC2CCOC2)C1 80371,C1(CC(C)NC(=O)NCC(c2nccs2)C)C=CCN1C(=O)C=C1CCCCC1 80372,C1(NC(=O)CNc2ccccn2)CCSC12CN(C(=O)C1=C(Cl)CC1)C2 80373,c1(CC(C(N2CC(C#N)(C(C)C)C2)=O)C)ccc(F)c(F)c1 80374,C1(C(=O)NC2C(C)C2C)CC2(CCN1C(C1CC(C)(F)C1)=O)CC2 80375,c1(OC(C)C)cnc2c(c1)C(NC1CCN(c3ccccc3F)C1=O)CCO2 80376,C(C1=COCCC1)(n1nnnc1C1(OC)CC(c2ccc(C)nc2)C1)NC(C)C 80377,CC#CCCCC(=O)NCC12CC(NC(=O)CCCOCCC)(C1)C2 80378,c1(C(=O)NCC2C(CNC(=O)CSc3cccc(F)c3)C2)c[nH]c2cccnc12 80379,C1(NC(c2c(CC)nns2)=O)CCC(C)N(C(C2(COC)COC2)=O)C1 80380,CCC(CN(C)C)C(=O)N1CCC=CC1C(=O)NCC(=O)O 80381,C1(NC(C(C)Oc2cccc(Cl)c2)=O)C2CN(CC(=O)N(CCOC(C)C)C)CC12 80382,c1(C(=O)NC2C(NC(c3c(C)nc(Br)o3)=O)CC2)cnc2ccccn12 80383,C1(CNC(c2cc(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)CC(C)C#N 80384,C1(CC(N2CC(C(C(=O)N(C3CCCCC3)CCOC)OC)C2)=O)CCCN(C)C1 80385,C1(C(N2CC(C(N)=O)(CNC(C3CCC(=O)N3)=O)C2)=O)CC2C=CC1O2 80386,C1(NC(c2cc(OC)no2)=O)CCC(NC(=O)C(C)OC2CCCC2)CC1 80387,N1(C(c2ncc(C)s2)C)CCN(CCc2ccccc2)CC1 80388,N1(C(c2cccc(-c3c(C)sc(O)n3)c2)=O)CCC2(CC1)CNC(=O)O2 80389,C1(CC(=O)NCCOCCCNC(C2CC(CC)C2)=O)CCCC2CCCCC12 80390,C1(NC(C2(CC(=O)OC)CC2)=O)C=CC(CC(=O)N(CCCCO)C)C1 80391,C1(C(=O)NC(C2(O)CN(C(c3cc(N(C)C)ccn3)=O)C2)C)CC(C2CC2)=NO1 80392,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1C(OC(c2cn(C3CCC3)nn2)C)CC1 80393,C(=O)(C(C)C(F)(F)F)N(C)CC1N(C(Cn2cc(C(C)O)nn2)=O)CCC1 80394,C1(=O)CCCCNC(=O)OC2CN(C(=O)C#CCN1)C2.C(=O)(C1CC1)OC 80395,N1(C(=O)C=Cc2cc(Cl)cc(Cl)c2)CCOC2(C1)CN(C(=O)COCC(F)F)C2.C 80396,CC(CC(=O)N1CC2(CNC(c3ccc4nnnn4c3)=O)CC1CO2)C(C)(C)C 80397,c1(C(C(=O)NCC(=C)CCNC(C2(C(=O)OCC)CC2)=O)C)cccc(OC)c1 80398,C(=O)(C1CCc2ccccc21)N1C(C(C)NC(c2cncs2)=O)CCCC1 80399,c1(NC(c2ccco2)=O)cc(Oc2ccc(F)cc2C(=O)NC2CC2)nc(Cl)c1 80400,C1(NC(=O)NCc2ncc(-c3cccnc3)[nH]2)CCCCCCC1c1ccccc1 80401,Cc1c(Br)cc(S(=O)(=O)N2CCCC3CN(C)CC23)c(C)c1.c1(CO)ccccc1 80402,c1(C(=O)NC2(CCC(=O)NCC(O)CC(F)(F)F)CCCC2)cccn2nccc12 80403,N1(C(C(C)NC(=O)NC)=O)CCC(Nc2ncc3c(n2)COC3)C2(CCC2)C1 80404,CC(C)(CC(F)C(=O)NC1CC2CC2C1)NC(c1cccc[n+]1[O-])=O 80405,N1(C(c2cn(C)c(Br)c2)=O)CCCC2C(NC(C3CCOC3(C)C)=O)C12 80406,Cc1nn(C)c(C(=O)NCCCN(C)C(C2CCCCN2C)=O)c1Br 80407,N1(C(COCCC(C)C)=O)CCC(CCCNC(C2(C)CCCO2)=O)CC1 80408,C12(C(=O)NC3C4CN(C(=O)Cc5cnn(C(F)F)c5)C3C4)CCCC1CCN2 80409,N1(C(c2n(COC)ncc2)=O)CCC(NC(=O)C(N2CCN(C)CC2)C)C12CC2 80410,CC1(C)CC(NC(=O)Cc2ccc(C#N)nc2)CN1C(=O)CSc1cccs1 80411,N1(C(C=C(CC)CC)=O)CCC(NC(=O)CC2CC2(C)C)C12CCC2 80412,c1(OCC(=O)NC(CNC(c2c(CC)c[nH]n2)=O)(C)CC)nn(C)cc1[N+](=O)[O-] 80413,C1(CC)(CNC(C2CCN2C(c2ccc(C)s2)=O)=O)CCOCC1 80414,C#CCC(C)C(=O)NC1(CNC(=O)CC2CCC(C)CC2)CCCCC1 80415,C(=O)(C1=NNC(=O)C1)NC1C(C(C)C)N(C(=O)CC(C)(C)O)CC1 80416,Cn1ccnc1NC(=O)C(F)(F)Cl.N12CCCC1CNCC2=O 80417,c1(COCC)cnc(N2CC3C(NC(=O)C(C)CCN(C)C)C3C2)nc1C 80418,C(c1cccnc1)=C(C)C(=O)NC(C)CC(C)NC(=O)Cc1ncc(C)[nH]1 80419,Cc1ccc(C(F)(F)C(=O)N(C2CC(NC(c3csc(=N)[nH]3)=O)C2)C)cn1 80420,C(=O)(C(C)(C)C(C)NC(C1CCCSC1C)=O)N1CCC(COC)(OC)C1 80421,c1(NC(c2n(CC)nnn2)C2(OCC)CCC2)cn(-c2ccccc2)nc1C 80422,C(=O)(CC(C(F)F)NC(=O)CCc1csnn1)N(CC)Cc1ccccn1 80423,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)Nc2cnc(C#N)cn2)CCC1(C)C 80424,C1(NC(c2cc(C)c(C)o2)=O)CC2CC(C1)N(C(=O)CCc1cn(C)nn1)C2 80425,C1(NC(c2c(C)cc(F)cc2)=O)C2CC(O)C1N(C(c1cn(C)nn1)=O)C2 80426,C1(C(=O)NC2CCCN(C(C3(C4(C)CC4)CC3)=O)C2)CCC2CC1CO2 80427,n1(CC(=O)NC(C)C(C)NC(=O)COC2CC=CC2)cc(C(F)(F)F)nn1 80428,CC1CN(C(=O)CCSc2ccccc2F)CC1NC(=O)Cc1ccccc1O 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80446,Cc1csc(=O)n1CC(=O)NCC(c1ccccc1)NC(C1CC12CC2)=O 80447,C(CCC(C)(C)NC(=O)C(C)CC1CC1)NC(C1CC(CC)(CC)C1)=O 80448,c1(C(=O)NC(CC(C)C)(C)CNC(=O)C=CS(C)=O)cnc2n1CCCC2 80449,Cc1cc(C(=O)NC2CN(C(=O)CC(C)c3ccncc3)CCC2F)cc(F)c1 80450,C1(NC(C2OCCN(C)C2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1C(N)=O 80451,C(=O)(C(CNC(=O)CSC)CCC)NCCC#CCC 80452,N1(C(C=CCOC)=O)CCCC(C(=O)NC(C)C(N)=O)C1 80453,c1(C(=O)NC2C(F)CCN(C(c3n(CC=C)ccc3)=O)C2)cccc2sccc12 80454,c1(SCC(=O)NCCC2(CNC(CCCOC)=O)CCC2)cc(C)ccc1C 80455,c1(C(=O)NC(C)CCO)ccc(C2COCCN2C(C2CC2C(F)(F)F)=O)n1C 80456,c1(C(N2C(CC)CC(O)C2)C(=O)NC(C)C)c[nH]c2c(F)cc(Cl)cc12 80457,C12(CC)CN(C(=O)CC(C)(C)O)C(CNC(c3ccc(N(C)C)nn3)=O)(C1)C2 80458,C(=O)(C(C)(C)C(=O)NN1Cc2ccccc2C(=O)N(C)C1=O)OCC 80459,C1(NC(Cc2cnc(C)[nH]2)=O)CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 80460,CCCC(C)(C)C(=O)NCC1(F)CCN(C(c2noc(C3CC3)c2C)=O)C1 80461,CC1(C(N2CCOC(C(=O)NCc3cn(C4CC4)cn3)C2)=O)CC2CC2C1 80462,C(c1cccc(CO)c1)=CC(=O)NC12CC(NC(=O)CC3CC4(CC4)CO3)(C1)C2 80463,Cc1ccc(-c2cc(F)ccc2CO)c2nc(C(=O)NCCc3ccc[nH]3)cn12 80464,N1(C(C(CNC(C2C(C)=CCS2)=O)O)=O)CC2CCCCCC2C1 80465,Cc1ccc(CC(N2CCCC2(C)CNC(c2cnccc2N(C)C)=O)=O)cc1Cl 80466,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(N(C(=O)C=CCO)C)C1)=O 80467,c1(C(N2CCCC(N(C(=O)CN3CCC(C)C3)CC)C2)=O)cnc(S(C)(=O)=O)s1 80468,c1(C(=O)NCC2CN(C(c3cnc(SC)s3)=O)CC2C)cc(C)c(F)c(C)c1 80469,CC1CN(C(C2CCC(C)C2)=O)CC1CNC(=O)Cn1ncc(C2CC2)n1 80470,c1(NC(C(CC=CC)NC(C2CCCN2C)=O)=O)cnc(C)nc1C 80471,C1(OC)(CNC(C2SCCS2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C1 80472,N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 80473,N1(C(C(C=CCCC)O)=O)CC2CCC1C(NC(c1cc(O)cc(=O)o1)=O)C2 80474,C1(C(=O)NC2(CNC(c3ccnc(O)c3)=O)CCCCC2)CC2(CCOC2)C1 80475,Cc1noc(C)c1SCC(=O)N(CCCNC(C1(O)CCOCC1)=O)C(C)C 80476,C=CCCC(F)(F)C(=O)NCCOCCNC(C1OCC2CCCC12)=O 80477,C(=O)(CCCC(=O)N1CC(C2CC2)(NC(C2CC(CC)CCN2C)=O)C1)OCC 80478,C12(CCC)CC(CO)(CN1C(C)=O)C2.N12CCN(CC1)C1CCC(CC1)C2=O 80479,c1(-c2ccc(CCCC)s2)ccc2c(c1)N(C(c1ncc(SC)cn1)=O)CC2 80480,CC1(C)OC2(C(=O)NCCn3cc(C4CCCO4)nn3)CCC1C2 80481,C1(CNC(=O)C(=O)Nc2cc(Cc3ccccc3)no2)CCCCNCC1 80482,c1(C(=O)NCC2CC(NC(C(CC(=C)C)C)=O)C2)cc2ccc(F)cc2o1 80483,C1(NC(=O)C2=CCC2)CCC2(CCCCC2)CC1 80484,n1(CC(N2C(CN(C(=O)C(N)=O)C)COCC2)=O)nc(C(F)(F)F)c2c1CCC2 80485,c1(C(=O)NCC(CNC(c2ccc(Cl)c(Cl)c2)=O)F)cccc2ccncc12 80486,CC1CC(C(=O)NCC(C)(C2CC2)NC(c2cc(O)nn2C)=O)CCC1C 80487,c1(N2CC(C(=O)NC(CCNC(CC(C)CF)=O)(C)C)C2)ccc(S(N)(=O)=O)cc1 80488,C1(C(=O)NCC2(NC(C3CCC(C)(CC)O3)=O)CC2)CN2CCN1CC2C 80489,CCC(CC)(C(=O)NC(CNC(C1CCCC(C(N)=O)C1)=O)C(C)C)OC 80490,C=C1CC(C)(NC(=O)CC2C(NC(=O)CC(C)OC)CC2O)C1 80491,C1(CC)CN(C(C2(Cl)CC2(F)F)=O)CC2(CCCOC2)O1 80492,CCC(F)(F)CC(=O)NC(c1nocc1C(=O)NC(CO)(CO)C1CC1)C 80493,C(=O)(CCC(F)(F)C(=O)N1CC(C)N(C(=O)CC(C)(C)CC)CC1C)OCC 80494,C(=O)(CCCn1nnnc1C(C1(CCO)CCC1)NCCCCO)OCC 80495,c1(C2(C(=O)NC3C4N(C(CCC=CC)=O)C(CC4)C3)CC2)ccc([N+](=O)[O-])cc1 80496,c1(C(N(C2CN(C(C(c3c(C)cccc3)C)=O)C2)C)=O)ccn(C(C)C)c(=O)c1 80497,C12(CNC(c3c(C)coc3)=O)CCCC(CN1C(c1cc(F)cc(F)c1)=O)C2 80498,C(=O)(C(CC1CCC1)NC(=O)C(O)c1ccsc1)NC(C(C)C)c1ccco1 80499,C(c1cc2ccccc2o1)=CC(=O)NCc1cc(Cl)ccc1OCCO 80500,c1(CCC(=O)NC2CCC2CNC(=O)COc2ccccc2)ccccc1F 80501,C1(NC(c2cn(CCC(C)C)nn2)=O)CCN(C(C2CCN(C)C2=O)=O)C1(C)C 80502,C(=O)(C(O)C(C)C)NCC1CC(NC(c2ccc(C3C(C)C3)o2)=O)C1 80503,C1(C(=O)NCC(N(C(=O)Cc2ccccc2O)C)C2CC2)CN2CCC1(C)CC2 80504,C(CCC(O)C(=O)NC(c1noc(C)n1)CC)NC(c1c(CC)n(C)nc1)=O 80505,CC#CCC(C(=O)Nc1ccc(SC)nc1)NC(c1cc(C)no1)=O 80506,c1(C(C2CCN(OC(=O)COCP(C)(C)=O)CC2)C)ccc(N)cc1[N+](=O)[O-] 80507,Cc1ncn(C)c(=O)c1C(=O)NCCC1CC(NC(=O)Cc2ccsc2C)C1 80508,C1(NC(N2C(C(=O)OC)(COC)CCCC2)=O)CCOC2(CCCC2)C1 80509,C1(C(=O)NC2CC(C)(CSC)C2)CNC(=O)CN1C(=O)CCC1CCCOC1 80510,c1(C(=O)NC2(C)CN(C(C3(COC)CC3(F)F)=O)C2)cc(C)ccc1OC 80511,c1(C(=O)NCC2(NC(c3ccc(C#N)o3)=O)CC(OC)C2)ccc(F)c(Cl)c1 80512,C1(CCO)(CNC(C(=O)NCCC(=O)NC(CC)C)=O)CCCC1 80513,Cc1cncc(C(=O)NCc2c[nH]nc2C(F)(F)F)n1 80514,c1(NC(C)=O)ccc(S(=O)(=O)NCC2CCN(c3ccc(C)c(F)c3)CC2)cn1 80515,CC1(CNC(C2CCC(=O)NC2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)C1 80516,c1(OCC)ccc(C)cc1C(=O)NC1CCN(C(C2(C)COCCO2)=O)CC1F 80517,N1(C(=O)CCOC2CCC2)CCC2C(CCN2C(=O)CCSc2ccccn2)C1 80518,c1(C(=O)NC2CCN(C(c3cccc(OC)c3)=O)C2)c(Cl)ccc2c[nH]nc12 80519,N1(C(C(c2cccc(OC)c2)OC)=O)CCC(C)(C)C(C(=O)NC2CC(O)C2)C1 80520,C1(C(N2CC(C)(NC(=O)C(Cc3ccccc3)SC)C2)=O)(CC)CCOC1 80521,c1(C(N(C2CCN(C(=O)COC3(C)CCCC3)C2)C)=O)cn(C)nc1C1CC1 80522,c1(C(N2CC(CC)C(NC(c3c[nH]nc3C)=O)CC2)=O)cc2c([nH]1)COCC2 80523,C#Cc1cc(OC(c2ncc(COc3ccc(Br)cc3)cn2)=O)ccc1Cl 80524,C(CO)(C(=O)N=c1ccn(C(F)F)[nH]1)N(C(=O)Cc1c(F)cccc1Br)C 80525,c1(CCNC(C2CCCC(NCc3ncc[nH]3)C2)=O)c(Cl)ccnc1Cl 80526,CCCCC(CCCC)C(=O)Nc1ccccc1CN(C)C 80527,C1(NC(CCCNC(C)=O)=O)CCN(C(c2ccc(C)c(C3CC3)c2)=O)CC1F 80528,C(N=c1[nH]c2c(c(=NCCOCCC3CC3)[nH]1)COC2)C1(C)CCCC1O 80529,N1(C(CCC2CCC(NC(CC3CC(C)(C)C3)=O)C2)=O)CCC(C#N)C1 80530,CN1N=C(CC(=O)NCCC2CCCN(C(c3c[nH]c(=N)s3)=O)C2)CC1=O 80531,Cn1ncc(CNC(=O)C(F)(F)C2CCOCC2)c1CNC(C1CCOC1)=O 80532,c1(C(=O)NC(CCNC(c2c(NC)cccc2)=O)C)ccc(F)c(F)c1 80533,c1(C(=O)N(C2CCCN(CC(=O)C3CC3)C2)CCCN)cnc(OC)nc1.C1(N)CC1 80534,c1(CC(=O)N(C(c2ccccc2)CN(C(=O)C(C)(C)C)C2CC2)C)cnnn1C 80535,Fc1cncc(-c2nc(-c3ccc(Cn4ccnc4)o3)n(CCCO)n2)c1 80536,C12(C(=O)NC3C(CC)CN(C(c4scnc4C)=O)CC3)CCOC1CCOC2 80537,c1(C(c2n(CC)nnn2)NCC(c2nccs2)C)cc(Br)nn1C(C)C 80538,CCC(CNC(NOC(=O)CCC(=O)c1cc(C)sc1C)=O)CC(F)(F)F 80539,c1(CCC(=O)NC2CN(C(C3(OC)CCC3)=O)CC2C)ccc2[nH]ccc2c1 80540,C1(NC(C#CCNC(C=C(C)C(C)C)=O)=O)CCCCCCC1 80541,C1(C(N2CCC(CC)C2CNC(=O)Cc2coc(C)c2)=O)CC12CCC(=O)CC2 80542,N1(C(C(C)NC(c2ccc(Cl)s2)(c2nnnn2C)CC)=O)CCN(C(=O)OC)CC1 80543,C(C)(C)(C(=O)N1CCC(CCNC(=O)C(c2cnn(C)c2)C2CC2)C1)OC(C)=O 80544,N1(C(C(CNC(CSC2(C)CCC2)=O)O)=O)CC2CCCC1C2 80545,c1(C(=O)NC(C)C(=O)N(C2CC(C(N)=O)C2)C)cn2ccccc2n1 80546,N1(C(c2nc(C(C)(C)C)oc2)=O)CCN(CCN(C(=O)C(C)(C)CF)CCO)CC1 80547,CC(C(=O)NCC1C=CCN1C(=O)CCOC1CC1)S(=O)(=O)c1ccc(Cl)cc1 80548,C1(N(S(C)(=O)=O)C)CC12CCN(C(=NCc1ccc(Cl)c(Cl)c1)NCC(F)F)CC2 80549,c1(C(=O)OC)c[nH][nH]c1=NCCNC(=O)C(C)OC 80550,C1(C#CC(=O)NCC=CCNC(=O)CCc2cncnc2O)(CC)COC1 80551,c1(C(=O)NCC(C)NC(=O)CCC2CCCN(C)C2)cncc(Cl)c1 80552,CC1CN(C(C23CCCC2N(C(=O)CN2CC4CC4C2)CC3)=O)CCN(C)C1 80553,Cc1ccc(C(N2CCCC(N(C)C(c3ccnn3C)=O)CC2)=O)nc1F 80554,CC1C(C(N2CC(OCCNC(=O)CC3NC(=O)NC3=O)C2)=O)CC(C)(C)C1 80555,CC(C(=O)NCC1CCCCN1C(C1CCn2ncnc2C1)=O)P(C)(C)=O 80556,N1(CC(=O)NC2CC(NC(C3N(CC(C)C)CCC3)=O)C2)CCCCCC1 80557,c1(C(C)C)ccc(C(=O)NCCCCCCNC(=O)CC2CC2CO)cc1 80558,C1(CCC)COCCN1C(=O)CNC(=O)CCCc1nc(C(C)OCCOC)no1 80559,N1(C(C2CC(SC)C2)=O)CC2CCN(C(c3nc(Cl)ccc3N)=O)CCC2C1 80560,C1(NC(c2ccoc2)=O)CC2CC(C1)CN(C(=O)Cn1cc(CO)nn1)C2 80561,C#CCCCCN=C(NCCc1cccs1)NC1CCN(CC(F)(F)F)C1 80562,Cc1nn(CCC(N2CCOCC2C(C)(C)OC(=N)O)=O)c(C)c1[N+](=O)[O-] 80563,CC1CN(c2ncncc2Cl)CC1NC(=O)CCCN1C(=O)CNC1=O 80564,Cc1cccc(C)c1-n1cc(NC(C2(F)CCOC2C)=O)cn1 80565,c1(C(=O)NC2C(CC)N(C(c3ncccc3F)=O)CCC2)ccc(Cl)c(Cl)c1N 80566,C1(C(N2CC(CCNC(C3COC(=O)N3C)=O)(OC)C2)=O)CC(C)CC(C)C1 80567,c1(CNCC2OCCN(C(c3cnc(Br)cn3)=O)C2)ccc2c(c1)CCCO2 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80585,C1(C(N(C(CCO)C(C)(C)C)C)=O)N(C(=O)OC(C)(C)C)CC12CCCC2 80586,N1(C(C2C(C=CCC)CN(C(C3(CSC)CC3)=O)C2)=O)CCC2(CNC(=O)C2)C1 80587,C1(CNC(CC2CCC(C)C2)=O)CC2CCC(C1)N2C(c1ccc2nonc2c1)=O 80588,c1(OCC=C)ccccc1C(N1CCC(C)(CNC(c2n[nH]c(C)c2F)=O)C1)=O 80589,C1(C(=O)OCc2ccc(C#N)o2)CCCc2ccccc2C1 80590,c1(CSC)cc(=NC(=O)NCCCc2ccc(Br)c(F)c2)[nH]n1C 80591,CCC(C)(CCC(C)C)C(=O)NCC1CCN1C(=O)C(C)S(=O)(=O)C(C)C 80592,c1(C(N(CCNC(=O)CC23CC(C2)C3)CC)=O)ccc(F)c(F)c1 80593,C1(CC(=O)NCc2cccs2)CCN(C(=NCCc2ccncc2F)NCC)C1 80594,C(N=c1[nH]ncs1)C1(NC(C=C(C)C)=O)COC1 80595,C=CC1CN(C(=O)C=CBr)CC1NC(C1CC(C)(C)O1)=O 80596,C1(COCC(=O)NCCC(=O)NCC(CO)C2CCC2)CCCCO1 80597,c1(C(=O)NC2CN(C(C3(SC)CC3)=O)C(C)CC2)nccn2c(C)nnc12 80598,C1(NC(CC(CC)(F)F)=O)CN(C(=O)CC2CCC(OC(C)=O)CC2)CC12CCC2 80599,c1(CC(N2CC(F)(C(N3C(CO)CC3CO)=O)C2)=O)ccn2ccnc2c1 80600,c1(-c2nc(C(C)Oc3ccc(CCOC)cc3)on2)cc(Br)c(C)nc1F 80601,Cc1nc(C(N2CC=CC2(C)C(=O)NCC2(CO)CC3CC3C2)=O)cc(O)n1 80602,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CC(=O)N(C(C)C)C2)=O)C(CC(C)(C)C)C1 80603,c1(CNC(=O)CSc2cn[nH]c2)cn(CC(N2CC3CC3C2)=O)cn1 80604,C(C1=CCCN(C)C1)NC(C(Cn1cccn1)NC(c1[nH]cc(C(C)=O)c1)=O)=O 80605,C(=O)(C(C#N)C(C)C)NCCNN(CCOCCC(=O)C(C)=O)CCO 80606,C(=O)(C(F)(F)C1=CCOCC1)NC1C(CNC(C(C)SCC)=O)CCCC1 80607,c1(C(=O)OCc2cnc(C)s2)ccc2c(c1)S(=O)(=O)N(C)C2=O 80608,Cc1cc(Cl)cc(C)c1OCC(=O)NCC(C)NC(=O)CC1(O)CCOC1 80609,Cc1cc(C(=O)NCC(F)CNC(=O)CCC2CCN(C)CC2)ccn1 80610,CON=CC(=O)N1CCC(N(C(=O)Cc2ccco2)CCn2ccnc2)C1 80611,C1(CNC(Cc2cn(CC)nn2)=O)CC(C)(C)CN1C(=O)Cc1ccnc(F)c1 80612,N1(C(c2c(C)nsc2)=O)CCC12CN(C(=O)C(O)C(C)(C)C)C2 80613,n1(CCOC)cc(C(=O)NCC2CC(F)(CNC(C3CCC(C)C3)=O)C2)cn1 80614,N1(c2cc(N3CCCC(N(C)CCO)C3)ncn2)CC2C3CCC(CC3)C2C1 80615,C1(NC(CCOC(C)=O)=O)CN(C(c2cn(Cc3cccnc3)nn2)=O)CC1C 80616,C(=O)(C1=CCC(C(F)(F)F)OC1)NC(CC)CNC(c1cnoc1C)=O 80617,C1(C(=O)NC2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)CCC=CCCC1 80618,c1(C(=O)NC(C)(C)CN2CCCCC2=O)cnn2cc(F)cc(F)c12 80619,C1(N(C)C(c2cc(-c3ccccn3)no2)=O)CN(C(C2(C)CSC2)=O)CC1F 80620,c1(CC(N2CCC(CN(C(C(CC)F)=O)CC)C2)=O)ccc(Cl)cc1F 80621,C(C(C)(C)CC(=O)N(CCC(C)O)C)NC(c1nc(C(C)C)oc1)=O 80622,N1(C(CN(C)C)=O)CCN(Cc2ccc(OC#N)c(I)c2)C2CC12 80623,C12(NC(=O)CC3CC4(CCC4)C3)CCN(C(C3CC4(CC4)C3)=O)CCC1C2 80624,C1(NC(c2ccc(C3CC3)s2)=O)CCCC12CN(C(=O)COCC1CCC1)C2 80625,c1(NC(C)=O)c(F)ccc(F)c1CN1CCN(C(=O)C(c2ccccc2)O)CC1 80626,c1(C(N(CC(O)CN(C)C(C2CC3(CC3)C2)=O)C)=O)c[nH]nc1-c1ccccc1 80627,Cc1cccc(-n2ncc(C(N3CCC(N(c4cccnn4)C)CC3)=O)c2C)c1 80628,c1(C(=O)NCCCN(C(=O)C=CCOC2CCCC2)C)cc(C2CCCCC2)no1 80629,O(C1CCc2c(Br)cccc21)CC1(C(C)(C)O)CC1 80630,c1(C(=O)NC(CCCNC(C2(C)CCC(OC)CC2)=O)C)ccc(C#N)c(C)c1 80631,CCCCCCCCC(C)C(=O)N1CCC(N(C(=O)CC2CCOC2)CCC)C1 80632,C1(C(=O)NC2(C(F)F)CC(C(=O)NCC3CC(OC)C3)C2)CC(C)(C)CO1 80633,C=CCC(C)(C)C(=O)NC(C)CCNC(=O)C=C1CC1 80634,CC1(C)CC(C(=O)NC2COCCC2NC(=O)CCN2CCCC2)CCO1 80635,Nc1cccc(C(=O)NC2(CCNC(=O)CC3C=CCC3)CC2)c1Br 80636,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)=C(C)CC)CCC1C 80637,C(=O)(C1=CCCC1(C)C)N1CC(CN(C(c2cncc(C#C)c2)=O)C)OCC1 80638,c1(C(N(C(C)C)Cc2cc[nH]c(=N)c2)=O)ccccc1CC(N)=O 80639,N1(CCCNC(c2nnnn2C2CCCC2)(CC2(C)CC2)C)CCNC1=O 80640,N1(C(CC(=O)Nc2nc(CCC)c(CC)s2)=O)CCc2ccccc21.C1C(=O)O1 80641,c1(C(=O)NCCC2(CNC(C3(C)CCC3)=O)CC2)cccc2sncc12 80642,C(=O)(CC(F)(F)C(C)C)NC1C(CNC(c2c(C)noc2)=O)CCC1 80643,N1(C(c2nccc(OC)c2)=O)CCCOC(CNC(c2ccncc2OC)=O)C1 80644,C1(C#N)(COCCCNC(C2CC(C(=O)OC)C2)=O)CC12CCC2 80645,C1(C(=O)Nc2c(C(=O)OC)n[nH]c2)C2CN(CCn3cnnn3)CC12 80646,N(C(=NCc1ccccc1)N1CCC(O)CC1)CCN1CCCC(CN)C1.CO 80647,C(=O)(C1CCCc2c[nH]nc21)N1CCC(N(CC#C)C(C2C=CCC2)=O)CC1 80648,Cc1cc(C(N2CCCC2)=O)c(Br)cc1F.N12CCCCC1CNC2=O 80649,c1(C(N(c2ncc(SC)cn2)C2CCNCC2F)=O)cc([N+](=O)[O-])c(F)cc1F 80650,C#Cc1c[nH]nc1C(N1CC2CC2(CNC(C2(COC)CCCC2)=O)C1)=O 80651,N1(C(c2c(C)n(C)nc2)=O)CC2CCCC2(NC(C2CC=CC(O)C2)=O)C1 80652,c1(C(N2CC(C3CC3)(C(=O)NOC3CCOC3)C2)=O)cccc2ccoc12 80653,CC(CC(=O)NCCCCCNC(C1(O)COC1)=O)c1cccnc1 80654,C#CC1(O)CCCN(C(=O)C(C)(C)CN(C)C(C2SCC=C2C)=O)C1 80655,n1(CC(=O)NCC(CCOC)C)c(C)cc(C(=O)Nc2cc(C(C)=O)cs2)c1C 80656,C1(OC)CN(c2cc(C(F)(F)F)ncn2)CCC1NC(=O)Cc1ccc(F)cn1 80657,C1(N(C)C(C2C=CCS2)=O)CCCOC1.C1(=O)COCCC2(CC2)CN1 80658,N1(C(c2cn(CC=C)nc2)=O)CC2=C(C1)CN(C(c1cc(C)c(O)c(C)c1)=O)C2 80659,C1(C(=O)Nc2ccccn2)CC12CCN(Cc1cncnc1)CC2 80660,N1(C(CCOC)=O)CCCC2(NC(=O)CNC(c3cc(F)ccc3F)=O)CC12 80661,CC(C)C(C)(Cc1ccccc1)C(=O)NC1CC1NC(C1CCC(F)(F)CC1)=O 80662,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NC(C1(O)CC1)C1CCC1 80663,N1(CCC(=O)NCC2(F)CN(C(c3cc(CCO)on3)=O)C2)CCNC(=O)C1 80664,C12(C(=O)NCCSCCOC)C(NC(=O)CN3CCOC3=O)C3CC1C2C3 80665,c1(CC)nc(=N)[nH]cc1C(=O)NC1CC(NC(C2CC2c2ccccc2F)=O)C1 80666,c1(C(C)OC)nc(NC(=O)NC2(C(N)=O)CCC2)cc(=NC2CCC(=O)NC2)[nH]1 80667,C1(CCC(=O)NCCC=C)CCCCN(C(c2scnc2CC)=O)C1 80668,C1(NC(CCC(C)C)=O)C2COCC1CN(C(c1cccc3ncoc13)=O)C2 80669,CC12CN(C(=O)COC3CC3)CC1(C)CN(C(C1(F)CC1)=O)C2 80670,c1(C(N2CCCCC(NC(=O)C=CCBr)C2)=O)cc(I)ccc1[N+](=O)[O-] 80671,C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(c2cccc3c2CCC3)=O)CCCC1 80672,Cc1nn(C)c(C(F)F)c1S(=O)(=O)N1CCC2(CCCCC2)C1 80673,C(CC1=CCN(c2ncc(OC)cn2)CC1)NC(C1N(CC)CCOC1)=O 80674,C12(C(N(C3CCN(C(C45CC(F)(C4)C5)=O)C3)C)=O)CCOCC1C2 80675,N1(C(c2occc2F)=O)CC2(C1)CN(C(C1CC(CC3CCC3)C1)=O)CC2CO 80676,N1(C(C(COCC)N=[N+]=[N-])=O)CCCC2(CCN(C(=O)C=CCF)CC2)C1 80677,C1(CC)CCCC(C(N2CCC(OC)C2)C(=O)NCC2CCCO2)C1 80678,CCCC(CCO)N=c1[nH]c(=NCC2(COC)CC2)[nH]c2cc(OC)ccc12 80679,C1(NC(C=C2CCC(C)CC2)=O)CC(NC(C2CCS(=O)(=O)CC2)=O)C12CCC2 80680,C(CC(=O)Nn1cnn(C)c1=S)ONC(Cn1nc(C)oc1=O)=O 80681,C1(NC(CC2(C)CCN(C(=O)C(F)C3CCCC3)C2)=O)C(O)C2CCOC12 80682,C1(C#N)(C(=O)NCC(C)N(C(=O)C(O)C2CC2)C)CCN(C)CC1 80683,C1(NC(=O)CSS(C)(=O)=O)CC2CCC(C1)N2C(=O)CCc1nnc(O)nc1O 80684,c1(C(=O)NCC(C)(C2CC2)NC(CNC(=O)OC)=O)ccc2scc(C)c2c1 80685,c1(C(=O)NC(CN(C(C=CC)=O)C)CC)cc(Br)c2[nH]nnc2c1 80686,N1(C(CC2CCC(C)CO2)=O)CCC2(CC(C(=O)NCC3CCCC3)C2)C1 80687,c1(C(=O)NC2C(OC)CN(C(=O)C=CC(=O)N(C)C)C2)cc(C)c(C)cc1N 80688,C1(OC)CCCN(C(=O)C(C)(C)Cc2ccccc2)C1.c12nscc1N2C 80689,N(C1CC(C)n2ccnc21)C(C=CCNC(c1cccc(C)c1O)=O)=O 80690,N(C1CC2(CCN(C(=O)CC#N)CC2)Oc2ccccc21)C(C(CCC)C)=O 80691,N1(C(C(C)OCCC#C)=O)CCCC1CN(C(c1c[nH]nc1F)=O)C1CC1 80692,N1(C(C2CCCC(=O)O2)=O)CCCC2(CCCN2C(C23CSC(C2)C3)=O)C1 80693,C(=O)(CC(C)(O)CCC)N(CC(=C)C)CC1CC(C)NC(C)C1 80694,N(C1CCSc2ccc(Cl)cc21)C(=O)NC1(C(=O)OC)CC1(F)F 80695,Fc1cc(CN2CCCC(Cn3cc(C4COCCO4)nn3)C2)cc(Br)c1 80696,N1(C(CSCCC=C)=O)CCCN(C(c2cc(F)ncc2OC)=O)C(C)C1 80697,c1(C(N(C(CNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)cc(F)c(Cl)cc1F 80698,C1(CNC(CN(C)CCO)=O)CN(C(C2CCCCC2O)=O)CCC12CCC2 80699,C1(NC(c2ccc(CF)cc2)=O)(CO)CCN(C(c2cc(F)cc(F)c2)=O)CC1 80700,c1(OCC(=O)NCC2N(C(C(C)=C3CC3)=O)CCC2(C)C)cc(C)c(Cl)c(C)c1 80701,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(=O)CSc3cnn(C)c3)CC2)C1 80702,c1(OC)nc(C)ccc1C(=O)N(C1CCCN(C(=O)C(C)S(C)(=O)=O)C1)C 80703,N1(C(C(C2CN(C(c3nc(CC)oc3C)=O)C2)OC)=O)CCc2nncn2CC1 80704,C1(C2CC2)(CNC(CCC(=O)NC)=O)CCN(C(=O)CC2(C#N)CCOCC2)C1 80705,c1(C(=O)NC2CN(C(C3N(C)CCC3)=O)CC3(C2)CC3)c[nH]c2ccccc2c1=N 80706,C(CO)(CCCCNC(C1CCCC(O)C1)=O)NC(c1c(C)nc(C)s1)=O 80707,c1(CC(CN(CC)Cc2nonc2CN)OC(C)(C)C)ccccc1Cl 80708,c1(NC(=O)Cc2nc(-c3ccccc3)no2)ccncc1I.C1CN1CCO 80709,n1(NCCC2CCC(NC(C3(CC4CC4)CC3)=O)C2)cc(C(C)=O)cn1 80710,CCCCCC(C(=O)NC1CC2C(NC(C3CC(OC)C3)=O)C2C1)C(C)C 80711,S(=O)(=O)(c1ccccc1Cl)N1CCCC(CNC(c2cnc[nH]2)=O)C1 80712,N(C(=NCCCOC(C)(C)C)NCNC1CCN1C(C)(C)C)CC1CCC(SC)C1 80713,CCCCCCC(CC)(CC)C(=O)N1CC(C(=O)OCC(C)(C)COC)C1 80714,C1(NC(=O)C(N2CCC(C(F)F)C(O)C2)=O)COc2ccccc2C1 80715,Cc1oc(C(C)C)cc1C(=O)NC(C)Cc1ccc(CNC(=O)C(N)=O)cc1 80716,Nc1ccc(Cl)c(NC(=O)NCC(c2ccccc2)c2nnc(O)s2)c1 80717,N1(C(C(C)OCCN(C)C)=O)CC(C(=O)NCC2(F)CC(O)C2)C(C)(C)C1 80718,c1(N2CCC(NC(C3CCCOC3)=O)C2)ncc2scc(Br)c2n1 80719,N12CCC(F)(CC1)C(=O)NC(=O)CC1(CCCCC1)C2=O.CC(F)C(C)N(C)C 80720,CC1CC(C)CN(C(=O)Nc2cccc(C(N3CCCCCC3C)=O)c2)C1 80721,c1(NC(C(C)(C)OCC)=O)ccc(NC(c2cc(C)n(CC3CC3)n2)=O)cc1C 80722,c1(C(=O)NCC2C3CN(C(COCC)=O)C2C3)ccc2nc(C)n(C)c(=O)c2c1 80723,Cc1c(Cl)cccc1S(=O)(=O)NC1C2CN(C(c3ccc(Br)[nH]3)=O)CC12 80724,c1(CC=C)cccc(C(N2CCC2C(=O)N(C)Cc2ccn(C)c2)=O)c1 80725,C1(NC(=O)C(c2ccc(F)cc2)CO)CN(C(c2coc(Cl)c2)=O)CC1CO 80726,CC1(C)CCC(C)(C(=O)NCC2(F)CCN(C(=O)CC3CCCOC3)C2)CC1 80727,c1(C(=O)NCC2CN(C(=O)C(F)Cc3ccccc3)CC2O)cc(O)ncc1F 80728,c1(SC)nnc2n1CC(NC(c1cc(C(F)(F)F)cc(O)n1)=O)CC2 80729,N1(C(C(C)OCC=C)=O)CC(CO)C2(C1)CN(C(=O)CCCC1CCOCC1)C2 80730,C=CC(C)(C)CN=C(NCC(C)(C)C)NC1CC12CCC2.OC(F)(F)F 80731,C(C(C(C)C(C)C)NC(=O)C=CCCC=C(C)C)NC(C1(CC=C)CCC1)=O 80732,C#Cc1cccc(CNC2(c3nnnn3CCCCCC)CN(C)CC2C)c1 80733,CCCC(C)(CC)C(=O)NC1CC(CNC(c2cnn3c2N(C)CC3)=O)C1 80734,CC#CCCCC(=O)N1CC(C2(C)C(=O)N2)C1.c1(C)noc2c1CCC2 80735,C1(CNC(C(C)N2CCC2C2CCCC2)=O)CCCCN1C(c1cn[nH]c1)=O 80736,O=C1CCC(C(F)C(=O)NCCCNC(C2C3(CC3)C23CC3)=O)CC1 80737,N1(C(Cc2cccc(C)c2)=O)CC2CC(NC(c3ccc(CN(C)C)s3)=O)C1C2 80738,c1(C(=O)NCC2C(NC(C3(COC)CCCC3)=O)C2)cnc(S)nc1 80739,N1(C(C2CCCOC2)=O)CCC2C(CCCN2C(=O)CC23COCC(C2)C3)C1 80740,C12(CC)CCN(C1)C2=O.C1(C)(OC)CN(C(c2ncoc2C2CC2)=O)C1 80741,C1(NC(c2c(C)sc(C(F)(F)F)n2)=O)CC2(CCCCN2C(=O)C=C(Cl)Cl)C1 80742,CCC(CNC(c1cncs1)=O)(CC)NC(=O)CCCn1ccnc1C 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80760,c1(-n2c(C3CC34CCOC4)nc(CCC(C)C)n2)ccc(Br)c(F)c1 80761,C1(N(C(=O)Cn2nnnc2C2CC2)C)CCC(NC(=O)C(C)(C)C2CCC2)CC1 80762,c1(OC)cc(C(=O)NCC2(OC)CN(C(=O)C(C)CC(N)=O)C2)ccc1C(F)F 80763,C1(CNC(C2C(CC)C2)=O)CC(F)(F)CN1C(=O)CCc1n[nH]c(=N)s1 80764,N1(C(C2CC(CCNC(c3nc(CCC)oc3)=O)C2)=O)CCOC(CSC)CC1 80765,C1(NC(C2(CC)CCC(O)CC2)=O)CCC2(CC1)CN(C(=O)C=C(C)Cl)C2 80766,C1(C(=O)NCCN(CC(C)O)C(c2cc(C3CCC3)[nH]n2)=O)CC1[N+](=O)[O-] 80767,CC1CCC(CC(=O)NC2CCN(C(c3ccc(F)cn3)=O)C2C(C)C)OC1 80768,O=C(C1CCCc2ncnn21)NCC1CCC(NC(C2CCCSS2)=O)C1 80769,N1(C(c2ncn(CC)c2)=O)CC(C)C(C)(CNC(C2CCS2(=O)=O)=O)C1 80770,C(c1cncs1)=CC(=O)NC12CC(C(=O)NCCCCN3CCCC3)(C1)C2 80771,C(=O)(C(=O)CCC(C)C)NC1(C)CC(NC(C2CN(CC)C(=O)C2)=O)C1 80772,C(=O)(C(F)C(C)(F)F)N1CC(C)(CC(N2CC(C(C)O)C2)=O)C1 80773,Cc1ccc(C(N2CCCCC2CCNC(C2CCCCNC2=O)=O)=O)cc1Cl 80774,C(=O)(C(F)(F)c1cnn(C)c1)N(CC(O)CNC(=O)COCCF)C 80775,c1(C(N2CCN(C(COCCOCC#C)=O)C(C)C2)=O)cc2c(cn1)COCC2 80776,C1(CNC(CC(=C=C)C)=O)CN(C(c2nn(C)c(C)c2N)=O)CC(C(F)(F)F)O1 80777,c1(C(N2CC(NC(c3c(CC)[nH]cc3)=O)C(C)C2)=O)sc(Cl)c(Cl)c1OC 80778,C(C(CO)C(F)(F)F)Nc1cc(NC(=O)CC2CCS(=O)(=O)C2)ncn1 80779,C(=O)(C1=C(Cl)CC1)NC(C)(CNC(c1occc1Cl)=O)C1CC1 80780,CN=c1ccc(C(=O)NC(CO)CCCCNC(c2ccc(F)cn2)=O)c[nH]1 80781,C(=O)(C1=CCC(C)(C)CC1)NC(C1CCN(C(C(C(CC)CC)C)=O)CC1)C 80782,Cc1cc(NC(C2(NC(C3CC4(CCO3)CC4)=O)CSC2)=O)cc(Cl)c1 80783,c1(Oc2c(C)cccc2)ccc(CN(c2ccccc2N)C(=O)CNC(N)=O)cc1 80784,c1(CC(=O)OC(c2c(C)nn(C(C)C)c2)=O)cccc(Br)c1F 80785,C(=O)(C1CCc2nccn21)N1CC(O)(CNC(C(=C(C)C2CC2)F)=O)C1 80786,c1(OC)ccc(NC(N2CCN(CC(C)O)C(C)C2)=O)c(OC(F)(F)F)c1 80787,c1(C(C2(OC)CCC2)NC2(C(=O)NCC)CCC2)nnnn1C1CCC1 80788,Cc1c(C(=O)NCCNC(=O)CCc2ccc(Cl)s2)c(=O)oc2ccccc12 80789,c1(C(=O)NC(C)CCN2CCCCC2)ccc2occc2c1 80790,C1(C#CC(=O)NCCn2cc(C(=O)NC3CC=CCC3)cn2)(CC)COC1 80791,N1(C(COCCC#C)=O)CCc2ccccc2C(N(C)C(=O)C(CCC)OCC)C1 80792,Cc1nc(N2CCC(CC3CC4C(C3)C4(C)C)C2)c(F)c(C)n1 80793,C1(NC(C(CC=C)(F)F)=O)CC2(CCN(C(c3nocc3C(C)(C)C)=O)C2)C1 80794,C(CC(=O)NC1CCCO1)N(C(=O)C(C)OCCC=C)CC#C 80795,c1(C(CC(=O)OC)C)ccc(NC(=O)CNC(=O)C(C(C)C)OC)cc1 80796,N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCN(C(N)=O)C2)=O)C(CCO)C1 80797,N1(C(CN2C(=O)COCC2)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CCC12 80798,c1(C(=O)NC2CCC(NC(c3ccn(CCC)n3)=O)CC2)cc(C)cc(F)c1 80799,C1(C(C)C)COCCN(C(c2csc(C(F)(F)F)n2)C(=O)Nc2ccccc2)C1 80800,c1(OC)ccc(CC(=O)NC(CCN(C)C(C2(C)CCCS2)=O)C(C)C)cn1 80801,C(=O)(C1=NOC(CNC(C2CCC(=O)N(C)C2)=O)C1)N1C(CCCC)CCC1 80802,C(CCCC(C)C)NC(c1n(CCOC)nnn1)CCc1ccc(F)cc1 80803,C(=O)(C(Cn1ccnc1)CC(C)C)N1CC(CNS(CC(=O)OCC)(=O)=O)C1 80804,N1(C(c2n(CC)ccc2)=O)CC2OCCN(C(=O)Cn3nc(O)ccc3=O)C2C1 80805,C1(CNC(c2c(C)cco2)=O)CC2(CCC2)CN1C(=O)C(C)OC(C)(C)C 80806,N1(c2nnc(CCC)s2)CC2(C1)C(NC(c1cn(C)cn1)=O)CCS2(=O)=O 80807,CC1(C)CC(CC(=O)NC2CC(O)C2)CN1C(=O)Cc1cccnc1 80808,CCS(=O)CC(=O)NCc1ocnc1C(=O)NCCC1(O)CCCC1 80809,N1(C(CC(=O)NCC)=O)CCC(C(N2CCCC(C#N)C2)=O)C12CCC2 80810,C1(NC(=O)CSc2nncs2)CC2CC1N(C(=O)CCOC1CCCCC1)C2 80811,C1(C(=O)NC(CCC)CNC(C2(C)CC2)=O)CC2COCC(C1)C2 80812,c1(C(N2C(CNC(=O)Cn3cc(CO)nn3)CCC2)=O)ccc(Cl)cc1Br 80813,N1(C(Cc2cc(C)nn2C)=O)CCN(C(=O)Cn2nc(C(F)F)cc2C)C2CCC12 80814,N1(C(C=C(C)C(C)C)=O)CC2CCC(NC(C3CCCC(CF)C3)=O)CC2C1 80815,N1(C(c2cn(CC=C)nc2)=O)CCN(C)C(CNC(=O)C=Cc2cnn(C)c2)C1 80816,C1(c2c(C(=O)OC)ncs2)CCCN(N2CCCC2CC(N)=O)C1 80817,C1(C(C)(C)C)CCCC(c2nnnn2C2CCOCC2)(NC2CCCC2CF)C1 80818,Cc1nc(Cl)ccc1C(=O)NC1(CCNC(=O)CCCC(F)F)CCC1 80819,Cc1ccc2nc(N3CCOCC3CNC(C3CN(C4CCOCC4)C3)=O)sc2n1 80820,c1(C(=O)NC2C(NC(C(C)SC(F)(F)F)=O)C2)cc(=O)n(CCF)[nH]1 80821,N1(C(c2nc(C)n(C)c2C)=O)CC(NC(=O)CCP(C)(C)=O)CC12CCCOC2 80822,N1(C(c2cncc(C)n2)C(=O)NCCOCC)CCSc2ccccc21 80823,C1(CCC)CCCN(N2CC(S(=O)(=O)NC)(NCC3CCCO3)C2)CC1 80824,c1(C(=O)NC2CN(c3cc(C)ncn3)CC(C)C2)cccn2ccnc12 80825,C1(CNC(C2N(CC)CC2)=O)CCCCC1NC(=O)Cc1ncc(Cl)s1 80826,C1(CNC(CC2CCN(C(C)=O)C2)=O)CN(C(c2ccoc2Cl)=O)CCCO1 80827,N1(C(C(C2CC2)OC)C(=O)NCc2ccc(C)s2)CCOCC(C)(F)C1 80828,Cc1cccc2[nH]cc(CN3CCSC(C(=O)NCCc4cc[nH]n4)C3)c12 80829,Cc1c(-n2cc(-c3cccc(NC(c4occ5c4CCC5)=O)c3)nn2)cccc1Cl 80830,C(CNC(=O)Cc1cc[nH]c1)(CC(C)C)NC(c1c(CC)scc1)=O 80831,N1(C(C2(CC)CCNC2=O)=O)CCC(N(C)Cc2ccnn2C)C(C)C1 80832,C1(N(C(C)CCOC)C(c2ccoc2C(=O)OC)=O)CCC(=O)NC1 80833,Cc1c(C(=O)NCCC2CCCN(C(c3ccc(F)cn3)=O)C2)cc(O)cc1N 80834,C(CCC(=O)NCCOCC)NC(=O)OC.c1(NC(=O)CO)cn[nH]c1 80835,C1(C(N2CCC(N3CCC3CF)CC2)=O)OC2CCC1CC2 80836,N1(C(c2cc(SC)oc2)=O)CC(NC(=O)C(F)=CC2CC2)CC12CCCCCC2 80837,C1(C(=O)NCCC2(NC(CNC(=O)OCC=C)=O)CC2)(CC)CCCNS1(=O)=O 80838,c1(C(=O)NC(CC)CN(C(=O)CC2CC3(CC3)CO2)C)cc2ncccc2[nH]1 80839,N1(C(C(n2ccc(C3CC3)n2)C)=O)CCC2(CCCN2C(C2CC(CF)C2)=O)C1 80840,C1(C2(OC(C)(C)C)CC2)CCCCN1C(=O)Cn1cnccc1=O.C1CCC(=O)N1 80841,N1(C(COCCCOC)=O)CCc2sccc2C1CNC(=O)C(F)n1ccnc1 80842,c1(CN(C)CC2CCOC2)ccnc(F)c1N 80843,c1(C(=O)NCC2CCN(C(c3cnn[nH]3)=O)C2)cc2c(s1)CCCCCC2 80844,N1(C(c2c(C)cco2)=O)CC2CCN(C(=O)Cc3ccc4c(c3)CCO4)CC2C1 80845,CCCC(C(O)C(=O)NCC1(C)CC(C)=NO1)NC(=O)CN(C(=O)C(C)C)C 80846,C(=O)(C1=C(C)OCCS1)N1CCC(NC(C(CC)OC)=O)(CO)C1 80847,N1(C(CS(CC)(=O)=O)=O)CCC(C2CN(C(C34COCC3C4)=O)C2)CC1 80848,c1(C(=O)NCC(c2ccccc2F)NC(C(C)=CC)=O)cccc2nccn12 80849,c1(C(=O)NCC(CNC(CCNC(=O)NC)=O)F)cnc2[nH]nnc2c1 80850,O=C(C#CC1CCOC1)NC1COC2CN(C(c3ccccc3Cl)=O)CC12 80851,C1(NC(C=C(CC)C)=O)CCCN(C(C2CCN(c3ccncc3)C2)=O)C1 80852,N1(C(C(=O)c2ccco2)=O)CCC2(CCCN2c2ncnc3n[nH]c(I)c23)CC1 80853,C=C(C)CCC(C(=O)Nc1ccccc1C)N1CCNC(=O)C1 80854,C1(C(N2CCCC2C2(C(=O)N(C3CCCS3)C3CC3)CC2)=O)CC2CCC1O2 80855,C1(C(=O)NC2CC(CNC(=O)Cc3cc(Cl)cs3)C2)(OC)CCC12CCC2 80856,CC1C(C(N2CCCCC2)=O)CCN1C(c1ccc(O)cc1)=O 80857,C1(C#CC(=O)NC2CN(C(=O)CCC(C)SC)CC2(C)C)(CC)CC1 80858,c1(C(C)C)cc(C(=O)N(C2CC(NC(C3(CN)CC3(F)F)=O)C2)C)n(C)n1 80859,c1(CC(C(=O)NCCC(C)C)NC(=O)CC2CC(C)C2)ccccc1Br 80860,N1(C(C(CC#C)O)=O)CCOCC(C)(CNC(=O)CCCNC(=O)OC)C1 80861,C1(C#N)(C(N2CC(N(C)C)C(C)(C)C2)=O)CC2CCC1CC2=O 80862,N1(C(c2c(C)ccnn2)=O)C2CC=C(C(=O)NC3(CF)CCCC3)C1CC2 80863,N1(C(CC2N(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C)CSC)CC2 80864,CCCC(C)CC(=O)NC1CC(F)(CNC(C2CCCCN2C(N)=O)=O)C1 80865,C(=O)(C1=C(C)CCCC1(C)C)NC1CN(C(C(C=C)(C)O)=O)CC1N=[N+]=[N-] 80866,C1(OC)CCCC(=O)O1.C(c1cnc[nH]1)=C(C)C(=O)N(C)C 80867,C1(CNC(C(CC)NC(N)=O)=O)CN(C(=O)Cc2ccsn2)C(C)(C)C1 80868,c1(C2C(C)C2)cn(CCNC(C2(CF)CC2)=O)nn1.C1CC(=O)NO1.C(N)=O 80869,c1(C(=O)NCC(C)CNC(C2CCC2C(C)(C)C)=O)ncoc1-c1ccccc1 80870,N1(C(CCC=C=C)=O)CCOCC(F)(NC(=O)Cc2csc(N(CC)CC)n2)C1 80871,C1(C(=O)NC2C(n3cc(CCCCC)nn3)COC2)CCCC(C)CC1 80872,C1(n2cc(C)nn2)(C(=O)OC)CCN(C(C)=O)CC1.C1(C)(CC2CC2)CCC1 80873,N#Cc1ccc(C(=O)NC2CCCC2NCc2nc(Cl)ccc2F)c(O)c1 80874,CC1CCCC1C(=O)NC1CCC1C(=O)NC1CC(CN(C)C)C1 80875,N1(C(C2CCCN(C(=O)C#CC3CCOC3)CC2)=O)CCc2cncnc2C1 80876,C1(CNC(C(CC)N(C)C)=O)CCCCN1C(=O)CCc1cccc(O)c1 80877,N1(C(c2cc(C(N3CC=CC3(C)SC)=O)oc2)=O)CCC2(CCC2)C(O)C1 80878,C#CCC(C(=O)N1CCC(C(=O)N(C)CC2CCCCC2O)C1CC)C1CC1 80879,C#CCC(CO)NC(=O)CN(C(=O)C(CO)NC(=O)C(C)OC)C 80880,C#CC1(C(=O)NC(CCN(C(=O)Cc2ncc(Cl)s2)C)C(C)C)CCCC1 80881,Cc1ccc(C(C(N2CCCC2CNC(c2[nH]cnc2C#N)=O)=O)C2CC2)cc1 80882,C#Cc1ccc(C(N2CCN(C(=O)C(n3nccc3C)C)C(CO)C2)=O)c(C)c1 80883,Cc1ccc(NC(=O)CC2CN(C(C3CCCS3)=O)CCO2)nc1C 80884,c1(SCC(O)Cn2ccc(-c3cccs3)n2)ccc(Br)c(Cl)n1 80885,N1(C(C2(OCC)CCCC2)=O)C2CCC(C(N)=O)C1C2.c12cccc(c1)C(=O)N2 80886,N1(C(C(c2ccncc2)C)=O)CC(O)(CCNC2CCCN2CCC#N)C1 80887,C(C)(C)(CCCO)NC(C1(CNC(C2CCC(C)O2)=O)CC(=C)C1)=O 80888,C1(O)(C(C)NC(C2CC2(C)C)=O)CCN(C(=O)CC2CCCC(=O)C2)CC1 80889,Cc1sc(C)c(C(=O)NCCN(C(C2CCCOC2C)=O)C(C)C)c1C#N 80890,c1(C(=O)NC(CN(C(CC(C=C)c2ccccc2)=O)C)C)nc(Cl)c(=O)[nH]c1N 80891,CC1(C)CCC1CNC=O.C12COCC1n1cc(nn1)CCC(=O)N2 80892,n1(CC)cc(C(=O)NCCN(C2CCCCC2)C2CC=CCC2)cn1 80893,C(N=c1cc[nH]cc1[N+](=O)[O-])c1nc(CNC(=O)NC)nc(O)c1.C1(C)C(=O)N1 80894,C1(C2CCN(C(COCC(=O)NC)=O)C2)CCCCN1C(c1c[nH]c(=O)cn1)=O 80895,c1(C(N2CCC(F)(c3ccccc3)C2)=O)cccc(N2CCCS2(=O)=O)c1 80896,C(CCO)(C(F)(F)F)NC(C1C=CCN(C(c2nn(CC)c(O)c2)=O)C1)=O 80897,C(C(O)C(F)(F)F)NC(=O)CCC1CCN(C(c2ccc(C3CC3)o2)=O)C1 80898,C(N=c1c(Br)c[nH]cc1[N+](=O)[O-])C1CC(NC(C(C)C(C)S(C)(=O)=O)=O)C1 80899,C1(C(N2C(CNC(c3cscc3Cl)=O)CCCC2)=O)CCCCC12CC2 80900,CC1(C(=O)NC2CC2NC(=O)Cc2cccc(F)c2)CC=CCC1 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80919,N1(C(c2cc(C)nc(C)n2)=O)CCN(C(c2n[nH]cc2N(C)C)=O)C(C)C1C 80920,Cc1nn(C)c2c(NCCCc3cnn(C)c3)nc(=NCC3CCCC3O)[nH]c12 80921,c1(SC)cccc(N(C2CC3CC2CN3)C)n1.C12CCC(CC1)NC2=O 80922,C1(C(C)C)(NC(c2nccn2C)=O)CCN(C(C23CC(O)C2C3)=O)CC1 80923,N1(C(C2(CCC)CC2)=O)CCC2(CCCCC2NC(C2CCCCN2C)=O)C1 80924,c1(C(=O)NC(c2n(CC)cc(Br)c2)=O)ccc(C)c2c1CCCN2 80925,c1(C(=O)NCC(CNC(c2ncsc2Br)=O)OC)ccc2c[nH]nc2c1 80926,CCC(CC1CCCC1)C(=O)NCCN(C)C(c1c[nH]nc1-c1cccnc1)=O 80927,CC(C)CCC(=O)C(=O)NCC1CCCC(CNC(C2CC(F)(CO)C2)=O)C1 80928,c1(C(=O)NC(c2ccc(NC(=O)C3CC3)cc2)C)cc2cc[nH]c(=O)c2s1 80929,c1(C(N2C(C)CC(CNC(CC3(OC)CC3)=O)C2)=O)ccc(OC)c2ccsc12 80930,C(=O)(CCS(C)(=N)=O)NC(C1CCCC1)CNC(c1cn(C(C)C(=O)O)nn1)=O 80931,C1(C(=O)NCCC2(NC(CC3CCN(C)C3)=O)CC2)CN=C2N=CNN2C1 80932,CCC(F)(F)C(C)(C)C(=O)NC1CC(CC(=O)NCc2cn(C3CC3)nn2)C1 80933,C(=O)(CC1CCc2ccc(O)cc21)NC1CC(O)(CNC(CSS(C)(=O)=O)=O)C1 80934,c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)sc2cc(F)ccc2c1Cl 80935,CC(C)CC(C)(C)C(=O)N1CCC1C(=O)Nc1ccc2[nH]ccc2c1 80936,CCC(C(=O)OC)N(C(=O)CC1CSC1)CCCC(CNC(=O)C(C)C)(C)C 80937,c1(OCCC)ccc(CNC(=O)CCCN(C(C)C)CC)cc1OC 80938,c1(C(=O)NC(CC)CNC(=O)C(C)C(=O)OC)cccc(C=C(F)F)c1 80939,C1(NC(C2(SC)CC2)=O)CC(C)CN(C(C2(C)CC(F)(F)C2)=O)C1 80940,CCC(CC)(CCC(=O)N(CC(O)CNC(=O)Cn1cncc1C)C)[N+](=O)[O-] 80941,c1(CC(=O)N(CC(C)O)CCNC(C2CCC2)=O)ccc(C2CC2)cc1 80942,C1(C)(CN(C(=O)CCCc2ccsc2)C)CCC(=O)N1.c12csc(c1)CNC2=O 80943,N1(C(CN(C(C(C)CC2CCC2)=O)C2CC2)=O)CC(C)C(C)(CO)C1 80944,C1(NC(C(C)OCCOCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C 80945,c1(C(N2C(C(C)NC(=O)C=Cc3cc[nH]n3)CCC2)=O)cncc(O)c1Cl 80946,C12(CNC(C3CCCC3)=O)CN(C(c3cc4cccnc4s3)=O)CC1CCO2 80947,c1(C(=O)NC2C(NC(Cc3n(C)ncc3)=O)CCOC2)ccc2c[nH]nc2c1 80948,Cn1c(=O)n(C)c2c(NC(C3(C)CCN3S(=O)(=O)c3ccc(Br)s3)=O)cccc12 80949,N(C1CCCc2n[nH]cc21)C(C1N(C(CCC(=C)Cl)=O)CCC(C)C1)=O 80950,c1(NC(C(CSCC)NC(C2CC(C)(C)C2)=O)=O)ccc(C)nn1 80951,N1(C(C=C(C)C(C)(C)C)=O)CCN(C)C(C(=O)NCc2nn(C)cc2C)C1 80952,C(=O)(CCCC(C)(C)C#N)N1CCC(CNC(CC2CC(CC)C2)=O)C1 80953,C12(C(=O)Nc3n(CC)nnn3)CC(CO)(CN1C(c1ccnn1C1CC1)=O)C2 80954,CCS(=O)CC(=O)NC(C1CCCCC1)CNC(=O)CCC(=O)OC 80955,CC(C)CC(C)(C)C(=O)NC(CNC(c1cnc(O)n1C)=O)C1CC1 80956,C12CCN(CC1C)C2=O.C1(C(=O)OC)CCN(C(=O)c2nc(Cl)oc2C)O1 80957,C#Cc1ccc(CC(=O)NCC(C)C(F)C(=O)NCc2ccc(O)c(F)c2)cc1 80958,C1(C(=O)NC(CCC)CCCNC(c2ccsn2)=O)CCc2ncc(C)n2C1 80959,Cc1nn(C)c2c(N3CC(C)C(F)C3)nc(=NCCCOC3CCOC3)[nH]c12 80960,N(C1CC2(CC(NS(=O)(=O)c3sccc3C#N)C2)Oc2ccccc21)C(C)C 80961,c1(C(N(C2CCC(NC(C(CC)C(C)C)=O)CC2)C)=O)cnc2sccn2c1=O 80962,N1(C(C(CCC)C)=O)CCN(C(c2ncc(OC)cn2)=O)CC(O)C1 80963,c12cc(I)c(Cl)cc1NC2=O.N1(CC)CCN(C(=O)Nc2csc(Br)c2)CC1 80964,CC1CC(C)CN(Cc2ccc(-c3ncc(Cc4ccccc4F)s3)cc2)C1 80965,c1(CC)cncc(C(=O)NCCC2(O)CN(C(=O)C(O)Cc3cn(C)cn3)C2)c1 80966,C(C(O)CCNC(C1C=CCS1)=O)NC(c1cnc(C2CCCO2)s1)=O 80967,C1(C2CCN(C(=O)CSC(F)(F)F)CC2)(NC(c2cc(C)n(C)c2)=O)CC1 80968,N1(C(C2C(C)OCC2)=O)CC2(CC2)CC1CNC(c1ccc(CO)cn1)=O 80969,Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCCC1NC(C1CCCN1C1CC1)=O 80970,CC1CCN(CC(N2CCC(C(=O)NCC3(Cl)CC3(F)F)C2C)=O)CC1 80971,CC1CN(C(=O)Cc2csc(Br)c2)CCN1C(=O)C(C)(C)CC#N 80972,C1(C(C)C)C(=O)N1.C(CC(C)CCNC(=O)C=C(Cl)Cl)NC(C)=O 80973,C(C)(c1cccc(Cl)c1)=CC(N1CC(C)(NC(C2C(OCC)C2C)=O)C1)=O 80974,N1(C(CCCCCNC(c2nccc(C#C)c2)=O)=O)CC2(CCCN2C)C1 80975,CC1(C)CN(C(=O)Cc2cc(Cl)ccc2Cl)CC1NC(C1(O)CCOCC1)=O 80976,N1(C(CNC=O)=O)CCSCC1C(=O)NCc1cncs1 80977,CC1CN(C(C2C=CC=CC=C2)=O)CC2(CCN(C(c3cc(F)cc(F)c3)=O)C2)O1 80978,C(=O)(C1=CS(=O)CCC1)NCC(C(C)(C)C)NC(COCC(C)(C)C)=O 80979,c1(-c2ccc(N(CCCC)CC)cc2)cc(C)ccc1S(N)(=O)=O 80980,CC1(C)CCCC1CNC(c1csc(CNC(c2scnc2Cl)=O)c1)=O 80981,C12(NC(C(C)OCC=C)=O)CC(CNC(c3csc(Cl)c3)=O)(C1)OC2(C)C 80982,C1(C(=O)NCCn2cc(C3CCOC3)cn2)CC2(C1)CC1CCC2O1 80983,C(C(=O)NNC(=O)CNc1nnc2cnccn12)OC(CC)(C)C 80984,CCC1=NOC(C(=O)N(CCCNC(c2snc(Cl)c2Cl)=O)C(C)C)C1 80985,N1(C(c2nn(C(F)F)cc2Cl)=O)CCC(NC(c2cc(OC)ncn2)=O)CC1C 80986,C1(CNC(Cc2cc(C)sc2)=O)CCCCCN1C(=O)C=CC(=O)OC(C)(C)C 80987,C(C(C)(O)C(=O)NCC1CN(C(c2c(C)cnn2C)=O)CCO1)OC 80988,c1(C(=O)NC(CNC(CCCOC)=O)(C)C)nccnc1C(N)=O 80989,N1(C(C(C(C)C)Oc2ccccc2)=O)CCOc2c(Cl)cncc2C1 80990,CCCCCCCC(=O)N(CCC)CCNC(=O)CCC(F)F 80991,N1(C(C(C(CCC)NC(=O)CC(C)(C)CC)O)=O)Cc2ccc(O)cc2C1 80992,CC1Cc2cc(Br)ccc2N1C(=O)N(C1CC(c2ccccc2)C1)C 80993,c1(C2C(C(=O)NCCN(C(CNS(N)(=O)=O)=O)C3CC3)C2)ccccn1 80994,c1(C(=O)NCC2(C(N3CC(C(C)(C)O)C3)=O)CC2)cccnc1C(F)F 80995,N1(C(COCc2nnc(C)s2)=O)CC(NC(c2cccnc2C)=O)C(C)C1 80996,CC1CN2CCN1C(C(=O)NC(C)CN(C(=O)COc1cccc(F)n1)C)C2 80997,N1(C(c2nc(CC)oc2C)=O)CCN(C(=O)C(C)CCc2ccccc2)CC(O)C1 80998,C1(COC)CCCCN(C(CCC2OCCO2)C(=O)NC(C)COC)C1 80999,Cc1sc(O)nc1C(N1CC(CC(=O)NC(c2cn(C)nn2)C)CC1C)=O 81000,c1(C(N2CCCC(COC)C2)=O)ccc2c(C)cc(Cl)nc2c1 81001,N1(C(C2(C=C)CCC2)=O)CCC(NC(C)=O)C(C)C1.C(=O)(CN(C)C)N 81002,O=C(C1=C(Cl)CCCC1)N1CCCC(CCCCNC(C2(O)CC2)=O)C1 81003,N1(C(C(C=C)CC)=O)CCC(C)C(CC(=O)NCCC2(C)CCOC2)C1 81004,C1(C(=O)NCC(C)NC(=O)CC2CC3(CC3)CO2)CCC(C(N)=O)N1C 81005,c1(C(=O)NCC2N(C(c3cc(C)cc(O)n3)=O)CCOC2)ccn2ccnc2c1 81006,c1(C(N2CC(O)(CNC(C(CC)OC)=O)C2)=O)cc2n(n1)CCCC2=O 81007,c1(C(N2CC(C)(NC(=O)CCC3CCCC(=O)N3)C2)=O)cnc2nccnc2c1 81008,N1(S(c2ccc(N3C4CC(C)CC3CC4)nc2)(=O)=O)CC(=O)N2CCCCC2C1 81009,c1(C(N2CCC(NC(C(C)SCC)=O)CC(O)C2)=O)cc(O)nc2ncccc12 81010,C1(C(=O)NC(C)Cc2cnccn2)CC=CC(NC(=O)CN=[N+]=[N-])C1 81011,Cc1nc2c(C(N3CCC(C)C(NC(=O)C(C(C)O)N(C)C)C3)=O)ccnc2[nH]1 81012,C1(CC)CC(C(N2CC=CC(NC(c3ccccc3SC(F)F)=O)C2)=O)CCO1 81013,N1(C(CCOCCCC)=O)CCCC2(CCCCC2NC(=O)CC(C)N(C)C)C1 81014,C1(C(=O)NC(C(C)(F)F)(C)C)CCc2cc(S(N)(=O)=O)ccc2O1 81015,Cc1cc(C)n(CCC(=O)NCC2C=CCN2C(=O)Cc2c[nH]nc2C)n1 81016,C1(CC#C)(C(=O)N(CC(C)(C)NC(=O)Cn2cc(Br)cn2)C)CCOC1 81017,S(=O)(=O)(c1ccsc1C(=O)NCCOCCn1cc(COC)nn1)NC 81018,Cc1cc(C(N2C(CO)CCC2C)=O)nnc1O.c12cc(no1)C(=O)NCC2 81019,C#CCC(C)C(=O)NC1(CO)CN(C(C2CCOC(c3ccccc3)C2)=O)C1 81020,N1(C(CC(C)SC)=O)CCN(C2CCN(C(c3ccnnc3O)=O)C2)CC1 81021,Cc1nnsc1-c1noc(C(N)CCC2CC2C)n1 81022,c1(OC)cc(C(N2CC3(NC(=O)C(=O)NCC4CC4)CCC2C3)=O)cnc1O 81023,C1(=O)C(O)CCCO1.C1(NC(=O)OC(C)(C)C)SC2C=CC1CC2 81024,N1(CCN(C(CC#C)=O)C)CCN(C(c2ccc(C3CC3)o2)=O)CC1 81025,N1(C(Cn2c(=N)nc[nH]2)=O)CC(O)CC1C(=O)NCCc1ncc[nH]1 81026,N1(C(C(C=C=C)C)=O)CCCN(C(c2cccc3ccnn23)=O)CC1CO 81027,N1(C(c2cnn(CC)n2)=O)CC(NC(=O)CCc2cccnc2)CC12CCOC2 81028,Cc1ccc(Br)c(CN2CC(C)(C(N3CCS(=O)(=O)CC3)=O)C2)c1 81029,c1(C(=O)NC2(CNC(c3c(N)cncc3)=O)CC2)cc2c(F)ccc(F)c2[nH]1 81030,CC1(C)CC(NC(=O)C(O)C(F)(F)F)CN(C(C2C3CCCC23)=O)C1 81031,C(C(C)(C)C(F)(F)F)NC(C(C)(C)CNC(=O)CC1(O)CCCC1)=O 81032,C1(CC)(NC(=O)C(O)c2ccsc2)CCN(C(=O)CCC(=O)c2cnn(C)c2)C1 81033,C1(NC(C(C)Sc2ccc(C(=O)N)nc2)=O)CCCCC1n1cc(C(N)=O)nn1 81034,CC(C)CC(C(=O)NCc1cccnc1F)N(C)C(C1CC12CCOC2)=O 81035,CC(CCC(C)(C)C)C(=O)NC12CCCC1N(C(=O)CC1C=CCCC1)CCC2 81036,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(F)(F)C2)=O)ccc2cnccc2n1 81037,Cc1nc(Cl)ccc1S(=O)(=O)N1CCn2nc(-c3ccc(N(C)C)cc3)cc2C1 81038,N1(C(CC(C)O)=O)CCC(N(C)CCNC(C23CCOCC2C3)=O)CC1 81039,C1(NC(C(C2CC2)OCC)=O)CCOC(C(=O)NCCC2CC2)C1 81040,C1(N(C(=O)CSC(F)F)CCC)CCN(C(=O)C=Cc2ccnn2C)CC1 81041,CS(=N)(=O)C1CN(C(=O)C(=O)NC2CCCCC23CC3)C1 81042,Cn1ncc2c1CC(C(N1CC(NC(c3cc(C#N)c[nH]3)=O)C(C)(C)C1)=O)CC2 81043,CC(c1cccc(F)c1)=CC(=O)NC1(CO)CCCN(C(=O)Cn2cncn2)C1 81044,N1(C(C(CC)CC)=O)CCC(C(N2CCOCC2C)=O)C(C)(C)C1 81045,N1(C(C(CCCC)C)=O)CC(C2CN(C(c3ccnc(F)c3Cl)=O)C2)C1 81046,C(c1cc(C)no1)=CC(=O)NCCN(C1CCCCC1)C(C1CN(C(C)=O)C1)=O 81047,C1(CNC(=O)OCC)CCN(C(=O)Cc2ncc(C(=O)OC(C)(C)C)s2)CC1 81048,c1(C(N2CCC3C(NC(C=CC(C)(C)SC)=O)C32)=O)cc(O)ccc1C 81049,c1(C(N(C2CN(C(c3cn(CC=C)nc3)=O)C2)C)=O)cn2c(n1)CCC(C)C2 81050,C(=O)(C(C(C)(C)C)N(C)C)NC1C(CNC(C2(CC=C)CCC2)=O)C1 81051,n1(CCOC)cc(C(=O)NC(C)C(C)(C)NC(=O)CCc2cc[nH]n2)c(C)n1 81052,C=C(C)CC(C(=O)NC1CC(c2ccn(C)c2)C1)NC(C1CC2CC(=O)C1C2)=O 81053,c1(C(=O)NC(C(C(=O)N(CC#CC)C)C)C)cncc(F)c1C 81054,CC(C)(C)C(CO)C(=O)N1CCCCC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)C1 81055,O=C(O)CCC(C[N+](=O)[O-])N1CCCC(Nc2nc3ccccc3o2)C1 81056,C(C)(CC(=O)NC1(C)CC(NC(=O)C(C)(F)c2ccon2)C1)SC 81057,c1(NC2CC(CNC(C3(O)CCCCCC3)=O)C2)ncnc2ccc(Cl)cc12 81058,C1(CCC(=O)N(CCCNC(c2ncc[nH]2)=O)CCC)CCCCC1 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81076,N1(C(C2CCCC(NC(C3CN(C)C(=O)CC3)=O)C2)=O)Cc2cccc(C#N)c2C1 81077,c1(C(N(C2CCN(C(C(C)OCCC#C)=O)C2)CC)=O)nn(C)cc1SC 81078,C1(NC(CC(=O)NCC)=O)CCN(C(C2CC(C)(C)CO2)=O)CC1O 81079,C1(CC(N2C(c3n(CCCCCC)ccn3)CC2)=O)CCC(F)(F)C1 81080,C1(C(=O)NC(c2cn(CCO)nn2)CCC)CNC(=O)N1C 81081,C12(C(=O)NCC3N(C(C4C=CCC4)=O)CCC3)CC3CC(CC(C3)C1)C2 81082,C1(CC(=O)NC2CCCC2)CN(C(=O)C(N)CN2CCC2)CC2(CCC2)O1 81083,c1(C(C)C(=O)NCCOCCNC(=O)Cc2cncs2)ccnn1C 81084,C(=O)(C(CC(C)C)NC(=O)C(C[NH+])NC(=O)CC1CCOCC1)OC.C(C)(=O)N 81085,CON(CCCO)C(=O)C(c1cn(C)nn1)NC(c1cnsn1)=O 81086,N1(CC(C)N(c2ccccc2)C)CCN(C2CCN(C)CC2)CC1 81087,C(CC(C)C)(C(=O)C(C1(NC(C)(C)C)CC1)=O)NC(N(C)C)=O.C12(C)CN(C1)C2 81088,CCCC(C(=O)NCC1CCC1NC(=O)Cc1ccsc1Cl)c1cccc(Cl)c1 81089,C1(=O)C(COC)C(CC)C(CNC(CN(CC)CC)=O)SCCN1C 81090,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2Cl)=O)(C)C)cc(F)cc(C)c1O 81091,C#CC1CCCN(C(C2(NC(c3cc(C)ccc3C)=O)CCC2)=O)C1 81092,c1(OCC)c(Cl)cc(C)nc1C(=O)NCC(C(C)(C)C)NC(=O)CCCN=[N+]=[N-] 81093,N#Cc1cncc(CC(=O)NCCSCC(=O)Nc2conc2C(N)=O)c1 81094,C1(C(N2C(C)(C(=O)NC)CC2)=O)CC(O)C(O)CC1CNC(C1(O)CC1)=O 81095,N1(C(C(C)C2CC2)=O)CC(CNC(c2ccc(NS(C)(=O)=O)o2)=O)OC(C)(C)C1 81096,N1(C(CCCOC)=O)CC(CNC(c2cccnc2SC)=O)C2(CC2)C1 81097,C12(C(=O)NC3CC(CNC(C4CC(OC(C)(C)C)C4)=O)C3)CC1COC21CCC1 81098,c1(C(C(N2C(C(C)NC(c3ccsc3C(F)(F)F)=O)CC2)=O)C)ccc(F)c(F)c1 81099,C1(C)(C(N2C(CNn3cc(CCN(C)C)nn3)CCC2)=O)CS(=O)(=O)C1 81100,c1(OC)ccc(Br)c(C(=O)N(CC(c2cccc(Br)c2)O)C)c1C 81101,CC(C)(C)C(CNC(=O)CCCc1ccccn1)NC(=O)C(c1ccccc1)F 81102,N1(C(CCC=CC)=O)CC2(CC(NC(=O)CCc3nccn3C)CO2)C1 81103,c1(N2CCCC(CN(C(=O)CCC[N+](=O)[O-])C)C2)ncnc2c(F)c(F)ccc12 81104,c1(C(=O)NC2CC(C(=O)Nc3c(C(N)=O)ccs3)C2)cccc(O)n1 81105,c1(C(N(C)CC2(NC(c3ccc(C)c(F)c3)=O)CC2)=O)cnc2c(c1)OCCN2 81106,C(=O)(Nn1cnn(CC)c1=O)c1n(CCN2C(CC(=O)OC)CC2)cnn1 81107,c1(C(C(=O)NC(C)Cn2ccnc2)N(N2CCOCC2)C)ccc2c(c1)CCC2 81108,c1(CC)nn(C)c(C)c1C(N1CCC(N(C(=O)Cc2ncccc2C)CC)C1)=O 81109,N1(C(C(c2n(C)ncc2)(C)C)=O)CCCC(C2(NC(=O)CC(C)(O)C3CC3)CC2)C1 81110,c1(C(C)C)cnc(Cl)nc1N1CCCCC(NC(=O)C(C)CN2CCOCC2)C1 81111,c1(CC2CN(C(C(n3ncc(C)c3)C)=O)C2)cnc(N)c(-c2nn[nH]n2)c1 81112,CC1CC(C(=O)Nc2cnn(-c3ccc(Cl)cc3)c2)=NO1.C12CN(C1)C2=O 81113,N1(C(C2CC(C)(F)C2)=O)CCC2(CCN(C(C3CC(OC(F)(F)F)C3)=O)C2)C1 81114,N1(C(Cn2cc(CCN(C)C)nn2)=O)CCC12CCC2 81115,c1(CC)cnc(Cl)cc1Cl.CC1(C)CCCC(=O)N1.C1(CC(=O)N)CC(O)C12CCC2 81116,N1(C(CCCN(C)C)=O)CCN(C(c2ncn(C(C)(C)C)n2)=O)C2CC12 81117,c1(CCC(=O)N(CC(C)Cn2ccnc2)C2CC2)ccccc1OC(F)(F)F 81118,c1(OC)ccccc1NC(=O)C(=O)N(CCCNC(=O)C=CCSCCOC)C 81119,Cn1cnc2c(N3CC(NC(=O)CCCn4cccn4)C3)nc(Cl)nc12 81120,c1(C(=O)NC2CN(C(CC3(C#N)CC3)=O)CC2F)c(O)cccc1F 81121,N1(C(CCOC(C)=O)=O)C2CCC1C(CNC(=O)C(c1ccc(F)c(C)c1)=O)C2 81122,c1(C(=O)NC2CN(C(Cc3c(OC)ccnc3)=O)CC2O)cnc2nccn2c1 81123,C1(N(C(C)C(N)=O)C)CCCCCC1.n12cc(nn1)C1(CC1)C2 81124,Nc1cccc(F)c1C(=O)NCC1CC1NC(=O)COCC(F)(F)F 81125,c1(C(=O)OC)cc2cc(NCc3cn(-c4ccn(C)n4)nn3)ccc2cn1 81126,CCCC(C)CN=C(NC(=O)NC1CCCO1)NC1CCN(C2CC2)CC1 81127,c1(C(=O)NCc2c(C(N(CC(F)F)CC#C)=O)c[nH]n2)sc(F)cc1C 81128,CC(C)(C)CC(O)C(=O)NCC1COCC1NC(C1SC2C=CC1CC2)=O 81129,C1(CC)CN(C(C2CC(=O)N(C)C2)=O)CCC1CNC(c1nc(C)oc1OC)=O 81130,N1(C(C=C(COC)C)=O)CCC2(CC1)CN(C(=O)CC1CC1C)CC(C)O2 81131,C1(CNC(c2nc(CC)[nH]n2)=O)CN(C(C2CCN(C(C)=O)C2)=O)C(C)(C)C1 81132,C12(NC(c3ccc(C)c([N+](=O)[O-])c3)=O)COCCC1CN(C(=O)COC(C)C)C2 81133,Cc1cccc(CC(=O)NC(CNC(=O)Cc2c(C)noc2C)CO)c1F 81134,C1(N(c2ncccn2)C(c2c(C)cc(Cl)cc2)=O)CCNCCC1(F)F 81135,C1(C(=O)NC2(CCC)CC2)C2CCC(C2)N1C(=O)CCc1ccc[nH]1 81136,N1(C(C)C)CCCC(CC(=O)NCC(C(C)(C)C)NC(c2cccnc2O)=O)C1 81137,Cc1ccc2c(CC(N3CCN(C(=O)CCn4cccn4)C4CC34)=O)c[nH]c2c1 81138,C=CCC(CC(F)F)C(=O)N1CCCC1CCNC(c1ccc(CC)nc1)=O 81139,C1(C(=O)OC)CCN(Cc2ccccc2C(F)(F)C(=O)OC(C)(C)C)CC1(C)C 81140,C(CC(=O)N1CCC(N2CC=CC2)C1)(C(F)F)NC(Cc1nc(C)sc1)=O 81141,C1(C(=O)NC(C2CCN(C(=O)CCC3CC3(Cl)Cl)C2)C)CCS(=O)CC1 81142,N1(C(COCCC=C)=O)CC2C(C(=O)NCC(N3CCCCC3=O)C)C2C1 81143,c1(C(=O)NC2CC(NC(c3cc(OC)ncn3)=O)C2)cccc2oc(C)nc12 81144,C(=O)(CC(C(C)(C)C)NC(=O)C(O)CC1CCCC1)NCC(C)CC1CC1 81145,C1(N(C(=O)C(F)OC(F)(F)F)CC)CCC(NC(=O)C(O)CSC)CC1 81146,N1(CCNC(C(CC)n2ccc(C3CC3)n2)=O)CCC(NC(=O)C(C)C)CC1 81147,c1(C(=O)NC2(C)CCCN(C(C(C(CC)O)C)=O)C2)n[nH]c2c1COCC2 81148,c1(C(=O)NC2CCC2)ccnc(OC)c1.c1(C(=O)OCCCS)ccc(C2CC2)o1 81149,N1(CC(C)NC(C)=O)CCN(C(=O)CCCC(N)=O)CC1c1ccc(Cl)cc1 81150,c1(C(c2nnnn2C2CCOC2)NS(CCOC)(=O)=O)cnn2c1CCCC2 81151,C(=O)(CC(CNC(C1(OC(C)(C)C)CCOC1C)=O)OCC)OC 81152,c1(OC)ccn2ncc(C(N3CCCC(NC(=O)C(C)C4CC4)CC3)=O)c2c1 81153,C#CCC(C)(C(=O)NC(c1ncc(C)[nH]1)CC)NC(c1cnc(Cl)s1)=O 81154,CC1(CNC(C2C3CCCCCC23)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 81155,C1(CN=[N+]=[N-])CCCN(C(=O)C(C2CCN(C(c3cc[nH]c(=N)n3)=O)C2)F)C1 81156,C1(CNC(C2C(C)(Br)C2)=O)CC2CCC1N2C(=O)C(C)(Cl)Cl 81157,c1(C(=O)OC)cc(-c2onc(CCN)c2C)c(Cl)cn1 81158,N1(C(=O)CNC(=O)OC(C)(C)C)CCC2CCCOC2(CC(=O)NCCCC)C1 81159,Cn1ncc2nc(Cl)nc(N3CCCC(CCNC(=O)CCOCC(F)F)C3)c12 81160,N1(C(C(C)OCCOC)=O)CC2C(CC(=O)NCCCCCF)C2C1 81161,N1(C(C2CCC(C)(C)CC2)=O)C2CCC1C1CC1(NC(=O)CCc1cnn[nH]1)C2 81162,CCC1=C(C(=O)NCC2CN(C(C3Cc4nnc(C)n4C3)=O)CCO2)CCCO1 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81600,N1(C(Cc2cnc(C)o2)=O)CCCC2(CCC(NC(C3(C)CC(F)(F)C3)=O)C2)C1 81601,C1(C(=O)NCC(=O)N(c2ccc(NC=O)cc2)C)(C(=O)O)CCOC2(CCC2)C1 81602,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 81603,c1(C(N2CC(C)(C(=O)NC(CCSC)CO)C2)=O)cc(C)c(F)cn1 81604,C1(CNCC(C(=O)OC)C)CC(O)CN1c1nccc(-n2cc(C)cn2)n1 81605,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 81606,C1(C(=O)NCC2CC(O)CN2C(=O)CCc2ccc(F)nc2)CCC2CC2CC1 81607,C(=O)(CC(C)(C)CC(=O)NCC=CCNC(C1CCC1(F)F)=O)OCC 81608,c1(C2N(C(=O)NCC3(C)CN(CC(=O)OCC)C3)CCC2)nc(C)n(C)n1 81609,N1(C(COC(CC)C)=O)C(CNC(c2ccc(C)nn2)=O)CC2COCC12 81610,N1(C(c2cc(CC)on2)C(=O)NCc2cccs2)CCCCC1c1cncnc1 81611,N1(C(c2c(CC)c[nH]c2)=O)CCOC2CCN(C(c3ccc(SC)cc3)=O)CC12 81612,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 81613,c1(OC)cccc(C)c1C(=O)NCC1CC(OC)CN1C(c1cc(N)ccn1)=O 81614,c1(OC)cc(F)c(S(=O)(=O)Nc2ccc(F)cc2OC(C)C)cc1F 81615,n1(CCOC)cccc(C(N2CCOC(Cc3nn[nH]n3)C2)=O)c1=O 81616,C1(C(C)CO)CCN(C(C2CCC(NC(=O)CCn3cncn3)CC2)=O)CC1 81617,C1(C(=O)NC2(C)CCN(C(=O)Cc3ccnc(O)c3)C2)COCCN1C=O 81618,N1(C(C2C(NC(COC3(C)CCCC3)=O)C=CCC2)=O)CC2CCC(C1)O2 81619,c1(OCC)ncc(Br)c(N2CCC(COc3cccc(C)c3F)C2)n1 81620,C12(C(=O)NC3CC(N(C(C(C)Cc4ccncc4)=O)C)C3)CCC(C1)OC2 81621,C(=O)(C(C(C)C)NC=O)NCc1cn(CC(C)NC(C2CC(=O)N(O)C2)=O)nn1 81622,c1(C(N2CC3CCN(C(CC(CCC)C)=O)CC32)=O)cc2c(nn1)OCCS2 81623,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)O)NC(=O)C2CCC12 81624,c1(C(C(=O)NC(C)C(CO)NC(=O)Cc2ccc(Cl)s2)C2CC2)ccc(F)cc1 81625,c1(N2CC(O)(CCNC(C3CCC(C)C3)=O)C2)cc(F)ncn1 81626,C1(CNC(CS(C)(=O)=O)=O)C2CCC(C2)N1C(=O)Cn1cc(Br)c(=N)[nH]1 81627,C(=O)(CCCCC(F)F)N1C(CN(C(c2ccc(C(=O)OC)[nH]2)=O)C)CCC1 81628,N1(C(COC(C)C)=O)CCC(O)(C(C)NC(=O)CCc2cnn(C)n2)C1 81629,Cn1cc(C(=O)N(CC(N)=O)Cc2ccc(Cl)cc2)nc1O 81630,C1(OC(c2cncc(OC(C)(C)C)n2)=O)CCC=CCCC1 81631,C(c1cccc(Cl)c1)=CC(=O)NCCCOCCCNC(C1(C)CC1)=O 81632,C1(NC(C2CCCC3(CCC3)C2)=O)CN(C(C2CC(F)(F)C2)=O)C2CCCCC12 81633,N1(C(c2cncc(COC)c2)=O)CC(NC(=O)C(C)(F)F)CC12CCOC2 81634,c1(CC(=O)NC2CCCC(CN(C(COC(CC)C)=O)C)C2)ccc(C#N)nc1 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81809,CC1CCN(C(=O)CC2CC(C)(C)C2)CC1CNC(c1cc(N)nc(Cl)c1)=O 81810,N1(C(c2c(C)ocn2)=O)CC(CNC(=O)C(O)C2CCCC2)C(S(C)(=O)=O)C1 81811,CC(F)(F)C(C)(C)C(=O)N1C2CCC(C(N3CC(n4cnnn4)C3)=O)C1CC2 81812,CS(=O)(=O)C1CC(F)(C(N2CC(OCCNC(=O)CCc3ccccn3)C2)=O)C1 81813,Cc1ccc(F)c(C(=O)N(C)CC2CCCN(C(C3CCC(C)O3)=O)C2)c1F 81814,Cc1cc(C(N2CCC2CNC(=O)C(C)(O)c2ccccn2)=O)nn1CCO 81815,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC23CC3)cc2c(s1)CCCC2 81816,Cc1c(C(N2CCC(O)(CNC(c3cncnc3)=O)C2)=O)cnn1C1CCC1 81817,C1(NC(C(C)Cc2cccc(Cl)c2)=O)CCC(C)N(c2nnc(C(C)(C)C)s2)C1 81818,C1(CNC(=O)Nc2nc3ccccc3[nH]2)COC2(CCCC2)OC1 81819,c1(C(N2CC(CNC(=O)C(F)CC3CCC3)C2)=O)c[n+]([O-])ccc1[N+](=O)[O-] 81820,C1(NC(C(=O)NC(C)C)=O)CCOCC1C(=O)NCCOC(=O)C1CC1 81821,n1(CC(=O)NCC(CC)NC(c2ccc(N)cc2F)=O)cc(C)c2ccccc12 81822,C1(C(=O)NCC2CCN(C(c3c[nH]c(C(F)(F)F)c3)=O)C2)(C2CC2)CCOCC1 81823,C(=O)(C(F)(F)C(F)F)N1CCC(N(C(=O)CC2CCCOC2)CCC)CC1 81824,C(c1cnc[nH]1)=C(C)C(=O)NC(C)C(=O)NC1CC2(CC2)C1 81825,N1(C(CCCC(C)=O)=O)CCCC2(NC(=O)CCC3CCC(=O)N3)CC2C1 81826,c1(-c2cn(CC(=O)O)nc2)cc(NCc2ccno2)nc2ccccc12 81827,c1(-c2nnc(N(C(c3cccn3C)CC)C)n2C)cccc(F)c1C 81828,c1(NC(C)CN(C)C(c2c(O)cc(F)cc2F)=O)ncc2ncn(C)c2n1 81829,N1(C(c2c(C)cn(C)c2)=O)CCC(CO)(CNC(c2cnc(S)[nH]2)=O)CC1 81830,CCCCCC(O)C(C)C(=O)NCCCCN(C)C(c1ccn2ccnc2c1)=O 81831,Cc1cc(C(=O)NCC(F)CNC(=O)CCn2ccccc2=O)ccc1F 81832,C1(NC(C(C)SCC)=O)CC(F)(CNC(c2csc(-c3ccncc3)n2)=O)C1 81833,C1(CNC(C(CC)=CC)=O)CC(NC(c2cc(C(C)C)n(C)n2)=O)C(O)C1 81834,c1(C(N2C(CNC(C(C)C3CCOC3)=O)CCCC2)=O)cccc2nc[nH]c12 81835,N1(C(c2cc(CC)c(C)s2)=O)CCN(C(=O)C(N2CCOCC2)C)CC1C1CC1 81836,N1(C(COC)=O)CCOC2(C1)CN(C(=O)NC1(C)CCC1)C2 81837,C1(OC)(CNC(c2ccc(Cl)s2)=O)CCN(C(=O)Cn2ccccc2=O)C1 81838,C(CN=c1[nH]c(=NCc2ccnc3ccccc23)[nH]c2cc(C)ccc12)(C1CC1)OC 81839,CON(CCO)C(=O)C1(C)CCN(C(=O)Cc2cccnc2C)C1 81840,C1(CNC(C(C)CF)=O)CN(C(c2cc(C(F)F)on2)=O)CCC12CCC2 81841,C1(NC(C2C(C)CN(C(=O)C3=C(Cl)CC3)CC2)=O)CC2CC1CC2(C)O 81842,CC(C)C(C(=O)NC1CCN(C(c2cc(C(N)=O)co2)=O)C1C)n1cncn1 81843,C=Cc1cncc(C(=O)NCC2CN(C(=O)C(C)OC(C)(C)C)CCO2)c1 81844,c1(C(N2CCC(c3cccc(F)c3)(CO)C2)=O)ccc2ccc(Cl)nc2c1 81845,C(c1cc[nH]c1)=CC(=O)NCC1CC1NC(=O)CC1CC1C(F)(F)F 81846,C1(NC(C(CSC)OC)=O)COCCC1NC(=O)CC1CC(C)(C)C1 81847,C#CCCC(C(=O)OC)C1(C2(C(=O)OC)CC2)CCC1 81848,C1(C(=O)NC(CC(C)NC(=O)CC2COC(=O)N2)C)CN2CCN1CC2 81849,c1(C(N2C(CNC(CS(CC)=O)=O)CCCC2)=O)ccc2n[nH]cc2c1F 81850,C1(C)(CC)CCCN(C(=O)C(c2cn(C)nn2)NC(=O)CCC(C)=O)CC1 81851,C(C)(N=c1[nH]c(Cl)ncc1Br)C1N(CC(n2nnc(-c3ccco3)n2)C)CCOC1 81852,Cc1cc2c[nH]nc2cc1C(=O)NCCN(CC(C)O)C(C1CNC(=O)N1)=O 81853,c1(C(=O)NC(CNC(C2(C3CCCO3)CCC2)=O)C2CC2)cc(Br)no1 81854,C1(NC(c2ccc(C)s2)C2CC2)CCCC2(CC1)OCCO2 81855,c1(C(N2CC(CNC(C(C)(C)OC)=O)C(O)C2)=O)cc(C)c(N)cc1Cl 81856,C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(C2CCCC(C#N)C2)=O)C2CCCC2O1 81857,C12(NC(=O)Nc3cnn(-c4cc(CC)cc(F)c4)c3C)CC3CC(CC1C3)C2 81858,O(C=CC(=O)NCCN(C)C(c1ccn(CC)n1)=O)CC 81859,C1(NC(c2cccc(CC)n2)=O)CC2CC(NC(=O)C#CC3CCCO3)CC2C1 81860,Cc1ccc(F)cc1C(=O)N(CCC(=O)NCC(CNC(N)=O)OC)C 81861,C1(CNC(c2coc(C3CC3)n2)=O)CC2CCC1N2C(=O)CCn1cncn1 81862,C1(C(N2CCC(OCC3CC3)C2)=O)CCC(OCc2cccc(F)c2)CC1 81863,C(CCCC(=O)NC1CC(=O)N(COC)C1)N(C(COCC#C)=O)C 81864,CC(O)C(C(=O)NCC(=O)NCCN(C(=O)CCCCO)CC1CC1)N(C)C 81865,C1(C(N2CCC(O)(CNC(=O)CCc3nc[nH]n3)C2)=O)CCC2(CC1)OCCO2 81866,CC(C)CC(C(=O)N1CCCC(O)(CN(C)C)C1)NC(=O)CCNC(=O)CO 81867,N1(C(=O)N(C(CN2CCCC2)CO)C2CC2(F)F)CC(O)(CCO)C1 81868,c1(C(=O)NC(CN(C(C2CCC(C)(C)C2)=O)CC)C)cccc(N=[N+]=[N-])c1 81869,C12(NC(CS(N)(=O)=O)=O)CCN(C(c3cccc(-n4cncn4)n3)=O)CC1C2 81870,Cc1c(C(N2CCN(C)CC2CNC(=O)C(O)CF)=O)cccc1CO 81871,C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(=O)CSCc1ncc[nH]1 81872,NS(=O)(=O)CCC(=O)NCC12CC(CO1)N(C(=O)CN1CCSCC1)C2 81873,C1(C(=O)NCC(CC)C(C)C)CN(C(=O)CC2CC2COC(C)=O)CC1(C)C 81874,N1(C(CC(C)SC)=O)CC(CN(C(=O)CSc2nncn2C)C)C(O)C1 81875,c1(C(=O)NC2CCC(NC(C(C)OC)=O)CC2)cccc(Br)c1OC 81876,n1(CCCNC(COCCC)=O)cc(CCNC(C2COCC2C(N)=O)=O)nn1 81877,CCC(C)CCC(=O)NC(CCN(C(=O)CC1(O)CCCC1)C)C(C)C 81878,N1(C(CC(C=C)C)=O)CC2(C(=O)NC(C)CC=CC)CC1CCO2 81879,C(=O)(C1=C(c2ccccc2)CCCC1)NC(C)(C#N)CCc1ccccc1 81880,N1(C(CCc2ncc(C)[nH]2)=O)CCCC(NC(=O)CC=CC(C)(C)C)C1C 81881,CC(C)(CCCF)C(=O)NCCC1CCCN(C(=O)CC2(N(C)C)CCCC2)C1 81882,N1(CCC(=O)NC)CCC2C(C1)NC(=O)CN2S(=O)(=O)CCS(=O)(=O)CC1CC1 81883,c1(N2CC(C)CC(C(=O)Nc3ccc(OCOC)cc3)C2)nc2cccnc2s1 81884,C(C(C(=O)NC1(CO)CCC1)C(C)(C)C)NC(CCC(C)(C)OC)=O 81885,c1(OC)cc(C2(C(=O)O)CC2)ccc1C.c1(C(C)(C)C)ccc(Cl)c(F)c1 81886,C1(N=[N+]=[N-])(C(N2CC(C)OCCC2)=O)CCN(C(=O)CC2COCCO2)C1 81887,C(=O)(C1CCCc2nncn21)NC1C=CCN(c2cc(CC=O)nc(Cl)n2)C1 81888,C12(SCc3n(-c4ccn(CC)n4)nc(-c4cncs4)n3)CC3CC(CC(C3)C1)C2 81889,N1(C(c2c(C)nc(C)[nH]2)=O)CC(N(C)C(C2CCCSC2)=O)C(C)(C)C1 81890,CCC1=C(C(=O)N2CCC(n3cc(-c4cc(F)ccc4OC)nn3)C2)CCCO1 81891,N1(C(C(CCCC)F)=O)CCC2(C1)CN(C(c1ccc(CCC(N)=O)cc1)=O)C2 81892,c12ccnc(c1)NC(=O)C(c1cc(C)c(C)s1)N(CC)C2.C(CCC1CC1)SC 81893,C=CCC(C)C(=O)NC(C(=O)NCc1ccc(OC)cn1)C1CCCO1 81894,C(=O)(C(C)N1CC(C)C1)NCC=CCNC(C1C(COC)C1)=O 81895,CC1(C)CN(C2CCN(C3CCCCC3)C2=O)CCC1NC(=O)CC(F)(F)F 81896,C1(CN(C)C(c2cc(C(F)F)n(C)n2)=O)CCN(C(=O)COCC2CCOC2)CC1 81897,CCC(CNC(C1CC=CCC1)=O)(CC)NC(c1nc(Cl)cs1)=O 81898,CC#CCC(C(=O)NC1CC2CCC2C1)NC(c1ccc(C2CC2)o1)=O 81899,C1(C(C(=O)N(CC(C)(C2CC2)OC)C)C)CCN(C(=O)Cc2nc[nH]n2)CC1 81900,C1(C(=O)NC(CNC(C=CC(C)(C)C)=O)(C)Cn2cccn2)CCCS1(=O)=O 81901,CCC(CSc1ccccc1)N=c1[nH]c2c(c(=NC3CN4CCC4C3)[nH]1)CSC2 81902,N1(C(C(C)N(CCC)C(c2cc(Cl)no2)=O)=O)CCCCCC1C 81903,N1(C(C(C)OC)=O)CCN(C(=O)C=CC(=O)OC(C)(C)C)C(n2cccn2)C1 81904,C(=O)(CC(C)(C)C1CC1)NCC(CC)NC(C1CCN(C(C)C)CC1)=O 81905,C1(CCNC(c2nn(C)c(C(N)=O)c2)=O)CN(C(=O)C(C)(C)CO)CCS1(=O)=O 81906,c1(C(COCC(CC)n2cncn2)SC)nnnn1CCCSC 81907,Cc1cccc(C(=O)NCC2(F)CCC(NC(=O)C(c3ccccc3Cl)C)C2)n1 81908,C12(NC(C(c3ncccn3)C)=O)CCCN(C(c3cncc(F)c3)=O)CC1C2 81909,N1(C(CSC)=O)CCN(C(=O)C(F)OC(F)(F)F)C(c2ccncc2)C1 81910,C1(CNC(c2c(C)cncc2)=O)CN(C(=O)CN2CCOCC2=O)CCCO1 81911,N1(C(=O)CCF)CCC(NC(c2cccc(NC3CCCC3)c2)=O)C12CC2 81912,N#CC1(NC(=O)Cc2cn[nH]c2)CC12CCCC2.N12CCC=C(CC1=O)C2 81913,N1(C(=O)C2=CCCSC2)CCC2CCN(C(c3occc3C3CC3)=O)C2C1 81914,n12ncc3ccc(cc13)-c1c(CC)cc-2cc1.N1(C(=O)OC)CCOCC1CC 81915,C1(C(=O)NCCCc2ccncc2)C2CC1N(Cc1cscc1Br)C2 81916,Cc1cc(Br)c(N)cc1C(=O)NC(C)(CNC(=O)CCCC(C)C)CO 81917,c1(NC(CC(C)(C)NC(C(C)=CC(C)(C)C)=O)=O)cnc(F)cc1C 81918,CCCC(C(=O)NC1CCN(C(c2ccc(OC)c(C)c2)=O)C1C)S(N)(=O)=O 81919,CC(CC(=O)N(C)Cc1ncnn1C)C(C)(C)NC(=O)C(O)Cn1cncn1 81920,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CNC(=O)COCC2CCCOC2)C1(C)C 81921,C(C(C)(C)CNC(=O)CCNC(c1ccc(Cl)o1)=O)SC 81922,C1(NC(C2C(CNC(c3cc(COC)no3)=O)CC2)=O)CN(C)CCN(C)C1 81923,N1(C(CCCCC=C)=O)CCOC2(CCN(C(c3cnc(OC)cc3C)=O)C2)C1 81924,C12(NC(C=NOC)=O)CCC(CC1)N(C(c1coc(CC3CCC3)n1)=O)C2 81925,C1(CCNC(=O)Cc2ccccc2)CCC(C(=O)NCC(=O)NC2CCC2)C1 81926,c1(NC(CC)CNC(c2cc(O)n(C)n2)=O)nc2c(cc1C#N)COCC2 81927,C(N=c1[nH]c(O)nc(=N)[nH]1)C1CCN(C(C(N2CCCC2=O)C)=O)C1 81928,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCO3)CC2)cc1C#N 81929,c1(NC(=O)NC(CC)C(c2ccccc2)OC)cc(CNC)cc(F)c1 81930,c1(CN(C(=O)NC2CC(C(=O)OC(C)(C)C)C2)C2CC2)cnc2[nH]c(=N)sc2c1 81931,C#Cc1nc(C(=O)N(CC(C)(C)CNC(C2(C(F)F)CC2)=O)C)cs1 81932,C1(CNC(CNS(NC)(=O)=O)=O)CCCCN1C(=O)C=Cc1cnc[nH]1 81933,C1(C(N2CC(CCCCNC(c3cc(C(C)C)[nH]n3)=O)C2)=O)COCC(C)O1 81934,C1(CC(C)NC(C2CCS2(=O)=O)=O)CCN(C(=O)CCc2cccs2)CC1 81935,Cc1ccc(F)cc1C(=O)NC(CO)C(=O)N1CCC(CCCO)C1 81936,C1(C(=O)NCC2CCOC2=O)CN2CCN1CC2.C12C=CC(C1)NC2=O 81937,Nc1ccc(C(F)(F)F)cc1NC(N1CCC1CNC(c1ccc(Cl)nn1)=O)=O 81938,C(=O)(CC(C1CC1)NC(=O)CCn1cc(C)cn1)OC.C12(CC1)C(=O)N2 81939,c1(C(N(CCCN(C)Cc2c(C)scc2)C)=O)cccc(-c2nc(O)n[nH]2)c1 81940,Cc1cc(C(=O)NCCC2(O)CCN(C(=O)Cc3[nH]cnc3C)CC2)ccc1Cl 81941,N(C1CCCc2cc(C(=O)Nc3cnc[nH]3)ccc21)C(c1ccc(C)c(I)c1)=O 81942,CC1(C)CN(C(=O)C(C)(C)CC2CC2)CCN(C(=O)CC(O)c2ccccc2)C1 81943,c1(NC(CNC(Cc2c(C)nc(N(C)C)s2)=O)(C)C)ncccc1[N+](=O)[O-] 81944,c1(C(N2CCC(C(C)(C)NC(COCCCC)=O)C2)=O)cc(C#N)c(N)cc1O 81945,S(=O)(=O)(c1ccccc1[N+](=O)[O-])CC1CN(CC(CC)O)C1 81946,N1(C(COC(CC)(C)C)=O)CC2CCN(C(=O)CC3(OC)CCOCC3)C(C2)C1 81947,C(=O)(CC(C)C1CC1)NC(C1CCCCC1)CNC(CC1CC(=C)C1)=O 81948,c1(SC(C(=O)N(C(C)CCNC(C2CCCO2)=O)C)(C)C)nc2ccccc2[nH]1 81949,c1(C(=O)NC2CCCCN(C(C(CCC)OC)=O)C2)coc(=O)c2ccccc12 81950,C(=O)(CCCCCN(C)C(C1CC1(F)Cl)=O)N1CC(=C)C1 81951,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 81952,c1(C(=O)NC(C)CCNC(c2ccccn2)=O)occ2c1CCC2 81953,CC(C(C)(C)C(=O)NC1C=CCCC1)NC(=O)C=CC(F)(F)F 81954,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)CC1CC 81955,N1(C(CCC(C)OC)=O)CCC2CCC(C1)N2CC(C)C(C)C 81956,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(c2cnn[nH]2)=O)CCO1)C 81957,c1(CNc2ccc3ncn(C)c3c2)cccc2c1OCCN(C(=O)OC(C)(C)C)C2 81958,N1(C(CCc2n(C)ncc2)=O)CCCC1(C(=O)NC12CC(C1)C2)C(N)=O 81959,c1(C(=O)NCC(=O)NCCCNC(c2csc(C3CCCO3)n2)=O)ccccc1 81960,CCCCCCCCC(C)C(=O)N1CC=C(CC(=O)N(C)CC2CCCS2)CC1 81961,C(CC(F)F)(C(=O)N1CC=CCO1)N(C(c1ccc(SC)o1)=O)C 81962,C(=O)(N1OC2CCC1CC2)c1c(C)oc(CNC(c2cccc(O)c2F)=O)n1 81963,c1(NC2(CO)CCN(C(c3cncn(C)c3=O)=O)CC2)nc(O)c2c[nH]nc2n1 81964,N1(C(CC2(OCC)CCC2)=O)CCOC(C(=O)NC2CCCC2(F)F)CC1 81965,C1(N(C(C2C=CCS2)=O)CC)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 81966,CC1(C)CC(C)(C(N2CCN(CCO)CC2)=O)CN1C(c1cscc1Cl)=O 81967,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C(C)C(C)C)=O)C(C)C1 81968,C(C)(CC(C)C(F)F)NC(C(C)=CC(=O)NC1CCC2(CCC2)C1)=O 81969,c1(NC(C23C(CN(C(C(C(C)C)OC)=O)C2)C3)=O)c(F)c(F)nc(F)c1F 81970,Cc1ccc2[nH]c(C(N3CCN(C(=O)CSCC(=O)N(C)C)CC3)=O)cc2c1C 81971,CCCC(CC(=O)NCCC(C)n1cccn1)NC(=O)CCc1nc[nH]n1 81972,N1(C(C(C2CC2)NC(C(=O)N(CCCO)CCC)=O)=O)CCC(C)CC1C 81973,N1(C(c2ccc(CC)o2)=O)C(CNC(=O)COCc2ccnn2C)CC2CC12 81974,C1(NC(C2CN(C(C)=O)C2)=O)COC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 81975,N1(C(CCC(=O)NC)=O)CCN(CC2CCC(CCCC)CC2)CC(O)C1 81976,Cc1ccc(N2CCC(NC(C3(F)CCCCC3)=O)C(O)C2)c([N+](=O)[O-])c1 81977,Cc1ccc(C=CC(=O)NCCC2C(C)CCCN2C(=O)C(C)N(C)C)c(C)c1 81978,C(C(=O)NCCC1(O)CN(C(C2CCCC2SC)=O)C1)(C(C)(C)C)OC 81979,c1(OC)nccc(CNC(c2ccnn2C2CC2(F)F)=O)n1 81980,C1(C(N2C(CC(=O)N(C)C)CC2)=O)CCCN1C(=O)Cc1cncs1 81981,NC(C(=O)NNC(=O)c1ncoc1Br)c1c(F)cccc1Cl 81982,c1(SC)ccccc1-n1cc(C2CN(C(=O)C(c3ccc(F)nc3)C)C2)nn1 81983,c1(C(=O)NC2CC(NC(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 81984,O=C1NCC2(CO1)CN(C(=O)CC1COCCN1C(=O)C(=O)NCC1CC1)C2 81985,N1(C(=O)C(O)C2CC2)CCC(C2CN(C(c3coc(-c4cccnc4)n3)=O)C2)C1 81986,C1(NC(CCC#C)=O)CN(C(=O)CSc2nncs2)CC1C 81987,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(O)C3)=O)C2)C)cn1 81988,n1(CCCC)ncc(C(=O)NCC(CC(C)C)NC(c2cnnc(O)c2)=O)c1C 81989,C(CO)(CCC(C)C)NC(CC1(C)N(C(C(C)SC)=O)CC1)=O 81990,C1CN=C2C=CN=C(N2)O1.C1(CN(C)CCN(C)C)CCC(C)(C)CO1 81991,C(c1cn(C)cn1)=CC(=O)NC1CCN(C(c2nc(CC)oc2)=O)C1 81992,C1(C(=O)NC2C(NC(CC(=O)OC)=O)CC2)CCCN(CC(F)(F)F)C1 81993,CC1(c2cn(C3CCC(C(=O)NCCC4(O)CCCC4)C3)nn2)CCOC1 81994,Cc1cc(CNCc2ccc(-c3ccc(F)cc3)o2)sc1Br 81995,C1(=CC(=O)NC2CCC2NC(=O)CC2CC=CC2)CCCC1 81996,C1(CNC(C=C(C)Cl)=O)CC2CN(C(=O)CS(=O)(=O)NC3CC3)CCN2C1=O 81997,c1(C(=O)OC(C)Cc2ccc(Br)s2)ccc(C2CCCC2)c(F)c1 81998,c1(NC(N(C2CCOC(c3cncn3C)C2)C)=O)ccn2c1CCC2 81999,N1(CC)CC(C(=O)N(CCCNC(=O)CC(C)F)C)CC1=O 82000,N1(C(C(c2c(C)cccc2Br)NC(C(COCC)C)=O)=O)CCCCCC1CC 82001,C1(CNC(C(C)=CC)=O)C2CN(C(=O)C)CC12.c1(-c2nocc2)cc(C)nn1C 82002,C12(CNC(Cn3ncc(C)c3)=O)CN(C(=O)Cn3ncn(C)c3=O)CC1CCO2 82003,c1(C(N2CC3(CC(NC(=O)Cc4c[nH]nc4O)C3)C2)=O)cnn2c1OCC(O)C2 82004,Cc1cccn2cc(C(N3CCC4CN(C(=O)C(O)C5CCC5)CC34)=O)cc12 82005,O=C1CC2(CCN(C(=O)CC3CC(NC(C4CC5(C4)CC(O)C5)=O)C3)C2)CN1 82006,C1(CNC(C2(OC)CCCC2)=O)CCC(CNC(C2CC(F)C2)=O)CC1 82007,N1(C(C2OCCN(CC)C2)=O)CC2(C(=O)NCc3nc(C)nn3C)CC1CO2 82008,C1(NC(Cc2cccc(OCC)c2)=O)CCN(C(C2(C)CCCS2)=O)CC12CC2 82009,C1(C(=O)NCC2(C)CC=CCC2)COC2(C1)CN(C(C1CC=CC(O)C1)=O)C2 82010,C(C(C)(O)CNC(C1(N2CCOC2=O)CC1)=O)NC(C1(N(C)C)CC1)=O 82011,CC1COCCC1N=c1[nH]c2c(c(=NCCCNC(C3CCCC3)=O)[nH]1)COC2 82012,C(=O)(C(C)(C)CNC(N)=O)NCC1CCC(NC(C(C)NC(=O)C(C)(C)C)=O)C1 82013,C12(C(N3C(C)CN(C(C4(C#N)CCC4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 82014,C1(C(=O)Nc2csc(O)n2)CN(CC2CN(C3CC4CCC3C4)C2)CCS1(=O)=O 82015,c1(SC)cc(C(=O)NCC2(NC(=O)Cc3cnn(C(F)F)c3)CCCC2)c(C)o1 82016,c1(C(N(CC(CC)NC(c2cnn(C3CCCC3)c2)=O)CC)=O)cnnn1C 82017,C=CCC(C)(C(=O)NC1CCN(C(=O)Cn2nc(C)nc2C)C(C)C1)N(C)C 82018,Cc1[nH]c(=NCC2CCn3c(O)nnc3C2)nc2c1NC(=O)CN2C 82019,C1(CNC(CC2CCC(C)CC2)=O)CN(c2cc(C(C)(C)C)ncn2)CCN1C 82020,c1(CNC(C(c2ccccc2F)C)=O)cnn2c1CN(C(=O)CCS(C)=O)CC2 82021,C1(C(=O)OCCN2CCOC2=O)CN(Cc2cccc(SC(F)(F)F)c2)CC1O 82022,c1(C(=O)NC2C(NC(c3c(C)nncc3)=O)COC2)cc2ccccc2[nH]1 82023,N1(CC(=O)NC(CN(C)C(C2CCC(CO)CC2)=O)(C)C)CCCC(N(C)C)C1 82024,C(C1CN(C(=O)CCc2ccn(C)n2)CC1C(N1CC(c2ccon2)C1)=O)=CC 82025,C1(C(=O)OC(CNC(C)(C)C)=O)CC2C(CC1c1ccccc1)C2(F)F 82026,CCCC(O)CC(=O)NCC1CCCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 82027,C1(C(=O)NC(C)C(CO)NC(=O)Cn2ncc(C#N)c2N)COCCN1C=O 82028,c1(SCC2CC(CC)C2)cc(C(=O)OC)ncc1[N+](=O)[O-] 82029,N1(C(C2N(CC#C)CCC2)=O)CC(NC(c2cc(N)cnc2C)=O)C(C)(C)C1 82030,c1(C(=O)NC(CCCNC(CC(CC)CC)=O)(C)C)ccn2nccc2c1 82031,C1(CNC(=O)C(O)c2ccsc2)CCCN1CC(F)F 82032,N1(C(CCOCC(=O)OC)=O)CC(C2CCCN(C(C3(C)CCC(=O)NC3)=O)C2)C1 82033,C12CN(C(C3C(CCC)C3)=O)CC1CCSS2.c1(C(=O)OC)cncc(SC)n1.C 82034,C1(NC(CC(=O)N(C)C)=O)CCCCC1NC(=O)Cc1ccc(O)cn1 82035,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2CCN(C)C(=O)C2)=O)CC1)C 82036,C1(=CCNC(C2CC(=C)C2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 82037,C(=O)(C1=CCCCO1)Nc1c(C2CCN(Cc3c(C)nsc3C)C2)ocn1 82038,C1(NC(c2c(C)nco2)=O)CN(C(c2c(Br)cnn2C2CCC2)=O)CC1C 82039,C1(NC(=O)Cn2ccnc2)CCC(C(=O)NCc2cccc(C(=O)O)c2)OC1 82040,c1(C(N2C(C)CCN(C(=O)C3=CCOC3)CC2)=O)cc(S(C)(=O)=O)ccc1F 82041,C1(CNC(C2CC(O)C2c2ccc(F)cc2)=O)CCC(C(F)(F)F)CC1 82042,C(=O)(CCCCCCOCC)N1CC(CSCC)(CNC(=O)C(F)C(CC)CC)C1 82043,c1(C(N(C2CCN(C(=O)C=C(C)C(C)C)CC2)C(C)C2CC2)=O)cc([N+](=O)[O-])c(C)s1 82044,N1(C(CCN(CC=C)C(C2CCC2OC)=O)=O)CCCC(C2CC2)CC1 82045,C1(NC(c2cn(C(C)(C)C)nc2)=O)CCC(O)CN(C(C2CCCN2C=O)=O)C1 82046,Cc1cc(Br)c(N)cc1C(N1CCC2C(NC(C3CC34CCOCC4)=O)C12)=O 82047,c1(C(C(=O)NCCN2CCC3CC23)Sc2ccccc2)ccc(F)cn1 82048,C1(C(=O)NCC(c2cccs2)C)(NC(=O)CCN2CCCC2=O)CC(F)C1 82049,C(C(C)(C)C(=O)NC(C)CCNC(=O)CN1C(=O)CNC1=O)SC 82050,C1(SC)CN(C(=O)CCN2CCCCC2=O)CC1NC(=O)C(c1cncn1C)O 82051,c1(C(N(C)C)=O)cccc(C(N2CCC(C3CC(N)CCN3)CC2)=O)n1 82052,c1(C(N(C)CC2CN(C(C(OC)OCC)=O)C2)=O)ccn(C)c(=O)c1O 82053,Cn1c(C(=O)NCC2CCCC2NC(C2CCCCC2C(F)(F)F)=O)cccc1=O 82054,C1(C(=O)NCC(c2ccsc2)NC(CCN(C)CC)=O)CCCN1C1CC1 82055,c1(CC(=O)NC2CN(C(c3c(C)nc(C4CC4)o3)=O)C(C)C2)nc([N+](=O)[O-])n[nH]1 82056,C(c1cncs1)=CC(=O)N(CC(=O)NCCCOCC)CC1CC1 82057,CC1CN(C(=O)CC2CCC2)CC1NC(C1CC1c1cccs1)=O 82058,N1(C(c2n(C)nc3c2CCC3)=O)CCOC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 82059,C(=O)(C#CC1CCCCO1)N1CCC(NC(CN(C)S(N)(=O)=O)=O)C12CC2 82060,c1(CC(N2CC(F)CC(NC(=O)C3=CCC3)C2)=O)cncc2ccccc12 82061,Cc1cc(CC(=O)N(CCCCN(C(=O)CCOC2CCC2)C)C)ccc1F 82062,C1(NC(C(=O)NC(C)CC2CCCCO2)=O)CCCN(CC(=O)N(C)C)C1 82063,C1(C)(NC(=O)OCC(C=C)OC)CCCC1COC(C)(C)C 82064,CC1CN(C(C2CC(C)(C)C2)=O)CC1NC(C1CCCC12CC2)=O 82065,n1(CC(=O)NC2C(NC(c3n(C)c(=O)ccc3)=O)C2)cc(P(C)(C)=O)cn1 82066,C(C(C)(C)C(=O)NCCC1CCNC1=O)NC(CCNC(=O)OCC)=O 82067,C(=O)(CP(=O)(C(C)C)C(C)C)N1C2CC(NC(C(F)=CC)=O)CC1CC2 82068,c1(C(=O)NCC2N(C(C(=Cc3cccnc3)C)=O)CC2)ccn2nccc2n1 82069,C12(CNC(C(CC)(F)F)=O)CC(C1)C(NC(=O)Cc1ccccc1CC#N)CO2 82070,n1(C(C)C)ncc2c(N3CCC(NC(c4csc(S)n4)=O)C3C)nc(Cl)nc12 82071,c1(CCCC)cc(C(=O)N(C2CN(C(c3cc(C(C)C)oc3C)=O)C2)C)c(C)o1 82072,N1(C(C(c2ccccc2)NC(CCCCC=CC)=O)=O)CCOC(C)(C)CC1 82073,N1(C(C(c2ccc(Cl)cc2)C(C)C)=O)CC(NC(C23CC4CC2C3C4)=O)CC(C)C1 82074,CC(CC(N)=O)N=c1[nH]c(N2CCN(C)C(=O)C2)nc(=NC(C)C)[nH]1 82075,N1(C(CC2(C)CC2(F)Cl)=O)CCOC2(CCN(C(c3cccn(O)c3=O)=O)CC2)C1 82076,N1(Cc2c(C)ccnc2)CCC(NC(C2(C)CC2(F)F)=O)CC(C)(C)C1 82077,N1(C(c2n(C)ccc2)=O)CCCC(O)(CNC(=O)CC2CCC(=O)N2)C1 82078,C1(CNC(C(c2ccccc2)OC)=O)CCC12CN(C(=O)C1=COCC1)C2 82079,N1(C(C=C(C)C(C)C)=O)CCC2CN(C(c3cnco3)=O)CCC12 82080,N1(C(c2cn(C)nc2)=O)CCN(C(C2CC23CCCCCC3)=O)C2(CC2)C1 82081,n1(CC)ncc(Br)c1C(N1CC(OCCNC(=O)C(C)(C)C)C1)=O 82082,N1(C(CNC(N)=O)=O)CCOC2(CCN(C(C3CCC(F)C3)=O)CC2)C1 82083,c1(CC(C)C)cccc(C(C)NC(=O)NCCCCCCO)c1 82084,Cc1ccc(C(N2CCC2CNC(c2cccc(CC(F)(F)F)c2)=O)=O)cc1 82085,c1(C(=O)NCCCN(C(c2snc(C)c2N)=O)CC)cc(C(F)(F)F)c(Cl)cn1 82086,c1(C(=O)NC2CC(F)(CNC(C3CC(OC)(OC)C3)=O)C2)nc[nH]c2nccc1-2 82087,C1(O)(C(=O)NC(COC)(C)C)CCN(C(c2ccc(OC(C)C)nc2)=O)CC1 82088,N1(C(C2(OC)CC(C(F)F)C2)=O)CCCOC(CNC(=O)CN(C2CCC2)C)C1 82089,C1C(C)C(=O)N1.C(C=C(Cl)Cl)=CC(=O)N=CCC 82090,N1(C(c2cc(CCC)on2)=O)CC2C=CC1C(C(=O)N(C(C)(C)CC)C)C2 82091,C(CCCCC(=O)NC(C)(CO)C(=O)NCCC1C=CCC1)OC 82092,C(=O)(C(C)(C)C)N(C1CN(C(=O)C(C)OCCOC)C1)CC 82093,C(=O)(C(Cc1ccco1)C(=O)NC1CC(CNC(=O)Cc2nnc(C)s2)C1)OC 82094,N1(C(C2(CO)CC(C)(C)C2)=O)CCC(C)(C)C(CNC(C2C(COC)CC2)=O)C1 82095,CC(Cc1ccccc1)C(=O)NCCNC(=O)CCC1CCOC1 82096,c1(NCCC(C(C)C)OCC)ncccc1S(=O)(=O)NC(CCSC)C(C)C 82097,C1(N(C(C(C)C(C)(C)C)=O)C)CCC2CN(C(=O)CC3CCSC3)CC12 82098,c1(OC)cn(CC(=O)NC2CC2NC(=O)CCCC(N)=O)c(C)cc1=O 82099,C1(OC)CC(CNC(=O)Cc2cnc(C)s2)N(C(=O)CCc2ccc[nH]2)C1 82100,C(=O)(C1=CCC(F)(F)CC1)N1CC(C)C(N(C)C(c2cnc(Cl)cc2N)=O)CC1 82101,N1(C(C(Cc2c(C)cccc2)C)=O)CC2CCN(C(C3CCC3)=O)C2C1 82102,N1(C(C2C(=C)C2)=O)CCCCC1c1cn(-c2ccccc2C(=O)N)nn1.C1(C)CC1 82103,N1(C(C(C(CC)C)O)=O)CC2(CCC(CNC(=O)CCc3ccnc(C)c3)O2)C1 82104,N(S(=O)(=O)N1CCCC1C)(CCO)CC1S(=O)(=O)CCC1 82105,c1(C(N2C3CN(Cc4cnc(O)nc4O)CC23)=O)ncc(Cl)cc1Cl 82106,c1(NC(=O)OC)nccc2cc(OCC(=O)Nc3ccc(C(C)C)cc3)ccc12 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82302,CC1CN(c2cc(C(=O)NC(CCN)C(F)F)ccn2)CCO1 82303,c1(C(=O)NCC(CNC(CCOCC#C)=O)(C)O)cc(C)n(C(F)F)n1 82304,C12(NC(C3C(=C)CC3)=O)CCC(C1)N(C(c1ccnc(-c3ccco3)c1)=O)C2 82305,N1(C(C2CCC(CC)O2)=O)CCC2(CC1)CN(C(=O)CC1CC(O)C13CCC3)C2 82306,Cc1nc(CN(C(=O)CCCN(C(=O)C=CC(F)(F)F)C)C)n[nH]1 82307,N1(C(C=CC)=O)CCN(CC2CCCN(C(C)C(F)(F)F)C2)CC1 82308,C12CCN(CC1O)C(=O)CC1(CCC1)N2CCOC.C(C(=O)OC)N(CCC)C 82309,c1(CC)ccoc1C(=O)NCCCC(c1ccccc1)NC(c1cnc(C)s1)=O 82310,CCCC(CNC(c1n[nH]c2c1COC2)=O)C(=O)N(C1CCC(O)CC1)C 82311,C1(CCC)CN(C(=O)C(C)(C)CC#N)CCN1C(=O)Cc1ccc(C)s1 82312,C1(C#N)(C(=O)NC2CCCN(C(CN(CCC#C)C)=O)C2)CCOCC1 82313,C(=O)(CCCCCCCCCO)N(C1CN(C(C2CC3CC2CC3(F)F)=O)C1)C 82314,N1(C(C(C)SC)=O)CCCCC1CCCNC(=O)CC1C=CCC1 82315,C#Cc1ccc(C(=O)NC2CC23CC(NC(=O)C(O)CC2CCCCC2)C3)nc1 82316,S(=O)(=O)(c1cccnc1)NCC(=O)NCC1N(C(C=NOC)=O)CCCC1C 82317,CN1CC(NC(=O)C=CCNC(C2CCOC2)=O)CC1=O 82318,C1(NC(CCCSC)=O)CC2CCC1N2C(c1cccc(C(N)=O)c1N)=O 82319,N1(C(CN(C)CC)=O)C2CCC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 82320,CC1=NNC(=O)C1CC(=O)NCC(O)CN(C(=O)C(=C1CCCCC1)F)C 82321,C12(C(CNC(C3CCCC3C)=O)NC(C(C)=C(C)C)=O)CCC(CC1)C2 82322,C1(=CC(=O)NC2CCCC(NC(=O)Cc3ccoc3)C2)CN2CCC1CC2 82323,C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 82324,C1(NC(c2ccc(OCC)cc2)=O)CCC12CCN(C(c1scnc1Cl)=O)CC2 82325,C=CC(C)(CC)C(=O)N1CCN(c2ccnc(CCSC(F)(F)F)n2)C(C)C1 82326,c1(CNC(=O)CC(O)C2CC2)ccc(-c2cn(-c3ncc(Br)s3)nn2)cc1 82327,C(N=c1ccnc(S(C)(=O)=O)[nH]1)C1OCCN(C(C(CCC)(C)C)=O)C1 82328,c1(CC(=O)N(C)CCc2cn(CCCOC(=N)O)nn2)cccc(C(C)(C)C)c1 82329,C(=O)(CC(C)C(C)(C)NC(=O)Cc1nc[nH]n1)N(C)CC1CC(OC)C1 82330,C1(NCc2c(OC(c3nccc(C(F)F)n3)=O)cccc2)CCN(CC)CC1C 82331,C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(c1cc3n(n1)CCC3)=O)C2 82332,C=C1CC2(C1)C(=O)NC2.N1(CCC(=O)NC(c2ccsc2)C)CCCC1 82333,C1(C(=O)NC(CCC)CCC)CCCCN(C(=O)CCN(C)CCOC)C1 82334,c1(NC(CC(=O)OC)=O)c(OC(C)(C)C)cccc1O.C1CCC(=O)N1CCN 82335,C1(C)(C(N2CC(CCCCC)C2)=O)CCN(C(=O)C(C)(CC)OC)C1 82336,O(N=C1CCCCCC1)CC(=O)NCC(N(C(C(C)OCC)=O)C)C1CC1 82337,N1(C(C(C(C)C)NC(=O)OCC)=O)CCN(C(=O)CC2CCCO2)CC1C 82338,N1(C(c2ccc(NC)c(F)c2)=O)CCN(C(=O)Cc2c(C)noc2C)C(C)C1C 82339,C(=O)(CCCS(C)(=O)=O)NC1CC(NC(c2ccc(C)nc2C2CC2)=O)CC1O 82340,CC(C)S(=O)(=O)CC(=O)NC1(CNC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C 82341,N1(C(C2(COC)CCOCC2)=O)CCCC(CNC(c2cc(OC)cs2)=O)CC1 82342,Cc1oc(C(=O)N(CCCN(C)C(c2csnc2Cl)=O)C)cc1CO 82343,C1(C(=O)OC)C(C(=O)NCCCN(C)CCn2ccnc2C)C12CC2 82344,N1(c2c(C=O)scc2)CCC(F)(CNC(C2C(OC)(OC)CC2)=O)C1.N(C)(C)C 82345,c1(C(=O)NC2C(NC(c3ccc(C(O)CF)cc3)=O)C2)ncc(F)cc1F 82346,Cc1nccc(C(N2CCCCC2CCC(=O)NC2(CO)CCC2)=O)n1 82347,C(C)(C(=O)NC1CC(OC)C1)(C(C)C)OC.C12(CCCOC1)C(=O)N2 82348,C1(C(N2CC(C)C(N(C)C(C34CC(C#N)(C3)C4)=O)CC2)=O)CN2CCN1C(C)C2 82349,C1(C(=O)NCCSCC)CC2CCC1N2C(=O)CC1CCCO1 82350,c1(C(=O)NCCC(C)NC(C(COC(C)(C)C)N(C)C)=O)cc(Br)ccc1O 82351,C(c1cn(C)cn1)=CC(=O)NC(CCOC)CNC(C1CCCN1C1CC1)=O 82352,C(c1ccc([N+](=O)[O-])cc1)=CC(N1CC2(CCN(C(=O)C=C3CCC3)CC2)C1)=O 82353,C1(CNC(c2cc(CCCC)oc2C)=O)CCC(C)(C)CN1C(c1cnc[nH]1)=O 82354,N1(C(CNS(N(C)C)(=O)=O)=O)CCN(C(=O)C(C)(O)C2CC2)CC(CO)C1 82355,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCc1cc2c(s1)CCC2)NCC 82356,c1(C(C)(C)C(N2CCC(C)(CNC(=O)Cn3cnnc3)C2)=O)ccnc(C#N)c1 82357,C(CCC(C)CO)NC(C1(NC(CC)=O)CCSC1)=O 82358,C=C1CC(C(N)=O)N(Cc2ncc(-c3ccccc3)[nH]2)C1.n12cc(cn1)NC2 82359,Cc1nnc2n1CC(C(=O)NC13CC1CN(C(C1(C)CC=CC1)=O)C3)N(C)C2 82360,Cc1nc(-c2cccs2)oc1C(N1CCCC1C(C)NC(C1C=CCC1)=O)=O 82361,C(CN=C(NCC1CCCCN1CCC1(OC)CCOCC1)N(C)C)SC 82362,C1(C(N(CC(c2nn[nH]n2)C)C2CC2)=O)CCCN1C(=O)CCc1ccoc1 82363,n1(CC)nccc1C=CC(=O)NC1C2CC1N(C(c1nn(C)nc1C)=O)C2 82364,c1(CCN(C(C2CC(F)(F)C2)CO)C)ccc(N)c(Cl)c1 82365,c1(C(=O)NC(C(=O)NCCn2c(CC)ncc2)CN(C)C)cc(Cl)cn1C 82366,C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)Cc1ccc(Cl)cn1)CC 82367,N1(C(c2ccc(OCC)cc2)=O)CCN(C(=O)C=C2CCC2)C(COC)C1 82368,Cc1nc(-c2cccs2)sc1C(N1CCCC1CN(C(=O)C(=O)NC(C)C)C)=O 82369,CC(C)C(O)C(=O)NC1CC(n2cc(C3(C)CCOC3)nn2)C1 82370,c1(C(CCC(N2CC3C(C(N4CCC(C)CC4)=O)(C3)C2)=O)=O)cc(F)ccc1F 82371,c1(C(N2C(CN(C(C3(CC(C)C)CC3)=O)C)COCC2)=O)nccc2cc[nH]c12 82372,c1(C(N(C)CC2C(C)OCC2)=O)c(CNC(C2SCCS2)=O)nnn1C 82373,C1(CSc2ccc(NC(c3ccc(Cl)cc3)=O)cc2)CN(C2=CCCC2)CCO1 82374,C1(C(=O)NCC(C2CCCCC2)NC(=O)C2=CCCC2)CCC(F)(F)CC1 82375,c1(CC)ccc(CNC(=O)CC(C)NC(C2CCOC2C(C)C)=O)cc1 82376,CC1(C(=O)NCCC(O)C(=O)NCc2cn(C3CC3)nn2)CCCC1O 82377,CC1CC=C(C(=O)NC2COCC2NC(=O)C(=O)NCCC(N)=O)CC1 82378,c1(CC)ccc(F)cc1C(=O)NC(C(C)NC(c1cnc(C)cn1)=O)C(C)(C)C 82379,C1(NC(CCC(=O)NCC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)CC2 82380,Nc1cc([N+](=O)[O-])ccc1NC(C1CCN(Cc2cscc2Br)CC1O)=O 82381,c1(C(=O)NC(CCCNC(c2c(CC)nc[nH]2)=O)C)ccnc(OC2CCC2)c1 82382,c1(NC(C2C(=C)COC2)=O)nc2c(F)cccc2n1C 82383,C1(CC)CN(C(c2ccnc(F)c2F)=O)CCN1C(C)=O.c12ccccc1S2 82384,c1(N2CC(C)C(NC(C3(F)CCOC3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] 82385,N1(c2n(CCCOC)c(CC(C)(C)C)nn2)CC2CC(OC)C(C2)C1 82386,N1(C(C2N(CC)CCOC2)=O)C2CCC(C2)C1C(N1CC(C(N)=O)C2(CC2)C1)=O 82387,N1(C(C2(COCC)CC2)=O)CCCC(CCNC(C2CCCC(O)C2)=O)CC1 82388,c1(CC(=O)NCC(C2CCOC2)NC(CC2(OC)CCCC2)=O)ccncc1F 82389,CC1CN(C(=O)Cc2ccon2)CC2(CCN(C(C3CC(C)(F)C3)=O)C2)O1 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82425,Cc1coc(C)c1C(C1CCCC1N(C)C)NC(=O)C(=O)NCC(Cl)(Cl)Cl 82426,Cc1cc(=NC(=O)N(C(C)(C)C)C(c2ccnc(F)c2)COC)cc[nH]1 82427,Nc1cccc(C(=O)NCCC2CN(C(=O)CC3CCCC(=O)N3)CCO2)c1O 82428,CCC(CC(C)C)C(=O)NCC1CCCCN(C(=O)CS(=O)CC)C1 82429,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82430,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82431,c1(C(=O)NCCN(C(c2ncoc2C(C)C)=O)CC)cnc(CC(C)C)cn1 82432,CCCC(O)CC(=O)N1CCOCC1CNC(c1sc(C)nc1CC(C)C)=O 82433,C1(C(=O)NC(C(=O)NC2CN(CCC)C(=O)C2)C2(O)CCC2)CN(C)CCN1C 82434,CC1CN(C(=O)COCC(C)(C)C)C(C)CN1C(c1cc(Cl)ncc1N)=O 82435,Cc1cccc(C(=O)NCc2csc(CNC(=O)C(N3CCCCCC3)C)n2)n1 82436,Cc1nc(-c2nnc[nH]2)ncc1C(N1CC(O)(CCNC(=O)CCF)C1)=O 82437,c1(C(N2CCCC(CNC(=O)CCc3cn[nH]c3)C2)=O)ccc2[nH]nc(Cl)c2c1 82438,C(=O)(C(F)C(=O)NCCN(C(=O)CCCNC(C)=O)C1CCCCC1)OC 82439,CCC(C(=O)NC1CC(O)(CNC(=O)C(C)CC2CC2)C1)OC 82440,C(C)(C(=O)NOCc1cccc(C)n1)(N(C(C(COC)N)=O)C)C1CC1 82441,CCS(=O)(=O)C=CC(=O)NC1CCCC(N(CCO)CC2CC2C)C1 82442,C12(C(N3CC(CCNC(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CCC(CC1)CC2 82443,c1(C(N(C(C)CNC(=O)C(C)NS(C)(=O)=O)CC)=O)ccc(C)n1C 82444,C1(CN(C(c2[nH]cc(C(=O)OC)c2)=O)C)CCCCN1C(C1CC1C)=O 82445,C1(NC(C2C(C(C)(C)C)C2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1cnccn1 82446,C1(C(=O)NC(CNC(c2onc(C)n2)=O)CC(C)C)CSc2ccccc2O1 82447,C1(C(=O)NCC(C2CCN(C(=O)CCSCC(N)=O)CC2)(C)O)CC12CCCC2 82448,Cn1cnc2nc(=NCC3C(F)(F)C34CCC4)[nH]c(NCc3cncs3)c12 82449,C(C)CCC(c1nnnn1C(C)C)NCCOC(C)(C)C.C1CO1 82450,CC(C)CC(C(=O)N(C1CCCN(C(c2cn3ccnc3s2)=O)C1)C)C(C)C 82451,c1(CNC(C2N(C(C)=O)CC2)=O)cccc(Oc2ccccc2C(N)=O)c1O 82452,C(=O)N=c1[nH]onc1C1CC1.c12cn(nn1)C(COC)C(=O)N(CC)CC2 82453,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 82454,C1(C(=O)NC2C(C(=O)OC)COC2)CC(NS(C)(=O)=O)CN1c1ccc(Cl)cc1 82455,C1(N(C(C(C)N=[N+]=[N-])=O)C)CCCN(C(=O)C(c2cncnc2)C)CC1 82456,C12(C(N3CC(C#C)OCC3)=O)COCCC1CN(C(C)=O)C2 82457,Cn1cc(C(=O)NC2CCCCC2NC(c2nc(C3CC3)cs2)=O)nc1O 82458,C12CN(C)CCN1C(=O)NC2.CC(CN1CCCC1)CC(F)F 82459,C1(OC)CC(NC(C2(c3ccno3)CCC2)=O)CN(C(=O)C=C(C)C)C1 82460,c1(OC)cc(OCC(C2(C)CC2)OC(=O)C2CC2)ccc1OC 82461,C(CSC)(C(=O)NC(Cn1cccn1)C(=O)N1CCC(COC2CCCC2)C1)OC 82462,Cc1cc(C(N2CC3CCC3(CCNC(c3cnc(N)cn3)=O)C2)=O)cc(C)c1 82463,C1(NC(CCC(=O)OCC)=O)CN(C(=O)C(c2cnn(C)c2)O)CC1C1CC1 82464,CC(CC(=O)c1ccc(F)cc1)C(=O)OC(C)(C)C(=O)N(C1CCCCC1)C 82465,c1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2F)c[nH]c2cnccc12 82466,c1(NC(C2CCN(C(c3cc4sccc4[nH]3)=O)CC2)=O)nc2ccccc2s1 82467,C1(OC)CC(C(=O)NC2CN(C(=O)CCc3cnccn3)CC23CC3)C12CCC2 82468,c1(OC)cc(C(=O)NCC(O)CCNC(=O)CCNC(c2ccoc2)=O)cc(F)c1 82469,c1(NC(CC(C)C2CCNCC2)=O)c(Br)c(C(C)C)nn1C(C)(C)C 82470,C12(C(N3CCCCC3C(N3CC(=C(F)COC)C3)=O)=O)CCCC1CC(=O)C2.CCS 82471,C12(C)CC(CCO1)NC2=O.c1(CC)ccc(-c2nn[nH]n2)cc1F 82472,n1(CC)ncc(Cl)c1C(N1CCCCC1Cc1cn(C(C)CC2CCC2)nn1)=O 82473,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(O)C4)=O)C2)cc1C#N 82474,C1(C(N2CCC(C(C)NC(Cc3c(C)nc[nH]3)=O)CC2)=O)OCCOC12CCC2 82475,c1(NC(C2CCC(N(C)C)CC2)=O)ncc(Br)c(OCC2CCOC2)n1 82476,c1(C(=O)NCC2(C)CCC(NC(c3cc[n+]([O-])cc3)=O)C2)cnc2n1CCC2 82477,c1(CNC(c2ccnnc2)=O)nc(C)c(C(=O)NC(COCC)C(C)C)s1 82478,CC1C(=O)N(C)CCN1C(=O)C(C)(C1CC1)N(C)C(c1ccc(C)s1)=O 82479,Cc1cc(N2CC(NC(=O)C3=C(Cl)CCC3)CC(C)(C)C2)cc(C#N)c1[N+](=O)[O-] 82480,CCCC(C(=O)NCc1ccccc1)N1CCCC1CC 82481,c12cn(nn1)CCC2.c1(SCCOCC(=O)NC(C2COC(=O)C2)C)ccccc1 82482,c1(OCCCC(N)C(=O)O)ccc2cccnc2c1 82483,C1(NC(C=CCOC)=O)C=CCCC1C(N1CC(c2nc(O)n[nH]2)C1)=O 82484,N1(C(C(CC)OC)=O)CCN(C(c2nc[nH]c2C(C)(C)C)=O)CC(C)(C)C1 82485,c1(C(N(CCC(=O)NC(C2CCCC2)C)CCO)=O)cccnn1 82486,CC#CC1CCN(C(C2CC2CNC(c2cc(C(N)=O)nn2C)=O)=O)CC1 82487,Cc1cc(O)ncc1NC(C1(C)CC(O)CN1C(=O)C(C)C(F)(F)F)=O 82488,c1(N2CCC(NC(=O)CCC(F)F)CC2)ncnc(Cl)c1Br 82489,C1(CC(=O)NCCC(=O)NO)CCCCC1NC(C1CC1C(F)(F)F)=O 82490,N1(C(c2c(COC)cco2)=O)CCCCC1CCN(C)C(c1c(C)nsc1N)=O 82491,C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2c(C)noc2N)=O)CC1 82492,CN1C2CCCC1CN(C(=O)C1=NOC(CNC(=O)C3=CCCCCC3)C1)C2 82493,Nc1cc(C(=O)NCC2CCC(NC(=O)C=CCO)C2)cc(N)c1 82494,C1(F)(C(N(CCOCCC(=O)NC(c2nc(C)[nH]n2)C)C)=O)CCCCCC1 82495,C(=O)(CC(C)(C)COC)NCC1N(C(c2cc(C(C)=O)oc2)=O)CC(OC)C1 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82741,N1(C(c2ccc(CSCC#C)cc2)=O)CCCC(NC(=O)C=C(Cl)Cl)CC1 82742,C1(C(C)C)CN(C(=O)CC2(n3cncn3)CC2)CCN1C(C1CCCCO1)=O 82743,C(N1CCN(CCC(C)C)C(C)(C)C1=O)n1cc(CC(C)C)nn1 82744,Cc1nc(N2CC(C(C)NC(=O)C(C)(C)C3CCCCC3)C2)ncc1Br 82745,C(=O)(CCCC1CC1)N(C(C)C(=O)N)CCOC(=O)C(C)(C)C.C(CCO)CC 82746,N(C(=NCCSC)N1Cc2ccc(OC)cc2C2(CC2)C1)CC(CCC)CC(C)C 82747,C(CNC(c1csc(F)c1)=O)(C(=O)NC1(C2CC2)CC1)N(C)C 82748,c1(CC(=O)NC2(CC)CN(C(=O)Cn3ccnn3)C2)cccc2c1OC(C)(C)C2 82749,Cc1cc(CC(=O)NCC2CCCCN2C(=O)Cc2cccnc2O)ccc1Cl 82750,CP(C)(=O)c1ccc(C(N2CCCC2CNC(=O)CSC(F)(F)F)=O)nc1 82751,N1(C(c2cc(C)ns2)=O)CC2CCC(NC(=O)C(C)S(C)(=O)=O)(C2)C1 82752,N1(C(CCC(=O)NC)=O)CCCC2(NC(=O)Cc3nncn3C)CC2C1 82753,c1(SCC(O)CCO)ccc2nc(Cl)ccc2c1 82754,c1(C(N2C(CNC(C3CCC4(CCC4)CC3)=O)CC2)=O)cccc2ccsc12 82755,c1(C(=O)NCc2cn(CCNC(c3ccn(C)n3)=O)nn2)[nH]cnc1C#N 82756,C1(C(=O)NCC(CNC(c2cccc(F)c2)=O)O)CC2(C1)CC2(F)F 82757,c1(SC)nc2ncnc(N3CCCC3C3(NC(=O)Cn4nnc(=N)[nH]4)CC3)c2s1 82758,c1(C(N(C(C)C)CCNC(C2CCC3(CCC3)O2)=O)=O)ccnc2c1CCC2 82759,c1(CSC2CCN(c3cccc(N)c3)C2)cc(Cl)nnc1O.CC(C)(C)OC(=O)N 82760,C=C=C(C)CC(=O)NCC1C(CC(N2CCC(c3ccsc3)C2)=O)C1 82761,C1(C)(CNC(c2nc(COC)oc2)=O)CCC(NC(=O)Cc2cnc(C)s2)CC1 82762,CC(C)(CNC(=O)CCCn1ccnc1)CC(=O)NC(C1CCOC1)CO 82763,c1(CN2C3CCN(C(C(=O)N(C)C)=O)CC2CC3)csc2ccccc2c1=O 82764,c1(C(=O)NC(CC)CNC(=O)C(C)(C)c2ncco2)cc(Br)ccc1O 82765,C=CC1(O)CCN(C(=O)CC)C1.c1(CC(=O)N2CCCC2)nncn1CC 82766,c1(C(=O)NC(C(N2CC(SC)C2)=O)C2CCCO2)ccc(C)c(C#N)c1 82767,N1(C(c2cc(F)cc(Br)c2)=O)CCC2C1CCN2C(c1cc(Cl)cnc1Cl)=O 82768,Cn1cc(C(N2CC=CC2(C)C(N2CCCCC2CC(N)=O)=O)=O)ncc1=O 82769,c1(NC(C)=O)ccc(F)c(F)c1.c12ncccc1C(=O)CNC(=O)C(C)O2 82770,c1(C)ccc(NC(c2n(CCSC)nnn2)c2cscn2)c(Cl)c1 82771,c1(C(C(=O)OC)NC(c2ccc(Br)cc2)CCCOC)ccc(S(C)(=O)=O)cc1 82772,c1(C(=O)NCC2(C(N)=O)CN(C(CC3C(C)CCCC3)=O)C2)cc2cccnc2[nH]1 82773,C1(CC)CC2CCC(C1)N2C(C1CN(C(C2COCCN2C)=O)CCO1)=O 82774,c1(C(N2CCCC(C(C)NC(c3c(COC)ccs3)=O)C2)=O)ccc(C)c(O)n1 82775,C1(NC(=O)CC2CC2CNC(C2COCC2O)=O)CCCC(O)CC1 82776,Cc1ccc(CN(C(=O)CCOCCCNC(=O)Cc2conc2C)C)cn1 82777,c1(C(=O)OC)ccc(NC(=O)N(C)C(=O)NCC2CC3(C2)CC3F)cc1 82778,C=CCC(CNC(C1CC12CC(NC(=O)CCCNC(N)=O)C2)=O)CC(C)C 82779,c1(C(=O)Nc2cncc(C#C)c2)cc(F)c(F)cc1F 82780,c1(C(=O)NC2C3(CC(NC(CC(C)n4cccn4)=O)C3)C2)ncc(F)cc1F 82781,C1(CCNC(=O)CN=[N+]=[N-])(OC)CN(C(=O)CCSC)C1 82782,c1(C(N2CC(C3(NC(=O)Cc4cccs4)CC3)C2)=O)cc2c(=O)[nH]ccn2c1 82783,C1(NC(c2cnc(OCC)s2)=O)CC(NC(C2CC3CC3C2)=O)C(O)C1 82784,C(CCN=C(NCCC1(C(F)(F)F)CCC1)NC1Cc2ccccc21)OCC 82785,C1(C(=O)NC(CNC(=O)C(C2CC2)C2CC2)C2CCC2)CC12CCCC2 82786,Cc1ccc(C(C)C(N2CCCC(CNC(c3cc(F)c[nH]3)=O)C2)=O)cc1 82787,c1(C2N(C(C(C)OC3CCCC3)=O)CC2)cn(Cc2ccccc2)nn1 82788,c1(CC)cc(NC2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)ncn1 82789,N1(C(C2(CC=C)CCN(C(=O)CC(F)(F)C(F)F)C2)=O)CCC2(CCCO2)C1 82790,N1(C(c2oc(C)c(Br)c2)=O)CCC2(COC(CNC(C3CCOC3)=O)C2)C1 82791,c1(C(N(CCN(C(CC(=O)OC)=O)C)C)=O)cccc2c3c([nH]c12)CCCC3 82792,c1(COC)ccc2c(c1)CN(C(=O)C=Cc1c(OC)cccc1Cl)C2 82793,c1(NC(C)C(=O)NC(=O)NC2CCCN(C)C2)cccc2c1CCCCC2 82794,C12(CCNC(=O)CCc3cnco3)CCC1CN(C(c1cc(O)cc(=O)o1)=O)C2 82795,C#Cc1ccc(C(=O)NCCC(C)N(C)C(c2cc3scnc3[nH]2)=O)c(C)c1 82796,c12cc[nH]c1C(=O)NC2.C1(C(C)(C)OC)CCN(C(=O)CC2CC2F)C1 82797,C1(CCN)COCCN1C(=O)Nc1ccc(N2CCCC2)cn1 82798,C(C)(C(F)(F)C(F)(F)F)=CC(N1C2(CN(C(C3CCC(=C)CC3)=O)C2)CC1)=O 82799,C12CCCC(CC1)NC(=O)c1ccc(o1)CSCC(=O)N2.C(C)(=O)OC 82800,C1(C(N2CC(O)(CN(C(c3occ(C)c3)=O)C)C2)=O)CCCCCC1 82801,c1(CNC(c2n(CC=C)nnn2)(CCC)C2CC2)nc2c(n1C)CCCC2 82802,c1(C(=O)OC)cnc(N2CC3CC2CN3C(c2ccc(F)c(O)c2)=O)nc1C 82803,C1(N(C)C)(C(=O)NCCN(C(=O)CCCN(S(C)(=O)=O)C)C2CC2)CC(CO)C1 82804,C(=O)(CCCC(F)(F)CO)NC(CNC(c1n(CC)ccn1)=O)(CC)CC 82805,Cn1cc(C(CO)NC(=O)NCCC2CCCN2Cc2ccccn2)cn1 82806,c1(C(=O)NCC2N(C(C3N(C(C)=O)CCC3)=O)CC2)ncc(C#N)cc1Cl 82807,c1(CCC)c(C(N2CC(C)(NC(=O)CCCCN(C)C)C2)=O)cnn1C 82808,C(CCC(C)C(=O)NCC(C)(C)CCNC(c1sccc1OC)=O)OC 82809,N1(C(CC(C)(C)O)=O)CCC2(CCCC2NC(c2ccc3c(c2)OCCO3)=O)C1 82810,C#CCCCCCCC(=O)NC1CCC1CNC(c1ccc(F)cc1C(F)F)=O 82811,C1(C(N2CCC(O)(CCNC(C3(C)COC3)=O)C2)=O)CCCC12CCOCC2 82812,C1(C(N2CC3CC(NC(C(CC=C)N(C)C)=O)C3C2)=O)CCS(=O)(=O)C12CCC2 82813,C(Cn1cncn1)(C(=O)NC1(C(O)CO)CC1)NC(C=C(C)C(C)C)=O 82814,C1(CCNC(c2c(C)scn2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)(C)O 82815,Cc1oc(C(=O)NC2CCN(c3ccnc(C(C)(C)C)n3)C2C)cc1Br 82816,C1(C(=O)NC(C2CCCCC2)C#C)CCCCC1CNC(=O)CC1OCCC1C 82817,C(=O)(C(C)C(=O)NCC1(CC(=O)NC(c2cncs2)C)CC1)OC 82818,N1(C(C2(CC#C)CCN(C(=O)C(C)CSC)C2)=O)CC2(CNC(=O)N2)C1 82819,C1(c2ccccn2)(C(=O)NCC(C)(C)Cn2cc(COC(=N)O)nn2)CCCCC1 82820,c1(OC)cc(C(N2CCC(O)C2C(=O)NCCCc2cnn[nH]2)=O)n(C)n1 82821,c1(C(=O)NCC2=CCN(C(c3ccc(CCF)cc3)=O)CC2)cc(Cl)ncc1F 82822,c1(CC)ccccc1CC(=O)N(CCCCCCNC(=O)CC1CCCC(=O)N1)C 82823,C(CCC(C)(C)C(c1nnnn1Cc1ccc(F)cc1)NCCC1(C)CC1)OC 82824,c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC(O)C2)cncc2sccc12 82825,c1(NC(c2ccc(CC)s2)=O)cc(C)n(C(C)CC)n1 82826,c1(NCCC(=O)Nc2c(C(=O)NC(COCC)C)cccc2)cccc(F)c1C 82827,CC(C)CC(C(=O)NC1CCC(N(CC(F)(F)F)C)CC1)NC(=O)C(C)N(C)C 82828,C1(CNC(CC(CCC)(C)O)=O)CC2(CCOCC2)CN1C(c1occc1Cl)=O 82829,N1(C(C2(CNc3ncc(C(=O)OC)nc3)CC2)=O)CCC(O)C(F)(F)C1 82830,N1(C(C(CC=CC)NC(c2ccsc2)=O)=O)CC2CC(C)C2C1 82831,C12(n3c4ncc(s4)c3=O)CCC(C1)N(C(=O)C(C)C1CC1)C2.c1(OC)nccs1 82832,N1(C(c2cc(C)sc2)=O)CCC(N(C)C(C2CCC(=O)NC2)=O)C2(CC2)C1 82833,c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)c2cccs2)ccc(C2CC2)nc1 82834,N1(C(C=Cc2n(C)ncc2)=O)CCC(NC(c2ccoc2)=O)C(F)(F)CC1 82835,C1(C(C)(C)C(=O)Nc2cc(C(F)(F)F)ccn2)CCN(Cc2cccnc2)CC1 82836,Cn1c(C(=O)NC2CC(NC(=O)CCCCCF)C(O)C2)cc2sccc12 82837,CN=c1[nH]c(=NCC2CCOC2C)[nH]c(=NCCS(=O)(=O)NC)[nH]1 82838,c1(CC)nn(C)cc1C(=O)NC(C(=O)Nc1cccc(OCC)c1)C1(C)CC1 82839,c1(C(=O)NCC(C)N(C(C(C)c2ccon2)=O)C)c(F)cccc1Br 82840,C1(C(N2C(C3(C(=O)NC(c4ccc(O)cc4)C)CC3)CCC2)=O)CC1C1CCC1 82841,C1(O)(CNC(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc(C3CC3)nc2)=O)C1 82842,C1(NC(C(CC)O)=O)CC(F)(F)CC1NC(c1ccc(Cl)cc1)=O 82843,c1(NC2C(NC(CCNS(C)(=O)=O)=O)CC2)cccc([N+](=O)[O-])c1F 82844,C1(CC(=O)NC2CCN(C(CCCCC#C)=O)CC2O)CCCC2(CCC2)O1 82845,C(=O)(CC(C(C)(C)C)NC(C1CCCS1)=O)N(C)Cc1nc(C)on1 82846,S(=O)(=O)(c1ccc(Br)cn1)N1C(C(=O)Nc2ccccc2S)CC(F)(F)C1 82847,C1(C(=O)NCC(CC)(O)CC)CCCCCN1C(C1CC1COC)=O 82848,CCCC(CCCNC(=O)C(O)CF)NC(=O)CNC1(CO)CC1 82849,C#CCCCC(C)C(=O)NC1CC12CCN(C(c1ccccc1C(C)=O)=O)CC2 82850,CC1(C)CC(C)(NC(=O)CNC(=O)C2=COCC2)C1 82851,Cc1ccc2c(C(=O)NC3C4CCC(C4)N3C(c3ccccc3)=O)n[nH]c2c1 82852,C1(C(=O)NCc2cnsn2)CCCCC1Cn1cc(-c2ncccn2)nn1 82853,C1(C2CCN(C(C3CCCC3C)=O)C2)(NC(C2CC(C)=C(C)CC2)=O)CC1 82854,C1(CNC(CCCOCCC)=O)C2CCC(C2)N1C(c1ccccc1COC)=O 82855,C=CCC(CC)C(=O)N1CCC(C)C(CNC(=O)C(C)(C)C(F)F)C1 82856,C1(NC(COC(CC)C)=O)COC2C(Nc3nc(SC)nc(=N)[nH]3)COC12 82857,CCC(CN(C)C)CC(=O)NCc1cn(C2CCN(C(=O)CSCC)CC2)nn1 82858,c1(C(=O)NC23CN(C(c4cn(CCC)nn4)=O)C(CC2)C3)ccc2occc2n1 82859,N1(C(CC(C=C)(C)O)=O)CCN(C(=O)C(C2CCOCC2)O)C2(CCC2)C1 82860,CC(C(=O)N1CCC(N(C(=O)Cc2cc[nH]c(=N)c2)C)C1)C(F)(F)C(F)F 82861,c1(C(=O)NCC2(NC(c3nsnc3O)=O)CCC2)ncc2ccccc2c1O 82862,c1(C(N2C(C(C)(C)NC(CCC=C(C)C)=O)CCC2)=O)cc(C(F)F)cs1 82863,CCCCC(CNC(c1[nH]nnc1CC)=O)NC(C1(C(=O)NCC)CCC1)=O 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82969,c1(C(N2CCC(NC(C3C(C(=O)NCC#C)C3)=O)CC2)=O)ccsc1S(N)(=O)=O 82970,C(=O)(C(C)(F)C(=O)NC1CCCC1C(=O)NCc1nnc2n1CCC2)OC 82971,CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)N1CCN(CCF)CC1)N(C)C 82972,c1(C(N2CC3C(C2)C3(C)C)=O)cc2ccc(-c3cncs3)cn2n1 82973,N1(C(COCC=C)=O)CCC(C2CCN(C(c3cc(CSCC)on3)=O)CC2)C1 82974,c1(C(C)NC(c2c(CC)occc2=O)c2n(CC=C)nnn2)ccc(Cl)c(C)c1 82975,c1(CN2CC(CNC(C(C(C)C)c3ccncc3)=O)C2)ccc(F)cc1F 82976,C(=O)(C(F)C(C)(C)O)N(C(CC)C(=O)NCC(C)C)CC 82977,C1(COCC)CCCN1C(C1CCC(n2cc(C(O)C(C)(C)C)nn2)C1)=O 82978,c1(C(N2CC(C#N)C2)=O)cnc2c(c1)CCN(Cc1cnc(-c3cccs3)s1)C2 82979,CC1CC(CNC(c2cncn2C)=O)CN1C(c1cc(C2CCCC2)nn1C)=O 82980,c1(C(=O)NC2CC(C(N(CC#C)CC3CCCCO3)=O)CC2O)ncc(F)cc1F 82981,CC12CN(C1)C(=O)CSn1cc(nc1)CNC(=O)C2.c1(C2CC2)ccccc1 82982,Cc1cc(Br)cc(C)c1CN1CCN(C(=O)NCC(C)C)C(CC(C)C)C1 82983,N1(C(c2nc(CCNC(=O)C(C3CC3)C3CC3)oc2)=O)CCCC(C2CC2)CC1 82984,N1(C(C(CNC(c2c(CC)ncnc2)=O)O)=O)CCN2CCCCC1C2 82985,c1(C(=O)NCCNC(C2(CC(N)=O)CCOC2)=O)ccccc1SCC(F)(F)F 82986,C1(C(N(C(CCC)C)C2CC2)=O)CN(C(c2cnn(CCF)c2)=O)CC12CCC2 82987,c1(OC)ccc(CC(=O)NC(C)C(C(C)C)NC(C)C)cc1[N+](=O)[O-] 82988,C1(C(N2C(C)C(NC(=O)Cn3cccc3)CCC2)=O)CC(C)(C)SC(C)(C)C1 82989,C#CCCCC(C)C(=O)NCCC1CC(CNC(=O)CC=CCOC(C)(C)C)C1 82990,N1(C(C(C(=O)OC)OC)=O)CCOC2(C1)CN(C(=O)COC1CCCCCC1)C2 82991,C#CC1CCC(CN2CC(C)CC(C(=O)NCc3c(C)cccc3F)C2)CC1 82992,C1(OC2(COC(F)F)C(=O)OCC2)CCC12CCCCC2 82993,N1(CCNC(=O)C=C(C2CC2)C2CC2)CCN(C(=O)CC2COCC2O)CC1 82994,CC1(CNC(=O)CC2CCCN(C(C3(F)C(C)(C)C3(C)C)=O)C2)NC(=O)NC1=O 82995,c1(C(=O)NCC(=O)NCC(=O)NC(c2nncs2)C)cccnc1S 82996,N1(C(CCCNC(C)=O)=O)CCC(CO)(CNC(=O)CN2CCNC(=O)C2)C1 82997,c1(C(N2CC(NC(CCCN=[N+]=[N-])=O)C3(C2)CC3)=O)cc2scc(Cl)c2[nH]1 82998,C#Cc1cncc(C(=O)OCC(c2ccn(C)n2)=O)c1 82999,C1(CN(C(C(C)SCC)=O)C)CCN(C(=O)C(O)CC2CCOCC2)CC1 83000,C#CCC(CC(F)F)C(=O)NC1CCC(CNC(=O)C2=C(Cl)CCC(C)C2)CC1 83001,c1(CC)cc(C(=O)NCC2CC(CNC(=O)CCC(=O)N(C)C)C2)nn1CCO 83002,Cc1c(CCC(N2CC(O)(C(C)(C)CNC(=O)C(CCO)N(C)C)C2)=O)cnn1C 83003,c1(C(N(CCC(C)NC(C(CCC#C)O)=O)C)=O)cncc2n[nH]cc12 83004,C1(NC(C2(c3cccc(Cl)c3)CC2)=O)C2CCC(C2)N1C(c1ccc(Cl)s1)=O 83005,c12cnn-1c2.O=C(CCC1CC1)N1CCC1C1CC1 83006,c1(N(C)C(=O)C2CC2)cc(Br)ccc1S(=O)(=O)NC(c1ccc(Cl)nc1)CC1CC1 83007,CCC(CC(=O)N(C)CCOCCNC(c1ccc(COC)s1)=O)OC 83008,C1(C(=O)NCC2(O)CN(C(c3ncn(C)n3)=O)C2)CN(CP(C)(C)=O)C1 83009,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)C2)=O)ccc2sccc2c1 83010,c1(C(=O)NCC(CC)(C)NC(C2(C)CCCCO2)=O)cc(C2CC2)nn1CC 83011,CC1CCCCN1C(=O)CCOC1CN(C(N)=O)C1.C12(CCCCC1)N(C)C2 83012,Cn1cccc(CN2CCC(O)CC2C(=O)NC2CC23CC(O)C3)c1=O 83013,C(C(CC1CC1)C(=O)NCC1CC2CCC2C1)NC(c1ccc(CC)o1)=O 83014,c1(C(=O)NC2C(C(=O)Nc3c(=N)cc[nH]c3)C2)cccn2nccc12 83015,CC1CCN(Cc2ccc(Cl)cc2Cl)CC1NC(c1cnn(C(F)(F)F)c1)=O 83016,CCCC(CNC(C1CCCCCN1C)=O)C(=O)N(C1CCCCC1(C)C)C 83017,N=c1[nH]cc2c(c1CN=c1cc(NCCCN3CCNCC3)nc[nH]1)CCC2 83018,N1(C(CCCC(C)O)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)n1C)=O)C2 83019,C1(C(=O)Nc2cn(CCC=C)nc2)C2CCC(C2)N1C(=O)CC1(C(=C)F)CC1 83020,C12(CC)CCCCC(C(N3CCCC(NC(c4coc5c4COC5)=O)C3)=O)(C1)C2 83021,CCCCCC(C)(C)C(=O)NCC(O)CNC(c1nnn(CC)c1C)=O 83022,c1(C(=O)NCC2C3CN(C(c4cc(C)c(C)nn4)=O)CC32)cccc2nsnc12 83023,N1(S(c2cc(SCC)[nH]c2)(=O)=O)CCCC2(CCCN2C(=O)C(C)(O)CCC)C1 83024,c1(NC(C2N(C(c3c(C)nsc3)=O)CC(O)C2)=O)ccc2c(c1)C(=O)N(C)C2 83025,C=CCCCC=CCC(=O)NCCC1(NC(=O)CC2OCCC2C)CCCC1 83026,C12(C(=O)NC3C(C)CN(C(C4(C)CC4(F)Cl)=O)CC3)CC3CC(C1)CC(C)(C3)C2 83027,C(=O)(C(C(C)(C)O)NC(=O)C(C)c1cccs1)N(C)Cc1c(COC)noc1 83028,N1(C(C(CC=CC)C)=O)CCc2cc(CNC(c3cccs3)=O)ccc2C1 83029,c1(C(=O)NC(CCC)CO)cc(NC(c2ccc(C(C)(C)C)cc2)=O)cn1C 83030,c1(C(=O)NCCC2CC(NC(C3N(CC)CCOC3)=O)C2)cccc2cc[nH]c12 83031,N1(C(C(C)OC)=O)CCOCC(CNC(c2ccc(-c3cnn(C)c3)o2)=O)C1 83032,C(=O)(CCCCC(C)(C)C)NC1CC1.c12ccc(nc1C)C(=O)N(CC)C(C)C(=O)N2 83033,CN1C(=O)C(NC(c2cccc(C#N)c2Cl)=O)c2cc(Br)ccc21 83034,N1(CC(=O)NC(C2(O)CCN(C(C3CC(=C)C3)=O)C2)C)OC(C)(C)CC1=O 83035,C(=O)(CC(C)C(=O)N(C)CCN(C(=O)C=Cc1ccc(OC)cc1)C(C)C)OC 83036,N1(C(C(C)C(F)F)=O)CCN(C(C2(C#N)CCSCC2)=O)CC1CF 83037,N1(C(C2C3CN(C(C4N(C)CC(O)CC4)=O)CC32)=O)CCC12CCOCC2 83038,N1(C(CCCn2cc(-c3cnc(C)nc3)nn2)=O)CCC12CC(C(=O)N(C)C)C2 83039,C=C1CC(C(=O)Nc2ccccc2C)N(Cc2ccnc(COC(C)(C)C)c2)C1 83040,CC(C)S(=O)(=O)C(C)C(=O)NCC(C1CC1)N(C(=O)Cn1nc(O)ccc1=O)C 83041,c1(C(=O)NC(C2CCCCC2)C(=O)NC(CC)C2CC2)oc(C)nc1C 83042,C#CC1CN(C(C2(NC(=O)C=Cc3cocn3)CCSC2)=O)CCO1 83043,C1(NC(c2cccc3cccnc23)C)CCc2c(Br)cccc2C1 83044,C1(C(N2CCC(NC(=O)CC3CC4(CC4)C3)C2)=O)CC2(CCC2)C1 83045,c1(N2C(C)CC(CNC(c3c(C)cncc3F)=O)C2)ccc2c(n1)CCC2=O 83046,C1(C(=O)NCCN2CCCCC2)N(C(C(CCC)N(C)C)=O)CCCC1(C)C 83047,N1(C(Cc2n(C)ncc2Cl)=O)CC2CCC2(NC(C2(F)CCOC2)=O)C1 83048,C1(C(=O)NCc2ccc(C)n2C)CCCN1S(=N)(=O)N(C)C 83049,N1(C(C2(CC)CC2(F)F)=O)CCC(C(C)NC(=O)CCCOC(C)C)CC1 83050,CC(C)C(F)C(=O)NCC1(CN(C)C(c2csc(Br)n2)=O)CC1 83051,C(c1ccc(S(=O)(=O)N(C)C)cc1)=CC(N1CCN(C(C(CC#C)C)=O)CC1)=O 83052,CC1C(=O)NC(=O)CN1C(=O)C(CN=[N+]=[N-])NC(c1ccc(C(N)=O)o1)=O 83053,N1(C(c2c(CNC(C(CC#C)O)=O)cc[nH]2)=O)CCCC12CCNC2=O 83054,c1(C(=O)NCC2CC(NC(CC(COC)(C)O)=O)C2)ccc(P(C)(C)=O)s1 83055,Cc1nnc(O)c(C(=O)NCC2CC3CN(C(=O)Cn4cnnn4)CC23)c1C 83056,C(=O)(C1=CCCOCC1)N1CCC(NC(c2ccsc2-n2cnnn2)=O)(CF)C1 83057,C(=O)(C(CO)C(F)(F)F)NC1CN(C(c2cccc(C(C)(C)C)c2)=O)CC1SC 83058,CC1OCCC1(O)CNC(c1ccc(CNC(C23CSCC2C3)=O)nc1)=O 83059,c1(OC)ccc(CC(=O)NC2CCC2NC(c2sc(N)nc2C)=O)cc1F 83060,C1(CC)CCCN(C(=O)CC2(NC(C3CC3C)=O)CCCCC2)C1 83061,C=CCC(CNC(=O)C(C)(C)COC)C(=O)Nc1cncc(C(C)C)c1 83062,CCCC(CCC)C(=O)NCCNC(c1c[nH]nc1-c1ccccc1Br)=O 83063,Cc1cnc(NC(=O)CCNC(=O)CCCOC2CCOCC2)s1 83064,N1(C(CCOCC(C)C)=O)CC(NC(C2C3CCCCCC23)=O)CC(F)C1 83065,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83066,C1(C(N(C2CCCN(Cc3ccc(C)nn3)C2)CCC)=O)CC12CCSCC2 83067,C(=O)(CCC(C(C)C)NC(C1CCCSC1C)=O)NC(CCCCCC)C 83068,c1(CNC2(C(N3CCC(C(=O)O)C3)=O)CCC2)cc(Cl)c(F)c(Cl)c1 83069,Nc1c(C(=O)NC2C3CN(C(C4CC5CC5C4)=O)CC23)ccc(F)c1Cl 83070,C1(CCNC(=O)C(=O)NCC2CCCC(C(=O)OC)N2)CCc2ccccc2N1 83071,c1(C(=O)NCC(=O)NCc2cncn2C2CC2)cc2ccccn2n1 83072,N1(C(c2cnnc(C)c2C)=O)CC(C(N2CCCC(OC(C)=O)C2)=O)CC(C)C1 83073,Cc1ccccc1OCC(=O)NC1CC(C(=O)NCC(C)CC2CCC2)C1 83074,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83075,N1(C(CN(CCCCC)C)=O)CCCC(C2(NC(=O)CCc3cnn[nH]3)CC2)C1 83076,O=C(CCCCc1cccs1)NCCOC(C1(c2ccc(F)cc2)CCCCC1)=O 83077,N1(CC)CCCC(N=c2[nH]c(=NCCc3cccc(C)n3)[nH]c3cccnc23)C1 83078,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83079,C1(CCNC(C2(CC)COC2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC1C 83080,C=C(Cl)CCC(=O)NCCN(C(=O)CCC1CCCC1O)C 83081,CC#CCCCC(=O)N1CCCC(CCNC(=O)CS(=O)(=O)NCC)CC1 83082,N1(C(c2c(C)oc(CO)c2)=O)CC2(CNC(=O)C(CO)NC(N)=O)CC(F)(C1)C2 83083,CCC(C)C(C(=O)NC1CCN(C(=O)C(F)F)C1C(C)(C)C)OC 83084,c1(C(C)C(=O)N(C)C)nnc(N2CC(CC(=O)NC3CC3)C2)s1.C1CC1 83085,c1(C(C)NC(C2CCN(C(=O)C(C)c3ccsc3)C2)=O)nn(C)cc1O 83086,C1(NC(CCC)=O)CN(C(c2cc(C(N)=O)ccc2F)=O)CCC1C(F)(F)F 83087,C1(C(F)(F)F)(NC(CC(C)(C)C)=O)CCCN(C(=O)C(F)C2CCOC2)C1 83088,c1(C(=O)NC2CC(NC(c3c(CCC)n[nH]c3)=O)C2)cc(CS(C)(=O)=O)c(C)s1 83089,C1(CC(=O)Nc2ccc(Cl)cc2)CN2CCC1CC2.C12CN(C3CC13)C(=O)NC2 83090,C12(C(=O)OC)CCC(CNc3ccc(OC4CCOC4=O)cc3)(CC1)S(=O)(=O)C2 83091,C1(NC(C(C)CO)=O)CCCC(NC(c2ccccc2C(=O)NC2CC2)=O)C1 83092,c1(C(N(C2(CC(=O)NCc3ccon3)CC2)C)=O)cnnn1C 83093,c1(CC2(CC(=O)Nc3ccco3)CCC2)ccc(F)nc1 83094,C1(CC=C)(NC(=O)Cc2ccnn2C2CCCC2)CN(C(=O)C(C)OC)C1 83095,CCCCCC(C)CC(=O)NC(CCN(C(=O)CCS(C)(=O)=O)C)C(C)C 83096,C1(CNC(CCC(N)=O)=O)(NC(C2CC(=O)N(C(C)C)C2)=O)CC2CCC1CC2 83097,c1(-c2cc(OC)no2)nc(-c2ccnc(Cl)c2)nn1CCC(C)C 83098,N1(C(=O)CCN2CCOCC2)CCCCCC1CNC(C1C2C3CCC(C3)C12)=O 83099,C1(C(=O)NC(C2CCN(c3nnco3)CC2)=O)CC12CN(Cc1ccccn1)C2 83100,C1(C(=O)NC(C(C)C)c2nc[nH]n2)(CC)CCCN1C(c1ccncn1)=O 83101,c1(OC)cc(CNC(c2oc(CNC(c3c(C)ncn3C)=O)nc2C)=O)ncn1 83102,CC1CC(C(=O)N(CCCCN(C(=O)COc2cccnc2)C)C)C(=O)O1 83103,C#CC(CNC(=O)CC(CCCC)NC(C1CCC1C#N)=O)CC(C)(C)C 83104,c1(C2(C(=O)NC(C)CNC(C3CCCSC3)=O)CCC2)ccc(F)cc1C 83105,C(=O)(CCCC(N)=O)NCC1OCCN(C(C2(CC=C)CCOC2)=O)C1 83106,C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(CCNC(C(C(C)C)SCC)=O)CC1 83107,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83108,Cc1noc(N)c1C(=O)NCCOCCNC(=O)Cc1ccccc1F 83109,C1(NC(c2cn(CC(N)=O)nn2)=O)CCSC12CN(C(C1CC3CCC1O3)=O)C2 83110,c1(C(=O)NCCCN(c2ncc3ncnc-3[nH]2)C)cc(=O)c2ccccc2o1 83111,C1(OC)CN(C(c2ccc(C(C)C)cc2)=O)CC1NC(c1scnc1C)=O 83112,c1(NC(C(CC2CC2)NC(C(CO)OC)=O)=O)ccc(C)nc1 83113,N#CC1CN(C(=O)CC2CCN2C(=O)C2=CCOCC2)CCO1 83114,C(=O)(C1=CC2CCCCCCC12)NCCC(C)NC(=O)C(c1cccc(F)c1)O 83115,N1(C(C(C)(C)F)=O)C2CCC1C(F)C(NC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 83116,C(C(=O)C(C)(C)C)C1CCN(C(C)CC#N)C1 83117,N1(C(C(CCSC)OC)=O)CCC(C=CC(=O)NCc2nccc(C)n2)CC1 83118,c1(OC)cc(F)c(F)cc1C(=O)NCC1(C)CCCN(C(C2CC3CC2C3)=O)C1 83119,c1(-n2cc(CNC(c3n(C)cnc3Br)=O)nn2)cccn2ccnc12 83120,c1(CC)cccc(C)c1Cl.c1(C(=O)NC2CNC2)c[nH]nc1C(F)F 83121,Cc1occc1CNC(=O)C(C1CCCCC1)NC(C1CC1(F)Cl)=O 83122,Cc1nc(C)c(C)c(=NCC2CCCN2C(C2CCC(OC(F)(F)F)C2)=O)[nH]1 83123,CC1CN(C(=O)CS(=O)CC)CC1(C)C(=O)NCC(N1CCCC1)=O 83124,C=CC1OCCC1C(=O)NC1CC(O)C1N(C)CC.N12CC(C1)C2=O 83125,N1(C(c2cc(C)c(O)nn2)=O)C2COCC1CC(O)C2 83126,C1(NC(C2CC3(CC3)C2)=O)(Cc2cccc(Cl)c2)CCN(C(=O)CCC2CC2)C1 83127,C(=O)(C1CCOc2ccccc21)Nc1c(C#N)ncc(Br)c1 83128,c1(C(=O)NCC(C2(O)CN(C(C3CCCN(C)C3)=O)C2)(C)C)cnn2ccn(C)c12 83129,c1(C(N2CC(CN(C)C(C3CCCC(F)C3)=O)C2)=O)ccccc1-n1cncn1 83130,N1(C(C2(CCC)CCC2)=O)CC(C)CN(C(c2cncc(C)c2Cl)=O)CC1C 83131,C(=O)(C(F)(F)CC)N1CCC(N(CCC)C(C2CCCCO2)=O)C1 83132,N1(C(C(C=C)(C)O)=O)CC2(CC(NC(c3ccc(N(C)C)cn3)=O)C2)C1 83133,C1(C2CCC2)(CNC(C(C)(C)OCC)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1 83134,c1(C(N2CC(CCNC(c3n(C)cc(Cl)c3)=O)OCC2)=O)ccc2sncc2c1 83135,C1(C(N2C(C(C)(C)CNC(c3ccc(Cl)nc3)=O)CCC2)=O)CC2(C1)CC(O)C2 83136,N1(C(c2c(OC)nc(C)s2)=O)CCN2C(=O)N(C)C(=O)C2C1 83137,Cc1cc(C)c(C#N)c(NC(C)(C)CCNC(c2c[nH]cc(C)c2=O)=O)n1 83138,S(=O)(=O)(c1cccc(=NCc2nnc(C3CC3)s2)[nH]1)NC1CCCN(C)C1 83139,C1(CNC(c2c(CC)cccc2)=O)CC(C(=O)N2CC(N=[N+]=[N-])C2)=NO1 83140,N1(C(Cc2nc(=N)[nH][nH]2)=O)CCOC2(CCN(C(=O)CN3CCCCC3=O)CC2)C1 83141,N1(C(C(COC)C)=O)CC(NC(c2cn3ncccc3n2)=O)CCC(O)C1 83142,c1(OC)nc(C(=O)NCCCC(C)NC(=O)C(C)N2CCC2)sc1C 83143,C(C1CCCN1C(c1ccnnc1C)=O)=CC(=O)NC(C=C)(C)CC 83144,C1(OCCC)CCN(N2CC[SH](OCF)C2)C1 83145,Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NC1CCN(C(=O)C(Cl)=CCl)C1C1CC1 83146,c1(C(N2C(C(=O)NC(C3CCCOC3)C)CC2)=O)ccc(C(=O)N(C)C)cc1 83147,N#Cc1cccnc1Nc1cnn(CC2(O)CC2)c1.C12CCC(CC1)CNC2=O 83148,c1(C(=O)NC2CCC(C)(CNC(CC=C=C)=O)C2)ccc2cc(F)ccc2n1 83149,c1(N(C(C)=O)C)cccc(NC(C2CCN(c3cccnc3)CC2)=O)c1 83150,C12(C(=O)NCCCN(C(=O)CCc3ccccc3)C3CC3)CCCC1C2(F)F 83151,C(=O)(C1CCCc2nncn21)N(CCC)CCNC(=O)Cc1ccnc(O)c1 83152,c1(OCC)cc(Cl)c(C)cc1C(=O)OCc1ccccc1SC(C)C 83153,c1(CC)cc(OC2CC(NC)C23C(=O)N3)ccn1.C12(CC1)NC2.OC.CC 83154,N1(C(C(C)(C)C)=O)CC2CCCC2(Nc2cc3nncn3cn2)C1 83155,C1(NC(c2scc(COC)c2)=O)CC2CCC1(Cn1cc(-c3cc[nH]n3)nn1)C2 83156,C12(NC(c3c(C#N)ccs3)=O)CC3CCC(C1C2)N3C(=O)Cc1ccon1 83157,N1(C(C(=O)NC(CC)C)CC2CCC2)CCCC(C(=O)N(CCO)C(C)C)C1 83158,C1(C(N2C(C#C)CC2)=O)CCCCN1C(C1CC(N(C)C)C1)=O 83159,CC1(C)OC(=O)CC1C(N1CC(NC(=O)C=CCN2CCCCC2)C2(CC2)C1)=O 83160,c1(COC)c(C(=O)N(C)Cc2cn(CC(C)C)nc2C)oc2ccccc12 83161,C(=O)(C(C)CS(C)(=O)=O)N1CC(C)C(c2cc(Cl)ccc2F)C1C 83162,c1(C(=O)NCC2C(NC(c3cc(CO)[nH]n3)=O)CCC2)cccn2c(O)nnc12 83163,CC(C(=O)NC1CC(O)(CNC(=O)CCC(F)(F)F)C1)C(C)(C)C 83164,C1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)(C(=O)OCC)CCOCC1 83165,C(C(C)(C)C(=O)NCCOCCNC(=O)CSC(F)(F)F)SC(C(=O)SC)C 83166,CC(Cl)(Cl)C(=O)NCCO.C(C(=O)CC=O)OC(F)F 83167,c1(NC(C)C)nc(C(=O)NC2CC3CCC(C2)N3)cc2ccc(Br)cc12 83168,N(C1CC(C)n2ccnc21)C(=O)Nc1ccc(OC)c(-n2cnnn2)c1 83169,Cn1ncc(C(=O)NC(Cn2cncn2)C(=O)NCCCC(O)CO)cc1=O 83170,c1(C(=O)NCC(C)(CO)NC(c2n[nH]c(C)c2Br)=O)nccc(Cl)c1F 83171,N1(C(C2C3(CC(NC(CCC(=O)OC)=O)C3)C2)=O)CC(C(N)=O)OC(C)C1 83172,c1(OC)cccc(C(C)C(=O)NCC2(NC(=O)CCC(C)C)CC2(F)F)c1 83173,N#CCCCCC(N)C(=O)Nc1ccc2nnc(O)n2c1 83174,N1(C(CCc2ccn(C)c2)=O)CCC2(NC(=O)C3=NOCC3)CCCCC12 83175,c1(C(=O)OC(c2cc(C)c(Br)c(C)c2)C)noc2c1CC(C)(C)CC2 83176,c1(C(=O)NCC2(CNC(c3c(C)cnn3C)=O)CC2)ccc2cccnc2c1N 83177,c1(CNC(c2c(C)cccn2)c2nnnn2C2(C)CC2)cc2ccccn2n1 83178,c1(C(C)C)cccc(F)c1C(N1CCC(C)C(CNC(C2(C#N)CC2)=O)C1)=O 83179,Nc1ccc(C(=O)ON2CCN(C(=O)CC3C=CCC3)CC2)nc1C(F)(F)F 83180,C(C(=O)N1CCC(CCC(=O)O)C(NC(=O)CCC2CC2)C1)(C(C)(C)C)SC 83181,C(=O)(CC(C)(C)C1CC1)NCC1N(C(C(CC)C2CCC2)=O)CC1 83182,N1(C(CC(CC)C)=O)C(C)CN(C(=O)CC2CC3CCC2CC3)CC1C 83183,C1(C(C)C)CN(C(c2ccc(Cl)cn2)=O)CCN1C(C12COC(CF)(C1)C2)=O 83184,C1(NC(C(COCC(C)C)C)=O)CCCCC1CNC(=O)CC1CS(=O)(=O)C1 83185,N1(C(C(C)(C)C#N)=O)CC2(NC(=O)Cc3sc(O)nc3O)CCCC2(F)C1 83186,c1(-n2cc(CC(C(N)=O)NC3(C(C(=O)OC)OCC)CC3)nn2)ccc(Br)nc1 83187,Nc1c(C(=O)NCC2(O)CN(C(=O)C(F)=CCCF)C2)sc2ncccc12 83188,C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CC(=O)NCC2CCN(C)C2C)C1 83189,C1(CC#C)(C(=O)NCCCCO)CCN(C(=O)C(C2CC2)OCC)C1 83190,N1(C(c2c(C)cc(Cl)cc2)=O)CCN(C(=O)C=CC2CC2)C2CCC12 83191,c1(N2CC(C(=O)NCC3CC(=O)NCC3)C(F)(F)CC2)ncnc2c1CCCC2 83192,C1(C(N2CCC(c3nc(=N)[nH][nH]3)C2)=O)CCN(C(=O)C(=O)c2ccco2)CC1 83193,c1(OC)nc(Br)ccc1C(=O)Nc1ccccc1Br.N12CC(C1)N(C)CC2=O 83194,C(Cc1ccccc1)(C(=O)N1CC(CC(C)NC(=O)CCSC)C1)NC(=O)OC 83195,N1(C(C(C)N(CC)CC)=O)CC2CCN(C(C3CN(C)CCN(C)C3)=O)CC12 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83356,c1(C(N(c2nccc(CC(=O)OC)n2)CCOC)=O)coc2ccc(C)cc12 83357,c1(C(N(C2CCN(Cc3cc(Cl)c[nH]3)C2)CCC)=O)cc(-c2ccccc2)on1 83358,C(=O)(C(C)C(C)NC(=O)COC1CCC1)NCc1c(CC)nco1 83359,C1(CSCCC)CC(NC(CCCNC(c2nc(C)c(C)s2)=O)=O)C12CCC2 83360,Cc1cc(C(=O)NCC(CC2CC2)C(=O)NC2CC2C(C)(C)C)ccc1F 83361,C1(C(=O)OC)CC2CCC1N(C(C1CCCCO1)=O)C2.C12CCC(C1)NC2=O 83362,CCCCCC(O)C(=O)N1CC(NC(C23CCC(C2)C3(C)C)=O)C(F)C1 83363,C1(C(N2CC(C3CN(C(CC4N(C)CC=CC4)=O)C3)C2)=O)CCc2nnnn2CC1 83364,C12(C(=O)NCC#CCNC(c3n(C)ncc3C(F)F)=O)CCCCC1NC(=O)C2 83365,CCC(O)C(C)(C)C(=O)NCC1(CNC(=O)C=CC(=O)NC)CCCC1 83366,C(=O)(CC(C(F)(F)F)C1CCOCC1)N1C(CC(CC)O)CC1 83367,n1(CC(=O)NC2C(CNC(C(CC)OCC)=O)COC2)ncn2nccc2c1=O 83368,CCC(C(F)(F)F)NCCc1cn(-c2cccc(C(=O)OC)c2)nn1 83369,c1(CC(=O)NCC2(C(N)=O)CN(C(C(C)OCC)=O)C2)c(C)cnn1C 83370,c1(C(=O)NCc2ccccc2)cc2cccc(-c3ccc(C(F)(F)F)s3)c2s1 83371,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCC(C1)N2C(=O)Cn1ccnc1C 83372,N=c1nc(Cl)cc(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)[nH]1 83373,c1(C(N2C3(CNC(COC)=O)CC(C2)C3)=O)cc2ccccc2c(C)c1F 83374,N(C(=NCCOC(=N)O)NC1CCC1)Cc1cc(-c2ncn(C)c2)on1 83375,c1(C(N2CCC2CO)=O)ccc(N)cn1.C12CCCC1C(=O)NC2 83376,C(=O)(C(O)Cn1cncn1)N(C(C)C)CCC1CCCCC1 83377,c1(CNC(C)=O)cc(F)c(C(C)Nc2cc(C)c(C)s2)cc1Br 83378,c1(SC)cccc(C(N2CCC(CCNC(=O)CCc3cccc(O)n3)C2)=O)n1 83379,C(=O)(C#CC1CCOC1)NC(c1ccnn1C)C(=O)NC(CC#C)CC(F)F 83380,C1(C(C)(CO)NC(=O)NC(CNC(C)C(=O)C2CC2)COC(C)(C)C)CCCCC1 83381,CC1C(C(=O)N(C2CCSC2)C)CCN1C(C1C2CCCOC12)=O 83382,Cc1cc(=NCc2cccc(NC(c3ccc4ncccc4c3)=O)c2)[nH]c(C)n1 83383,N1(C(c2c(OC)nc(Cl)cc2)=O)CCCc2nc(Cl)ccc21 83384,C1(C(=O)Nc2c(C)ccc(O)c2)CCC2(CN(Cc3cccc(C(F)F)n3)C2)O1 83385,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(CNC(C1C(C(=O)OCC)C1)=O)C 83386,N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(S(C)(=O)=O)CCC1C 83387,c1(C(=O)NCC2(NC(c3cc(C)sc3C)=O)CCOC2)ccnc(C)c1N 83388,[N-]=[N+]=Nc1ccc2c(c1)CN(Cc1cc(F)ccc1F)CC2 83389,c1(CC(=O)NCC2(C)N(C(CCCN(C)C)=O)CC(O)C2)cc2ccccc2s1 83390,c1(C(=O)NC(CSCC)C(=O)OC)cn(C)c(C(=O)N(C)Cc2cscn2)n1 83391,CC(C)CC(C)CC(=O)NC1CN(C(c2cc(O)ccc2OC(F)F)=O)CC1F 83392,C1(C(N2C(CCNC(C(CCCOC)C)=O)CCCC2)=O)CC1C1CCCCC1 83393,C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1OCCN(C(C2CCC(C)(C)OC2)=O)C1 83394,N1(C(c2c(COC)ncs2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83395,C1(CCC)CN(C(=O)CCc2ccncc2)CC1NC(c1c(Cl)noc1C)=O 83396,C1(CC)COCCC1(c1nnnn1C)NCC1(OC)CC(SC)C1 83397,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3CCC(=O)C23)=O)C1)=O 83398,c1(C(=O)NCCN(C(C(C)SC)=O)CCCN(C)C)cnc2[nH]c(C)nc2c1 83399,c1(OCC)cccc(C(=O)NCC2CCN(CCF)CC2c2cnn(C)c2)c1N 83400,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83401,Cn1nc(C2CCC2)ccc1=O.c12nc(nn1C1CCOC1)COc1n[nH]cc1-2 83402,Cc1cc(C)c(C(N2CC=CC(NC(=O)C(=Cc3cccnc3)F)C2)=O)c(N)c1 83403,Cn1c(CC(N2CCC(F)(c3cn(-c4ccccc4)nn3)C2)=O)nnc1S 83404,c1(CNC(C(CNC(CCC=C(C)C)=O)O)=O)cccc(C#N)c1 83405,n1(CCNCCCc2nccs2)cncc1C(c1nnnn1CC1CCCO1)OC 83406,c1(OCCO)ccccc1Br.C12CC(C1)NC(=O)C1CC(C1)C(=O)N2 83407,N1(C(c2cc(C)ns2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83408,CCCCCC(C(=O)NC(C1CN(C(=O)Cc2coc(CC)n2)CCO1)C)C(C)C 83409,N1(C(c2c(C)scc2)=O)CC(CNC(c2ccn3cncc3c2)=O)CC12CCC2 83410,C#CCC(C)(C(=O)N(C(C)CCC(C)C)C)NC(=O)C=Cc1ccsc1 83411,N1(C(C2(CSC)CC2)=O)CC(CCNC(=O)CN2CCC2)C1 83412,c1(CCCC)nc(OCc2ccccc2)c(N(C2CC(OCC)C2)C)c(Cl)n1 83413,Cc1cc(NCC2CC(NC(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83414,c1(C(N2CCC(CC(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83415,Cc1ccc(C2CC2C(=O)NCC2(NC(=O)CC(C)C(C)C)CCC2)c(Cl)n1 83416,Cc1c(C(N2CC(C(O)C(=O)NC3CC(C)(CO)C3)C2)=O)cccc1C#N 83417,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)on2)=O)CC1C 83418,Cc1cnc2c(C(N3CC(NC(=O)Cn4cnnc4O)CC(F)C3)=O)cccn12 83419,C1(C(=O)NC2CCC(CNC(C(COC)(C)O)=O)C2)CC(C(N)=O)=NO1 83420,N1(C(c2[nH]nc(C)c2Cl)=O)C2CCC(C2)C1CNC(c1c(F)ccnc1F)=O 83421,c1(C(N2CCC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)=O)cnc2cc(Cl)ccn12 83422,C12(C(N3CCCC(CC)(NC(=O)C=CCO)C3)=O)CCC(C#N)(CC1)CC2 83423,CC(CC(=O)NC1CS(=O)C1)N(C(=O)CCc1ccn(C)n1)C 83424,c1(OCC=C(C)C)ccc(Br)cc1O.C12CCC(C1)OC2=O 83425,C(CCCCCCC(=O)NC1CC2CN(C(c3occc3Cl)=O)CC2C1)SC 83426,O=C(N1OC2C=CC1CC2)C12CC(CN1C(c1ccon1)=O)C2 83427,C(=O)(C(CCC)C(C)C)N(C1CCCN(C(Cc2c(NC)nccc2)=O)CC1)C 83428,C(=O)(CC(C)(C)OC)NC(C1(O)CN(C(C2N(S(CC)(=O)=O)CCC2)=O)C1)C 83429,C12(CCN(C(=O)C(=O)N(C)C)CC1)C(=O)NCC2.c1(C(C)N(C)C)cnn(C)c1 83430,C(=O)(C(C)(C)C(C)(F)F)N(C(C(N1CCCC(C#C)C1)=O)C)CC 83431,C(=O)(CCCCC(F)F)NCC1C(NC(c2cnn(C)c(=O)c2)=O)CC1 83432,c1(C(=O)N(CCN(C(C2CC(CC(C)(C)C)C2)=O)CC)CC)ccc(Br)nc1N 83433,C1(C(N2C(CNC(=O)CP(C)(C)=O)CC(OC)C2)=O)CC(C(C)(C)C)=NO1 83434,c1(C(=O)NC(CNC(c2c(CC)noc2C)=O)(C)C)ccc(Cl)cc1C 83435,c1(CNC(C2CCCCCC2)c2n(CCOC)nnn2)ccc(C(N)=O)cc1 83436,N1(C(c2c(C)n(C)nn2)=O)CCN(C(c2ccnn2C)=O)CC1c1cccnc1 83437,CC(C(=O)NC1C2CC1N(C(C1CCCCC1C(F)(F)F)=O)C2)C(C)(C)C 83438,CC1(C)CCN(C(=O)CCc2ccccn2)CC1NC(C12CCCC1C2(F)F)=O 83439,C=CCC(CNC(=O)Cn1ccnc1)C(=O)N1CC=CCO1 83440,C1(CN(C(=O)C(C)Sc2nncn2C)C)CCN(C(=O)C=CC(C)(C)C)CC1 83441,CN1CCN(N2CCC(N3CCN(C(C4CCCC(=O)O4)=O)CC3)C2)CC1 83442,c1(C(N(C2CCN(C(=O)Cc3c[nH]nc3O)C2)C)=O)cc2cnn(C)c2s1 83443,CC(CC(=O)NCCC1(CNC(c2ccn(C)c(=O)c2)=O)CC1)CC(F)(F)F 83444,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(=O)Cc3cn(C)cn3)C2)C1 83445,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCOC(CC)=O)=O 83446,c1(C(N2C(CCC(=O)NC(CC(=C)C)C)CCCC2)=O)n[nH]cc1[N+](=O)[O-] 83447,c1(CC)ccc(I)c(O)c1.c12ccc(cn1)NC(=O)C1CN(CCO1)C2=O 83448,C=CCC(CC(=O)NC(CC)C(F)(F)F)NC(=O)Cc1ccc(C)s1 83449,c1(CNC(C(CCOCC)NC(=O)C(F)(F)CSC)=O)sc(C)c(C)c1C 83450,C(=O)(C1CCCc2nncn21)C(C)=O.C1(CCC(C)C)C(=O)N2CC3(C2)CN1C3 83451,C1(NC(c2c(CC)nco2)=O)CN(C(C2CC(=C3CC3)C2)=O)CCC1F 83452,C1(C(N2C(CNC(C34CCC(CC3)CC4)=O)CCCC2)=O)CC1C1CCCCC1 83453,c1(C(N(C2C3CN(C(c4c(C)ncnc4)=O)CC32)C)=O)ccc2nn[nH]c2c1 83454,CC1(C)CCCCC1C(=O)NCCN(C(=O)C1=CCCCC1)C1CCCCCC1 83455,N1(C(C)CC(=O)N2CC(OCCNC(=O)C(O)c3ccsc3)C2)CCCCC1=O 83456,C1(O)(C(=O)NC2CCC(NC(c3cc(OC)nn3C)=O)C2)CC2(CCOCC2)C1 83457,C1(CNC(=O)Cc2ccsn2)CCN(C(=O)CCC2CCOCC2)CC1O 83458,Cc1noc2cc(C(N3CC(CCNC(=O)COC(C)C)C(C)C3)=O)ccc12 83459,CCCC(CC)S(=O)(=O)NCc1cnn(-c2ccccc2)c1C(=O)O 83460,c1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)c(C)cc(C)cc1N 83461,CC1CCN(C(C2CC(=O)N(C)C2)=O)CCN1C(=O)CCN1CCCCC1=O 83462,N1(C(Cn2c(C)ncc2)=O)CCCC2(CCN(C(=O)C(F)C3=CCCCC3)C2)C1 83463,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 83464,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 83465,c1(OCCC)ccc(-c2nc(CCC(C)C)nn2-c2ccn(C)n2)cc1OCC 83466,C(C)(CO)(C(=O)NCC1CC(NC(c2cnn(CCO)c2)=O)C1)NC(=O)OC 83467,CC(C)(C)CCCCNC(C1(NC(c2cc[nH]n2)=O)CCSC1)=O 83468,N1(CC=CC(=O)N(CC(C)N(C(CC)=O)CC)C)CCCCCC1 83469,c1(NC2CCN(CCC)CC2)[nH]c(=NCC(CC)C(C)(F)F)nc2sccc12 83470,c12cc(no1)CNC2=O.C(=O)(C(C)C1CCOC1)N(CC=C)CCO 83471,C(=O)(C(C)C(C)(C)C)NC(c1conc1C(C)C)C(=O)Nc1c(C)cccc1 83472,N1(C(CCCC#CC)=O)CC2CCC(C1)C2CC(N1CC(OC)CC(F)(F)C1)=O 83473,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 83474,Cc1cc(NC(C2C3CCC(C3)N2C(c2csc(C3CC3)n2)=O)=O)c(C)cn1 83475,C(=O)(C(C)(C)CC(F)F)NC1(CF)CCN(C(c2cnn(C)c2C(C)(F)F)=O)C1 83476,C(C(C)(C)S(C)(=O)=O)NC.Cc1n[nH]c(C)c1CN(C1CCN(C(=O)N)CC1)C 83477,C#CCCN=C(NCC(=O)NC1(OC)CCS(=O)(=O)C1)NC(c1cccc(F)c1)C 83478,C1(NC(C(C)SCC)=O)CC2CN(C(c3nc(C)n(C4CC4)c3C)=O)CC12 83479,N1(C(COCC=C)=O)Cc2n[nH]cc2C1C(=O)N(C1CCCCCC1)C 83480,C(c1c(N)cnn1-c1ccccc1C)=CCNC(CCCCC1CC1)c1nccs1 83481,c1(C(C(N2CCC(n3cc(COCC=C)nn3)C2)=O)(C)C)cccc(OC)c1 83482,c1(CN2CCC(O)(Cc3ccccc3)C2)noc2c1COCC2 83483,CCC(C)CC(=O)NCC(C1CC1)NC(=O)Cc1n[nH]cc1C 83484,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 83485,c1(CC)cc(C(N2CC3CC3(NC(=O)C(C)C(C)(C)C)C2)=O)cc(C(F)(F)F)c1 83486,O=C(C1=CCCOC1)N1CCN(C(=O)C(F)n2cccn2)C(CF)C1 83487,c1(NC(C)=O)ccc(F)c(C(c2nnnn2C2CC2)NC2(C=C)CCCC2)c1 83488,N1(C(CCN(c2n[nH]c(C)c2[N+](=O)[O-])C)=O)CCc2ccc(N=[N+]=[N-])cc2C1 83489,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 83490,CC1CN(C(C2CCN(C)C2=O)=O)CCC1NC(=O)C(C)Cc1cccc(Cl)c1 83491,N1(C(CCc2n(C)ccn2)=O)CCN(C(C2CC(=O)NC(=O)C2)=O)CC(C)(C)C1 83492,c1(OC)cc(C=CC(=O)OCCNC(C2CCCC2(F)F)=O)ccc1OC 83493,C(C)(c1ccc(F)cc1)=CC(=O)NCC1N(C)CCN(C(C(C(CC)O)C)=O)C1 83494,c1(C(=O)NCC(c2ccccc2F)NC(C(C2CC2)OC)=O)cc(C#N)[nH]c1C 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83634,C(=O)(CC(C)NC(N)=O)NCC(CO)OCC.C1(C2C(=O)N2)CC=CCC1 83635,Cc1nn(Cc2nc(-c3cc[nH]n3)nn2CC)c2ncccc12.c1(C)cccnc1 83636,N1(CC(=O)NCc2ncoc2CCn2cc(CCCC)nn2)CCCCCC1 83637,c1(CNC(c2n(CC=C)nnn2)c2sccc2C)cc(C)cc(C)c1 83638,C1(CC)(CC)CN(C(=O)NC23CC(CO)(C2)C3)CCS1 83639,C(C(=O)N1CC(NC(c2cc(O)n(C)n2)=O)CC1(C)C)(C(C)(C)C)NC(C)=O 83640,C(N=c1cc(-c2ccccc2)nc(Cl)[nH]1)C1CC(C)N(C(=O)C(F)C2CCC2)C1 83641,N1(C(CC2C(C)CCC2)=O)CCC(CCNC(C2(n3cc(Cl)cn3)CC2)=O)CC1 83642,CCC(CC)CCC(=O)NCC(c1ccc(F)cc1)NC(c1cc(OC)ns1)=O 83643,Cc1ccc(C(=O)NCc2cc(C(=O)NC3(C)CCCC3O)ccn2)cc1Cl 83644,N1(C(CC(=O)NCC)=O)CCC2(CC1)CC(CNC(=O)CC(C)C(F)F)CO2 83645,C(C)(N=c1[nH]c(N(C)CC2CC2(F)F)nc(=NC)[nH]1)C1Oc2c(OC)cccc2C1 83646,C1(C(N2CC(CO)(NC(=O)CC(=O)OCCC(C)C)C2)=O)(CC)CCCC1O 83647,N1(C(C#CC2(C)COC2)=O)CCC2CCN(C(c3nccnc3C(N)=O)=O)C2C1 83648,N1(CCC)CCCC(CCNC(C2CCCCN2C(=O)COC2CC=CC2)=O)C1 83649,C=CCC(CC(C)C)C(=O)NCC(CCC)C(=O)NCc1ncc(F)cc1F 83650,CC(CC(=O)N1CCCN(CCNC(C23COCC(C2)C3)=O)CC1)CC(C)(C)C 83651,C(C(C)(C)CC(=O)NCC(C)(C1CC1)NC(=O)CC(C(F)F)N(C)C)OC(C)=O 83652,C(=O)(CCCN(C)N=O)NCCC1OCCN(C(CC2C(C)CCCC2)=O)C1 83653,c1(C(N2C3CN(C(C4N(CC)CCCC4)=O)C(C3)C2)=O)oc2ccccc2c1C 83654,C1(C(=O)NC2(C(=O)NCc3nccc(C)c3)CC2)C2CCC(C2)C1C 83655,C(C)(CNC(C1(c2ccnn2C)CC1)=O)(C(C)C)NC(c1c(C(C)=O)ccs1)=O 83656,N1(C(C2CCC(C)(C)O2)=O)CCC2CC2(C(=O)N(C23CCC(CC2)C3)CCO)CC1 83657,CC1=CCC(C(N2CCC(C)(NC(c3cnoc3-c3ccc(C)o3)=O)C2)=O)CC1 83658,S(=O)(=O)(C1(CSc2cccc(Cl)c2)CC1)NC.N12CCC(C1)NC2=O 83659,N1(C(C(C)CC2CCCO2)=O)CCC(CN(C)C(C2(n3cccn3)CC2)=O)CC1 83660,C1(OCC(C)C)CC2CCC(C1)N2C(N1CCC(C(=O)OC)CC1)=O 83661,N1(c2nc(OC)nc(C)c2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 83662,C1(N(C(c2c(CC)n[nH]c2)=O)C)CCCN(C(=O)CN(C)C(C)=O)C1 83663,N1(C(c2cccc(C#C)c2)=O)CCCCCCC1C(=O)NCC1CCC(C)C1 83664,C(=O)(C(C)(C)C(N)=O)N(CCC(C)NC(c1cnn(C(C)C)n1)=O)C 83665,N1(C(C(Cc2ncn(C)c2)O)=O)CCC(F)(C2CC(NC(=O)CS(C)(=O)=O)C2)CC1 83666,n1(C(C)C)cnc(C(N(C2CCC(NC(=O)C(=O)N(C)C)C2)CCO)=O)c1 83667,C=CCC(CC)C(=O)NC(C)(C)CCC(=O)N(CCC(=O)OCC)C 83668,c1(OC)ccc(CC(N2CCCN(C(C3CN(C4CC4)C3)=O)CC2)=O)cc1F 83669,N1(CC(C)S(=O)(=O)NC(=O)CNc2nccnc2C#N)CCc2ccccc21 83670,CN1CC(CNC(=O)NCC2CN(Cc3ccnn3C)CCO2)CC1=O 83671,c1(C(=O)OC)cc(F)cnc1NC(C1CC12CN(C(c1cc(C)nc(C)n1)=O)C2)=O 83672,c1(C(N2C(CCNC(CCC=CCC=C)=O)CSCC2)=O)cc(F)cc(C)c1N 83673,C(C)(C)(C#Cc1cn(CCCCCO)nn1)NC(c1c(Br)ccc(C)c1)=O 83674,CCCC(CNC(c1ncn2c1CCC2)=O)C(=O)NC1CC2(C1)CC2OC 83675,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)NCCc1ccns1)C1CC1 83676,C(=O)(CCCCC(=O)N1CCN(C)CC1CNC(=O)C(O)C1=CCCC1)NCC 83677,CN1CCC(=CC(N2CC3C(CC(=O)NC4(CCO)CCOCC4)C3C2)=O)CC1 83678,Cc1csc2ncc(NC(=O)NCC3(O)CCCN(C(=O)OC(C)(C)C)CC3)n12 83679,c1(C(=O)NC2(C(=O)NC(C(C)SCC)C)CC2)ccc(C(=O)OC)nc1.C1CC1 83680,C(CCCCCCCC(=O)Nc1cnc(O)nc1O)n1cc(CSCC)nn1 83681,c1(-c2cn(C3CCC(C(=O)NCc4cncn4C4CC4)C3)nn2)ccc(Cl)cc1 83682,C(=O)(CC(C)CN(C)C)NC1CC(CC(=O)NC(c2cccc(Br)c2)C)C1 83683,C(CN=c1[nH]c(N2CCCC(C(F)F)C2)nc2ccsc12)=C(C)C 83684,N1(C(=O)Cn2nccn2)CC2CCC(C1)N2C(c1ccc(I)cc1Cl)=O 83685,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 83686,c1(CC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cnn2c1OCCC2 83687,N1(C(C2(C#C)CCOC2)=O)CC2=C(C1)CN(C(c1cc(F)ccc1CC)=O)C2 83688,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)C)cccc(C(C)=O)c1 83689,CC(C(F)(F)C(F)F)NC(C1CCCN(C(=O)NC2CC2)C1)=O 83690,C(=O)(C(Cc1ccco1)NC(=O)CCC1CCCOC1)NC(C=C)C1CC1 83691,N1(C(C2CCC(CCC)CC2)=O)CCN(C(=O)CCCCCSC)CC1COC 83692,c1(CC)cc(C(=O)NC2CCN(C(=O)CC3(C(F)(F)F)CC3)C2)c(C)o1 83693,c1(CNC(=O)CC2CC(NCc3ccnc(O)c3)C2)cccc2c1CCC2 83694,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)C(C)OC1CCCC1)OC 83695,c1(CC(N2CC3CC(CNC(C4(C)CC4)=O)C3C2)=O)ccc2ncsc2c1 83696,N1(C(CC2N(CC)CCOC2)=O)CCC2OCCN(C(=O)CC(CC)OC)C2C1 83697,C1(C(N(C)CCNC(c2ccc(C3CC3)cc2Cl)=O)=O)CSc2ccccc2O1 83698,C12(CNC(CC(C=C)(C)O)=O)CCCC(CN1C(=O)C=Cc1ccc(C)cc1)C2 83699,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 83700,S(=O)(=O)(c1cccc(C(F)F)c1)N1C(C2CCN(C(C(=C)F)=O)CC2)CCC1 83701,c1(N(C(c2ccccc2O)C(=O)NC)CC)ccc(OC)cc1.C(C(=O)OC)OCC 83702,c1(C(C)C)cc(F)ccc1C(=O)NCC(CNC(=O)COCC1CC1)CO 83703,C1(NC(CN(C(C2(C)CCCN(C)C2)=O)CC2CC2)=O)CCCN2CCCCC12 83704,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(CC3CC3)c2)=O)C1 83705,c1(CC)c(C(=O)N(C2CCN(C(=O)C(C)Sc3ccccc3)C2)CC)nnn1C 83706,C(=O)(CC(CC(C)C)NC(=O)CC1CC2CCC1C2)Nc1onc(C)c1C 83707,N1(C(CC(C)(F)F)=O)CCCC(C2CCCN(C(c3cnc(N)c(N)c3)=O)C2)C1 83708,N1(C(C2CCN(C(C3CC3C3CCC3)=O)CC2)=O)CC2CCCCC2(CO)C1 83709,C(C)(CNC(c1c[nH]nc1C1CC1)=O)(C(C)C)NC(C(CO)OC)=O 83710,C1(N(C(=O)CCc2cnoc2)C)CCC(CNC(C2C3CCC2CC3)=O)CC1 83711,c1(NCc2c(OC)ncc(F)c2)cnc2ccc(F)cc2c1 83712,N(C(=NCCF)NCc1ccc(Cl)s1)Cc1cnc(C(=O)OC)o1 83713,C1(C(=O)NC(C)CNC(=O)C(C)SCc2ccccn2)CCCCC1(F)F 83714,c1(OC)c(C(=O)NC2CCC(NC(C3(C)CCNC3=O)=O)C2)c(C)nn1C 83715,C1(O)(CNC(=O)C(C2CCCCC2)O)CCCN(C(=O)CC2CCC2)C1 83716,CCC(COC1CCOC1)(CC)C(=O)N1CCC(C(=O)NC2CC2)O1 83717,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCCOCC1)=O 83718,c1(C(=O)NC2(CNC(=O)C(O)C3CCC3)CCOC2)cc2ccccc2cn1 83719,Cc1c(C(N2CCC(C(C)NC(=O)CSc3ncccn3)CC2)=O)nnn1C 83720,C1(n2cc(CNC(=O)CO)nn2)(C(=O)OC)CCN(C(c2ccc[nH]2)=O)C1 83721,C1(OCC)CCC(C(=O)NC2C(CNC(C)=O)C2)CC1.C1(Br)(C(=O)N)CC1 83722,C(=O)(C(C)(C)C(N)=O)N1CC(C2C(=O)N2)C1.c1(COC)cnc(O)c(F)c1 83723,N12CCCC(C1)C(=O)NC1C=CCCC1C(=O)NCC2.C1(O)CC1(F)F.CS 83724,CC(=O)CC(C)(C)C(=O)N1C2CCC(C(=O)NCC3CC(O)C(O)C3)C1CC2 83725,C1(C(=O)NCC(=O)OCC)CCC(C(C)C)N1C(=O)C=Cc1cc[nH]n1 83726,c1(C(=O)NCC(C2CCCCC2)NC(c2cncn2C2CC2)=O)ccncc1F 83727,c1(C(N2CC(NC(C3(C(N)=O)CC3)=O)C(F)C2)=O)cnc2n1CCOC2 83728,C(CO)(CCCCNC(=O)CCc1cscn1)NC(c1nc(C(C)(C)C)sc1)=O 83729,c1(C(=O)NCCCNC(CC2COCC(C)O2)=O)cccc(F)c1F 83730,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 83731,C1(C(=O)NCC2(CCC)CC2)CCCCN(C(=O)C(C)(CO)OC)C1 83732,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(C2SCCS2)=O)C1)C 83733,N1(Cc2ccc(-c3ccc(OC)cc3)nc2)CCOC(C2CC2)CC1 83734,c1(CNC(CCN(CCC)C)=O)ocnc1C(=O)NCC1CCN(C(C)C)C1 83735,c1(C(=O)NC2CC(NC(c3c(C)cco3)=O)C23CCC3)sc2ccsc2c1C 83736,N1(C(C2CCN(NC(C(CC)C)c3ccccc3)CC2)=O)CCN(C)CC1.C(C)=O 83737,c1(NC(C(C(C)C)SC)=O)ccc(NC(=O)C(C2CCC2)N(C)C)cc1C 83738,C(=O)(C(C(C)(C)C)C1CCCCC1)N(CCCNC(c1cn(C)nc1O)=O)C 83739,CC1CN(C(C2(c3ccccc3F)CC2)=O)CCN1C(c1ccc(O)nc1Cl)=O 83740,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CC2)=O)C1 83741,Cc1cc(F)c(C(=O)NCC(C)CNC(c2csc(C(N)=O)n2)=O)cc1Br 83742,CCC(CNC(c1cnc(C)c(C)c1)=O)(CC)C(=O)NC1CCC1N(C)C 83743,Cc1scc(C(=O)NCCC2(O)CCN(C(=O)CCC3CCCOC3)C2)c1C 83744,CC1(C)COC(CCC(=O)NCCCOCCNC(=O)CCn2cncn2)C1 83745,c1(CNC(NCC2CCOC2)=NCCCCl)cc(F)cc2nc[nH]c12 83746,Cc1cc2[nH]c(C(=O)NCC3(NC(C4(C(=O)OC(C)(C)C)CC4C)=O)CC3)cc2o1 83747,C(CC(C(=O)NC)NC(=O)CCC1CCCO1)OC.c1(COC)nnnn1C 83748,C12(NC(C=C(CC)C)=O)CCCC1N(C(c1ccc(C(N)=O)cn1)=O)CC2 83749,N#Cc1ccc(C(C(N)=O)NC(=O)NC2CCN(c3ncc(F)cn3)C2)cc1 83750,CC(O)C(CC(=O)NC1CCN(c2ccncc2)C1)c1ccccc1 83751,Cc1cc(C(N2CC(O)CCC2C(=O)N(C)C)=O)cc2ccoc12 83752,C1(C(=O)NC(C)CSC(F)F)CCCCN1C(C1CCCCO1)=O 83753,C1(NC(=O)CCCc2ccc(F)c(F)c2)C2CC3CN(C(=O)C4=CCC4)C1C3C2 83754,c1(C(=O)NCC2CCC(O)CN2C(=O)CN2CCCCC2)cn2ncccc2n1 83755,C(CNC(=O)CSCC(N)=O)(CN(C)C)OC.C1(=O)CCN1 83756,C1(C)(CNC(C(c2cccc(C(F)F)c2)C)=O)CN(C2CCC2)CCO1 83757,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 83758,c1(C(N(CCCF)C)=O)cc(CNC(C2C3CCC(=O)C23)=O)nn1C 83759,CCC(CC1CCCC1)C(=O)N(C)CCN(C)C(C1CC(C)(F)C1)=O 83760,C(=O)(C1=CC(C)(C)C1)NC(CC=C)CNC(C1CC1c1ccc(F)cc1F)=O 83761,c1(C(N2CC(CNC(C(C)N(CC)CC)=O)C(O)C2)=O)cccc2ccoc12 83762,C1(C(=O)NCc2nnc(C)n2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 83763,N1(C2(c3csc(C)c3C)C(=O)NCC2(CC)SC)CCC(F)(F)C(C)C1 83764,c1(N(CCNC(c2ccc3ocnc3c2)=O)CC)nc(O)c2c[nH]nc2n1 83765,c1(NC)cnccc1C(=O)NC1C=CCN(C(=O)CS(=O)(=O)NCC2CC2)C1 83766,CN1CCC(NC(C2CCCCN2C(C2CC3CCCC3C2)=O)=O)CC1=O 83767,C1(CNC(c2cc(OC)ncn2)=O)CC2(CC(NC(=O)C(F)(F)CC3CC3)C2)C1 83768,C1(NC(C(CC)CC=C)=O)CCC2(C1)CN(C(=O)Nc1cc3cn[nH]c3cn1)C2 83769,N1(C(C=CC2N(C)CCC2)=O)CC2CCC2(CCNC(c2cnnn2C)=O)C1 83770,N1(C(CCC)=O)CCC2(CCCN(C(c3ccc(Br)c(Cl)n3)=O)C2)C1 83771,CC1CCC(C)(CNC(c2coc(CNC(=O)C(C)(O)C3CCC3)n2)=O)CC1 83772,C1(N(C)C)C2CN(C(=O)C(CO)NC(c3csc(Cl)n3)=O)CC12 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84085,C1(C(=O)NCC(O)CNC(c2cccnc2O)=O)(OC)CCCC(C)(C)CC1 84086,C(C1c2ccccc2CN1C(C1CC(F)(CO)C1)=O)NC(CP(C)(C)=O)=O 84087,N1(C(C2(C)CCN(C)C2)=O)CCN(C(c2ccsn2)=O)CC(C)(C)C1 84088,N1(C(c2ccc(F)cc2Cl)=O)CCC(N=c2[nH]nc(C(F)F)s2)(CO)CC1 84089,Cc1cc(C(=O)N(C(C)(C)CC(=O)NC2CCCC2(F)F)C)nc(O)c1 84090,C1(C(=O)NCC2(C(C)NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 84091,C1(COC)CN(C(C2CC3CCC(C2)O3)=O)CCN1C(C1(C(=O)OC)CCC1)=O 84092,N1(C(c2c(OC)c(C)ccc2)=O)Cc2ccnn2CC(NC(=O)CCCC#N)C1 84093,c1(C(N2CCC(N(C(=O)COCc3nnc[nH]3)CC)C2)=O)cccc2sncc12 84094,c1(C(NC(=NCC2CC(OC)C2)NC2CCC2)C)ccc(F)cc1C 84095,N1(C(C2(COC)CC2)=O)CC2C(C(=O)NCCc3cncnc3)C2C1 84096,C=CCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NC1COCC1C=C 84097,c1(OC(C(=O)NC2CC(CNC(c3c(C)cns3)=O)C2)C)ccc(Cl)cc1 84098,C1(NC(Cc2cc(C)nn2C)=O)CCC2CC1CN2C(=O)CCCCC(C)C 84099,C1(C(N(CCOCCNC(c2cnc(C(C)O)s2)=O)C)=O)CN2CCC1CC2 84100,N1(C(C(F)=CCC)=O)CCC2CCN(C(c3ccc(F)c(C(F)F)n3)=O)CC2C1 84101,c1(OCC(=O)NCC(C)(C(C)C)NC(Cc2nc(C)[nH]n2)=O)c(Cl)cccc1Cl 84102,N1(C(C2CN(C(C3(COC)CC3)=O)C2)=O)CCC(C#N)C1 84103,C(CC(C)(C)C(=O)NCC(CO)NC(C1(F)CCN(C(C)(C)C)C1)=O)OC 84104,c1(C(N(CCCCNC(CC(CC)OC)=O)C)=O)cc2cccc(Cl)c2[nH]1 84105,c1(C(=O)NCc2ccc(C(C)NC(COCC)=O)cc2)nnn2c1CCCCC2 84106,C(=O)(C(C)C1=CCCC1)NC(CC)CNC(=O)CC1(c2ccc(C)cc2)CC1 84107,N1(C(CS(=O)(=O)NC)=O)CC2(C1)CN(C(C13CCC(C)(CC1)OC3)=O)CC2CO 84108,C(=O)(CCN=[N+]=[N-])NCCCC(=O)N(C1(c2nc(=O)o[nH]2)CCC1)C 84109,CC(N=c1[nH]c(N2Cc3ccc(C#N)cc3C2)nc2cc[nH]c12)C1CC1 84110,C1(OC)CCC2CCC1N2C(=O)CC1(O)CCCCCC1.C=CC1CCCN1C 84111,Cc1cc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C2)=O)ncc1C(N)=O 84112,C1(C(N(CC#CC)C)=O)CC2(CC2)CN1C(C1CC12CCC2)=O 84113,c1(C(=O)Nc2c(C)cc(NC(C3CCCO3)=O)cc2)ccnc2c1cnn2C 84114,C1(CNC(=O)Cc2ccnn2C)CCCOCC1.C1CC(=O)N1C(C)C 84115,C(C(C(=O)N1CCC(SC)C1)NC(=O)C(O)CN(C)C)OC 84116,C1(NC(C=CCC)=O)C2CCCCCC12.C12CCC(CC1)N2C(C12CCCC1C2)=O 84117,S(=O)(=O)(c1cc(Br)c(C)cc1F)N(CC(C)C)Cc1c(C)ccc(C)c1 84118,Cc1ccc2c(CC(=O)NC(C)CN(C(=O)C(O)P(C)(C)=O)C)coc2c1 84119,N1(C(C(CCOC)C)=O)CC2(CCCC2NC(C2(OC)CCOCC2)=O)C1 84120,N1(C(c2c(C)nc(Br)s2)=O)CCC2C(CCN2C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 84121,CCCC(CCC)C(=O)N(C1CN(C(=O)Cc2cc[nH]n2)C1)C 84122,C1(NC(c2nnn(C)n2)=O)CCCCN(C(c2cc(C#N)no2)=O)C1 84123,C(C(C(C)C(C)C)NC(=O)Cc1csc(S)n1)NC(CC=CC=C)=O 84124,C1(NC(c2ccc(OC(F)F)cn2)=O)C2CC1CN(C(=O)C=C1CCC1)C2 84125,N1(C(C(C)N(C)C)=O)C2CCCC1CN(C(=O)CON=C1CCCCCC1)CC2 84126,C1(NC(CCOCC)=O)CC(C)(NC(c2cnc[nH]2)=O)C1 84127,C1(CNC(c2ncccn2)=O)CCCCN(C(=O)CCOCC2CCC2)C1 84128,N1(C(C2C(C)OCCO2)=O)CCC=C(CNC(=O)Cc2cnsc2)C1 84129,C1(CNC(c2ccc(O)c(F)c2)c2n(CCOC)nnn2)CCOC(C)(C)C1 84130,N1(C(c2c(C)cc(C)nc2)=O)C(CNC(=O)CC2CN(C)C2)CC2COCC12 84131,c1(-c2ccc(C(C)=O)cc2)cc(=NC(=O)C(C)(C)CCCF)[nH][nH]1 84132,N1(C(COCc2n(C)c(S)nn2)=O)CC(CNC(=O)C(C)(C)C#N)CC12CCC2 84133,Cc1cccnc1CC(=O)N(C1CCN(C(c2ccc(Cl)cc2)C)CC1)C 84134,c1(C(=O)NCC(CC)NC(=O)CCCCCSC)c(C)cccc1O 84135,C1(C(N(CC(F)F)CCC)=O)COC(CNC(=O)Cc2cc[nH]n2)C1 84136,C1(CC(=O)NCC=Cc2cccnc2)CN(C(=O)C(F)CC2CCCC2)CCO1 84137,C(C(C)CC(=O)N(C(C)C(C)(C)O)C)NC(c1c(C)nco1)=O 84138,Cc1nc(CC(=O)NC2(CCCC(=O)N3CC(c4ncc[nH]4)C3)CCC2)cs1 84139,CC1CC(C)N(C(c2coc(C(F)F)n2)=O)CCN1C(=O)CCNC(=O)C(C)(C)C 84140,C(=O)(C#CC1CCCOC1)N1CC(NC(c2cc(F)cc(F)c2)=O)CC(OC)C1 84141,Cc1nc(CC(F)(F)F)sc1CC(=O)NCC1CCCCC1C.C12CCN(C1)C2=O 84142,C1(C)(C(N2CCC(NC(C)=O)CC2)=O)CC2CC2N1C(c1ccc(O)cc1C)=O 84143,C12(NC(C(C)=C3CC3)=O)CCCC1N(C(c1cnn3c1OCC3)=O)CCC2 84144,C12(NC(C(N)=O)=O)CC1CN(C(c1cnn(CCc3ccccc3)c1F)=O)C2 84145,C1(NC(CC(CCC)(C)O)=O)CCC2CCN(C(c3cc(C)nn3C)=O)C1C2 84146,C1(CCN)(OC)CCN(CC=Cc2cccnc2)C1 84147,CC(C)COCC(=O)NCC=CCNC1(CC(N)=O)CC1 84148,C1(CNC(COCCOC)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 84149,N1(C(CNCC)=O)Cc2cccn2CC(C(=O)NCCN(CC(C)O)C)C1 84150,CC1CC(CNC(=O)CCN2CCCC2=O)CN1C(c1cc(C(N)=O)co1)=O 84151,C1(CCCNC(=O)C(=O)NC(c2ccc(F)cc2F)CF)Cc2ccccc2C1 84152,C12(NC(c3cn(CCC)nn3)=O)CCCC1(F)CN(C(c1ccn(CC)n1)=O)C2 84153,CC1CC2(CC(C(=O)NOCC(=O)NCC(O)C3CC3)C2)C1 84154,N1(C(CCc2ccc(OC)c(OC)c2)=O)CCN(C(=O)CC(C)F)CC2(CC2)C1 84155,C1(NC(CC(C)(C)C#N)=O)CCCCCN(C(=O)C2=CCCC2(C)C)C1 84156,N1(C(C(CC)OCC)=O)CCN(C(=O)C=Cc2c(C)coc2C)C(CC)C1 84157,c1(NC(C(c2csc(Cl)c2)N(CC)CC2CCOC2)=O)ccc(F)cc1 84158,c1(C(C)NS(=O)(=O)CC2CCCCC2)cc(C(=O)O)ccc1F 84159,C(C(CNC(=O)C(C)Cc1ccnn1C)S(C)(=O)=O)NC(c1c(CC)nns1)=O 84160,C1(OCC)CCCCCN1N1CC(O)C(F)C1 84161,c1(N2CCCC(C)(CNC(C3CC(C)OC3)=O)C2)ccc([N+](=O)[O-])cc1C(N)=O 84162,Cc1nn(CC(=O)NC(C2(CNC(=O)COCCN(C)C)CC2)C)c(=O)n1C 84163,C1(C(=O)NCCC2CCC3CC23)CC2CCC(C1)N2C(=O)CC1CC(F)C1 84164,c1(CN2C3CN(C(C4N(C)CCC4)=O)C(C3)C2)ccc(F)c([N+](=O)[O-])c1 84165,C1(C)(CNC(C2C(C)(Br)C2)=O)CCN(C(C2CC23CC(O)C3)=O)C1 84166,C1(C(N(CCCN(C(Cc2cccc(SC)c2)=O)C)C)=O)CCCC(C)(C)C1 84167,c1(C(N2CC3C(NC(CCC(=O)NCC)=O)(CC3)C2)=O)c(F)cc(Br)cc1Br 84168,c1(CCC(=O)NC2C(CNC(C3CC4COCC4C3)=O)CC2)c(F)cccc1F 84169,C(CC(=O)NC1CCC(NC(=O)C=CSc2nc[nH]n2)C1)(C(F)(F)F)OC 84170,C1(C(N)=O)(NC(C2C(C(=O)OC)C2)=O)CCCN(c2ccc(C#N)cn2)C1 84171,C1(CC(C)C)(C(=O)N(C2CCC(n3cc(CO)nn3)CC2)C)CCNC1=O 84172,CC1(C)CCCC(CC(=O)NCC2(C)CCCC2NC(=O)Cn2cccnc2=O)C1 84173,N1(CC(=O)NCC(C)NC(CN(C(C)C(=O)N(C)C)C(C)=O)=O)CCNC(=O)C1 84174,C(=O)(CCCC(F)(F)F)N1CC(C)C(n2cc(C3CCn4ccnc4C3)nn2)C1 84175,C1(OC(CN(C(C)(C)C)C(N(C(CC)C)CC(C)C=O)=O)=O)CCC(C)(C)C1 84176,c1(C(=O)NC(c2ccc(F)cc2)CC)cc(C)c2sccc2c1 84177,N1(C(c2nc(N(C)C)oc2)=O)CCC(NC(=O)CNc2ccoc2)C(C)(C)C1 84178,C1(NC(C2CC=C(C)CC2)=O)CC2CC1CC2C(=O)N(CC(C)C#N)C(C)C 84179,c1(C(N2CCC(n3cncn3)C2)C(=O)NCC(=C)C)cc(F)ccc1Br 84180,C(Cc1ccoc1)(C(=O)NC1C2CCCC12)NC(=O)CO.CC(C=O)n1cncn1 84181,c1(CC)cc(C)cc(C)c1CN(c1ccc(C)c(C)c1)CC1CCCC1.N 84182,N1(C(c2c(C(C)C)ocn2)=O)CCC(NC(c2nncn2C)=O)C(C)C1 84183,c1(C(=O)Nc2ncc(C)nc2Cl)n[nH]c2c1CCN(C(c1ccc(O)cn1)=O)C2 84184,C=CCC(C)(O)C(=O)NC1CCCCN(C(C23CCC(C2)C3(C)C)=O)C1 84185,C1(NC(C(C)(C)F)=O)CCN(C(c2cccc(NS(C)(=O)=O)n2)=O)CC(O)C1 84186,C=CC1OCCCC1C(=O)N(C)CCOCCN(C)C(c1ccc(F)cc1N)=O 84187,C1(C(N2C(CCN(C)C)CCC2)=O)CCN(C(=O)CCN2CCOCC2)CCO1 84188,C1(CNC(c2ccc(O)nc2)=O)CN(C(C2(C(F)F)CCCC2)=O)CCCO1 84189,C(=O)(C1=CCS(=O)(=O)C1)N(C(CNC(C12OC(C)C(C1)C2)=O)C1CC1)C 84190,CCCC(C(=O)NCC(C)(C)C(=O)NCC1OCCC1C)N(C)C 84191,C(CN=C(NCC1(c2ccc(F)cc2)CC2CC2C1)N1CCC1)NS(C)(=O)=O 84192,c1(NC(=O)Nc2ccc(NC(N(C)CC)=O)cc2C)ncc([N+](=O)[O-])c(O)n1 84193,C#Cc1ccc(C(=O)NCC2C(C)CCCN2C(=O)CCCN2CCCC2)cn1 84194,N1(C(Cc2c(C)ocn2)=O)CCC(C)C(CNC(c2cc(C(C)C)no2)=O)C1 84195,C1(NC(C(COC)C)=O)CN(C(=O)COCc2nnc(C)s2)CCC12CCC2 84196,c1(C(=O)NCCC(C)N(C)C(C2(C)CCCCC2)=O)cc(Br)cn1C 84197,CCC(C)CC(=O)NC1(CCNC(=O)CNC(N2CCOCC2)=O)CCCC1 84198,C1(F)(C(N(CCCCC=C)C)=O)CCN(C(C2SCC=C2C)=O)CC1 84199,Cc1cc(-c2nc(C3CCCCC3)nn2-c2cccc(Br)c2)c(C)[nH]1 84200,C(=O)(C1SCCc2sccc21)NCCN1CCN(C(C(CC)SC)=O)CC1 84201,C1(N(C(=O)COC2CCOC2)CC)CCN(C(=O)CCc2nnc(S)n2C)CC1 84202,C1(C2CCN(C(=O)CC3CC4(CC4)CO3)CC2)(NC(=O)C(=O)N(CC)CC)CC1 84203,N12CC3(CCCC3)C1C2=O.C1(NC(=O)OC(C)(C)C)C2CCC(C2)C1CO 84204,Cc1c(N(C(C(=O)NCCC2CCCC2)C)C)ncnc1Cl.CC 84205,N1(C(C(C)NC(=O)C2CC2)=O)CC2(C)CC1(C(N1CC(O)C(F)C1)=O)C2 84206,c1(C(N2CCC(CN(C(=O)Cc3cccc(O)c3)C)C2)=O)cnc(O)cc1O 84207,c1(-c2cn(CC(C)(C)CNC(=O)CN3CCCS3(=O)=O)nn2)cc(Cl)cc(Cl)c1N 84208,c1(C(=O)NCC2(O)CN(C(C3CCC4CC34)=O)C2)c(F)cccc1[N+](=O)[O-] 84209,C1(C(=O)NC(C(C)NC(c2n[nH]cc2Cl)=O)(C)C)CCCN(CC(F)F)C1 84210,C1(CC)C(NC(=O)CSCc2ccccc2)CCN1C(c1ccc(SC)nc1)=O 84211,CC1CN(C(c2ccoc2)=O)CC2(CCN(C(c3cccc(N)c3O)=O)CC2)O1 84212,C1(NC(CSCCOC)=O)CC(O)CN(C(c2ccc(Cl)nc2Cl)=O)C1 84213,C(=O)(C(CO)C(F)(F)F)N1CCC(=C)CC1C(=O)N(C)Cc1c(C)cnn1C 84214,c1(C(=O)OCC)nc(NC(C2CCN(CC3CCC3)C2)=O)[nH]c(=N)n1 84215,Cc1cc(C(=O)N(C2CCCN(C(C3CC(C)C3)=O)C2)CCO)cnc1O 84216,CN1C2CCC1CC(CN1CCC1C(N1CC3(CCOCC3)C1)=O)C2 84217,c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C#N)(NC(c2ccsc2)=O)C1)=O 84218,S(=O)(=O)(c1cn(C)nc1C)N1C(NCc2c(C)ccc(Cl)c2)C(O)CC1 84219,C(=O)(C(C)(C)C1CCN(C(=O)CC2CC2(C)C)C1)NC(C)Cc1cn[nH]c1 84220,CC(CN(C)C)CCC(=O)NCC(N1CC=CC1)=O.C12C=CC(C1)NC2=O 84221,c1(C(N2CCN(CC#CC)CC2)C(=O)NCCC2(C)CC2)nc(Cl)cc(C)c1Br 84222,c1(C(N2CCC(c3cccc(C(=O)NC(C)(C)C)c3)C2)=O)cc(Cl)cc(Br)c1F 84223,C(=O)(CC1OCCc2ccccc21)N1C(CNC(C2(C)CC=CC2)=O)COCC1 84224,C(N=c1nc(NCCCS(C)=O)c2c([nH]1)CCC2)c1cc2cccc(OC)c2o1 84225,c1(C(C)C)cc(C(=O)NC2CCC2NC(c2cncn2C)=O)ccn1 84226,CCC(C)CCCCC(=O)NS(=O)(=O)c1cn(C)nc1C(F)(F)F 84227,c1(Nc2nccc(SC)n2)ccc2nccnc2c1Cl 84228,c1(C(C)NC(=O)C(=O)NCCc2cnn(C)c2)ccc(C(C)(F)F)cc1 84229,C1(C(N2C(CNC(c3n(C=C)ncc3)=O)CCC2)=O)CCc2nnc(O)cc2C1 84230,CC1(CCNC(C2CCCC(=O)O2)=O)CCN(C(C2(n3nccn3)CC2)=O)C1 84231,c1(C(=O)NCC(CC)NC(c2c(COC)n(C)nc2)=O)cnc(N(C)C)nc1C 84232,C1(C(=O)NC(C=C)COC)N(C(=O)C(CC)SC)CCC1(C)C 84233,Cc1ccc(F)cc1NC(=O)CN(C1CCCO1)CCN1CCCOCC1 84234,C(=O)(C1=NOC(C)(C)C1)N(C)CC1CCCN(C(c2c(C)ncc(C)c2)=O)C1 84235,C1(NC(C(C)(C)NC(c2cn(C)nc2)=O)=O)CC12CC(O)C2 84236,C(=O)(CCCC=C)NCC(CC=C)NC(c1cn(C(F)(F)CO)nn1)=O 84237,C#CCC(C)(C)C(=O)Nc1cccc(F)c1.C12CCCN(C1)Cc1cn(nn1)C2C 84238,N1(C(c2ccc(CSCCOC)o2)=O)CCCC(C)C1CO.c1(C(=O)N)cncs1 84239,NS(=O)(=O)N1CC(C(=O)NCC(C2(O)CCN(C(C3CCCCC3)=O)C2)(C)C)C1 84240,N1(C(CCN(CCC)C)=O)CC(c2ccccc2)(NC(c2occc2Cl)=O)C1 84241,C1(NC(CSCCC(C)C)=O)CCN(C(C2COC(C)(C)CO2)=O)CC12CCC2 84242,c1(CO)c(Br)cc(F)c(F)c1F.Cc1ccc(CN2C3(CCC2)C(=O)O3)c(Br)n1 84243,c1(C(C)NC(C2(CCNC(C34CCC(C3)C4)=O)CC2)=O)ccn(C)c1 84244,c1(NC(c2ccc(N3C(C)CCC3)cc2)C(F)(F)F)cc2cc(Br)ccc2s1 84245,C(=O)(CCCCC(=O)NC1CN(C(c2nnc(O)nc2O)=O)CC2(CC2)C1)NC 84246,C1(Cc2ccccc2)CCOC1(C)C.C(=O)(CCCC1CCC1)N1CC(C(C)N)C1 84247,C(C(C)(C(=O)NC1CCC1NC(C1(CCc2ccccc2)CC1)=O)OC)OC 84248,n1(CC)nc(C)c(C(N2CC3CC2C3CNC(C23CCOC(C)(C2)C3)=O)=O)c1Cl 84249,N1(CCC2(C)CCN(C(Cn3c(C)cc(C(F)F)n3)=O)C2)CCC(O)C(C)C1 84250,Cc1cc(C(=O)NC2(C)CC(NC(C3CC(=O)NC(C)C3)=O)C2)cc(C)n1 84251,COn1cnc(C)c1C(N1CC(NC(c2c[nH]c(=O)cn2)=O)C(F)C1)=O 84252,N1(C(CC2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCCC1 84253,CC1OC(C)(C)CC1C(=O)N(C)CCOCCNC(=O)C(C)C1CCCC1 84254,C1(CNC(CC(C)F)=O)CN(C(c2ccc(NC3CC3)cc2)=O)CCC12CCC2 84255,c1(N2CC(C(=O)NCC34CCCN3CCC4)SCC2)ncnc2[nH]c(Br)cc12 84256,N1(C(C(C2CCOCC2)C)=O)CC(NC(C2(O)COC2)=O)CC2(CCC2)C1 84257,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84258,C1(NC(c2ccc(SC)s2)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C2CC2)C1 84259,c1(C(C)C(C)C)ccc(C(=O)NC2CCN(C(c3cc(F)c[nH]3)=O)C2)cc1 84260,C1(C(N(C(c2cc(C)on2)C)C)=O)CCN(C(C2C3CN(C)CC23)=O)CC1(C)C 84261,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(CCCOC)CC1 84262,N1(C(C)(C)C)CCC(NC(=O)CCC2CC(NC(c3ccc(C(F)F)o3)=O)C2)C1 84263,c1(CC(=O)NCC(C)(O)CNC(=O)COCCOC2CCCC2)cccnc1Cl 84264,C1(CCNC(=O)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCS(=O)(=O)C1 84265,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(SC)cnn2C)=O)CC1 84266,C(=O)(C(F)CC(CC)CC)NCC(=C)CCNC(C1(C2CCCO2)CCOCC1)=O 84267,CC1(C(N2CCCC(c3cccs3)C2)=O)CCCN(C(=O)Nc2ccc(Cl)cc2)C1 84268,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(C)C)Cc2ccccc2C(C)(C)C1 84269,CC1CSCC1(c1ccc(Br)cc1)NC(=O)NC1CCC(N(C)C)CC1 84270,c1(CCC(=O)NCC#CCNC(C2OCCN(C)C2)=O)ccc(F)cc1F 84271,C1(NC(C(c2cnn(C)c2)NC(C2C(CC)CCO2)=O)=O)CCOC2(CCC2)C1 84272,Cc1cc(C)c(C(N2CC(c3ccccc3)C(Cl)C2)=O)[nH]1 84273,C(=O)(NN(CC(=O)OC)C1CCc2ccccc21)NC1CCC(CC)C1 84274,C1(N(CCC(=O)NC(=O)CNC2CCCC2)C(=O)NC)CCOCC1C1CC1 84275,CC1CN2CCN1C(C(=O)NC1CC1CNC(=O)C(C)(C)C)C2 84276,C1(CC(=O)NCc2c(C)nc(CC)o2)CN(C(c2n[nH]c(C)c2Cl)=O)CC1(C)C 84277,C(C(C)(O)CC(=O)NC1CCOCC1C(=O)NCCc1cn(C)nc1C)OC 84278,N1(CC(CC)CC(C)(C)C)CC(C(=O)OC)C2(CN(C(=O)OC(C)(C)C)C2)C1.OC 84279,N1(S(C)(=O)=O)CCN(C(C2CC2(F)C(=O)N(CCF)C2CC2)=O)CC1 84280,C1(NC(CNC(CCC)=O)=O)CC(C)(C(=O)OC)C1 84281,c1(N2CC(CN(C(C(COC)(C)O)=O)C)OCC2)cc(=O)n(C)c(O)n1 84282,C1(C(N2CC(CNC(C(CC)n3ccnc3)=O)OCC2)=O)CC(C)(C)C(C)(C)C1 84283,C1(NC(=O)C(C2CCCCC2)O)CCCC1OCc1cccnc1 84284,FC1CC2CC1CC2NCc1cccc(C2CC2)c1 84285,N1(C(c2cncc(Cl)c2Cl)=O)CC2CCCC(C1)N2C(C1CCCCC1(F)F)=O 84286,c1(C(=O)NC(C)CCNC(c2cc(Br)co2)=O)n[nH]cc1[N+](=O)[O-] 84287,c1(C(=O)OC)sc(-c2ccc(NC(=O)NC3CCCCC3)cc2)nc1C 84288,Cn1cc(C(=O)NC2C3CC2N(C(=O)Cc2ccc(C#N)nc2)C3)ccc1=O 84289,C#CCCCCCC(=O)N1CCCC(CC)(NC(c2cccnc2)=O)C1 84290,N1(CC(=O)N(CC(C)CNC(=O)CCN(C)C)C)CCCCC1 84291,c1(C2OCCN(C(c3nnc(C(=O)OC)s3)C(=O)NCC)C2)ccc(F)c(F)c1 84292,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(OC2CCN(C(=O)C(C)(C)C)C2)CC1 84293,c1(C(N2CCC(NC(C=C(CC)CC)=O)C23CC3)=O)cccc2c1NCCC2 84294,c1(C(N(C)Cc2cccc(CC)c2)=O)ccnc2ncc(C)cc12 84295,N1(C(c2c(Br)n[nH]c2Br)=O)CCC2(CCCN2C(c2ccoc2)=O)C1 84296,C1(F)(CNC(c2ccon2)=O)COCCN(C(c2ccc(Br)cn2)=O)C1 84297,C1(CCC)CC(C(=O)NCC(C)(O)CNC(=O)CN(C2CCC2)C)CCO1 84298,c1(C(=O)NC(c2cccc(OC(F)(F)F)c2)C)cc2cc(Br)ccc2[nH]1 84299,N1(C(C(CC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CCN(C)C1C 84300,CC(=O)CCCC(=O)N1CC(CNC(=O)CCC(C)(C)F)CCC1C 84301,C1(NC(c2cc(C(=O)OC)sc2)=O)CS(=O)(=O)CC1NC(c1c(Cl)cnn1C)=O 84302,c1(CNCC2N(C(c3c(OC)cncc3)=O)CCOC2)cc(F)ccc1Br 84303,N1(C(C)C)CCN(C(C(=O)NCC(C)C)C(C2CC2)C2CC2)CC1 84304,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3COC(=O)C3)C2)C1 84305,C1(CNC(C=CCOC)=O)CCN(C(c2cc(OC)cc(C)n2)=O)CC1C 84306,C(=O)(C1CC(=O)c2c(F)cccc21)NC(CNC(Cc1c(C)cccc1Cl)=O)C 84307,c1(OC(CCNC(c2n(CCCSCC)nnn2)C2CC2)=O)c(OC)cccc1Br 84308,C1(NC(C2(C)C(C)(C)C2(C)C)=O)CC(N=c2ccn3nccc3[nH]2)C1(C)C 84309,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC2(C)CN(C(=O)CC(C)SC)CC2(C)C1 84310,N1(COc2c(OC)cccc2)CC2CN(C(c3c(F)ccc(F)c3C)=O)CC2C1 84311,c1(C(N(CCN(C(=O)CN(C)C2CC2)C)C)=O)cc(Cl)cc2c1NCCC2 84312,C(C(=O)NC1CCC(NC(=O)C2=CCSC2)CC1)(C(C)C)OCC 84313,c1(C(N2CC(C)OCC2)=O)ccc(O)c(-c2ccc(Cl)cc2)c1 84314,C1(NC(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CC2CCOC2)C12CCC2 84315,C(=O)(C(CNC(=O)C(C)(C)O)C(C)C)NCC(=O)OCC(C)C 84316,CN1CCn2ncc(C(=O)NC3(C)CCCN(C(=O)CC4CC5CC5C4)C3)c21 84317,N1(C(c2ccc(N)cc2F)=O)CCC2(NC(=O)C(F)CC3CC3)CCCCCC12 84318,C1(C(=O)NC2C=CCN(C(CCc3scc(C)n3)=O)C2)CCc2cnnn2C1 84319,Cc1ccc(C(N2CCC(CCF)CC2)C(=O)NCC(F)F)c(O)c1 84320,CC1CC=C(C(=O)NC2CCN(C(=O)Cc3cccc(Cl)c3F)C23CC3)CC1 84321,c1(SCC2CN(C(=O)C(N3CCCC3)C3CC3C(F)(F)F)C2)ccccc1 84322,CN1CCCC(F)(C(=O)NC(CNC(c2cncc(C(F)(F)F)n2)=O)CO)C1 84323,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84324,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84325,O=C(C1=CSCCO1)NCC(Cc1ccccc1)NC(=O)CC1CCCO1 84326,N1(C(c2c(CC)cco2)=O)CC(NC(c2ccc(Cl)[nH]2)=O)C2(CCOCC2)C1 84327,N1(C(CCC=C)=O)CCCC(C(C2CCCN(C(=O)C(C)C(F)F)C2)(C)C)C1 84328,c1(-c2cnc(C)s2)ncccc1NC(c1cncc(C(F)(F)F)c1)=O 84329,c1(NC(c2ccc(OC)cc2)C2CC2)cccc(OC(C)=O)c1C 84330,CC1=C(C(=O)NCc2ccnc(OC(F)F)c2)SCCO1.C12CC(C1)C(=O)N2 84331,C1(CNC(C(C(C)C)N2CCCS2(=O)=O)=O)CN(C)CCN1C(c1cnco1)=O 84332,c1(C(c2nccc(=N)[nH]2)NCc2c(OC(C)C)cccc2)cc(Cl)ccc1[N+](=O)[O-] 84333,C(CC(C)(C)C(CCC=C)Oc1cc(C)ncn1)(C(=O)OC)OCc1ccccc1 84334,c1(C(N2CC(C(C)NC(=O)CC3(C#N)CC3)C2)=O)cccc(C2CCOCC2)c1 84335,c1(C(N(CCCOCCNC(CC(C=C)C)=O)C)=O)c(F)ccc2n[nH]cc12 84336,C1(C(C)C)CN(C(C2CC(=O)C2C)=O)CCN1C(C1CS(=O)(=O)C1)=O 84337,C(=O)(C(C)(C)C(=O)N1CCC(C(C)NC(=O)C(C)C2CCCO2)CC1)OCC 84338,c1(C(N(CC=CC(N2C(C(C)O)COCC2)=O)C)=O)coc2ccccc12 84339,c1(C(=O)NCC(CC)NC(=O)C(C)(F)CC)cnc2c(ccn2C)c1 84340,N1(CCC(N2CCC(NC(C3CCC(C#C)CC3)=O)C2)=O)Cc2ccccc2C1 84341,c1(C(=O)NCC2CC(NC(CCCCC)=O)C2)ccc2c(c1)CC(OCC)C2 84342,N1(C(C2CC(=C)C2)=O)CCC2(CCC2NC(c2ccc(F)c(CO)c2)=O)CC1 84343,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(Cl)c2)C(C)C)CCC1 84344,C1(NC(Cc2c(C)noc2)=O)CCCC(NC(=O)C(C)C=Cc2ccccc2)C1 84345,C1(C)(C(=O)NC2CCC(C(=O)NC(CCC)c3ccco3)C2)CCC(=O)N1 84346,C1(C(=O)NCC#N)CC2CC2N1C(C1(F)CC1)=O 84347,c1(CN(C(C(C)OC)C)C(=O)CC2CC2)ccnn1C 84348,c1(NC(C23CC(C(=O)Nc4ncnc5sccc45)(C2)C3)=O)ccc2cc[nH]c2c1 84349,c1(C(=O)NCCCN(C(c2cc(C)nnc2)=O)C)ccc2[nH]c(=O)c(=O)[nH]c2c1 84350,c1(C(N(CCC)CCNC(C23CCC(F)C2CC3)=O)=O)nc(O)nc(O)c1F 84351,C1(C)(NC(CN2CC(C)CC(C)C2)=O)CCCN(C(=O)C(N)=O)CC1 84352,C(N=c1[nH]cncc1I)C1(NC(C(C(CC)C)O)=O)CCC1 84353,Cc1ccc(C)c(C(N2CC(N3CCN(C(C4CC4C#N)=O)CC3)C2)=O)c1C 84354,N1(C(C2CCC(=O)N2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84355,Cc1cc(C(=O)NC2COCC2NC(=O)C#CC(C)C)c(C)c(O)c1 84356,C1(NC(CC=C)=O)CN(C(C2CCN(CCF)CC2)=O)CC12CCC2 84357,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84358,c1(CC)cnccc1C(=O)N(C1CCCN(C(=O)C(N2CCOCC2)C)C1)CC 84359,CC1CC(NC(=O)Cc2cc(F)cc(Cl)c2)CCN1C(c1cnc(Cl)n1C)=O 84360,c1(C(=O)NCCC(CCNC(c2c(C)nc(COC)s2)=O)C)cc2c[nH]nc2s1 84361,C1(C(=O)NC(CC)CCC(=O)NCCOCC(F)F)C2CCC3C(C2)CC13 84362,c1(C(=O)NCC(C(C)C)NC(CC(CCSC)O)=O)cnc2sccc2c1 84363,C12(COC)CCCC1(C(=O)NC1C3CC1N(C(=O)OC(C)(C)C)C3)OCC2 84364,C1(CC(N2CC(=C(F)CNC(C3(O)CCC3)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 84365,CCC(C)C(C(=O)NC1CCN(C(C)C)C1=O)NC(c1ccsc1OC)=O 84366,C1(NC(CCC=CC)=O)CN(C(C2(F)CCCC2)=O)CCC1CO 84367,N1(C(=O)Nc2c(-c3n(C)c(Cl)cn3)cccc2)CC(S(N)(=O)=O)C1 84368,N1(CC)CC2(CCN(C(=O)CCc3nc(C)no3)C2)C1.C12C(CC1O)NC(=O)C2 84369,C1(CC)CN(CC(CC)CC)CCC1(F)F.[nH]1cc(C(C)C2CC2)nn1 84370,Cc1cn2c(n1)CC(C(=O)NC1CCN(C(=O)COCCO)CC1C(C)C)CC2 84371,c1(NC(C2NCCN(C(c3c(C)nc(C)s3)=O)C2)=O)cc2c[nH]nc2cc1Cl 84372,C1(NC(c2cc(OCC)no2)=O)CN(C(c2nnn(C)c2CC)=O)C(C)(CC)C1 84373,N(C1CCCc2ccc(C(C)(C)C)cc21)Cc1n(C(C)C)nc(-c2cccs2)n1 84374,c1(CN2CCC(=CCC)C2)ccc(-n2cncn2)c(F)c1 84375,CCCC(C(=O)NCCC(C)N(C)C)NC(=O)Cn1cnnc1O 84376,c1(N(C(=O)CCCc2cccs2)CCCc2nn[nH]n2)cc(Cl)cc(Cl)c1 84377,n1(CCC)cccc1NC(=O)NCc1ccn(CCF)n1 84378,C=CCC(C)(CC)C(=O)N1CCCC1CC(N1CCC(N(C)C)C(C)C1)=O 84379,C1(N(C(C(N2CCCCC2)C)=O)CCO)CC12CCNCC2.c12ccccc1C2 84380,C1(S(C)(=O)=O)(C(=O)NCC2C(NC(C(CC)(C)OC)=O)CCC2)CCOCC1 84381,c1(C(N(C)CC2CCN(c3nnc(C(N)=O)s3)C2)=O)cc(Br)cc2ccccc12 84382,N1(C(c2cncc(C)c2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1CC1CC1 84383,N1(C(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(C2(F)CCOC2)=O)CC1 84384,C(=O)(C1=CCCC1C)NCCN(CCCCCC)C(c1ccc(F)cc1C)=O 84385,C1(OCCC(N2CC(CC(C)NC(C=C(CC)CC)=O)C2)=O)CCOCC1 84386,c1(C(=O)NCC2CCN(C(CSCC=C)=O)C2(C)C)ccc2c(C)noc2c1 84387,N1(NCCCCN(CCN(C)C)CCN)CC(C)(C)OC1=O 84388,C=CCCCCCNC(c1ccccc1Cn1cc(CCC(=O)CC)nn1)=O 84389,c1(CN(C(=O)Nc2c(C(C)C)cc(F)cc2)C(C)C)ccc2c(c1)OCCCO2 84390,C1(NC(C(CC)C)=O)(CF)CCN(C(c2ccc(NC(C)=O)cn2)=O)C1.CC(F)F 84391,C1(C(=O)OC)CCCCCN1C(=O)CN1CCCNS1(=O)=O 84392,NC(=O)C(F)(F)CCNC(=O)C(C1CC1)NC(=O)CCN1CCCC1=O 84393,CCC(CNC(=O)Cc1ccccc1F)(CC)NC(=O)C(C1CCOC1)OC 84394,c1(N(C)CC2CCCO2)nc(=NCCCCCO)[nH]c2c1SCC2 84395,C(C(CC(F)(F)F)NC(C1(c2ccno2)CCC1)=O)NC(=O)Cc1cn[nH]c1 84396,C(C)(CC(=O)NOCC(O)C(C)C)N(C(C1C(C)C1)=O)C 84397,c1(C(N2C3C(CNC(c4cc(OC)n[nH]4)=O)C(C3)C2)=O)cc2n(n1)C(C)CCC2 84398,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(=C)CC2CC)=O)C(CC)CCC1 84399,C1(OC)CN(C(c2ccc(O)c(F)c2)=O)C(C)(CNC(=O)C=CC(C)C)C1 84400,C(CC(=O)N=c1ccn(C)[nH]1)C1(NC(C(C)Cc2ccc(F)cc2F)=O)CCCC1 84401,c1(OC)cnc(F)c(C(=O)NCC2CCN(C(=O)CN3CSCC3=O)C2)c1 84402,N1(C(C2N(CC)CC2)=O)CCOC2(CCN(c3nc(O)c4ccccc4n3)C2)C1 84403,N1(C(C2C(C)C2)=O)CCC(C2CCN(CCCc3ccc(Br)cc3)CC2)CC1 84404,c1(C(=O)NCC2C(C)CN(C(c3csnn3)=O)CC2)cc2c(F)ccc(Cl)c2[nH]1 84405,C1(CN(C(=O)NCC(c2nccs2)C)C2CC2)C(C)(C)C1(F)F 84406,c1(C(=O)NCCCN(C(C2(COC)CCCC2)=O)C)c(Cl)cccc1[N+](=O)[O-] 84407,c1(C(N2CCC(NC(C(C)=CC)=O)C(F)C2)=O)ccc([N+](=O)[O-])c(C)n1 84408,c1(C(=O)NCC(CC)NC(c2nc(OCC)oc2)=O)cnc(O)cc1C 84409,N1(C(CN(C(C2C(C(N)=O)CC2)=O)CC2CC2)=O)CCSC2CCC12 84410,CCCCC(C(=O)NCCc1[nH]cnc1C)NC(=O)C=Cc1ccc(C)cc1 84411,C(CC(C)(C)C(=O)NCC1(CNC(c2ccc(Cl)nc2N)=O)CC1(F)F)OC 84412,c1(CC)cnc(C(C)NCc2ncc(-c3ccccn3)s2)o1 84413,C1(C(=O)NC2CCC(NC(c3cccc(Cl)c3Cl)=O)CC2)CCC2CC1CO2 84414,N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCC(C2CCCN2C(C2CCC(=O)C2)=O)CC1 84415,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84416,C1(C(=O)NC(c2nnc(O)o2)C)CNC(=O)CN1C(=O)C=CCN1CCC1 84417,Cc1cc(NCC(C)NC(N2CCCCC2c2ccc(CO)cn2)=O)cc(C)c1 84418,C1(C)(OC(C)=O)CCC(C(=O)N(C)C)O1.C1C(=O)O1 84419,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cn(C)cn3)=O)CC12 84420,C1(C(=O)NC(C2(O)CN(C(=O)CCCn3cccn3)C2)C)CCc2cnn(C)c2C1 84421,Cc1cc([N+](=O)[O-])cc(C(=O)NCC2CCN(C(=O)C#CC3CC3)C2)c1Cl 84422,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)CC3CCSC3)C(C)C2)=O)c1 84423,c1(OC)cccc(CC(=O)NCC2CC(O)CC(CN)C2)c1Cl 84424,C1(CCC(=O)N(C2CN(CCC(C)C)C2)CCNC(C(C)O)=O)CCCC(=O)N1 84425,n1(C(C)C)cc(C(=O)NCCOCCCNC(C2CCCS2)=O)cn1 84426,C1(OCC)CCN(S(C)(=O)=NC(=O)c2cnn3cccc3c2)C1 84427,C1(C#N)(C(=O)NC2C(C(N(C)CC3CCCCC3)=O)CCC2)CCCCC1 84428,c1(C(N2CC(OCCNC(CC3CC(=C)C3)=O)C2)=O)nn(C)nc1C(N)=O 84429,CCC(CC(=O)Nc1cccc(O)c1)NC(C1(C(=O)OCC)CC1)=O 84430,Cn1nc(O)cc1C(N1CC(NC(=O)C(F)=CC2CC2)CC1CO)=O 84431,C1(NC(C(C(C)(C)C)=O)=O)CC(N=c2[nH]c(Cl)ncc2F)C12CCC2 84432,C(CSC)(C(=O)NCC=C(C)C)NC(CN(CCC)C)=O 84433,N1(C(C(=O)NCC2CCCCC2Nc2cccc(F)c2)=O)CCSCC(F)(F)C1 84434,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2ccc(OC(C)C)cn2)=O)CC1C 84435,N1(C(CCNC(C)=O)=O)C(C(=O)NCc2ccco2)C2CC(O)C1C2 84436,C(CCC)(CCCNC(=O)C(C)=C1CC1)NC(C(CC=C)NC(C)=O)=O 84437,c1(N(CCC)CCNC(=O)CCC(C)C)cccc(F)c1C#N 84438,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 84439,c1(C(=O)NCCC2N(C(C(C)NC(C)=O)=O)CCSC2)c(C)[nH]c2ccc(O)cc12 84440,N1(C(C)C)CCOC(C(=O)NCCN2CCC(NC(C3CCC3)=O)CC2)C1 84441,c1(C(N(C)CC2OCCN(C(C(CC)CC)=O)C2)=O)cc(C(=O)OC)ccc1F 84442,n1(CC)c(N2CCC=C(F)C2)nnc1Cc1cccnc1 84443,c1(C(=O)OCc2c(C(=O)OCC)oc(Br)c2)cn2ccccc2n1 84444,N1(C(C(C)OCCCC)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 84445,N1(C(C(C)c2cc[nH]n2)=O)CC2CCC(NC(=O)C3=CCN(C)C3)(C2)C1 84446,C1(CC(=O)OC)COCCN(C(C2CCN(S(=O)(=O)CC(C)C)CC2)=O)C1 84447,C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)CC1 84448,c1(CC)nc(C(=O)NCC2C(CNC(=O)CC(C)OC)C2(F)F)cs1 84449,C1(C(=O)OC(C)(C)C)CCN(C(=O)NC23CCCN(CC2)C3)C2(CC2)C1 84450,C1(CN(C(C(N2CCC(NCCOC)C2)=O)C2CC2(Cl)Cl)C)CCN(C)CC1 84451,N12CCCC1(C)C(=O)OCC2=O.c1(NC)ccccc1Cl.c1(C=O)cnsn1 84452,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 84453,N1(C(C2(C#C)CC2)=O)CCC(C2CCN(C(c3ccnc(SCC)c3)=O)CC2)C1 84454,c1(NC(=O)NC(CCNC(C)=O)C(C)C)c(C)nn2cc(N(C)C)cnc12 84455,C(=O)(C(C)C(O)C(C)C)NC(CN(C(c1n(CCC)ncc1)=O)C)(CO)CO 84456,C(=O)(CCC(=O)c1cc(Cl)sc1Cl)NC(CN(C(C)C)C)C 84457,C1(CC(=O)NC2CCC(NC(C3(C)CCCOC3)=O)CC2)CCC(=O)NC1=O 84458,N1(C(c2c(C)c(CO)ccc2)=O)CC(CNC(C2(C(C)C)CC2)=O)CC(C)(C)C1 84459,c1(-c2nc(CCCCCC)nn2CCCNC(C2CCOC2)=O)ccc(Cl)c(Cl)c1 84460,C=CCC(CNC(c1cnco1)=O)NC(=O)C(C)CN1CCOCC1 84461,N1(C(c2c(CC)scc2)=O)CC(C)(C)OCC1CNC(=O)C(c1ccc(C)o1)C 84462,C=CC(CCC)CC(=O)NCC(C1CC1)NC(C1(c2cccs2)CCCCC1)=O 84463,c1(NCCC(C)OC)nc(N2CCCOCC2)c2c(n1)c(C)nn2C 84464,C1(C(=O)NCC(CC)N(C)C(C2(C)CCCOC2)=O)CCC12CCC2 84465,N1(C(C2N(C)CCCC2)=O)CC2(CNC(=O)C(C)(C)c3ccccn3)CC1CO2 84466,N1(C(COCC)=O)CCCC(n2cc(CNC(=O)C(=Cc3cscn3)F)nn2)C1 84467,C1(CNC(c2cc(CNC(C3CCCN(C)C3)=O)ncc2)=O)CCCS(=O)(=O)C1 84468,N1(C(c2csc(C)c2N)=O)CCC(NC(=O)CCC2CC2(F)F)CC(O)C1 84469,C1(C(=O)NCC2CC(N(C)C(c3c[nH]nc3C(F)F)=O)C2)COCCN1C1CC1 84470,c1(C(N(C)CCN(C)C(c2cnc(C3CCOC3)s2)=O)=O)csc2nnsc12 84471,CCC(C(=O)NCC1CC(CNC(c2cnsn2)=O)C1)c1ccccc1 84472,Cc1sc(N)c(C(=O)NCC2CCCC2NC(c2cnn(C)c2C(F)F)=O)c1C 84473,N1(C(=O)NC2CN(CC)C2)CC2(CCCNC(=O)C2)C1 84474,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ccoc2)=O)C2COCC12 84475,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 84476,Cc1n[nH]cc1CNC(=O)C=CCC1(NC(=O)CCn2ccnc2)CCC1 84477,C12(CNC(Cc3cc(C)sc3)=O)CC1CN(C(C13CCCC1(C(N)=O)C3)=O)C2 84478,c1(OC)ccccc1CN(C(c1csc(-c2cccs2)c1)C(=O)NCC(C)C)C 84479,N1(C(c2cc(C)n(CC#C)c2C)=O)CCC(N(C(=O)CCSC)C)C2(CC2)C1 84480,c1(C(N(C(CNC(CC(=C)C)=O)C2CC2)C)=O)cc2cc(N)ccc2[nH]1 84481,c1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)Cl)ccc2occc2c1 84482,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C23CCC3)c1 84483,N1(C(=O)NC(C)(C)Cn2nccc2-c2ccccc2)CCCC(O)C1 84484,CC1(C)NC(=O)N(CCC(=O)NC2CCN(C(c3ccco3)=O)CC2C2CC2)C1=O 84485,S(=O)(=O)(c1cc(NC)ccc1OC(F)F)N1CC2C(C(=O)OC)C(COC2)C1 84486,c1(CCC)cccc(C(N2CC3(NC(c4cc(C5CC5)ccn4)=O)CC2C3)=O)c1 84487,N1(C(C23CCC(OC)C2C3)=O)C2CC=C(C(=O)NC(C)C(=O)OCF)C1CC2 84488,C1(NC(C(n2ccc(C)n2)C)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 84489,C(N=c1cc(C)nc(N2CC(C3CC3)OC(C)C2)[nH]1)C1(OCCOC)CCC1 84490,c1(C(N2CCN(C(=O)OCC)CC2)C(=O)NCCCF)ccc(F)c(F)c1 84491,N1(C(C2(C=C)CC2)=O)CCN(C(c2nn(C)c3c2CSCC3)=O)C2CCCCC2C1 84492,CCN=C(NCC1CCCC1OC(C)C)NCCC1CCN(C(C)=O)CC1 84493,C1(NC(CC(C)CF)=O)CCC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 84494,C1(NC(C2(C(=O)NC)CC2)=O)CN(C(c2ncc(Br)cn2)=O)CC1C 84495,c1(NCC(CC)O)cc(Br)ccc1OC(F)F 84496,C1(CCC)C(=O)NCCN1C(C1CCCN1CCC(C)C)=O 84497,CCCC(C)C(=O)NC1CCCC1CNC(c1sc(=N)[nH]c1C1CC1)=O 84498,c1(N2CCC(NC(C(C#N)=CC(C)C)=O)C(C)C2)ncnc2c(F)c(F)ccc12 84499,C1(NC(c2c(Br)cn(C)n2)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 84500,C1(CC)C(C(N(CCC2CC2)C(C)C)=O)CCN1C(c1cnc(OC)s1)=O 84501,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)CCN(C)CC2 84502,C=CC1OCCCC1C(=O)NCC1CN(C(=O)CSCC(N)=O)CCC1C 84503,C(C(C(=O)NCC1(O)CC(NC(=O)CCCc2ccc(C)s2)C1)OC)OC 84504,C(C(C)C(=O)NC(CN(C)CCN(CCCN(C)C)C)C(=O)SC)N 84505,Cn1ncc(C(N2CC=C(C(=O)NC3CCCN(C4CC4)C3)C2)=O)c1C#N 84506,C1(CC(=O)N(C2CCCN(S(=O)(=O)C(F)(F)F)C2)CCC)CCC(F)(F)CC1 84507,N1(C(C(C)N(C)CC)=O)CC2CCC1(C(=O)OC(C)(C)C)CC2 84508,Cc1c(O)nnc(C(=O)NCCCc2ncc(-c3ccc(Cl)cc3)[nH]2)c1C 84509,N1(C(c2cc(C(CC)CC)no2)=O)CCN(C(c2nn(C)cc2Cl)=O)C2CC12 84510,c1(CN(CCSC)C)ccc(F)cc1F.C12(C3C(=O)N3)CCN(CC1)CC2 84511,C1(C(N(CC#C)CC)=O)CC2CC1CN(C(C1CCC(=O)CC1)=O)C2 84512,c1(C(=O)NCC2CC(NC(=O)CCN3CCCCC3)C2)cc2ccccc2[nH]1 84513,N1(C(C2CCN(C)C2)=O)CCCCC1CCCNC(C1CCC(C(F)F)CC1)=O 84514,N1(C(COCCCC)=O)CC2CN(C(=O)C(c3ccccc3F)(C)F)CC2(C)C1 84515,c1(C(N2CC(NC(c3n(CC)ccn3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cc1C 84516,N1(C(C(CC)(C)CC)=O)CCC2(NC(c3ccnc4ccsc34)=O)CCCC12 84517,C1(NC(C=CCCC)=O)CC2CN(C(=O)C(Cc3ccccc3Br)OC)CC2C1 84518,C(=O)(C#CC1CCCCC1)NC1C(NC(=O)Cn2cnnn2)CCCC1 84519,N1(C(C(CSC)(C)NC(c2c(C)nsc2C)=O)=O)CCCC(C2(C)CC2)C1 84520,c1(NCC=CCSC(C)C)ccc(C(=O)NC23CC(C)C2C3)cc1.c1ccccn1 84521,c1(NC(C2CCCN(CC3(CC)COC3)C2)=O)ncc(Br)c(N(C)C)n1 84522,c1(C(N(CC(CC)NC(=O)CC(C)n2ccc(C3CC3)n2)C)=O)ccncc1F 84523,N1(C(CC(C(C)C)O)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1C 84524,CCC(C#N)C(=O)NC1CCN(C(=O)CC(C)(C)C)C1C1CC1 84525,c1(C(=O)NC23CC(NC(=O)C=Cc4cnccn4)(C2)C3)ccc(C(F)F)nc1O 84526,C1(CC(N2CCCC(N(C)C(c3n[nH]cc3F)=O)C2)=O)NC(=O)CNC1=O 84527,C1(C(N2CC(C#N)(SC)C2)=O)CN(C)CCN1C(C1CCCCC1(C)C)=O 84528,C1(CNC(c2ocnc2C(F)F)=O)CCC2CN(C(c3ccc[nH]3)=O)CCC2C1 84529,C1(NC(C2C(CC)CCC2)=O)CCC(NC(c2cc(OC)c(Cl)s2)=O)CC1 84530,S(=O)(=O)(c1cccc(F)c1)NCCN(CC)CC1CC1NC(=O)Cn1cccc1 84531,N1(C(=O)CCCCCn2cc(C3CCCO3)nn2)CCCC2(CCNC2)C1 84532,N1(C(c2cccc(OC)c2OC)=O)CCCCC12CN(C(c1ccoc1C)=O)C2 84533,C1(CCCC)CN(C(=O)Cc2ccco2)CCN1C(=O)CN(C)CCOC 84534,Cn1ccc(C(=O)NC2(C(=O)NC3CC(CO)C34CCC4)CCOCC2)cc1=O 84535,N1(C(c2ccc(C)o2)=O)CCC2CCN(C(C3CCCCC3)=O)CC12 84536,C1(O)(C(C)NC(=O)C(F)C2CCOC2)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 84537,CCC(CC(=O)N1CC(OCCC(=O)NCC2CC[Si](C)(C)C2)C1)C(C)C 84538,Cc1cccc(Br)c1C(C(=O)NC1CC1(C)C)NC(C1CCC2(CC2)C1)=O 84539,Cc1ccc(C)n1CC(=O)NC1C=CC(C(=O)NCC2CCC(C)C2)C1 84540,c1(OC)cc(O)c(C(N2CCC2C(=O)NC(C)(CO)CO)=O)cc1O 84541,C1(C(N2CC(NC(c3csc(Cl)c3Cl)=O)C(O)CC2)=O)CCCC2(CCC2)C1 84542,c1(C(=O)NCC(=C)CCNC(c2c[nH]nc2C)=O)csc(C)c1C1CC1 84543,CC(C)(C#N)CCCC(=O)NC1CCCC1NC(C12CCC(CC1)C2)=O 84544,C(=O)(C1COc2ccccc21)NC(C1CCN(C(Cc2c(C)[nH]nc2O)=O)CC1O)=O 84545,C(=O)(CC1OCCc2ccccc21)NCc1cc(C)n(C)n1 84546,C1(NC(Cn2ncn(C)c2=O)=O)CC2CCC1CC2NC(=O)CC1CC2C=CC1C2 84547,c1(C(N(C(CNC(C(CC)=CC)=O)CC)C)=O)nccc(C)c1O 84548,N1(C(c2nn(C)c(C#N)c2)=O)CC(NC(=O)CN2CCS(=O)CC2)CC(O)C1 84549,C(N=c1[nH]cncc1OC)C1N(C(CC2CC(CC)OCC2)=O)CCCC1 84550,c1(C(N2C(C)CC(NC(=O)CS(N)(=O)=O)CC2)=O)ccc2n[nH]cc2n1 84551,O=C1CC(NC(c2cc(C3(O)COC3)on2)=O)C2(CCC2)C1 84552,C(=O)(C1=NOC2(CCOC2)C1)NCC1(OC)CN(C(=O)C(F)n2cccn2)C1 84553,N1(C(c2c(C)snc2)=O)CCC(O)C(NC(C2(C)CC23CCC3)=O)C1 84554,C1(NC(CN(CC)CC)=O)CN(C(=O)C(CC(C)C)OC)C(C)(CC)C1 84555,N1(C(C2C(C)OCC2)=O)CCC(C(F)F)(CNC(=O)COC(F)(F)F)C1 84556,N1(C(c2ncccc2Cl)=O)CCC2(CCCC2Nc2nccc(CO)n2)CC1 84557,c1(C(N(C(CNC(C2(C(=O)OCC)CC2)=O)C)C)=O)ccc(N)cc1C 84558,C1(CNC(CCC(=C)Cl)=O)COCC2(CCN(C(=O)CC3=CCCCC3)C2)O1 84559,CC1CN(C(C2CCC(c3ccccc3)C2)=O)CC1CO 84560,C1(C)(CC)C=C(C(=O)Nc2cccc(NC(C3(OC)CCS(=O)(=O)C3)=O)c2)C1 84561,N1(C(=O)OC)CC(C)CN(Cc2nnc3n2CCOC3)c2ccccc21 84562,N1(C(c2ncc(CC)nc2)=O)CC2(C1)SCCC2NC(=O)C1=CCCCO1 84563,N1(C(Cc2ccc(OCCCC)c(OC)c2)=O)CC(O)(C2(C(=O)O)CCC2)C1 84564,C1(NC(CCc2onc(C)n2)=O)CC2CCC(C1)N2C(c1ccnc(Cl)c1F)=O 84565,C12(NC(COCCCCC)=O)CC(C(=O)NCC3(F)CC3)(C1)C2 84566,C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCN(C(c2ccoc2Cl)=O)C1 84567,C=CCC(F)(F)C(=O)NCC1CC2CC1CN2C(c1c(C)cccc1F)=O 84568,C12(CNC(=O)Nc3[nH]c(=N)sc3)CNCCN1CCOC2 84569,C(=O)(CS(=O)(=O)CCO)N1CCCC(Nc2cc(C(N(CC)CC)=O)ncc2)C1 84570,N1(C(COCCOC)=O)CCC2CCN(C(c3cc(F)c(C)cc3C)=O)CC12 84571,C1(C(=O)O)(C(=O)NCc2cncnc2)CC2CCC1CC2 84572,N1(C(C(C)OC2CCCCC2)=O)CCCCC1CNC(C1CC1c1ccsc1)=O 84573,Cn1ccn2ncc(C(=O)NC3CCCN(C(c4cc(F)c(N)c(F)c4)=O)C3)c12 84574,N1(C(C2CC(CCNC(c3nc(CC)oc3)=O)C2)=O)CCC(CO)C(F)(F)CC1 84575,C=C(C)C1OCCC1C(=O)NCC1(NC(=O)C(F)C(C)(C)O)CCCC1 84576,N1(C(c2c(CC)scn2)=O)CCC2(CCCN(C(c3ncccn3)=O)C2)C1 84577,c1(NC(C2CCC(NC(=O)C=CC(F)(F)F)C2)=O)cncc(C2CC2)c1 84578,c1(C(C(=O)NCCCF)NCc2ncn(C)c2)cccc(Cl)c1Cl 84579,C1(C(N(CCC(=O)NCCC(=O)NCCOC)CC#C)=O)CCC(=O)N(C)C1 84580,CC1CCCC(CC(=O)NCc2csc(C(N3CCC3CF)=O)c2)C1 84581,C(c1ccncc1)=C(C)C(=O)NCC1CCCCC1NC(C1CC2CCC1C2)=O 84582,N1(C(C2N(C(C3CCC(C)C3)=O)CCOC2)=O)CCCC(O)(CN(C)C)C1 84583,n1(CC(N2CC(NC(C3C(C)OCC3)=O)C(O)C2)=O)nc2c(n1)CCCC2 84584,C1(OC(C2(c3ccccc3)CCC2)=O)CCCC1NC(=O)OC.C1(=O)CCO1 84585,C1(C(=O)NCC2(CNC(C(C(C)C)C3CCC3)=O)CCC2)Cc2nccn2C1 84586,c1(C(N2CCCC2CCNC(C2CS(=O)(=O)C2)=O)=O)nc[nH]c2nccc1-2 84587,c1(CC)nc(Cl)c(CC)c(=NC2CCCCC2NC(=O)CC2CCC(=O)N2C)[nH]1 84588,N1(C(Cn2c(CCC)ncn2)=O)CCC(NC(=O)C(O)C(C)(C)C)C12CCCC2 84589,c1(OC)ccc(F)cc1CCC(N1CC(NC(=O)Cc2cncn2C)C(C)C1)=O 84590,C1(C2CC2)(C(N2CC3C(CNC(C4CCS(=O)(=O)N4)=O)C3C2)=O)CC=CC1 84591,C12(C(=O)NCc3c(CNC(CCCCC#C)=O)cccc3)CCC(OC)(CC1)CC2 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84747,C(=O)(C(F)CC(C)C)NCC(=O)N(C1CCN(C(C=C(C)C(C)(C)C)=O)CC1)C 84748,N1(C(C)=O)CCCCCC1CN1CCC(C(=O)Nc2ccc(C(N)=O)cc2)CC1 84749,C(C)(C)(CC(=O)N1CCCCC1CCNC(=O)Cc1coc(C(F)F)n1)OC 84750,C1(C2(O)CN(C(c3cccc(Cl)c3Cl)=O)C2)(CNC(C(C)C(C)(C)C)=O)CC1 84751,c1(C(N2CC3CN(C(c4c(C)nsc4)=O)CC32)=O)cc2cc[nH]c2cc1Cl 84752,CC(C)(O)C(C)(C)NC(C1CCC(CNC(c2ccncn2)=O)O1)=O 84753,C1CCC(=O)N1.C1(C(C)COCC)CCCN1C(=O)C(CC)OCCN(C)C 84754,c1(N2CC(C(C)NC(=O)C(c3cccc(Cl)c3)(F)F)C2)cc(C)ccc1[N+](=O)[O-] 84755,c1(NC(Cc2cccc(NC(C)=O)c2)=O)ncc(Cl)cc1C#N 84756,c1(C(=O)NC2CC(C)(NC(CSc3n(C)ccn3)=O)C2)ccc(O)nn1 84757,C1(COC)(NC(=O)Cn2nnc(=O)[nH]2)CCN(C(=O)Cc2cc(C)no2)CC1 84758,Cn1nnnc1C(c1nnnn1CC1CCOC1)NC1(n2cc(Br)cn2)CC1 84759,C1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)CN2CCC1CC2 84760,c1(N2CCC(CC(=O)NC)C2)nc(=NCCC(O)C(C)C)[nH]c2c1SCC2 84761,C1(C(=O)NCC(COC)(C)CO)CCCN(C(C2CC3CCCC3C2)=O)CC1 84762,C=CCC(C)(C)CC(=O)N1CSCC1C(=O)Nc1cnccc1SC 84763,Cc1ccc(O)c(C(N2CCOC(C(=O)NCC(CO)C(C)C)C2)=O)c1 84764,N1(C(C(COC)NC(C)=O)=O)CCC(C(=O)NC2(C)CCSC2)C1(C)C 84765,Cc1ncc2cc(C(N3CC4C(NC(=O)C(F)(F)c5cscn5)C4C3)=O)ccn12 84766,CN1CC(NC(C2(CCNC(=O)C(=O)N(C)C)CCCC2)=O)C(O)C1 84767,c1(CCC23C(CN(C(CN4CC(C)C4)=O)C2)CC3)csc2c1CCC(C)C2 84768,N1(OC(Cc2cc(C)no2)=O)CCCCCC1.C12(CC1)C(=O)N2C 84769,C12(C(=O)NCc3c(C)nn(C)c3)CCCC1CN(C(C1CCCCO1)=O)C2 84770,Oc1cc(CSCC2CCS(=O)(=O)C2)ccc1F 84771,CCC(C(=O)OC)C(C)N=c1[nH]c(=N)[nH]c(=NCCCOCOC)[nH]1 84772,c1(SCC)cncc(C(=O)NC2CCCN(CCNC(=O)CNC(C)=O)C2)n1 84773,c1(C(=O)NCC2(COC)N(C(CCC=CC)=O)CCC2)cc2cc(C)ccc2[nH]1 84774,CCCCCCC(F)C(=O)N1CC(NC(c2ccc(CC)cc2)=O)C1 84775,C1(C(=O)NCCC(C(=O)OC)O)CCCCC1(C)NC(C1CCCCCC1)=O 84776,O=C(C1=C(Cl)CC1)N1CCC1CC(N1CCC(n2cnnn2)C1)=O 84777,C(C(C)C(C)C(=O)N(CC(=O)N(C)CC1CCCC1)C1CC1)OC 84778,C(=O)(C(C)CN(C)C)N(CC(CC)NC(=O)C(C)CN(C)Cc1ccccc1)C 84779,C=CC(CC)CC(=O)NCC(COC)OC.C1=CCN(C)C(=O)CC1 84780,C1(CC)CN(C(c2cn(C)nc2C)=O)CCC1NC(=O)Cc1ccns1 84781,c1(NC(C(CC)NC(=O)CC2C=CCCC2)=O)cccc(CSC)c1 84782,C1(C(=O)NC2CCCN(C(CNC(CC(C)C)=O)=O)C2)CC2CC1CC2(F)F 84783,CCCC(CCCNC(C1OCCCO1)=O)NC(C1(C(=O)N(C)C(C)C)CC1)=O 84784,CC1CN(C(=O)CC2NC(=O)NC2=O)CC1NC(=O)CCc1nc(C2CC2)no1 84785,CCC(CCC(=O)NCC1CC2(CCC2)CO1)NC(=O)C=CC1CCC1 84786,C12(N(C)C(C3CC3(C)C)=O)CC(C(F)(F)F)(C1)C2 84787,CON=C(C(=O)NCC1CCC1NC(c1coc(S(N)(=O)=O)c1)=O)c1ccco1 84788,C1(C(=O)NCCC(C)(C)O)CC2CCC1N2C(c1cccc(Cl)c1)=O 84789,C1(NC(C2(COC)CCN(C(=O)CC(C)C)CC2)=O)CC2(CCCCCC2)C1 84790,C(=O)(CC(C(F)F)NC(C1C2CCC(C2)C1C)=O)NCCc1ccc(C)s1 84791,c1(C(=O)NCCC(=C)C)cc(C)c(CC)o1.C1(=O)CCO1 84792,c1(CCNC(=O)Cc2cc[nH]n2)nc(CCNC(c2csc(C(F)F)c2)=O)no1 84793,N1(C(c2c(OC)nsc2)=O)CC2CCC1(CNC(C1(C(F)(F)F)CC1)=O)CC2 84794,N1(C(CC2CCCN(C(C(C)OCOC)=O)C2)=O)CC(O)C(O)C1CO 84795,O=C(C1=CS(=O)CCC1)NC1CCCCN(C(C2(O)CC2)=O)C1 84796,c1(CC(=O)NC(C(C)C)CNC(=O)Cc2cnoc2)ccccc1N=S(C)(C)=O 84797,C1(NC(C(Cc2cnc[nH]2)NC(C(C)C2CC2)=O)=O)CC2(CCC2)C1 84798,c1(C(=O)NCCC(C)NC(c2coc(Cl)n2)=O)ccc2c(c1)OCCCO2 84799,c1(C(N2CC(N(C)C(C3CC3(Cl)Cl)=O)C2)=O)cc2n(n1)CCCC2 84800,c1(C(N(CCN(C(C)C)CC=O)C)=O)nocc1C(C)C.S(=O)(=O)(Cc1ccsc1)N 84801,N1(C(C(=O)N(C(C)COC)CCOC)=O)CCCCCCCCCC1 84802,c1(C(C(=O)NCC(CNC(C2(C(C)C)CCC2)=O)C)(C)C)cc(Cl)cc(Cl)c1 84803,C(=O)(CS(=O)(=O)N(C)C)NCC(CNC(C1CC1F)=O)OC 84804,O=C1CCC(CC(=O)N(CCCNC(c2ccc(F)o2)=O)C2CC2)C(=O)N1 84805,c1(NC)ccccc1C(N(CC(CNC(C1(OC(C)C)CCOC1)=O)O)C)=O 84806,C(CCC)(C(=O)NCc1cccnc1CNC(C1CC1COC)=O)=CCC 84807,C12CCCCC1OCCN(C)C2=O.C1(OCC)CC(C(=O)N(C)C)C1.C1CO1 84808,CC(C(=O)N(C(=O)NC(C)(C)C)C(c1ccccc1)=O)C(C)NC12CCC(C1)C2 84809,C(=O)(CCCCC(=O)OC)N1CCC(N(C(CC(CCC)O)=O)CC)CC1 84810,c1(C(N2C(C)CC(NC(=O)CC(=O)NC3CC3)CC2)=O)nnc2ccccc2n1 84811,C(C)(C(=O)NC(C1CCCC1)CNC(c1nc(Cl)ccc1N)=O)(C(C)C)OC 84812,C1(NC(C(CC)NC(=O)C(C)N2CC(C)C2)=O)CCOC(CC)C1 84813,c1(C(N2CC(C(N)=O)(CNC(c3cn(C)nc3O)=O)C2)=O)c[nH]c2ncccc12 84814,c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)C2)ccc(S(N)(=O)=O)cc1 84815,c1(C(N2CC(N(CCC3=NNC(=O)C3)C)C2)=O)cnc2cccc(Br)n12 84816,CC(=O)CCN=C(NCC1CC2(C1)CC(C)(C)C2)NCC1CCC2CC1C2(C)C 84817,c1(N(C2CCN(C(c3ccsc3)=O)C2)C)ncc2ncnc-2[nH]1 84818,c1(CCCOCC)nc(-c2ccnc(Cc3ccccc3)c2)n(C2CCOC2)n1 84819,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCc1cnc(C)s1)NCCC 84820,c1(C(C)NN(CCCc2cnn(C)c2)C)ccc(-c2nc(C3CC3)no2)c(Cl)c1 84821,CC(CC(C)(F)F)C(=O)NCCC1(NC(=O)CC(F)(F)C(F)F)CCOCC1 84822,c1(OC)ccc(CC(=O)NC(C)CCCNC(=O)C(C=O)OC)c(OC)c1 84823,CN1CCCCC1CCC(N1CCC(C(=O)NCC23CCC(CC2)C3)(CO)C1)=O 84824,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 84825,N1(C(c2cc(C)c(C)[nH]2)=O)CC2CCC(C1)N2C(c1c(C)noc1C)=O 84826,CC1=C(C(=O)N2CC(CNC(C3CC4(C3)CC3(CC3)C4)=O)CCC2C)SCCO1 84827,C(=O)(C1=CCC2CCC1N2C(c1cccs1)=O)Nc1c(C)n(C(C)C)nc1 84828,C1(C(=O)NC2CC(OCC(=O)NCC3=NOCC3)C2)CC2CCC(C1)O2 84829,c1(C(=O)NC2C(NC(=O)C=CBr)CCC2)ccc(F)c2ccccc12 84830,Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CC(NC(c2c[nH]c(=N)nc2C)=O)C1 84831,N1(C(C(CC)(F)F)=O)CC2CC(NC(c3cc(C4CCCC4)no3)=O)CC2C1 84832,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 84833,N1(C(C(C(C)C)NC(c2n(C=C)nnc2)=O)=O)CCN(C)C(C)C1C 84834,CC1CC(NC(c2nccn2C)=O)CN1C(c1snc(O)c1Cl)=O 84835,c1(C(=O)NCCN(CCC)C(c2coc(Br)c2)=O)ccnc(C(F)F)c1 84836,CCC(CC(F)(F)F)C(=O)NCC(C)(CC)NC(C1CC2C=CC1C2)=O 84837,Cc1ccc2c(c1)CC(C(=O)NC1CC3CN(C(c4ccccc4Cl)=O)CC13)S2 84838,c1(CC)ccc(C(=O)OC)cc1F.C(F)(F)(C(F)(F)F)O 84839,C(=O)(C(Cc1cn[nH]c1)NC(=O)COCCF)NCCN(CCC)C(C)C 84840,CCC(F)(F)C(=O)N1CCC(C(C)(C)NC(=O)CN2CC(C)(OC)C2)CC1 84841,c1(C(=O)NC2CC(C)(CNC(CCCOCC)=O)C2)ccc2[nH]cc(C#N)c2c1 84842,CCC(C)C(C)(O)CNC(=O)C(C1CCCC1)NC(=O)CCCn1cccc1 84843,c1(N2CCN(C(C)C#N)CC2)nccc(=NCCc2cccc(Cl)c2)[nH]1 84844,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C(C)C)nn(C)c2c1CCCC2 84845,c1(C(=O)NC23CC2CN(Cc2ccncc2Br)C3)ccc(O)cc1O 84846,C1(C(N2CC(N(C(C3=NOC(C)C3C)=O)C)C2)=O)COC2(CCC2)CO1 84847,CC1=C(C(=O)NCc2cc(C(=O)OC(C)(C)C)on2)CCO1.C(CCCC1CC1C)C 84848,C1(C(=O)NCC2N(C(C(CCC)C#N)=O)CC=C2)CCc2nnnn2CC1 84849,C(c1cccc(F)c1Cl)=CC(=O)NC(C(C)C)(C)CNC(=O)C1=CC(C)CC1 84850,C(CC(C)(C)C(=O)N1CCC(C)C(CNC(=O)C#CC2CC2)C1)OC 84851,c1(OC)cccc(C(CNC(=O)NCC2CC2(F)F)CO)c1 84852,S(=O)(=O)(c1cccc(=NC2COC3(CCCCC3)C2)[nH]1)NC(c1cc(Br)cs1)C 84853,CC1(C)CC(NC(C2CC(N3CCOCC3)C2)=O)CN1C(=O)C(F)C(F)(F)F 84854,C#CCCC(C(=O)NCC(C)OCC=C)NC(=O)C(C)CC 84855,c1(C(=O)NCC(=O)NC(C(C)C2CC2)=O)cn(CSC2CC2)cn1 84856,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 84857,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 84858,N1(C(C(C)Oc2ccccc2)=O)CC2CCC(NC(=O)CSC3CCCO3)(C2)C1 84859,N1(C(c2c(CNC(C(C)(C)n3cnnn3)=O)cco2)=O)CC2C=CC2C1 84860,C(=O)(C(C)S(=O)c1ccccc1)N1CCCC(F)(C(=O)NC2(COC)CC2)C1 84861,c1(C2C(CNC(=O)NC(C)CC3CCN3)C2)ccc(F)cc1F 84862,N1(C(c2c(C)oc(C3CC3)c2)=O)CCCC(c2ccccc2)CC1 84863,c1(C(=O)NCC(CO)NC(C(c2ccccc2Cl)C)=O)cnc2ccccc2c1 84864,C(=O)(C1=CCCCO1)NCCCC(C)NC(=O)CC1CCOC1C 84865,N1(CC(=O)NCCCCN(C(=O)C=CC2CC2)C)CCC(F)(F)C1 84866,CC1CCCN(C(C23CC(CN2C(N)=O)C3)=O)C1CO.c1(C=O)ccc(C2CC2)nc1 84867,CC1OCCOC1C(N1CCCC1C=CC(=O)NC1CCCOC1)=O 84868,CCC(O)CN(C(=O)C(C1CC1)N(C(=O)CNC(=O)CN(C)C)C)C 84869,c1(CC)[nH]c(=N)sc1C(=O)N(C(C)CNC(=O)C(C)(C)CC1CC1)C 84870,Cc1cc(C(=O)NC(C2CCCCN2C(=O)CSc2nncn2C)C)ccn1 84871,C(CC(C)C(=O)N1CCCC(OC2(CC(=O)NOCC)CC2)C1)=CC 84872,Cc1nc(-c2cccs2)c(CNC(N2CC(F)CC2c2ccccc2)=O)s1 84873,Cc1ccc(C(=O)NCCCC2(CNC(=O)C(C)(Cl)Cl)CCCC2)c(Cl)c1N 84874,c1(NC(C2CC(OC)CN2C(=O)Cc2ccc(Cl)s2)=O)ccc(O)cc1Br 84875,N1(C(C2(CC(C)C)CCC2)=O)CC=C(CNC(C2CCOC2C)=O)CC1 84876,C#CC1(NC(C2(CF)CCN(C(C3CCC3)=O)C2)=O)CCCCCC1 84877,c1(C(=O)NC2CCN(C(CCC)=O)CC2C)c(Cl)nc2cc(Cl)ccn12 84878,c1(CN(C(=O)CSS(C)(=O)=O)C)ccc(CNC(C2(C)CCCC2O)=O)cc1 84879,c1(C(c2nnnn2C(C)C)NCC(c2ccccc2)C)cc(OC(F)F)ccn1 84880,c1(CCC(=O)NC2CC(SC)OC2)ccccc1-n1cc(-c2cccnc2)nn1 84881,CC1(C)CC(NC(=O)C(CN=[N+]=[N-])NC(c2nc[nH]n2)=O)C(=O)O1 84882,Cn1ncnc1C(=O)N(CCCN(C)C)CCNC(C1(C)CC1F)=O 84883,c1(CCNC(C(C)(C2(C)CC2)N(C)CC)=O)cn(Cc2ccccc2)nn1 84884,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 84885,C1(C(=O)NCC=C(C)C2CC2)CC12CCN(C(=O)C(N1CCOCC1)C)CC2 84886,C(=O)(C1(C)OCCc2ccccc21)NC(CNC(c1cncc(NC)c1)=O)(C)C 84887,Cn1nnc2c1CCN(C(=O)C(C1(O)CCC1)NC(C1CCCOC1)=O)C2 84888,C(C)(C(=O)OC)(C(C)C)N(Cc1n(CC)c(-c2ccc(Cl)cc2)nn1)CC.OC 84889,C(=O)(CCN(OC)C(=O)C=Cc1cncn1C)N(C1(CCC)CCC1)C1CC1 84890,n1(CC)ccc(CC(=O)NC2CCN(C(=O)C(C)(C)c3cscc3Cl)C2)n1 84891,CC1CC(N(C(=O)C(C2CCC2)NC(c2ccoc2Cl)=O)C)CC(C)C1 84892,N1(C(c2c(C)scn2)=O)CCN(C(=O)CC23CCC(CC2)C3(C)C)C2CCCC12 84893,Cc1c(C(=O)N(CCCCN(C(=O)CC2(C)CCCCC2)C)C)cnn1C(C)C 84894,C1(C(F)(F)F)(NC(C2C(C)CCO2)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1 84895,C(=O)(CCCCCCCCC1CC1)N(C)CCNC(c1nc(Cl)cs1)=O 84896,C1(C(=O)NCc2ccno2)CSCN1C(C1(Cl)CC1)=O 84897,N1(C(C2(CCCC)CC=CC2)=O)CCC(C)C(CNC(c2nc(C)sc2C)=O)C1 84898,c1(C(=O)NCCOCCN(C(C2C(C)CCO2)=O)C)ccc(F)c(F)c1O 84899,N1(C(C2(SC)CN(C(=O)Cc3ccnn3C)C2)=O)CCC(F)CC1 84900,C1(COC)(CO)CN(C(=O)COC(C2CC(OCCSc3ccccc3)C2)=O)C1 84901,C(=O)(C(F)C(C)(C)O)NC(C1CC1C(=O)N(C1CCCC(O)C1)C)C 84902,C(=O)(C(CC(C)C)C(C)C)N1CC(C(C(=O)N(CCCCCC=C)C)O)C1 84903,N1(c2cc(OC)nc(C(F)(F)F)n2)CC2CC1CN(C(=O)CC(C)C(C)C)C2 84904,C12(C(=O)NC(C)CNC(C3CCSCC3)=O)CC(CO)(C1)OC21COC1 84905,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCCS3)=O)CC1CCO2 84906,c1(C(N2CCC(CC(N3CCCC(CCO)C3)=O)C2)=O)ccncc1Cl 84907,Cc1nc(C(=O)NCC(C)(C2CC2)NC(c2ccn(-c3ccncc3)n2)=O)co1 84908,CC1(C)CCCCC1C(=O)NC1CC(NC(c2cccc(SC(F)(F)F)c2)=O)C1 84909,CC(CC(F)(F)F)C(=O)N1CC(c2ccccc2)(NC(C2CCC3CC23)=O)C1 84910,c1(CC(=O)NC(C2CCN(C(CCCC(C)C)=O)C2)C)ccc2cnccc2c1 84911,c1(CCCC#N)ccc(NC(C2(CCC(=O)O)CCC2)=O)o1 84912,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 84913,Cn1nc(Cl)c(C(N2CCN(C(=O)CC3COC4CC3C4)CC2C2CC2)=O)c1Cl 84914,CC1CC(NC(=O)CC2CC(=O)C2)CCN1C(C1CCCCC1)=O 84915,CC1(C)CC(CC(=O)OCC2CC(C)(F)C2)C1 84916,C(c1scnc1C)=CC(=O)NCCc1nc(C)[nH]n1 84917,C1(CC)C(NC(c2c[nH]nc2OCC)=O)CCCN1C(c1ncnc(C)c1C)=O 84918,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(=O)Cc1nc(=N)[nH][nH]1)C2 84919,C(C(Cc1ccccc1)C(=O)OC)Sc1ccc(Nc2snc(CC)n2)cc1 84920,Cc1nc(C(=O)NC2CCCC2NC(c2ccc3snnc3c2)=O)ccc1[N+](=O)[O-] 84921,N1(C(C(C)N(C)C)=O)CC2(NC(=O)Cc3ccnn3C3CCCC3)CCCC1C2 84922,N1(C(C2N(CC)CCCC2)=O)CC(C(=O)N(C)CCN(C)C)CC2COCCC12 84923,C=CCC(C)C(=O)NCC(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O 84924,S(=O)(=O)(c1ccc(C(=O)NC2(CN(C)C(c3c[n+]([O-])cnc3C)=O)CC2)o1)NC 84925,Cc1scc(CNc2ccc(OCC(O)CN(C)C)cc2)c1C 84926,c1(OC)cc(OC)cc(CC(=O)NC2CC(C)CN(C(=O)CC3CN(C)C3)C2)c1 84927,C(C(=O)NNC(=O)C(c1ccccc1)N(C)C)NCC(c1cc(C)c(F)cc1)O 84928,CC1(CCC(N2CCN(C(=O)CCS(C)(=O)=O)C(CF)C2)=O)CCOCC1 84929,c1(C(C)NC(CC2(CC=C)CCCC2)=O)c(OC)cc(C(=O)OC)cc1OC 84930,CC(C)CC(=O)NCCC(C)N(C(=O)C(n1cc(Br)cn1)C)C 84931,c1(C(=O)NC2C(C(=O)NC(C3CCCC3)C#C)CC2)cc(C#N)n(C)n1 84932,c1(NC(NOC(NOCCC=C)=O)=O)ccc(CC)cc1 84933,c1(C(=O)NCC(C)N(C)C(c2cn(C3CCCCC3)nn2)=O)cccn(C)c1=O 84934,C1(CNC(CCCN(C)C)=O)CN(C(c2cc(CCO)on2)=O)C2CC12 84935,C1(NC(C(c2scc(C)n2)C)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCCC12 84936,C1(C(N2C(CNC(c3ncccc3C(F)(F)F)=O)CC2)=O)COC2COCC2O1 84937,c1(N(CC(c2n(CCC)nnn2)NCC(C)C)C)ccc(F)cc1SCC 84938,CC1CC(C(N2CCC(C)C2CNC(=O)C=C2CCSCC2)=O)CCS1 84939,N(C1CCCc2c[nH]nc21)C(C1=CCC(NC(C#CC(C)C)=O)C1)=O 84940,N1(C(c2c(C)[nH][nH]c2=N)=O)CC2(C1)CN(C(c1ccc(C(C#N)C#N)cc1)=O)C2 84941,N1(c2nnc(CC)o2)CCC(NC(C2CCCOC2)=O)C1(C)C 84942,c1(C(=O)NCC(CC)NC(=O)C=CCc2ccc(C)cc2)cccc(OC)c1C 84943,c1(CN(C(=O)C(=O)NCc2cscc2Cl)CCOC)ccccc1Cl 84944,c12cc(ncn1)N1CCCC(C1)NC2.c1(CC)cccc(-c2nc(=O)o[nH]2)c1 84945,c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 84946,N1(CCC(=O)OC)CCN(C(=O)Cc2ccc(O)nc2)CC1.C12(CC1)C(=O)NC2 84947,C(CCCC(=O)N1CCCC(C(=O)NCCCN(C)C)C1)N(C)C 84948,c1(C(=O)Nc2cc(F)cc(F)c2F)ccc2c(c1)OCO2.CC12CCN1NC2=O 84949,Cc1ccc(F)c(C(=O)NC2CCC(NC(C3CC4(CCCO4)C3)=O)C2)c1Br 84950,C(=O)(NN1CCCC1C(=O)NCC1C(C)(C)C1(F)F)c1c[nH]c(C)c1.NC=O 84951,c1(N2CCN(CC)CC2)nc(=NCc2nnnn2C2CCOC2)[nH]c2cc[nH]c12 84952,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 84953,C1(C)(C(=O)NCCC2CCC(CC)O2)CCN(C(=O)C(C)(C)OC)CC1 84954,c1(C(N2CC(NC(=O)CC(C)C(C)C)CC(OC)C2)=O)cc2n(n1)CCN(C)C2 84955,C(=O)(CS(=O)C(F)(F)F)N1CC(NC(C=Cc2c(C)ccs2)=O)C1 84956,c1(-c2ccccc2)ccc(F)cc1F.n1(CCC(=O)N2CCNCC2)ccnc1 84957,N1(C(c2n(C(C)C)cnc2)=O)CC(C2CCCN(C(=O)C(C)(C)CC3CC3)C2)C1 84958,Cc1cc(CNC(=O)NC2CC(O)C23CCC3)c2n[nH]cc2c1 84959,Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C(=O)CSCC(N)=O)C 84960,C1(C(=O)NCCC(=O)NC(C)C(c2cccs2)NC(=O)CO)CCCCC1 84961,C(=O)(C(CC(C)(C)C)OC)N(CCCN(C(C1COCOC1)=O)CC)CCC 84962,c1(OC)cc(OC)cc(C(N2CC(C(C)NC(C3CCCC3(C)C)=O)C2)=O)c1 84963,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 84964,C1(C(N2C(CC)CCCC2)=O)C(C2CC2)CCN1C(=O)CC1CC(C)C1 84965,Cc1nccnc1C(=O)NCC1CC1CC(=O)NC(C)(CO)C1CCCC1 84966,c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)cc(O)c2ccoc2c1 84967,C1(COC)(COCC(=O)OCCF)CCN(C(=O)C(C2CCC2)C2CC2)C1.OC 84968,c1(C(=O)NC23CC(C2)N(C(C2COCCO2)=O)C3)cnc(O)c2ccsc12 84969,CC(C)(C)CCC(F)C(=O)N1CC(CNC(c2cncc(Cl)c2)=O)C2(CCC2)C1 84970,C(=O)(C(C)(C)CNC(=O)CC(C)CNC(=O)C(C1CCC1)OC)OC 84971,C(C(O)C(F)(F)F)NC(C1CC(NC(C2CC(C)(F)C2)=O)C1)=O 84972,c1(NC(c2ccc(CNC(c3scc(C)c3Cl)=O)nc2)=O)ccc(I)cc1Cl 84973,c1(CC)ccc(NC(=O)CN2CC(c3ccc(F)cc3)C(N)C2)cc1 84974,c1(C(=O)NCCCNC(CN(CCOC)C)=O)ncc(N)cc1C 84975,c1(N2CC(F)(F)C3(C2)CCC3)nc(N2CCC3OCCCC3C2)c2ccccc2n1 84976,C(=O)(C(C(C)(C)C)NC(c1cc(OC)ccc1N)=O)NCCCOCC 84977,CC1(C)CN(C(=O)COC2CCOC2)CC1C(=O)NCCn1cccnc1=O 84978,c1(C(N2CC(C)N(C(=O)CN3CCCCC3=O)CC2)=O)ccn2[nH]c(=N)nc2c1 84979,Cc1c(Br)ccc(NC(C2CCC(NCc3ccc(O)cc3Cl)CO2)=O)c1F 84980,C(CC(=O)NC12CC(NC(=O)C(C)=C(C)COC)(C1)C2)(OCC)OC 84981,c1(OC)c(F)cc(C(=O)NCC2CC2NC(=O)C(F)C2CCC2)cc1Br 84982,C1(CNC(c2c(N)ncc(C)c2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC(C)(C)C1 84983,c1(C(=O)NC2(C)CC(NC(CSc3cccc(C)c3)=O)C2)cc2scc(Cl)c2[nH]1 84984,CC(CC(=O)NCC12CCCC(CN1C(C1COCCOC1)=O)C2)CC(F)(F)F 84985,CC(C)C(C(=O)N(C1CN(C(=O)CCF)C1)C)n1cccc1 84986,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)NC(C(CC)SC)=O 84987,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(c1occc1C1CC1)=O 84988,c1(N(CCNC(CC2C(C)C2)=O)C2CC2)nc2ccc(O)cc2s1 84989,CCC(CC(=O)N1CC(C(=O)NCC(c2ccncc2)O)C2(CCC2)C1)C(C)(C)C 84990,N1(C(CN(C)C(N)=O)=O)CCC(C)(C)CC1C(=O)NCC(F)(F)CC 84991,Cc1c([N+](=O)[O-])ccc2cc(C(=O)NCCN(C3CC3)Cc3ccccc3)[nH]c12 84992,c1(C(N(C2CN(C(CC(C)C3CC3)=O)CC2O)C)=O)cc2c(cnn2C)nc1O 84993,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 84994,CC1=C(C)CC(C)(C(=O)NCC(O)CNC(c2sccc2C2CC2)=O)CC1 84995,c1(C(=O)NC2CCC(N(C(CC(=C=C)C)=O)C)C2)c(OC)ccnc1O 84996,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 84997,Cc1cc(C)c2nc(NC3CCN(C(c4cnc(C(C)O)s4)=O)C(C)C3)sc2c1 84998,C1(C(=O)OCC)=C(N=[N+]=[N-])CCN(C(C2CC23CC3(F)F)=O)C1 84999,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85000,c1(C(C)=O)ccccc1OCC(=O)NCC(C)(C)CNC(=O)C=CCO 85001,c1(C(=O)NCC(C2CCC2)NC(C2(C)CCCS2)=O)ncn2ccccc12 85002,c1(N(C)Cc2cc(C)ncn2)nc(N2CC3CC3(CO)C2)nc2sccc12 85003,C1(C)(NC(CCc2ncn(C)c2)=O)CCN(C(C2(CCF)CCC2)=O)C1 85004,N1C2CC=C(C(=O)C(c3nc(CC)oc3)=O)C1CC2.c1(CN)nonc1C 85005,c1(C(N(C(CN(C(c2nc(C(C)=O)sc2)=O)C)C)C)=O)ccc2sncc2c1 85006,Cn1ncc(Br)c1C(C(=O)NC(c1cccc(Cl)c1)(C)C)N1CCC1 85007,N1(C(CC(C)C)=O)CCCC(N(C(=O)Cn2ccccc2=O)CCO)C1 85008,N1(Cc2onc(CC)n2)CCC(NC(C)=O)C(C)C1 85009,C#Cc1ccc(OCC(=O)NCC2CC2NC(=O)C(C2CCC(=O)CC2)F)cc1 85010,C1(CNC(c2c(C)nc(O)s2)=O)CCC12CCN(C(=O)Cc1ccsc1)CC2 85011,C1(N(C(C(CNC(C)=O)(C)C)=O)CC(N2CCSCC2)=O)CCC2(CC1)CNC2 85012,Cc1cc(C(=O)NC2CCC(NC(c3ccc(O)nc3C)=O)CC2)cnc1C 85013,C=C(C)CN=C(NCC(C)C)N(C)CC12CC3CC1C2C3 85014,C1(C(=O)NC(CC)CNC(=O)C(C)C)CC(c2cnn(C)c2)=NO1 85015,Cc1ccccc1-c1ccc(C(N2CC(C3COCCN3C)C2)=O)o1 85016,CC(C)(CCC#N)C(=O)NC1CCC2(CCC2)O1.C(=O)(CSCC(=O)O)C(=O)CO 85017,N1(C(C2CC(OC)C2)=O)CCCC(C)C1CNC(c1cnn(C)c1Cl)=O 85018,Cn1ccc2[nH]c(CO)cc12.C12CN(CCC1NC(=O)COCCF)C2=O 85019,N1(C(c2c(OC)cc(O)nc2)=O)CCC2(CCC2NC(=O)C(C)=C2CCC2)CC1 85020,c1(-c2cc(OC(C)C)cc(C)c2)cccc2c1oc1ccccc21 85021,NCC(C(F)(F)C(F)(F)F)NC1CCCCC1c1ccccc1 85022,S(=O)(=O)(c1c[nH]ccc1=NCCn1cnc(C)c1C)NCC1C(CCC)CCC1 85023,c1(C(=O)NC2CN(C(C3(C=C)CCC3)=O)CC3(C2)CC3)ccnc2c1cnn2C 85024,C1(C2NCCN(C)C2)CCC(F)(F)CC1.n12cc(nn1)C1CCOC1C(=O)CC2 85025,C(CC(C)(O)c1ccccc1)N(C(=O)CCc1nc(-c2ncccn2)no1)C 85026,c1(C(N(CCCNC(CC2CC(CC)C2)=O)CC)=O)ccc2nc(=N)[nH]n2c1 85027,C(C(CC(=O)NC1(C)CCC1)C1CCC1)NC(C(C)C#N)=O 85028,C1(NC(CCc2cnc(C)o2)=O)C(C)CCN(C(=O)CCS(N)(=O)=O)C1C 85029,Cc1cn2cc(CC(=O)NC3CC(NC(=O)CC(C)c4ccccc4)C3)nc2s1 85030,N1(C(C=CCOC)=O)CCN(CC(C)NC(c2cnc(C)s2)=O)CC1 85031,c1(OCC)ncc(C(=O)NCC2CCCN(C(C3(C)CCCO3)=O)C2)cc1Cl 85032,C=CCCCCCCCCC(=O)NC1CCSC12CN(C(=O)Cc1ccoc1)C2 85033,Cc1cc(C(=O)NC2CN(C(c3cncc(Cl)c3)=O)CC2C)nn1C 85034,c1(C(=O)NCC=CCNC(c2c(OC)cco2)=O)cc(C2CC2)nc2ccccc12 85035,CC(O)C(F)(F)C(=O)NC1CCN(C(c2ccc(Br)cc2)=O)C1 85036,Cn1nccc1C=CC(=O)NCC1CC2CC2N1C(=O)CSc1n[nH]c(=N)s1 85037,N1(C(c2cc(Cl)cc(C)c2N)=O)CC2(CCCCN(C(=O)C(F)(F)C(F)F)C2)C1 85038,N1(C(C2(NC(C(CC=C)C)=O)CC(SC)C2)=O)CC2CN(C)CC2C1 85039,N1(C(C(NC(CCC)=O)=Cc2cccs2)=O)C(=O)CCC1C(N)=O 85040,N1(C(c2[nH]nc(OC)c2Cl)=O)CCCC(C)(CNC(=O)C(c2nc(C)cs2)C)C1 85041,C(C(=O)N(C(CNC(=O)COCC1CCCO1)C1CC1)C)(C1CC1)OC 85042,C1(CCNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2(F)F)CC1 85043,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85044,c1(C(=O)NC2CN(C(CCN(CC)CC)=O)C3C2C3)cc([N+](=O)[O-])cnc1O 85045,C(C(CNC(C1OCCC1(C)C)=O)S(C)(=O)=O)NC(C1(CO)CC(C)(C)C1)=O 85046,N1(C(C2(N(C(c3c(C)con3)=O)CC)CCCC2)=O)CCCC(CCCC=C(C)C)C1 85047,C(CC(C)C(=O)N(C)CC1CCCN(C(=O)CSc2cccc(F)c2)C1)OC 85048,N12CC(N(C)NCC)(C1)C2=O.c1cnn(CC(=O)NCC)c1.N(C)(C(C)=O)CC 85049,C1(C(N2C(CCNC(C3(CCC)CC3)=O)CCC2)=O)CC2CC(C(N)=O)CC12 85050,CCCC(C)(CCC)C(=O)N1CC2(CCN(C(c3[nH]nnc3C)=O)C2)C1 85051,c1(C(C(=O)NCCNC(C(CC)(C)OC)=O)OC)ccc(OC)c(F)c1 85052,N1(C(C(C)OCCOC)=O)CC2(CC2)CC1CC(=O)NCC1CCOCC1C 85053,c1(C(=O)NC2CC3(C2)CC3COC)cc(NC(C2(C#C)CCCC2)=O)cnc1C 85054,N1(C(CC(=O)OCC)=O)CC(F)CC1CN(C)C(c1ccccc1)=O 85055,c1(CN(C)C)ccc(C(=O)NC(c2ccccc2)CNC(C2(Br)CC2)=O)cn1 85056,c1(CNC2C(SC)NC(=O)N2)cc(C)ccc1-n1ccnc1 85057,N1(C(C(CC)F)=O)CCC2(CNC(=O)CCN3CCCCC3C)CCCCC12 85058,C(=O)(CCCCCN(C)C)N(CC(C(=O)NCC(C(C)C)OC)O)C 85059,C(Cc1ccccc1)(C(=O)NCCCN(C(=O)CC1(C(F)F)CC1)C)NC(C)=O 85060,N1(C(c2c(C(C)C)ncnc2)=O)CC2CC(NC(=O)CCCCCF)CC1C2 85061,C#CCC(C(=O)N(CCCC(F)(F)F)C)NC(C1CCC(OC)CC1)=O 85062,C(C(C(=O)NC1CCC(C)(O)CC1)C(C)C)NC(c1c(CC)c[nH]c1)=O 85063,c1(C(N2CCC(CNC(COc3cn(C)nc3)=O)C2)=O)cccc(C(C)(F)F)n1 85064,N1(C(C2C(CNC(C(CCC)OC)=O)CCC2)=O)CCCC(C)(OC)C1 85065,C1(C(=O)NC(c2cccnc2)c2nc(C)no2)(CC)CCC(F)(F)CC1 85066,O=C1CCCCC(C(N2CCC2CNC(C2CC(O)C2)=O)=O)N1 85067,c1(C(=O)NCC(CNC(c2cc(F)n(C)n2)=O)OC)cc(F)c2ncccc2c1 85068,Cc1ccc(OCCOCc2cn(CC)nn2)cc1.c1(C(=O)O)nn(C)c(C(F)F)c1C 85069,c1(CC(=O)NC(C)Cn2cc(CNC(=O)CCN(C)C)nn2)ccccc1Cl 85070,N1(C(c2c(C)nn(C3CC3)c2)=O)CC2COCCC2(NC(=O)CC#N)C1 85071,c1(-n2ccc(CN(C(Cc3c(C)cccc3)C)C)n2)ccc(F)cc1F 85072,c1(CC)cc(C(=O)NCC2CC2NC(c2coc(C)n2)=O)oc1CC 85073,Cc1cccc(C(=O)NCC2(C)CCN(C(c3nc(C4CC4)sc3Br)=O)C2)c1 85074,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(C)=C(C)C)CC2C)c(F)c1Cl 85075,C1(NC(CC2C(C)(C)C2)=O)CC2(CCN(C(=O)CSCCN(C)C)C2)C1 85076,N1(C(CC2C(C)OC(C)C2)=O)CC2CC1CN2C(C1CCCC(O)C1)=O 85077,c1(OC)cc(Cl)c(C)cc1C(N1CCC1NC(=O)OC(C)(C)C)=O.C(=O)(CS)N 85078,N1(C(c2cc(C)ns2)=O)CCC(CNC(N)=O)CC1C 85079,c1(CN2CC3(CN(C(c4c(C)cco4)=O)C3)C2)cc(C)c(Br)cc1C 85080,N1(C(c2cc(OC)n[nH]2)=O)C2CCC1(CNC(=O)C(C)CC1CCOC1)CC2 85081,c1(C(=O)NC(CSC2CC2)C2CC2)cc(O)nc2c(Br)cccc12 85082,C1(NC(C(CCSC)O)=O)CC2CCC1(C(=O)NCc1nncn1C(C)C)C2 85083,C1(C)(CC)C=C(C(=O)NCC2CC2CNC(C2CCC(C(F)(F)F)CC2)=O)C1 85084,c1(C(=O)NC(CNC(C2CCC(C)O2)=O)(C)CO)ncccc1N 85085,Cc1cc(C)c(C(=O)NCC2CCN(C(=O)CN(C(=O)Cc3ccsc3)C)C2)[nH]1 85086,c1(CC(=O)N(C(C)COc2cnn(-c3ccccn3)c2)C)cc(CN(C)C)n[nH]1 85087,Cc1cc(I)c(C(=O)N(C2CCN(Cc3c(F)ccc(F)c3Cl)C2)C)cc1C 85088,C(CN=C(NCc1ccc(Cl)nc1)NCC1(CC(N)=O)CC1)C(C)(F)F 85089,C(=O)(CCCNC(=O)CNC(=O)C=CC1CCC1)OCC 85090,N1(C(C2(C#C)CCCC2)=O)CC2CC(O)C1C2NC(c1c[nH]nc1C)=O 85091,Cc1ccc(OCC(O)CNCCCC2CC2C)c(C)c1Br 85092,c1(NC(C2CC(=C)CN2C(C2(C)CC2)=O)=O)cccc(Br)c1OC 85093,C1(NC(c2cnc3ccsc3c2)=O)CC2CCC1N(C(=O)C1CC1)C2 85094,c1(C(=O)NCC2CCCN(C(C(CC=C)(C)C)=O)CC2)c(Cl)nc2ccccn12 85095,c1(C(N2CCOC3(CCSC3)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 85096,CC1CCCCC1(CNC(=O)C(F)(F)CC1CCCO1)NC(=O)COC1CCC1 85097,n1(CC(N2CC3CC(NC(CNC(CC)=O)=O)C3C2)=O)cc(C#N)c(O)nc1=O 85098,N1(C(c2cc(-c3cccs3)[nH]n2)C(=O)NCCC)CC(C(=O)OC)C(CC)C1 85099,N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(=O)C(C)(C)C 85100,C1(C(=O)NC2C=CCN(C(=O)CCC3CCCO3)C2)CC2CCCC(C1)C2 85101,n1(CC(=O)NC(C(C)NC(c2[nH]cc(C)c2)=O)CO)cccc([N+](=O)[O-])c1=O 85102,C1(C(=O)NC(C(=O)OCC)C2CC2)CCC(C)(C)N(C(c2cccc(CC)n2)=O)C1 85103,C(=O)(C(C)(CC)CO)NCc1cn(CCCC(=O)NCC2(CC)CC2)nn1 85104,N1(CC=CC(=O)OCC2(C)CC2)CCCCC1Cc1cccc(F)c1 85105,c1(SCC)nccc(C(=O)Nc2scnc2C2CC2)n1 85106,CON(CCC(=O)NCCCn1nccn1)C(=O)C(C)OCCOC 85107,C1(C(=O)OCC)CC(NC(=O)C(=O)Nc2cccc3nc[nH]c23)C2OC(C)(C)OC12 85108,N1(C(C(C2CCOC2)NC(C)=O)=O)CCCN(C(=O)CC2CCCC(C)(C)C2)CC1 85109,N1(C(C(=CC2CCCC2)C)=O)CCN(C(c2ccc(CF)cc2)=O)C(CCO)C1 85110,Cc1cc(NC(C2CCCC2C)=O)ccc1NC(c1c(Cl)nsc1Cl)=O 85111,c12ccc(c(F)c1)Cn1c-2nc(CCC2CCCCC2)n1.CC(F)(F)C1CCC1 85112,C1(CCCNC(c2onc(COC)n2)=O)CCCCN1C(c1coc(Br)n1)=O 85113,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CSCC(N)=O)N(C)C 85114,c12ccc(C)c(c1)NC2.Cc1cc(C)c(C(=O)N(C)CCOC(C)C)o1 85115,C12CCN(C(=O)CNC1=O)O2.C1(C(C)C)CCN1C(N)=O 85116,C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC(CC)NC(C1(CC(C)C)CCC1)=O 85117,CCC(Cc1ccc(N)cc1)C(=O)NCCCN(C)Cc1nnc(CO)o1 85118,c1(-c2c(C(C)C)n[nH]c2)nc(C2CCN(C(C)C)C2)nn1C(C1CCCCC1)C 85119,c1(C(C2CCCCC2)CCCC)cccc(Cl)c1.C1C(C2CC2)NC(=O)CO1 85120,C1(OC(=O)CC2OCCO2)CC2(CCOC2)C1 85121,c1(N(C)Cc2cc(F)ccc2Cl)ccc2nc(NC3CCNCC3O)[nH]c2c1 85122,C1(C(=O)NCC(C(=O)NCc2ccc(F)cc2)N(C)C)CSCC(=O)N1 85123,c1(C(=O)NCCCCNC(C2C3CNC(=O)C23)=O)cncc2ccsc12 85124,CC1=NOC(C)(C(=O)NCC(C2CC2)NC(c2cc(C)c(CC)s2)=O)C1 85125,c1(C(=O)NC(C)Cn2cnc3ccccc23)cnc2ncnn2c1O 85126,C1(CC)CN(C(c2cnc(C3CC3)[nH]2)=O)CCN1C(c1cccc(CC#N)c1)=O 85127,C1(C(=O)NC(CN(C)C(C2CCC23CCC3)=O)(CO)CO)CCCCCCC1 85128,C(CCN(C(=O)C(O)CC(C)(C)Cc1ccccc1Cl)C)(C(C)(C)C)NC(C)=O 85129,C1(NC(c2ccc(OC)cc2F)=O)CCCCN(C(=O)C(=O)NCC2CC2)CC1 85130,C1(C(=O)NCCN(C(=O)CCc2cccn2C)C(C)C)CCNC1=O 85131,C1(C(N2C(CNC(Cc3cn(CC)nn3)=O)C(C)CC2)=O)CCn2cncc2C1 85132,c1(C(C)(C)C)ncc(C(C)NC2(C3CCC3)CCC2)cc1Cl 85133,N1(C(C(CNC(c2ccc(C(N)=O)[nH]2)=O)O)=O)CCC2(CCCOC2)C1 85134,Cc1nccc(C)c1CCCCNC1CC(F)(F)CN1CC1OCCCC1(C)C 85135,C1(NC(C2(CCNC(=O)CC34CCCC3C4)CCC2)=O)CC2CC1C(O)C2O 85136,c1(NC)nc2ccc(C(N3CC(F)(CNC(=O)C(F)n4cccn4)C3)=O)cc2[nH]1 85137,N1(C(C(c2cn(C)nn2)OC)=O)CCCC(NC(=O)Cc2ccc(Cl)cc2)CC1 85138,C(=O)(C(C)(O)C(C)C)N(C)CC1N(C(c2cc(CCOC)on2)=O)CCCC1 85139,C1(=CC(=O)NC(C2CCCC2)CNC(C(CCSC)O)=O)CCCCC1(C)C 85140,c1(CN2CCCC(CNC(CCS(CC)=O)=O)C2)ccc2c(c1)oc(=O)n2C 85141,Cc1cc(OCCNC(=O)NCC2CC2F)cc(C)c1 85142,c1(CC(=O)C(=O)CO)ccnc(O)c1.C1(C(C(=O)NCC(C)C)N)CC=CCC1 85143,c1(C(N(C)CC2CCN(C(CC3CC(OC)C3)=O)C2)=O)c(C)noc1Cl 85144,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85145,C(=O)(C1CCOc2ccc(Br)cc21)NC1C(NC(c2c(C)c[nH]n2)=O)CCCC1 85146,C1(C)(CC)CC(NC(c2ccc(CO)cn2)=O)CN1C(=O)C=Cc1ccccn1 85147,c1(C)csc(C#N)c1.Cc1csc(C(CC)NC(=O)C(C)SC(C)(C)C)n1 85148,C1(CNC(CN(c2ncccn2)C)=O)CN(C(=O)CC2CCCCCC2)CCO1 85149,C(=O)(CC(C)CC(C)C)N1C(C(=O)OC)CC(n2cc(-c3c[nH]nc3OC)nn2)C1 85150,CC(C)C(C(C1CCCCC1)NC(=O)CC1CCCC1)NC(c1nc(Cl)cs1)=O 85151,C1(C(=O)N(CC(F)(F)Cl)C)(CC)CCN(C(c2cc(Cl)ns2)=O)C1 85152,C1(N(c2cccc(O)c2F)C(c2n[nH]c3c2CCC3)=O)CCC2(CCNC2)CC1 85153,C1(C#N)(C(N(C)CCc2nc(C(C)(C)C)no2)=O)CN(C(=O)OC(C)(C)C)C1 85154,N(C1CCc2c(Cl)ccc(Br)c21)S(c1c(C)cccc1Cl)(=O)=O 85155,C(=O)(C(C)(O)C(F)(F)F)NCC(C)NC(CCC#C)=O 85156,C12(C(=O)NCC3CCC(NC(C=NOC)=O)C3)CC(C)(C1)OC21COC1 85157,C1(N(C(CSC(C)(C)C)=O)C2CC2)COC(CNC(=O)C(C2CCOCC2)O)C1 85158,c1(C(=O)NCC2C(NC(C(=CC3CCCC3)C)=O)C2)c[nH]c2c(F)cccc12 85159,C1(C(=O)NCC(CC)(CC)NC(c2cc(OC)n(C)n2)=O)CC2(CCCC2)CO1 85160,c1(C(c2n(C(CC)C)nnn2)NCc2ccnn2C2CC2)ccc(C2CC2)cc1 85161,Cc1ncc(CCC(=O)N(C2CCN(C(C3CC3C(C)(C)C)=O)C2)CCO)o1 85162,CCC(CCC(=O)NCC1CC1CC(N1CC2(C1)CN(C)C2)=O)OC 85163,C1(C(CNC(C2C(OC)CCC2)=O)(C)C)CCN(C(=O)C(C)(C)C)CC1 85164,CC1CC(NC(c2c(CNC(=O)CN(C)C(N)=O)cnn2C)=O)CCN1C 85165,c1(C(=O)NCCCN(C)C(C2CCCN2C2CCOCC2)=O)ccncc1N 85166,c1(NC(C(C)(C)NC(c2cn(CC)nc2)=O)=O)cn(C)nc1C 85167,Cc1nocc1CCNC(=O)NC(c1ccccc1)C1(CC(C)C)CCC1 85168,c1(CC)[nH]ccc1C(=O)NC(C(N1CCC(CCOC)C1)=O)c1cccs1 85169,C(C)(CCCC(C)C)NC(CCC1CC(NC(C2C(=C)C2)=O)C1)=O 85170,CN=c1ccc(C(=O)NC2(C(=O)Nc3cnccc3C)CCCC2C)c[nH]1 85171,c1(SC)nc(C(N2CCC(NC(C3(C)CCCOC3)=O)C2)=O)c2ccccn12 85172,c1(CNC(C(c2ccoc2)NC(COC(C)C)=O)=O)c[nH]nc1O 85173,c1(-n2c(C3(OC)CCC3)nc(C3CC=CC3)n2)cc(F)cc(F)c1 85174,C1(C(=O)NCC2N(C(c3n(CC)ccn3)=O)CC(O)C2)CCC2(CCC2)CC1 85175,C=CC(C)(CC)C(=O)NC1C2CC1N(C(c1ccsc1OC)=O)C2 85176,C(=O)(C1(C)CCn2ccnc21)N1CCC(O)(CN(C)C(C2(C)CCCC2)=O)C1 85177,Cc1cc(=NC2C(C)C2C)[nH]c(N2CCOCC3(CCOCC3)C2)n1 85178,c1(C(N2C(C)CC(CNC(=O)C(C)(C)CC3CCC3)C2)=O)cnc(O)c(F)c1 85179,C1(C)(C(=O)NCCC(=O)NC)CCN(C(=O)C(C(C)O)NC(N)=O)C1 85180,c1(C(=O)NCC(F)CC)cccc(C2COC2)c1.C(CC(=O)NCCOCC)NC=O 85181,C(=O)(CC(=O)N1CC(CC(C)NC(=O)CC2C=CCC2)C1)NCC 85182,c1(C(=O)NC23CC(NC(C(C(C)C)OC)=O)(C2)C3)csc2ccc(Br)cc12 85183,C1(C(=O)NCCCOCC#C)CC(OC)CN1C(C1CCC(O)C1)=O 85184,CCCC(C)CC(=O)N1CCCC1C(N(C1(C(O)C(F)(F)F)CC1)C1CC1)=O 85185,c1(CN2C(CC(=O)NCc3cc(C)c(Br)nc3)COCC2)ccc(C#N)cc1F 85186,N1(C(C2C(C)CCO2)=O)CCC(C)CC1C(=O)NC1CC1.C12CCN(CC1)C2=O 85187,Cc1cc(C(=O)NCC(C2(O)CN(C(c3ccccc3F)=O)C2)(C)C)cc(C)n1 85188,C(C#Cc1cccnc1)NC(c1cccc(-c2ccco2)c1)c1n(CCC)nnn1 85189,Cc1ncc(CCC(N2CCN(C(=O)CCNS(C)(=O)=O)C3CC23)=O)c(O)n1 85190,C=C(C)CC(C(=O)N1CCCC1C(C)NC(=O)C(C)(C)C)c1ccccc1 85191,CC1(C)CC(C)(CNC(=O)CC2CCC(=O)O2)CN1C(=O)Cc1cc[nH]n1 85192,O=C(CC1CN(C(=O)COCCF)C1)NOC1CCOC1 85193,c12cccc(c1)S(=O)(=O)N2.CC(C)C#CC(=O)OCCC(=O)NC1CC1 85194,c1(C(=O)N(CC2CC2)CC2CCCCO2)cc2c(=O)cc[nH]c2s1 85195,CC1(C)CC(CO)CN1C(=O)C(c1ccco1)NC(C1CCCCC1)=O 85196,CC(C)(C#N)CCC(=O)NC1CCCC1CNC(c1cc(F)cc(F)c1O)=O 85197,C1(CNC(c2n(CCC)ncc2)=O)CN(C(=O)C=CSC)C2CC12 85198,C(Cc1cc[nH]n1)(C(=O)NCC1(C)CNC(=O)O1)NC(CCC=C(C)C)=O 85199,c1(C(=O)NC2C(C)CCN(C(C(C)c3cccs3)=O)C2)cc2ccc(F)cc2[nH]1 85200,C1(CNC(CC(C)F)=O)CCN(C(C2CC2c2ccncc2F)=O)CC1(F)F 85201,C(=O)(CCCC(N)=O)NCCC(C)NC(=O)COCc1nccn1C 85202,N1(C(C(F)=CCC)=O)CC2C3CCC(C2C1)N(C(=O)C(c1ccnn1C)C)C3 85203,c1(OC)nn(C)cc1C(=O)NC(C1CCCN1C(C1CCC1OC)=O)(C)C 85204,c1(C(N(CCCNC(=O)C=CC2CCOC2)C(C)C)=O)cc2c(o1)CCCC2 85205,Cc1c(C(C)N(C)C)cnn1Cc1ccccc1.C1(=O)C(=O)N(CCN(C)C)N1 85206,C=CCC(F)(F)CNC(=O)C(c1ccco1)NC(C12CC(CO)(C1)C2)=O 85207,c1(OC)cc(N)c(C(=O)NC2CN(C(=O)Cc3ccc(C)nc3)C2)cc1F 85208,N1(C(CCN(CCCCC)C)=O)CCN(C(C2(C)CC=CCC2)=O)CC1C 85209,C12(C(N3CC(CNC(CCCc4ccc(C)cc4)=O)C3)=O)C3CC(CC13)C2(F)F 85210,C(CC(C(C)C)NC(=O)CC1CC(C)C1)NC(C1(SC)CC(O)C1)=O 85211,N1(C(CCC(=O)N(C)C)=O)CCC12CN(C(=O)C(CC1CCC1)N(C)C)C2 85212,c1(C(=O)NCC(CC)NC(c2ccc3occc3c2)=O)cccn2cc(C)nc12 85213,N1(C(=O)Nc2cncc(F)c2Cl)CCn2c(C(F)(F)F)nnc2C1 85214,N1(Cc2c(C)n[nH]c2C)CC2CCC(NC(=O)CCCC(=O)N(C)C)CC2C1 85215,C(C(Cc1ccco1)C(=O)N(C1(CC)CC1)C)NC(c1n(CC)ccc1)=O 85216,c1(C(N2CCC(C(C(N3C(C(=O)OC)CC3C)=O)F)C2)=O)nnn(C)c1C 85217,c1(C(N(CC(C)NC(=O)CC(=O)NC2CC2)CC)=O)ccccc1OC(F)F 85218,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)N(C(c2cc(O)ccc2F)=O)CC1 85219,CC1CN(C)CC(CCC2CN(C(=O)Cn3cc(C4(C5CC5)CC4)nn3)C2)O1 85220,c1(C(N2C(CNC(C3CN(CC)C3)=O)CCC2)=O)cc(F)ccc1-n1ccnc1 85221,Cn1ncc2c(O)nc(=NCCC=CCNC(C3COC4COCC34)=O)[nH]c12 85222,c1(CC)cscc1C(=O)NCCN1CCC(NC(=O)CSCc2csc(C)n2)C1 85223,C(N=c1[nH]nc(C)o1)C1CCCC(NC(CC(=O)NC(c2nccs2)C)=O)C1 85224,N1(C(C(C)O)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)CCC1C 85225,CC(CC#N)C(=O)NCCCn1ccnc1.N1CCCCC1 85226,C1(CC(=O)N(CCN(C(c2c(SC)cncc2)=O)C)C)OCCOC1(C)C 85227,C(C(C)(C)CC(=O)NC1CCCN(C(=O)C(C(C)C)n2cnnn2)CC1)OC 85228,c1(C(=O)NCCC(=O)N(C2CCN(CC)C2)CC)cc(C(F)F)ncn1 85229,CC1(CNC(=O)CCS(N)(=O)=O)CCN(C(=O)CSc2ccc(C#N)cc2)CC1 85230,C(CCCCC(=O)NC1CC1CNC(c1cc(Br)nn1C)=O)SC 85231,c1(-n2cc(CCCCC)nn2)ccccc1C(=O)NC1CC2CC2(C)C1 85232,Cc1ncc2c(n1)CNC2C(=O)N1CCC(O)C(C)C1 85233,C(=O)(CC1=CCCC1)N(C1CC2CCC1O2)C(=O)CC1C=CC(CO)C1 85234,CCCCC(CNC(=O)C(C)N(CC)CC)NC(c1csc(C)c1C)=O 85235,c1(NC(CC)=O)ccccc1C(=O)NC1CC1NC(=O)OC(C)(C)C 85236,C1(C)(CNC(c2cccc(N(C)C)c2)=O)CC(F)(F)CN1C(=O)COCCF 85237,CN1CCC(C)(C(=O)NC2(c3ccccc3)CCN(C(=O)C(F)(F)C(F)F)C2)C1=O 85238,N1(CC(N2CCC(CN(C)C(c3sncc3Br)=O)C2)=O)C(=O)CCC1=O 85239,C(=O)(CCCC(C)(C)C#N)NC1CC(NC(c2c(CC)noc2)=O)C12CCC2 85240,CC(C(C)C(=O)NOCCCO)NC(c1cnn2cccc2c1)=O 85241,C#CCCCCC(=O)NC(CO)C(=O)NCCCC1CCC1 85242,C=CC1CCN(C(=O)C(C2CC=CCC2)NC(C2CCCN2C=O)=O)C1 85243,N1(C(c2ncn(CC)n2)=O)CC(CNC(c2ccc(C(F)F)s2)=O)C(O)C1 85244,N1(C(CN2C(C)CC2)=O)CCCCC1CN(C(=O)C(F)(F)CN(C)C)C 85245,CN1CC(C(N2CCCC2C2(C(N3CC=CC3(C)CO)=O)CC2)=O)NC1=O 85246,C1(CNC(C=CC=CC)=O)CCC12CCN(C(c1coc(C(C)(C)C)n1)=O)CC2 85247,N1(C(c2cnc(C(C)C)s2)=O)CC2CCCC2(CNC(=O)CCF)C1 85248,N1(C(c2c(CC)cno2)=O)CC2CCCC(C1)N2C(=O)CCn1cccn1 85249,N1(C(c2n(CC)c(O)nc2)=O)CC2CCC(N(C(=O)CCSC)C)C2C1 85250,C(C(C)N=c1[nH]c(=NCCOc2ccc3c(c2)COC3)[nH]c2c1CCC2)OC 85251,O=C1CCC(C2(C(N3CC4CCC3CN4C(=O)Cc3ccon3)=O)CCC2)CN1 85252,Cc1nc(O)nc(C)c1CC(=O)NCCC1CCC(NC(=O)CC2CC2(Cl)Cl)C1 85253,C(=O)(C#CC(C)(C)C)N1CCC(N(C(COC)=O)CCO)C1 85254,c1(C(=O)NCC2(C)CCCN(C(c3ccc([N+](=O)[O-])s3)=O)C2)ccc2ccoc2c1 85255,C1(C(=O)NC(CNC(C(COC)(C)C)=O)C)CCc2ccccc2O1 85256,C1(C(=O)NCC2C3CN(C(c4c(Cl)cn(C)n4)=O)CC32)CCCCS1(=O)=O 85257,N1(C(=O)OC(C)(C)C)CC2(CC(NS(=O)(=O)NCCCF)CO2)C1 85258,C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCC1NC(=O)CCN1CCOCC1 85259,c1(C(=O)NC(C=CC(=O)N(CCOCC=C)C)(C)C)cccc(F)c1 85260,CC1N(C(C2CC2C2CN(C(=O)CNC=O)C2)=O)CCCC12CCC2 85261,N1(C(c2c(OC)cncc2)=O)CC(C2CCCN(C(=O)C(C)(C)C3CC3)C2)C1 85262,c1(NC(=O)NCc2nc(C(C)OCC)sc2)ccc(C(C(C)OC)(C)C)nc1 85263,C1(NC(c2ccc(F)c(OC)c2F)=O)CC2(CCN(C(=O)CC3CC(=O)C3)CC2)C1 85264,c1(C(=O)OC)cnc(C)cc1N1CC=CC(NC(=O)C(C)OCC(C)C)C1 85265,C1(NC(c2c(C)nc(C3CCC3)o2)=O)CC2CC(C1)N(C(C1CCCSC1)=O)C2 85266,c1(C(N2C(CNC(=O)CN3CC4CC4C3)CC2)=O)c[nH]c2c(F)cccc2c1=O 85267,c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)C(F)C2)=O)nc2ncc(CCO)cn2n1 85268,C1(NC(CCC#CC)=O)CCN(C(=O)C(C)CC2CCCCC2)CC1O 85269,c1(CNC(C2CN(C3CCOC3)C2)=O)c[nH]nc1C1CCC1.C12CCN1C2=O 85270,C12(COC)CCC(C(N3CC(CNC(=O)C=CC4CC4)C3)=O)(CO1)C2 85271,C1(OC)CC2(C1)CC(C(N1CCCC1CN(C(=O)Cc1ccsn1)C)=O)C2 85272,c1(C(N2CC(C)(NC(c3c(CC)onc3)=O)C2)=O)ccnc(Cl)c1O 85273,c1(C(=O)NCC2C(NC(C(COCC)C)=O)C2)cc(F)c2nc(C)cn2c1 85274,CCCC(C(=O)OC)C(=O)NCC1CCC(C(=O)NCc2nc(C)ccc2O)C1 85275,C1(C)(NC(c2c(C)[nH]nc2C(F)F)=O)CCN(c2ccnc(-c3nccs3)n2)CC1 85276,Cc1ccnc(C)c1C(=O)NC1CC(C(F)F)(NC(C2CC23CC(C)(C)C3)=O)C1 85277,N1(C(C(c2scc(C)n2)C)=O)CCCC2CN(C(c3ccsc3C)=O)CCC12 85278,N1(C(CC(C)=C(C)C)=O)CCN(C(=O)C(F)C(C)(C)O)C(CC(C)(C)C)C1 85279,c1(C(=O)NC(c2ccsc2)CNC(=O)CSC(F)F)cccn2nnnc12 85280,C12(CNC(C(CCSC)O)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C=CCF)C1)O2 85281,N1(C(Cc2c(C)ncs2)=O)CCC(C)(C)CC1C(N1CCN2CCC1C2)=O 85282,CCCCC(C)CCC(=O)N1C(C(=O)NCc2ncccn2)CCC1C 85283,C12(C(N3CCC(CCNC(C4CN5CCC4CC5)=O)C3)=O)CCC(CC1)CO2 85284,N1(Cc2scc(-c3occ(C(=O)O)c3)c2)CCC(O)C(F)(F)C1 85285,CCC(C)CCCCC(=O)N1CC(OCCNC(c2c(F)cc(O)cc2F)=O)C1 85286,C1(C)(CNC(C2CN(C(C)=O)C2)=O)CN(C(=O)CN2CC3C=CC2C3)CCO1 85287,C1(CC(=O)N(CC(C)OC)C)CC(NC(=O)CCC(=O)N(C)C)C1(C)C 85288,c1(CNC(=O)NC(c2nc(C)sc2C)C(C)(C)C)ccc(C)c(Br)c1 85289,N1(C(C2CCN(C3CC3)C2)=O)CCCCCCC1C(N1CCC(F)(CF)CC1)=O 85290,C1(C(=O)NC(CC)(C)CNC(c2nccn2C)=O)CCOC(C)C1 85291,C1(CN(C(=O)Cc2ccco2)C)CCC(=O)N1.C12(CC1)C(=O)NC2 85292,CC1(C(=O)Nc2ccns2)CC12CCN(CC(N1Cc3ccccc3C1)=O)CC2 85293,c1(CC(=O)NC(C2(C(=O)NCCNC(C3CCOC3)=O)CC2)C)ccccc1 85294,c1(-c2c(=O)cc(C)n(C3CCS(=O)(=O)C3)n2)ccc(C)c2ncccc12 85295,N1(C(c2nc(N3CCOCC3)ncc2Br)=O)CC2(CCOC2)c2ncccc21 85296,c1(C(N2C(C=C)CCCC2)=O)coc2c1CN(C(=O)CCc1nncn1C)C2 85297,C1(NC(C2CC(C(=O)OC)C2)=O)CN(C(=O)C2=CCSC2)CC1C(F)(F)F 85298,N1(CC(=O)NCC(n2cc(-c3cc(C4CC4)no3)nn2)C)CCC(=O)CC1 85299,C1(C(=O)NC(CNC(C(Cc2ccc(OC)cc2)C)=O)(C)C)CCN(C)S1(=O)=O 85300,C1(NC(CSCC=C)=O)(CNC(=O)C(N2CCN(C)CC2)C)CCC12CCC2 85301,N1(C(c2cc(CC(C)C)n[nH]2)=O)CCC(C)C(NC(=O)CNS(C)(=O)=O)C1 85302,c1(OC)ccc2oc(C(N3CCCC3C(C)NC(=O)COCC(F)F)=O)cc2c1 85303,c1(NC(CC)COC)ncnc(NCC(C(C)(C)C)OC)c1C 85304,C12(C(=O)NCCNC(C3C(Cl)(CCOC)C3)=O)CC(CN1C1CC1)C2 85305,O(N(C)C(=O)CC(C)(C)N(C(=O)C(C)C1(O)CCC1)C)CC=C 85306,Cc1ccsc1CC(=O)NC1(CNC(=O)C(C)CN(C)C)CCOC1 85307,C1(NC(CN(C(c2n(CC#C)ccc2)=O)CC)=O)CCCCCC1F 85308,C1(c2scc(C)n2)CN(C(=O)Cn2cc(CN(C)C)nn2)CCO1 85309,N1(C(CCOCC#C)=O)CC(NC(=O)C=Cc2ccccc2F)CCC1C 85310,CC1(O)CCN(C(=O)CCCc2ccccn2)CC1(O)c1ccccc1 85311,c1(N2CC(CCNC(C3CCSC(C)C3)=O)(OC)C2)ncnc2ccc(Cl)cc12 85312,C(C)(C)(CCCNC(C1NC(=O)CC1C)=O)NC(COCc1nnc(C)s1)=O 85313,C1(C)(C(=O)NCC(CCC)O)CCN(C(C)=O)C1 85314,CCCCC(F)(F)C(=O)NC(CC1CC2C=CC1C2)C(=O)NOCCCC1CC1 85315,C1(S(C)(=O)=O)(C(N(CCNC(=O)Cn2c(C)c(C)sc2=O)CC)=O)CCOCC1 85316,c1(OC)c(C)cc(C(N2CCC(NC(C3CC3C(N)=O)=O)C2(C)C)=O)cc1C 85317,C(=O)(NNC(=O)c1ccc(C)o1)NC(CCCC)=O 85318,C1(N(C(c2c(CNC(Cc3cc(C)[nH]n3)=O)noc2)=O)C)CCCC1(C)O 85319,c1(OC)ccc(C=CC(=O)NC2CCCC2NC(=O)C(c2cccn2C)=O)c(C)c1 85320,C(=O)(C(CCC1CC1)NC(=O)C(F)C1CCCC1)N(C)CCOCCO 85321,C1(C(N(C23CCC(CC2)CC3)C)=O)CC2C=CC1N(C(c1ncccc1N)=O)C2 85322,O(P(C)(=O)CN1CCCCC1)c1c(OCC)cccc1 85323,c1(C(=O)NCCN(C(=O)CC2CCCCC2C)CCOC)c(C)[nH]c(C)c1C 85324,O=C(C(F)C1=CCCCC1)N1CCCCC1CNc1nc2ccc(O)cc2s1 85325,C1(OC)(CNC(=O)CCc2cncs2)CN(C(C2CC2Sc2ccccn2)=O)C1 85326,N1(C(C(C)=CC#N)=O)CCOCC(C(=O)NC(C)CNS(C)(=O)=O)C1 85327,C1(CNC(C=NOC)=O)CN(C(c2cccc3c2CCC3)=O)C2COCC2O1 85328,Cc1nc(C)c(C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)o1 85329,N1(C(C(CC)NC(N)=O)=O)CC(C(N2CC(CC3CCC3)C2)=O)CC(C)C1 85330,CCC(C)C(C(=O)NC(CN(C)C)CC)NC(=O)C(CN(C)C)NC(C)=O 85331,C(=O)(C(C)(CC)OC)NCC(CC=C)NC(c1ccoc1Br)=O 85332,c1(CC(C)C)cccc(CNC(c2nnnn2C2CC2)C2CC=CC2)c1 85333,Cc1cnc(C(=O)NC(C)C(C)C(=O)NCc2cccnc2O)c(F)c1 85334,CC(C)CC(C)C(=O)NCC(=O)NCC(=O)N(C1CCCCOC1)C 85335,c1(CN2CC(C(N3CCN(C(=O)OC)CC3)=O)C2)cc[nH]c(=NC)c1 85336,C1(NC(C=CC=CCC)=O)CC(CNC(c2cc(CC)cc(Cl)c2)=O)C12CCC2 85337,C(=O)(CCCC(C)C)NC1CN(C(CS(CC)=O)=O)CC1CC1CC1 85338,C1(CC(=O)NCc2ccccc2CNC(c2ccncc2O)=O)CCC1C1CC1 85339,Cc1c(CN2CCC(O)(C(N3CCC(CN)C3)=O)CC2)cccc1Cl 85340,CC(CCC(C)(C)C)C(=O)N1CC2C(c3cn(Cc4cc(C(F)F)no4)nn3)C2C1 85341,N1(C(COC(C)C)=O)CCC2CCCC12CNC(=O)C(F)(F)CO 85342,C(=O)(C1CSc2ccccc21)N(CCCN(C)C(c1n[nH]cc1Br)=O)C 85343,C(CC(C(=O)NCCCCC1CC1C)N(C)C)NC(CC1C(CC)C1)=O 85344,N1(C(c2cscc2Br)=O)CCCC(C2CC2NC(C2(F)CCCC2)=O)C1 85345,c1(C(N(C2CN(C(C3CC(OC)C3)=O)C2)CC)=O)nc2c(cc1Cl)OCCO2 85346,N1(C(=O)NCC(C)N(C(=O)CCCNC(=O)C2CC2)C)CCCC1C1(C)CC1 85347,N1(CC(C2CC2)OC)CCC(C(C)NC(c2ccnn2-c2ccncc2)=O)CC1 85348,c1(CN2CCCC(C(=O)NC(c3nnc(C)o3)C)C2)ccc(F)c(Br)c1F 85349,N1(C(=O)CC2CCCO2)CCC2CN(C(=O)COCC(F)(F)F)CC2C1 85350,C1(NC(C(CC)OCC)=O)CC2(C1)CC2C(=O)NCc1ccc(Cl)cn1 85351,c1(SCC)ccc(C(C)NC(C23CC2CN(CC(C)O)C3)=O)cc1 85352,CC(N=c1nc[nH]n2cccc12)C1CN(C(C2(CCF)CCOCC2)=O)CCO1 85353,c1(C(N(CCCNC(c2c(F)ccc(C)n2)=O)C)=O)cn(C)c2ccc(F)cc12 85354,c1(NC(C)=O)cc(C(=O)NC2CCCC2CNC(=O)C(F)SC(F)(F)F)ccn1 85355,C(=O)(CC(C)CC(C)(C)C)NCc1cc(C(=O)NCC(C(C)O)(C)C)n(C)n1 85356,CC1(C)C(C(=O)NCCCc2ccc(-c3nn[nH]n3)cn2)C1(F)F 85357,CC1(C)CN(C(c2ccnnc2O)=O)CCC1C(N1C(CO)CC1CO)=O 85358,N1(C(c2cn(-c3ccccc3)nn2)C)Cc2cccc3c2C(C3=O)C1 85359,c1(C(=O)OCC)sc2cnccc2c1NC(c1[nH]nc(OC)c1Br)=O 85360,c1(OC(C(=O)NCC2(OC)CN(C(=O)Cc3csnn3)C2)C)ccc(C)cc1C 85361,CC(C)CC(C)CC(=O)NCC(C(=O)NCP(C)(C)=O)C(C)C 85362,N1(CCO)CCN(CCC(F)(F)F)CC1.N1(C(C(=O)N)=O)CCCC1C1CCCC1=O 85363,c1(C(=O)NCCC2CCN(C(C(CC)OC)=O)CC2)cc2c(C)ccc(F)c2o1 85364,N1(C(C2C3(CCN(C(c4ncc(OC)cn4)=O)C3)C2)=O)CC(O)(C2CCC2)C1 85365,Cc1cc(C(=O)NCC2(O)CN(C(c3cccc(Cl)c3C)=O)C2)[nH]c1C#N 85366,c1(C(N2CC(CNC(=O)C(F)=CC3CC3)OCCC2)=O)cnc2c(c1)CCOC2 85367,c1(C(=O)NCC(CO)NC(=O)CC23CCCC2C3)ccc(-c2cn[nH]c2)cc1 85368,O=C(C1CCOc2ccccc21)N1CCC(c2nn[nH]n2)(C(F)(F)F)C1 85369,c1(C(=O)NCC23CN(C(C=COCC)=O)C(C2)CO3)cc(=O)n2nccc2[nH]1 85370,CC1CN(C(=O)C(CCF)NC(C2CCC(O)C2)=O)CCS1=O 85371,C1(NC(c2c[nH]nc2C2CC2)=O)CC1C1CCCN(C(=O)C(F)=CCCF)C1 85372,C1(SC)CCCN(C(C2CCC(NC(=O)OC(c3ccc(C)cc3)C)CC2)=O)C1 85373,Cc1cccc(SCC(=O)NC2CCN(C(=O)CC(C)n3ccnc3)C2)c1 85374,CCCC(C)C(CO)NC(c1cnn(CCNC(=O)CC2CNC(=O)O2)c1)=O 85375,CC(C)CC(C(=O)NC1(CCO)CC1)NC(=O)Cc1ccn(C(C)C)n1 85376,c1(SC)cccc(C(N2CCCCC2CN(C(=O)C(Cl)=CCl)C)=O)n1 85377,C1(NC(c2nncc(C)c2)=O)CN(C(C2(O)CCCC2)=O)CCC1CO 85378,C12(C(=O)NC3CCCN(CC)C3)CCC(CC1)N2Cc1csc(C2CCCO2)n1 85379,c1(C=O)cc(C)cc2ccoc12.C(C(C)(C(=O)NCCC(F)CC1CCC1)O)OC 85380,c1(C(=O)NC(CN(CC(=O)N(CC)CC)C)C)cc2nc(F)ccc2o1 85381,C#CC1(NC(C2COCCN2C(c2c[nH]nc2Cl)=O)=O)CC2CCCC12 85382,Cn1nnc2c1CCC(C(N)=O)C2.C12CCCN(CC1)c1ccc(nn1)NC2=O 85383,c1(C(N(C2CN(C(C(C)(C)OCC)=O)CC2F)C)=O)cc2c(nc1O)CCOC2 85384,C(=O)(C(C)(C)CC1CC1)N1CC(O)(CN(C)C(c2cocc2C(N)=O)=O)C1 85385,CCCCCCn1cc(CNC(=O)C(C)SCCC2CC(N(C)C(C)=O)C2)nn1 85386,C(=O)(CCCCCC(C)O)N1CC(NC(c2c(C)[nH][nH]c2=N)=O)C(C(F)F)C1 85387,C1(O)(CN(C(=O)COc2ccon2)C)CCN(C(=O)COC2CCCC(C)C2)CC1 85388,C1(O)(C(N2CCCC(CNC(C(C)(C)OC)=O)C2)=O)CN2CCC1CC2 85389,C1(CC(=O)N(C)Cc2c(C)occ2)CN(C(=O)C(C)(C)CN(C)C)CC12CC2 85390,C1(C(=O)NC2(CNC(CCc3c(C)noc3)=O)CC2)CCN(C)CC1 85391,c1(-c2nc(NC(N3CC(Cc4cc(Cl)ncc4F)C3)=O)sc2)ccc(F)c(Cl)c1 85392,C(=O)(CCC(=O)NC(C1CCCN(C(=O)CSCC(F)(F)F)C1)C)NCC 85393,n1(C(C(=O)NCCN(CC)CC)C)cc(SCCCNC(C)(CC)CNC(N)=O)nn1 85394,c1(C(C2CCCNC2)N(C(=O)NCC2CCCCC2)CCO)ccc(F)cc1 85395,C1(CNC(=O)CO)(NC(c2cccn2Cc2ccccc2)=O)CCOC1 85396,c1(C(=O)NCC2C(NC(C(CCC)(C)O)=O)C2)ccc(Br)c2ccccc12 85397,C1(CNC(C(CC)C)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1(F)F 85398,c1(OC)c(C(N2CC(O)(CCNC(=O)Cn3cc(C)cn3)C2)=O)occc1=O 85399,c1(N2CCCC(NC(C3CC(O)C3)=O)C2)ncnc2c(F)cccc12 85400,Cc1ncc(C(=O)NCC2CC2NC(c2cc(O)nn2C)=O)n1C(F)F 85401,N12CCN(CC1)CCCc1ccc(nc1)OC(C)C2=O.C=CCCOCC 85402,N1(C(c2c(C)c[nH]n2)=O)CCC2(CC1)OCCC2NC(=O)C1=CCCOC1 85403,N1(C(COCC(C)(C)C)=O)CCC(NC(C2CCC3CC3CC2)=O)C(F)C1 85404,C=CCC(CC)C(=O)NCC(CNC(=O)Cn1nc(Cl)ccc1=O)C(F)(F)F 85405,N1(C(C2(C(C)=O)CC2)=O)CCC2C(NC(c3sc(C)nc3C)=O)C2C1 85406,c1(C(N(C2CCN(C(CS(=O)(=O)NC)=O)C2)CCO)=O)onc2c1CCCC2 85407,C1(NC(=O)CCCF)CC2CCC1CN2C(=O)Cn1cnnc1 85408,c1(CC(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2O)c[nH]c2cccc(Cl)c12 85409,C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(c2c(C)cnn2C)=O)CCC1 85410,c1(OC(C(=O)NCC2CN(C(C3C(C)C3C)=O)C2)C)ccccc1C(C)(C)C 85411,C1(C=O)CCS(=O)CC1.C12OCCC1CCCNN(CCC)CCNC2=O 85412,C12(CCNC(C=CSC)=O)CCC(C1)N(C(c1ccco1)=O)C2 85413,CC1(C)CCCCCC1NC(=O)CN(C(c1cc(F)cc(F)c1)=O)C1CC1 85414,Cc1ccc2c(c1)CCN2C(=O)CC(C(C)C)NC(=O)Cn1ncccc1=O 85415,c1(C(=O)NCC2CCC(NC(C3C4COCC34)=O)C2)ccc(F)cc1OC(F)F 85416,C1(CC(=O)NCC(CNC(C(C)Oc2cccc(C)c2)=O)CO)CC2(CCO1)CC2 85417,N1(C(CC(C)C(C)(C)C)=O)CCCC2(CCCN2C(c2cc(C3CC3)ns2)=O)C1 85418,c1(NCC2C(C(=O)NC3CC(OCC)C3)C2)c(F)cc(C#N)cc1[N+](=O)[O-] 85419,C1(NC(C2(C(C)(C)O)CC2)=O)CCCCN(C(=O)CC(O)c2ccccc2)C1 85420,C1(NC(=O)Cc2ccncc2)CC2CCC(C1)N2C(c1cccnc1Cl)=O 85421,CCCCCCCC(C)NC(=O)C(CC)N(C(=O)C(C)(C)OC(C)C)C 85422,C1(NC(=O)CCc2nc(-c3nc[nH]n3)no2)C2CC1CN(C(C1CC1CF)=O)C2 85423,N1(C(C2(NC(C)=O)CCCC2)=O)CCC(NC(C2NC(=O)OC2C)=O)CC1C 85424,C1(C(N2CC(C)C(NC(=O)CC3=CCOCC3)C2)=O)CCc2nnc(O)cc2C1 85425,c1(C(=O)NC2C(CNC(C(N3CCCCCC3)C)=O)C2)ccc2oc(S)nc2c1 85426,C1(C(=O)NC(N2CC3CC2(CC2(CO)COC2)C3)=O)C2CC3C(C2)C13 85427,C1(O)(N(C(CCOCCN(C(=O)Cn2ccnn2)C)=O)C)CCOCC1 85428,c1(C(=O)N)conc1C(C)NC(C1CS(=O)C1)=O.N(CCC1CC1)CC 85429,C(C)(C)(CC(C)NC(=O)CC1CCC(NC(=O)C(F)CC2CCOC2)C1)OC 85430,C1(CNC(=O)CC2CCC2)CCC(C(=O)NCCC(O)C2CCCC2)CC1 85431,CC(CC(C)N=c1[nH]c(C(C)(C)C)nc2[nH]cnc12)NC(c1cnn(C)c1)=O 85432,S(=O)(=O)(c1ccc(C(=O)O)cc1)NC1CN(C(=O)Cc2cc(Br)cs2)CC1O 85433,C1(C(C)C)CN(C(=O)CN2CC3CC3C2)CCN1C(=O)C(=O)Nc1ccccc1 85434,C(=O)(C#CC(C)(C)O)NCC1N(C(C(c2cccc(Cl)c2)C)=O)CCC1C 85435,CC1C(NC(=O)CCF)CCN1C(c1n[nH]cc1Cl)=O 85436,c1(C(N2CC(CCCCNC(=O)C=CC=C(Cl)Cl)C2)=O)coc2c1CS(=O)(=O)C2 85437,N(C(=NCCSC(C)C)NCC(c1ncc(F)cc1F)(C)O)C(c1ccccn1)C 85438,N1(C(C2C(C(N(CC#C)C)=O)C2)=O)CCCC1CCCNC(C1CC(C)=NO1)=O 85439,c1(C(N2CCC(OCCO)C2)C(=O)NCCSC)oc2ccccc2c1Cl 85440,c1(ON=CC(=O)NC2CCN(C(C(C)C#N)=O)C2)c[nH]c2ccccc12 85441,N1(C(C(C2CCC2)OC)=O)CCC(NC(c2csc(Cl)n2)=O)CC1 85442,Cc1ccccc1C=CC(=O)NC1(CC=CC(N2CCOCC(O)C2)=O)CCC1 85443,CC(C)(CC(=O)N1CCCCC1C(N)=O)NC(c1coc(N(C)C)n1)=O 85444,N1(C(C=Cc2ccc(C)o2)=O)CCC(C)(CNC(C2CC(=O)N(C)C2)=O)CC1 85445,CC1(CNC(=O)CC2(C)CC2(F)Cl)CCN(C(c2cnoc2-c2cccs2)=O)C1 85446,C1(C(=O)NCCC(=O)NCCCN(C(C2CCOC2)=O)CC)CN2CCN1CC2 85447,C(=O)(C1CCCc2nc(C)[nH]c21)N1CCCC(N2CCN(C(C=C)=O)CC2)C1 85448,c1(C(=O)NC(c2ccc(Cl)cc2)C2CC2)cc(C2CCCCC2)nc2ccc(Br)cc12 85449,N1(CC(=O)Nc2cc(OC)c(F)cc2)CCn2nnc(Br)c2C1 85450,c1(C(N2CC3(CCCCN3C(c3cnns3)=O)C2)=O)ccc2ncccc2n1 85451,N1(C(CCN(C)CCO)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C2CCCCC12 85452,N1(C(CC(C)OC)=O)CCOCC(C)(CNC(c2c(C)cc(C)nc2C)=O)C1 85453,CC1CC(NC(=O)CC(=O)NC2CCCC2)CN(C(c2cc(C(F)F)on2)=O)C1 85454,c1(C(N2CC(N(C(=O)COCC3CCC3)C)C2)=O)cccc(CF)c1 85455,C1(CNC(N(CCC#CCC)C)=O)CCC(F)CC1 85456,C(=O)(C(O)C(C)c1ccc(C)cc1)NCCN(C(=O)CCN1CCCC1)CCC 85457,CC1(C)CN(C(=O)CCC2CCCN(C(c3ccc(CF)cc3)=O)C2)C1(C)C 85458,Cc1cc(C(=O)NC2CCCN(C(=O)Cn3ccnc3)CC2)cc(C)c1 85459,c1(CNC(N(C(C2CCCC2)C)C)=O)ccc2nc(O)[nH]c2n1 85460,C1(CNC(c2c(C)cn(C(C)C)c2)=O)C(C)CCCN1C(c1ncccc1F)=O 85461,C(=O)(C1CCc2c[nH]nc21)CCN1CCCC(C(=O)NCCC)CC1 85462,N1(Cc2nc(C)on2)CCC2(CCCN(C(=O)CCc3ccncc3)C2)C1 85463,CCC(CC(C)C)C(=O)NC(c1nocc1C(=O)N1CC(C)(O)CO1)C 85464,CCCC(CCCNC(=O)Cn1nnc(C)n1)NC(=O)C(CO)c1ccccc1 85465,C(=O)(C1=C(F)CN(C(C2CC=C(C)CC2)=O)CC1)NC(CC)C1CCC1 85466,CN=C(NC1CCC2CC2CC1CC)N1CCc2nc(C(=O)OCC)sc2C1 85467,C(=O)(C(CO)C(C)(C)C)NCCCC1N(C(c2cc(C)cc(C)c2)=O)CCC1 85468,N1(C(C(N2CCCC(C)C2CCC2CC3CCC2C3)=O)=O)CCN(C)CC(C)C1 85469,N1(C(C2(N(C(c3cc(C(C)=O)[nH]n3)=O)C)CC2)=O)CCC(O)(C(F)F)C1 85470,CC(CN=c1[nH]c2c(c(=NCc3cocn3)[nH]1)CSC2)Oc1ccccn1 85471,c1(NC(C2CN(C(COCC(C)C)=O)C2)=O)cnn2c1OCCC2 85472,C1(C(=O)OCC)CCN(C(=N)Nc2cccc(C3COCCN3)c2)CC1 85473,c1(C(C)=O)cc(C(=O)NCC2CCCC(CNC(=O)CCc3cscn3)C2)n(C)c1 85474,C1(C(N2CC(O)(CNC(Cc3cc(COC)on3)=O)C2)=O)CCCC(=O)N1C 85475,C1(COC)(OCC(F)F)CN(C(=O)C(=O)Nc2ccc(-c3csc(C)n3)s2)C1 85476,C(=O)(C(C)C(C)(F)F)NCC1(F)CC(NC(CN(S(CC)(=O)=O)C)=O)C1 85477,C1(CN(C(c2c(C)c[nH]n2)=O)C)CN(C(=O)C(CO)c2ccccc2)CCO1 85478,N1(C(C=CC)=O)C2CCC1CC(F)(CNC(C1(c3ccncc3)CC1)=O)C2 85479,c1(C(=O)NCC(CO)NC(C(COC)N(C)C)=O)ccc(=N)[nH]c1 85480,c1(OC)nc(C(=O)NCC2CC(C)N(C(c3ccc(Cl)nn3)=O)C2)cc(O)n1 85481,C1(NC(C(CC)N2CCCC2=O)=O)CC2C1CCN2C(c1cc2n(n1)CCC2)=O 85482,c1(C(=O)NC(CCCC)CNC(=O)C(C2CC2)OCC)occc1S(C)(=O)=O 85483,C(=O)(CCC(=O)NC(C1CN(C(=O)C=CC2CCCC2)CCO1)C)NCC 85484,c1(OC)cc(OC)nc(C(N2CCN(C(=O)CCn3cccn3)CC2)=O)c1 85485,Cc1cc(C(=O)NC(CNC(=O)CC2CCCS2(=O)=O)C(C)(C)C)cc(C#N)c1 85486,CC(C)C(F)(CNC(C1(C)CCCCCC1)=O)C(=O)NCC(C)(CO)O 85487,N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)C2=CCN(C)C2)C(CC)C1 85488,c1(C(C)C)ncc(Br)c(N2CC(C(C)NC(=O)CC3CC3)C2)n1 85489,C(=O)(C1=CCN(C(=O)Cc2cccc(Cl)c2F)CC1)NCC1CC(C)OC1 85490,CN1CCCC(O)(CC(=O)NCC2CCC(NC(C34CCC(CC3)CC4)=O)C2)C1 85491,C(=O)(CCCCC(F)(F)F)N1CC(N2CCN(C(CC)=O)CC2)OC(C)(C)C1 85492,c1(C(N2C(C)CC(NC(c3ccc(C(F)F)nc3)=O)C2)=O)cnc2cccnn12 85493,C1(CNC(C2(Cl)C(C)(C)C2)=O)(NC(=O)C(O)c2ccsc2)CCC(F)(F)CC1 85494,c1(C(=O)NC2C(NC(=O)CSC3CCOC3=O)CCC2)ccc(C(F)(F)F)nn1 85495,c1(CC(=O)NC2(C)CCN(C(c3oc(CC)c(C)c3)=O)C2)ccc(F)cc1C 85496,C1(N(C(=O)Cc2nncs2)C)CCC(NC(=O)NC(c2cnnn2C)C)CC1 85497,C=C(F)C1(CC(=O)NC(c2ccccn2)C(N2CCC(N(C)C)CC2)=O)CCC1 85498,C1(CC(=O)NCC(C)OC2CCCCC2)CN(C(C2CCSC2)=O)CC12CC2 85499,c1(CC(=O)NCC2CCN2C(c2cc(F)c[nH]2)=O)nc(F)c(F)cc1F 85500,CCC(C(=O)NCCCN(C(=O)CSCC(F)(F)F)C(C)C)Nc1nc(C)cs1 85501,C(CC(=O)NCCCNC(=O)Cn1cnc(C)cc1=O)(C1=CCCC1)NC(C)=O 85502,c1(C(N2C(CC)C(C(=O)N(C)Cc3cnn[nH]3)CC2)=O)cccc(F)c1O 85503,n1(CC)ccc2nc(NC3CC(NCc4ccc(O)c(I)c4)C3)ncc12 85504,c1(C(=O)NCC2(CNC(=O)Cn3cc(CO)nn3)CC2)cnc2nccn2c1 85505,C1(CC(=O)NCCN(C)C(c2ccc(C(=O)N(C)C)cn2)=O)CC(=O)NC(=O)C1 85506,C1(C(=O)NC2CCC(NC(c3c[nH]nc3-n3cnnn3)=O)C2)CC2(CCOC2)C1 85507,C1(CNC(C(CC)N(C)C)=O)CCN(C(c2ccc(C(C)(C)C)cc2)=O)C12CC2 85508,c1(N(CC(=O)NCC(C)NC(CC(=O)OC)=O)C)cc(C)nc2c(C)cccc12 85509,C=C=CCC(=O)N(C1CC(NC(=O)CCC=C(C)C)C1)C 85510,N1(C(C2C(OCC)C2C)=O)CCCC(NC(c2conc2C2CCCC2)=O)C1 85511,c1(C(=O)NC2CN(C(=O)CN3CCCCC3=O)C2)cncc2c(O)nccc12 85512,N1(C(CCC(C)SC)=O)CC2(CCC2)CC1CNC(c1cc(C)ns1)=O 85513,C(=O)(C(CNC(=O)Cn1cnnc1C)CC(C)C)NCC(C(F)(F)F)OC 85514,C1(N=[N+]=[N-])(C(=O)NC2CN(C(C(C)OCC)=O)CC2C(F)F)CCOCC1 85515,N1(C(c2c(CC)nccc2)=O)CCN(C(C2CC3(CCO2)CC3)=O)C(C(C)C)C1 85516,c1(C(N(C2CN(Cc3ccc(C(C)(C)C)[nH]3)C2)CC)=O)nocc1C(C)(C)C 85517,CCCCCC(C(=O)NCC(C1CCCC1)NC(C1CCCN1C(C)=O)=O)C(C)C 85518,c1(C2CCN(C(=O)NCC(=O)NC3(n4cncn4)CC3)C2)c(F)cccc1F 85519,N1(C(C(=O)Nc2cccc(F)c2)=O)CCC(S(=O)(=O)N2CCCC2)CC1 85520,C=CCCC(F)(F)C(=O)NCC1CN(C(c2nccc(Cl)c2C)=O)CC12CCC2 85521,c1(C(=O)NCCC(C)NC(c2c(F)cc(O)cc2F)=O)cnn2ccncc12 85522,Cc1ccc(CC(N2CCOC(CCNC(=O)C=Cc3cnc[nH]3)C2)=O)c(Cl)c1 85523,C1(CC(=O)NC2CC(NC(Cc3c(C)noc3)=O)C2)CCCN(C(C)C)C1 85524,C(CC(O)CC(=O)NCCCC1CCCCN1C(=O)C(c1ccccc1)C)SC 85525,n1(C(CC)C)nnnc1C(C)(C(C)NC1CC(C)(SC)C1)N.SC 85526,c1(OC)cnc(C(=O)NC2C3CC(NC(C4CC(CC5CC5)C4)=O)CC23)cn1 85527,c1(CNc2cc(N3CCC(SC)C3)nc(C(C)C)n2)cc2c[nH]nc2cc1C 85528,C(c1ccccc1)=C(C)C(N1CC(F)CC1C(=O)NCC1CCC(F)(F)C1)=O 85529,Cc1cc(CC(N2C(C(=O)NCCCC(=O)O)CSC2c2ccco2)=O)cc(C)c1 85530,C(=O)(NNc1cc(F)c(F)cc1Cl)c1cc(OC)nnc1SC 85531,c1(OC)ccc(C(=O)NC2CN(C(c3cnn(-c4ccc(F)cc4)c3)=O)C2)cc1 85532,N1(C(C2(C#N)CC3(CC3)C2)=O)CCN(C(c2cccc(CCO)c2)=O)C2(CC2)C1 85533,c1(C(N2CC(CNC(CC(C)C)=O)C(O)C2)=O)ccc(Cl)c(Cl)c1 85534,CC1=C(C)CC(C(=O)NCc2cncc(C(=O)NCC3CNC(=O)CO3)c2)CC1 85535,c1(C(=O)NC)ccc(CCC(=O)NC2C3CN(C(=O)CC(F)(F)F)CC23)cc1 85536,CC1CN(C(=O)CCC2CCOCC2)CC1(C)C(N1CC(C(N)=O)C(O)C1)=O 85537,c1(NC(C2CCCCN2C(=O)Nc2ccnnc2)=O)ccc(I)nc1 85538,Cc1ccc2c(C(=O)NCC3COCCN3C(=O)Cn3cccc3)ccnc2c1 85539,c1(CO)nc(Cl)sc1C.C1(CCOC)(C(=O)N2CC2)CC1 85540,C#Cc1cccc(OCCC(=O)NC(C)CNC(c2c[nH]nc2F)=O)c1 85541,C1(C)(OC(C2(C(=O)OCC)CC2)=O)CCCC1(C)C.C1C(C)=CC(=O)N1 85542,Cc1sccc1C(=O)NCc1cc(C(=O)NCCCC(C)O)cs1 85543,C1(C(C)(C)C)CC(NC(=O)C(=O)NCCc2ccno2)C1 85544,c1(C(N2CC=C(CNC(c3cc(Cl)cc(Br)c3)=O)CC2)=O)cc[nH]c2nccc1-2 85545,Cc1c(CC(N2CC(c3cn(-c4cccnc4)nn3)C2)=O)ncn1C 85546,c1(OC)ccc2c(c1)CCN(C(c1ccc(NC(=O)CSC(C)=O)cc1)=O)C2 85547,Nc1ncc(Br)nc1C(=O)NC1CC(F)CN(C(C2CC=CCC2)=O)C1 85548,C(=O)(C(C)C(O)C(C)C)N1CCC(NC(=O)NCc2c(C)nsc2)C1 85549,c1(C(=O)NC(C)CC2CN(C(c3nn(C)cc3Cl)=O)CC2C)nc2ccccn2n1 85550,Cc1ccc(C(=O)NCC=CCNC(=O)C=C2CCCC2)cc1CO 85551,N1(C(CC)F)CCCC(C(=O)N(CCCC2CCCN2C(=O)C(O)CC)CC)C1 85552,CCCCC(O)C(C)C(=O)NCC1CCC(C(=O)NC2C3CCC4C(C3)CC24)O1 85553,c1(OC)cc(CN2CC(F)(C(=O)Nc3cccc(Br)c3O)C2)c([N+](=O)[O-])cc1O 85554,N1(c2snc(CC)n2)CC(C)(C)CC1CNC(=O)CC(C)C1CCCC1 85555,c1(C(=O)NCC23CC(NC(CC4CC(=O)C4)=O)(C2)C3)ccc(=O)n(CCOC)n1 85556,c1(C(=O)NCC(CNC(c2cn(CC)nn2)=O)CO)c[nH]c2c(C)cccc12 85557,Cc1cc(S(=O)(=O)O)cc(NC(C2CCN2Cc2ccc(C#N)cc2F)=O)c1F 85558,N1(C(COCC=C)=O)CC(C2CC2C(=O)NCC2CC2Cl)C1 85559,N1(C(CC=CC=C)=O)CCC(C2CCN(C(=O)CCOCC(F)(F)F)C2)C1 85560,C(=O)(C1=CC2(CCOCC2)C1)NC(CN(C(c1c(C)nc(CC2CC2)s1)=O)C)C 85561,C1(NC(C(c2cccs2)OCC)=O)CC2CN(C(c3sccc3OC)=O)CC12 85562,N1(C(c2cc(CNC(C(C)S(C)(=O)=O)=O)[nH]n2)=O)CC2CC(C)(C)C2C1 85563,c1(-c2scc(CNC(C3(COC)CC3(F)F)=O)n2)ccc(Cl)nc1N 85564,c1(C(=O)NCC(C(C)C)(C)NC(=O)C=CC2CCCCC2)c(F)cccc1Br 85565,CC#CCC(C(=O)N(C)CC1CC1(C)C)NC(=O)CCc1ncnn1C 85566,C(C1CSc2ccccc21)N(C1COC2(CCNCC2)C1)C(C1CC(C)(C)C1)=O 85567,C(CCCCCC(=O)NN(C(C)C)C)n1cc(C(C(CO)C2CC2)C)nn1 85568,CCC(CC(=O)N(CC(C)NC(=O)CCCN(C)C(C)C)C)C(F)F 85569,CCCC(C(=O)NCC1(C)CCN(C(c2ccnc(CSC)c2)=O)C1)N(C)C 85570,Cc1ccc(-n2nccn2)c(C(N2CC3CC2C3NC(=O)CS(C)(=O)=O)=O)c1 85571,C1(NC(=O)NNC(=O)c2ccc(Cl)cc2)CCCC(C2CC2)CC1 85572,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)C(C)C2)cnc2ccnn2c1C 85573,C1(NC(C(C)N(CCC)C(c2nn(C)cc2C)=O)=O)CN2CCC1(F)CC2 85574,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)COC(C)C(C)C)C2(CC2)C1 85575,C12COCCN1C2=O.C(C(=O)NCCCOCCOC)OCCOCC#C 85576,CC1CN(C(=O)CCCC2CCCN2C)c2ccc(C(F)(F)F)cc2O1 85577,C(=O)(C#CC1CCCCC1)N1CC(CCNC(c2nc(C)sc2)=O)OC(C)C1 85578,CC1CC(CNC(c2ncccc2F)=O)CCN1C(=O)C(F)n1cccn1 85579,C(=O)(CCC(C)C)N1C(C(N2CCC(CCC)C2)=O)CC1C 85580,C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NC2CC3CC4C(C3)C24)(CC)C1 85581,c1(CNC(C2(SC)CN(C(=O)C3=CCSC3)C2)=O)c(C)noc1C 85582,CCN=C(NCC(C)NC(C)C)N1CC2C(CNC(=O)OC(C)(C)C)C2C1 85583,Cc1cc2ccc(C(=O)NCC(C3CC3)NC(=O)CN3CCCC3C)cn2c1 85584,CC(C)(C)CCCCCC(=O)N1CCN(C(=O)C#CC2CCC2)CC1C(F)F 85585,O=C(C(O)C(F)(F)c1ccc(F)cc1)NCc1nc(C2CCC2)n[nH]1 85586,C(c1cncnc1O)=CC(=O)N(CCCCNC(CC1C(C)OCC1)=O)C 85587,O=C(C#CC1CCCOC1)N1CCC2C(C1)CN2C(c1coc(CO)c1)=O 85588,Cc1cc(Cl)cc2cc(C(N3CCC(C)C3CNC(=O)CC(F)(F)F)=O)[nH]c12 85589,C1(CCOC)(NC(C(C)OCCC#C)=O)CCN(C(C2CCC(O)CC2)=O)C1 85590,c1(OCC=C)cccnc1C(=O)NCCC1CCC(NC(c2cc(C)co2)=O)C1 85591,C(CN=c1[nH]c2c(c(=NCC34CCC(CC3)O4)[nH]1)COC2)n1ncc(SCC)c1 85592,c1(C(=O)NCCCN(C(=O)Cc2cccc(OC)c2)CC)cc2sccc2[nH]1 85593,Cc1nc(NCC2CCCCN(C(c3cc(C4CC4)on3)=O)C2)ccc1[N+](=O)[O-] 85594,C=C(C)CC(C)C(=O)NC1CC(F)(CNC(c2c[nH]nc2OC)=O)C1 85595,C1(CC)CN(C(=O)C=C(C)Cl)CCC1NC(C1COC(=O)C1)=O 85596,CC1CC(C(N2CC(F)(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)Cc2nn[nH]c21 85597,N1(C(c2c(OC)cc(CO)cc2)C)CCC(C(C)C)CCC1C 85598,C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(C2(F)CCC2)=O)CC2(CC2)C1 85599,CC1CN(C(C2CC(=O)C2C)=O)CC(C)N(C(C2CC3CCC2CC3)=O)C1 85600,C1(C)(CNC(C(CCOC)NC(C=CCC2(SCC)CCC2)=O)=O)CC2CCC1C2 85601,C1(OCC)CC(NC(=O)COc2cccc(Cl)c2)C12CCC2 85602,C1(NC(C(CC=C)CNC(C2CC3CCC(C2)O3)=O)=O)COC2(CCCC2)C1 85603,N1(c2ccc3c[nH]nc3n2)CCCC2(CCN2C(N(C(C)(C)C)C)=O)C1 85604,N1(C(C(c2ccccc2)NC(c2n[nH]cc2Cl)=O)=O)CCCN(C(=O)C2CC2)CC1 85605,C1(CNC(c2ccc(OCC)o2)=O)CN(C(C)=O)C(C)(C)C1.c12ccc(cc1)[nH]2 85606,C1(NC(c2ccc(COC)[nH]2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 85607,c1(OC)ccc(NC(C2(C)CCCN2C(c2cc(C)oc2C)=O)=O)c(Br)n1 85608,c1(N2CCC(=O)OCCC2)ccccc1.C(CCC)N(CC)CC 85609,N1(C(CC2(COC)CCC2)=O)CCCN(C(c2ccnn2C)=O)CC1C 85610,N1(C(C2(C#C)CCN(C(=O)Cc3ccc[nH]3)CC2)=O)CCOCC(C2CC2)C1 85611,c12noc(n1)CCC(=O)NC2.c1(C(N2CC(CCSC)C2)=O)cnc(C(C)O)s1 85612,C12(CNC(C(=O)NCCNC(C)=O)=O)CC(CN1C(=O)CC1CC1(Cl)Cl)C2 85613,N1(C(c2c(C)cc(=O)n(C)c2)=O)CCC2CN(C(C3(C)CC3(C)C)=O)CC2C1 85614,C(=O)(CCCNC(=O)CSC(F)F)N(C)CC1CCC1 85615,c1(CNCC(C)NC(C2c3nnc(C)n3CC2)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 85616,N(C1CCOc2ccc(Br)cc21)C(C(c1c(N)cccc1)c1ccccc1)=O 85617,Cc1ccc(Cl)c(C(=O)NC(CNC(C2(C(F)F)CC2)=O)CC(C)C)c1N 85618,c1(OC)cccc(C(N2CCCC(N(C)C(C3COCC3(C)C)=O)C2)=O)n1 85619,C(C)(C)(CCC(=O)N(C)CCN(C12CCCC1C2)C)n1cc(SC)nn1 85620,C1(NC(C2CCC(NC(C)=O)CC2)=O)CC2CCC(C1)N2C(=O)Cn1cccn1 85621,N1(C(C=C(CCC)C)=O)CCCC(CC(=O)Nc2cnn(C3CC3)c2CC)CC1 85622,C1(C(F)(F)F)(C(N2CC(NC(c3cc(COC)on3)=O)C2)=O)OC2CCC1CC2 85623,C(=O)(C1=CCC(NC(=O)CC2(O)CCCCC2)C1)N(C1CCOC1)C 85624,C1(C(=O)NCC2(CNC(c3c(C)c[nH]n3)=O)CC2)CCCCN1C(N)=O 85625,c1(C(=O)NC(CC#CC)C(=O)NCCP(C)(C)=O)cc2cc[nH]c2cn1 85626,C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2 85627,C1(C(=O)NCc2ncc(C(N3CC(OC)(CO)C3)=O)cn2)CCOCC1(C)C 85628,N1(C(CCSCC)=O)CCC2(C1)CN(C(C13COCC(C1)C3)=O)CCO2 85629,c1(OC)ccc(F)c(CNC(=O)C(=O)NCC(F)F)n1 85630,C1(C(=O)NCCOCCNC(=O)CC2CCS(=O)(=O)CC2)CC2(CCC2)CCO1 85631,Cc1cc(C(N2CC(O)(C(C)(C)CNC(=O)CC(O)CN3CCCC3)C2)=O)co1 85632,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3(c4cncnc4)CCCCC3)=O)CC2)C1 85633,c1(OC)ccc(CN(c2cc(N3CCc4sccc4C3C)nc(SC)n2)C)c(F)c1F 85634,C1(CCNC(C=CSC)=O)CCCN(C(=O)CC2COC(C)(C)CO2)CC1 85635,C1(NC(C2(OC)CCCC2)=O)(CNC(c2nc(C)ccc2C)=O)CCCCC1C 85636,CC1(C)C(CC(=O)NC2(C)CCN(C(c3ccccn3)=O)C2)C1(C)C 85637,N1(C(CC(CC)SC)=O)C2CC=C(C(=O)NCC3C(C)C3(F)F)C1CC2 85638,N1(C(C(C(C)C)CO)=O)CC2(CCC2)CC1CNC(=O)COC1(C)CCOCC1 85639,c1(C(=O)NC(C)Cn2cc(CCC3CCCN3C)nn2)cncc(O)c1Cl 85640,C12(CNC(C3(CCCC)CC3)=O)CCC1CN(C(=O)C=Cc1c(Cl)n[nH]c1C)C2 85641,N(C1=NCc2ccc(o2)C(=O)NC2(C)CCN1C2)CC.N1(CC)CCN(C)CC1 85642,C1(F)(C(=O)NCc2occ(C(=O)NC(CCC=C)C)n2)CCCCC1 85643,c1(NC(C2C(C(=O)OCc3nc(C(C)OC)no3)C2)=O)cccc(C#N)c1 85644,CC(CC(=O)NCC1(F)CN(C(C2(CF)CC2(F)F)=O)C1)c1ccncc1 85645,CCCCCCCCCC(=O)N1CC(C)(NC(c2ccc(C(F)F)s2)=O)C1 85646,N1(CCNC(C2(CC#C)CCCC2)=O)CCN(c2nnc(SC)s2)CC1 85647,C1(C(N(CCCN=[N+]=[N-])CC(N2CC(CCC)C2)=O)=O)CCCCC1CO 85648,C1(n2cc(CC(c3ccccc3)C)nn2)CCN(C(C2COCCO2)=O)CC1O 85649,Cc1cc(C)c2cc(C(N3CC(CNC(c4c(C)[nH][nH]c4=N)=O)C3)=O)oc2n1 85650,C(=O)(C(C)C(CC)CC)N(C1CCN(C(c2c(CC)n[nH]c2)=O)C1)CC 85651,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 85652,c1(C(N2C(CNC(CC(C)OC)=O)CCCC2)=O)ccc(F)c(F)c1N 85653,C1(NC(c2nc(CC)sc2)=O)CCCC1(C)NC(=O)C(C)c1ccsc1 85654,c1(-c2scc(C(N(C)CC3(NC(C(CC)SC)=O)CC3)=O)n2)ccc(C)cc1 85655,CC1(NC(c2ccc(O)c(Cl)n2)=O)CCN(C(=O)CC2CCCCO2)CC1 85656,c1(Nc2ccc(CC(=O)OCC)cc2)c(Cl)nc(C)nc1Cl.C12CN(C1)NC2=O 85657,C12CCN(CC1)C2.Cn1ccc(-c2n[nH]cc2C(=O)NC(c2cnccn2)=O)n1 85658,n1(C(C)C)cnc(C(=O)NC(C)(C)CN(C(=O)Cc2cncs2)C)c1 85659,N1(C(c2n(CCOC)ncc2)=O)CCCC(N(C)C(C2CCCS2)=O)C1 85660,N1(C(CN2CC(C)C2)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 85661,C1(NC(c2ccc(C)nn2)=O)CN(C(=O)Cn2ncc(Cl)c2C)C2(CCC2)C1 85662,N1(C(C2C(C(N)=O)C2)=O)CCN(C2CCCN(C(c3ccco3)=O)C2)C(=O)C1 85663,C(C(C)(C)CC(=O)N1CCCC(CC(N)=O)C1)NC(C(CC)SC)=O 85664,C(C(C(=O)NCC1CCCCC1)N1CCN(CC2CC2)CC1)(C1CC1)OC 85665,c1(COC)ccccc1-c1nc(-c2c[nH]cc2C)n(Cc2cccc(OC)c2)n1 85666,N1(C(c2c(C)nc(Br)s2)=O)CCN(Cc2cccc(Cl)c2O)C2CC12 85667,C12(CC(=O)NCCCC(C)O)CCC1CN(C(=O)COc1ccsc1)C2 85668,CCCC(CNC(C1CSCCN1C(=O)C(C)=CC1CC1)=O)CCO 85669,c1(C(=O)NC2CN(C(CC(C)OC)=O)C2)sc2nccnc2c1N 85670,C=CCC(CNC(=O)COC1CC1(F)F)C(=O)N(C)Cc1nc[nH]n1 85671,N1(C(C(CC)N(C)C)=O)CC(NC(c2ccnc(OC)n2)=O)C2CCCCC12 85672,N1(C(c2c(C)ccnc2C)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2(C#N)CCC2)C1 85673,c1(CCC(=O)N(CCC(=O)O)CCO)cnccn1.c12cn(nn1)C2 85674,C12(CNC(c3cccc(C)c3)=O)CCCC1CCN2C(c1cccc(Cl)n1)=O 85675,CCN=C(NCCCC(F)(F)F)NCC(c1ccccc1O)(C)O 85676,c1(SCCC(=O)NC(C2CCN(C(C34CC(F)C3C4)=O)C2)C)ccc(F)cc1F 85677,C1(CNC(=O)COC2CCCC2)CCC2(CO1)CC(NC(=O)C(O)C1CCC1)C2 85678,N1(c2c(C)c(NC3CCC4(CC4)C3)ncn2)CC2CC3CC2C1C3 85679,c1(NC(C2C=CC(CC(=O)NC3(C)CC(C)C3)C2)=O)cc[nH]c(=N)n1 85680,c1(OC)ccc(C(F)F)cc1C(=O)NC1CC1NC(=O)C(C)CF 85681,Cc1cc(C(=O)NCC(C2CCCCC2)NC(=O)CC23CC(C2)C3)ccc1[N+](=O)[O-] 85682,c1(OC)ccc(C=CC(=O)NC(C)CC2CN(C(=O)C(O)C(C)(C)C)C2)cc1F 85683,c1(C(N(CC=CC(=O)N(CC#C)Cc2cccnc2)C)=O)cccnc1O 85684,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 85685,c1(SC)ncc(C(=O)NC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c(O)n1 85686,c1(C(=O)NC2CC(C)(C(N3C(C)CN(C)CC3)=O)C2)ccn2ccccc12 85687,c1(CC(N2CCC(NC(CC(C)OC)=O)CC2C)=O)coc2c(C)c(Cl)ccc12 85688,C=C(C)CC(C(=O)NCC(C)(O)CC)NC(c1cc(OC)sn1)=O 85689,CC1CC(NC(c2cccc(=O)o2)=O)CN1C(=O)Cc1ccccc1Br 85690,N1(C(COCCOCC)=O)CC(NC(c2c(Br)n[nH]c2C)=O)CC(O)C1 85691,Cc1ccc2sc(C(N3CCC(C(C)(C)NC(=O)C(F)(F)C(C)O)C3)=O)cc2c1 85692,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 85693,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)NC1(N(C(C)C)C)CCC1 85694,c1(C(C2CCN(C(C(=O)NC)=O)CC2F)=O)cccn2c(C)nnc12.CC(=O)N 85695,C12=CNC=CC1=NC(=O)CC13CC1CN(C3)C(=O)CO2.c1(C(=O)OC)nc[nH]n1 85696,CC(F)(F)CCNC(=O)C(O)C1(CC(N2CCC(C(N3CCCC3)C)C2)=O)CC1 85697,CC1(NC(c2coc(Br)n2)=O)CCN(C(=O)CCCn2ccccc2=O)C1 85698,N1(C(CCC(=O)NCC)=O)CCC(CO)C(NC(=O)CCCn2ccnc2C)C1 85699,N12CC3CC4CC3C1C4NCC1(CC1)C2=O.O=CCc1ccccc1C1CC1 85700,N1(C(CC(C)n2cccc2)=O)CC(NC(=O)CCc2ccncc2Br)C(O)C1 85701,N(C(=NCCc1ccc(F)cc1)NCCc1nc2c(s1)CCC2)CC1(O)CCC1 85702,c1(CC(=O)N(CCCNC(c2cc(OC)ncn2)=O)C)cc(C)cc(C)c1 85703,N1(C(C(C=C)(C)O)=O)CC2CC(NC(c3ccc(CC)c(Br)c3)=O)C1C2 85704,C1(N(C(C2C(=C)C2)=O)C)CCCC(N(C)C(c2occc2OC)=O)C1 85705,c1(C(=O)NC2CC(NC(c3cccc(C(=O)O)c3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 85706,N(C(=S)N1CCC2(CC2)C1)c1ccc(C(c2nnnn2CCC2CC2)C)cc1 85707,c1(N(CCCNC(=O)CC(C)C2CCCO2)CC)ncncc1OC 85708,CC(C)(CCCNC(=O)CC(F)(F)F)C(=O)NCC1CCCS1 85709,c1(OC)cc(C(=O)NC(C)(C)CCCNC(C23CCN(CC2)CC3)=O)cc(F)c1 85710,c1(NC(c2ccccc2)CNC(C(CN(C)C)O)=O)nccc(C#N)n1 85711,N1(C(C)=O)CCC(O)(C(F)(F)C(=O)N2CCC2C(=O)OC(C)(C)C)C1 85712,CN(Cc1c[nH]nc1-c1ccoc1)N1CC=C(C(C)(C)C(C(F)F)C)CC1.C1(O)CC1 85713,N1(C(C2C(COC)CC2)=O)CC2CC2(NC(C2CC(C(C)C)C2)=O)C1 85714,c1(C(N2C(C)CS(=O)CC2)C(=O)NCc2ccco2)cc2ccccn2n1 85715,N(C(=NCc1cocn1)NCC(C)(O)CN1CCCC1)C(C=C)C 85716,C1(CC(N2CCCC(CCC#C)C2)=O)CN(C(c2cncn2C)=O)CCC1C 85717,c12cc(ccc1C)C(=O)c1scc(n1)C(=O)N2.c1(CO)c(F)cncc1Br 85718,C(CCCC)(c1n(CC(CC)O)nnn1)N1CCOC1.c1(OC)cccc(C)c1 85719,FC1(F)CCC2C(CNCCC3CCN(c4ncccn4)CC3)C12 85720,c1(-n2cc(CC(CC(=O)OCC)N)nn2)cccc2ccsc12 85721,C(=O)(C1=COc2ccccc2O1)C(c1cccc[n+]1[O-])=O.C12C3CN(CC13)C2=O 85722,N1(C(C2C(=C)C2)=O)CCC(CNC(=O)Cc2nc(C(N)=O)cs2)C1(C)C 85723,c1(C(N2CC(CNC(C3CCCO3)=O)OCCC2)=O)cc2cccnn2c1 85724,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 85725,Cc1c(O)c(=O)ccn1CC(=O)NCC1(F)CCN(C(=O)CN2CCSCC2)C1 85726,c1(N(CCNC(C)=O)C(C2(CF)CC2)=O)c(C2CCC2)cnn1C 85727,Cn1cnc2cnc(N3CCN(C(c4ccccc4)C#N)CC3)nc12 85728,C(CC(C(C)(C)C)NC(=O)C=CC(C)C)N(CCCNC(c1c(C)noc1N)=O)C 85729,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 85730,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 85731,c1(C(N(C)CCN(C)C(C2CCC(c3nc[nH]n3)O2)=O)=O)ccnnc1S 85732,C1(NC(C(CCC)C#N)=O)Cc2ccccc2C1NC(=O)Cc1cnn(CC)c1 85733,CC(Cc1ccccc1Br)N=c1[nH]c(=NCCN2CCC(O)C2)[nH]c2cccnc12 85734,N1(CC(N2CC(NC(C(C(C)C)OC)=O)C(SC)C2)=O)CCN(C)C(=O)C1 85735,c1(C(=O)NCC2(O)CN(C(=O)CC34CCC(CC3)CC4)C2)ncnc2sccc12 85736,c1(C(N2C(C)(CNC(Cc3nnc(C)o3)=O)CCC2)=O)noc2ccc(F)cc12 85737,C(C(C(=O)N1CC2CC1C2CNC(c1ccc2c[nH]nc2c1)=O)C(F)(F)F)OC 85738,c1(C(N(C2C(C)CCN(C(=O)CC3(C)CC3)C2)C)=O)ccc(Cl)c2ccccc12 85739,C1(NC(C(c2c(C)nn(C)c2)C2CCCCC2)=O)CCC2CN(C(C)C)CC2C1 85740,c1(NC(C2(N(C(=O)C(C)(C)C#N)C)CC2)=O)ccc(Cl)cc1Cl 85741,N1(C(COC(C)=O)C)CCN(C(c2coc(C)n2)C(=O)NC2CCCC(C)C2)CC1 85742,C1(C(N(CCNC(C2(c3ccccc3)CCOC2)=O)CC)=O)CC2CCC(C1)C2 85743,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)NC(C)C1CC1 85744,c1(CC(=O)N(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 85745,c1(OC)ccc(C(=O)NCC2CCN(C(C3(CO)CC3)=O)CC2)nc1 85746,C(=O)(C1=CCCOCC1)N1CCC(CCOC)(NC(C2C(C)(CC)C2)=O)CC1 85747,C1(CC(=O)NC2CN(CC)CC2C)N(C(=O)CSC)CCC1(C)C 85748,C(=O)(C1=NNC(=O)CC1)NC(C1CCCCC1)CNC(COCCOC)=O 85749,N1(C(c2cc(CN(C)C)on2)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 85750,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 85751,c1(CC(=O)NC2C(C(N(CCOCC#C)C)=O)C2(C)C)cc(C)ccc1O 85752,CC(C)C(C(=O)NCCC(C)N(C(=O)C(N)=O)C)NC(=O)OC(C)(C)C 85753,C1(C(=O)NCC2CC(CNC(C(C)OCC#C)=O)C2)CCc2nnnn2C1 85754,c1(C(=O)NCC(CC)NC(=O)C(C#N)CC)cn(C)nc1-c1cccs1 85755,C1(C)(C(N2CCC(OC)C2)=O)CCCN(C(=O)CCC2(C#N)CCC2)C1 85756,C1(NC(CC2CCN(C)C2)=O)CCC2CN(C(c3nc(Cl)ccc3F)=O)CC2C1 85757,Cc1cccc(C)c1NC(=O)C(c1ccc(CC(C)C)s1)N(C)CC1CCCO1 85758,N1(C(CN(C)CC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCCO2)=O 85759,c1(C(=O)NCC(C)CN(C)C(c2cc3sccc3n2C)=O)cc(F)c(F)cc1F 85760,N1(C(CCSCCC)=O)CC(CC(=O)N(CC(C)(C)CSC)C)C(C)C1 85761,C1(CN(C(CN(CCC)C(c2ccc(C#N)o2)=O)=O)C)C(C)(C)C1(C)C 85762,N1(C(CCCCC(C)C)=O)CC=C(C(C)(C)C(=O)NCC2CCC(F)C2)C1 85763,c1(C(=O)NCCC(C)C(F)F)cc2nccc(C(F)(F)F)n2n1 85764,c1(C(=O)NCC2(NC(C3CCSCC3)=O)CCC2)ccc(F)cc1[N+](=O)[O-] 85765,C12(CNC(C(CCC)C#N)=O)CN(C(c3c[nH]nc3C3CC3)=O)CC1CCO2 85766,Cc1nc2cncc(C(N3CC4(CCN(C(c5ccc(F)cn5)=O)C4)C3)=O)c2[nH]1 85767,CC(C)CCCCN(CC(c1cccc(OC2CCC2)c1)O)C(=O)CN(C)C 85768,C1(NC(CC2(OC)CCC2)=O)COCCC1NC(C1CCC(CO)CC1)=O 85769,c1(C(N2CC(NC(C(CCCC)O)=O)(CO)C2)=O)n[nH]c2ccccc12 85770,C(CNC(c1ccc(C2CC2)o1)=O)(C(C)(C)C)NC(CCc1n(C)ccc1)=O 85771,C(=O)(CC(C(=O)N(C)C)NC(=O)C#CC(C)C)NCC1CCC(C(=O)OC)C1 85772,C=CC(C)CC(=O)NC1CC(CNC(c2ccccc2OC(F)(F)F)=O)C1 85773,c1(C(C)C)cc(-c2cscc2NCCCCC(C)C)ccc1F 85774,Cc1cc(C(=O)N(C2CCN(C(=O)COCC3(F)CC3)CC2C)C)ncc1C#N 85775,N1(CCC)CC(C(=O)C2CC2)CC1=O.c12cccc(n1)NC1CC(C1)CNC2=O 85776,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCC2(CCN(C(=O)C(=O)NCC(F)F)C2)C1 85777,c1(C(=O)NC(CC)CNC(=O)CC(C)(C)C#N)cc2c(C)cc(OC)cc2o1 85778,c1(C(=O)NCC(CO)NC(c2cn(C(C)C)c(=O)cc2)=O)n[nH]c2cccnc12 85779,N1(C(C(CN(C)C)(C)C)=O)CCOCC(CNC(=O)CCCCCO)C1 85780,C1(O)(CC(=O)NCCCCNC(CSc2nc(C)[nH]n2)=O)CCCOC1 85781,Cc1ccc2cc(C(=O)NCCCNC(=O)C(F)=CCCF)nn2c1 85782,CC1CC(C(N2CCOC(CN)C2)=O)N(C(=O)CC2(C#N)CCC2)C1 85783,C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2c[nH]ccc2=O)=O)C1 85784,c1(N(c2ccccc2-c2cn(C3CCCCNC3)nn2)C)nccc(S(C)(=O)=O)n1 85785,c1(C(=O)OC)cccc2c(CSC3CCCCC34CC4)cccc12 85786,N1(C(C(CC2CC2)N(C)C)=O)CCCC(NC(c2ccccc2)C2COC2)C1 85787,C1(CNC(CC=C)=O)CCN(C(=O)CCc2nc3ccccc3o2)C12CCC2 85788,C(=O)(CC(C)(C)C=C)NC(CC(=O)N(CC#C)CC1CC1)CC 85789,N1(C(=O)OC)CCc2nc[nH]c2C1.c1(-c2ccc(F)cc2)nc(Cl)ccc1Cl 85790,N1(C(C2CC(N(C)CC)C2)=O)CC2(CCCN(C(c3nc(C)no3)C)C2)C1 85791,C1(C(C)NC(=O)CCc2cnn(C)c2)CCCCN1C(=O)COC1CCCCC1 85792,c1(C(=O)OC)nn(C)[nH]c1=NC(=O)C1(c2noc(C)n2)CC1 85793,N12C(CC3CC13)C(=O)NCc1ccc([nH]1)C2.c1(C(=O)OC)cnccc1C(C)C 85794,CC1(C)NC(=O)CC1C(N1CCSCC1CCNC(c1ccnnc1S)=O)=O 85795,C1(NC(c2c(C)snc2)=O)CCC12CN(C(C1CCN(CC(F)(F)F)C1=O)=O)C2 85796,C=CC(O)C(=O)NC(C)(CNC(Cc1cc(COC)no1)=O)CO 85797,O=C(CCCC1CC1)NC1C(C(c2ccccc2)NC(c2cnn[nH]2)=O)CC1 85798,N1(C(C=C(C)c2ccco2)=O)C(CC(=O)NC2CC=CCC2)C2CCCC12 85799,c1(OCC(=O)OC)cccc(S(=O)(=O)Nc2cccc(N3CCCNC3=O)c2)c1 85800,C1(CNc2c(NC(=O)NCC(N)=O)cccc2)CCc2nnnn2C1C(=O)O 85801,CC1CN(C(=O)CCN2CCC2)CC1CNC(=O)CN1CC(=O)NC1=O 85802,c1(C(=O)NCCC2CN(C(C3CC(F)(F)C3)=O)CC(C)O2)cn2ccncc2n1 85803,c1(CSC)cc(C)n(C)c1C.C12CC(C1)NCC(=O)N(C)CC(=O)N2 85804,c1(C(=O)OC2(CC)CCOC2(C)C)nc2c(OC)cccn2n1 85805,C(=O)(CCCC(=O)OC(C)(C)C)NC(CNC(CC1(OC)CC1)=O)(C)CO 85806,C1(CC(=O)NC2(C(N(C3CC34CCCC4)CC)=O)CCOCC2)CCOC(C)(C)C1 85807,N1(C(c2cnc(C(C)C)nc2)=O)CCC(F)(C(=O)NCC2COCC(C)O2)CC1 85808,c1(C(N2C3CCC(NC(C(Br)=C(C)C)=O)C(C3)C2)=O)cnn2ccc(O)nc12 85809,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 85810,Cc1cn(C)c2nc(N(C(C3CCNCC3)C)Cc3cc(Br)ccc3F)ncc12 85811,c12cc(ncc1OC)NC2=O.c1(C(c2nc(COC)on2)C)ccccc1F 85812,c1(N2CCC(N(C(=O)Cc3cncn3C3CC3)CCC)CC2)ccc(C#N)nc1 85813,C1(CC(N2C(C(c3cn(CCOC)nn3)CC)CCC2)=O)CCC2CC2C1 85814,C1(NC(=O)C(F)n2cccn2)CCCC(NC(=O)CC23CCCC2C3)C1 85815,N1(C(CC)C(=O)NCc2nc(OC)ncc2N)CCc2ccccc21 85816,c1(OC)ccc2nc(C(C(=O)N(C)C)N(C)CCCc3ccccc3)ncc2n1 85817,CC1NC(=O)C2=C1N(CC(=O)O)C(=O)NC2c1cc(C(F)(F)F)c(O)c(=O)o1 85818,c1(C(=O)NC(C)CCCCNC(=O)C2CC2)snc(-c2ccccn2)c1C#N 85819,N1(C(C(C(C)C)C2CCC2)=O)CCCCC(C(=O)NC(c2cccc(O)c2)C)C1 85820,C#Cc1ccc(C(=O)NCC(C)(C)CNC(c2c[nH]cc2C2CC2)=O)nc1 85821,N1(C(C(C)NC(C)=O)=O)CCCC(CNC(c2conc2C2(C)COC2)=O)CC1 85822,Cn1cnc2nc(NCC34CCC(CC3)N4C(c3ccn(C(F)F)n3)=O)ncc12 85823,C1(SC)CN(C(=O)C=CC2CCC2)CC1NC(=O)CN1CCOC1=O 85824,c1(C(C(=O)OC)NC2CCN(CC(F)F)C2)ncc(C)cc1C.C1(N)CC1 85825,Cc1noc(CC(C)C)c1C(N1CCCC(c2nccn2C)C1)=O 85826,CN1CC2CCC(C1)N2C(=O)C(O)CCCNC(=O)CC1CCC(=O)C1C 85827,C(C(C(=O)OCC)O)CC.C(=O)(C(C)(C)Oc1ccccc1)N1CC(CCOCC)C1 85828,C12(NC(C3CC3F)=O)CC3CCC(C1C2)N3C(=O)Cn1ncc2ncccc12 85829,C(CCCCC(=O)NCC1(C(C)NC(=O)CCc2cncnc2O)CC1)SC 85830,C(=O)(C1CCCc2scnc21)NCC(C)(C)Nc1nc(Cl)nc2c1CCC2 85831,N1(c2nnc(CCC)s2)CCN(C(c2ccc(CC)[nH]2)=O)CC(C)(F)C1 85832,CCCC(C(O)C(=O)N1CC(C)(CF)C1)NC(C12CCCC1OCC2)=O 85833,N1(C(C2CC(C(C)C)C2)=O)CCOC(CC(=O)NCC2CCCC2(C)C)C1 85834,C1(CNC(=O)Cn2nccc2-c2ccco2)CN(C(=O)C(F)CC2CC2)CCO1 85835,Cc1cc(CNC(C2CC(C)CN(C(c3c[nH][nH]c3=N)=O)C2)=O)cc(F)c1 85836,N1(C(CN(CC)CC)=O)CCCCCC1CNC(c1cncc(C(F)(F)F)c1)=O 85837,CCCC(CNC(=O)Cn1ccnc1C)C(=O)N1CCCC1CN(C)C 85838,N1(C(C2C(CCC)CN(C(C3CNC(=O)N3)=O)C2)=O)CCn2nccc2C1 85839,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 85840,C1(C2CCCCC2)(C(=O)NC2C(NC(c3nc(CC)sc3)=O)CS(=O)(=O)C2)CC1 85841,c1(CN2CCC(C)C(C)(C)C2)ccc2cc(F)cc(Br)c2n1 85842,c1(-c2c(OC)cccc2C(=O)N=c2cc[nH][nH]2)ccc2[nH]nc(CO)c2c1 85843,N1(C(C(CCCCC)F)=O)CCOC2CCN(C)CC12 85844,Cc1nn(C)c2sc(C(=O)NC3CC(C)N(C(=O)CCCF)C3)cc12 85845,Cc1c(C(=O)N(C(C)CN(C)C(c2cccnn2)=O)C)cnc2ncnn12 85846,C1(NC(C=CC(=O)N(C)C)=O)C=CC(NC(=O)C=CCO)C1.C(C=O)=C 85847,c1(SC)cnn(C)c1C(=O)N(CCCNC(=O)C(c1ccc(C)s1)C)C 85848,c1(C(N2CC3CC2CN3C(c2cscc2C(F)F)=O)=O)cc2n(n1)CCC2 85849,C12(CNC(c3c(CC)ncs3)=O)CCC1CN(C(=O)CN(C)C(=O)OC)C2 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85902,c1(C(N2CC(C)N(c3cc(C4CC4)ncn3)CC2)=O)cc2ncccc2[nH]1 85903,c1(Cn2ccnc2)nc(-c2ccccn2)nn1C1CC2CCC1C2 85904,c1(C(N2CCC(N3CCNC3=O)CC2)C(=O)NCC2CC2)cnc2cnccn12 85905,c1(C(=O)NC2CC(C)N(C(=O)C=CC3CCC3)C2)cc2nc[nH]c2cc1N 85906,C1(NC(C(C)OCC#C)=O)CCS(=O)(=O)C12CN(C(=O)COC1CCC1)C2 85907,N1(CC(=O)NCCCC)CCc2c(OCC)cccc21.c12ccc-1c(F)c2 85908,C(=O)(CCS(=O)(=O)CC(C)C)NCC1CCN(C(CN2CCC(C)CC2)=O)C1C 85909,Cc1cc(C(=O)NC2CCC(CC(=O)NC(c3ccnc(C)n3)C)C2)cnn1 85910,C(=O)(C(F)(F)CCNC(C1CCS(=O)(=O)N1C)=O)NCCCCN(CC)CC 85911,C1(CCCNC(C(CO)N(C)C)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 85912,C(=O)(C1=CC(O)CCC1)N1C(CNC(=O)CO)CC1 85913,CC(C)CCCCCC(=O)NC(C(N1CCC1(N)CO)=O)C1CC1 85914,c1(C(N(C)Cc2ccc(Br)s2)=O)cc2c(-c3ccns3)cc(N)cc2s1 85915,c1(C(=O)NC2(CCCNC(C(=O)N(C)C)=O)CC2)cn2c(Br)cnc2s1 85916,N1(CC)CCC(C23CC(C2)C3)C1.c1(-n2c3nc(n2)C(C)S3)ccc(C)c(F)c1 85917,CC1Cc2sc(C(=O)NCCCN(C)C(c3ccncc3O)=O)cc2C(C)C1 85918,C1(NC(COC(CNC(CCCN(C)C)=O)(C)C)=O)CCC(C)(C)C1 85919,c1(C(N2CCC(N(C(C(CCC)C)=O)C)C2)=O)cc(OC)ccc1O 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86008,C(=O)(C1COc2cc(C)c(C)cc21)NC(C(C)NC(c1c(CC)scn1)=O)(C)C 86009,N1(CC(=O)Nc2cn(CCCC)nn2)CCc2cc(C)ccc2C1 86010,c1(NC(c2c(F)ccc3c2CCC3)=O)ccc2nc(OC(F)(F)F)[nH]c2c1 86011,C1(CC)CN2CCN1N1C(CC1)C2=O.c1(C)cc(C)ccc1F 86012,O(NC(=O)C(CCNC(=O)C(CC)SC)OC)CCCC#C 86013,c1(CN(C(=O)NCC(C)O)CCO)cccc(CN(C)C)c1 86014,Cn1ncc(CN(C=O)CCSc2ncc(C(F)(F)F)[nH]2)n1 86015,CC(C)C1=NOC(C(=O)NCC=C2CCN(C(C3CC(C4CC4)C3)=O)CC2)C1 86016,c1(NC(C2SCCN(C(C=C(C)C(=O)O)=O)C2)=O)cc(F)cnc1Br 86017,CCC(C)(C)C(=O)NCC1(F)CC(NC(c2ccc(C(C)(C)CC)cc2)=O)C1 86018,C1(NC(C(c2ccc(C)cc2)=O)=O)CN(C(=O)CC23CCCC2C3)CC1(C)C 86019,c12c(C)[nH]c(c1C)C(=O)N(C)C2.c1(C(C)=O)c[nH]c(C(N2CC(C(N)=O)C2)=O)c1 86020,C(=O)(C(C)CC(F)(F)F)NCC1COCCN(C(Cc2ccc(C)cc2)=O)C1 86021,N1(C(CC2CC(CC)OCC2)=O)CCOC2(C1)CN(C(=O)CC1CCC1)C2 86022,Cc1c(CC(=O)NC(C)(CNC(=O)CC2CC2CC(C)(C)C)C(C)C)cnn1C 86023,c1(-n2cc(CCC(=O)NCC(c3ccccn3)(C)O)nn2)ccc(S(N)(=O)=O)cc1 86024,N1(C(COCCC)=O)CCC2CCN(C(c3cscc3OC)=O)CC2C1 86025,c1(C(N(CC(CNC(C(CC)CCOC)=O)O)C)=O)occ2c1CCCC2 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86044,C1(C)(NC(C(C)Cc2ccccc2)=O)CCC(NC(=O)COCC2(F)CC2)CC1 86045,C1(C(=O)NC2CC(CNC(c3ccc(OCCO)cc3)=O)C2)CCC(F)(F)CC1 86046,c1(-c2nn(C(C)C)c(-c3cccc(OCCOC(C)C)c3)n2)cccc(C#N)c1 86047,C1(CN(C(CCC)=O)CC)CC(F)(F)CN1C(=O)C(O)Cc1ccccn1 86048,c1(C(N(CCC(N2CCC(C(=O)N(C)C3CC3)C2)=O)CCO)=O)cc[nH]c(=N)n1 86049,Cc1nn(CC(=O)NCC(CNC(C2(C3CC3)CCCO2)=O)CO)c(=O)n1C 86050,N1(C(CC2CC(=O)OC2)=O)CCC(O)(CNC(C2(CO)CCC2)=O)CC1 86051,c1(C(=O)OCC)c(C)ccnc1NCc1cc(C2CCCO2)n[nH]1 86052,N1(C(n2ncc(C(=O)OC)c2)=O)CC(n2cc(CNC(=O)C=NOC)nn2)C(C)C1 86053,c1(OC)ccc(C(N2CCC2CNC(c2nc(C)n(C)c2C)=O)=O)cc1F 86054,CON=CC(=O)NCCCN(C(C1CCC(C(C)(C)C)O1)=O)Cc1ccccc1 86055,C(=O)(CS(=O)(=O)C1CCCC1)Nc1cccc(NC(C2C(C)(C(C)C)C2)=O)c1 86056,CC(C)(Cn1cnnn1)C(=O)N(C1CCCCCC1)Cc1cc[nH]n1 86057,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1(CNC(C(CC)OC2CCCC2)=O)CCC1 86058,C(=O)(CC(=O)NC1CC1)NC(C1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O)C 86059,CC(C)C(O)C(F)(F)C(=O)N1CC2CCC1C(CNC(c1ccc(=N)[nH]c1)=O)C2 86060,C1(C(=O)NC2(CO)CN(C(C(CC#C)C3CC3)=O)C2)CC2(C1)CC2(F)F 86061,C1(C(=O)NC(C)(C)CCNC(=O)Cc2cncnc2)CCCC(N(C)C)C1 86062,CCC(CC(=O)NC1(COC)CN(c2ncoc2-c2ccon2)C1)c1ccccc1 86063,C(=O)(C(Cc1ccccc1)C(F)(F)F)NCC(CO)NC(Cc1n(C)cnc1)=O 86064,c1(C(=O)NCCC2N(C(C(C=C)OC)=O)CCOC2)cc(C)c2[nH]nnc2c1 86065,CCC(C(=O)NCC(n1cc(C2CCCOC2)nn1)C)N1CCCC1 86066,c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NC1CC1NC(=O)CCn1cnnn1 86067,Cc1ccnc(C(F)(F)C(=O)NC2CCC2NC(C2COCC2(C)C)=O)c1 86068,c1(CNC(=O)C(=O)Nc2cc(CO)ccn2)cc(F)c(NS(C)(=O)=O)c(F)c1 86069,C1(NC(CCC(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C 86070,c1(CC)cncc(NC(C2CCC(C)N2C(c2cc(C(C)C)no2)=O)=O)c1 86071,C1(NC(Cn2nnc(C)n2)=O)CCS(=O)(=O)C12CN(C(=O)CCS(C)=O)C2 86072,C1(NC(C2C(OC)C2)=O)CCCCC1C(=O)NCc1ccccc1OC(F)(F)F 86073,c1(C(N2CC(NC(CC(C)(C)C)=O)C3(C2)CC3)=O)cc2ccc(F)cc2[nH]1 86074,C=CCC(C)(C)CC(=O)N1CCC(C)CC1CNC(=O)CC1(N(C)C)CCC1 86075,c1(C(N2CCCC2CNC(C2CC(F)(CF)C2)=O)=O)ccc2c[nH]nc2n1 86076,c1(C(N2C(CNC(CCCC(C)=O)=O)CCCC2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 86077,c1(C(=O)NC(CC)CN(C(=O)C(c2ccnn2C)O)C)cc(O)ncc1F 86078,CC(C)CC(C)C(=O)NCCCC(c1ccccc1)NC(c1csnc1Cl)=O 86079,Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)cc1C 86080,N1(C(=O)OC)CSCC1C(N1CC(O)(C(C)NC(c2c[nH]nc2C(F)F)=O)C1)=O 86081,c1(-n2cc(CCCC)nn2)cccnc1C(=O)N(CC(C)C(C)(C)C)C 86082,C1(CNC(C(C(=C)C)(C)C)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CCC12CCC2 86083,C1(c2nnnn2CCCF)(NC(C2CC3(CCC3)C2)CC)CC2COC1C2 86084,C1(NC(c2[nH]cc(C)c2)=O)(CNC2(c3ccccc3)CCC2)CCCCC1C 86085,C(=O)(CCCCCNC(c1ccsc1OC)=O)NCC(CC(=O)OC)O 86086,c1(OC)ncc(C(=O)NC2CC(F)(CNC(=O)CCCN(C)C(C)=O)C2)c(C)n1 86087,N(C(=NCC1CCCO1)Nc1n(C2CC(F)(F)C2)nnn1)CC(F)(F)F 86088,n1(CC)nnc(C(F)F)c1CC(=O)NCC(CNC(=O)C=CCOC(C)(C)C)CO.O 86089,c1(NCC(N2CC(NC(CC=CC=C)=O)C(F)C2)=O)ccc(C)cc1C 86090,c1(CC)c(Cl)cc(Br)cc1Cl.O1C=CC(=O)N2CCC(C2)n2cc(nn2)CC1 86091,c1(CC(=O)NCC2C=CCN(c3nncs3)C2)ccc2c(c1)CCCC2 86092,N1(C(CN2C(C)CCC2)=O)CCOC(CNC(C2(N(C)C)CCCCC2)=O)C1 86093,c1(C(C)C)ncsc1C(N1CCC(OCCNC(N)=O)C1)=O 86094,c1(NCC2(CSC)CC(F)(F)C2)nccc(=NC(C)C2CCC2)[nH]1 86095,C1(NC(CC(C)(C)O)=O)CC2CC(C1)N(C(c1cnncc1O)=O)C2 86096,CCCC(C(=O)N1CCCCC(NC(c2ccnn2C2CCC2)=O)C1)S(N)(=O)=O 86097,c1(CNC2CCCC(C)CC2)coc(S(C)(=O)=O)c1 86098,CC(CNC(=O)C(=O)NCc1c[nH]nc1C(=O)O)CC(C)O 86099,C1(NC(=O)Cc2cccnc2O)CN(C(c2ccoc2)=O)CC2CCCC12 86100,c1(C(=O)NCCNC(C2C(C(C)C)C2)=O)nc(N(C)C)ccc1F.C1CO1 86101,c1(C(=O)NCC(CNC(CCc2ccc(C(C)C)cc2)=O)C)cc2n(n1)CCO2 86102,C1(CNC(C2CCC(CC)C2)=O)(NC(=O)C(C)(C)CF)CC2CCC1CC2 86103,C1(C(N(C(c2ccc(F)cc2)(CC)C)C)=O)COCCN(CC2COC(=O)N2)C1 86104,c1(CC)ccccc1C(N)=O.c12nc(no1)CNC(=O)N1CC(C1)C2 86105,c1(CC(=O)NCCN(C(C2CC2(C)Br)=O)CC)cn[nH]c1 86106,c1(SCCC(=O)NC2C(NC(C3(C)CCC(=O)C3)=O)C2)ccc2ccccc2c1 86107,C12CC3CN(CC13)C2=O.CC(C(C)SC)NC(=O)C=CCNC(=O)OC(C)(C)C 86108,c1(NC(Cc2c(C)cc(F)cc2)C)ncnc2c(F)cccc12 86109,CN1CCc2[nH]nc(C(=O)Nc3ccc(C(F)(F)F)nc3)c2C1 86110,c1(C(N2CCC(NC(C(C(C)C)OC)=O)C23CC3)=O)ccc2c(C)noc2c1 86111,CCC(CCCC(=O)NCCC1CCSC1)NC(c1ccccc1O)=O 86112,N1(C(Cc2cc(C)no2)=O)CCC(C)(C)C1CNC(C1CCCCC1)=O 86113,c12cnc(s1)C2.n1(C(C)C(=O)N2CCCC2)ccc(C(F)(F)F)n1 86114,c1(C(=O)NCCN(C)C(c2ccc(F)nc2)=O)cnc(O)c(Br)c1 86115,S(=O)(=O)(c1ccc(NC2C3CCC(F)(F)C23)c(C#N)c1)N(C)CCC1CCCO1 86116,c1(OC)ccc(C)cc1C(=O)NC1CC12CC(NC(=O)Cc1csc(=N)[nH]1)C2 86117,c1(C(C)C)nccc(=NC(C)C2CCN(C(=O)COCC3CCOCC3)C2)[nH]1 86118,N1(C(C(c2ccccc2)C)=O)CCC(CNC(c2cncc(N)n2)=O)C12CC2 86119,C1(=CCNC(=O)CC(F)F)CCN(C(C2(F)CCOC2)=O)CC1 86120,C(CCC(=O)NC1CC1CNC(=O)C=CC1CCCO1)N(S(C)(=O)=O)C 86121,N12CC(F)(F)CC1CNC(=O)c1cn2c(SCCC(C2C(C(N)=O)COC2)=O)n1 86122,C(=O)(CCC(=O)NCc1cc(C(N2CCC(C)CC2)=O)cs1)NCC 86123,c1(C(=O)NC(CN2CCN(C(C)=O)CC2)(C)C)nc(C)c(C)nc1C 86124,C=C(Cl)CCC(=O)NCCN(C(=O)CSCc1cccnc1)CC1CCCC1 86125,c1(NC(C(=O)NCC)=O)ccc(OC)c(OCCN2C(C)CCC2C)c1 86126,c1(C(=O)NC(C)CCCNC(=O)C#CC2CC2)ccc2nnc(S)n2c1 86127,c1(CC(N2CCC(n3cc(CCCCC(N)=O)nn3)CC2)=O)cc(Cl)nnc1Cl 86128,c1(C(=O)NCCN(C2CCCC2)C(=O)Cc2cn[nH]c2)cccc(O)n1 86129,c1(C(=O)Nc2nccc(CC)c2)nc(C2=CCC(O)CC2)c2ccccn12 86130,c1(NC(C2(C(=O)OC)CC2)=O)cn(C)c(NC(c2cocn2)=O)n1 86131,CC1=C(C(=O)NCc2occc2C(=O)N(C(C)CC(C)C)C2CC2)CC1 86132,N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(C(=O)NC2CCOC(C)C2)CC1(C)C 86133,c1(N2CCCC(CC)CC2)nc2ccc(Cl)cc2c(=NCCNS(=O)(=O)NC)[nH]1 86134,C1(NC(C(CSC)(C)C)=O)CN(C(=O)CN(C(=O)COC)C)CC1O 86135,c1(OC)cc(C(=O)OCC2CCCN2Cc2cc(C)on2)ccc1N 86136,c1(C(=O)NC2CC(C(=O)NCC=CCl)C2)csnc1Cl 86137,n1(CC)nnc2cc(C(N3CCCCCC(NC(C4CC(F)C4)=O)C3)=O)ccc12 86138,CCCCC(C(=O)OC1CNCCNC1=O)OC 86139,CC(CCCc1ccccc1)C(=O)N1CC(OCC(=O)Nc2cnccn2)C1 86140,C(CC(C)C)(C(=O)N1Cc2ncsc2C1)NC(CCc1ccc(C)o1)=O 86141,N1(C(C(CCC2CC2)NC(CSCC)=O)=O)CC2(CCNC(=O)O2)C1 86142,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86143,C1(C)(CC(=O)N(CCC(=O)NC(c2ccn(C)n2)C)C)OCCO1 86144,N1(C(CCCOC)=O)CCC(NC(C2CC2Oc2ccccc2F)=O)C12CCC2 86145,N1(C(C(C)N(C)C(c2nnsc2N)=O)=O)CCC12CCOCC2 86146,N1(C(C(C)(C)c2ccno2)=O)CCC(C)(C)C(C(=O)NC2COCC2O)C1 86147,c1(OC)ccc(Cn2nc(-c3cncs3)nc2-c2cnc(Cl)s2)cc1 86148,C1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CCC2)C(C=C(C)C)C1(C)C 86149,S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CC(C(=O)Nc2cncnc2O)SCC1 86150,c1(C2C(N(CC(=O)NCCC)CCc3ccccc3)C2)ncccc1F 86151,c1(C(=O)NC2COCCN(C(CCC(=C)C)=O)C2)cc2ccccc2oc1=O 86152,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)NC(c1ccco1)C#C 86153,N1(C(C2(C)CCCC2)=O)CCC(C(F)F)(CNC(C2CCC3CC3C2)=O)C1 86154,c1(NC(=O)OCC)cccc(C(N2CC3CC3(CC(=O)CCN(C)CC)C2)=O)c1 86155,c1(CC(=O)NCc2ccc(CCNC(C3(O)CCC3)=O)cc2)cc(Cl)cc(Cl)c1 86156,c1(-c2cn(CCN3C(N4C(=O)OCC4)COCC3)nn2)ccc(F)c(Br)c1 86157,N1(C(C)=O)CC2CC(C1)C2NC(=O)CN(C)S(N)(=O)=O 86158,CC1(NC(=O)CC2CCSC2)CCCCC1C(=O)NC1C=CCCC1CO 86159,C1(N(CCCc2cccc(F)c2)C)COc2ccc3ccccc3c2C1 86160,Cc1c(C(=O)NCC2CC(C)N(C(c3cnc[nH]3)=O)C2)cc(F)cc1Br 86161,CCCCCCCS(=O)(=O)CC(=O)NCC(C1CCOC1)NC(=O)C1=COCC1 86162,N1(C2CN(C(C)=O)C2)CCN(C(=O)COc2ccc(C(F)(F)CF)cc2)CC1 86163,n1(CCC)ccc(=NC(=O)C2CCC(C(C)C)N2C(C2CC2Cl)=O)[nH]1 86164,C1(CNC(CNS(N)(=O)=O)=O)COCCN1C(C1C(C(F)(F)F)C1C)=O 86165,c1(NC(C(C(=C)C)C)=O)cc(O)nc2ccccc12 86166,C(=O)(CC(O)C(C)CC)NC1(CC)CCN(C(=O)C=Cc2ccsc2Br)C1 86167,C(C(CNC(=O)C=CCOC)S(C)(=O)=O)NC(C1C(CC(CC)C)C1)=O 86168,CCC(C(=O)N(C1CN(C(C2(c3cccc(Cl)c3)CC2)=O)CC1O)C)C(C)(F)F 86169,C1(NC(C=CC)=O)CCN(C(=O)CSCc2ccccc2)CCC1CO 86170,N1(C(C2CCC(F)(F)CO2)=O)CCC2(CC1)CCN(C(C1C=CCCC1)=O)C2 86171,c1(C(=O)NCCC(C)(C)NC(c2cc(=NC)[nH]cc2)=O)csc(=NC2CC2)[nH]1 86172,CS(=O)(=O)c1ccc(F)cc1NC(=O)CC1CN(Cc2cc[nH]c2)C1 86173,C1(CN(C)C(C2CC2c2cn[nH]c2)=O)CN(C(C2CC(F)C2)=O)CCO1 86174,N1(C(c2ncc(C)s2)=O)CCCC(F)(C(=O)Nc2cc(Cl)nc(C)n2)C1 86175,CC1OC2(CNC(=O)CCN3CCC3)CC1(NC(c1cc(N)nc(Br)c1)=O)C2 86176,C1(NC(CCOC)=O)CCN(C(=O)CC2CCC(=O)N2C)C12CC2 86177,C=CCC(C)(C(F)F)NC(=O)C=CCC1(NC(=O)CC(C)=CCC)CCC1 86178,C(=O)(C1Cc2ccccc21)NC1CN(C(C=C(C)C)=O)CC12CCC2 86179,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86180,c1(C(N2C(C(C)NC(=O)CCC=CBr)CCC2)=O)cnc2ccccn12 86181,c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2)=O)noc2c1CCCC2 86182,CC1CCCCCCN1C(C(=O)NCCCOCCOC)c1cncs1 86183,S(=O)(=O)(CCC(=O)N1CCCC(N2CCN(C(C3CC(C#N)C3)=O)CC2)C1)NC 86184,N1(C(CSCC(=O)OC)=O)CCC(C)(F)C1.C1(Cc2ccco2)C(=O)N1 86185,N1(CCCC)CCN(C(=O)C=CCN(C(=O)C(CC)NC(=O)CC)C)CC1 86186,C1(NC(CCOCCC)=O)CC(C)CN(C(=O)CC2CC(O)C2(C)C)C1 86187,C(CC(=O)NOC1CCOCC1)(C(C)OC)NC(C(CC)NC(C)=O)=O 86188,C(=O)(C1=CCCC1(C)C)NC(C)CCNC(c1cc(OCC(F)F)ccn1)=O 86189,C1(CNC(C2CC(C)N(C)C2)=O)CC2(CCN(C(c3ccnn3C)=O)CC2)CO1 86190,Cc1nnc(NC2CCC(C)(CNC(c3nc(C)ncc3Cl)=O)C2)c(C#N)c1C 86191,O(NC(=O)C(C)(C)CCCF)CC(=O)NCC(C#C)CCC 86192,c1(C(N2C(NCc3cnc(CCCC)[nH]3)CC3CC32)=O)ccc(I)cc1Cl 86193,C1(C)(NC(=O)COC2CCC2)CN(C(C2(C(=O)OC)CC2)=O)C1 86194,C1(F)(C(=O)NCSC2C(NC(=O)CNC(c3ccco3)=O)C2)CCS(=O)(=O)C1 86195,c1(OC)ccnc(C(=O)NCC(C)NC(=O)CC(C)n2ccnc2C2CC2)c1F 86196,C1(CC(=O)NC(C(=O)NCC(N2CCCCC2)C)CO)CCC(C)(C)C1 86197,Cc1ccc(CN2CCOCC(C(=O)NCC3=CCCCC3)C2)c(C)c1 86198,N1(C(=O)CCn2cc(CNS(=O)(=O)C(F)F)nn2)CCOC(c2ccc(F)cc2)C1 86199,C1(C(=O)Nn2cnnn2)CC12CCN(c1cc(=O)n(-c3ccc(F)cc3)[nH]1)CC2 86200,C1(C(=O)NCC(C(=O)OC)O)CC(O)CN1C(=O)CC1(C#N)CC1 86201,N1(C(C2(COC)CC2)=O)CCC(CNC(=O)C(C(C)C)NC(N)=O)C1(C)C 86202,c1(OC)ccc2c(CN3CCC(O)C(C(N4CCCC4C#N)=O)C3)c[nH]c2c1 86203,c1(C(=O)NCC(COC)NC(CC(C)OCC)=O)c(F)cccc1F 86204,C1(CNC(c2c(CC)scn2)=O)CCC2(CCC2)C1NC(=O)CN1CCSCC1 86205,C1(CNC(C=C(C)C)=O)(NC(C2CCCC(=O)N2)=O)CCCCC1C 86206,c1(C(N2C(CNC(C(C=C)O)=O)CC2)=O)cnn2cccc(C)c12 86207,c1(C(N(CC(C)NC(=O)Cn2cc(C#N)cn2)C)=O)ncccc1OC(F)F 86208,c1(CC)ccc(C)c(C(N2CCCC3(CNC(=O)CN4CCCCC4)CC23)=O)c1 86209,CS(=O)(=O)c1ccc(CN2CC3CC3(C(=O)Nc3ncc(I)nc3Cl)C2)cc1 86210,c1(C(N2CCC(NC(C3N(C)CCCC3)=O)C23CC3)=O)ccc2ncn(C)c2n1 86211,C(C)(CCC(=O)NOCCCC(=O)OC)NC(c1cccc(CC)n1)=O 86212,C1(NC(C2(CC=C)CC2)=O)CC2CC1CC2C(=O)NC(CC1CC1)C1CC1 86213,C1(C(=O)NC(C2CCN(C(=O)CNc3ccccc3)C2)C)CCS(=O)(=O)N1 86214,C1(NC(c2ccc(C(N)=O)nc2)=O)CCC2(CC1)CN(C(C1CCO1)=O)C2 86215,C1(NC(CCC(CC)CC)=O)CC(C2CCN(C(C3C4CN(C)CC34)=O)CC2)C1 86216,C=CCC(CNC(C1CCCCN1C)=O)C(=O)Nc1ccc[n+]([O-])c1 86217,C(=O)(C#CC1CCCOC1)N1CCN(C(c2c(COC)scc2)=O)C(COC)C1 86218,N1(CCCC)CCN(C(c2ncc(CC)[nH]2)C(=O)NCc2cccc(Cl)c2)CC1 86219,c1(C(C(=O)N(CCC(=O)N(C2(CC)CC2)C)C)O)cncn1C 86220,CS(=O)(=O)CCC(=O)NCC1CCN(C(=O)Nc2ccc(OC3CCC3)cc2)C1 86221,N1(C(C2N(C)CCCC2)=O)CC2CCC(NC(=O)C(F)(F)C3CC3)CC2C1 86222,C12(C(N(C(C)CCNC(=O)C(C)C3CCOC3)C)=O)CC=CC(C1)OC2 86223,Cc1ccc(C(N2CC(NC(C3(F)CCCC3)=O)C(F)C2)=O)c(N)c1C 86224,C1(C(=O)NCC(C)(F)F)CC(F)(F)CN1Cc1cccc(-n2cncn2)c1 86225,c1(C(C(=O)N(C)CCNC(=O)CCC2CC2)=O)cccc(Cl)c1 86226,N1(C(C2C(C)C2C)=O)CCC(CCCNC(C2(C)CCCOC2)=O)CC1 86227,c1(C(N(CCNC(c2ccccc2)=O)CC)=O)ccc2nnn(C)c2c1 86228,C1(CNC(c2c(C)[nH]nc2Br)=O)COCCN(C(C2CN(C)CCO2)=O)C1 86229,c1(C(N(C2CCN(C)CC2)C(C)C)=O)cc(C2CC2)n(C(F)F)n1 86230,c1(NC(c2c(C(C)NC(=O)CC(C)(C)F)noc2)=O)cccc2c1CCO2 86231,C1(C(=O)NC2C=CC(CNC(=O)CSc3nc[nH]n3)C2)CCC2(CCOC2)O1 86232,C(=O)(C(CCC(N)=O)N)N(CCC)CCNC(=O)C(C)Sc1ccc(Cl)cc1 86233,N1(C(C2C(C(N)=O)COC2)=O)CCC(C2CN(C(C3CCO3)=O)C2)CC1 86234,C1(NC(CCNC(=O)OCC)=O)CCN(C(c2ccc(C3CC3C)[nH]2)=O)CC1 86235,C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCN(C(c2scnc2Cl)=O)CC1(C)C 86236,Cc1cnccc1C(=O)NCC12CC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 86237,C1(OCC)CCC(CCC(=O)NCCN(C2CC2)CC2CC3C=CC2O3)CC1 86238,C(CCC(O)CO)N(C(CC1(C)N(C(C=CC=CC=CCC)=O)CC1)=O)C 86239,N#Cc1cccc(F)c1NC(C1CC(F)CN1C(c1ccc(S)cc1)=O)=O 86240,N1(C(=O)OC(C)(C)C)CC(C(=O)O)C(C2CCCC2)C1.N12CCC(CC1)CC2=O 86241,C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCCOC)(C)CO 86242,C1(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C)Cc2c[nH]cc2S1(=O)=O 86243,N1(C(Cn2cc(C(CC)(C)C)nn2)=O)CCC(C(=O)O)C1(C)C 86244,C1(C(N2CCCC(C(N(CCN(C)C(=O)C3CC3)C3CC3)=O)C2)=O)CCCC1(C)C 86245,C1(CC(=O)NCc2ccc(Br)cc2)CC(C)(C)CN1C(CCS(C)=O)=O 86246,C1(NC(c2cc(N)cc(F)c2)=O)CC12CCC(NC(C1CC1F)=O)CC2 86247,c1(N2CC(C)OC(C)(C)C2)nccc(=NCCCCc2ccccc2)[nH]1 86248,CCS(=O)CC(=O)N1CCC(C(=O)NC(C)CF)(C(C)C)C1 86249,N1(C(c2cnn(C)c2C#N)=O)CCCC2(CCCN2C(=O)C(F)C2CC2)C1 86250,Cc1ccc(C(N2CCCCC2CCNC(=O)C(O)C(F)(F)F)=O)cc1Cl 86251,c1(C(N(CC(O)CN(C)C(C2CC2F)=O)C)=O)ccc(N)cn1 86252,C(=O)(CC(C)(C)C1CC1)N(C(C)C(=O)NCc1coc(SC)c1)CCC 86253,c1(CN(C(C(=O)NC(C=C)CO)=O)C2CC2)csc(Br)n1 86254,CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CC3C(C(N)=O)C3C2)=O)CC1=O 86255,Cc1cc(C)c(C(=O)NCC2CC3CCC2N(C(=O)CC(C)F)C3)c(C)n1 86256,c1(C(C(N2CCC(Cn3cc(C4(C(=O)O)CC4)nn3)CC2)=O)O)ccccc1Br 86257,c1(N2CCC(N(C(C(=C(C)C3CC3)F)=O)C)CC2)nc(Cl)nc2c1ncn2C(C)C 86258,C1(NC(CCC2CC(C)C2)=O)CCC(C(=O)NN2CC=CC2CF)CC1 86259,C(=O)(C(F)C(C)(F)F)N1CCC(N(CCC)C(C2(CO)CCCO2)=O)CC1 86260,N1(C(C2(CC=C)CN(C(=O)CC3(O)CCOC3)C2)=O)CCC12CN(C)C2 86261,N1(C(C(C=C)CC)=O)CCC(CNC(c2cc(C3CCC3)on2)=O)C12CCC2 86262,Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCSCC(C)C)nn1C(C)C 86263,C(=O)(CCC(C)(C)C)N(CCCCN(C(=O)CC(O)c1cnc(Cl)s1)C)C 86264,C1(C(C)C)CCOCCN1C(=O)CC1CC(O)CN1C(c1cccs1)=O 86265,N1(C(=O)CC2C=CCC2)CCC2C1CCCN2C(c1cc(F)c2ncccc2c1)=O 86266,c1(C(=O)NCCNC(CC(C=C)c2ccccc2)=O)cc(CC)nc(Cl)n1 86267,c1(C(=O)NC(C(N2CC(C)CC(CC)C2)=O)CN(C)C)c[nH]c2cccnc12 86268,c1(OC)cnccc1C(=O)NCC1C(C(=O)NC2CC3CC3C2)C1(C)C 86269,C(CC(C(=O)NC)NC(=O)CN(C(=O)C=Cc1ccncn1)C)=CC 86270,CC(C(=O)NCC1CCN1C(c1csc(C(C)(C)C)n1)=O)P(C)(C)=O 86271,C(C(C)(C)C(=O)N(C)C)NC(C1N(C(C=CC(=O)N(C)C)=O)CSC1)=O 86272,C(C(C)(C)CC(=O)NC(c1c(CC)[nH]cc1)=O)NC(C1(CO)CCC(C)C1)=O 86273,c1(C(=O)NC(CNC(C(C)OCCCCCC)=O)CO)ccn2cccc2c1 86274,C1(CNC(c2cnn(C)c2C(F)F)=O)CCC2(CN(C(C3CCCOC3)=O)C2)O1 86275,N1(C(C(C=CC)O)=O)CC2CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2C1 86276,c1(CC)cc(N)c(C(=O)NCC2CCCN2C(=O)C(C)CC2CC2)cc1F 86277,c1(C(=O)NC2CC3CC2N(C(=O)CNc2ncccn2)C3)ccc2n[nH]cc2n1 86278,Cc1nc(C(=O)NCC2(C(N3CC(C)(CO)C3)=O)CCC2)c(C)s1 86279,N1(C(C=C(CC)C)=O)CCCC(O)(CNC(=O)CC2CCCN(C)C2)C1 86280,N1(C(C(C)NC(CC)=O)=O)CCC2(CCN(C(c3nc(Cl)sc3C)=O)C2)C1 86281,c1(CCC(=O)Nc2cc(OC)c(F)cc2)ccc2[nH]ccc2c1 86282,c1(C(=O)NC2CN(C(C(C=C)(F)F)=O)CC2C(F)F)ccc(Cl)c(C)c1N 86283,C(=O)(CCC(=O)c1ccc(Cl)s1)NC(CC)CNC(C1CC1c1cnn(C)c1)=O 86284,CC1CCC(C(=O)NC2(CO)CC(F)(F)C2)N(C(c2cn(C)cn2)=O)C1 86285,C1(C(=O)NCC2CC(C(=O)NCCN(C(CC)C)C)C2)CCCCC1O 86286,Cc1cc(C(=O)NC2CC2CNC(=O)C=C2CCC2)ccc1Cl 86287,Cc1cc(C(=O)NC2CCN(C(C3CCC(C)(C)C3)=O)C(C)C2)c(F)cc1F 86288,N1(C(CC(C2CCCCCC2)C)=O)CC2CCC1CN2CC1CCOC(=O)CC1 86289,C(CCCCCN=c1[nH]nco1)NC(=O)CCC1(c2ccccc2)CCC1 86290,CC1CCn2c(CNC(c3cc(-c4ccc(CO)cc4)nc(O)c3)=O)cnc2C1 86291,c1(OC)cc(C=CC(N2CCN(C(=O)C(C#N)C(C)C)C(CO)C2)=O)ccc1O 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86346,C(C(C)(COC)CC)NC(C1(CC)CN(C(c2nc(COC)oc2)=O)C1)=O 86347,c1(N2CCC(c3n(C(C)C)cnn3)C2)nc2ccsc2c(=NCC#CC2CC2)[nH]1 86348,N1(C(C2OCCC(C)C2)=O)CCC2(CCC2CNC(=O)CN2CCCCC2)CC1 86349,Cc1cc(F)cc2c1CCN(c1nc(N3CCOC(C#N)C3)nc3scnc13)C2 86350,N1(C(CCC(C)(C)C)=O)CC(NC(=O)CN=c2cc[nH]cc2)CC2(CCC2)C1 86351,C(=O)(C1=Cc2ccccc2C1)NCC(CC(=O)N(CC(F)F)C)C1CC1 86352,C1(CC(=O)NC(c2csnn2)C)COCCN1C(=O)CC1(n2cccn2)CCC1 86353,c1(C(=O)NCC2C(NC(COCc3cccc(OC)c3)=O)C2)cc(N)cnc1Cl 86354,CCCC(CNC(=O)CCCC1CCCO1)C(=O)NC(C)(CC)CCO 86355,C(CC1CCC1)(C(=O)NCC1CC(O)C1)NC(C(C)OCCCC)=O 86356,c1(C(=O)NCC2CCC(NC(C3CCC(C)C3)=O)C2)ccc2n[nH]cc2c1 86357,N1(C(C=CC(C)(C)SC)=O)CCCCC1CC(=O)NCCc1cc[nH]n1 86358,CC#CC1CCN(C(=O)C(CCF)NC(C2CC3COCC3C2)=O)CC1 86359,C1(C(N2CCC(C(C)NC(C=C(C)C(C)C)=O)CC2)=O)CC2CCCCN2C1 86360,N1(C(CN(C2CCCC2)C)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 86361,C1(NC(CSC)=O)CCC2(CCCN(C(=O)Cc3ccncc3)C2)C1 86362,c1(C(N2C(c3cn(CCCC(=O)OCC)nn3)CCC2)=O)cc(C)cnc1C 86363,N(C1CCCc2ccoc21)C(=O)NCCC1CCCC1(F)F 86364,C1(C(=O)NCCCOC)CCC=CC1NCc1ccc(C)cc1 86365,c1(C(N2CCCC(NC(C3C4COCC34)=O)C2)=O)ccc(C(F)(F)F)cc1Br 86366,CS(=O)(=O)CCCC(=O)OCc1nnc(C(F)(F)F)s1 86367,N1(C(c2ccnc(C)n2)=O)CCN(CCO)C(C)C1.c12ccoc1C(=O)NC2 86368,CC(O)CCCC(=O)NC(C)CN(C)C(C1(P(C)(C)=O)CC1)=O 86369,C1(C(N(C2CN(C(=O)CCc3ccccc3[N+](=O)[O-])C2)C)=O)CC(=O)OC1(C)C 86370,c1(C(=O)NCC(CNC(CN(C(=O)OCC)C)=O)(C)F)ncncc1C 86371,C(=O)(C(CO)C(C)(C)C)N1CCC(O)(C(C)NC(=O)Cn2cccn2)C1 86372,C(=O)(C1=NOC(C)(C)C1)NC1CN(Cc2nc(C)sc2C)C(C)CC1 86373,CC(CC(F)F)C(=O)N1CCCCC(C(=O)NOC(C2(C)CCCN2CCF)=O)C1 86374,CC(O)C(C(=O)N(CC(=O)Nc1cocn1)C)NC(=O)C1CC1 86375,c1(SCC(=O)NCC2C(NC(c3n(CCOC)ncc3)=O)C2)ccc(F)cc1 86376,c1(C(C(=O)NCC2(NC(CN(C(C)C)C)=O)CC2)C)ccccc1C(F)(F)F 86377,C1(N(C(C2CCOC2CSC(F)F)=O)CC)CCN(C(c2ccco2)=O)CC1 86378,Cc1ccn(C(C)CC(=O)NCC2CN(C(=O)C(C)C)C2)n1 86379,CS(=O)(=O)C1CN(C(=O)C(O)C2CC2)CC1NC(=O)CC(O)c1ccccc1 86380,C1(C(=O)NCC2CN(C(c3c(SC)ccs3)=O)CC2O)CC2(CCC2)CCO1 86381,c1(C(=O)NCCCC(c2ccccc2)NC(CNC(=O)NC)=O)sc(C)cc1Cl 86382,C1(C(=O)NC(CCSC)C(N)=O)CC12CCN(C(c1c[nH]nc1C(C)C)=O)CC2 86383,C1(C(=O)NCCCOCCN(C(CC=C=C)=O)C)Cc2ccccc2O1 86384,CC(C)C(C(=O)N1CCC(N(C)C(c2cnn[nH]2)=O)CC1)Sc1ccccc1 86385,C(=O)(N=c1[nH][nH]c2c1CN(C(C1CC1(F)F)=O)C2)c1cc(C)c(=O)n(C)c1 86386,C12(CC)CN(C(c3ccsn3)=O)C(CNC(c3sc(F)cc3C)=O)(C1)C2 86387,C1(C)(CC)CC(C(=O)NC2CC(CCNC(c3csc(S)n3)=O)C2)C1 86388,c1(C(=O)OC(C)C(=O)NC(c2ccccn2)C)ccc([N+](=O)[O-])c(N(C)C)c1 86389,c1(C(=O)NC2(CCCCNC(C3(C)ON=C(C)C3)=O)CC2)cc(C)c(C)cn1 86390,N(C(=NCCF)NC1CC(OC(C)(C)C)C1(C)C)C(C#C)(C)C.OCC 86391,c1(CCOC)cc(C(=O)NC(CC(=O)NC2CC(C(F)(F)F)C2)C2CC2)no1 86392,N12CC3CCC(C1=CC2=O)C3.N1(C(C(C)(C)C)=O)CCCC(n2cc(CO)nn2)C1 86393,C12CCCCC1OCCSn1ncc(n1)-c1nc2no1.N1(CC)CCCOCC1 86394,N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCN(C(=O)CC2(O)CCCCC2)CCC1C 86395,N1(C(CC2CCC(NC(c3cc(C)n(C)c3C)=O)CC2)=O)CCC(C)C(C)(C)C1 86396,N1(C(C(C=C)(C)C)=O)CCC(C)N(C(c2ccc(C(F)(F)F)s2)=O)CC1 86397,c1(C(N2CC3C(N(C(c4c(NC)cnnc4)=O)C)C3C2)=O)cc2c([nH]1)CCCC2 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86538,C1(F)(CNC(C(C)C2CC2)=O)CN(C(=O)C(F)(F)c2cnn(C)c2)C1 86539,c1(C(=O)N(C(C2CCN(C(=O)CC3CS(=O)(=O)C3)C2)C)C2CC2)cnc(N(C)C)s1 86540,N1(C(c2c(C)cncc2)C(=O)NC2CCOC2)CC(C)(C)C12CCC2 86541,c1(NCC(C2CC=CCC2)NC(C(=O)OCC)=O)ccc(OCC(F)(F)F)nc1 86542,c1(CC)ccc(C(N2CC(NC(C3CSCCS3)=O)C(F)C2)=O)cc1 86543,c1(C(CNC(C(C(CC)(C)C)O)=O)NC(=O)C2CC2)ccc2ccccc2c1 86544,N1(C(C(C)=C(CC)C)=O)CCN(C)C(CNC2COCCO2)C1 86545,C1(C(N2CC(C(C)C)C(NC(=O)COCCN(C)C)C2)=O)CCC12CCOCC2 86546,n1(CCC(=O)OCC)nnnc1C(CCc1cnccn1)NCC(C)C(C)C 86547,C(=O)(C#CC1CCCOC1)N1CCC(C)C(NC(c2cc(O)nc(O)n2)=O)C1 86548,C1(NC(C(C)SCC)=O)CCC(C)(C)N(C(C2(Br)CC=CCC2)=O)C1 86549,c1(CC)nn(C)c(Cl)c1C(=O)NCC(C(C)C)NC(C1CN2CCC1CC2)=O 86550,N1(C(CCc2ccc(C)o2)=O)CC(O)CC1(C)C(=O)N(CCC(C)C)C 86551,c1(C(C)C(=O)N2CC(NC(=O)CCc3cncn3C)C2)ccc(C#N)cc1 86552,O=C(C1CCCc2c[nH]nc21)NCC1CN(C(=O)Cc2ccc(Cl)cc2)CCO1 86553,C(=O)(C(O)CCCNC(=O)C(CN(C)C)C(C)C)NC(C=C)C1CCC1 86554,c1(CC)cc(C(=O)N(C2CN(C(c3nocc3C)=O)CC2(C)C)C)c(C)nn1 86555,C1(C(N2CC(C#C)(F)C2)=O)CC2C=CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 86556,O=C(CCS(=O)(=O)c1ccc(F)cc1)NC1CCN(C(C2CC2(F)F)=O)C1 86557,c12cccc(c1)CC(=O)N2.c1(OC)cnn(C)c1 86558,C(=O)(C(c1cn[nH]c1)N(C)CCc1cccs1)NCCSC 86559,c1(C(N(CC=C)CC2CC2)=O)oc(CNC(=O)CC(C)C2CCCC2)nc1C 86560,C1(NC(CC)=O)CCCC(OC)CC1.c12cc(OC)cc(c1)OC2=O 86561,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)C(C)(C)O 86562,c1(N2C(CNC)CC(O)C2)ncnc2ccnn12 86563,c1(C(=O)NC2C(NC(C(C3CCC3)OC)=O)CC2)cc(C)c(Cl)c(C)c1 86564,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 86565,N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(=O)Cc1ccc3nn[nH]c3c1)CCO2 86566,N1(C(COCC=C)=O)CCC(CCNC(c2cc(C)nnc2O)=O)C(F)(F)CC1 86567,c1(C(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)[nH]c2ccc(Cl)cc2c1Cl 86568,C1(F)(C(=O)NCCN(C(COCCC(C)C)=O)C(C)C)CC1(F)F 86569,CC1(C)CCOC1CC(=O)NCC1CCCCC1NC(=O)C1=CCCC1 86570,c1(C(=O)NCC(CCOC)NC(C2(C#N)CCC2)=O)cncc2nc(C)[nH]c12 86571,C(C)(C)(C(c1cccnn1)N(C)C)OC.C12(CC1)C(=O)N2 86572,C(C(=O)NCc1cccc(C)c1)(C(=O)NC)NC(C1C(OCC)C1)=O 86573,c1(C(=O)NC2C(OC)CN(C(c3sccc3SC(F)F)=O)C2)cnc(C)c(C)c1 86574,CP(C)(=O)c1cncc(C(N2CCCC(NC(=O)COC3CCOC3)C2)=O)c1 86575,N1(C(c2cc(N)cc(C)c2F)=O)CC(CNC(C2CC2C)=O)C2(CCOCC2)C1 86576,C1(C(=O)NC)CCCC(NC(=O)NCc2cc(-c3ccccn3)[nH]n2)C1 86577,c1(NC(C2(C)CCN(Cc3cnc(OC)c(Br)c3)C2)=O)ccc(F)cc1[N+](=O)[O-] 86578,N1(C(=O)Cc2ccnc(F)c2)CCC2C1CCN2C(c1cc2cccnc2[nH]1)=O 86579,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 86580,C(CCCC(=O)N1CCC(CN(C)C(c2cnc(N(C)C)o2)=O)C1)OCC 86581,N1(C(C2(C)C(C)C2)=O)CC2CCC1CN2C(C1(c2ccno2)CCC1)=O 86582,C(C(CC(F)(F)F)NC(c1snc(O)c1Cl)=O)NC(C(C(C)C)OC)=O 86583,C1(O)(C(C)NC(CCOC(C)C)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 86584,CCC(C(=O)NC(N)=O)N(CC(=O)OC(C)C)C.C12(CC(F)C1)C(=O)N2 86585,C1(NC(CC2CC(=C)C2)=O)CC(O)CN(C(c2csc(-c3cnn(C)c3)n2)=O)C1 86586,N1(C(Cc2c(C)cccn2)=O)Cc2ccccc2C(NC(c2ccsn2)=O)C1 86587,C(=O)(C(S(C)(=O)=O)C1CC1)NCCCN(C(=O)C(O)CC(N)=O)C(C)C 86588,C1(NC(C2(C)C=CCN2C(C2CC(N(O)C)C2)=O)=O)(CO)CC2CCCC12 86589,C1(CNC(c2c(C(C)C)ocn2)=O)CCCC2CN(C(C3(C#N)CC3)=O)CC12 86590,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(c2nc(O)nc(O)n2)=O)C1 86591,Cc1ccc(O)cc1C(=O)NCCC1CC(C(=O)NC2CCCCC2(C)O)C1 86592,CCC(C(=O)NC1CC(NC(=O)Cn2cc(C)cn2)C(O)C1)C(C)(F)F 86593,N1(C(c2scc(CC)n2)=O)CCC(C(=O)NCCc2cn(C)nc2C)C12CC2 86594,N1(C(Cn2nc(C)oc2=O)=O)CCN(C(C2(C3CCC3)CC2)=O)C(C)C1 86595,N1(C(C(Br)=C(C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3F)CC2C1 86596,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 86597,c1(C(=O)NCCC2(OC)CN(C(C3(C)CC=CCC3)=O)C2)cc(F)cnc1O 86598,C(=O)(C1CCCc2nccn21)N1CCC(CNC(c2ccc(CC)cc2)=O)CC1 86599,N1(C(CC=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 86600,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCCn1cccn1)SC 86601,C(=O)(C(C(=O)NC1(C(=O)NC2C=CCCCC2)CCCCC1)OC)OCC 86602,c1(C(=O)NCC2N(C(CC(=C)Br)=O)CC2)cn(C)nc1Oc1ccccc1 86603,C=CC(C)(O)CC(=O)NC(CNC(c1[nH]ccc1C1CC1)=O)C1CC1 86604,N1(CC)CC(C(=O)NCC2(O)CC(NC(C34CC(CCO3)C4)=O)C2)CCC1=O 86605,C1(NC(c2occc2Cl)=O)CCC2(CC1)CN(C(C1CC3(CCC3O)C1)=O)C2 86606,C1(C(=O)NC2CCCN(C(CCn3ccc(C)n3)=O)C2)CN2CCC1(C)CC2 86607,Cc1oc(C#N)cc1C(=O)NC1CCCC1NC(c1ccc(CO)s1)=O 86608,C(=O)(C(O)CC(C)C)N(CC(CNC(C(CCC)C)=O)O)C 86609,c1(NC(N2C(COC)(CNC(c3ncccn3)=O)CCC2)=O)cc(C)ncc1Cl 86610,N1(C(CCC(CCC)CC)=O)CCC2CCCC(C1)N2C(C1(O)CCSCC1)=O 86611,C(c1ccc(C(C)(C)C)cc1)=CC(=O)N(CCCNC(=O)C(N)=O)C 86612,N1(C(CCCOCC)=O)CCN(C(c2ccc(C)cn2)=O)C2CC12 86613,N1(C(c2n[nH]c(CC)c2Br)=O)CCSCC1c1nc(C)no1 86614,C1(C(=O)NC(C)C(=O)N(C)Cc2cccs2)CCCN1C1CCCCC1 86615,[N-]=[N+]=NC1COCC1n1cc(C2CC3(CCN3C(C3C4CCCC34)=O)C2)nn1 86616,c1(C(N(C2COCC2S(C)(=O)=O)C)=O)cc2cc(Cl)ccc2[nH]1 86617,N1(C(C2C(C)CC2)=O)CCN(CC(=O)N(C)C(c2cnnn2C)C)CC1 86618,N1(C(C(CC)C)=O)CCC(NC(c2cn(CC3CC3)nn2)=O)C(CC)C1 86619,c1(OC)ccc(C(=O)N(C(C)CNC(=O)CCCOc2ccccc2)C)nc1 86620,CC(C(=O)NCC1CC(NC(=O)Cc2cccs2)CCO1)C(F)(F)F 86621,C(=O)(C(C)S(C)(=O)=O)N(C1CCCN(C(COCCC(C)C)=O)C1)C 86622,C#CCC(CC(=O)OC)NC(=O)CC(CCC)NC(=O)C1=C(C)CC1 86623,C1(CC(N2CCC(NC(C3(F)CCOC3)=O)C(F)C2)=O)CN2CCN1CC2 86624,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 86625,c1(OC)c(C(N2CC3CCN(c4nccc(SC)n4)C3C2)=O)cccc1[N+](=O)[O-] 86626,c1(C(=O)NCC(CN(C(=O)CC23COC(C)(C2)C3)C)O)c(N)cccc1Cl 86627,S(=O)(=O)(c1ccc(C(F)F)cn1)N(C)CCNC(=O)Cn1nnc2c1CCCC2 86628,CC1=NNC(=O)C1CCC(=O)N1CC(CC(=O)NOC(C)C)C1 86629,N1(C(C2=NNC(=O)C2)=O)CC2(CCC2)CC1CNC(=O)C(C1CCOCC1)=O 86630,C(C(=O)NNC(=O)C(N)C(C)c1cccnc1)n1cc(CCN(C)C)nn1 86631,C1(C(=O)NCc2c(C(N(CCN(C)C)C)=O)cccc2)CC2COCC2C1 86632,C1(C(N2CC(O)(C(C)NC(C3(OC)CCSCC3)=O)C2)=O)CCN(C)S1(=O)=O 86633,N1(C(CSCC(=O)OC)=O)CC2(C(=O)NCC(CC(C)C)SC)CC1CCO2 86634,C#CCCN=C(NCCC1CC2CC1O2)N1CCC(C(N)=O)(C(N)=O)C1 86635,N1(C(c2c(C)nsc2)=O)CCC(c2cn(CCNS(C)(=O)=O)nn2)CC1 86636,C(=O)(C(=O)N(C)C)NCCNC(C1(CC(C)C)CC1)=O.C1CN1 86637,c1(CN(C)Cc2cc(NCCC(=O)O)ns2)ccc(OC(F)F)cc1 86638,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 86639,C(C)(C)(CCCNC(=O)CC1OCCC1C)NC(Cc1cn(CC)nn1)=O 86640,C1(CCC)CN(C(=O)C(C)(c2cccs2)NC(=O)C(C)=C(C)C)CC1OC 86641,Cc1ccc2c(C(=O)NC(C)CCCNC(C3CC(F)C(=O)N3)=O)c[nH]c2c1 86642,c1(C(N(C)CC2(NC(C(CO)N(C)C)=O)CC2)=O)ccc(CC2CCCO2)nc1 86643,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)CCCC2)nn1)CC(C)(C)C 86644,C(=O)(C(C)S(N)(=O)=O)NC1(CNC(C(C)SCC)=O)CC1 86645,c1(C(N(CCNC(C2CCCN(C(C)=O)C2)=O)CC)=O)ccc(O)c([N+](=O)[O-])c1 86646,N1(C(=O)OC)CCN(C2CC2CC2CCCN(C(C3CC(F)(F)C3)=O)C2)CC1 86647,CC(C(=O)N1CC(n2cc(C3(O)CC3)nn2)CO1)N(C)C 86648,c1(C(=O)NC2CC(N(C)C(C3CCCCS3)=O)C2)cccn2cc(C)nc12 86649,c1(NC(C2N(C(C)=O)CC(O)C2)=O)n[nH]c2c(F)cccc12.C12CCN(CC1)C2 86650,N1(C(c2c(C)nns2)=O)CCC2(CCC(N3CCC(O)(CF)CC3)O2)CC1 86651,N1(C(=O)CC2CCCOC2)CCC2(C1)CN(C(c1cc3occc3s1)=O)C2 86652,CCC(COC)C(=O)N(CCC(=O)NCC1CC=CCC1)C 86653,C1(O)(CNC(C=CC(=O)N(C)C)=O)CCN(C(C2CC(=O)CO2)=O)CC1 86654,O(C1CCc2cc(OC)ccc21)C(CCCC(CC)C(=O)O)=O 86655,C1(C(=O)NCC2CCN(C(CC)=O)C2)CC2(CCN1C(C1CCCO1)=O)CC2 86656,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(NC(C=C(C)C)=O)C1C)=O 86657,c1(C(N2C(C(=O)Nc3nnco3)CC3CC32)=O)ccc2nccc(Cl)c2c1 86658,N1(C(=O)OC)CCOC(C)C1C(=O)NCCCF 86659,CCC(CCC(=O)NCCN(C(=O)C(c1ccccc1F)O)C1CC1)OC 86660,C(=O)(C#CC1CCCCO1)N1CCCC(CNC(c2c(C)cn(C)c2)=O)CC1 86661,Cc1nccc(CN(C2CCCCN2C(=O)Nc2cnc(Cl)n2C)C)n1 86662,C1(NC(C(CC#C)C2CC2)=O)CC12CCN(C(c1ccc(Cl)c(C)c1N)=O)CC2 86663,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 86664,C=CCCC(C(=O)NC1CCOC(C)(CC)C1)NC(c1ccc(CC)o1)=O 86665,Cc1cnccc1C=CCNC(=O)N(CC(C)O)CC1CC1 86666,C12(NC(c3cnc(SC)s3)=O)CCC(CNC(=O)CN(C)C)(C1)OC2 86667,N1(C(C2=C(C)OCC2)=O)CCCC2CCN(C(c3c(C(F)F)cnn3C)=O)CC12 86668,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC(C)(O)CNC(c1cc(C(F)F)[nH]n1)=O 86669,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 86670,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1C)=O 86671,N1(C(COCC(N2CCCC2)C)=O)CCC2(CC2NC(c2ccc(C#N)cn2)=O)C1 86672,C12(C(=O)NC(CC)CO)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 86673,c1(C(=O)NCCC(C)NC(=O)C(F)n2ccnc2)ccc2c(c1)CCO2 86674,C(=O)(CCCC(C)=O)NCC(CC(=O)N(C(CC(CC)C)C)C)C 86675,C(C(=O)N1CCN(C(C)CNC(C2(C(F)F)CC2)=O)CC1)(C(C)C)OC 86676,c1(C(=O)NCCCN(C(=O)C(F)OC(F)(F)F)CC)cc(CC)nnc1C 86677,c12c[nH]nc1C(=O)NCC1CCC(C1)NC2.c1(CCC(=O)OC)ccccc1 86678,C#Cc1ccc(OCC(C)(C)C(=O)NC2CCN(C(=O)CC(=O)OC)C2)cc1 86679,CS(C)(=O)=Nc1ccc(C(=O)NC2CCC2NC(=O)Cn2c(O)nnc2O)nc1 86680,Cc1ncsc1C(C)NC(=O)CCN(C(=O)C(C)Cn1ccnc1)C(C)C 86681,c1(Nc2c(CC(N3CCC(CO)C(O)C3)=O)cccc2)ncnc2occc12 86682,c1(CC)ncncc1C(=O)NC(C1CCN(C(=O)CCc2cccnc2)C1)C 86683,C(C(C)C(F)C(=O)N(c1cn(C)nc1C)C(C)C)NC(CCc1cc(C)on1)=O 86684,c1(COC)ccnc(NC(C2CCCC(NC(c3cscc3C)=O)C2)=O)c1 86685,C12(C(N3CCCC(OC)C3)=O)C(NC(=O)C(C)C(C)C)C3CC1C2C3 86686,C1(NC(c2n(CC)c(O)nc2)=O)CN(C(=O)CC2CCCCC2O)CCC1F 86687,C1(C(=O)NC(C(C)=O)=O)CCN(C(=O)CC2CCC(C)C2)CC1(C)C 86688,c1(C2(CC)CC2)ccccc1C(=O)NC1CCC(NC(=O)OC(C)(C)C)C1 86689,Cn1nccc(C(=O)NC2CN(C(=O)Cn3nccn3)CC2O)c1=O 86690,N1(C(Cc2n(C)c(S)nn2)=O)CC(NC(c2csnc2C2CC2)=O)CC(F)C1 86691,N1(C(c2nc(C)n(C)c2)=O)C2CCCC1CN(C(=O)CC1CCCC(C)C1)C2 86692,c1(OC)c(-c2ccc(C#N)s2)cccc1S(=O)(=O)Nc1nccc(C(F)(F)F)n1 86693,C1(C)(C(=O)NCC(=C)CCNC(c2cnc(C(=O)OC)s2)=O)CC(O)CN1C 86694,C1(c2n(CC)nnn2)(NCc2nn(COC)nc2C)CCC(c2nc(C)no2)C1 86695,C12(C(=O)NCc3cccc(C)c3)COCC1CN(C(=O)C(C)Cn1ccnc1)C2 86696,N1CCC(C)(C)C(C)C1.N1(N(C)C)CCCCC1NC(N)=O 86697,C(C(C(=O)NC(c1nn(C)cc1O)C)C(C)(C)C)NC(C(C(=O)OCC)(C)C)=O 86698,c1(C2(C(=O)NC(CC(C)NC(=O)CSCC#N)C)CC2)ccc(O)cc1 86699,c1(CC)cccc(C(=O)NC2CC(NC(=O)Cc3c(Cl)cnn3C)C2)c1F 86700,[N-]=[N+]=NC1CN(C(c2csc(CO)n2)=O)CC1NC(C1CC(=O)NC(=O)N1)=O 86701,N1(C(c2cccc(NC)n2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C)C1 86702,c1(CNC(=NCC)NCC2CCCC2(C)C)c(OC)ccc(Cl)c1Cl 86703,C(=O)(CC(C)C)NC1(C(=O)NC2(C(=O)NCC)CC2)CSC1.NC 86704,c1(CC)nc(O)c(C(N2CCC3(NC(=O)CCc4ncc[nH]4)CC3C2)=O)cc1C 86705,N1(C(CCC(CC)CC)=O)CCCCC2(C1)CN(C(=O)Cc1cnnn1C)C2 86706,C1(NC(C(CN(C)C)(C)C)=O)CC2(CCCN(C(=O)C=Cc3cccnc3)C2)C1 86707,Cc1scc(NC(=O)NCC(C(F)F)NC(=O)OC(C)(C)C)c1N 86708,C(=O)(C(CNC(=O)CN1CCCCC1=O)(CC)CC)NC(C#C)C(C)(C)C 86709,C1(CNC(c2c(C)cnnc2)=O)CCCCN(C(=O)C(C2CCCCCC2)C)C1 86710,Cc1nc(N)cnc1C(=O)N(C)CCOCCNC(=O)CC(C)n1ccnc1 86711,C1(NC(c2ccc(C)[nH]2)=O)CN(C(C2CC23CCOCC3)=O)CC2(CCC2)C1 86712,c1(C(C)C)cc(N2CCC(NC(=O)C3=CCCCC3)C(C)C2)n2ncnc2n1 86713,C(=O)(C#CC1(C)CCCO1)NC(CC)CNC(C1CCC2(C1)CC2(F)F)=O 86714,C=C=C(C)CC(=O)N1CCC(C(C)CNC(=O)C(c2ccccc2F)(F)F)C1 86715,C1(CN(C(C(C)OCCC(C)C)=O)C)CN(C(=O)CC=CC(C)(C)C)CCO1 86716,CC1CCN(C(=O)O)CCC1N1CCSC1.C1(NC(C)(C)C)CCCNCC1 86717,c1(C(=O)NCCCCNC(Cn2ccc(C)n2)=O)cccc(F)c1F 86718,c1(C(N2CC3C(NC(=O)CN4C(=O)C=CC4=O)C3C2)=O)c(F)c(F)c(O)c(F)c1F 86719,C1(NC(CN2CCC(C)CC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 86720,c1(OC)ccc(C(=O)NCC#CC(=O)NCC(=O)NC2CCCC2)s1 86721,N1(C(C=NOC)=O)CCOCC(C)(CNC(C2NC(=O)C3CCC23)=O)C1 86722,c1(C(=O)NCC2(F)CCC(CNC(C34CCC(C3)OC4)=O)C2)ccc(F)cc1Cl 86723,c1(OC)c(C(=O)NCC2CC(C)N(C(C3CC(OC)C3)=O)C2)sc(Cl)c1Cl 86724,N1(CC)CC(C(=O)NCCN(C(C2(c3ncc(C)o3)CC2)=O)CC)CC1=O 86725,N1(S(C)(=O)=O)CCCCC1C(N1CCCCC1CNC(C1(C)CS(=O)(=O)C1)=O)=O 86726,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 86727,c1(NC(C2CCC(NC(=O)Cc3cccc(Br)n3)C2)=O)cc(F)c(Cl)c(Cl)c1 86728,N1(C(C(N(C(C(C)OCC(C)C)=O)C)C2CC2)=O)CCCC[Si](C)(C)C1 86729,CCCCN=c1[nH]c(=NCc2n[nH]c3c2COCC3)[nH]c2c1SCC2 86730,c1(C(N(C2CN(C(=O)C(C)(C)O)CC2O)C)=O)c[nH]cc(Br)c1=O 86731,N1(C(CC(C(F)F)NC(c2cc(C)c(F)cc2)=O)=O)CCC2CCCC2CC1 86732,Nc1sc2c(c1C(N1CCC3(CC(NC(=O)CCC4CC4(Cl)Cl)C3)C1)=O)CCC2 86733,[N-]=[N+]=NCCCCCC(=O)NC1CCN(C(c2ccc(CO)o2)=O)C12CC2 86734,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 86735,c12ccccc1NC1CCN(C1)C(=O)C1CCN1C2=O.N1(C)CCOCC1.CCO 86736,c1(C(=O)NC2C(NC(CNC(=O)NC)=O)COC2)nnc2n1CCCCC2 86737,c1(OC)ccc(NC(C(N2CCCC2C(=O)N(C)CC2CCOC2C)=O)=O)cc1 86738,C(=O)(CCC=CBr)N(CCCNC(c1ccc(C2CC2)s1)=O)CC 86739,Cc1nc(C(=O)Oc2cccc(Cl)c2)c(C)s1.N12CCN(CC1)CCOCC2 86740,N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 86741,N1(C(C2CNC(=O)N2)=O)CC(C2CC2)(C(=O)NC2C3C=CC(C3)C2CO)C1 86742,c1(CN(C)C(=O)NCCC2CCCCO2)c(F)ccc(Br)c1F 86743,c1(C(N2CCCC(NC(CCOCC#C)=O)C2CC)=O)cnc([N+](=O)[O-])n1C 86744,N1(C(C(C)=CC)=O)CCCC(NC(=O)CCc2nnc(C3CC3)o2)CC1 86745,C1C2=CCN(CC2)C(=O)C1OC.c1(CC2(C(=O)OC)CC2)ccncc1 86746,c1(C(N2CC3C(C(=O)Nc4cnc(OCC)nc4)C3C2)=O)cn(C)c(=O)nc1O 86747,C1(F)(CNC(C(C)OCC=C)=O)CCN(C(c2cccs2)=O)CC1 86748,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 86749,C1(NC(c2ccc(F)c(F)c2)C(C)C)CC2CCC1C(N)C2 86750,C(=O)(CC(O)CC(C)(C)C)NC(CCNC(C(=O)NCCCCC)=O)(C)CC 86751,C1(C(=O)NCC(C)CO)CC(O)CN1C(c1cc(Cl)no1)=O 86752,N1(C(C(C(CC)C)NC(C2CCNC2=O)=O)=O)CCC2CN(C)CC2C1 86753,C(=O)(CCCCCOC)N1CC(OC)C(NC(=O)CCC2(C)CC2)C1 86754,c1(NC(CCC)CNC(=O)Cn2cc(Cl)cn2)c([N+](=O)[O-])c(CC)nn1C 86755,CC1(NC(C(CC2CN(C(=O)Cc3nnc(O)o3)C2)F)=O)CC1(F)F 86756,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCSc1nccn1C 86757,N1(CC2CC(=O)N2)CCCN(C(c2noc(C3CC3)n2)C)CC1.C(C)(=O)OCC 86758,C1(C(=O)NC(CC(=O)NCC(=O)N(CC(C)C)C2CC2)C)CCCCC1O 86759,c1(NS(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCCN3C3CC3)=O)C2)cn1 86760,CC(C)(CCC(=O)NC1CC(CNC(=O)C(O)(C2CC2)C2CC2)C1)[N+](=O)[O-] 86761,CC(CC(=O)N1CC(O)CC1C(=O)NC1CC(CO)C12CCC2)C(F)F 86762,c1(C(C(=O)N2CC(F)C2)NC(CCOC(C)C)=O)cnn(C)c1 86763,C12(NC(=O)CCNc3ccccn3)CCC1CN(C(c1c[nH]c(=O)cn1)=O)C2 86764,c1(C(N(C2CC(NC(CN(CCC#C)C)=O)C2)C)=O)cc2occc2n1C 86765,N1(CCNC(C=Cc2ccc(OCC)o2)=O)CCCC(C)C1 86766,C(CN=c1cc(C)nc(C)[nH]1)C1(O)CCN(C(C=CC=CC=CC)=O)CC1 86767,c1(-n2ncc(C(C(=O)OC)OC)c2)ccc(C)cc1 86768,CC1c2ccc(F)cc2CCN1C(c1ncsc1Br)C(=O)Nc1cccc([N+](=O)[O-])c1 86769,c1(NCc2cn(CC(C3CCOCC3)OCC)nn2)c(OC2CC2)ncnc1Cl 86770,CC(CC(C)NC(C1CCCN1c1ccncn1)=O)NC(=O)C(C)(C)C 86771,c1(CC(N2C(CCC(=O)NC(C3CC(=C)C3)C)CCC2)=O)nn(C)cc1C(C)=O 86772,c1(C(N(CCC(=O)N(C(CC)C)CC)CCO)=O)c[nH]nc1CC 86773,C1(C(=O)NC(c2ccccc2)CC)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 86774,C1(N(C)C(C2(C)CCCN2C(=O)OC(C)(C)C)=O)CCC(=O)NC1=O 86775,C1(C2CCCN(C(=O)C(C)(C)CC#N)C2)(NC(C(c2ccccc2)C)=O)CC1 86776,CC1CN(C(c2ccn(CCNC(C3C4CCC(=O)C34)=O)c2)=O)c2cccnc21 86777,C(=O)(C(CNC(C1CNC(=O)N1)=O)CC1CCCC1)N.C(C)(CC(N)=O)(C1CC1)OC 86778,c1(OCC(=O)NCC2(NC(c3c[nH]c(=NC)o3)=O)CCC2)cc(C)c(Cl)c(C)c1 86779,CC(Cc1ccc(F)cc1)C(F)C(=O)N1CC2C(c3cccc(F)c3)C2C1 86780,N1(C(C)C)CC2CC1CN2C(c1nc(C(=O)Nc2ccc(O)c(F)c2)cs1)=O 86781,c1(COC)nc(OC)cc(N2CCCCC2CNC(c2csnc2C2CC2)=O)n1 86782,c1(C(=O)NCC2N(C(C(CC)OC3CCCCC3)=O)CC2)cc2ccccc2s1 86783,C1(C(N2CCN(C(CCOC)=O)CC2C)=O)CC2CC1C1C2C1(F)F 86784,C1(CC(=O)NCCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 86785,C1(N(CC=C)C=O)CN(C(=O)C(CC)=C(C)C)CCC1(C)C.OCC 86786,c1(C(N2C(C(C)NC(c3cc(Cl)cnn3)=O)CCC2)=O)cncc2nc[nH]c12 86787,CN1CC2(CN(C(=O)C(O)C3CN(C(=O)Cc4ccccc4F)C3)C2)C1 86788,C1(NC(NCC(C)C)=NCC2CC(=O)N(c3ccccc3)C2)CCOC(C)(C)C1 86789,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 86790,C1(CNC(C2CC(=C3CC3)C2)=O)CCCN1C(C1(c2cccnc2)CCCC1)=O 86791,CC1CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C(=O)Nc1cccc(Cl)c1 86792,c1(NC(C2(C)CN(Cc3ccc(O)c(O)c3)C2)=O)ccc(OC(F)(F)F)cc1Br 86793,C=C(C)C1CCC(NCc2ccc(Cl)c(CO)c2)CC1 86794,c1(CC)oc(C(=O)NC2(C(=O)NCCCN3CCC(O)C3)CCN(C)C2)cc1C 86795,C1(CC)CCN(C(=O)C(C)C2(O)CCC2)C1C(=O)NCCS(=O)(=O)NC 86796,c1(-n2cc(C(C3CC=CCC3)NC(C(C)O)CO)nn2)ncccc1OC(F)F 86797,c1(C(N2CCC3CN(C(C(CCCOC)C)=O)C3C2)=O)cc(C#N)c(O)nc1N 86798,C1(NC(C(C)NC(c2ccc(NS(C)(=O)=O)cc2)=O)C)CCC(=O)N(C2CC2)C1 86799,N1(C(C2N(C)CCCC2)=O)CC2CC1CC2NC(c1cc(Cl)ncc1F)=O 86800,C1(CN(C)C(c2sc(F)cc2Cl)=O)CN(C(=O)Cc2cncs2)CCO1 86801,N1(C(C2(CC=C)CCCC2)=O)CC(NC(=O)C(C)Oc2ccccn2)CCC1C 86802,C1(C)(OC)CCCN(C(C2OCCC2NC(=O)C2=C(C)CCC2)=O)CC1 86803,Cc1c(C(=O)OC2CCCC2C2CCCC2)sc2c(F)cc(F)cc12 86804,C1(CC)CN(C(c2cocc2C)=O)CCC1NC(C1(C)CC(F)C1)=O 86805,c1(C2CNC(=O)N2)cccc(Cl)c1.CC(CCc1cn[nH]c1)N(C)C 86806,C(=O)(CCCCN(C(=O)C(C)(F)c1ccon1)C)NC(c1cc(O)n[nH]1)C 86807,c1(OC)ccc(CCC(=O)NC2CN(C(C3CCSC3)=O)C2)cn1 86808,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 86809,c1(C(=O)NC(CCOC)CNC(=O)C=Cc2cnc[nH]2)ccc2c(c1)OCCO2 86810,N12CCN(CC1=O)C(=O)CC1CN(CCO1)C2=O.C1(CC)CCC(C2CC2)CC1 86811,Cc1cc(C(=O)NC(C2CC2C(=O)NCc2ccn(C(C)C)n2)C)n(C)n1 86812,C(CO)(CCCCNC(C1(C)CCCC1)=O)NC(C=CC=CC)=O.COC 86813,C1(CNC(C2C(C=C)C2)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 86814,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OCC(F)F)c1)=O 86815,CC1(C)CC(C)(NC(C2COCCN2C(c2cc(=O)cc[nH]2)=O)=O)C1 86816,Cc1cc(NC(C2C=CCN(C(c3cc(Cl)n(C)n3)=O)C2)=O)n(C)n1 86817,c1(C(=O)NCCOC2CN(C(=O)CCOC3CC3)C2)nnc2ccccc2n1 86818,C12(C(N(CC(CC)NC(=O)Cc3cc(C4CC4)on3)CC)=O)CCCC1CC2 86819,c1(C(N2CCC(OC)(CF)C2)=O)c2c(nn1C)CCS(=O)(=O)C2 86820,CCCC(C)C(CC)(c1nnnn1CCCOC)NC12CC(CCO1)C2 86821,N1(C(C=C(C)c2ccsc2)=O)CCC2CN(C(c3cn4c(n3)COCC4)=O)CC12 86822,c1(C(N2CCCC(NC(c3cncc(CSCC)n3)=O)C2)=O)ccc(C)nc1O 86823,c1(CC(N2CC=CC(NC(CN(CCC#C)C)=O)C2)=O)ccc(S(C)=O)cc1 86824,CS(=O)(=O)c1cc(Br)ccc1NC(C1CC(NS(=O)(=O)c2ccncc2)C1)=O 86825,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 86826,CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCC(C)(C)CC1)C 86827,c1(OC)ccoc1C(=O)NCCC(O)CNC(c1ccc(CN2CCCCC2)o1)=O 86828,N1(C(C(C2CCC2)NC(C2CCN(CC)C2)=O)=O)CCCC(C2CC2)CC1 86829,C1(NC(NCc2ccc(O)cc2)=NCC2CC2)CCc2nncn2C1 86830,C(=O)(C(C)(F)C(=O)N(C)CCN(C)C(c1ccnc(C(C)C)n1)=O)OC 86831,N1(CC2CCC3(CCC3)C2)CCCC(C)(C)C1C.C1(O)COCCC1N 86832,c1(C(=O)NCCC(C)CCNC(=O)CC2CC2(C)C)cncn(C)c1=O 86833,C1(c2cn(CCCN(C)C)nn2)C=CCN(C(c2cccc(CO)n2)=O)C1 86834,N1(C(c2ccc(Cl)o2)=O)CC(C2CC2)(C(=O)NCC2(CO)CCCCC2)C1 86835,Cc1ccc2c(c1)C(C(=O)NC(CNC(=O)Cn1cc(C(C)O)nn1)C(C)C)C2 86836,c1(OC)ncccc1CC(=O)NC1CCN(C(C)Cn2cccn2)CC1 86837,C(=O)(NNc1ncc(Br)c2ccccc12)C1CCC(NC(CCC(=C)C)=O)C1 86838,C1(CCC(N2CC(CC(C)NC(=O)CN(c3ccccc3)C)C2)=O)CCCN1C 86839,C12(C(=O)NCC(C)(C3CC3)NC(=O)CC34COCC(C3)C4)CCC(CC1O)C2 86840,NC(=S)C1(NCCN=[N+]=[N-])CCN(C(=O)C(O)CO)CC1 86841,c1(C(N2CC(CNC(C3(C)CC(C#N)C3)=O)OCC2)=O)ncn2c1CCCC2 86842,c1(NC(C(C)OC(=O)CC(c2ccccc2)N(C)C)=O)nnn(C)c1N 86843,C=CC1(C(N2C3C=CCC2CC3)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C1 86844,c1(C(=O)NCCCCCNC(c2sccc2F)=O)ccc2n[nH]cc2c1F 86845,C1(NC(c2ccc(C(N)=O)cc2)=O)CC2CCC1N(C(c1cc(Cl)c[nH]1)=O)C2 86846,C(CCCCCO)NC(CC(C)N(C(CN1CCC(C)C1)=O)C)=O 86847,C(=O)(C(C)C(C)NC(c1cnc(OC)cn1)=O)NCC1CN(CCC)C1 86848,CN1CCOC(CC(=O)NC(CCN(C)C(c2ccco2)=O)c2cccs2)C1 86849,Cc1cc(S(=O)(=O)NC2CN(C(=O)Cc3ccc(Cl)cn3)CCO2)c(Cl)cc1Cl 86850,N1(C(C#CC2(CC)CC2)=O)CCCN(C(c2cccc(C3(C)CC3)c2)=O)C(C)C1 86851,C12(C(=O)NC(C#C)CC)CCC(NC(C3CC34CCCCC4)=O)(CC1)C2 86852,Cc1cc(Cl)cc(C(=O)NCC2CC2CNC(=O)CCCC(F)(F)F)c1C 86853,CN1CCOC(C(=O)NCC(C2CC2)NC(c2cccnc2N)=O)C1=O 86854,c1(CC)ccsc1C(=O)NC(C(=O)NCc1cncn1C1CC1)C1CC1 86855,Cc1ncc(N)cc1C(=O)NCC(C)N(C)C(c1nc(Cl)c(Cl)s1)=O 86856,c1(C(=O)NCC2N(C(C(CC)C(=O)OC)=O)CCCC2)noc2c1CC(C)CC2 86857,C=CCCC(F)(F)C(=O)N1CC2CCC(C1)C2NC(C1(C)CC2CC2C1)=O 86858,c1(C(C(=O)NCC(C(C)C)NC(=O)C(=O)NCC(F)F)C)cncc(F)c1 86859,c1(CN(c2nc(OCC)c(OC)cn2)C2CCCNC2)ccc2c(c1)ncn2C 86860,c1(OC)cc(NC(=O)Nc2nc[nH]n2)cc(O)c1OCC1CC1.N1(CCC)CCCC1 86861,C(=O)(C(C)(C)C(N)=O)N1CC(NC(C2C(C)OCCC2)=O)C1 86862,CN1CCN(C(=O)C(O)CCN(C)C)CC1CNC(c1cccc(N(C)C)c1)=O 86863,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 86864,c1(C(N(C(C)C(=O)NCCC2CCC(=O)N2)CCC)=O)ncc(F)cn1 86865,Cc1cc(=O)n(CCCCC2CCCN2C(=O)C(C)(C)c2cscc2Cl)cn1 86866,C1(C(N(CCNC(c2cc(-c3ccco3)[nH]n2)=O)CC2CC2)=O)CCC12CCCO2 86867,N1(C(c2c(COC)n(-c3cccc(Cl)c3)nc2)=O)CCCN(C)C(=O)C1 86868,Cc1ccc(C(=O)NCC2C(C(N3CC(O)(CCO)C3)=O)C2(C)C)s1 86869,N1(C(C(C)(C)OC)=O)Cc2occ(C(=O)NC3CN(C)CC3C)c2C1 86870,C#CCCCC(C)C(=O)N(CCCNC(C1(C)COC1)=O)CCC 86871,C(CCCCCNC(=O)CC1CCC(=O)C1C)N(C)C(C1(c2ccno2)CC1)=O 86872,n1(CCC)ncnc1C(N1CCC(C(=O)NCCC2CC2)C1)C(=O)NC 86873,CC1CN(C(=O)Cc2ccn(C)c2)CC(C)N(C(c2[nH]ccc2C2CCC2)=O)C1 86874,c1(C(C)NC(C(C)N(C(C(C)=CCC)=O)C2CC2)=O)ccnn1C 86875,Cn1cc(C(=O)NC23CCCC(NC(=O)C(F)C(F)(F)F)(C2)C3)ccc1=O 86876,CN1CCCCC(C(=O)NCCCN(C)C(c2cn3c(n2)SCC3)=O)C1=O 86877,C(=O)(CCCCC1CC1)N1CC(OCCNC(C(C)CC2CCCO2)=O)C1 86878,c1(C(=O)NC2(CCNC(C3(CC)CC(O)C3)=O)CCCC2)cc(O)cc(=O)o1 86879,N1(C(c2c(Cl)ccc(C#C)c2)=O)CCCC2(NC(=O)Cn3ccc(C)n3)CC2C1 86880,c1(C(N2C(C3(NC(CNS(NC)(=O)=O)=O)CC3)CCC2)=O)cc(C)n(CCO)n1 86881,C1(NC(C(C)Cn2cccn2)=O)C2CC3C1C3C2C(=O)Nc1cc(O)cc(F)c1 86882,Nc1c(C(N2CC(NC(=O)Cn3ncnn3)CC(F)(F)C2)=O)ccc(Cl)c1Cl 86883,S(=O)(=O)(c1c[nH]ccc1=NCCCNC1CC1)NC(CC)CCOC 86884,c1(CC(N2CCCC(CN(C(C(C)(C)CO)=O)CC)C2)=O)ccc2occc2c1 86885,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(N(C(CC3C(OC)CC3)=O)C)C2C1 86886,N1(C(C2(SC)CCC2)=O)CCC(C)C(NC(=O)C(C)(c2ccccc2)N(C)C)C1 86887,C(=O)(C(CC)C(C)(C)CC)N1CCC(CCNC(CC(=C)C)=O)C1 86888,C(CC(C)C)(C(=O)NCCC(CC)CO)NC(C1(CC)CNC(=O)C1)=O 86889,c1(OC)cc(C)c(CC(c2ccn(C)n2)Nc2cc(N(C)C)nc(C)n2)cc1C 86890,S(=O)(=O)(c1cccnc1NCC(CO)C1CCC1)NCC(C(C)O)(C)C 86891,C(=O)(C(CC(C)C)NC(C1(CC=C)CC1)=O)N(CC(=O)NCC=C)C 86892,CCCCCC(O)C(=O)NC1(CCC(=O)N(C(CO)C2CC2)C)CCC1 86893,CN1CC2C(CCCN2C(=O)NC2CCCN(Cc3ccccc3)C2)C1=O 86894,CC1(C)CCC(C(=O)NC(CCO)C2CC2)CN1C(C1(O)CCCC1)=O 86895,CCC(C)(COC)C(=O)N1CSCC1C(=O)NCc1nn(CC)nc1C 86896,C(=O)(C=C1SCC(=O)N1C)N(CCC(C)NC(=O)CC1CC(=O)NC(=O)C1)C 86897,C1(CNC(c2c(C(C)C)con2)=O)CN(C(C2CCOC(=O)CC2)=O)CCCO1 86898,N1(C(C=CC=CCC)=O)CCCCC1C(C)(C)CNC(c1ccc(N(C)C)cn1)=O 86899,C1(F)(CNC(C(C)OCOC)=O)CN(C(=O)CCNC(c2ccco2)=O)C1 86900,N1(C(CN(C(c2cc(C)on2)=O)CCO)=O)CCN(C(=O)Cc2ccco2)CC1 86901,c1(OC)cc(NC(=O)C(=O)N(C)C)ccc1CN(C(C)CC(C)O)C 86902,C1(C(=O)NCC(=O)NC(CCC)C)COCOC1 86903,c1(C(CC)=O)ccc(C(=O)NCC2CC2NC(=O)CN(C2CCC2)C)cc1 86904,C1(C(N(CC#C)CCF)=O)CN(C(=O)C=C(C)C2CC2)CC1(C)C 86905,c1(C(N(C2CCC(NC(C(C)C)=O)CC2)C)=O)nc2ccc(Cl)nn2n1 86906,C=C=CC(C)C(=O)NCCC1CCCN(C(C2(C)COC2)=O)C1 86907,c1(CCC)noc2ncc(C(N3CCN(C(=O)CNC(N)=O)C4CCC34)=O)cc12 86908,O=C(C1=CCCCCC1)NC(C1OC(=O)CC1OCc1ccccc1)C(=O)O 86909,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 86910,c1(C(=O)NCCN(C2CCCCC2)C(CC2(C)OCCO2)=O)cccc(Cl)c1O 86911,Cc1cncc2cc(C(N3CCOCC(NC(c4cn[nH]c4)=O)C3)=O)sc12 86912,c1(-c2nnc(NC(=O)CCCNc3cccc(C)n3)o2)c(F)cccc1F 86913,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 86914,CC(C)C(C)(CNC(c1ccc(C2CC2)nn1)=O)NC(C1CCC(=O)C1)=O 86915,C1(C)(C=O)CCCOC1.C12(CCC1)C(=O)NCC2.C(C)(CNC)OC 86916,c1(NC(N2CCCC2C(=O)Nc2ncccc2Br)=O)ccc2nonc2c1 86917,c1(OC)nccc2c(C(N3CCCN(C(=O)CCS(N)(=O)=O)C(C)C3)=O)c[nH]c12 86918,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 86919,C(CCC(C)CC(=O)N(CCNC(C1(C(C)(C)O)CC1)=O)C1CC1)=C(C)C 86920,c1(SC)cc(Br)ccc1C(=O)OC(C)C(=O)NCC(F)F 86921,C1(C)(C(=O)NC2ON=C(C(=O)OC)C2)CN(C(=O)CC2(O)CCCCC2)CCO1 86922,N1(C(c2c(CC)csc2)=O)CC(NC(=O)Cc2cccc(C#N)c2)CCC1C 86923,CC(CN=c1[nH]cnc2c(F)c(F)ccc12)N(C(=O)Cc1ccc(Cl)cn1)C 86924,N12CCCCC1CNC(=O)CNS(=O)(=O)CC2.c1(CC)ccc(COC)s1 86925,C(=O)(C1=CCN(C(c2c(OC(F)F)ccnc2O)=O)C1)NCC 86926,C(C)(CCS(C)(=O)=O)NC(C(=O)Nc1ccc(N(CCC)C)nc1)=O 86927,c1(C(=O)NC2CC(N(C)C(C3CCCSC3)=O)C2)cccc(N(C)C)n1 86928,C(=O)(C1Cc2ccc(F)cc21)NC1(CNC(CC(C)C2CC2)=O)CCCC1 86929,Cc1cccc2nc(NCCCC3CCCN3C)[nH]c12 86930,N1(C(=O)Cc2ccc(F)c(F)c2)C2CCC1CN(C(c1ncsc1Br)=O)C2 86931,N1(C(CCCSC(C)(C)C)=O)CCC(CCNC(=O)C(c2cncn2C)O)C1 86932,C=CCCC(=O)N(CCNC(c1cscc1Cl)=O)Cc1ccccc1 86933,C1(C(N(CCCNC(C2CCN(C(=O)N(C)C)C2)=O)CC)=O)CC2CCC1O2 86934,N1(C(C(C)O)=O)CCCCC(NC(=O)C=CC2CCC2)C1 86935,C1(C(N(C2CSC2)CC#C)=O)CCOCC1NC(c1cccn1CCC)=O 86936,C#CCCC(=O)NC12CC(C(=O)NCCC(C)(O)C3CC3)(C1)C2 86937,c1(OCC(=O)N(CCNC(C2(CC(C)C)CCCC2)=O)C(C)C)cccc(O)c1 86938,Cc1nc(C2CCN(C(c3cc(CNC(=O)C(C)CC4CC4)on3)=O)C2)n[nH]1 86939,c1(C(=O)NCCCC(C)NC(=O)CSc2cccs2)ccccc1CC(=O)OC 86940,C12(C(=O)NC(C(C(C)C)NC(C3CC4(CCOC4)C3)=O)C)CC3CC1C2C3(F)F 86941,c1(CC)nc(C(N2CCCC2CN(C(=O)C(F)=C(C)C)CC)=O)c2ccccn12 86942,CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)C=C(Cl)Cl)CCC12CCC2 86943,C(CN=C(NCC1CC1)N1CCC(NCCN(S(C)(=O)=O)C)C1)N1C(C)CCC1 86944,C1(C)(OC)CC(C(=O)Nc2nncs2)C1(C)C.C1CCNC(=O)N1 86945,c1(NC(C)C)cccc(Cn2cccn2)c1.N12CCC(CC1)NC2=O 86946,C1(C(N2CCC2CNC(C2ON=C(C)C2C)=O)=O)(CC)CC(F)(F)C1 86947,c1(C2C(C)(C)C2)nc(CCc2cc[nH]n2)cc(=NCC2CCC3(CCC3)O2)[nH]1 86948,C(=O)(C1=C(SC)CCCC1)NCC1CCN(C(c2c(CC)csc2)=O)CC1C 86949,C1(OC)(OC)CCN(CC(=O)Nc2ccc(Cl)cc2SC)CC1O 86950,c1(CCC(N2CCCC(N(C(=O)Cc3ccns3)CC)C2)=O)cccc(C#N)c1 86951,c1(SC)ncc(C(=O)NC2CN(C(C3CCC(C)(C)C3)=O)CCC2C)c(O)n1 86952,C1(Cn2cc(CCCCC)nn2)CCCN(C(c2cnccc2CC)=O)C1 86953,N1(C(C(C)CO)=O)CCC2(CCC2)C(CNC(=O)Cc2cc(C(F)(F)F)n(C)n2)C1 86954,Cc1cc(=NC(=O)C2CC(F)CN2S(=O)(=O)Cc2cccc([N+](=O)[O-])c2)cc[nH]1 86955,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cnc[nH]3)CC12 86956,C1(C)(C(N(C2CCCN(C(=O)Cc3cn[nH]c3)C2)CC)=O)CCC2(CC1)CC2 86957,N1(C(=O)CC2COCCN2C(=O)Cn2cc(CO)nn2)CCC2(CC1)OCO2 86958,CC1=C(C(=O)N2CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C(F)C2)CCO1 86959,C(c1cc(Cl)sc1Cl)=CC(N1CCC2C(NC(C3C(C)(C)C3)=O)C21)=O 86960,C(c1ccc(C#N)cc1)=CC(=O)NC1(CN(C(C2CC(C)SCC2)=O)C)CC1 86961,Cc1cc(O)nc(C)c1C(=O)NCCC1(CNC(C2(C)CCNC2=O)=O)CC1 86962,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OCC1 86963,C1(OC)CC(NC(C2(C)CCCS2)=O)CN(C(=O)C(=O)NC2CC2)C1 86964,C(N=c1cccc(S(=O)(=O)N(C)CC2(OC)CCOC2)[nH]1)c1ccc(NCC)o1 86965,N1(C(c2cnc(C)s2)=O)CCC2(CC1)CC2(C)C(c1ccccc1)NCCC#N 86966,Cc1cc(Cl)c(CN(C=O)Cc2ccoc2)cc1[N+](=O)[O-] 86967,c1(OC)cc(NC(C2CC(NCc3cc(C)cc(O)c3)C2)=O)nc(Cl)c1 86968,c1(C(C)N(C23CCC(CC2)C3)C(N2CCC(F)(C(F)(F)F)C2)=O)ccc(Br)cc1 86969,C1(C(N2C(Cn3cc(S)nn3)CCC2)=O)CC2(C1)CC2(F)F.CS(=O)(=O)NCC=O 86970,CC1(C)CC(CO)CN(C(CCC2CC2)C(=O)NCc2ccccc2Br)C1 86971,N1(CC)CCN(C(C2CSCCN2c2ncc(F)cn2)=O)CC1=O 86972,c1(CCC(=O)N(C2CC(NC(CC3(OCC)CC3)=O)C2)C)cc(Cl)ccc1F 86973,C(=O)(C#CC(C)(C)CNC(=O)OC(C)(C)C)Nc1ccc(C)cc1Br 86974,N1(C(C(F)=CC)=O)CCN(C(=O)Cc2cnn(C(C)(C)C)c2)C2CS(=O)(=O)CC12 86975,C1(NC(=O)CSc2ccccn2)CN(C(C2CC(n3cnnc3)C2)=O)C2CC12 86976,C(=O)(CCCCC(N)=O)NC1(C)CCN(NCCc2nc(C(F)F)no2)C1 86977,C1(NC(c2nnc(C)s2)=O)CCC2(CCN(C(C3CC(C)(O)C3)=O)C2)C1 86978,N(C)(C1CCc2c(OC)cccc21)CCN(C(c1cccc(OC)c1)(C)C)C1CC1 86979,C(COC)(CC(=O)NCC1(CC)CC1)NC(C(C)=CC=C)=O 86980,c1(C(N2CCCC(C)(NC(C(C)=C3CCCC3)=O)C2)=O)ccn2cc(C)nc2c1 86981,C1(C(=O)NC(CCOC)(C)C)(C(C)C)CCCN1C(C1CCC(C)CC1)=O 86982,c1(N2CCCN(CCC)CC2)nc(=NCC2CNC(=O)C2)[nH]c2cc(C)ccc12 86983,CCCCC(O)CC(=O)NCC(C1CCCCCC1)NC(c1ncccc1Cl)=O 86984,C1(n2cc(CN(C)CCOC(C)(C)C)nn2)CCCCCC1O 86985,N1(C(CCC(C)OC)=O)CC2CC1CCC2NC(=O)CC1CCCCC1C 86986,C(=O)(CC(C)(C)C(F)F)NC(CCCC)CNC(c1cc(C2(O)COC2)on1)=O 86987,C(c1cn(C)cn1)=CC(=O)N(C)CCOCCNC(C1C=CCCC1)=O 86988,Cc1nc[nH]c1C(C(=O)NC(=O)C(F)C1CCCC1)NC(c1cc(C(C)C)[nH]n1)=O 86989,c1(NC(C2(C)CCN2c2ncncc2I)=O)cccc2ncsc12 86990,Cn1ccc(CCNC(C2CC(C)N2C(=O)Cc2ccc(Cl)s2)=O)n1 86991,c1(N2CCCC(C(=O)OCC)C2)ncc(F)c(OC)n1 86992,C#Cc1ccc(CC(N2CCC(NC(=O)Cc3c(C)noc3Cl)C(CO)C2)=O)cc1 86993,c1(OC)ccnc(C(N2CC(O)(CNC(=O)CC3C=CCC3)C2)=O)c1F 86994,C1(C(N2CC(O)(C(C)NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)CCC(C(C)C)CC1 86995,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1CC(N)=O)=O 86996,c1(C(N2C(CN(C)C(C3CN(S(C)(=O)=O)C3)=O)CCC2)=O)cccc(O)n1 86997,Cc1cnc(NC2(C)CC2)c(S(=O)(=O)NCCC(C)c2cn[nH]c2)c1 86998,c1(OC)cc(C(=O)NC2CCOCC2N2CCCCC2)c2ccccc2c1 86999,C1(CCN(C(CC)C(=O)NC2(OC)CC2)CC)CCN(C(=O)C(C)(C)CSC)CC1 87000,c1(CC)cc(=NC(CNC(c2coc(COCC)n2)=O)c2ccccc2)[nH]c(Cl)n1 87001,c1(C(N2CC(NC(C3C(C)(C)C3)=O)C(F)CC2)=O)ccc2c(c1)OCCO2 87002,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NCc3ccncc3)C2)=O)c1 87003,N1(C(CC(CC)SC)=O)CCC(O)C(NC(=O)C(C)(C)CBr)C1 87004,C(=O)(CC(C)(C)N(C)C(c1sccc1CO)=O)N(C)CC1CCOC1 87005,CC(Cn1cccn1)N=c1cccc(S(=O)(=O)NC2CC3CCCCC23)[nH]1 87006,C(=O)(CC1=CCN(C(=O)CCC2(C)CCCN2C(=O)C(C)N=[N+]=[N-])CC1)OC 87007,c1(NC(CC2C(NC(C=CCOC)=O)CCCC2)=O)cc(C2CC2)ccc1C 87008,Cc1sc(C(=O)NCC2CCN2C(=O)C(C)(C)c2ccccc2)nc1O 87009,N1(C(c2cc(OC)ns2)=O)CCC(C)N(c2ncnn3c(Br)ccc23)CC1 87010,c1(OC)ccc2nc(S(C)=O)[nH]c(=NCc3cnn[nH]3)c2c1 87011,c1(CC(=O)NCCN2CCN(C(c3c(C)onc3)=O)CC2)ccc(Cl)cc1Cl 87012,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(C(C2CC2)OC)=O)C(C(F)F)C1 87013,Cn1cncc1C=CC(=O)NC1C2CN(C(=O)C(N3CCSCC3)=O)CC12 87014,Cc1ccc(C(=O)NCCCCCCNC(C2CC(C)(C)C2)=O)nc1C 87015,C#Cc1cnn(C)c1C(=O)NCC1CN(C(C2CN(C)C2)=O)C2CC12 87016,C1(N(C)C)CN(C(=O)CC(C)SC2CCC2c2nc[nH]n2)CC1O 87017,c1(C(N(C2CC(NC(C(C(CC)CC)C)=O)C2)C)=O)cnn2cccc(OC)c12 87018,CN1CCc2[nH]nc(C(=O)NCC3C=CCN3C(=O)CCCC(F)F)c2C1 87019,CCC(C)C(C(=O)NCC1CN(C(C23CC(C)(C2)C3)=O)CC1(C)C)OC 87020,C(=O)(C(C)CC(F)(F)F)Nc1c(C)cc(NC(C2(N(C)C)CCC2)=O)cc1 87021,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NCC(CC)N(C)C)CCSC1 87022,c1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C2)ccc(-n2cncn2)nc1 87023,N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(N(C(=O)C(O)C(C)C)C)C2(CC2)C1 87024,c1(OC)ccc2nc(N3CC4CSCC(C4)C3)nc(N3CCC4(CCO4)C3)c2c1 87025,N1(C(c2c(C)n(C3CCC3)nn2)=O)CCC(CNC(=O)Cn2cncn2)C12CC2 87026,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87027,c1(CC(=O)N(C2CN(C(C3(CN(C)C)CC3)=O)C2)C)ccn(C2CCOCC2)n1 87028,O=C(C1=CS(=O)CCC1)NCCNC(C1(C(F)(F)F)CCCCC1)=O 87029,O=C1CC2CCCC2(C(N2CCCC(NC(c3cc(CO)ccn3)=O)CC2)=O)C1 87030,c1(N(CC(=O)O)C=O)ccccc1.c1(C(COC(=O)C2CC2)=O)snnc1C1CC1.C 87031,Cc1cc(N(C)CC2CC(Cl)(Cl)C2)nc(N2CC=CCC2)n1 87032,N1(CC(=O)NCC2CCCC2C(N2CC(O)(c3nn[nH]n3)C2)=O)CCOCC1=O 87033,C(N=c1ccnc(C)[nH]1)C1CC(NC(Cc2c(C)ccc(C)c2)=O)C1 87034,c1(C(=O)NC2C3(CN(C(c4occ(C)c4)=O)C3)CC2)coc(S(=O)(=O)N(C)C)c1 87035,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87036,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87037,N1(C(C(C)=C(CC)C)=O)CC(CO)C2(C1)CN(C(c1cc(Cl)cn1CC)=O)C2 87038,C1(C(N)=O)CN(C(=O)COc2cccnc2)CCO1.C12CCC(O1)CNC2=O 87039,c1(OC)ccc(OCCCNC(=O)N(c2ccc(F)cc2)C2CC2)cc1 87040,OC1CCCCN(Cc2ccc(OCCn3nccn3)cc2)C1 87041,CCC(CNC(=O)C(C)OC(C)=O)(CC)C(=O)Nc1ccc(O)c(Cl)c1 87042,C(=O)(C#CC1(C(F)(F)F)CC1)NC1C(CNC(CCCN(C)C)=O)CCC1 87043,N1(C(=O)CSc2nc[nH]n2)CCCC2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 87044,CC1CN(C(=O)CS(=O)(=O)N(C)CCO)C(C)CN1C(c1cnn(C(F)F)c1)=O 87045,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)NC2(CCO)CCOCC2)C1 87046,CCCCN=C(NCC(C)Sc1ccccc1)N1CCC(COC)C1 87047,C1(C)(CC(=O)NC2CCC(C(=O)NCC(C#C)CC3CC3)C2)CCCCC1 87048,c1(C(N(C)CCN2CCN(C(c3cn[nH]c3)=O)CC2)=O)ncc(F)cn1 87049,N1(C(C)=O)CCCCC1C(=O)NC(C)CCNC(c1cnc(NC(C)=O)cn1)=O 87050,c1(OC)cc(NC(N2CC3CC2CN3Cc2cncn2C)=O)c2ccccc2c1 87051,C1(C)(CNC(C2C(OCC)C2C)=O)CCN(C(C2CNC(=O)N2)=O)CC1 87052,N1(C(C(CC#C)N(C)C)=O)CC2N(C(=O)C(C)CCC(=O)OC)CCC2(C)C1 87053,C1(F)(C(=O)NC2CC(CNC(c3c(COC)noc3)=O)C2)CCCOC1 87054,c1(CN(c2cc(C(N)=O)cc(C3CC3)c2)C)sc2ccccc2c1C(=O)O 87055,c1(C(=O)NC(C)CN(C)C(c2c[nH]nc2-c2ccccn2)=O)cc(N)cc(O)c1 87056,C(=O)(C#CC1CCCOC1)NC(CNC(c1ccc(C(=O)NCCC)cc1)=O)C 87057,C12(C(N3CCC(NC(=O)C=CC=C(Cl)Cl)C3)=O)CCOCC1C2 87058,C1=NC(=O)C2C1CN(C(=O)C(O)CC1CC1)C2.N1(CC)CC(n2cnnc2)C1 87059,Cc1cccc2[nH]cc(CC(N3CC(NC(=O)Cc4ccsc4Cl)C(C)C3)=O)c12 87060,c1(C(=O)OC)c(NC(C2CC2C(=O)OC)=O)cc(C#N)c2ccccc12 87061,N1(C(C(N2CCSCC2)C)=O)CC(NC(c2ccc(F)s2)=O)CCC1C 87062,C1(CC=C)(NC(=O)C(F)C2CCOC2)CN(C(C2CCCN2CC)=O)C1 87063,N1(C(CCN(C(C2CC(CN=[N+]=[N-])C2)=O)CCO)=O)CC2CC1C2SCC(N)=O 87064,C1(C(N(C)OC(C2(CC)CCOCC2)=O)=O)Cc2nccn2C1 87065,c1(NC2CCCN(C(=O)OC)C2)nc2cc[nH]c2c(=NC2CC=CCC2)[nH]1 87066,C1(C(=O)NC(CCCCNC(C(C)NC(=O)NC)=O)(C)C)COc2ccccc2C1 87067,c1(C(=O)NC2CN(C(CSCC)=O)CC2(C)C)sc2ncccc2c1Cl 87068,N#Cc1cccc(OCC(=O)NCCCCCCNC(C2CCC(F)(F)C2)=O)c1 87069,CC1(C)NC(=O)CC1C(N1CCC1CNC(C1CCCC1)=O)=O.C1(=O)CCN1 87070,C(=O)(C(CCC(N)=O)N(C)C)N(C(C)CCNC(=O)CCc1ccncn1)C 87071,c1(C(N(C2CCCN(C(c3c(C)scn3)=O)C2)C)=O)c(C)nc(=N)[nH]c1C 87072,C1(CNC(C2C(COC)CC2)=O)CCCCN1C(=O)CC(C)n1cccn1 87073,C(CC1=CCN(C(c2cccc3c2NCC3)=O)CC1)NC(CCC1C(C)(C)C1)=O 87074,c1(C(N2CCN(c3ncc(CC(=O)O)cc3F)CC2)=O)cc(Cl)c(Cl)c(Cl)c1 87075,N=S1(=O)CCCC(NC2c3cccc(c3)C23CCC3)C1.C(=O)C1CC1.N(C)C 87076,CCC(C)(C(=O)NCC1CC(NC(c2cc(-c3cccs3)on2)=O)C1)C(N)=O 87077,C1(OC)CCCN(C(C2(NC(=O)CC(C)O)CC(F)(F)C2)=O)CC1 87078,N1(C(c2c(C)cccc2)=O)CCC2(CC1)CC2C(=O)Nc1c(C)ncnc1C 87079,N1(C(=O)NCc2ccc(F)c(F)c2)CC2CC=CCC12 87080,C1(NC(C2CCC(C)O2)=O)CCC2(CC1)CN(Cc1cncc(F)c1)C2 87081,N1(C(c2c(CNC(C3(C(=O)OC)CC3)=O)cco2)=O)CC(C)CCCC1C 87082,N12CCCC1C(=O)N(C)CC2=O.C(=O)(CC1CCC1)NC1CCC1 87083,Cc1cc(C(=O)NCC2COC(CNC(c3cc(C(N)=O)[nH]n3)=O)C2)nn1C(F)F 87084,N1(C(CC)C)CCOCC(CNC(c2cn(C)nc2-c2ccc(C)o2)=O)C1 87085,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)CN2CCCCC2=O)C(C2CC2)C1 87086,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(-c3ccccc3)no2)=O)C(C)C1 87087,Cc1nc(NCC2=CCCOC2)cc(=NCC2CCOCC2C)[nH]1 87088,N1(C(c2oc(C)c(Br)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C(C)C1 87089,N1(C(C2(C#C)CCC2)=O)CC2COCC(C1)C2NC(C12CCCN(CC1)C2)=O 87090,C(CCCCC(=O)NC1C=CCN(C(c2cc(Cl)c(Cl)n2C)=O)C1)OCC 87091,c1(C(=O)NC(C2CCCN(Cc3ncccc3O)C2)C)cccc2nccn12 87092,C(C(C)(C)Cc1nccn1C)NC(c1nnnn1C1CCOCC1)C1(CC)CCC1 87093,c1(C(=O)NC(CN(C(c2cnc(OCC)s2)=O)C)C)cnc2[nH]cnc2c1 87094,c1(C(=O)NCC2CCCCN2C(=O)CC2CCCCO2)cncc2nc[nH]c12 87095,CCCCCC(NC(=O)CNC(N)=O)NC1(CCC(=O)OC)CCN(C(N)=O)C1 87096,N1(C(C(CC=C)CNC(C2CC2(Cl)Cl)=O)=O)CC2(CNC(=O)C2)C1 87097,N1(C(C#C)COC)CCC(C#N)(c2cccc(F)c2)CC1 87098,N1(C(c2c(C)csc2)=O)CC=CC(NC(=O)CSc2ccccc2C)C1 87099,c1(C(=O)Nc2cnc(C)s2)cc2c(-c3nn[nH]n3)cc(O)nc2o1 87100,c1(C(=O)NC2(C3CN(C(C(CC)CC)=O)C3)CC2)cc2nc[nH]c2cc1F 87101,CC(CN=C(NCC1(Cc2cccc(Cl)c2)CC1)NC1CC1)c1cccnc1 87102,CCCCC(C(=O)NCC(C)(C)OCCNC(c1ccc(F)cc1O)=O)N(C)C 87103,Cc1cc(C(=O)N(CC(O)CN(C)C(c2ocnc2C(C)C)=O)C)sc1Cl 87104,C1(NC(C2(C3CCCO3)CC2)=O)(CO)COc2ccccc2C1 87105,C(CCCC(=O)NCCN(C(c1ccccc1)=O)C(C)C)OC(C)=O 87106,N1(C(CC2(CNC(=O)CC3CCCC34CC4)CC2)=O)CC2CCCC(O)C2C1 87107,CC1CC(NCc2nn(C)c3c2COCC3)c2ncnn21 87108,N1(C(C2N(CC)CC2)=O)CCC2(C(=O)NC(CO)CCC3CC3)CCCC12 87109,n1(CC(=O)NCC2N(C(CS(CC)=O)=O)CCC2(C)C)[nH]cc2c(=O)ncnc1-2 87110,C1(NC(C23CCC(OC)(CC2)C3)=O)CCCN(C(C2(C)CCN(C)C2)=O)C1C 87111,CC1(C)CC(CC(N2CCC(CF)(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)NC1=O 87112,c1(CCC(=O)NCC(COCC=C)O)ccccc1N 87113,N1(C(CCCOCC)=O)CCC2(CC1)CCN(C(c1ccc(F)c(F)c1F)=O)C2 87114,N1(C(C(CC)OCC)=O)CCOC2CN(C(c3cccc(C)n3)=O)CC12 87115,C12(NC(C3C(CN(C)C)C3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 87116,C(CCC(C(=O)NCCC1CC(C)C1)NC(=O)C(c1cncnc1)C)OC 87117,CC(CC(=O)NC1(c2cn(C(C)C(=O)O)nn2)CCC1)c1ccncc1 87118,CC(C)C(C)C(=O)NC1(CNC(=O)CCc2coc(-c3ccccc3)n2)CC1 87119,C1(NC(=O)CC2CCCN(C(=O)CCCCF)CC2)CC2C=CCC(C1)C2 87120,C1(C(=O)NC(CCCC)C)CCC(F)(CNC(=O)C(C)CCN(C)C)CC1 87121,c1(C(=O)NCC23CCC2CCN3C(c2ccc[nH]2)=O)ccc2ccccc2n1 87122,C(=O)(CCCN(C)C)N(C1CCC(NC(C2(F)CCC2)=O)C1)C 87123,C1(F)(CNC(C(COC)(C)C)=O)CCC(CNC(c2ccc(C(F)F)s2)=O)CC1 87124,C1(NC(CSc2ccc(OC)cc2)=O)C(C)CN(C(=O)Cc2cn[nH]c2)CC1C 87125,C1(NC(=O)Cc2ccc(Cl)cc2)CCN(C(c2ccnc(F)c2Cl)=O)CC1O 87126,N1(C(C)=O)CCCC(CNC(c2sc(F)cc2C)=O)CC1 87127,C(C(=O)N1OC2CCC1C2)C1N(OC(CCCCSC)=O)CCC1 87128,CC1OC2(C(N3CCC3CNC(=O)CCN3CCN(C)CC3)=O)CC1C2 87129,N1(C(CN2C(C)CCC2)=O)CCCN(C(=O)C)CCC1.c1(OC(C)=O)cncc(Br)c1 87130,N1(C(C2N(C(CC(C)(C)N(C)C)=O)CC(=O)NC2)=O)CCC2(CCC2)CC1 87131,c1(C(=O)NC(c2cnc[nH]2)C)coc(CNC(c2ccsc2Cl)=O)n1 87132,Cc1cc(C(=O)NCCN(C(=O)Cc2cncc(C#N)c2)C2CC2)ccc1Cl 87133,O=C1CC(C(=O)NC23CCN(C(=O)CCc4ccc(F)cc4)CC2C3)CC(=O)N1 87134,c1(C(=O)NC2CC(C)N(C(c3cnc(O)nc3O)=O)C2)cc(Cl)c(Cl)cc1N 87135,C1(CC)(CNC(=O)NC(=O)C=CS(C)=O)CCNCC1 87136,Cc1cn2cc(C(=O)NC3CC3CNC(c3cnc(C(C)(C)C)s3)=O)nc2s1 87137,N1(C(C(CCC)O)=O)C2CCCC1CN(C(=O)C(C)(c1ccccc1)OCC)C2 87138,c1(CNC(C2(CC)CCN(C(C(C=C=C)C)=O)C2)=O)ccc(C#N)c(C)c1 87139,N1(C(c2ccc(C(=O)OCC)s2)=O)CCCC(Cc2ccc(C(C)=O)cc2)C1 87140,CCCCCC(C)(C)C(=O)NC(CO)CCCCNC(c1c[nH]nc1[N+](=O)[O-])=O 87141,C=CCC(C(=O)OCCC1CCC(CNC(=O)OC(C)(C)C)C1)NC(=O)C(C)C 87142,C=CCCCCCCCC(=O)NCC1CC1CNC(=O)CC1CCCC(CC)C1 87143,c1(OCC)cccnc1C(=O)NCCCCNC(C1(C)CCC(=O)N1)=O 87144,CC(C)CCC(O)C(=O)NCCCCC1CCN(CCOCCOC)CC1 87145,c1(OCOC)n[nH]c(=NC(=O)Nc2ccc(-c3ncc[nH]3)cc2)s1 87146,N1(C(C(CC)CN(c2nocc2Cl)CC)=O)CCCC(C)(NC(=O)C2CC2)C1 87147,c1(CC(N2CC(CCNC(=O)C(F)C3CCOC3)C2)=O)ccccc1O 87148,C1(C(=O)NC2CN(C(C=Cc3cncc(OC)c3)=O)C2)CCc2ncncc2C1 87149,C1(NC(c2occ(C)c2)=O)COC2C(NC(=O)C(F)F)COC12 87150,C1(C(=O)OC)COCCN1C(C1CCCCN1C(C12COCC(C1)C2)=O)=O 87151,c1(CC)nc(C(=O)NC(C)(C)CN(C(=O)CC2CCCCC2O)C)c(C)o1 87152,c1(C(=O)NC2(CNC(c3n[nH]cc3F)=O)CCOC2)cnn2c1OCCC2 87153,c1(CC)cc(NC(=O)CCC2CC(NC(=O)COC3CCC3)C2)ccc1F 87154,N1(C(C(C=CC)O)=O)CC2CC1(C(N1CCC(C(C)C)CC1)=O)C2 87155,C1(CNC(c2ccc(C#C)cc2)=O)COC(C)(C)CN1C(=O)C(C(C)C)N(C)C 87156,C1(N(C(=O)CSCC(=O)O)C)CCN(CCc2ccccc2)CC1 87157,c1(CC)ccc(C(N2CC(CNC(=O)Cc3n[nH]c(C)n3)C(C)C2)=O)c(F)c1 87158,C1(NC(CCOC(C)C)=O)CC2CN(C(=O)CC3CCCCC3(C)C)CC2C1 87159,CC1CN(C(=O)C=C2CCCC2)CCN(C(c2ccc(C3CCOC3)s2)=O)C1 87160,n1(CCC(N2CCC(O)(C(C)NC(c3nc(C)oc3)=O)C2)=O)ccc(O)nc1=O 87161,N1(C(c2c(OCCC)cccc2)=O)CC(NC(=O)C(C)n2cccc2)CC(C)C1 87162,C=CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)CCc2cnn[nH]2)C)C1 87163,C1(CC)CN(CC(C)C)CCN1Cc1c(C)coc1CBr 87164,c1(C(=O)NCCCC(C)NC(=O)CC2CCCC(C)(C)O2)nn(C)c2c1CCC2 87165,Cc1nn(C)c(O)c1CNC(=O)NCc1ccnn1C1CCCCC1 87166,C1(NC(C(c2ccccc2)OCC)=O)CCN(C(c2cccnc2C)=O)CC1C 87167,N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C=CC(=O)NC2CC(=C3CC3)C2)CC1 87168,C1(C(N(C2CCN(C(=O)CC3CCC(O)C3)CC2)CC#C)=O)CCN(C)C(C)C1 87169,C1(O)(C(=O)NCCCN(C(c2c(C)cns2)=O)C(C)C)C2CC3CC(C2)CC1C3 87170,C(C(CC(C)C)C(=O)NCc1nc(C(N)=O)co1)NC(CC(=C=C)C)=O 87171,C1(CNC(C2CCCN(C(C(C)C)=O)C2)=O)CN(C(=O)CC2(C)CC2)CCCO1 87172,N1(C(C2C(CCOC)C2)=O)CC(NC(C2CC(C)(C(C)=O)C2)=O)CC2(CCC2)C1 87173,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87174,C1(C(=O)NCC(C(C)C)NC(C2(c3cncnc3)CCCC2)=O)CCC(C)CC1 87175,c1(C(=O)NCC2(NC(C34CC(C#N)(C3)C4)=O)CC(OC)C2)ccc2ccoc2c1 87176,c1(OC)nc(NC(C2CC2NC(c2scc(C)c2Cl)=O)=O)cnc1C#N 87177,c1(C(N2C3C(NC(C(C)O)=O)CC(C3)C2)=O)nccc2n[nH]cc12 87178,C#CCCC(O)C(=O)NCCC1(NC(c2cc(C(N)=O)cnc2O)=O)CC1 87179,C1(OCC(N)=O)CCN(C(=O)CCOC2CN(C(C3CC(CCO)C3)=O)C2)C1 87180,N1(C(C=CCCC)=O)CC2(CCCN(C(C)=O)C2)C1.C1(CO)CC2CN1C2 87181,C1(C(=O)NC(C2(O)CN(C(c3nc(OC)oc3)=O)C2)C)CC(C)(C)C(C)(C)C1 87182,c1(N2CC3CC(=O)NN3CC2)nc(N2CCN3C(=O)OCC3C2)c2cnn(C)c2n1 87183,C12CCCN(CC1)C2=O.C(CS(=O)(=O)C(C)C)n1cc(CCCC)nn1 87184,c1(C(=O)NCC2CN(C(C3OCCO3)=O)CCO2)ccc2c(F)cc(F)cc2n1 87185,CC1CC(C(N2CC(CO)(NC(=O)CCc3ccc(F)cc3)C2)=O)CCO1 87186,N1(c2nccc(C(=O)OC)n2)CC2(CCCC2NC(=O)CCC(C)C)C1 87187,Cc1cc2ccc(C(=O)NCC3CN(C(C4CC(=O)N(C(C)C)C4)=O)C3)cn2c1 87188,Cc1cnc(NC2CC(NC(=O)Cn3nc(O)ccc3=O)C2(C)C)nc1O 87189,c1(C(N(CCN(C(c2cccc(C)c2)=O)C(C)C)C)=O)ccc2nn[nH]c2n1 87190,C1(C(=O)OC)CN(C(C2(C)CC(OC(C)(C)C)C2)=O)CCN1.C(=O)OC 87191,CCC(C)C(C(=O)NCc1cc(OC)nn1C)NC(=O)CC1CC1C(C)C 87192,N1(C(C(=O)NCCC2(C)CC2)CCc2ccccc2)CCC(S(=O)(=O)C(F)F)C1 87193,c1(CCC(=O)NC2C(C)(NC(=O)CC3C=CCCC3)CCC2)c(F)cccc1Cl 87194,c1(OC)cc(C(N2C(C(=O)Nc3scnc3C#N)CCC2C)=O)cc(I)c1OC 87195,Cc1cccc(N(C(=O)C(=O)Nc2ccnn2Cc2ccccc2)C(C)C)c1 87196,CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)s2)CC1COC)C(F)F 87197,c1(OC)cccc2c(CC(=O)NCCN3CC=CCC3)c[nH]c12 87198,Cc1cccc(N)c1NC(C1C2CC1N(Cc1ccc(N3CCCC3)nc1)C2)=O 87199,c1(CC)onc(C)c1C(N1CC2CC2(C(=O)NCc2cccc(Br)n2)C1)=O 87200,c1(C(N(C(CC)C)C(=O)CN2CCCC(OC)C2)=O)ccc2c[nH]nc2c1 87201,c1(C(=O)NCC(C)N(C)C(c2cnc(C(F)F)s2)=O)cnn(C)c1C1CC1 87202,C1(C(N2CC(C=C)OCC2)=O)CC(O)C(O)CC1CNC(C1(CSC)CCC1)=O 87203,c1(C(=O)NCCCNC(C=Cc2ccc(C3C(C)C3)o2)=O)cc(N)c(Cl)c(O)c1 87204,Cc1cc(N)c(C(=O)NCC2CN(C(c3ncccc3Br)=O)CCO2)cc1F 87205,c1(C(=O)NCC2(OC)CCN(C(=O)C=C(Cl)Cl)C2)ccc2c(c1)OCC2 87206,C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(=O)Cc1ccnc(OC(C)(C)C)c1)C2 87207,c1(C(=O)NCC(C(C)C(C)C)NC(Cc2cnc(C)[nH]2)=O)cc2ccccc2o1 87208,c1(C(C(=O)NC(CNC(C(CC)OC2CCCC2)=O)CO)F)ccc(C)cc1 87209,c1(CC)cc(CC)nc(C(=O)NC(CS(C)=O)C(C)(C)C)n1 87210,C1(NC(CC(c2ccc(OCOC)cc2)C)=O)CCNCC12CC2 87211,CC(CCC(=O)NC(C(=O)NC)C1(C)CC1)NC(=O)COCCN(C)C 87212,C(C1=CCCN(C(C2C3CCCOC23)=O)C1)NC(=O)Cc1cnco1 87213,c1(NC(C2CCN(C(c3cnn(CC)n3)=O)C2)C)ccnc(S(C)(=O)=O)n1 87214,C1(CN(C)C(c2cccc(O)n2)=O)CCCCN1C(C1(C)CCC(=O)C1)=O 87215,c1(C(=O)NCC2C(C(=O)NCC(=O)OCC)CCC2)ccccc1C(F)(F)F 87216,C1(C(=O)NCCN(CCOC)C)CC2CC2N1C(=O)CC1OCCCO1 87217,c1(C(=O)NCCC(=O)N(C2(C(N)=O)CCOC2)C)ccc(CC#N)cc1 87218,c1(CNC(=O)CCOc2ccc3cccnc3c2)cccc2c1OCCO2 87219,C1(C(=O)NCC2CC2C(=O)NOCCCC2CC2)C=CCOC1 87220,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3nc[nH]c3c2)=O)C1 87221,c1(C(=O)OC)cccc(C(=O)NCC(C)CNC(C2CCCC3CC23)=O)n1 87222,C1(NC(CNC2(F)CCN(C(C3C(C)C3)=O)C2)=O)CC2C=CCC(C1)C2 87223,N1(C(C2N=C(C)SC2)=O)CCC(C(C)NC(c2sc(C)nc2C(F)(F)F)=O)CC1 87224,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SC)=O)CC1CC1 87225,C=CCCCCC(=O)NC1COCC1CNC(c1c[nH]c(Br)c1)=O 87226,N1(C(c2occ(C)c2)=O)CC2OCCN(C(c3cnn(CCF)c3)=O)C2C1 87227,C(C1=CCCOC1)N(C(CC1N(C(C(CN(C)C)O)=O)CC1)=O)C 87228,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(c2cnc[nH]2)C)[nH]c1C 87229,c1(OCC)cncc(C(=O)NC2CC3CC3N2C(=O)Cc2nc(C)c(C)s2)c1 87230,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)COCC3CCCCC3)CC2C1 87231,c1(CCC(=O)NCC2(CNC(=O)Cc3nnc(O)s3)CCC2)ccccc1F 87232,C1(NC(=O)Cc2cscn2)CC2(C1)CN(C(c1ncoc1C1CC1)=O)C2 87233,Nc1ccc(C(=O)C(=O)NCC2CCN2C(C2COCCN2C(N)=O)=O)nc1 87234,C1(C(=O)NC2CCCC(CNC(COCC(=O)OCC)=O)C2)CN(C)CC(C)O1 87235,N1(C(CNS(C)(=O)=O)=O)CC(CNC(C2CCCCN2C)=O)C(O)C1 87236,c1(C(=O)NC(C2CCN(C(CCC(=C)C)=O)C2)C)cn2ccccc2n1 87237,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(C3CC34CCOCC4)=O)C2)n1 87238,c1(CNC(NC(CC)C)=NCC2CN(C)CCO2)ccc2c(c1)CCCC2 87239,c1(C(=O)NC(C(N2C(CC)CCC2)=O)Cn2cncn2)cccc(O)c1F 87240,C=Cn1nccc1C(=O)NCC1CCN(C(=O)Cc2cnn(C3CC3)c2)C1 87241,CCCCCCCCC(=O)N(CCC(N1CCC2(CO)CCCC12)=O)CCC 87242,c1(OC)ncc(S(=O)(=O)NCC(c2ccccc2Cl)N)cc1Cl 87243,C1(C(N2CC(CC)N(C(c3ccc(C)n3C)=O)CC2)=O)CN2CC3CC2(CO1)C3 87244,N1(C(C(C2CC2)SC)=O)CCC(CNC(c2ccc(Cl)c(CO)c2)=O)C12CC2 87245,Cc1csc2ncnc(N3CCCC(C(=O)Nc4cnnn4C)C3)c12 87246,c1(CC(=O)NC(C)CCNC(c2csc(-c3cnc[nH]3)n2)=O)c[nH]c(=N)nc1O 87247,C12(CNC(c3cc(C)c(F)cc3)=O)CCCC1N(C(C1CC(=O)N1C)=O)CC2 87248,C(CC(F)F)(C(=O)N(C(C)C(=O)NC)C)NC(CCN(CCC)C)=O 87249,C=CCC(C(=O)NCC(CO)N(C)C)NC(=O)CCCN1CCCC1 87250,Cc1nc(NCCN2CC(CF)C2)cc(=NCc2ccc(F)cc2Br)[nH]1 87251,C1(C(N(CCOC)CCNC(=O)CC=C(C)C)=O)CCCCC1C(F)(F)F 87252,c1(COC)nc(N2CC(CNC(C3CN4CCCC3C4)=O)CC2C)cc(C)n1 87253,c1(OC)ccc(CC(N2CC3(CCC3NC(=O)CC3CCC4CC34)C2)=O)c(Cl)c1 87254,c1(C(=O)NC(CNC(CC2(CC=C)CCCC2)=O)C(C)C)coc2c1COC2 87255,N1(C(CC(CC)(F)F)=O)CC2CCN(C(c3ccc4sc(C)nc4c3)=O)CC2C1 87256,c1(C(C)NC(c2cc(-c3n(CC)ncc3)[nH]n2)=O)cc(F)cc(Cl)c1 87257,c1(NC(c2cccc(CCC)c2)C(=O)NC2C(N(C)CC)C2)ccc(C#N)cc1 87258,c1(CC)nn(C)c(CC(=O)NC(C)C(CO)NC(=O)C(O)Cc2cnc[nH]2)c1Cl 87259,N1(C(C2CC=C(C)CC2)=O)CCC2C(C1)CN2C(c1cc(C)cnc1C)=O 87260,C(c1c(C)nn(C)c1Cl)=CC(=O)NC(CC)(C)CNC(C1CN2CCC1CC2)=O 87261,C1(CO)CCN(C(C2CCCCC2OCCN(C(CNC(CC)=O)=O)C)=O)CC1 87262,N1(C(c2ncc(C(=O)OC)nc2)=O)CCC2(CCN(C(=O)CNC(N)=O)C2)C1 87263,c1(C(=O)NC(C(C)NC(=O)C(C)(Cl)Cl)CO)cccc2c1OCC2(C)C 87264,CC1CCN(C(C2CCC=CO2)C(=O)Nc2ccc(Cl)cc2F)CCS1 87265,FC1CN=C(N2CCCCC2CC2CC2)N1 87266,C(=O)(C1CCCc2ccccc21)NCc1ccc(-c2ccc3[nH]nc(CC)c3c2)o1 87267,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87268,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(C(C)(C)C)c[nH]c1)=O 87269,c1(OC)ccccc1OCC(N1CCC(N(C)C(C2C3CCCC23)=O)C1)=O 87270,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(C2CC(CCC(=O)NC)C2)=O)CC1 87271,Cc1cnn(C)c1CC(=O)NCC1(CNC(C2CC2Cl)=O)CCCC1 87272,CCC(C)(C(=O)NC1(CCNC(C2CCCC2(C)C)=O)CCC1)OC 87273,c1(CNC(c2ncn(C)c2)=O)ncc(C(=O)NCCOCC2CCC2)cn1 87274,C(CNC(c1ccsc1)=O)(CC(C)C)NC(C(C)OCCCCCC)=O 87275,c1(N(C)C)cnccc1C(=O)NC1CCCC(NC(=O)CC2CCCCO2)C1 87276,C(C)(CCCC(=O)NC(C1CC(C)(C)C1)C)NC(C(CSC)OC)=O 87277,C(=O)(CCS(C)(=O)=O)N(C)Cc1ncoc1-c1cn(C2CCCC2O)nn1 87278,C(=O)(C1=C(Cl)CCCC1)N(C)CC1N(C(CC(OCC)OCC)=O)CCCC1 87279,N1(C(c2ccc(CC)s2)=O)CCN(C(=O)Cn2ncnn2)C(CC)C1 87280,c1(OC2CC2)cccc(Cl)c1.C1(C)C(=O)N2CC(C2)N(C)C(=O)CCN1C(=O)NC 87281,CC1(C(=O)NCC2(C)CN(C(C3CC(O)C3)=O)C(C)(C)C2)CCc2ccccc21 87282,N12CC3C4CCC(C3C1)N(C4)S(=O)(=O)c1ccccc12.C1(F)(C(N)=O)CC1.C=O 87283,N1(C(Cc2ccn(C)n2)=O)CC2CCC2(CC(=O)NC(C)(C)CF)C1 87284,N1(C(C(C)c2cc[nH]n2)=O)CCC(C(O)CNC(=O)C=CCC2CCCCC2)CC1 87285,CC1(C)CC(NC(c2ccc(F)s2)=O)CN(C(C23CCC(=O)N2CCS3)=O)C1 87286,C1(CNC(C2CCCC2(F)F)=O)CN(C(c2csnn2)=O)CC12CCC2 87287,c1(OC)ccc2cc(C(N3CCOCC(NC(=O)C(F)C(C)(C)O)C3)=O)sc2c1 87288,N1(C(C2(c3ccno3)CCC2)=O)CCCC(N(C(=O)Cc2cncnc2)CCF)C1 87289,Cc1ccc(C#N)cc1S(=O)(=O)N1CC(C(=O)Nc2c(C(F)(F)F)cccc2Br)C1 87290,CC#CCC(C(=O)N1CCCC(CC)(COC)C1)NC(=O)C(CCC)N(C)C 87291,c1(OC)ccc2c(c1)c(C(c1nnnn1C1CCC1)NC1CCC(Br)C1)nn2C 87292,C(=O)(C(C)CNC(C1(C)CCC1)=O)N(CCCN(C(C)=O)C)C(C)C 87293,c1(OCC(=O)NC2C3CN(C(=O)CC4C=CCCC4)CC23)cc(F)cc(F)c1 87294,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(Cl)cc2)CC1 87295,C1(CCC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)CC1CCC1 87296,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87297,C1(NC(C(CC#C)C2CC2)=O)CC2CC1N(C(c1ccoc1Br)=O)C2 87298,C(=O)(C(CCC1CCC1)NC(=O)CC1CCC(=O)NC1)NCc1ccn(C)n1 87299,c1(C(=O)NC2CN(C(=O)COc3ccc(F)cn3)C2)cccc2ncc(Br)n12 87300,C1(C(N2CCC(C(=O)OC)C2C)=O)CCC(O)CN1C(=O)CN1CC2CCC1C2 87301,N1(C(CC(C)CN(C)C)=O)CCCN(C(=O)CCc2ccccn2)C(C(C)C)C1 87302,C(CC(F)F)(C(=O)N1CCOC(CN(C)C)C1)N(C(C=CC(CC)C)=O)C 87303,c1(C(C(=O)Nc2cccc(C#C)c2)(C)OC)ccc2c(c1)OCO2 87304,N12CCC(C)(CC1)C2=O.CCCC=CC(=O)NCC1(C(=O)OC)CC1 87305,N1(C(C2C(C(=O)OC)C2)=O)CCC(C)(C)CC1C(N1CCCC(C)(CO)CC1)=O 87306,c1(NC(=O)NC(CC)C2(c3cc(C)cc(C)c3)CC2)ccc(Br)cc1C(F)(F)F 87307,C12COCCN(C1)C(=O)C2.C(C(=O)NCCN(C)CCOC)=CCC 87308,c1(C(C)=O)cccc(OCC(N2CCC(C)C2CNC(=O)C(C)(Cl)Cl)=O)n1 87309,c1(CC(C)NC(C2(CNC(c3c[nH]c(=S)cn3)=O)CCOCC2)=O)cccc(F)c1 87310,Cn1c(NC(=O)C(O)C(c2ccccc2Cl)O)nnc1C1CCCCC1 87311,C(C)(C)(CCNC(=O)CCc1scnc1C)NC(C1C(C)(COC)C1)=O 87312,CC1(C)CCCCN(C(C2N(C(=O)CC3OCCCO3)CC23CCCC3)=O)C1 87313,C1(C(N2CC(C)C(CNC(C3(F)CCCCC3)=O)C2)=O)Cc2c(F)cccc2O1 87314,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87315,C1(CN2CC(CC(=O)NC3(C(C)C=O)CCC3)C2)CCCOC1c1cn(C)nn1 87316,C=CC1(O)CCN(C(=O)CC(C(C)OC)NC(c2cncc(CC)c2)=O)C1 87317,C(=O)(C(C1=CCSC1)N1C(C)CCCC1C)NCCCCCS(=O)(=O)C(C)(C)C 87318,c1(NC(N(C(C)C2CC2)Cc2ccccc2Cl)=O)ncc(Cl)cc1[N+](=O)[O-] 87319,C(C(C)(C)CC1CN(C(=O)C(C)(C)C)C1)NC(C1(CSC)CCC1)=O 87320,c1(OCC)cccc(C(N2CC(F)CC2C(=O)NCc2cnc(C)o2)=O)c1 87321,C(C(CC(=O)NCCCCC1CC1C)NC(C)=O)OC.C1(=O)CN1 87322,c1(NC(N2CCN(C3CCOC3)CC2)=O)cncc(-c2ccnnc2)n1 87323,c1(C(=O)NC2CCC(n3ccnn3)C2)ccc(CCc2ccccc2)cc1 87324,C1(C(=O)NCc2nccc(OC)c2)CC12CCN(c1nc(Cl)ncc1F)CC2 87325,CC(C(=O)N(C1CC(CO)C1)C)C(C)NC(=O)CCc1cnn[nH]1 87326,CCCC(C)(C)C(=O)NCc1cnn(C)c1C(N1CCCC1(C)CCCO)=O 87327,CC1CCC(O)C(NC(=O)CC2(N(C)C)CCC2)C1.c12occc1CNC2=O 87328,N1(C(C(c2ccc(C)cc2)=O)=O)CCC2C(CCCN2C(C2CCS2(=O)=O)=O)C1 87329,N1(C(=O)CSc2ccccc2)CCC2CCN(C(c3ccnn3C3CC3)=O)C2C1 87330,N1(C(CCOc2ccc(C)cc2C)=O)CCN(C(=O)C(F)=CCCF)CC(O)C1 87331,CC(C)C(CN(C)C)C(=O)NC(c1nc(-c2c(F)cccc2Cl)cs1)C 87332,c1(CC)ccc(CC(N2CC=CC(NC(=O)CCN3CCC(F)C3)C2)=O)cc1 87333,c1(CCC=O)cccc(CC)c1.C(=O)(CN(C)CC)OCCC 87334,C1(CN(C(C=CSC)=O)C2CC2)CC(C)CN(C(=O)C(N2C(=O)CCC2=O)C)C1 87335,C1(N(C(=O)CN(C2CCSC2)C)C)CN(C(=O)CC2CCC(O)C2O)CC1(C)C 87336,C(N=c1[nH]c(=NCC(C(C)C)N2CCN(C)CC2)[nH]c2c1CCCCC2)C1(C)CC1 87337,CC1(CC(N2CCC(CCNC(=O)CCCc3nncn3C)C2)=O)CC1(F)Cl 87338,c1(C(=O)NC(C2CCN(C(c3c(CC)scc3)=O)C2)C)occ2c1CCOC2 87339,C(c1cccc(Cl)c1)=C(C(N1CC(OC)C(NC(C2CCCOC2)=O)C1)=O)C 87340,N1(C(C2(C)C(C)(C)C2)=O)CC2COCC(C1)C2NC(=O)C1=C(Cl)CC1 87341,N1(C(C(CC)OCC)=O)CCCC2CN(Cc3ccc(S(C)(=O)=O)cc3)CCC12 87342,c1(C(N2CC(COC)(CNC(=O)C(C#N)C(C)C)C2)=O)nc2ncccn2n1 87343,c1(CN(C)C(C2(CCNC(=O)CCc3cncs3)CC2)=O)cccc(F)c1 87344,C1(OC)CCCC1Nc1nnnn1C1CCOC1.C1(C)CCCCO1 87345,c1(C(C(=O)NCCC(C)F)NC(C2CC(=C3CC3)C2)=O)cccnc1 87346,CCC(COC1CCSCC1)N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1 87347,N1(C(CCCCCSC)=O)CCC2(CCOCC2)C(NC(C2CC(SC)C2)=O)C1 87348,C1(CC)CCN(C(=O)C=Cc2ccncn2)C1C(=O)NC1CCC(CO)CC1 87349,N1(C(C(C)OCCN(C)C)=O)CCC(CNC(=O)C(C)(C)N2CCOCC2)C(C)C1 87350,C(CCCCCC(=O)NC(C1CCN(C(c2ccc(C(N)=O)cc2)=O)C1)C)SC 87351,N1(C(c2cn(C)c(=O)nc2O)=O)CC(CO)C2(C1)CN(C(C1CC1C1CC1)=O)C2 87352,Cc1ccc(C=CC(=O)NC(C)CN(C(=O)CC23CCCC2C3)C)cc1 87353,CC(C)C(C)CNC(CNC(=O)CC1C=CC(NC(=O)CNC=O)C1)=O 87354,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87355,C12(C(=O)NC(CN(C(c3n(CC)cc(Cl)c3)=O)C)C)CCC(F)(CC1)CC2 87356,C(=O)(CCC(C)N(C)C)N(C1CCC(C(NOCC(=C)Cl)=O)CC1)CC 87357,C(CCCCC(=O)NCC1CCC(C#N)C1)n1cc(C2(CC)CCC2)nn1 87358,N1(C(c2ccc(F)c(C)c2Cl)=O)CCC2(CC1)CN(Cc1c(O)cc(Br)cc1F)C2 87359,c1(CNC(C(COCC)C)=O)ccc(CN(C)C(C2(CO)CC2)=O)cc1 87360,C1(NC(c2cn3nc(C)sc3n2)=O)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87361,c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncnn3)C2)ccn2c1CSCC2 87362,C1(NC(C(=Cc2cccnc2)C)=O)CCN(C(=O)CC2(C)CCC2)CCC1CO 87363,c1(OC)ccccc1-c1nccnc1CNC(c1ccccc1)C1(OC)CCC1 87364,C(=O)(N=c1ccn(C(F)(F)F)[nH]1)C1(C)CCCN1.c1(C(=O)N)cc(O)ccc1Br 87365,c1(C(=O)NC(c2cn(C(C)C(=O)OC)nn2)CC)ccccc1[N+](=O)[O-] 87366,C(c1ccccc1)=CCN(C(=O)COCC1CN(C(=O)CC2(C)CC2)C1)C 87367,C(=O)(C1=C(Cl)CCC1)NC1CCCN(C(c2c(C(C)C)n(C)nc2)=O)C1 87368,N1(C(C(C)(C)NC(C)=O)=O)CCC(C)(Cc2cccc(-n3nc(C)cc3C)c2)C1 87369,C=CCC(C)(CC)C(=O)NC1CCCC1CNC(c1cnnn1C1CC1)=O 87370,c1(N2CCC(N(C(=O)C(C)C(F)(F)F)CC)CC2)nc(C)nc(Cl)c1CC 87371,c1(CC(=O)NCC2C(NC(=O)CCN3CCCC3)C2)nccc2ncccc12 87372,C1(NC(C2C(C(=O)OC)CC2)=O)(SC)CN(C(c2nncn2C)=O)C1 87373,Cc1nc(-c2ccco2)ccc1C(=O)NC1CCCC(NC(C2CCCO2)=O)C1 87374,C(=O)(C(C)(C)C(=O)NC1CCCC(n2cc(CNS(N)(=O)=O)nn2)C1)N(C)C 87375,c1(C(C(=O)OC)NC(=O)COC2CCCOC2)ccccc1F 87376,CC1(C)CN(C(=O)NCc2snc(C(F)(F)F)c2Cl)Cc2cccc(Br)c21 87377,C(=O)(CS(=O)(=O)C1CCCC1)NCCC(C)N(C)C(C1CC2(C1)CC2(F)F)=O 87378,Cc1nc(C(=O)NCCCN(CCCNC(=O)CSC2CC2)C)c(C)n1C 87379,C1(NC(=O)C(F)(F)n2cc(Br)cn2)COC2(C1)CN(C(C1COC1)=O)C2 87380,CC1OCCCC1C(=O)NC1(c2ccccc2)CC(NC(=O)C(C)C)C1 87381,c1(C(C)(C)C)ccnc(C(N2CC3(C2)CN(C(=O)COC(=O)C2CC2)C3)=O)c1F 87382,CCC(COC)C(=O)N(C(C)(C(=O)NC(C)C(C)(C)CN(C)C)C1CC1)C 87383,C(CN=C(NC1CC1(F)F)NC1CCCCC1)N(C)C(C1CC=CCC1)=O 87384,C(=O)(C1=CCCOCC1)N1C(c2cn(CC(=O)OC)nn2)CC1 87385,N1(C(CC(C)N(C(C)=O)C)=O)CCCC(C(N2CCC(N3CCCCC3)CC2)=O)C1 87386,c1(C(C)=O)cc(Br)ccc1NCc1ccnc(C2CC2)n1 87387,CC1(NC(=O)CC2CCSCC2)CCCN(C(c2coc(CC3CC3)n2)=O)C1 87388,C1(O)(C(c2ccsc2)NC(c2cc(OC)no2)=O)CCN(C(=O)CCC2CCC2)C1 87389,C(c1cnn(C)c1)=CC(=O)CN1C(C)C2CC2C1=O.N1(N)CCOCC1CCO 87390,N1(C(c2c(C)ncnc2)=O)CCC2(CCSCC2)CC1 87391,CC1CN(c2cc(NCCCn3nccn3)ncn2)CCO1 87392,C12(CCCCC1)CC(=O)OC2.C1C(O)COC1=O.C(C)(C)(C)O.CC(=O)O 87393,c1(C(N(C2C(C)CN(C(=O)C=C3CCC3)CC2)C)=O)coc(=O)c2ccccc12 87394,C1(C(=O)NCC2(CNC(=O)Cc3csc(S)n3)CC2)CCCC1(F)F 87395,N1(C(C(CCSC)OC)=O)CC2CC1CN2C(c1ncn(C(C)(C)C)n1)=O 87396,Cc1cc(Cl)ncc1-c1noc(N2CCCC(N)C2)n1 87397,C1(CNC(C2N(C(C)C)CCC2)=O)CCCN(C(C2CCCN2C2CC2)=O)C1 87398,C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnns2)=O)cc1F 87399,C12(C(=O)NCCCOCCNC(Cn3nc(C)oc3=O)=O)CCC(C1)C2(C)C 87400,C(CCC(=O)N1CCCC1C(=O)N(C1CCC1)C)OC(C)C 87401,CP(C)(=O)C(O)C(=O)NCCOC1CCN(C(=O)CCC2CCCC(=O)N2)CC1 87402,c1(C(N2C(C)(C(=O)NC3(COC)CC3)C=CC2)=O)cc([N+](=O)[O-])c[nH]1 87403,c1(C(=O)NC2C(C(N(CC(F)Cl)C)=O)COC2)cc2cc[nH]c2cn1 87404,c1(OC)ccc(Cl)c(C)c1OCc1cnc2n1CCC(OCc1ccccc1)C2 87405,Cc1cc(C(=O)NC(C2CCN(C(=O)C=Cc3cn[nH]c3)C2)C)no1 87406,CC(C(F)F)C(=O)NCC1COCCN1C(c1ccc(C(N)=O)[nH]1)=O 87407,c1(CNCC(CC)OCC)cn(C)nc1OC(=O)CC1C=CCC1 87408,Cc1cncc(C)c1C(=O)NC(CCN(C)C(C1CCOCC1)=O)C(C)(C)C 87409,N1(C(C(C=C)C)=O)CCNCC1.c1(CN)ccc(Cn2cc(C)cn2)cc1 87410,c1(CC(=O)N(C2CCCC2)CCNC(C2C(C)CCCO2)=O)ncc(F)cc1F 87411,Cc1nc(C(N2CC(O)C(O)C2CNC(=O)CCCc2ccccc2)=O)cc(O)n1 87412,CC1=C(C(=O)N2CC(=O)NCC2C(N2C3CCC2COC3)=O)CCCO1 87413,c1(N(CC(n2ccnc2)C)C)nc(-c2ccccc2)nc(=NC2CCSC(C)C2)[nH]1 87414,C1(C(N2CCCC(N(CCC)C)C2)=O)CCC2(CC2)N1C(=O)CC(CC)OC 87415,N1(C(Cc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCCOC)C2)C1 87416,N1(C(c2ccc(C)cn2)=O)CC2(CCOCC2)CC1CNC(=O)C(C)C1CC1 87417,C1(C(=O)NCC(CNC(c2sc(N3CCCC3)nc2Cl)=O)F)Cc2cccnc2C1 87418,C1(NC(C(n2cc(Br)cn2)C)=O)CCCC(NC(C2CC(=O)N(C)C2)=O)C1 87419,c1(C(=O)NCC(C)NC(=O)C=CCN2CCOCC2)cc2c(F)c(F)ccc2s1 87420,c1(C(N2CC(CNC(c3cnn(C)c3F)=O)OCCC2)=O)cccc2cncn12 87421,C1(CNC(C2C(C=CC)CN(C(c3ccc(O)cn3)=O)C2)=O)CCCC(C#C)C1 87422,c1(OCC(=O)N(CCN(CCC)C(C2CCC2(C)C)=O)CC)ccc(C#N)cc1 87423,C1(CCNC(c2cc(C)n(C)n2)c2n(C(C(=O)OC)C)nnn2)CCN(C)CC1 87424,c1(N)ncc2[nH]ncc2n1.C12=CC(CN3CCCC4C(O)CC34)=C(C=N1)C2=O.CO 87425,c1(C(=O)NC2(C)CCN(C(C3(C#N)CCC3)=O)C2)cc2n(n1)CCNC2=O 87426,C(=O)(C(F)CCC(C)C)ONC(CSCC(=O)NCC(CC(C)C)OC)=O 87427,C1(NC(C(C(C)C)(C)O)=O)(CO)CC12CCN(C(=O)CNS(N)(=O)=O)CC2 87428,c1(C(=O)NCCOCCNC(Cn2nnc(C)n2)=O)cccc(C(N)=O)c1C 87429,c1(OCC)cc(S(=O)(=O)N2CC3(CCCNCC34CCN(C)CC4)C2)ccc1Br 87430,c1(C(=O)NC(CNC(c2n(C(C)C)ccc2)=O)C2CC2)ncccc1C(F)F 87431,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 87432,C1(C)(CN(C)C(C2(CN)CC2)=O)CCN(CCO)CC1 87433,c1(CC(C)NC(=O)C(c2cccs2)NC(=O)CC2(O)CCC2)cncnc1 87434,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)CC1CC1C)C2.c1(O)ccc(F)cc1 87435,N1(C(C2C(=C)C2)=O)CCCCC12CC(NC(=O)CCCOCc1ccccc1)C2 87436,C1(NC(c2cc(CC)c(C)s2)=O)CC2(NC(c3sc(OC)nc3Cl)=O)COC1C2 87437,CCC(CC)C(C)C(=O)NCCC1(OC)CN(C(=O)COCC(C)C)C1 87438,Cn1cnc2nc(N3CCC(NC(C4CCCNS4(=O)=O)=O)CC3)ncc12 87439,CN1CCC(CNC(=O)C(C2CCCCC2)=O)C1c1cccnc1 87440,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 87441,C12(C(=O)NC3CC(CC(=O)NCCOCC(C)C)C3(C)C)CCC(CC1)CC2 87442,n1(CC(=O)NCC2N(C(c3[nH]n(C)c(=O)n3)=O)CCCC2)cnc([N+](=O)[O-])c1 87443,CC1CC(NC(=O)Nc2ncccn2)c2nccn21 87444,c1(CC(N2C3C(NC(C(CC)COC)=O)C(C3)C2)=O)cc(Cl)ccc1[N+](=O)[O-] 87445,C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NC2(C(=O)NCC#C)CC2)C2CCC1C2 87446,C1(c2n(CCOCC)cnc2N)NC(=O)N(CC)C2=C1C(=O)NC1(CCSCC1)C2 87447,c1(CN(CCCCO)C)cc(Cl)ccc1OC.O=C(COCCO)NC1CC1 87448,c1(C(N2C3CCC2CC(N2CC(F)C2)C3)=O)ccc(OC(F)(F)F)cc1[N+](=O)[O-] 87449,c1(C(N(C)CCN(C(=O)C(F)=CCCF)C)=O)ncoc1C1(C(C)C)CCC1 87450,c1(CCN(CC)CC)cn(CCC(=O)N(CCC(C)(C)O)CC)nn1 87451,Cc1c(NCc2ccoc2)ncnc1N(CC(C)(C)C1(O)CCC1)C 87452,C1(CC)CCOC1C(=O)NCC1(O)CN(C(=O)C(C)CN2CCCCC2)C1 87453,c12cc(F)ncc1N2.C(=O)(CC(C)(C)C)N1C(C)(C(=O)NCC(=O)OCC)CC1 87454,C1(C)(CCNC(C(CO)OC)=O)CCN(C(=O)CC(=O)NC2CC2)CC1 87455,Cc1nc(CCC(=O)NC2CN(C(=O)C(N3CCC(O)CC3)C)CC2O)[nH]c1C 87456,CCCCC(C)CCC(=O)N(CCNC(C1CCCOC1CC)=O)CCOC 87457,C1(C(N(C)CCNC(=O)Cc2cncnc2)=O)CCNC(=O)C1 87458,N1(CC(=O)N(CCCOC)C(C2CCCCC2)C)CCC(O)(C(=O)OC)CC1 87459,c1(CC(=O)NCC(CCNC(=O)Cc2cn(C)nc2C)OC)ccnc(F)c1F 87460,Cc1ccc(Br)c(NC(C2CC(NC(=O)Cn3cc(Cl)cn3)C2)=O)c1 87461,C1(C#N)(C(=O)NC(CN(C(=O)CC2CC2c2ccccc2)C)(C)C)CCOCC1 87462,CON=CC(=O)NCC(c1cnn(C(C)C(N2CCCCC2)=O)c1)=O 87463,C#CCCC(C(=O)NCc1ccccc1O)NC(=O)CN1CCC(=O)CC1 87464,n1(-n2c(C)cnc2C)ncc(-c2nc(-c3nc[nH]n3)nn2C2CCC(C)CC2)c1C 87465,Cc1[nH]c(C)c(C(=O)N(C)CCOCCN(C)C(C2(C)CCN(C)C2)=O)c1C 87466,C1(CNC(Cc2cc(C)ns2)=O)CCCCN(C(=O)C(N2CCSCC2)C)C1 87467,CC#CCCC(=O)N1CCC(CCN(C(=O)C(C)C(C)SC)C)CC1 87468,CC(C)(C)CCCC(=O)N1C(C(=O)NCCCN2CCCCC2)CCC12CC2 87469,N1(C(c2cnc(C)c(C#N)c2)=O)CC(C)CN(C(C23CC2C3)=O)CC1C 87470,N1(C(c2cn(CCC)nn2)=O)CCC(CN(C)C(C)C)CC1 87471,C1(F)(C(=O)NC(C2CCOC2)CC)CCN(C(c2ccn(COC)n2)=O)CC1 87472,N1(C(c2c(F)cccc2[N+](=O)[O-])C)CCC(C2CCC3(CC2)OCCO3)C1 87473,N1(C(CCCCN(C(C)=O)C)=O)CC2(CCCN(C(=O)C(C)(C)S(C)(=O)=O)C2)C1 87474,C(=O)(C1=C2CCCN=C2NN1)NC1CCCN(C(C2C(OC)C2C)=O)C1 87475,C1(CC(=O)NCCOCCN(C)C(c2cc(C#N)on2)=O)SC2=NCCN2C1=O 87476,C(=O)(CCCC(F)(F)F)NC(CSCC)C(=O)N(C1CCN(C(C)C)C1)C 87477,C1(N(C(CC2(NC(c3ccc(C#C)o3)=O)CC2)=O)C)CCC(C)(C)CC1 87478,c1(CC(=O)NCC(CNC(c2c(OC)n(C)nc2)=O)CO)cc(F)ccc1C 87479,N1(C(CCC#C)=O)CCC2CC2(NC(=O)CCNC(c2ccc(F)cc2)=O)CC1 87480,CN1CC(CNC(=O)CCn2cc(-c3ccc(I)cc3)nn2)C(O)C1 87481,N1(C(c2nnn(CC)c2C)=O)CC(C)N(C(c2cccc(CSC)c2)=O)CC1C 87482,C(=O)(C(C)(C)C(F)F)N(C(c1nn(CC)c(O)c1)=O)CC1(N2CCCC2)CCC1 87483,O=C(C1=CCCC1)NCCC1CN(C(C2(C3CCCCO3)CCC2)=O)C1 87484,C1(CC(=O)N(C2CCN(C(C3(CC)CC3)=O)C2)CC)CCC(=O)N1C(C)C 87485,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CN(C(=O)Cn3nc(C)n(C)c3=O)CCC12 87486,c1(OC)c(C(N2C3CCC(C3)C2CNC(C2CCOC2)=O)=O)ccc(Cl)c1C 87487,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 87488,C1(NC(C(CC)OCC)=O)CCN(C(=O)C(C)=C(C)CC)CC1 87489,C#CC1(CO)CN(C(=O)C(CC)NC(=O)CCC)C1 87490,C1(CCC)(CO)CCN(C(=O)Cc2sccc2CNC(c2cccnc2C)=O)C1 87491,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 87492,C(=O)(C(C)CCCC)NC(CCN(C(=O)CCCNC(C1CCCC1)=O)C)(C)C 87493,N1(C(c2cn3c(n2)CCC3)=O)CC2CC(C1)C2N=c1ncc2c(Br)cccc2[nH]1 87494,CC1(C)CCCCC(C(=O)NCC(c2ccccc2)NC(c2ncccn2)=O)C1 87495,CC1CN(C(C2(NC3CC4CCCC34)CCCC2)=O)CC1c1ccccc1 87496,C1(N)CCC(C2CC2)C1.c1(O)c(CN(S(C)(=O)=O)CC)cnn1C.c12cncc-1c2 87497,C12(NC(CCc3cc(C)on3)=O)CC1CN(C(c1cnn(C)n1)=O)C2 87498,N1(C(Cc2cc(C)no2)=O)CC2CCCC(NC(C3CCCOCC3)=O)(C2)C1 87499,C1(CC)CCCC1(C)C(=O)NCCN(C(C1CC(=O)N(C2CCCCC2)C1)=O)CC 87500,C1(C[Si](C)(C)C)CCCN(C(=O)NCC(c2ccccc2)CO)C1 87501,c1(C(c2nnnn2Cc2cccs2)Nc2c(C)nsc2)ccc(F)nc1 87502,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)cc3O)=O)C2)=O)c(C)n1 87503,c1(C(=O)NCCCNC(c2cc(S(=O)(=O)NC)oc2)=O)ccc2sc(C)nc2c1 87504,n1(CC(=O)NCC2(NC=O)CCC2)ncc(=O)c2ccccc12.C1CCCC12CC2 87505,Cc1ncnc(C)c1OCC(N1CCN(C(C2CC2F)=O)C(C(C)C)C1)=O 87506,c1(CC)cnc(C(N2CCC(NC(c3ncccc3C(F)F)=O)C2C)=O)cn1 87507,C=CCC(C(=O)NCc1nccn1C)NC(C1CCCC1CCC)=O 87508,c1(C(C(=O)OC)C2CCC2)cccc(C(=O)NC2CC2)c1.C12C3CN(CC13)NC2=O 87509,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 87510,CCCC(CC(=O)N(c1cscc1C)C)NC(C1CCCN(C)C1)=O 87511,c1(C(C(=O)OC(C)(C)C)N(CCCCCNC(C)=O)C)cc(COC)nc(Cl)c1 87512,C1(NC(CSCC)=O)CCCC(N(C(=O)CC2CN(C)C2)C)C1 87513,N#Cc1cnn(COC2CCC2)c1N.N12CCC(CC1)NC2=O.C12CN1C2 87514,c1(C(=O)Nc2cc(NC3CCC(CO)C3)ncn2)cccc2nc(C3CC3)[nH]c12 87515,Cc1ncnc(C(N2CCSCC2N(C)C)=O)c1C.C1(CCF)C(=O)N1 87516,Cc1cc(-c2ccsc2)ncc1C(=O)NC1CCC(NC(c2cocn2)=O)CC1 87517,N1(C(CN2CCN(C(CC3N(C)CC=CC3)=O)CC2)=O)CC(=O)NCC12CC2 87518,N1(C(c2n(C)ncn2)=O)CC2C(NC(c3cccc(Br)c3)=O)C2C1 87519,c1(NC(C2CCC(NCc3cc(Cl)cc(Br)c3F)CO2)=O)ccc2c(c1)CCC2 87520,C1(NC(C2(CCC=C)CC2)=O)CCCN(C(c2ccc(C#N)c(O)c2)=O)CC1F 87521,Cc1ccc(NC(=O)CCN(C2(c3cccc(Br)n3)COC2)C)cc1 87522,c1(NC(N(C2CCOC3(CCCCC3)C2)C)=O)ccc2c(c1)CCCCC2=O 87523,C1(NC(CS(=O)(=O)NC)=O)CC2CCC1(NC(c1cncc(C(C)=O)c1)=O)C2 87524,N1(C(CCN(C(C2(OC)CC2)=O)CCO)=O)CCC(C)CC1C 87525,C1(C(C)C)N(C(c2cnc3c[nH]nc3c2)=O)CC12CCN(C(=O)C1CC1)CC2 87526,c1(C(=O)NC(CNC(C(C)CCN(C)C)=O)(C)CO)cccc(Cl)c1Cl 87527,N1(C(C=CSC)=O)CCCC(C)(C)C1CNC(C1C2CCCOC12)=O 87528,CC(C)CCC(C(=O)N1CC(CN(C)C)C1)NC(C1CCCC(=O)CC1)=O 87529,CC(CCCNC(=O)Cc1nccn1C)NC(c1cnc(Cl)s1)=O 87530,C1(c2cn(CC(CC(C)C)OC)nn2)CCN(C(c2cc(C)co2)=O)C1N(C)C 87531,C1(C(=O)NCC=CCNC(C(n2ccc(C)n2)C)=O)CC(C2CC2)=NO1 87532,C1(OC)CC(NC(=O)C(F)n2ccnc2)CN(C(C2CSCN2C(C)=O)=O)C1 87533,c1(CS(=O)(=O)N(C(C)C(=O)N(C)C)C)cccc2nccnc12 87534,CC(C)CC(C)(O)C(=O)N(C)CC1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 87535,N1(C(CCCCOC)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CC(F)(F)C1 87536,Cc1ccc(O)c(C(N2CCC(O)C(NC(C3CC4(C3)CC4F)=O)C2)=O)n1 87537,C1(NC(c2ccc(=NC)[nH]c2)=O)CC2CN(C(c3cc(SC)oc3C)=O)CC2C1 87538,N1(C(C2(CC3CC3)CCC2)=O)CCC2(C=C(C(=O)NCCO)C2)C1 87539,C1(C(=O)NCC2(OC)CN(C(C3CN(S(C)(=O)=O)C3)=O)C2)CC2CCC1O2 87540,C1(C(=O)Nc2nnco2)CN(Cc2ccnc(-c3ccccc3CO)c2)CCN1 87541,CP(C)(=O)c1ccc(C(=O)NC2COCC2NC(=O)Cc2cn3ccsc3n2)o1 87542,c1(C(N2CC=CC(NC(CCCCSC)=O)C2)=O)cnc2n1CCCCC2 87543,CC1(C)CCCN1CCn1cc(-c2ccn(C3CCCC3)n2)nn1.c1(C=O)cnc[nH]1 87544,c1(C(CNC(C(c2ncc(CC)o2)N(C)CC)=O)C2CC2)ccc(Br)cc1 87545,c1(C(N2C3CC(NC(=O)CC4CCOCC4)(C3)C2)=O)cnc2ccsc2c1 87546,C=C(C)CC(C)C(=O)NC1CN(C(=O)CCn2nc(C)nc2C)CC1O 87547,c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)ccc(Br)cn1 87548,CCCCC(=O)C(=O)NCC1CN(C(c2cc(C)sc2C)=O)CCC1C 87549,c1(C(C(=O)NCc2ccco2)N(C(CSC)C)C)cc(C2CC2)on1 87550,N1(C(C(C)=C2CCCC2)=O)CCCN(C(=O)C=CSCc2ccco2)C(C)C1 87551,C(=O)(C1CCCc2ncnn21)N(C)CCNC(C1(C)CC2CCC1C2)=O 87552,c1(C(N2C(C(N(CC(=O)OCC)CC)=O)C=CC2)=O)c[nH]c(=O)cn1 87553,C=C(Cl)CCC(=O)N(CCC(C)NC(=O)C(C)(C)c1cncs1)C 87554,Cc1ccccc1C=CC(=O)NC1CC(NC(=O)COC2(C)CCCC2)C(O)C1 87555,C1(C(=O)NC(C2CN(C(C(C)OCC#C)=O)C2)C)CN(C(C)=O)CCO1 87556,Cc1ncccc1CC(=O)NCC1(CNC(c2cnc(C(C)C)o2)=O)CCCC1 87557,N1(C(=O)C2=NOCC2)CCN(C(=O)C(C2CCOCC2)O)C(CC2CC2)C1 87558,c1(CN2CC(C(=O)Nc3cc(OC)n[nH]3)SCC2)ccc(Cl)nc1C 87559,c1(SC)ccc(C(N2CCC(CCNC(=O)C(CO)NC(N)=O)CC2)=O)cc1 87560,c1(CNC(c2n(CCOC)nnn2)C2C3COCC23)cccc(F)c1OC 87561,Cc1ccc(-n2ccnc2C)c(CN2CCSC(C)(C)C2)c1 87562,N1(C(c2cc(C)c(N)cn2)=O)CCN(C(C2CN(C)CCO2)=O)CC12CC2 87563,c1(C(N(C2CCCN(C(=O)Cc3ccccc3)CC2)C)=O)cnc2ccnn2c1 87564,C1(C)(C(=O)NCCC2(OC)CN(C(=O)C(F)(F)CN(C)C)C2)CCOCC1 87565,c1(C(=O)NCCN(C(C2CCC(OC)C2)=O)CC)cc(O)cc(=O)o1 87566,C=CC(CC)CC(=O)N(C(C)C(=O)N(C)CCN(C)C(=O)OC)CC 87567,N1(C(C(C(C)O)(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccn1 87568,C1(C(C)NC(c2ccc(C(C)=O)o2)=O)CCCCN1C(=O)CC1CC2(CC2)C1 87569,c1(C(N2CC(C(=O)Nc3ccc(CO)cc3)NCC2)=O)cc(Br)cc(Br)c1O 87570,Cc1nc(O)nc(C)c1CC(N1CCCCC(CNC(=O)C(N)=O)C1)=O 87571,c1(OCC(=O)NCC23CCC(NC(C(C)C)=O)(C2)CO3)ccccc1[N+](=O)[O-] 87572,N1(C(CSC(C)C)=O)CCCC(C)(CNC(c2ccc(OC(F)F)nc2)=O)C1 87573,C(C)(C)(C(=O)NCC=CC(=O)NC1CC1CN(C)C)SC 87574,c1(C(=O)NCC2(C)CC(NC(C=CC(CC)C)=O)C2)cncc(OC)c1C 87575,C(N=c1[nH]c(Cl)ncc1Cl)C1CCC(NC(c2c(C)noc2C)=O)C1 87576,C1(CCC)(NC(c2n[nH]c3c2COC3)=O)CCN(C(=O)CC(C)C)CC1 87577,c1(C(=O)NC2CCN(C(Cc3c(C)cncc3)=O)C2C)ccc(P(C)(C)=O)cc1 87578,CCCCN=C(NCc1ccc(F)cc1F)NCC1CCCN1C1CC1 87579,CC(C)C(C(=O)NCC1CCN1C(C1CCC1(F)F)=O)C(C)C 87580,Cc1csn1C(=O)NCC(=O)NCCC1CCCC1.C1C(=O)N1 87581,N1(C(CCC#C)=O)CC2(CCN(C(=O)CC3CC3CSc3ccccc3)C2)C1 87582,C(CC(=O)N(C1CN(C(=O)C=C2CCOCC2)CC1O)CC)(C(C)C)OCC 87583,C1(NC(c2cnc(NC(=O)OC(C)(C)C)c(F)c2)=O)C2CCN(C)C2C1(C)C 87584,c1(C(CCO)Nc2nc(C)c(Cc3cnn(C)c3)s2)ccc2ncsc2c1 87585,N1(C(=O)Nc2ccnn2C2CNC2)CCC2(CCCCO2)C1 87586,C(c1ccc(F)c(F)c1)=CC(=O)NC(C(C(C)C)NC(=O)Cc1nnc(O)s1)C 87587,Cc1c(C(=O)NOCCn2cc(-c3cn4ccccc4n3)nn2)ccc(Br)c1F 87588,n1(CC)nc(C)cc1C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 87589,c1(C(=O)NCC2N(C(c3cc(C)ncc3C)=O)CC2)ccc2nc(Cl)nn2c1 87590,N1(C(c2cccc(NC)n2)=O)CCC(C)C(NC(c2cc(O)cc(O)c2)=O)C1C 87591,C1(CNC(CC2(C)CCC2)=O)CC(F)CN1C(C1CCC1CN(C)C)=O 87592,c1(C(N2CCC(c3cnccn3)C2)C(=O)N)cnccn1.C1(C)(NC)CC1 87593,Cc1ccc(F)c(C(=O)NCCC2CCN(C(=O)Cn3nccc3C)C2)n1 87594,CCC1=NOC(CC(=O)N(C2CN(C(=O)C(=Cc3ccco3)C)C2)C)C1 87595,CCCCC(C(=O)NC1CCN(c2ncc(F)cn2)C1C)NC(N)=O 87596,N1(C(c2n(C)ccn2)=O)CC2CCOC2(CNC(c2ccsn2)=O)C1 87597,c1(OC(Cn2cc(C(=O)OC)nn2)=O)ccc(C)c(N(C)C)c1 87598,c1(C(C)(CNC(=O)C(F)F)NC(C(CC)C2CCOCC2)=O)cc(N)ccc1Cl 87599,c1(OCC)ccc(CCCNC(=O)CC2(C)CC2(Cl)Cl)cc1OCC 87600,c1(CN(C(=O)C(C2CC2)NC(c2ccoc2Cl)=O)CC)cn(C)nn1 87601,C1(C(N2C(C3(O)CN(C(c4c(SC)scc4)=O)C3)CCC2)=O)CCC(C2CC2)CC1 87602,N1(C(=O)NCCc2cscn2)CCS(=O)(=O)C(CSc2ccc(F)cc2)C1 87603,N1(C(c2c(C)csc2Cl)=O)CC2CCN(C(c3cccc(F)c3O)=O)CCC2C1 87604,C1(NC(C(=O)NCCC(N)=O)=O)CC(N=c2ccnc(Cl)[nH]2)C12CCOCC2 87605,CC(C)CCC(=O)NCC(C1CCCCN1C(C1(C2CCCCO2)CC1)=O)(C)C 87606,c1(NCC(=O)NCC(C2(C)CC2)NC(=O)CO)ccccc1C(C)SCC 87607,N1(C(CN(CCC)C)=O)CCC(C)(C(=O)NCC2CN(CC)CCCO2)CC1 87608,C1(C(=O)NCC(C2CC2)NC(CCc2cc(C)[nH]n2)=O)CC12CCC(F)(F)CC2 87609,Cc1ccc(N)c(C(=O)NC2CN(C(=O)Cn3c(C)csc3=O)CC2(C)C)c1 87610,C1(N(C(=O)CCc2csc(C)n2)CCCC)CCN(C(C2CCC2C)=O)CC1 87611,c1(C(=O)NC2CCC(N(C(=O)CSCC(N)=O)C)C2)ccc2nc[nH]c2n1 87612,N1(C(CC(C)(C)C)=O)CC2CCCC(NC(c3coc4c(F)cccc34)=O)C2C1 87613,N1(C(c2nccn3nccc23)=O)CC(O)C(O)C12CCC2 87614,c1(C(=O)NCC2C(NC(CCC=C)=O)CC2)c(C)ccc(F)c1O 87615,c1(C(N2C(CNC(C(C=C)(F)F)=O)CC(O)C2)=O)cc2c(cc1Cl)NCC2 87616,c1(NC(C2CC(NC(c3c(C)nc[nH]3)=O)C2)=O)nc(Cl)ccc1F 87617,C(=O)(C1CCc2c(Cl)cccc21)NCCCCCOC.C(=O)(COCC(C)C)N 87618,CC(C(=O)NC1CCCOC1C1CCN(C(C2OCCCO2)=O)CC1)C(C)(F)F 87619,C(C)(C)(CCCC(=O)N1CCC2C(O)CC12)NC(CCc1n(C)cnn1)=O 87620,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2n1)=O)NC(C(C)O)C(N)=O 87621,C1(OC)CCCC2(CNC(c3nc(Cc4ccc(C#N)cc4)no3)=O)CC12 87622,C(C(COC)C(=O)N1CCCC(CCCO)C1)OC 87623,CCC(C)C(O)C(=O)NC1CC(Cn2cc(C)cn2)C1 87624,c1(CCCCC)nc(C(=O)N(C2CC2)CC2CCCN2C(c2cc[nH]n2)=O)cs1 87625,C(=O)(C(CCF)NC(C1(C)CCC(=O)N1)=O)N(C)C 87626,N1(C(COCCSC)=O)CCC2CC1CN2C(C1CCCCC12CCC2)=O 87627,C(=O)(CC1OCCc2ccccc21)NC(CN(C(c1[nH]cc(CC)c1)=O)C)C 87628,C1(C(=O)NC2C(C)(CN(C(Cc3cc(C)on3)=O)C)CCC2)C(C)(C)OC1(C)C 87629,Cc1cc(C(N2CCN(C(=O)C3=CCOC3)C3CC23)=O)c(N)cc1F 87630,C(C(=O)NCCOCC(C)(C)O)(C(C)C)NC(Cn1ccc(C)n1)=O 87631,C#CCC(CC(=O)NCC1(CC)CC2CC2C1)NC(=O)CN(C1CC1)CC 87632,C(=O)(CCCCCC#N)NC1CC2(CN(C(c3n(C)c(S)nc3)=O)C2)C1 87633,CCCCC(C(=O)NCc1cn(C)nn1)NC(C1CS(=O)(=O)C1)=O 87634,Cc1nc(-c2cc(C(=O)NCC(C(C)C)NC(=O)CC3CC3)cs2)cs1 87635,N1(c2nccc(OC)n2)CCC(O)C(C(N2CCC(O)C2)=O)C1 87636,C(CCN=C(NCCOC)N1CCN(CCc2csc(C)n2)CC1)OCCC 87637,C1(=O)C(C(C)O)N1.C1(C)(OCC)CN(C(=O)CON(C)CCO)C1.CC 87638,C(=O)(C(C)P(C)(C)=O)N(CC=CC(=O)NC(COC)CO)C 87639,N1(C(C(CCCC)=O)=O)C(CNC(=O)C(c2cnn(C)c2)C)CC2CCCCC12 87640,C1(CO)C(=O)N2CC(C2)N(CCO)N1.C(=O)(CCNC(=O)CO)OC 87641,CN(C)NC(=O)CCC(=O)NC1(C)CCN(C(c2ccc(C#N)o2)=O)CC1 87642,c1(C(=O)NC2CCCN(Cc3ccc(F)cn3)C2)ncn2ccccc12 87643,C1(C(N(C2CCN(C(=O)C(=O)N3CCCC3)C2)C)=O)CCc2cncn2C1 87644,C1(CCNC(C)=O)CCCN(C(=O)COc2cccc(Cl)c2)C1C 87645,C(=O)(CC(C)(F)F)NC(CCNC(CCC#C)=O)C 87646,c1(C(N2CCC3CN(C(c4c(C)coc4)=O)CC3C2)=O)coc2cc(O)ccc12 87647,Cc1cncc(CC(N2C(C(N3CC(c4ccc(Cl)cc4)C3)=O)CC3CC23)=O)c1 87648,Cc1ccnc(O)c1C(=O)N(CC(O)CN(C(=O)CC1(N2CCCC2)CC1)C)C 87649,N1(C(Cc2c(C)cco2)=O)CC2C3CCC(C2C1)N(C(c1cocn1)=O)C3 87650,Cc1c(N)ccc(C(=O)NCC2CCCCN(C(=O)CCc3ccoc3)C2)c1C 87651,C(=O)(C(C)(C)C(=O)N(C)C)NC(C(=O)NCC(=C)Cl)COC(C)=O 87652,CC(O)(C(=O)NCC(O)CC(=O)NCC(O)CCC1CC1)C(F)(F)F 87653,C=CCCCCCCC(=O)NC1CC12CC(NC(=O)CN(C)C(=O)C1CC1)C2 87654,N1(C(CCNC(c2cnn(C(F)F)c2)=O)=O)CCn2nccc2C1 87655,c1(C(N(CCCCC)C)=O)ccc(CNC(C2(C)CCOC2C)=O)nc1 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87833,CS(=O)(=O)CCCCN=C(NCC(C)Cc1ccco1)NC1CCC1 87834,c1(OC)cnncc1C(=O)NC(C)CNC(=O)CCOCC(F)F 87835,CC(CC(=O)N(CCNC(=O)C1=NNC(C(F)F)C1)C1CC1)C(F)(F)F 87836,C1(C(=O)NCC2C(OCC)CN(C(=O)C(CC)SC)C2)CN2CCN1C(C)C2 87837,CCC(CC)CCCC(=O)N1CCCC1C(N1CCCC(N=[N+]=[N-])C1)=O 87838,C1(NC(c2cnn(C(F)F)c2)=O)CC2CCC1(C(=O)NC1C=CCCCC1)C2 87839,C(=O)(C1=NNC(C(F)(F)F)C1)N(CCCCn1cc(C(O)CC(N)=O)nn1)C 87840,c1(CC)c[nH]c2ncnc(N3CCC(CF)(NC(C4C=CCC4)=O)C3)c12 87841,O=C1CCCC(C(N2CCOC(CF)C2)C(=O)NCc2cnn(C3CC3)c2)CC1 87842,CON(C)C(=O)C(C)NC1CCCCC1n1cccc1 87843,N1(C(c2c(OC)ccs2)=O)CC2(CCC(NCc3ccc(Cl)c(F)c3Br)O2)C1 87844,c1(C(N2CC(SC)C(NC(C3(C)CCCC3)=O)C2)=O)ccc2n[nH]c(C)c2c1Cl 87845,N1(C(c2nn(CC)c(O)c2)=O)CCOC2(C1)CN(C(c1cc(C)cc(Cl)c1)=O)C2 87846,CC1CCc2[nH]c(-c3nc(C(F)F)nn3CCF)cc2C1 87847,N1(C(CC)=O)CCOCC2(COCCN2C(=O)C(O)C(C)c2ccccc2F)C1 87848,CC(C)C(C)(CNC(=O)Cn1nnc(C2CC2)n1)NC(c1cccnc1F)=O 87849,c1(CCC(=O)N(CCC(=O)NC2CCSC2)CC#C)ccnn1C 87850,c1(OC)ccc(COCCCNC(=O)C(=O)NC2CC(Cl)=NO2)cc1 87851,N1(C(C(C)NC(N)=O)=O)CCCCC1CNC(=O)CC1CCC(C2CC2)O1 87852,CN1CCC(C(=O)NC2(C3CCCN3C(c3cncc(Cl)c3)=O)CC2)C(C#N)C1 87853,C=CCCC(O)CN(C)C(C1(C)CCCN1C(=O)Cn1cccc1)=O 87854,C12(CNC(C(C(C)C)OC)=O)CCC1CN(C(c1nccc(C(F)(F)F)n1)=O)C2 87855,N1(C(c2cc(C)c(Cl)cc2F)=O)CCC(NC(C2CC(C)C2)=O)CC(C)(C)C1 87856,CC(C(C)(C)C)=CC(N1CCC(NC(=O)CCc2cc[nH]n2)C1)=O 87857,CCC(CO)C(=O)NCC(C1(O)CN(C(=O)C(F)(F)C2CCOCC2)C1)(C)C 87858,N1(C(c2ccc(CNC(c3cnc(CC)o3)=O)s2)=O)CCC(F)(F)C(C)C1 87859,C(CCC(=O)NC1CCOC1(C)C)(C(C)C)NC(CCn1ccc(C)n1)=O 87860,c1(CC(=O)NCC2(F)CC(CNC(C3CCC(=O)N3)=O)C2)nc([N+](=O)[O-])n[nH]1 87861,N1(C(C2(C)SCCCS2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CC=CC(F)(F)F)C1 87862,c1(NCCCC)ccc(C(N2CC(F)(CNC(C3CC3C#N)=O)C2)=O)cc1 87863,C1(OC)CCC2CN(C(C3(C)CN(C(C4CCOC4C(C)C)=O)C3)=O)CC12 87864,n1(CCNC(C2CC(C3CCCCO3)C2)=O)cc(C2CCCOC2)nn1 87865,O(N(Cc1ccccc1)CC(=O)Nc1ccccc1NC)C(S(C)(=O)=O)C 87866,C1(C(=O)NCC(CC=C)NC(C2CCOCC2)=O)CCCC12CCC2 87867,C1(CC)(OC)CCN(C(C2CCC(C(=O)O)CC2)=O)CC1 87868,CC(O)(CNC(c1conc1CNC(C1(CO)CCOC1)=O)=O)C(F)(F)F 87869,c1(CC(=O)N(C2CCN(C(c3ccc(C)cc3)=O)C2)CC)cc(F)c(N)cc1F 87870,N1(C(C2CCC(C)C2)=O)CCN(C(=O)C(F)(F)n2cccn2)CC1 87871,C1(N(C(=O)Cc2cn[nH]c2)C)CCCCC1N(C(=O)Cc1ccc(N)cc1)C 87872,C1(NC(c2scc(C)c2)=O)C2CC1N(C(=O)CSc1nc[nH]n1)C2 87873,c1(C(=O)NC2CC3CC(NC(C(C)SCC)=O)C3C2)c(C)cc(C)nc1C 87874,CN1CCN(CCC(=O)Nc2ccc(COc3cc(OC(F)F)ccn3)cc2)CC1 87875,c1(C(=O)NCC2CN(C(CC)=O)CC2C)ccc2c(c1)C(CC)C(=O)N2 87876,N1(C(CCN(C)CCO)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 87877,C1(CCOC)CCCN(C(C2CC(O)C(F)C2)=O)C1.c12occc1CNC2=O 87878,c1(CC(=O)NCC2CCCN2C(=O)CC2CCCC3CC23)ccc(F)c(F)c1 87879,C1(C(=O)NCC2C(NC(C3CC(OC)C3)=O)C2)COCCN1CC(F)(F)F 87880,C1(CCN(CC)CC)(CNC(c2cc(Cn3ccnc3SC)no2)=O)CCCO1 87881,C(CC(CNC(C1CCCO1)=O)C(c1ccccc1)C1(O)CCSC1)OC.C(=O)N 87882,CN1C2CCCC1CN(N1CCN(CCC(F)F)CC1)C2 87883,c1(CC2COC2)ccc(Cl)cc1.Cc1ccsc1-c1cccs1 87884,C(CCC(C)(C)NC(=O)C=CC(=O)N(C)C)NC(c1cn(CC(CC)O)nn1)=O 87885,CC1(C(=O)Nc2cnc(O)nc2)CCCN(C(=O)CCc2cnccn2)C1 87886,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2ncccc12 87887,N1(C(Cc2c(C)nccc2)=O)CCC2CCC12CNC(c1c(C)nc(C)n1O)=O 87888,C(=O)(CS(=O)(=O)CCO)NCC1(CO)CCN(C(C(F)OC)=O)C1 87889,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 87890,c1(NC(C)CCc2ccccc2F)nccc(=NCc2nnc(C(C)(C)C)s2)[nH]1 87891,c1(CCC(C)c2ccccc2)nc(-c2cncs2)nn1CC(=O)OC(C)(C)C 87892,N1(C(C(C(=O)OCC)F)=O)CCC2(C)CN(C(C34CCCN(CCC3)C4)=O)CC12 87893,C1(c2nnnn2C)(NCCOC)CCN(C(CC(C(=O)OC)F)(C)C)CC1 87894,N(C(=NCCCCC(F)(F)F)NC1CC(C)(C)C1)C(C)COCC(=O)NC1CC1 87895,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 87896,S(=O)(=O)(CC(=O)NC1CCCC1NC(c1nccn1CC(F)F)=O)N(C)C 87897,C1(CC(=O)N(CCCC=C)C)CCCN(C(C2CCCN2CC)=O)CC1 87898,C(=O)(C1CCCc2ncnn21)N1CC(O)CC(NC(C2(C)CCCCC2)=O)C1 87899,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 87900,Cc1cc(C(=O)NCc2cn(CC(C)C)nn2)n2nccc2n1 87901,c1(CC(=O)NCC(c2ccccc2)CNC(C2CCC(=O)N2)=O)cccnc1Cl 87902,N12CCCC(C1)NC(=O)C2.C(=O)(CC(F)F)NCC(C1CCCC1)CNS(CC)(=O)=O 87903,Cc1n[nH]c2cnc(C(=O)NCC(C(C)C(C)C)NC(c3nocc3Cl)=O)cc12 87904,N1(C(C(C)OC(C)(C)C)=O)CC(NC(c2cncc(O)c2Cl)=O)C(C2CC2)C1 87905,C1(CC)CC(C(=O)NC(c2cccc(Cl)c2)C)CCN1C(c1ncoc1CC)=O 87906,N(C1CCCc2cc(CNC(C3OCCO3)=O)ccc21)C(c1n(C)nc(O)c1)=O 87907,C1(OC)(OC)CCC1C(=O)NCCNC(=O)CCc1cnoc1 87908,C(=O)(C(=O)CCC(C)(C)C)N1C(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCC1 87909,N1(C(C2CC(F)(F)C2C)=O)CCN2CC1C(CC)C(CO)C1C(CC1(F)CO)C2=O 87910,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CN(C(C1Cc3nc(C)cn3C1)=O)C2 87911,c1(CC(N2C(C(=O)OCC)CC2C)=O)ccc(-c2ccnn2C)cn1 87912,C1(C(N(C2CCCC2)C)=O)COCCC1NC(C1(C)CC1)=O.C1C=CCO1 87913,Nc1ccc(C(N2CCC3(NC(=O)Cc4ccoc4)CC3C2)=O)c(O)c1Cl 87914,C1(NC(CC2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(C2(CC)CCNC2=O)=O)C1 87915,CC(CC(F)(F)F)C(=O)Nc1ncc(C(F)F)s1 87916,c1(OCC)ccccc1C(CC(=O)OC)NC(c1ncccc1C(F)F)C 87917,c1(NCC(CNC(C2OCC(C)C2)=O)O)cc(C(F)(F)F)ncn1 87918,C1(OCCN(C)C(=O)NCC2(C(C)(C)O)CCC2)CCC(F)(F)CC1 87919,c1(CN2C(C(=O)Nc3ccn4cnnc4c3)CC(F)C2)ccc2ccccc2n1 87920,N1(C(C(F)=CCC)=O)CCCN(C(c2n[nH]c(C)n2)=O)CC1 87921,CC1=C(C(=O)N2CCC(CNC(C34CC(F)C3C4)=O)CC2C)C(=O)OC1(C)C 87922,c1(CC(=O)NCC2(C(C)NC(C(N3CCOCC3)C)=O)CC2)cc(SC2CC2)no1 87923,C1(OCC)CN(C(C2(CO)CC2(F)F)=O)CC1CNC(c1ncccc1OC)=O 87924,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2C(N)=O)=O)CC1 87925,N1(C(C=C(CCC)C)=O)C2CCC(C(N3CC4CC3CN4C)=O)C1CC2 87926,CC(CN1CCOCC1)N=c1[nH]c2c(c(=NC(C)c3nncn3C)[nH]1)SCC2 87927,n1(C(C)NC(=O)OC(CCSCC(=O)NC(C(C)OC)C)=O)cc(Br)cn1 87928,c1(C(N(C(C)C)CCNC(C2OC3CCC2C3)=O)=O)ccnc(O)c1F 87929,c1(C(C)C)[nH]nc(C(N2CC(NC(C3(C)C=CCC3)=O)C2)=O)c1[N+](=O)[O-] 87930,N#CC1(C(N2CC(C3C(=O)N3)C2)=O)CCOCC1.c1(CCC)nnc(O)o1.CCF 87931,Cc1cc(CNC(=O)C=CC(C)(C)NC(c2coc(C(C)C)n2)=O)n(C)n1 87932,Cc1cnc2c(C(=O)N(C3CCN(C(=O)CC4CC(F)C4)C3)C)cnn2c1 87933,Cc1c(F)cc(C(N2CCC(NC(C3CCc4n[nH]cc4C3)=O)C2)=O)c(F)c1N 87934,Cc1nc(C(N2CCCC(NC(C3CCC4CC34)=O)C2)=O)c(C)o1 87935,c1(CNC(c2cc(CNC(C(C)OCCCC)=O)no2)=O)ccc(O)c(F)c1 87936,c1(NCCC)ccc(C(=O)NCCN(C(C2SCCS2)=O)C2CC2)cc1 87937,C(CNC(=O)C(c1cccn1C)=O)(CC(=O)N(C1(CCO)CC1)C)OC 87938,Cc1nc(CO)sc1C(=O)NCCC1CCN(C(c2nc(=N)cc[nH]2)=O)C1 87939,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 87940,Cc1nc[nH]c1CC(=O)NC1(C)CN(C(C2CCC(C)C2)=O)C1 87941,C1(NC(C2(COC)CCCC2)=O)C=CCC(C(=O)N(C2CCCC2(C)O)C)C1 87942,Cc1[nH][nH]c2ncnc(=NCC3CCN(C(c4csc5cncn45)=O)C3)c1-2 87943,C1(O)(C(N2C(C(=O)Nc3c(C)nc(C(=O)OCC)s3)C=CC2)=O)CCC(C)(C)C1 87944,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 87945,C1(NC(CC(C=C)(C)C)=O)CN(C(c2cc3ccccc3o2)=O)C2(CCC2)C1 87946,Cc1cnc(Cl)c(S(=O)(=O)N2CCCC2(C)C(=O)Nc2ccnc(Cl)c2I)c1 87947,C=CCC(C)(C)CC(=O)N1CCN(C(C2(C#N)CC(=O)C2)=O)CC1C 87948,c1(N2CCCC(C)(CO)C2)cc(Br)ccc1S(=O)(=O)NCCCC#N 87949,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 87950,c1(C(c2nnnn2C2CC(F)(F)C2)NC(CC)C2CCC2)cncc(Br)c1 87951,C1(OCC)(CNC(c2cc(=O)cc[nH]2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1 87952,c1(COC(C2CC(F)(F)C2)=O)cccc(-c2nc(O)n[nH]2)c1 87953,N1(C(c2cnc(SC)s2)=O)CCN(C(C23CC(C2)C3)=O)CC(C)(C)C1 87954,c1(OC)cc(C(N2CC(NC(c3cccc(F)c3C)=O)CC2C)=O)cc(N)c1N 87955,C12(C(=O)NC(C)CCN(C)C(c3cc(C(N)=O)[nH]n3)=O)C3CC(CC13)C2(F)F 87956,CC1CN(C(=O)CN(C)C(c2ccccc2)=O)CC1NC(C1(F)CC=CCC1)=O 87957,N1(C(c2c(OCC(C)C)ccc(Br)c2)=O)CC(S(C)(=O)=O)CC1(C)C 87958,N12CC3CN(C3C1)C(=O)CCn1cc(nn1)-c1ccc(cc1)CC2=O.CC(=O)O 87959,Cc1cc(F)ccc1C(=O)NCC(C1CCCN1c1ccccc1)(C)C 87960,C(=O)(CC1COc2cc(O)ccc21)N1CCN(C(C2(C)CC(F)C2)=O)CC1 87961,c1(C(N2CC3C(CNC(CCc4n[nH]c(=N)s4)=O)(C3)C2)=O)ccc2nccn2n1 87962,CC1COCCN(C(=O)CCN(C(=O)COC2(C)CCC2)C2CC2)C1 87963,N1(C(CCC(=C)C)=O)CCC2(CCOC2)C(CNC(c2csc(COC)n2)=O)C1 87964,N1(C(c2cn(CC(CNC(C(CCOC)OC)=O)(C)C)nn2)=O)CCNC(=O)C1C 87965,c1(C(=O)NC2CC(CNC(C(C)C3CCC3)=O)C2)n[nH]c2ccc(Cl)cc12 87966,c1(C(=O)NCC2N(C(CC(C)NC(N)=O)=O)CCC2)nn(C)nc1Br 87967,C(C(=O)N1C2CCC1(CNC(=O)C=Cc1nnn(C)n1)CC2)(C(C)(C)C)N(C)C 87968,CC1(C)CCOC1CS(=O)(=O)NC(=O)Nc1cnc(-c2cccs2)o1 87969,Cc1cccc2c1CCOC2C(=O)NC1(CNC(c2ccc(O)nn2)=O)CCC1 87970,C(=O)(CC(C)(C)C(=O)OCC)NC1(CNC(CCC=C)=O)CCC1 87971,C=Cn1ncc(C(=O)NCC(C(=O)N2CCC(CCO)CC2)C(C)C)c1N 87972,C1(CNC(CCCC(C)=O)=O)CN(C(=O)C(C)(C)C2CCCCO2)CCC1(F)F 87973,c1(OC)coc(C(=O)NC2CC(CCNC(=O)Cn3cc(C#N)cn3)C2)cc1=O 87974,C(CC(C)(C)C)(C(=O)N1CCC(C)(CC(=O)NCC2(C)CCC2)C1)OC 87975,C#Cc1cccc(C(N2CC(CN(C)C(c3cnn4ccn(C)c34)=O)C2)=O)c1F 87976,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 87977,CCCCCC(F)C(=O)N1CC(NC(=O)CCCCCn2cnnn2)C(C)(C)C1 87978,C1(NC(C2(C#C)CC2)=O)CCCN(C(=O)Cc2cc(C)n(C(C)(C)C)n2)C1 87979,N1(c2nc3n(n2)C(C)CC3)CC(C(=O)NC)OC2(CCC2)C1.C(=O)(C=CC1CC1)N 87980,c1(C(=O)OC)cncc(OC2CCN(C(c3ccccc3-n3cnnn3)=O)C2)n1 87981,C(=O)(CC(O)C(C)C)NC12CC(CNC(C3CCN(CC)C3)=O)(C1)C2 87982,C1(NC(C(CC)NC(C)=O)=O)CCC2CC1CN2C(=O)C(C)OCCC(C)C 87983,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(c2ccncc2Cl)=O)C1 87984,C1(C)(NC(CC2C=CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC(F)(F)C1 87985,c1(C(=O)NC2C(CNC(C)=O)CCC2)[nH]c2ccccc2c1-c1ccccc1 87986,Cc1ncnc(C(=O)NCC(CNC(c2cc(C3CC3)cs2)=O)S(C)(=O)=O)c1C 87987,C12(NC(CC(CC)C)=O)CCC(CNC(=O)CN3C(=O)CN(C)C3=O)(C1)OC2 87988,C(=O)(C(O)CC(C)(C)C)NCC1C(CC)CN(C(=O)Cc2cccc(C)c2)CC1 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88077,S(=O)(=O)(C1CC1)NCCCN(C(=O)C(C)n1cccn1)CC(=O)OCC 88078,C(CCC(=O)NCC(O)C(=O)NCC1(CF)CC1)OCC 88079,N1(CC(=O)NCC2C3CC3N2C(=O)CC2CC=CCC2)CCNC(=O)C1 88080,C1(C(=O)NC2CN(C)CC2O)CC(O)CCN1C(c1nccnc1N)=O 88081,N1(C(CN(C)C(c2ccccc2)=O)=O)CCCC(C2(C(N3CCOCC3)=O)CC2)C1 88082,c1(NC(C(CSc2cnn(CC)c2)NC(CCC)=O)=O)ccc(F)cc1C 88083,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NCC1CC(C(C)C)C1 88084,Cc1[nH]nc(C(=O)N(C(C)CN(C(=O)C(C)CF)C)C)c1C(F)(F)F 88085,C1(NC(c2c(SC)cccn2)=O)CN(C(=O)CCc2cnco2)CC12CC2 88086,C(=O)(CCCC(C)(C)C)N(C1CN(C(c2ccc(NC(CC)=O)cc2)=O)C1)CC 88087,C(=O)(C1=CCCCC1)NC1CC(NC(C(n2cc(Cl)cn2)C)=O)C(O)C1 88088,CN1CC(C(N2CCC(F)(C(=O)NCCc3ccncc3F)C2)=O)NC1=O 88089,C1(NC(C(COCC)NC(=O)CSC)=O)CC2(COCCO2)C1 88090,c1(N(CC(C)C#N)C)nc(N(C)CC2COC(=O)O2)c2cnn(C)c2n1 88091,C1(N(C(=O)CC2CC2)C)CN(C(c2ccc(Cl)cc2)C2C3CCC2CC3)CC1(C)C 88092,CC(C)C(CCNC(C12CC(CN1C1CC1)C2)=O)NC(C1(C)CCCC1O)=O 88093,Cc1[nH]c(=N)ccc1C=CC(=O)N(C(C)CNC(C1CCCC12OCCO2)=O)C 88094,C1(NC(=O)CO)CC2(CCN(Cc3ccc(OC4CCCC4)cc3)CC2)C1 88095,C(=O)(C1=CCOC1)Nn1ccc(=NC(CCC(C)c2nnnn2C)c2nn[nH]n2)[nH]1 88096,C(CCC1CCC1)(C(=O)NCC(Cc1ccc(Cl)cc1)CO)NC(CCC)=O 88097,C#CCCCC(C)C(=O)Nc1ccc(NC(C2CCCC(=O)N2)=O)c(C)c1 88098,Cn1nc(C(N2CCCC(Cn3cc(-c4nccs4)nn3)C2)=O)c2c1CCC2 88099,c1(OC)ccccc1OCCC(=O)NC1CC(CNC(C2COCC(C)O2)=O)C1 88100,c1(NC(=O)NCC2CCN(c3cccc(OCC)c3)C2)nc(C)c(Br)c(Cl)n1 88101,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CCO)C1 88102,c1(NCCCS(C)=O)ccc([N+](=O)[O-])cc1C(=O)OC 88103,C1(C(=O)NC(CCCC)C)CCC(C)N1Cc1ncccc1Cl 88104,n1(CC(=O)O)cccc(NC(=O)NC2CCC=CCC2)c1=O 88105,c1(C(=O)NC2C3CN(C(=O)Cc4cc[nH]c4)CC23)cccc(F)c1F 88106,CCCC(C)(CCC)C(=O)NC12CCC1CN(C(C1(CC)CCSCC1)=O)C2 88107,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(C2(Br)CC2)=O)C1 88108,N1(C(c2c(C(C)C)con2)=O)CCN(CCNC(C2CCCN2C)=O)CC1 88109,N1(C(C(C(C)C)n2ccc(C3CC3)n2)=O)CCN(C(=O)C(N)=O)C2(CCC2)C1 88110,C(C(C)(O)CC(=O)NC1CCCN(C(c2cc(C#N)cs2)=O)C1)OC 88111,c1(CNCC(Cc2c(C)cccc2)CO)ccc(-n2cccn2)c(F)c1 88112,C=C(C)CN=C(NCC(CO)C1CC1)NCC(N1CCNCC1)(C)C 88113,N1(C(CNc2cc(OC)ncc2)=O)CCN(C(=O)CC2CCOC2=O)C(CO)C1 88114,C(=O)(CC(CC)CC(F)(F)F)N1C(CN(C(CC(=O)NCC)=O)C)COCC1 88115,N1(C(=O)Cn2cc(C(F)(F)F)nn2)CCN(C(C2CC2(Cl)Cl)=O)CC1 88116,C12(C(N3CCCC(N(C(COC)=O)CCF)C3)=O)CCCN1S(=O)(=O)CC2 88117,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 88118,C(CC(CC)C(=O)NC1CCCN(C(c2ncccc2C(F)(F)F)=O)C1)=CC 88119,C(C(=O)N1CCC(NC(=O)COc2cccnc2)C1)(C(C)C)OC 88120,C1(OC)(CNC(=O)COCc2ccccn2)CCN(C(C2CCCO2)=O)C1 88121,N1(C(CP(C)(C)=O)=O)CC2(CCCN(C(=O)Cc3ccsc3Br)C2)C1 88122,C1(C(=O)NCC2CCOC2)(CC)CN(C(C2CCCN2C(C)C)=O)C1 88123,C1(F)(C(N2CCC(N(CCO)C(c3cc(CC4CC4)on3)=O)C2)=O)CC=CCC1 88124,c1(NC(NCCNC(c2cc(C)n(C3CC3)n2)=O)=S)ncnc2ncc(Br)cc12 88125,N1(Cc2cc(OC)c(C)cc2)CCCC(C2CCCN(C(c3cn[nH]c3)=O)C2)C1 88126,Fc1ccc(SC(F)(F)CF)c(F)c1CNCCN1CCCCC1 88127,Cc1ccc(NC(=O)Cc2ccccc2NCc2cccc(I)c2Cl)c(Cl)c1O 88128,CCC(CC)(c1nnnn1CCCC1CC1)NCC(C1CC1)C1CC1 88129,O=C(C1=C(F)CN(C(=O)CC23CCC(CC2)C3)CC1)NCC(O)C(F)(F)F 88130,n1(CCCC)nccc1C(=O)NC(C1CCN(C(=O)C(O)C2CC2)C1)C 88131,N1(C(N2CC3CCC3C2)=O)CCCN2CCCC12 88132,c1(SC)ccc(C)o1.C12CCC(C1)n1cc(nn1)-c1c[nH]nc1N(CC)C2=O 88133,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CCc2nnc(S)n2C)CC12CC2 88134,C(C(C)(C)CC(=O)N1CCN(CCNC(C2(C3CCC(C)(C)C3)CC2)=O)CC1)OC 88135,CC(C)(O)C(F)(F)C(=O)N1CC2(CC(C(=O)NC(CC3CC3)C3CC3)CO2)C1 88136,N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)Cc2cc(O)n(C)n2)C(C2CC2)C1 88137,N1(C(c2ccccc2)C(=O)NCC(CN(C(=O)CC(F)F)C)O)CCC(O)CC1 88138,CCC(C)C(O)CC(=O)NC(C)(C)CNC(=O)COCC(=O)Oc1ccccc1 88139,CC1CC(NC(=O)CCC2CCC2)CN1C(c1cc(-c2cc[nH]n2)ccn1)=O 88140,c1(OCC(=O)NC2CC(C(C)NC(=O)C(C)(C)n3cnnn3)C2)ccc(F)cc1 88141,C1(NC(=O)C=CCO)CC2CN(c3nccc(CN)n3)CC2C1 88142,Cc1ccc(CC(=O)NCC2CC3CN(C(C4CCCCC4O)=O)CC23)c(Cl)n1 88143,c1(CC)ccc(C(=O)NCc2ccc(C(=O)NC(C)CC3CCCCO3)o2)o1 88144,N1(C(c2cn(CC)nc2)=O)CC(C2CC2)(C(=O)NC(c2cccc(C)n2)C)C1 88145,Cc1cc(C)c(C=CC(=O)NCC(C)NC(c2cnc(O)c(F)c2)=O)cc1C 88146,N1(CCNC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CC2COC(C)(C)C2)CC1 88147,C1(CCC)CN(C(=O)COC(C)(C)C)CCN1C(c1ncn(CC)n1)=O 88148,C1(C(N2CC(NC(c3ccc(CCC)[nH]3)=O)C2)=O)C2CCC(F)(F)C12 88149,c1(OCC)ccc(C(=O)NC2CN(C(=O)Cc3cccnc3Br)CC2C)nn1 88150,N1(C(C(=O)NCCOC)=O)CC2CCN(C(=O)COC(=O)NC)CC2C1 88151,N1(C(C)=O)CCCC(C)(C(N2CCCC(N(C(=O)CN3CCOC3=O)C)C2)=O)C1 88152,c1(C(=O)NCC2(CNC(CCCOC)=O)CCC2)ccc(C#N)c(C)c1 88153,C12(C(=O)NC(CNC(CNC(C)=O)=O)C3CC3)CC(C1)C(C)(C)O2 88154,CCCCC(CNC(=O)CC1(C)CC1(F)Cl)NC(c1scc(C)c1OC)=O 88155,Cn1ccc(CC(=O)NCCCCNC(C2CCO2)=O)n1 88156,C(=O)(C(CN=[N+]=[N-])NC(c1cc(Cl)n[nH]1)=O)N(CCCN(C)C)C 88157,O=C1CCCC(C(N2CCCC(C(N3CCOC(C4CC4)C3)=O)C2)=O)C1 88158,CC1(C)CCCCC1N1C(=O)CCNC(=O)C1.C1C(=O)N1.O(C(F)F)CC1CC1 88159,N1(C(c2cnc(CC)nc2C)=O)CCC(CNC(=O)C(C)C(C)(C)C)C(F)(F)C1 88160,N1(C(c2c3cccc(CC)c3[nH]c2)=O)CCN(C(=O)C(F)F)C(C)CC1C 88161,c1(C(=O)NCC=CCNC(=O)Cc2cn3ccsc3n2)cc(O)cc([N+](=O)[O-])c1 88162,Cc1cc(C(=O)NCC2CCN2C(C2(C#N)CCCO2)=O)c(C)cc1Br 88163,C1(NC(CCCSC(C)(C)C)=O)CCN(C(C23CC(CO2)C3)=O)CC1F 88164,C=CCCCCCNC(=O)CC1(NC(=O)C(C)(C)Cl)CC1 88165,C1(SCC)CCC(C)(F)CC1.C12C(C1)CNC(=O)O2 88166,N1(C(C2(OC)CCCCCC2)=O)CC(C)CN(C(=O)CCCCO)C(C)C1 88167,Cc1cc(CNC(=O)C(CNC(C2(C)CCNC2=O)=O)CC2CCCC2)sc1C 88168,C(N=c1[nH]c(Cl)ncc1Cl)C12OCC(CNC(C=Cc3cn(C)nc3)=O)(C1)C2 88169,C(N=c1[nH]cc(C#N)c2ccsc12)C(CCC)C.C(c1cncc(F)c1)=CC(=O)N 88170,C1(CC#C)(C(=O)N(C)CCSC)CCN(C(=O)Cn2ccc(C)n2)C1 88171,O=C(C1=CCC2CCC1N2C(C1C(C2CC2)CN1)=O)NCc1cccc(F)n1 88172,c1(C(N2CCSC(C(=O)OC)C2)C(=O)NCCCC)ccc(Cl)c(C)c1Cl 88173,C#CC1CCN(C(C2CCN(C(c3scnc3C)=O)CC2)=O)C1 88174,c1(C(N2CCOC(CNC(C3CC(O)(C(F)F)C3)=O)C2)=O)cccc(Br)c1 88175,N1(C(C(C)SC)=O)CCC(C)(N(c2ccc(-c3ccccn3)cc2)C(=O)C(N)=O)C1 88176,C1(CC(=O)NCC2(NC(C(CC)=CC)=O)CCOC2)CCN(CC)CC1 88177,c1(CC(=O)NCC(CNC(CC2(C=C)CC2)=O)CO)nccc(OC)n1 88178,c1(NC(C(C)NC(C)=O)=O)c(O)cccc1O.C12CN(CC1O)C2=O 88179,C1(C(N2C(C3C(C)CCC3)CCC2)C(=O)NCCCF)CC2CC1CC2O 88180,Cc1cc(C(N2CCOCC2CNC(c2cc(O)ccc2F)=O)=O)c(O)c(Br)c1 88181,C1(C(=O)NC(c2csnn2)C)CC2(CCN1C(C1CCCCC1)=O)CC2 88182,N1(C(c2c(C)ccc(SC)c2)=O)CCC2(CCC2)C(NC(=O)Cc2cnsc2)C1 88183,C12(NC(CCC(=O)NCCC)=O)CCC(CC1NC(=O)C(n1ccnc1C)C)C2 88184,C=CC(CC)CC(=O)NCC1CC(OC)CN1C(C1CC1c1sccc1C)=O 88185,c1(C(=O)NCC(CNC(CN(C(COC)=O)C)=O)OC)cn(C)nc1O 88186,C(=O)(CC(C)CC(=O)NC(C)(C)C(C)NC(c1cnc(C)cc1Cl)=O)OC 88187,C12(NC(C(C)O)=O)CCC(NC(c3ccnc(OCCO)c3)=O)(CC1)C2 88188,S(=O)(=O)(CC(=O)N1CCN(CC2CC2NC(=O)C(C)Oc2ccccc2)CC1)NC 88189,c1(CN(C(=O)CC=CCNC(=O)CCn2cccn2)CC)cncn1C 88190,c1(CNC(CSCC=C)=O)ccc(C(=O)OCC(=O)NC2CCC2)c(F)c1 88191,C1(C(N)=O)(CNC(=O)COCC2CCC2)CN(C(=O)CC2CCCO2)C1 88192,N1(C(c2cccc(C(N)=O)c2)C(=O)NCC)CCC2(CC1)OCC(C)(C)CO2 88193,c1(C(N2CCN(c3cc(C)ncn3)CCC2=O)=O)cc(=O)c2ccccc2o1 88194,CCCC(C)C(=O)NCC(c1ccc(OC)cc1)NC(=O)C=C(C)CCC 88195,CC(C(C)C(=O)NCCc1cnc[nH]1)NC(=O)C=Cc1cccnc1 88196,c1(CNC(C(ONC(CC2ON=C(C)C2)=O)C2CCOCC2)=O)ccc(F)cc1 88197,c1(C(N(CC(=O)N(CC(C)(C)C)CCO)CC2CC2)=O)ccnc(O)c1F 88198,CC(CF)CC(=O)NCC(C1CCN(C(c2[nH]nnc2C2CC2)=O)CC1)F 88199,C(C#Cc1cnn(C)c1)NC(C1N(C(c2ccc(C)nc2C)=O)CCC1)=O 88200,Cc1cc(C#N)c(O)nc1C(N1CCC(F)C(NC(=O)C#CC2CCCCO2)C1)=O 88201,C1(F)(C(N(C2CC(C)OCC2)C)=O)CCCN(C(=O)CC2COC(=O)N2)C1 88202,c1(C(=O)NCC(C)NC(C(C)SCCCC)=O)ccc([N+](=O)[O-])cc1 88203,Cc1cn(C)nc1C(N1CCCC1CCCNC(c1cc[n+]([O-])cc1)=O)=O 88204,C1(NC(CCC(=C)Br)=O)(CO)CCCN(C(=O)C(C)C(O)CC)C1 88205,Cc1nn(CC(F)F)c(C)c1C(=O)NC1CN(C(=O)C(C(C)O)N(C)C)CC1C 88206,CC1(C)CC(O)CN1C(C1CN(C(C2CCC(O)C2)=O)C1)=O 88207,C(=O)(C1=CCCN(C(c2cc(Cl)n(C)n2)=O)C1)N(CC(CC=C)(F)F)C 88208,N1(C(C(C)CO)=O)C2CCC1C(F)C(NC(c1ccn3nccc3n1)=O)C2 88209,Cc1scnc1C(=O)NCCC(C)N(C)C(C1CSCCS1)=O 88210,c1(C(N2CC(C)CC(NC(C(C)SC)=O)C2)=O)c[nH]c2nccc(Cl)c12 88211,c1(C(N2CC(NC(C(C)CC3CCC3)=O)C(F)CC2)=O)nccc2c1CNC2=O 88212,N1(C(Cc2ccn(CC)n2)=O)CCC2CCCC12C(N1CCCC(C)C1)=O 88213,CCC(C(=O)NCCC1CN(C(C2CCCN2Cc2ccccn2)=O)C1)N(C)C 88214,N1(C(c2cc(C)c(O)nn2)=O)CCC2(CCN2C(=O)Cc2ccc(Cl)cc2Cl)C1 88215,C(C(C)(O)C(=O)NCC1CN(C(=O)C(F)n2cccn2)CC1C)OC 88216,C(N=c1nc(C2CC2)nc[nH]1)C1CCCC(NC(c2n(CC)c(O)nc2)=O)C1 88217,c1(CC)cc(C(=O)NC(CNC(C2CC(=O)N(C)C2)=O)CCOC)c(C)nn1 88218,c1(C(N2CC(C)(C)C(c3cn(CCO)nn3)C2)=O)csc2ccc(F)cc12 88219,C(=O)(CCCN(C)N=O)N1CCN(CCN(C(Cc2cc(C)ns2)=O)C)CC1 88220,N1(C(C(CCC(N)=O)n2cc(CCOC)nn2)=O)CCCn2nc(C#N)cc2C1 88221,N1(C(c2n(CC#C)ccc2)=O)CC2CCCC(NC(c3nncn3CC)=O)C2C1 88222,c1(C(=O)NC2C(NC(C3CCCO3)=O)C2)nccc2ccccc12 88223,C(=O)(C1=NOC2(CCC2)C1)NC(C)CC(O)c1cccs1 88224,C1(C(=O)NCC2(C)CCN(C(CCc3cncc(C)c3)=O)C2)CN2CCC1CC2 88225,c1(C(N2CCC(OCCNC(c3cnc(CC)[nH]3)=O)C2)=O)nnccc1C 88226,c1(OC)cccc2c1CCN(C(C1CCN(Cc3cnc(Cl)s3)C1)=O)C2 88227,C1(OC)CN(C(C2CC2F)=O)CC1NC(=O)CCN1CCOC1=O 88228,C1(C(=O)NC)(C(=O)NCC2(COC)CC2)CCOCC1.C12CCCC1NC2=O 88229,N1(C(C(C)N(C(C2CC(C#C)(O)C2)=O)C2CC2)=O)CCOCC(C(=O)OC)C1 88230,CC(C)CC(O)C(C)C(=O)NC1CC1NC(c1nnn(C(C)(C)C)n1)=O 88231,C1(NC(c2n(CC)ncc2Br)=O)CCN(C(=O)Cc2ccn(C)n2)C(C)C1 88232,CC(C)CCC(O)C(=O)N1CC(C(=O)NCCCN2CC=CC2)CCC1C 88233,c1(CC)nc(C)c(C(=O)N(C)Cc2cccc(CNC(C3(O)CCOC3)=O)c2)o1 88234,c1(C(N2CC(CNC(C(CCC)C)=O)C(C)C2)=O)cc(C)cc(Br)c1 88235,Cc1nn(C)cc1NC(=O)C(C)(C)NC(=O)CCCC1CCCC1 88236,C(=O)(C(CC1CC=CCC1)N1CCC(C(C)C)C1)NCCC(=O)OCC 88237,c1(OC)ccc(OCCC(=O)NCCCCNC(=O)C(C#N)C2CC2)cc1 88238,C1(NC(c2ncc(C(C)=O)s2)=O)CCC(C)(CNC(c2c(C)n[nH]c2C)=O)C1 88239,c1(C(=O)NC(C(=O)NCCCC)(C)C)cnc2onc(C(C)C)c2c1 88240,CCC(O)C(C)C(=O)NC(C)CCN(C(=O)CNC(c1ccccn1)=O)C 88241,CC(C(=O)N1CCN(C2CN(C(=O)CC3CC4(CC4)CO3)C2)CC1)C(F)(F)F 88242,N1(C(C(C(CC)CC)C)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC2(CC2)C1 88243,C(=O)(C1(C)CCc2ccccc21)NC1(C)CCN(C(C=CC=CC)=O)C1 88244,c1(OC)ccc(F)c(C(=O)NC(C)CNC(=O)C=CC2CCOC2)c1 88245,N1(C(C2(c3c(C)cccc3C)CC2)=O)CCS(=O)CCC1C 88246,CC(C)(C(=O)NCCC1CCC(NC(C2CC2C2CCCO2)=O)C1)c1cc[nH]n1 88247,CC1CC(CO)(NC(C2(F)CN(C(C3CCSC3C)=O)C2)=O)C1 88248,Cc1cnn(C)c1CNC(=O)CN(C(=O)C(Cn1cccn1)N(C)C)C 88249,C1(C(N2CCC(CNC(=O)NC3(c4cccnc4)CC3)C2)C)CC2CCC1CC2 88250,C1(CC(=O)N(C)CCN(C(C)C)C)CC(O)C1(C)C.c12nc(cs1)NC2=O 88251,C=CC1CN(C(C2CN(C(N)=O)C2)=O)CC1NC(c1ccc(SC(C)C)cc1)=O 88252,C#Cc1cnc(C(=O)NC2CC(CCNC(=O)C=C(C3CC3)C3CC3)C2)c(C)c1 88253,C=CCCCCCCCCNC(=O)NC1CCC(=O)NC1=O 88254,c1(C(=O)NC(C2CN(C(C(CO)OC)=O)C2)C)n[nH]c2ccc(OC)nc12 88255,C(=O)(CCCCC(C(=O)OCCN=[N+]=[N-])OC)OC.c12ccc(C#N)cc1OC2 88256,CC1CC(C)(CNC(=O)NCCCC2CCCC2(F)F)CC(C)O1 88257,c1(C(=O)NC(CC(C)C)CNC(C2CNC(=O)C2)=O)cc(O)ncc1Br 88258,CC(C)C(O)C(C)C(=O)N1CC2C(C(=O)N(C)Cc3nnnn3C)C2C1 88259,C1(NC(=O)CCOC2CCC2)CCC2(CC1)CC2NC(c1cc(C2CC2)ns1)=O 88260,NC(=O)CC(C(=O)NCC1C=CCCC1)NC(C1CC(C2CC2)C1)=O 88261,CC1=C(C(=O)NC(C)CC(C)NC(=O)CCC=O)S(=O)(=O)CCO1.OC 88262,C1(CNC(CSCCCC)=O)CC2CCC1N(C(=O)C(F)CC1CCOC1)C2 88263,CCC(C)C(O)CC(=O)NCC1CCCC1C(=O)NCC12CCC(CC1)CC2 88264,c1(C(N(CCCN(C(C2C(CC)CCCC2)=O)C)C)=O)cc(C)cc(C#N)c1 88265,CCCCCCCCC(C)CC(=O)NC1CN(C(=O)CS(=O)(=O)CC)CC1CC 88266,C1(C(N2CC(NC(CCSC)=O)C(CO)CC2)=O)C(C)(C)CCCC1(C)C 88267,C1(NC(=O)OC(C)(C)C)CCCC2CN(C(=O)Cc3cc(F)ccc3F)CC12 88268,n1(CC)cc(NC(c2cnc3ccccn23)=O)c2ccccc12 88269,N1(C(Cc2nc(C)oc2)=O)CCC(NC(c2nc(C)nn2C)=O)C12CCC2 88270,C1(n2cc(C3(OC)CCC3)nn2)CCN(CC(C2CCCC2C)=O)CC1.CC=O 88271,c1(C(N(CC(C)NC(c2c(CC)onc2Cl)=O)C)=O)cc(C)cnc1N 88272,C(C(=O)NCC(C)(C)CN(C(=O)Cc1conc1C(C)C)C)(C(C)C)NC(=O)OC 88273,c1(CC(=O)NC2C(NC(CC(C=C)C)=O)COC2)ccc(Cl)c(Cl)c1 88274,c1(C(N2CCC(CNC(C(CC#C)O)=O)(CO)C2)=O)ccc2cc(C)ccc2n1 88275,c1(C(N2C(C(=O)Nc3c(OC)ncnc3)CC2)=O)ccc(C(F)(F)F)c(I)c1 88276,N1(C(c2ccn(CCC)n2)=O)CCC(C)(C)C1C(=O)NC(c1ccncc1)C 88277,C1(NC(CSCc2c(C)noc2C)=O)CC(C)CN(C(=O)CCc2ccc[nH]2)C1 88278,N1(C(C2(CC#N)COC2)=O)CCOC2(C1)CN(CCc1ccc(F)cc1)C2 88279,c1(COC)nc(N(C2CN(C(C3(c4ccccc4)CCOC3)=O)C2)C)cc(C)n1 88280,CCC(F)(F)C(C)(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)C1 88281,C1(C(N(CC(=O)N(C)C)C)=O)CCCC1CNC(=O)CCn1cccn1 88282,c1(C(N2CCC(NC(CC(C(C)C)C)=O)(CO)CC2)=O)cnn2c1CC(F)(F)C2 88283,C12CCN(C(CC)C1)C(=O)C(N(C)C)CN2C.n1(CCC)nccc1C(=O)OC 88284,c1(C(=O)NCC2CCN(Cc3ccnc(C(=O)O)c3)CC2)cc(F)cc(F)c1F 88285,C1(CC(N2C3C(NC(C4CC45CC(O)C5)=O)C(C3)C2)=O)Cc2ccccc2N1 88286,C(C(=O)N=S(C)(=O)c1ccc(O)cc1)c1cccc(C)c1Cl 88287,c1(C(N2CCCC(F)(CNC(C(C)CF)=O)C2)=O)cn2cccc(Br)c2n1 88288,C12C3CC4CC1CC(C4)(C3)C(=O)N2.C1(CC(=O)OC(C)(C)C)(COC)CCCC1 88289,C1(CN(C)C(C23CC2CNC3=O)=O)CCCCN1C(=O)Cn1ccnn1 88290,N1(C(c2c(C)ncnc2)=O)CCC(C(F)(F)F)C(CNC(=O)CC2CCCO2)C1 88291,Cc1cnc2cccc(C(=O)NCC3CCN3C(=O)C=Cc3cc[nH]c3)n12 88292,C1(CNC(C(COC)COC)=O)CN(C(=O)Cc2ccc(F)nc2)C(C)(C)C1 88293,Cc1csc(=NCC(=O)NCC(C)NC(C2COC3COCC23)=O)[nH]1 88294,CCCC(CC)CCC(=O)NC(CCC1CC1)C(N)=O.C1C(C)CC(=O)N1 88295,C1(C(=O)NCC2CC(CC)C2)CCN(C(=O)Cc2cnn(C)c2)C12CCC2 88296,C(=O)(C1=CCCC1P(C)(C)=O)N(CC(=O)NCc1ncnn1C)C 88297,N1(C(C2(F)C(C)OCC2)=O)CCC2(CCC2)C(CNC(=O)C2=COCCO2)C1 88298,C(CCS(=O)(=O)c1ccc(F)cc1)NC(C1N(C)C(=O)NC1)=O 88299,N1(C(c2c(C)nsc2)=O)CCC(O)(CCNC(=O)CCC2CCCCN2C)CC1 88300,Cc1cc(CN2CC(O)CC2C(=O)NCCc2ccc(O)c(O)c2)c(C)cc1O 88301,C(C(F)(C(=O)NCCCC1CCOC1)C(C)C)NC(c1c(C)scn1)=O 88302,C(=O)(C1=NOC(C)(C)C1)N(C1COCCC1NC(c1cnc2[nH]ncc2c1)=O)C 88303,CN1CC(O)CC1C(=O)NC(CO)C(C)(C)C.C12CCC(O1)CNC2=O 88304,C(CO)(CCCCNC(C1(O)CCC1)=O)NC(=O)CCN1CCCCC1=O 88305,c1(C(N(CC(CNC(C(CCCC)N(C)C)=O)O)C)=O)c(C)ccc2n[nH]cc12 88306,c1(OC)cccc(Cl)c1CCN(C(C(=O)NCC(C)C)=O)C(C)Cc1ccc(Cl)c(Cl)c1 88307,Cc1c(C(N2CCSCC2C(=O)NC(c2ccno2)C)=O)oc2ccccc12 88308,c1(C(N2CC(C)C(NC(=O)Cc3ccc(F)cc3)C2)=O)cccc2c1ncn2C 88309,N1(C(C2COCCN(C(c3ccns3)=O)C2)=O)Cc2ccncc2C1 88310,c1(C(=O)NCC23CC(CN2C(C2CCC=CO2)=O)C3)cc2occc2s1 88311,C(CNC(=O)CSC(F)(F)F)(CC(F)(F)F)NC(Cc1cc(C)sc1)=O 88312,N1(CC(=O)NCC(CNC(c2c(C(C)(C)C)con2)=O)C)C(=O)CNC1=O 88313,N1(C(CCOC(C)C)=O)CC(NC(C2CC23CCSCC3)=O)CC(C)C1 88314,N1(Nc2ncnc(N3CCC4CCC(C3)S4)c2)CC2CC3CC(C2)CC1C3 88315,Cc1coc(C(N2CCCC2C(C)NC(c2n[nH]cc2C(C)C)=O)=O)c1 88316,N1(C(CCCN(C(C)C)C)=O)CC2(CCC2NC(c2ccc(F)cc2C2CC2)=O)C1 88317,CC(CN=c1ncc2ccccc2[nH]1)NC(C1(O)CC(COC)C1)=O 88318,c1(C(=O)NC(C)(CO)CO)cnc2c(-c3ccc4ccoc4c3)cnn2c1 88319,c1(C(=O)NCCCC2(NC(CC(CC)(C)C)=O)CC2)cccc2c1OCCCC2 88320,C1(C(C)C)CN(C(C2C=CC(NC(=O)CCc3cnoc3)C2)=O)CCN1C 88321,C1(CNC(CC(C)n2cccc2)=O)CCCCN(C(=O)COC(F)F)C1 88322,c1(C(N2CC(C)CC(NC(CN(C(C)=O)C)=O)C2)=O)ccc2ccc(Cl)cc2n1 88323,C1(CNC(C2C(C)C2C)=O)CC(F)CN1C(=O)COCc1ccncc1 88324,N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CN2CCC2C)CCF)C1 88325,C1(C)(OC)CC(N(C(c2ccc(C3CC3)nc2)C(=O)NC(C)(C)C)C)C1(C)C 88326,C(C(CO)C(C)(C)C)NC(C1CC(NC(CC2C(COC)C2)=O)C1(C)C)=O 88327,c1(NC2CCC(C(C)C(=O)NCC3CCN(C)CC3)C2)ccc(F)c(F)c1 88328,C=C=CCCN=c1[nH]c(N2CCC(C)(CN(C)C)C2)nc2c1COCC2 88329,C1(CC(=O)NC(C2(C(N3CC(n4cnnn4)C3)=O)CCCC2)C)COCC1O 88330,N1(C(c2c(C)cn[nH]2)=O)CC2CCN(C)CC(C2)C1 88331,C(=O)(C(F)CC(C)(C)NC(=O)CC#N)NC(C(C)(C)O)(C)C 88332,c1(C(=O)NC2CC(NC(C(COC)(C)C)=O)C2)cc(OC(F)F)cc(F)c1 88333,N1(C(CC(C)NC(Cc2cncc(C)c2)=O)=O)CC(CO)CCC1C 88334,C(CN=c1ccnc(NCc2conc2C2CC2)[nH]1)c1ccc(C)o1 88335,C1(C(=O)NCC=CCOCCO)(CC)CCN(C(=O)C=CC(F)F)C1 88336,C1(C(=O)NC2C(C(N)=O)CC=C2)C2CN(C(c3ccnn3CCF)=O)CC12 88337,Cn1ncc2nc(C(F)(F)F)c(C(=O)NC3CN(C(=O)CP(C)(C)=O)C3)cc12 88338,C(N=c1[nH]nc(C(C)(C)C)o1)(n1nnnc1CO)c1cnc[nH]1.CC 88339,c1(C(=O)NCCCCC(C)NC(CCCC#CC)=O)c[nH]c2cccc(C)c12 88340,c1(C(C)C)cccc(CNC(N2CCOC(CSc3cnc[nH]3)C2)=O)c1 88341,C(c1ccccc1)=CC(=O)NCCCCNC(C1(COCC)CCC1)=O 88342,C1(C(N2C(CCNC(C(C)(C)C(F)F)=O)CCCC2)=O)CCCC12OCCO2 88343,Cc1nc2cc(NC(=O)CC3CCC(NC4CNC(=O)C4)CC3)ccc2s1 88344,c1(COC(C2CC(=O)N(C(C3CCOC3)=O)C2)=O)ccccc1C(F)(F)F 88345,n1(COC)nccc1C(=O)NC(C)CC(C)NC(=O)CC1CCCC1 88346,Cc1n[nH]c(C)c1C(=O)NCC(C(=O)OC1CN(C2CCC2)C1)CC1CCCC1 88347,CC1CCc2[nH]nc(C(=O)N(CC(C)NC(c3cc(O)cs3)=O)C)c2C1 88348,C12(NC(C3N(C)CCCC3)=O)CCC(C(=O)NCC3CCC(O)CC3)(CC1)C2 88349,C1(C(N2CC(O)(C(C(=O)NCC#CCCC)F)C2)=O)CC12CCOC2 88350,N1(C(C2(C#N)CCCC2)=O)CCC2CCN(C(C3CC3C(N)=O)=O)CC2C1 88351,c1(C(N2C3(CNC(C4CC(=C)C4)=O)CCC2CC3)=O)cn2ccccc2n1 88352,N1(C(c2ccc(C)nc2)C(=O)NCC)CCc2cccc(OC)c21 88353,C1(C(=O)NC(c2c[nH]nc2C2CC2)CC)CCCN1C(=O)C=Cc1ccco1 88354,N12CCCC1C2=O.c1(CS(=O)(=O)NC)cn(CC(N2CCCC2)=O)nn1 88355,C1(C#N)(C(N(CCCCN(C(=O)CCCC#N)C)C)=O)CC2CCC1C2 88356,C(=O)(C1=NOC2COCC12)N1C(CN(C(c2c(C(C)C)nns2)=O)C)COCC1 88357,C(CN=c1[nH]ccnc1F)(c1ccccc1)NC(c1cn(CC)nc1)=O 88358,CC1CN(C(=O)CC(=O)NC2CCCN(C3C4CC3(C)CN4)C2)CC(C)O1 88359,N1(C(CC2CC(=C)C2)=O)CCN(C(C2(C)CC3CCC2C3)=O)CC(O)C1 88360,N1(C(C2(NS(N)(=O)=O)CS(=O)(=O)C2)=O)CCCCC(CNC(C2CCCO2)=O)C1 88361,C1(C(=O)NCCOCC2CC2c2ccccc2)CNC2(CCC2)C1 88362,c1(C(N2CCC(n3cc(CCC=O)nn3)CC2)=O)c(F)cccc1Cl.C1CC(F)(F)C1 88363,C1(NC(CN(C2CCC2)C)=O)C(C)(C)C(NC(=O)C2=COCCC2)C1(C)C 88364,Cc1cccc(OCC(=O)NN2CCCC2SC(C)CN(C)C)c1F 88365,c1(OC(F)F)ccc(F)c(-c2n[nH]cc2CC2(CO)COCCN2)c1 88366,C(=O)(C=C1SCC(=O)N1C)N1C(C)CC(NC(c2nc(C#C)sc2)=O)C1 88367,CC1(C)C(NC(=O)CC=C(Cl)Cl)CC1CC(=O)NCCC(F)(F)Cl 88368,N1(C(C(C)CO)=O)CCC2CCC(C1)N2C(c1cc(N)c(O)c(F)c1)=O 88369,C(C(=O)N=c1ccn(C)[nH]1)C1N(C(CCCC(CCCC)CC)=O)CCC1 88370,C1(C(=O)NCC(C)CNC(c2cnc3[nH]cncc2-3)=O)CCc2cnn(C)c2C1 88371,c1(C(=O)NCC(CC)(CC)NC(CC(CCC)O)=O)cc2cccnc2cc1F 88372,c1(C(N2CCOC(CNCC34CCC(F)C3CC4)C2)=O)ccc(Cl)cn1 88373,N1(C(c2cnc(CCC)s2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC12CCC2 88374,CC1(F)CN(C(=O)CCN)CCN(C(=O)C(=O)NCCC2CCCOC2)C1 88375,CCC(CCCC(=O)NCc1ncsc1C)NC(C1CCCCC1O)=O 88376,N1(C(C(C)Oc2ccccc2F)=O)CC2(CCN(C(C3CCCCC3)C)C2)C1 88377,CC1ON=C(C(=O)N2CCC(CNC(C3(C#N)CCN(C)CC3)=O)(OC)C2)C1C 88378,Cc1nn(C)c(Cl)c1C(N1CC(C)(NC(C2CC2F)=O)C1)=O 88379,CC1(C)CN(C(=O)COCP(C)(C)=O)CCN(C(C2CC3(CCC3)C2)=O)C1 88380,C=C=C(C)CC(=O)NCC1CCN1C(c1cncn1-c1ccccc1OC)=O 88381,c1(C(N2C(C3(NC(c4c(C)noc4)=O)CC3)CCC2)=O)cncc2cccnc12 88382,C(=O)(C#CC1CCCCC1)N1CCC2(CC(NC(CCCCCC=C)=O)C2)C1 88383,C(CC(C(=O)NCCCNC(=O)C(F)OC(F)(F)F)OC)OC 88384,N1(C(C2C(C(=O)OCC)C2)=O)CC(C(=O)NC2CCCCC2C#N)CC(C)C1 88385,C1(NC(c2c[nH]nc2C2CCCO2)=O)CC12CCN(C(=O)C1=COCC1)C2 88386,c1(C(N(CC(C)NC(=O)C=CC2CC2)CC)=O)cc(C#N)ccc1N 88387,CCC(CC)C(C(=O)N(C(CC(F)F)C(=O)N(CC(OC)OC(C)=O)C)C)OC 88388,N1(C(C(N2CC(C=CC)C2)=O)=O)CC(C)CC(C)C1 88389,CCC(C)C(CC(=O)NCC1(Cl)CC1(F)F)NC(=O)COc1cc(C)on1 88390,C1(CNC(c2ccc(OC)cn2)=O)CN(C(=O)C2=CCOC2)CCN1C 88391,c1(C(N2C(CC(N3CCC(CC(=O)OCC)C3)=O)CCC2)=O)cnn(C)c1Cl 88392,C1(NC(C23CCC(C)(C2)C3)=O)C2CC(O)C(C2)N1C(=O)C=CC1CCC1 88393,Cc1ccc(O)cc1C(N1CCCCCC1C(=O)NC(c1cn(C)nn1)C)=O 88394,c1(C(CC)NC(C2CCCO2)COC(C)C)ccc2nccnc2c1 88395,C1(CNC(C2C(C=C)C2)=O)CCCN(C(=O)C(C)(Cl)Cl)C1 88396,c1(C(=O)NCC2(CC(=O)NC3CCN(CC)C3)CC2)ccnc(C)n1 88397,C1(CNC(C2(C)C(C(=O)OC)C2)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)CC1 88398,N1(C(C2C(NC(c3ccn(COC)n3)=O)CC2O)=O)CC2(CCC2)CC1C 88399,C1(C(=O)NC(c2csnn2)C)N(C(=O)C2=CCCC2)CCC1(C)C 88400,N1(C(CCS(C)(=O)=O)=O)CC2(CCC(CNC(=O)CSC(F)F)O2)C1 88401,c1(OC(CNC(C=CCC)=O)C=CC)cc(Br)ccc1F 88402,c1(NC(C(CO)OC(COC2CCC(C)CC2)=O)=O)ccn2nccc2n1 88403,Cc1nn(C)cc1C(N1CC(C(O)C(=O)N2CC(c3cnn(C)c3)C2)C1)=O 88404,c1(COCC(=O)NC2(CC)CC2)ncc[nH]1.C(C)(C)(C)O.CC(O)NC(=O)O 88405,N1(C(c2ncn(C)n2)=O)CCCC1C1CCCN1C(=O)Cc1cc[nH]n1 88406,C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)NCC2CCCC(C)C2)OC)C1)OC 88407,C1(CC)CN(C(=O)C=Cc2ccnn2C)CCN1C(=O)CC(C)N1CCCC1=O 88408,c1(SCC(=O)NCC2C=CC2Br)ccccc1 88409,c1(C(=O)NC2C(NC(c3ccc(C)cn3)=O)COC2)cc(Cl)ccc1O 88410,CC1CCC(C(=O)NCCC(C)(C)O)CN1C(C1CCC(=O)O1)=O 88411,C(=O)(C1=C(Cl)CCCC1)N1C(C(=O)NC2CC(C(C)C)C2)(COC)C=CC1 88412,c12ccc(c(C)n1)[nH]2.C1(OCC(=O)OC)CN(C(=O)OC(C)(C)C)C1 88413,c1(CC(=O)NCCCn2cnccc2=O)ccccc1F 88414,C1(=O)C2=CCC(CC2)O1.C1(C(=O)NCC2(COCC)CCC2)CC2OC1C1CC21 88415,c1(C(=O)NC2C(C(=O)NCC3CC(COC)C3)C=CCC2)cnn2c1CCC2 88416,O=C(CC1=CCCC1)NCc1cn(C2CCCN(C(c3csnn3)=O)C2)cn1 88417,C12(CNC(C=CC)=O)CCCC1N(C(c1ccc([N+](=O)[O-])cc1)=O)CCC2 88418,Cc1ncccc1CCC(N1CCCC(NC(c2ccncc2Cl)=O)C1)=O 88419,C(=O)(NNc1ccc(F)c(F)c1F)Nc1cc(OC)cc(OC)c1 88420,c1(OC)cnncc1C(=O)NCC(O)C(=O)NCc1cccc(OC)n1 88421,c1(C(c2n(CCSC)nnn2)NCC(C)CC)cc(F)ccc1Cl 88422,c1(C(=O)NC(CCCCNC(C(C)OC)=O)C)ccc(-n2ccnc2)cn1 88423,C(=O)(N1CCC(C(=O)NC2(n3cnnn3)CC2)O1)c1cc(OC)ncn1 88424,C1(C2CCN(C(c3cnoc3Br)=O)C2)(NC(C(CC)OC)=O)CC1 88425,c1(C(=O)NCC2CCCC(CNC(C(CC)(C)CO)=O)C2)nccc2nn[nH]c12 88426,C1(NC(C=CC=CCC)=O)CCN(C(=O)CC(O)c2ccccc2)CC1(C)C 88427,Cc1cc(O)c(C(N2CCC(CNC(=O)Cn3ccccc3=O)CC2)=O)nn1 88428,N(C1CCOc2ncccc21)CC(O)CC1(O)CCCC1 88429,C1(CC)(NC(=O)CC(C)C(C)C)CCCN(C(c2csc(Br)c2C)=O)C1 88430,Cc1cc(C(=O)NCCC(C)N(C(=O)CC(C)(C)CN(C)C)C)cc(O)n1 88431,c1(OCC)ccc(NC(C(CC)OC2(CNC(=O)CC)CCC2)=O)cc1 88432,CC1CC(NC(=O)Cc2ccc(C(N)=O)cc2)CN1C(c1nocc1Br)=O 88433,Cc1ccccc1CN1CCCC(C(C)NC(=O)CC(C)c2ccccc2)C1 88434,C(=O)(C#CC1CCC1)NCc1ccc(C(N2CCCC(OCC)C2)=O)cc1 88435,C1(NC(CC(CCC)C)=O)CCN(C(c2ccccc2CO)=O)CCC1(F)F 88436,c1(C(C(=O)NCC2(NC(Cn3ncc(CC)c3)=O)CC2)C)ccccc1F 88437,CC(C)(C)CCC(F)C(=O)NC1CCCC(NC(c2ccc(N)c(Cl)n2)=O)C1 88438,c1(C(N(C2(C(N(C)Cc3cncn3C)=O)CC2)C2CC2)=O)ccc2[nH]ccc2n1 88439,c1(C(=O)NCC2CCN(C(COC(CC)C)=O)CC2)cc2cccnc2s1 88440,CC(O)C(C(=O)N(C)Cc1ccccc1CNC(C1CC1C(F)F)=O)N(C)C 88441,C1(NC(C=CC=CC)=O)CCN(C(c2ncc(OCC)cc2Cl)=O)C(C2CC2)C1 88442,C1(OC)(CSC2CC2)CCN(C(C2CC(C)(O)C2)=O)C1.C1C(=O)NC(=O)N1 88443,C(=O)(CC(CC)C(=O)OC(C)(C)C)NCC1OCCN(C(CCCCC)=O)C1 88444,C(C1CCCCCC1)=CC(=O)NC(CC(C)C)CNC(=O)CC1NC(=O)NC1=O 88445,CP(C)(=O)C1(C(=O)NC2CC(NC(=O)CC3CCC(=O)NC3)C(O)C2)CC1 88446,C1(NC(c2c(CC)cco2)=O)CCCC(C(=O)NCCc2c(C)n[nH]c2C)CC1 88447,c1(C(N2CCC(N(C)C(C3CC(F)C3)=O)C2)=O)ccc2nn(C)cc2c1 88448,C1(NC(C(C)=CC2CC2)=O)CCCC(NC(c2cccc(NC(N)=O)c2)=O)C1 88449,CCC(C)C(C)C(=O)NC1(C)CC(NC(c2c(Br)noc2C)=O)C1 88450,C(=O)(CCC(=O)N1CCCCC1CCNC(C1CCC(C(N)=O)C1)=O)NC 88451,N1(C(C2CN(c3c(C)cccc3)C(=O)C2)=O)CCC2(CCOCC2)C1 88452,CCCC(C)N=c1[nH]c(=NC2CC(N3CCOC3=O)C2)c2sccc2[nH]1 88453,C1(C(=O)NCCCN2CCC(C)CC2)COCCN(CC2CCOC2)C1 88454,c1(NC(c2n(CCC)nnn2)CN(CCC(F)(F)F)C)cccc(C)c1C 88455,C(=O)(C(C)CC(C)CC)NC1(C(N(CCCO)CC#C)=O)CCCCC1 88456,CC#CCCCC(=O)N1CCC(CNC(=O)COCc2ccc(C(C)C)cc2)C1 88457,C(CCC(CO)NC(=O)CC1CCCN1CC)NC(CCC=CC)=O 88458,CC(C)CCN=C(NCC1(C)CCN(C)CC1)N1CC2CC1CS2(=O)=O 88459,Cc1cc(C)n2cnc(C(N3CC(NC(c4cccc(F)c4)=O)C3)=O)c2n1 88460,O=C(CCCC#Cc1ccccc1)NCC1CCC(NC(C2CCCCO2)=O)C1 88461,CC1CCN(Cc2ccnc(F)c2)CC1NC(c1cncn1C)=O 88462,Cc1c(C(=O)NC(C)CCCNC(=O)CC2(C)OCCO2)sc(Cl)c1Cl 88463,C(=O)(Nn1ccccc1=O)C1(C)N(C(c2cncc(OC)c2)=O)CC1 88464,Cc1scc(C(N2CC(NC(=O)C(F)n3cccn3)CC2CO)=O)c1N 88465,N1(C(C=NOC)=O)CCC2C(CCCN2C(=O)CCc2nc3ccccc3[nH]2)C1 88466,c1(C(=O)NC2(C)CCN(C(=O)Cc3ccsc3Cl)C2)ccnc2ccccc12 88467,C1(CNC(=O)C2=CCC2)C2CN(C(=O)CC3CC4CC4C3)CC12 88468,CC1CCN(C(=O)CN2CCSCC2)CC1CNC(c1ccn(C(C)(C)C)n1)=O 88469,C1(n2cc(CCCN(C(C)C)C(C)=O)nn2)CN(C(=O)CC2(O)CC2)CC1C 88470,C(=O)(C1=COCCO1)N1C(COC)(CNC(c2[nH]cc(C)c2C)=O)CCC1 88471,n1(CCC)nccc1C(=O)NCC(C1CC1)N(C(=O)Cn1cncc1C)C 88472,C(C(C)(C)C(=O)NCC1(F)CC(NC(c2cnc(Cl)s2)=O)C1)OC 88473,CC(C)CC(C)(C)C(=O)NCC1CCCN1C(C12CC(CO1)C2)=O 88474,c1(N2CC(NC(c3ccc(F)c(SC)c3)=O)(CO)C2)nc(C)nc(C)c1F.C(C)(C)CC=O 88475,C(=O)(CCC(C)(C)NC(N)=O)NCC=CC(=O)NC(C(C)C)CO 88476,C1(NC(CCSCC(N)=O)=O)CCCC(CNC(c2cc[nH]c2)=O)C1 88477,C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1CCCCC1(F)F)=O 88478,C(c1ccc(OC)cn1)=CC(=O)N(C1CCN(C(C23CCC2CC3)=O)C1)CCC 88479,c1(CNC(C(=O)NC(c2noc(C)n2)CC)=O)c(F)ccc(Br)c1C 88480,C12(C(N3CC(OCCNC(C(n4cc(C)nc4)(C)C)=O)C3)=O)CCCCC1C2 88481,C1(C(N2CCCC(N(C)C)CC2)=O)(NC(c2c(CC)nns2)=O)CCC(C)(C)C1 88482,C1(NC(=O)C=CCF)CCOC12CCN(C(c1csc3c(Cl)cccc13)=O)CC2 88483,c1(C(=O)NCCCCCOC)nc(C2CCCN2C(=O)C(F)F)n2ccccc12 88484,C(CCC(=O)NCC1CNC(=O)C1)NC(C1CC(C(C)(C)C)C1)=O 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88502,c1(C(N2CCC(O)(C(=O)NC(CCCOC)CO)CC2)=O)cc2cccnc2[nH]1 88503,Cc1cccn(CC(N2CC3CC3(NC(C3CN(C)CCO3)=O)C2)=O)c1=O 88504,C1(N)CCN(C2CCC2)CC1.C1(C(C)O)CCCN(C(c2cc(C3CC3)ns2)=O)C1 88505,C1(C(N(CC(=O)OCC)C)=O)COC2(C1)CN(C(=O)C(COC)N(C)C)C2 88506,C1(NC(C(C)Oc2ccccc2)=O)C2CCC(C2)C1C(=O)NCCCO 88507,C1(NC(COCCC)=O)CN(C(c2cc(OC)no2)=O)C(C)(COC)C1 88508,CC1(C)CN(C(=O)C=Cc2ccc([N+](=O)[O-])s2)CCN(C(C2(C)CC2(F)F)=O)C1 88509,C(=O)(Nn1cccn1)C1N(C(CC(=O)OC(C)(C)C)=O)CC2CC21 88510,N1(C(c2nc(CC)oc2)=O)CCCCC1C(=O)N(CCn1cccn1)C1CC1 88511,c1(C(=O)OCC2CCC3C(C(=O)OCC)C32)cc2n(n1)CC(N(C)C)CO2 88512,C1(c2ccc(Br)cc2)(NC(C2CCS2)=O)CCCCC1 88513,Cc1cc(C(=O)NC2CC(O)CN(C(=O)CCCn3cncn3)C2)ncc1F 88514,Cc1cc(C)c(C(=O)NCC23CC2CN(C(c2cn(C)[nH]c2=N)=O)C3)c(C)n1 88515,C(=O)(C1CCCc2ccccc21)N1CC(C)N(C(c2cccc(O)n2)=O)CCC1 88516,C1(NC(C(C(=O)OC)C)=O)CN(C(=O)CCN2CCOCC2)CC12CC2 88517,N1(C(c2c(C)cco2)=O)Cc2ccccc2C1C(=O)Nc1cncc(C(N)=O)c1 88518,N1(C(CS(=O)(=O)N(C)C)=O)CC2CCC1CN2C(C1CCCC(O)C1)=O 88519,c1(-c2nc(C(=O)NCC3(C4(C)OCCO4)CC3)sc2)cccc(C#N)c1 88520,c1(C(C(=O)NCC(C)CNC(C2CC(=C3CCC3)C2)=O)O)cccnc1 88521,C1(C(=O)NCCC(CNC(=O)CN2CCCC2CO)O)CC2(CCC2)CO1 88522,c1(N2C(C)(CNC(CC)=O)CCC2)nc2c(F)cc(Cl)cc2s1 88523,CCC(C#N)C(=O)NC(CCSC)C(=O)N(C(C)C)CC1CC1 88524,c1(N(C)C)cccc(C(=O)NC2(CN(C)C)CN(C(=O)Cc3cc[nH]c3)C2)c1 88525,C(=O)(C(CC)CC(C)C)NCC1C(NC(CN(CCC#C)C)=O)C1 88526,CN1CC(C(=O)NC(CC2CCC2)C(=O)NCC2(C(F)(F)F)CC2)CCC1=O 88527,c1(C(N2C(CNC(COCC(C)(C)C)=O)CC2)=O)cc2sc(Br)cc2[nH]1 88528,N1(C(c2cc(C(CC)C)no2)=O)CC(CCNC(c2ncsc2C)=O)C(C)C1 88529,C1(C(N2CCN(C)C(CNC(=O)Cc3ccno3)C2)=O)CCC(S(C)(=O)=O)CC1 88530,C1(C(N(CCCOCCN(C)C(C2CC(F)CN2C)=O)C)=O)CC2(CC2)CN1C 88531,c1(C(=O)NCC(CNC(Cn2cc(C(C)=O)nn2)=O)O)csc(C#N)c1 88532,C1(C(=O)NC2CC3(C(NC(c4ccn(C)c4)=O)C3)C2)CC2(CCOCC2)C1 88533,Cn1ncc2ncnc(N3CCCC(CNC(=O)CN4CCCCC4=O)CC3)c12 88534,c1(OC)ccc(COCCCNC(C2CCC2C(N)=O)=O)c(F)c1.C1CC(=O)O1 88535,C1(CC(N2CC(OCC(C)C)C2)=O)C2CCCC2N1C(=O)C(C)(C)CN(C)C 88536,C12(C(=O)NCC3(NC(CCCSC)=O)CCCCC3)CCCC(CO1)C2 88537,C(=O)(N=c1cc(Cl)cn[nH]1)C1N(C(c2cc(C)c(Br)cc2C)=O)CC2(CC2)C1 88538,N1(C(COC2(C)CN(C(C3(C#N)CCC3)=O)C2)=O)CC2(C)CC1(C)CO2 88539,c1(OC)cc(C(N2CCCC2CNC(=O)C(c2ccccc2F)O)=O)ncn1 88540,C1(C(=O)NCC2(CSC)CC2)C2CN(C(=O)CC3CC4CC4C3)CC12 88541,C(=O)(CCC(F)(F)C(F)F)NC(c1cccc(Cl)c1)(C)C(=O)O 88542,N1(C(c2ccc3nn[nH]c3n2)=O)CC2(C1)CN(C(c1cc(=O)cc[nH]1)=O)CCO2 88543,C1(CNC(C(C)C2CCOC2)=O)(CNC(C2(C)COC2)=O)CC1(F)F 88544,c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)C2)oc(Br)nc1C 88545,C1(C(N2CCCN(C(CC3CCC(C)CC3)=O)CC2)=O)CCCCN(C)C1=O 88546,CS(=O)C=CC(=O)NCC1CC(NC(=O)Cn2cc(Br)cn2)C1 88547,C1(C#N)(NC(C2CN(C(C=CC(=O)OCC)=O)CC2C(C)C)=O)CCOCC1 88548,N1(C(c2n(CC)ncc2)=O)CCC(O)(CNC(=O)CC2CCC(=O)N2C(C)C)C1 88549,c1(C(=O)NCC(CN(C(C(CCC)=CCC)=O)C)C)cc2ncccc2[nH]1 88550,C1(C)(CC)CC(NC(c2c[nH]nc2OC)=O)CN1C(=O)Cc1ccnn1C 88551,C1(C(N(CCC)CCNC(c2ccn(CCF)n2)=O)=O)CCCCNC1=O 88552,c1(N(C)C)cncc(C(=O)NC2CC(NC(C3CC(n4ccnc4)C3)=O)C2)c1 88553,C12CC3(COC1C3)NC(=O)NC2.N#Cc1csc(C2CC(COC(C)(C)C)C2)n1 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88571,N1(C(C2CC(SC)C2)=O)CCCC1C1CCCN1C(C1CC(=O)CCO1)=O 88572,c1(C(=O)NC23CN(C(Cn4c(C)cc(C(F)F)n4)=O)C(C2)C3)ccc(F)c(F)c1 88573,S(=O)(=O)(c1ccc(NCC2(C)CCC(=O)N2)c(F)c1)N1CCC(SC)C1 88574,N1(C(C(C)O)=O)CC2CCCCC2(CNC(c2cncc3c(Cl)cccc23)=O)C1 88575,C#CC1(NC(=O)CCN(C(=O)CC2CCN(C)CC2)C2CC2)CCOC1 88576,N1(C(C2CN(Cc3csc(N4CCCCC4)n3)C2)=O)CC(O)CC(F)C1 88577,CC1(C)CC(C(=O)NC2CCCC2CNC(C2(Br)CC2(C)C)=O)=NO1 88578,C1(NC(CCc2cc(OC)no2)=O)CN(C(=O)CCc2cc(C)n(C)n2)CC1C 88579,Cc1cc(CCNC(=O)NC2(C)CCC(C)CC2)ccc1-n1cnnn1 88580,c1(C(=O)Nc2c(C(C)C)cc(Br)cc2)n[nH]c2cc(-c3ccnnc3)ccc12 88581,CCCCC(CNC(=O)CCOCc1ccccc1)NC(=O)C(O)CC 88582,c1(CC)n[nH]cc1C(=O)NCc1cc(OC)no1.C12(CC1(C)C)C(=O)N2C 88583,C1(CNC(C(C(CC)O)C)=O)CCC2CN(C(=O)Cc3nc(C)sc3C)CC12 88584,C#Cc1cccc(C(=O)NCC2CN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)c1F 88585,N1(C(CSCC(C)C)=O)CCCC(C(N2CC(C)(O)C2)=O)C1.C1(=O)OC1.C1CC1 88586,C(CCC(=O)NC(Cc1ccccc1)CCNC(=O)COC1CCOC1)OCC 88587,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 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88605,c1(OC)nc(C)ccc1C(=O)NC1CC(n2cc(C3CCOC3)nn2)C1 88606,N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 88607,C(c1c[nH]c2ccccc12)=CC(N1C(CCC(N2CCCC(C)CC2)=O)CCC1)=O 88608,C1(NC(CCN(C)CC)=O)CCN(C(=O)C(C(C)C)c2cnc(C)s2)C1(C)C 88609,c1(C(C)C(=O)NCCOC(C2(CC(=O)N(C)C)CC2)=O)cnn(C)c1 88610,C(=O)(C(C)(CCF)N(C1CC2CC2C1)C(C1CN(c2ccccc2O)C1)=O)OC 88611,C1(ONC(C2N(C(N3CCC(CO)CC3)=O)CCOC2)=O)CC2CCC1C2 88612,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)c2)=O)C1 88613,CC1CN(C(c2ccnc(OCCO)c2)=O)CC(C)C1NC(C1CCCC1O)=O 88614,C1(NC(C2(CNC(=O)C=CCF)CCCCC2)=O)CC2CCCC(C1)C2 88615,c1(CCC(N2CCC(NC(c3c(CCC)n[nH]c3)=O)C2)=O)ccc(F)nc1 88616,c1(OC)ncnc(NC(=O)CC2CCCN2C(c2ncccc2Cl)=O)c1C 88617,Cc1ncc(C(=O)NCC2CCCCN(C(c3cnc(C)s3)=O)C2)cc1N 88618,c1(C(=O)NC(CC)CNC(C2CCCO2)=O)c[nH]c2c(Cl)cccc12 88619,N1(C(C2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(c2cnc(Cl)[nH]2)=O)C1 88620,S(=O)(=O)(c1cccc(C)c1)N(C(C(CC(=C)C)OC)=O)CC(O)COCC 88621,C1(C(=O)NCC(C(C)C)NC(C2(C=C)CCOCC2)=O)CNC(=O)CC12CCC2 88622,C1(Nc2c(C(=O)OC)cn(C)n2)CC2CC1CN2C(C1(c2ccno2)CC1)=O 88623,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 88624,C(N=c1[nH]c(N2CCN(CC3CC3)CC2)nc2ccsc12)C1C=CCCC1 88625,N1(C(CS(CC)=O)=O)CCC(C2CC2)(NC(c2cnsc2)=O)C1 88626,c1(C(N2CC(CC(C)NC(=O)C(C)(O)C3CCC3)C2)=O)[nH]ccc1C1CC1 88627,Cc1nc(C)n(CCC(=O)NCC2(C(C)(C)O)CN(C(=O)CC(F)(F)F)C2)n1 88628,N1(C(C2CC3(C2)CC(F)C3)=O)CC2CCCC(C1)N2C(C1(O)CCCCCC1)=O 88629,n1(CCOC)nnc2c(N3CCC(NC(=O)C(C)CC(N)=O)(OC)C3)ncnc12 88630,N1(C(C(COCC)(C)C)=O)CC2(CC)CC1(CNC(=O)CC(C)n1cccn1)C2 88631,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 88632,c1(NC(C2(OC)CCN(C(C(CCCOC)C)=O)C2)=O)cn(C)c(=O)nc1O 88633,C1(CC=C)CCN(C(=O)CC2(NC(c3c[nH]c(=N)o3)=O)CC2)C1 88634,N1(C(c2ccc(F)c(F)c2Cl)=O)CCCC2C1CCN2C(c1ccncn1)=O 88635,c1(C(N(C)CC2OCCN(C(C(C)=C3CCC3)=O)C2)=O)ccn2cncc2c1 88636,C1(NCc2ccc(CF)cc2)CCC2COCCC2C1 88637,CC1(C)CC(C(=O)NCCNC(=O)CCc2ccc(Cl)cc2)C(C)(C)O1 88638,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 88639,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(C(C)CNC(=O)C(C)SC)C1)=O 88640,CC12CC(C(=O)NC3CCC(NC(C4CCSC4)=O)CC3)(C1)C1(COC1)O2 88641,c1(C(N2CC(CNC(CN3CCC(C)CC3)=O)C3C2C3)=O)ccc(Cl)cc1F 88642,C(C)(C)(CCC(=O)N(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)CCO1)OC 88643,c1(OC)cc(C(=O)NC2CC2C(=O)NCc2cc(CO)ccc2O)ccc1F 88644,c1(CCNC(=O)CC2C3CN(C(=O)CC4CC=CC4)CC23)cc(O)ncn1 88645,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 88646,c1(C(N2CCN(C(=O)Nc3cccc(C)c3)CC2)=O)cc(Br)cc2ncoc12 88647,c1(SC)ccc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CCOC2)o1 88648,c1(CNC(C2CCC(CNC(C3CCN(C)C3)=O)O2)=O)cnnc(O)c1 88649,C(=O)(CCCCN(C)C)NCC1CC(C)(NC(c2[nH]cc(C(C)=O)c2)=O)C1 88650,C1(C(N(C2CC3C(=O)NCC(=O)N3C2)C)=O)C2CC(C(O)C2O)S1(=O)=O 88651,CCC(C)N(OC)C(=O)C1CC=CCN1C(C1CC2(C1)CC2(F)F)=O 88652,c1(CC)nccn1CC(=O)N(CC(O)CN(C)C(C1CC1C(C)(C)C)=O)C 88653,CC(C)C(C)C(CNC(=O)Cc1c(Cl)cnn1C)NC(=O)COCC1CCC1 88654,C(C(=O)N=c1ccn(C(F)F)[nH]1)(C1CCOC1)NC(=O)CC1CCCC1 88655,CC(C)C(C)(CNC(=O)Cc1ccsc1)NC(=O)CCCOc1ccc(F)cc1 88656,N1(C(CCCOCC)=O)CC(NC(c2nc(C)n(C)n2)=O)CCC1C 88657,Cc1cccc(Cc2nc(-c3ccc(C)o3)nn2CCC(C)C)c1 88658,c1(C(=O)NC(C2CCN(C(c3ns[nH]c3=O)=O)C2)(C)C)ccc2ocnc2n1 88659,C(=O)(C1=CCCC1P(C)(C)=O)NC1CC(NC(C(C)(C)C(N)=O)=O)C1 88660,c1(OC(C)C(=O)N(CC(C)(C)CNCC)C)ccc(C#C)cc1NC(=O)CCOC 88661,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCC1 88662,C(=O)(CCCN1C(=O)C(=O)c2cccc(Cl)c21)N(CCCCNC(CCC)=O)C 88663,c1(OC)ccc(O)c(NC(=O)C=CCN(C(=O)CCCCCSC)C)c1 88664,C1(CC)CN(C(c2oc(CNC(=O)CCC=CC(C)C)nc2C)=O)CC(=O)N1 88665,c1(OC)cc(CC(=O)NC2CCN(c3cccc(C)c3)C2=O)ccc1Cl 88666,C1(NC(=O)Cc2ccccn2)CCC2CN(C(=O)CCCCC(F)(F)F)CC2C1 88667,c1(C(=O)NC2(CC)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 88668,c1(C(=O)OC)n[nH]c(=NC2CCN(C(C3CCCC3C)=O)CC2)s1 88669,N1(C(C(C(C)C)SCC)=O)CC2(C(N3CC(=O)NCC3C)=O)CCC1CC2 88670,N1(C(c2cncc(C#C)c2)=O)CCC2CN(C(=O)COc3cccc(Cl)c3)CC12 88671,C1(C(=O)OCC(=C)CC)CCCN(C(=O)C(N2CSCCSC2)=O)C1 88672,N1(C(c2cn(CC3CCOCC3)nn2)=O)CC(C(=O)NC2(CC)CC2)CC(O)C1 88673,CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(C1(CO)CCC1)=O 88674,Cc1cn2cc(C(=O)NC3CC(CNC(c4c(C)coc4C(C)C)=O)C3)nc2s1 88675,N1(C(CC2(CC)CCC2)=O)CC=C(C(=O)NCC2(CCOC)CC2)C1 88676,C1(N(C(CCNC(C)=O)=O)C)CCCCC1N(C(=O)CC1CCS(=O)(=O)C1)C 88677,C(CC(C(=O)NCCc1cnc(C)s1)NC(C1CCC1(F)F)=O)OCC 88678,C1(C(=O)Nc2cccc(C(N(C)C(=O)C3CC3)=O)n2)CCC2(CCC2)C1OC(C)=O 88679,N1(C(c2cc(C(F)F)ccc2F)=O)CC2CC(C1)CN(C(C1CC=CCO1)=O)C2 88680,C1(SCC(=O)N(C)NC(CN(C)C)=O)CCCN1C(c1cnoc1)=O 88681,c1(C(C)C)cc(C(=O)NCCOCCNC(C2COC(C)(C)CO2)=O)ccc1F 88682,C12C=CCCC1C(=O)N2.C1(C)CCCC12CC2.O=C1CCC(n2ccnn2)C1 88683,c1(C(=O)NC23CCN(C(c4c(N)non4)=O)CC2C3)cc(O)nc2c1CCCC2 88684,CC(O)CC(=O)NCC1(C(=O)NCCCC2CCCC2O)CC1 88685,C1(NC(C(C)c2ccsc2)=O)C2CN(C(=O)C(c3ccc(N)cn3)C)CC12 88686,Cc1cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc4c3CCC4)=O)C2)cc1F 88687,C1(N(C(=O)CNC(C)=O)CC#C)CCN(C(=O)C(N2CCOC2=O)C)C1 88688,c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cncc(N)c1.C1(O)CC1 88689,N1(C(C2C(CC)CCC2)=O)CCC(C2(O)CN(C(=O)C=CCCC=C(C)C)C2)CC1 88690,c1(C(c2n(CC)nnn2)N(C)C)ccc(C2CC2)c(F)c1.C(CCSC1CC1)N 88691,c1(C(=O)NC2CCC(NC(C(C)OCCC#C)=O)C2)ccnc2c1ncn2C 88692,Cc1c(C(C)C(=O)NC2(C)CN(C(C3CCCN3C=O)=O)C2)cccc1Br 88693,c1(C(=O)NCCNC(Cc2c(C)ccc(F)c2)=O)cccc2c(C)ccnc12 88694,Cc1c[nH]cc(C(=O)NC(C(C)NC(c2cn(C)nc2C(F)F)=O)C(C)C)c1=O 88695,c1(CNC2(COC)CCC(C)CC2)cccc2c1ncn2C 88696,N1(C(CC(=O)NCC#C)=O)CCC(CC)(NC(=O)C(c2cncnc2)C)CC1 88697,C(=O)(C1CCc2c[nH]nc21)N(CCC(N1CCC(O)C1CC)=O)CCC 88698,CCC(CCCC(=O)NCC(O)(CC)CC)NC(C1(CO)CCCCO1)=O 88699,N1(C(c2c(C)n(C(C)C)nn2)=O)CCC(F)(CNC(C2CC=CCC2)=O)CC1 88700,N1(C(C2CCC(C(N)=O)O2)=O)CCC2CCC(C1)N2C(=O)CCc1ccsc1 88701,N1(C(CCOCCC)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 88702,N1(C(=O)OC(C)(C)C)CCC(C)(CC(O)C(=O)N2CCC2C(F)F)C1 88703,N(C1CCCc2ccccc21)C(=O)NCC1CCC(N=[N+]=[N-])CC1 88704,Cc1cc(=NC(=O)N2CC(C)CCC2C2CC2)[nH]n1-c1ccccc1C(F)(F)F 88705,c1(CCC(=O)NCC2CN(C(CCS(C)=O)=O)CC2O)nc2ncccn2n1 88706,C1(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCCN1C(=O)COC1CCCC1 88707,C1(CNC(c2csc(O)n2)=O)C=CC(NC(c2coc(-c3ccsc3)c2)=O)C1 88708,N1(CC2CCC(C)O2)CCc2cnccc21 88709,C1(C(=O)NC2CC(CNC(=O)CCc3ccc(O)cc3)C2)CCn2nnnc2C1 88710,N1(C(c2ccccc2Cl)=O)CCCCC2C1CCCN2c1nnc(CO)s1 88711,N1(C(=O)CCc2cnn[nH]2)CCC(NC(=O)COC2(F)CC2)CC1 88712,c1(NCCC2CCN(N(C)C)C2)ccc(N2C(C(C)CCO)CC2)cc1F 88713,N1(C(CCC(CC)OC)=O)CC2CCCC2(NC(c2c[nH]nc2Cl)=O)C1 88714,c1(SC)cc(NC(=O)CNC(=O)CN2CCCCCC2)ccn1 88715,c1(N2CC(C(=O)NCC(CC)NC(=O)C(F)C(=O)OC)C2)ccccc1[N+](=O)[O-] 88716,C(=O)(CCC(C(C)C)NC(C1(C)CC(=O)C1)=O)Nc1ccc(C#C)nc1 88717,C1(C(N(CCCCCNC(C(C)N(CCOC)C)=O)C(C)C)=O)CCCC1(F)F 88718,N12CCC(F)C(C1)NC(=O)CSc1n(C)ccc1CC2=O.C1(C2CC2)CCCO1 88719,c1(C(=O)OC(C)(C)C)cccc(Cl)n1.C1(C2C(=O)O2)CCOC1=O 88720,N1(C(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)CC2CC2C)CC(O)C1 88721,c1(C(N(C2CCCC(NC(C3CC(=C)C3)=O)C2)C)=O)cnn2ccnc(N)c12 88722,O=CN1CCCC1C(N1CC2C(CNC(=O)Cc3cnoc3)C2C1)=O 88723,Cc1c(Cl)sc(Cl)c1NC(N1CCOCC(CNC(=O)Cc2c[nH]nc2O)C1)=O 88724,C1(NC(C(C)Cc2ccccn2)=O)CC2CCC1N2C(c1ccc(=O)n(C)c1)=O 88725,c1(CC)c(NC2CN3CCC23)nc(-c2ccccn2)nc1C.C12CCN(CC1)C2 88726,CCCCCCCCC(=O)N1CCN(C(=O)CCc2nc(C3CC3)no2)CC1C 88727,N1(CC(=O)N(CCNC(C2CN(C(C(C)N(C)C)=O)C2)=O)C)CCC(C)(C)C1 88728,CC1CCCn2c(NC(CN(C(=O)Cn3cnnn3)C)=O)cnc21 88729,C1(NC(c2n(C)ncc2)=O)CCCCC1NC(c1ccncc1F)=O 88730,N1(C(c2ccc3cnsc3c2)=O)CC2CCCC(C1)N2C(C1CN(C(N)=O)C1)=O 88731,C12(C(=O)NC3CCCN(C(c4ccc(OC)c(F)c4)=O)C3)CCCCN1CCC2 88732,N1(C(C(Cc2ccoc2)NC(c2c(OC)cnnc2)=O)=O)CC(O)CC(O)C1 88733,C1(NC(CC2(N(C(c3nccc(C)c3N)=O)C)CC2)=O)C2CCC3C(C2)CC13 88734,c1(CC)nc(NC2(COC)CCCN(C(=O)C(c3cccnc3)O)C2)cc(Cl)n1 88735,N1(C(c2c(C)ocn2)=O)CC2CCC1CN2C(c1nc(Cl)ccc1F)=O 88736,CC1CCN(C(C2CN(C)CCN2C)=O)CCN1C(C1CCC(C)C1)=O 88737,c1(SCC(=O)NC2CCCCN(C(CC(=O)N(C)C)=O)C2)cc2ccccc2o1 88738,CC1CN(C(=O)C=CCN(C(=O)CCc2ccnn2C)C)CC(C)S1 88739,C1(NC(c2ncn(C)c2)=O)CN(C(C2CC(=C(F)F)C2)=O)CC2(CCC2)C1 88740,c1(C(=O)NCC2C3CN(C(C(C=C)(F)F)=O)CC32)noc2ccc(F)cc12 88741,N1(C(CC2(C=C)CCC2)=O)CCCC1C1CCCN1C(C1CCc2nc[nH]c2C1)=O 88742,C1(C(C)NC(c2c[nH][nH]c2=N)=O)CCCN(C(c2cc(N)cnc2Cl)=O)C1 88743,Cn1cnc2cc(C(=O)NC3CC4(NC(=O)CC5(CO)CC5)COC3C4)ccc12 88744,C1(C(=O)Nc2c(OC)nsc2)COCCN1NC(=O)CC(C)c1ncc[nH]1 88745,C(C#Cc1ccccc1)OC1CC(NC)C1(C)C 88746,C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2nnn(CC)c2C)=O)C(CF)C1 88747,C1(C(N2CCC(CNC(c3onc(COC)n3)=O)C2)=O)CCCCNC1=O 88748,O=C(CC(C(F)F)NC(C1CC2CC2C1)=O)Nc1cnn(C2CC2)c1 88749,c1(C(=O)NC2CC(N(C(CC(C=C)C)=O)C)C2)cnc(O)n(C2CC2)c1=O 88750,C1(NC(CCCN(C)C)=O)CN(C(c2ccc(O)cn2)=O)CC1N=[N+]=[N-] 88751,c1(C2(NC(C3C(C(C)NC(C=CCCC)=O)C3)=O)CC2)ncco1 88752,c1(C(N(CCCN(C(c2nccc(C)c2O)=O)C)C)=O)cc2cccc(F)c2o1 88753,C#CCC(O)C(=O)N(CCCNC(=O)C(=Cc1ccccc1)C#C)CC 88754,C12(NC(C3C(C)=CCS3)=O)CCC(CC1)N(C(c1c(C3CC3)noc1C)=O)C2 88755,c1(C(N2C3CC(NC(c4cc5c(s4)CCC5)=O)C(C3)C2)=O)ccn2nnnc2c1 88756,CC(C)C(O)C(F)(F)C(=O)NCCC1CN(C(=O)C(c2ccc(Cl)s2)=O)C1 88757,c1(CNC(C2CC23CC3)=O)ccc2c(c1)CN(C(c1cn3ccnc3s1)=O)C2 88758,C1(CC(=O)NC2C(C)N(C(=O)Cc3csc(=N)[nH]3)CCC2)SC2=NCCN2C1=O 88759,Cc1c(C(N2CCC(F)C23CC3)c2ccccc2)cc([N+](=O)[O-])cc1[N+](=O)[O-] 88760,C1(NC(CC(C)OC)=O)CC2CCC(C1C)N2C(c1ccc(C(=O)CF)cc1)=O 88761,c1(C(N2CC(NC(CC(COC)(C)C)=O)C2)=O)ccc2c(c1)nc(C(F)F)n2C 88762,c1(OCC(=O)NC2CC2NC(c2ccnn2C2CCC2)=O)cccnc1 88763,N12CCC(O)(C1)CN(CCC)CCC2=O.OC 88764,N1(CC(=O)NC2(CO)CC2)CCC(CN(C)C(c2cc(C(F)F)[nH]n2)=O)CC1 88765,C1(CC(N2CC(C)(CSC)C2)=O)CN(C(C2CCC(C)CC2)=O)CCO1 88766,n1(CC)cc(C(N)=O)c(NC(N2CC(C3CCN(c4ncc(Cl)cn4)C3)C2)=O)n1 88767,n1(CC#C)cccc1C(N1CC(COC)(NC(=O)CCC2CCC2)C1)=O 88768,C1(CNC(C(C)(C)OC)=O)(CO)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C1 88769,C1(C(=O)NCC2CC(NC(C=C(C)C)=O)C2)C2CCCC12 88770,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 88771,C1(CC(N2CCOC(CNC(=O)CN3CCCCC3=O)C2)=O)(OC)CCCCC1 88772,c1(C(=O)Nc2c(C(=O)NC(C(=O)NC)C)scc2)ccc(Cl)c(F)c1 88773,C(CCC(C)NC(c1ccnn1C)=O)NC(C(=C(C)C1CC1)F)=O 88774,C1(C(N2CCN(CC3CCCC3)CC2)=O)(CN)CC2(CC(F)C2)C1 88775,c1(C(=O)NC(C)CCNC(c2nnn(C)c2C(F)F)=O)cc2n(c1)CCC2 88776,C1(C(C)(C)CN)CCN(c2ncccn2)CC1.c12cccc(c1)NC(=O)C(=O)N2 88777,C1(NC(C2(NC(C3N(C)CCC3)=O)CCC2)=O)CCC12CCCC2 88778,C#Cc1cnn(C)c1C(N1CCCC(N(C(=O)Cc2cn(C)nc2Cl)CC)C1)=O 88779,C1(CNC(=O)C(O)C2CN(C(C3CC3c3ccco3)=O)C2)COCC1O 88780,c1(N2C(N(CCOC)C)CCC2)nc(NCc2nnc(O)n2C)c2ncsc2n1 88781,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 88782,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CO)ccc(CC)c([N+](=O)[O-])c1 88783,c1(CNC(C(CC)OC2CCCC2)=O)cnn2c1CN(C(C1CC13CCC3)=O)CC2 88784,c1(SCCNC(=O)OC(C)(C)C)nn[nH]c1Cc1ccncc1 88785,C12(CNC(C3CC(=C)C3)=O)COC(CNC(=O)C(O)CCN(C)C)(C1)C2 88786,c1(C2C(CC)C2)csc(=Nc2cccc(OC)c2)n1CC1COCCOC1 88787,C(=O)(C(C(C)O)SC)NCCC(=C)CNC(=O)CCCCN(C)C(C)=O 88788,c1(C(N)=O)cc(C(=O)NCC(=O)NCCc2cn(CCO)nn2)co1 88789,CC1CCC(C)(C(N2CCC(O)(CNC(c3cc(Cl)sc3Cl)=O)C2)=O)C1 88790,C1(NC(CSCCOC)=O)CN(C(=O)C(C)(C)S(=O)(=O)C2CC2)CCC12CCC2 88791,Cc1cc([N+](=O)[O-])cc(C(=O)NCC2CCN2C(C2(CCF)CCC2)=O)c1Cl 88792,C1(OC)CC(N=c2[nH]c(=NC(C)c3ccncc3F)c3ncccc3[nH]2)C1 88793,N1(C(CNC(c2ccoc2)=O)=O)CCN(C(c2cc(O)ncn2)=O)C2COCC12 88794,n1(CCC)cc(C(=O)NCC2(NC(=O)Cc3cc(C)no3)CCC2)nn1 88795,c1(C(N2CC(C(=O)NCC3CC4(CCO3)CC4)C2)=O)ccc2c(c1)OCCCO2 88796,Cc1cc(C(=O)NCC(O)CNC(=O)C=Cc2cnc(C)s2)n(CCO)n1 88797,CC(C(=O)NC(c1nc(C(=O)N(C2CC3CC3C2)C)co1)C)C(C)(C)C 88798,C1(CNC(COCC(=O)NC)=O)CN(C(C23CSC(C2)C3)=O)CC1C(F)(F)F 88799,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 88800,N1(C(c2c[nH]c3ccncc23)=O)CCC2CCN(C(=O)CCOC3CC3)C2C1 88801,N1(C(C(C)OCC#C)=O)CCCCC(CC(=O)NCC(C)N(C)CCF)C1 88802,c1(CNS(NC)(=O)=O)ccc2occc2c1.N12CC(CC1=O)NC(=O)N1CC2C1 88803,CC1(C)CCCC(C(=O)NCC(C2CC2)NC(=O)Cn2ccc(C(F)F)n2)C1 88804,C12(C(=O)NCCCCC(=O)OC)COCC1CN(CCC(=O)N(C)C(C)=O)C2 88805,c1(C(N2CCN(C3CCCN(C(CCC(=C)Cl)=O)C3)CC2)=O)ccc(C)cc1Cl 88806,C1(NC(C)=O)CCC(CC(=O)NC(C)(CNC(=O)C(C)CC2CC2)C2CC2)CC1 88807,C(=O)(C(CCOC)OC)N(C1(NC(Cc2nc(COCC)sc2)=O)CC1)C 88808,CC(C)C(CCC(=O)N(CCO)CCN(C)C)NC(=O)CSCc1nc[nH]n1 88809,N1(C(C(C)OCC#C)=O)CCOC(CCCNC(=O)Cc2ocnc2CC)C1 88810,c1(OC)c(C)ccc(C(N2CC3CC2CCC3NC(=O)CC(C)O)=O)c1F 88811,c1(C(N(CC(CNC(CC(CC)C)=O)C)C)=O)c(N)c(Cl)cc(Cl)c1Cl 88812,c1(OC(C)=O)cc(C)c(C)cc1C(N1CC2(CC2)CC1C(=O)NC1CNC(=O)C1)=O 88813,C1(C(=O)NC23CCC(CNC(C(CC)(C)O)=O)(OC2)C3)CC2(C1)CC(C#N)C2 88814,C1(CNC(c2c(C)nccc2)=O)CN(C)CCN1C(c1cc(Cl)c[nH]1)=O 88815,N1(S(C(C)C)(=O)=O)CCCC2(CCCN(Cc3conc3C(F)(F)F)C2)C1 88816,Cc1cccc(Br)c1C(=O)NCC(C)C(=O)N(C(C)C(F)F)C 88817,N1(C(C2CCC(=C)CC2)=O)CCCC1C1CCCCN1C(c1ncncc1Cl)=O 88818,CC1CC(C(N2CC(NC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)C1(C)C 88819,N1(C(COc2c(C)onc2C(F)(F)F)=O)CCc2nnnn2CC1 88820,c1(C(=O)NC2CCCCC2F)c(Cl)ccc2ccncc12 88821,N1(C(=O)NCc2cc(C)c(C)nc2)CCNC(=O)CC1C 88822,Cc1c[nH]nc1NC(C1CCN(c2nncs2)C1)C.C1(C)C(=O)N1 88823,C(=O)(C(C)C(O)C(C)C)NC1CN(C(c2c(C)nc(CCC)o2)=O)CC1CO 88824,CC(CO)C(=O)NCC=CCNC(C1(CC2CC2)CCC1)=O 88825,N1(C(c2c(C)scn2)=O)CCCC(C(N2CCCC2CNC(N)=O)=O)(C(C)C)C1 88826,N1(C(C2(C)CCCOC2)=O)CCCN(CCNC(=O)Cc2cn[nH]c2)CC1 88827,CC(C)(O)C(C1CC1)NC(=O)CC1(NC(C2CNC(=O)N2)=O)CCOC1 88828,Nc1ncc(O)cc1C(=O)NCC1CN(C(c2ccc(CC3CC3)s2)=O)CCO1 88829,[N-]=[N+]=NC1CNCCC1NCc1ccc(Oc2ccccc2)cc1F 88830,N(S(=O)(=O)N1CCN(C(c2ccc(C(F)(F)F)cc2)C)C(=O)C1)C(C)C 88831,C1(c2n(CCCSC)nnn2)(NCC(c2cccc(Cl)c2)CO)CCN2CCCC12 88832,c1(CC(C(=O)NCCC(C)NC(c2cn(CC)nc2)=O)O)cc(Cl)cc(Cl)c1 88833,C1(NC(c2c(NC)cncc2)=O)CC2COCC1N2C(=O)COCCF 88834,N1(C(c2c(CC)ocn2)=O)CCC2CN(C(c3ccc(N)c(C)c3Cl)=O)CCC2C1 88835,C(=O)(C1=CCCOCC1)N1CCC(O)(C(C)NC(Cc2cccc(CC)c2)=O)C1 88836,N1(C(Cc2nc(CC)sc2)=O)CC(NC(=O)CC2CCC(C)(C)O2)C2(CC2)C1 88837,N1(C(C(CSC)OC)=O)CC(NC(C2CC3(C2)CC3F)=O)CC12CCOCC2 88838,c1(CC)ncc(C(N2CCCOC(CNC(=O)CCOC3CCC3)C2)=O)c(C)n1 88839,Cc1nc(C(=O)NC(C2CCCN2C(=O)C(c2ccccc2)C)(C)C)c(C)o1 88840,c1(N(CCCC)C)cc(O)nc(COC(=O)CC(C)(C)c2ccc(C)cc2)n1 88841,C=CC1(CC(=O)NC2COCC2NC(=O)CCCC2CCOCC2)CCCCC1 88842,S(=O)(=O)(c1cccc2c1OCCC2)N1CC(O)CC(OCC)C1 88843,N1(C(C(C)(CO)OC)=O)CCC2OCCN(C(=O)C=C(C)C(F)F)C2C1 88844,c1(C(N2C(C)CCC(NC(CCOC)=O)C2)=O)cc2c(OC)[nH]c(=N)nc2s1 88845,C(CCCCC(=O)NC1CCCCC1NC(=O)CCN(C)CC)=CC 88846,c1(C(=O)NCC2(O)CCN(C(C3(OC)CCC3)=O)C2)ccc(=O)n(CCF)n1 88847,N1(C(c2ccc(-c3cn(C)nc3)cc2)=O)CCC2CCN(C(=O)CNC=O)CC2C1 88848,Cc1ccc(C(=O)NCCC2(O)CN(C(C3CCOC3C)=O)C2)cc1N=[N+]=[N-] 88849,N1(C(c2c(SCC)cccc2)=O)CC2(C1)CN(C(C1CCC3CC13)=O)C2 88850,N1(C(CCC=C)=O)CCN(C(=O)Cn2cc(Br)ccc2=O)CC1CC1CC1 88851,C1(C(N2CCC(CC)C2)=O)CN(C(=O)C(C)COC)C(C)(C)C1 88852,CCC(COC)C(=O)NC(CNC(c1nncn1C1CC1)=O)(CC)CC 88853,C=CCC(CNC(=O)C=NOC)NC(=O)CSCC(=O)Nc1ccccc1 88854,c1(C(N2CC(CNC(=O)CC(O)C3CCCC3)C2)=O)cc([N+](=O)[O-])cnc1O 88855,N1(C(C2(F)CC2)=O)CC2CC2(Cn2cc(CCCO)nn2)C1 88856,C1(OCC)CN(C)C(C)(C(N2CCC(CN(C)C(c3ccccc3)C)CC2)=O)C1 88857,C=C(CNC(=O)COc1cnn(C)c1)CCNC(=O)C(n1ccc(C2CC2)n1)C 88858,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 88859,N1(OC(c2cc(F)ccc2F)C)CCC2(CC1)CCN(c1ncnc(=N)[nH]1)CC2 88860,c1(CCC(=O)NC2CN(Cc3ccccc3)C2)nc(O)n[nH]1.C12CN(C1)C(=O)N2 88861,c1(C(=O)NCCC2(O)CCN(C(CC(=O)NCC)=O)C2)ccc(C)c(C)c1Cl 88862,Cc1cc(C(=O)N(C2CN(C(c3ccccc3F)=O)C2)C)c2ccccc2n1 88863,N1(c2cc(C(=O)OC(C)(C)C)ncn2)CC(C2=NOCC2)C1.c12cnn(c1)C2 88864,n1(CCC(=O)NCC(C)CN(C)C(C2C3CC4C(C3=O)C24)=O)cc([N+](=O)[O-])cn1 88865,N1(C(C(=O)NCC)=O)CCC2CN(C(=O)CCSCCCc3ccccc3)CC12 88866,N1(C(C(CO)=C(NCC)C(=O)Cc2cc(Cl)ccc2Cl)=O)CC2CC1CN2CC 88867,CCC(O)C(C)C(=O)NCC1CCN(C(=O)CCC2CCCO2)CC1 88868,C(=O)(CCCCC(=O)OC)N1CC(O)(C(C(=O)NCc2c(C)nc(CC)o2)F)C1 88869,c1(N2C(C(=O)OCc3c(C)ccc(C)n3)CCCC2)ccc([N+](=O)[O-])c(C#N)c1 88870,C#Cc1ccc(C(=O)NCC2(O)CCN(C(C3(C#N)CCC3)=O)C2)cc1 88871,C(CCCCC(=O)N1CC(CNC(c2cc([N+](=O)[O-])sn2)=O)C2(CC2)C1)OCC 88872,C#CCCC(C(=O)N1CCC(N=[N+]=[N-])C1)NC(C1CC(=O)C1(C)C)=O 88873,Cc1nc(NC(=O)CCn2nnc3ccccc23)nc(Cl)c1I 88874,C(C(C)(C)C(=O)N(CC(O)CNC(=O)C(N1CCOCC1)C)C)OC 88875,C1(NC(CC(C)F)=O)CN(C(c2ccc(C(O)CF)cc2)=O)CC1n1cccn1 88876,C1(CCOC)(NC(c2n(CCC)ncc2)=O)CCN(C(=O)CC2CCN(C)C2)C1 88877,N1(C(C2(CC#C)CCCCC2)=O)CC2(CNC(c3c(C)coc3C)=O)CCC1C2 88878,c1(C(N(CC(CNC(CC(C=C)c2ccccc2)=O)O)C)=O)ccn(C)c(=O)c1 88879,C1(O)(CC)CCN(C(=O)C(=O)NC(c2cccc(-c3ccccc3)c2)C)CC1 88880,N1(C(CN(C2CCCC2)C(C(C2CC2)OCC)=O)=O)CCCC(O)CC1 88881,CC1(C)C(CNC(=O)Cn2cccn2)CCN1C(C1C2CC3C(C2)C13)=O 88882,c1(CN(C(=O)C(C)C)CCCNC(CSC)=O)ccc2c(C)csc2c1 88883,N1(C(C2(CCCC)CC2)=O)CCC2CC(O)CCC2C1.c1(OCCO)cc(C)on1 88884,c1(NC(C(C)NC(c2cccc(CC)n2)=O)=O)cnc(CO)nc1C 88885,C1(N(C(C(CC)N(C)C)=O)C)CCC2CN(C(c3cc(C)on3)=O)CC12 88886,C(C1c2ccsc2CCN1C(C1(C2CC2)CC1)=O)NC(Cc1nc(CC)sc1)=O 88887,Cc1cn(-c2ccccc2F)nc1CN1CC(O)(C(C)NS(=O)(=O)C(F)F)C1 88888,C(C)(CO)(CC(F)(F)F)NC(c1cc(OC)c(OCc2ccccc2)cc1)=O 88889,C1(CC)CCN(Cc2cc(C(C)(F)F)n[nH]2)C1C(=O)O 88890,C1(CNC(c2cc(CO)on2)=O)CCN(C(C2(CCO)CC2)=O)C1 88891,c1(SC)nccc(=NCC2CN(C(c3cn(CC4CCCO4)nn3)=O)CC2C)[nH]1 88892,C1(SCc2cn(C3C(C)CN(C4CC4)C3)nn2)CC(=O)N(C)C1c1ccccc1 88893,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(c2cc(C(N)=O)cn2C)=O)C1 88894,N1(C(C(F)=C(C)C)=O)CCOC(CCNC(=O)CCc2nccn2C)C1 88895,C12(NC3CCCN(C(=O)OC)C3)CCCN(C(c3ccc(O)c(N)n3)=O)CC1C2 88896,N1(C(C(CC)C(C)C)=O)CC2CCOC2(CNC(=O)C(C)=C(C)C)C1 88897,Cc1c(C(N2CC(CO)OC(CF)C2)=O)[nH]c2cc(Cl)ccc12 88898,CC#CCC(C(=O)NCCC1NC(=O)NC1=O)NC(c1cscc1Cl)=O 88899,C1(CC)CCCCC1C(=O)NCc1cn(C2CCCN(C(C3CSC3)=O)C2)nn1 88900,N1(C(C(CC=C)(C)C)=O)CCC2CCN(C(C3(F)CCN(C)CC3)=O)CC2C1 88901,c1(CNC2CCC(C(=O)NCC(C)O)C2)c(Cl)cc(F)cc1Cl 88902,Cc1cc(C(N2CC(NC(C3CCC4(CCC4)CO3)=O)C2)=O)c2c(n1)CCCC2 88903,N1(C(C(=O)NCC)=O)CCN(C(=O)CCCN2CCCC2)C(CC(F)F)C1 88904,N1(C(C2(CCC=C)CC2)=O)CCC2(CCCCC2NC(=O)CSc2cccs2)C1 88905,S(=O)(=O)(c1ccc(NCc2cnccn2)c(Br)c1)N1C(C)C(C)(C)CC1 88906,C12(CC(=O)NC(CCNC(C(CC)N(C)C)=O)C)CC3CC(CC(C3)C1)C2 88907,c1(CCCCOCC(c2n(CCOC)nnn2)(C)N)ccc(F)cc1.C1(O)CC1 88908,C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1(C)C 88909,Cc1c(-c2ccccc2)nn(C)c1C(=O)NC1CCN(C(=O)CC(C)F)C1 88910,c1(C(N2CCN(C(C3CC4CCCCCC34)=O)CC2)=O)cc(O)ccc1Cl 88911,C(C(C)(C)C(=O)NC(CN(C(=O)C(C)(C)F)C)C1CCC1)OC1CCOCC1 88912,c1(OC)ccc2nc(C(N3CCC(C(C)CNC(C4CSC4)=O)CC3)=O)cn2n1 88913,c1(C(N(CC(CC)NC(=O)C(CC)SC)C)=O)cc(C)c2c(O)n[nH]c2n1 88914,C(CC1=CCCCCC1)NC(C1(CF)CCN(CC(O)Cc2ccc(F)cc2)C1)=O 88915,c1(C(=O)NC2(CC(N)=O)CN(C(c3ccncn3)=O)C2)cc2cccc(Cl)c2s1 88916,N1(C(C(CC=C)(C)O)=O)CC(NC(C2CC2c2cnn(C)c2C)=O)C2(CCC2)C1 88917,C(=O)(CC1=CCCCC1)N1CCC(C)C1CNC(=O)COc1cccc(Cl)c1 88918,CC1(C)CCC=C1C(=O)N1CCC(CCNC(=O)C2CC2)C1 88919,N1(C(CSCCCC)=O)CCC2(CC2)CC1C(=O)NCC1CCN(C)CC1 88920,c1(C(=O)NCC(=C)F)ccn(CCNC(=O)CC(C)OC)c1 88921,c1(C(=O)NCCOCC(=O)Nc2cccc(C3CC3)c2)c(O)cccc1F 88922,N1(C(C(C=C)O)=O)CC2(C(=O)NCC(O)C(=O)OC)CC1CO2.C 88923,c1(C(=O)NC(CCNC(c2ccc(CC)nc2)=O)C)ccc2c(=O)cc[nH]c2c1 88924,Cn1ncc(C(N2CCOC(C(=O)NC3CC(C)(O)C3)C2)=O)cc1=O 88925,c1(Cc2cccc(C)n2)cc(=O)n2nccc2[nH]1.C12(CC1)C(=O)N(C)C2 88926,C(CCNC(C1C(NC(c2cc(Cl)ns2)=O)C1(C)C)=O)(C(C)C)OC 88927,C(CCNC(=O)C1=NOCC1)(C(=O)NCCOC1CCC(C)(C)C1)OC 88928,C1(CNC(C(CC)NC(N)=O)=O)CCN(C(c2nccnc2C(N)=O)=O)CC1 88929,c1(C(N(C2CCCC(NC(CNC(=O)NC)=O)C2)C)=O)ncn2cccnc12 88930,c1(CC(N2CCCC(C)(NC(CCCC)=O)C2)=O)ccc2cnccc2c1 88931,Cc1cn2cc(C(=O)NC3CC(CNC(C4CCC=CCCC4)=O)C3)ccc2n1 88932,N1(C(C(C)Cc2cnn(C)c2)=O)CC2(CCCCN2C(C2CCC(N(C)C)C2)=O)C1 88933,c1(CC(N2CCC(N(C(=O)CC(F)F)C)C2)=O)ccc2c(c1)ncn2C 88934,N1(C(c2ccncc2C)C(=O)NCC(=C)C)CCc2cc(Br)ccc21 88935,C1(C)(C(=O)Nc2nc(CC)sc2C)CCCN(c2ccncc2)C1 88936,C(=O)(C(CC)C(=O)N(CC(=O)NCC1(C)CCN(C)CC1)C)OCC 88937,c1(CC)c(C(=O)NC(C)CN(C(=O)C(C)(C)C2CCOC2)C)nnn1C 88938,c1(NC(C(C2(O)CN(C(=O)CCC3CCCO3)C2)F)=O)csc(CO)n1 88939,Cc1ccccc1N(C(=O)C(c1ccc(Cl)nc1)(F)F)C.N12CCOC(C1)C2 88940,c1(-c2cccc(C(N3CC(CO)C4CC34)C(=O)NC)c2)ccccc1C(F)(F)F 88941,c1(N(C(CCn2cc(C3(NC(C)=O)CC3)nn2)=O)C)ccc(-n2cnnc2)cc1 88942,Cc1cc(C#N)ccc1C(N1CCC2CCCC12C(N1CCC1C1CCCCC1)=O)=O 88943,C1(N(C)C)(C(=O)O)CCCN(Cc2cn(Cc3nncs3)nn2)C1 88944,c1(C(N(CC(NNC(=O)C2CCN(CC)C2)=O)C)=O)cccc(S(=O)(=O)NC)c1 88945,N1(C(c2n(C)ccc2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C(F)(F)C1 88946,CC(C)CC(CNC(=O)C=Cc1cncn1C)NC(C1CN(C)CCO1)=O 88947,c1(OC)ccc(C(=O)N(CC(C)CNC(=O)C=Cc2cncs2)C)cc1OC 88948,C=CCC(C(=O)N1CC(O)CC1C(=O)NCC(c1nncn1C)C)NC(C)=O 88949,CC1C(C=CC(N2CC(O)(CNC(=O)C(C)Oc3ccccc3)C2)=O)C1(Cl)Cl 88950,C(CCNC(C1(CSC2CC2)CC1)=O)OCC 88951,CCC(CC)C(F)C(=O)NC(CCCC)CC(=O)NCC#Cc1cnn(C)c1 88952,C1(CN(C(=O)CC2CC(CF)C2)C)CCN(C(=O)CC(Cl)Cl)CC1 88953,CCC(C)(CNC(c1cc(CCO)on1)=O)NC(C1CC1F)=O 88954,c1(NC(Cc2nc(NC(C(=Cc3ccccc3)C)=O)sc2)=O)ccc(C#N)c(F)c1 88955,c1(C(N2CCC(NC(c3c(COC)ccs3)=O)CC2)=O)cccc2c1CCCN2 88956,c1(C(C)NC(c2ccc(F)cc2F)c2ccccc2)cccc(S(N)(=O)=O)c1 88957,C1(C(N(C2CCCC2)CCCNC(CC(C)(C)O)=O)=O)C2CCCCCC12 88958,C1(C)(C(=O)NCc2ccc(CN(C(=O)CCC(=O)N(C)C)C)cc2)CCCS1(=O)=O 88959,C1(C(=O)Nc2cccc(NC(=O)C(F)Cc3ccccc3)c2)CCCCCCC1 88960,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCCC3)CC1C 88961,N1(C(C2(CC)CC2)=O)CC(CCNC(C2CC(=O)N2)=O)(OC)C1 88962,C=C1Cn2c(C(=O)NCCC3(CNC(C4(CC(C)C)CCC4)=O)CC3)nnc2S1 88963,c1(N(S(=O)(=O)C(F)(F)F)C(c2ccco2)=O)ccc(Br)c2c1CNCC2 88964,c1(CC)occc1C(=O)NCCOCCCN(C)C(c1c[nH]nc1C1CC1)=O 88965,c1(C(N(CC(CN(C(C2N(C)CCCC2)=O)C)O)C)=O)cn2ccsc2n1 88966,CN1CCOCC2(COCCN2C(C2CCC3(CN(S(=O)(=O)C(C)(C)C)C3)O2)=O)C1 88967,C1(CN(c2nccc(OCC)n2)CC)COc2ccccc2C1 88968,C1(C(N(CC(COC)O)C)=O)CC(F)(F)CN1C(c1cccc(F)c1O)=O 88969,c1(C(C)C)ccc(N2CCN(C(C3(N)CCSC3)=O)CC2)cc1 88970,C1(C)(NCCSCCCNC(C(c2cccnc2)OC(C)=O)=O)C(C)(C)C1(C)C 88971,c1(OCCC(=O)NC2CC(c3ccccc3)CO2)ccc(Br)cc1 88972,N1(CCC(=O)NCCCN(C(c2cnc(C)o2)=O)C(C)C)CCCCC1=O 88973,C1(C(C)NC(=O)Cn2nnc(-c3cccs3)n2)CCCN1C(=O)CCn1cncn1 88974,C1(CC)CC(C(=O)NCCc2csc(C)n2)CCN1C(=O)C(C)OC(C)=O 88975,C(CC(C)CCNC(C1CCN(C(C)=O)CC1)=O)NC(C1N(CC)CC1)=O 88976,c1(OC)c(-c2nc(C(C3CCCCC3)N)no2)ccnc1F 88977,C1(C(=O)NC(CC=C)CO)CC(N=[N+]=[N-])CN1C(=O)C(O)CN(C)C 88978,C(=O)(C(CCSC)SC)NCCCCCN(C(CC)=O)C 88979,CCC(CC)CC(F)C(=O)NC(CNC(C1CCC1)=O)CCOC 88980,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(=N)s2)C1)=O 88981,C1(C(=O)NCC2(NC(CCSC)=O)CCCCC2)CN2CCN1CC2C 88982,c1(C(=O)NC(C)CCC)ccc(Br)cc1.C12(CCC1)C(=O)N2.CC(C)OC 88983,N1(C(c2c(OC)scc2)=O)CC2CN(C(=O)CN(C3CCC3)C)CC2(C)C1 88984,c1(C(=O)NCC2N(C(CCSCCCC)=O)CC(C)CC2)cccc2nonc12 88985,N1(CC#N)CCN(C(=O)CC2CCCCN2C(C2(O)CC2)=O)CC1 88986,C1(NC(=O)Nc2cccc(C)c2)COCCN(C(C2(CF)CC2)=O)C1 88987,C1(OC)CC2CCC(C1)N2C(c1ccc(F)c(CC2CC(=O)N(C(C)C)C2)c1)=O 88988,c1(NC2CCN(C(=O)NC(c3ccccn3)CCC)CC2)cnc2n1CCOC2 88989,C1CS(=O)(=O)N1.C(C(O)CN1CCCC1)OC(C)(C)C 88990,C=CCCC(C)(C)CNC(C1(CO)CCN(C(=O)C(CC(=C)C)OC)C1)=O 88991,c1(N2C(C)C(NC(c3ccc(C(N)=O)cn3)=O)CCC2)ncc(C#N)cc1Cl 88992,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 88993,c1(-c2ccc(OCC)c(O)c2)ccc2cc(C(=O)NCC3CCC(F)C3)nn2c1 88994,CC1(C)CN(C(C2CCCSC2)=O)C1C1CCN(C(c2cnc(Cl)[nH]2)=O)CC1 88995,C1(NC(c2cn(C3CCOC3)nn2)=O)CC12CCN(C(c1cnns1)=O)C2 88996,c1(CNC(C2(CCNC(C3CCC4CC34)=O)CC2)=O)ccccc1SC(F)(F)F 88997,C#Cc1ccc(CC(=O)N(CC(C)O)CCNC(=O)C(=Cc2cccnc2)C)cc1 88998,C1(C(=O)NC(C(C)C)CNC(=O)C(C2CCCCC2)O)CCCCN1C 88999,CCCC(C)CCCC(=O)NCc1cc[nH]c2nccc1-2.C12(CC1)C(=O)NC2 89000,C1(C(=O)NCC2(NC(C3CCC(C)(C)CC3)=O)CCC2)Cc2ccccc2CO1 89001,c1(C(N2CC3CN(C(C#CC)=O)CC3C2)=O)c(C)cccc1[N+](=O)[O-] 89002,N1(C(COCC(C)C)=O)CC(NC(=O)CCCn2ccccc2=O)CC2(CC2)C1 89003,N1(C(CSCC#C)=O)CCc2ccc(CNC(=O)C(F)C(F)(F)F)cc2CC1 89004,c1(C(N2CCC(C)(CNC(C(CC#C)(C)C)=O)C2)=O)ccc2ncnn2c1 89005,N1(C(C(C(CC)C)NC(=O)C2=CCN(C)C2)=O)CC(F)(F)C(F)(F)C1 89006,Nc1nccnc1C(C(F)(F)F)NC(=O)CCNC(=O)CO 89007,N1(C(C=C2CCN(C)C2)=O)CC(NC(c2csc(N3CCCCC3)n2)=O)C2(CC2)C1 89008,C1(=O)C#CC(C)(C)CO1.C(C(F)F)(C1CCCO1)OC(C)=O 89009,c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)CCN(C)C2)cccc2c1CCC2 89010,c1(C(=O)NC2CC(NC(c3c(C)c(F)ccc3)=O)C2)cnc2[nH]c(=N)sc2c1 89011,C1(C(N2CC(C)C(NC(c3cccc[n+]3[O-])=O)C2)=O)CC2CS(=O)(=O)CC2C1 89012,CC1(CNC(C2CC(F)C(=O)N2)=O)CCCN1C(=O)C=CC1CCCC1 89013,C1(C(=O)N(C(C)C(=O)NC(C)CSC2CC2)C)(CC)CCNC1=O 89014,c1(CC)cccc(C(=O)NC2CCCC(CNC(c3c[nH]c(=N)o3)=O)C2)c1O 89015,c1cc(=NCCCS)[nH]c(NCC2CCCCCC2)n1.C1(C2(N)CC2)CCCO1 89016,c1(C2N3CCC(F)(CC3)CNC2=O)cccc(CO)c1F.CCCCCCOC 89017,CN1CC(O)(CCNC(=O)CC2(NC(=O)C=CC(=O)NC3CCC3)CC2)C1 89018,CC1CCN(C(=O)CSCc2cscn2)CCN1C(C1CCC(=O)N(C)C1)=O 89019,N1(C(C(CC)N(C)C(c2cc(COC)[nH]n2)=O)=O)CCCC(COC)C1 89020,c1(C(N(CCCNC(C(CCOC)C)=O)C)=O)cnc2nc(O)nc(O)c2c1 89021,c1(CC(=O)NC2C(OC)CN(C(c3ccsc3OC)=O)C2)cc(F)ccc1O 89022,C1(CNC(C2CCCC(=O)N2)=O)CN(c2ncnc(O)c2Br)CCC12CCOC2 89023,N12CCC(CC1)CC(C)C1CCCN1C2=O.C1(C(=O)OC)CC(C#N)C1 89024,c1(-c2ccc(C(N(CCC)CC)=O)cc2)nn(C)c2c(C#N)cccc12 89025,c1(C(=O)NCC(N2C(CN(C)C(C3C4COCC34)=O)CCC2)=O)cn2ccsc2n1 89026,c1(CNC(C(C2(C)CN(C(c3ccnn3CCF)=O)C2)C)=O)nc(C#N)cs1 89027,C1(CCN2CCC2)CN(C)CCN1C(=O)C(C)C.Cc1ccccc1NC(C=CC)=O 89028,c1(C(C)C)ccc(N)c(C(N2C3CCC2C(NC(C2(C)CCCC2)=O)C3)=O)c1 89029,c1(C(C(=O)NCC=CCNC(C(=O)NCCNC(C)=O)=O)C)cccnc1 89030,Cc1nn(C)c(C(F)F)c1C(=O)NCCCCN=[N+]=[N-] 89031,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89032,N1(C(CC2C(C)(C)C2)=O)CCC(C(=O)NCc2c(CC3CC3)cco2)CC1 89033,C(CC(C(=O)NC1CCCCC1)N(C)Cc1cnn(C)c1)SC 89034,C1(CCC(N2CC(CC(C)NC(=O)C(c3ccnn3C)O)C2)=O)C=CC=CC=C1 89035,C(=O)(CCN=C(Nc1nc2c(s1)CCCC2)N1CCCC1)N1CC(C)CC(C)C1.C 89036,Cn1cc(C(=O)NCC2CCC(NC(c3nccn3C)=O)CC2)c(C(C)(C)C)n1 89037,C1(C(=O)NC(COCCCNC(CCSC)=O)(C)C)OCCC1C 89038,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(=O)C(C(C)C)N(C)C)C(C2)C1 89039,Cc1ccc(C2CCCC2n2cc(Cc3ccc(Br)cc3)nn2)c(Br)c1 89040,C12(CNC(=O)C(c3ccc([N+](=O)[O-])cc3)O)CC=CCN1CCC2 89041,N1(C(CC)=O)CCCC(C(=O)NC2CCCC2NC(c2[nH]nnc2C(=O)O)=O)C1 89042,N1(C(c2c(CNC(c3c(CC)noc3)=O)occ2)=O)CC2CCC2(OC)C1 89043,C1(C(=O)NC2C(NC(COc3cccc(CC)c3)=O)CCC2)C(F)(F)C12CCC2 89044,C1(OCC)CC(F)CN(C(C2C=CC(NC(c3cccn3C3CC3)=O)C2)=O)C1 89045,c1(CC(=O)NC2CC3(C2)CN(C(=O)C(F)n2ccnc2)C3)cc(F)cc(F)c1 89046,C1(NC(C(C)S(C)(=O)=O)=O)CN(C(=O)CN2CCOCC2)CCC12CCC2 89047,c1(OC2C(n3cc(C(N(C)Cc4ccn(C)n4)=O)nn3)C2)cccc(C#N)c1 89048,O=C(CCCc1ccsc1)NC1CCCC1n1cc(CCN2CC3CC3C2)nn1 89049,N1(C(CCc2ccc(SC)cc2)=O)CCC(NC(C2C=CCC2)=O)C(O)C1 89050,C1(C(N(C2CCN(C(c3csc(O)n3)=O)C2)C)=O)CCS1(=O)=O 89051,C1(C(=O)NCCCN(C(CCC(CC)OC)=O)CCO)CCCC(C)(C)CC1 89052,N1(C(CC)CO)CC(=O)N(CC(=C)C)C1 89053,c1(C(N2C(C(C)NC(c3n(CC)cnn3)=O)CCC2)=O)cccc(C(F)(F)F)n1 89054,N1(C(c2ccccc2C(=O)NC2CCO2)=O)CCN(c2cccc(Cl)c2)C(=O)C1 89055,N12C(CCC1C(F)F)C(=O)NC1CCC(C1)NC(=O)CC2.C1(O)CCCCC1 89056,C(=O)(C(O)CC(C)C)NC(CC)(C)CN(C(=O)CC1CNC(=O)C1)C1CC1 89057,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89058,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89059,C1(NC(C(COCC)N=[N+]=[N-])=O)CC(N=c2[nH]cnc3cnccc23)C1 89060,c1(OC(C)C)ccc(F)cc1C(=O)NC1CCCC(NC(C2(CCO)CC2)=O)C1 89061,C12(CN3CCC(c4ccc(Br)cc4)CC3)CCCCCC1NCC2 89062,Cc1cncc(C(=O)N(C2CN(C(=O)CCC=CC(C)C)CC23CC3)C)c1C 89063,C12(NC(C(n3cc(C(C)C)nn3)C)=O)CCC(C1)C(O)C2O 89064,CCCC(O)CCN=c1nc(N2CCC(CF)C2)c2sccc2[nH]1 89065,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CC(O)C2CCCC2)C3)cc(C)c1 89066,c1(-c2cn(CC(=O)NC3CC3)nn2)ccccc1C1=CCS(=O)(=O)CC1 89067,c1(C2(C(F)(F)F)C(NC(CCS(C)=O)=O)CN2C(=O)C(C)(C)F)cc(F)cc(F)c1 89068,C1(CC(=O)NC(CC=C)CNC(=O)CCSC)CN(Cc2nc[nH]n2)CC1CC 89069,C(=O)(C1=CCSC1)NCc1c(C(=O)NCCC(CC)C)cco1 89070,C1(CC(C)C)C(=O)N1.c1(C(C)NC(C(COCC)OC)=O)ccc(C)nc1 89071,C(C)(C(O)C(=O)N(C)CCNC(c1ccc(C2CCCCC2)nc1)=O)OC 89072,C1(n2cc(C3CCOC3)nn2)(C(N(CCC2CC2)CC)=O)CCOCC1 89073,C1(CC(=O)NC(COCC)C)CC(C)N(C(=O)C=Cc2cncs2)C1 89074,C(=O)(C(C)C(C)(C)O)NC1C(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)COC1 89075,N1(C(CCCCSC)=O)CCC(NC(c2ccn(CC(F)(F)F)n2)=O)C(O)C1 89076,C(=O)(CCC(=O)N1CC(CC)C(c2ccnn2C)C1)Nc1nnc(CCC)s1 89077,C#CC1(C(=O)N(C)Cc2ccn(C)n2)CN(C(=O)C(=O)CC)C1 89078,CC1(C(=O)NCC2(NC(c3coc(Br)c3)=O)CC2)CC2CCC1C2 89079,c1(C(C(=O)NCC(=O)NC)NC(=O)CCOCCOCCCO)cnn(C)c1 89080,c1(CCC(=O)NCC(=C2CN(C(c3cc(Cl)no3)=O)C2)F)nnc(O)nc1O 89081,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(CC(C)C)nc2)=O)C12CC2 89082,N1(C(c2cscc2-c2ccccc2)=O)CC(O)C(O)C1CNC(C12CC(C1)C2)=O 89083,N1(C(C(CC2CCC2)NC(c2c(C)non2)=O)=O)CCC(O)C(C)(C)C1 89084,c1(C(=O)NCC2C(NC(C=C(C)c3cccs3)=O)CCCC2)cnc(O)cc1C 89085,O=NN1CCCCC1C(=O)N(CCCNC(=O)C(F)C(F)(F)F)CCO 89086,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89087,N1(C(c2ccn(C3CCC3)c2)C(=O)NC(CC)(C)C)CCC(F)(C(N)=O)C1 89088,O=C1CCCc2c(NC(C3CC(NC(c4ccc(Br)c(Cl)c4)=O)C3)=O)cccc21 89089,N1(C(Cc2nc(SC)sc2)=O)CCC(SCC(C)N(C)C)CC1 89090,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1(Br)CC1)=O 89091,c1(CN(C(=O)Cc2cccnc2)C(C)C)cc(Br)ccc1OC(F)F 89092,c1(C(N(CCCNC(c2coc(C3CC3)n2)=O)C)=O)ccnc(C(C)(C)C)n1 89093,CCC(C)(C(=O)OC(C)C(N1CC(OC2CC2)C(c2ccccc2)C1)=O)C(F)F 89094,C(=O)(CC(F)F)NCCOCCCN(C)C(c1ncccn1)=O 89095,c1(CC)nc(C)cc(=NCCC2CN(C(C3CCCCN3C3CCCC3)=O)C2)[nH]1 89096,C(C(=O)NC1CC(NC(C2(F)CCOCC2)=O)C1)(C(=O)OC(C)(C)C)OC 89097,Cc1cccn2cc(C(=O)NC3CCN(C(c4cncc(Br)c4)=O)CC3C)nc12 89098,Cc1ccc(C(F)(F)F)cc1C(N1CCC(C)(NC(c2ccccc2)=O)C1)=O 89099,c1(C(=O)NC2CN(C(C3C(=C)C3)=O)CC3(C2)CCC3)ccc2cccc(OC)c2n1 89100,[N-]=[N+]=NCCCCC(=O)NC1(C(=O)NCC2CCCC2O)CCC1 89101,C#CC1(C(=O)N(C)CC2CCCCCC2)CCN(C(=O)C(F)C(C)(F)F)C1 89102,C#CC1(CC)COCCN1C(=O)Nc1c(SC)n[nH]c1 89103,c1(OC)ccc(CC(=O)NCCCNC(c2cnc3n2CCC3)=O)cc1F 89104,c1(N(C2CN(C(C)=O)C2)C)nc(=NC)[nH]c(=NC2COCC2F)[nH]1 89105,N1(C(CCOCCC)=O)Cc2ccccc2CC1CNC(=O)C(C(C)C)OC 89106,Cc1noc(C)c1C(C)(C)C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C 89107,C(C(=O)NN1CCCC1C(=O)NCc1cnn[nH]1)OCC=C 89108,C1(CNc2cc(F)cc(F)c2)CCCC2OCCC12.C12CC(OC)(C1)c1nnnn12.OC 89109,C#Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCN2CCOC2=O)o1 89110,CN1CCOC(N(C(C(=O)NC(C)(C)C)C(C2CC2)C2CC2)C)C1 89111,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NCc2ccc(C)cc2)[nH]1 89112,c1(C(N2CC(CCNC(C3CCC3CF)=O)(OC)C2)=O)ccc(Cl)c(O)c1 89113,c1(C(=O)NC(CC)CN(C(=O)CCS(N)(=O)=O)C)ccc(S(N)(=O)=O)c(Cl)c1 89114,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89115,CC1c2nnc(CCSc3cn(CC(=O)O)nn3)n2CCN1C(=O)OC(C)(C)C 89116,c1(CC(=O)NCC(CNC(=O)C(CO)C2CC2)OC)ccc(CO)cc1 89117,Cc1ccc(C(CNC(c2nccnc2C)=O)NC(C2CCC(C)(C)C2)=O)cc1 89118,C(=O)(C#CC1CCCCO1)NC1C(C)(C)CCN(C(CCCCCC=C)=O)C1 89119,CC1(C)COCCC1C(N1CC2CC2(NC(c2csc(-c3cnc[nH]3)n2)=O)C1)=O 89120,c1(C(=O)NCC=CCNC(C2CC3CCC2C3)=O)c[nH]c2ccccc2c1=O 89121,c1(C(C(F)F)NC(CCn2cc(CCCOCC)nn2)=O)c(F)cccc1F 89122,C(=O)(C(F)CC(C)C)NC(CC)CNC(c1cc(SC(F)(F)F)c[nH]1)=O 89123,c1(NC(=O)NC2CNC=C(Br)C2)cc(C(F)(F)F)ccc1Br 89124,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89125,c1(C(=O)NCC2CCN(C(c3ccc(Cl)cn3)=O)CC2O)ccc2cc[nH]c2n1 89126,Cc1coc(OCCNC(=O)COC(=O)N(C2CC2)C)c1-c1ccccc1.C=O 89127,Cn1nc(-c2ccncc2)cc1C(=O)NCCNC(=O)CC1CCCN1C(N)=O 89128,Cc1c(C(=O)NCCCNC(=O)CCCOC2CCCCC2)cnn1CCC#N 89129,C1(C2CCCN(C(c3ccc(C)c(F)c3)=O)C2)(NC(C(C(COC)C)C)=O)CC1 89130,n1(C(C)C)cnnc1CC(=O)NC1(C(=O)O)CC1 89131,N1(CCNc2cn(C3CCCC(N)C3)nn2)CCC(C2CCC(F)(F)CC2)C1 89132,N1(C(c2ccno2)=O)CCN(C(C2CCC(O)C2)=O)C2CCCCC2C1 89133,N1(C(C=CCOC)=O)C2CCC(C(=O)NCCC3CCCCC3)C1CC2 89134,c1(OC)noc(C)c1C(=O)NC(CNC(=O)C(C)(C)COCC(F)F)C1CCC1 89135,c1(C(=O)OC)cc(N2CCOC(C(C)NC(c3ccoc3Br)=O)C2)nc(C)n1 89136,N1(CC)CCOCC1C(=O)OCc1cccc(CN2CCOCC2)c1 89137,N1(CC(=O)NCCN(C)C(c2snc(O)c2Cl)=O)CCC(c2ccccc2)CC1 89138,N1(Cc2cccc(C)n2)CCCC2CN(Cc3cccnc3)CCC12 89139,N1(CC=C)CCCN(C(=O)C#CCNC(=O)C(N)=O)CC1 89140,Cc1ccc2snc(C(=O)NC(C)(C)CNC(C3CCC4(C3)CC4(F)F)=O)c2c1 89141,CC1=C(c2ccccc2)CN(C(c2cccc(F)c2C)C(=O)NCC2CC2)CC1 89142,N1(C(C(CC)CC)=O)CC(NC(=O)CC2CC3CC3C2)C2(CCC2)C1 89143,N1(C(C(C)SCCCC)=O)CCC2(CC1)CCN(c1nc(Cl)ncc1F)CC2 89144,c1(CNC(N2CCCC(CC(=O)OCC)C2)=O)ccc(F)c(C)c1F 89145,C12(CNC(c3cc(C)ncn3)=O)CCC1CCN2C(=O)C=Cc1ccc(C)nc1 89146,Cc1nc(O)nc(O)c1CCC(N1CC(NC(=O)C(F)C(C)C)C(C)C1)=O 89147,C1(NC(C2(C=C)CCCC2)=O)CC2CC(NC(=O)C=COCC)CC12 89148,c12ncc(Cl)cc1C(=O)N2.Cc1nn(C)cc1CN1CCOC(CO)C1 89149,Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CCSc2ccccc2)cc1 89150,N1(C(CCCN(C(C)=O)C)=O)CCC2(CC2NC(c2cnn(C)c2N)=O)C1 89151,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCc1[nH]cnc1C 89152,C(=O)(C(F)(F)CF)NCCOC1CN(C(C(C)N(CC)CC)=O)C1 89153,c1(C(=O)NCCOC2CN(C(c3n(CC)cnn3)=O)C2)ccnc(C)c1Cl 89154,C(=O)(C1=C(C)OCCC1)N(CCNC(Cc1cccc(OC)n1)=O)C(C)C 89155,Cc1ccc(Br)cc1SC1N(C(CC(N2CCCC(C)(C)C2)=O)=O)CCC1O 89156,C(=O)(CCC(F)(F)C(F)F)NC1C(C(N2CCC(C(N)=O)CC2)=O)CC1 89157,CCCCC(CN=c1[nH]cnc2c(Br)cccc12)NC(c1ccc(=O)n(C)c1)=O 89158,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89159,C(=O)(C(C)(C)C(O)C(C)C)N(C)CC1CN(C(c2c(C)ncc(C)c2)=O)C1 89160,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89161,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CCO)C3)=O)ccn12 89162,C#Cc1ccc(Br)c(C(=O)NC(C)CN(C)C(C2(C)C=CCCC2)=O)c1 89163,C1(C(NOCCOC)=O)CN(C(=O)CCc2cn[nH]c2)CC12CC2 89164,c1(OCC(N2CC(NC(C(C)O)=O)CC3C2COC3)=O)c(F)c(F)cc(F)c1F 89165,N1(C(C(C)CN(C)C)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CCC1C 89166,c1(NC(=O)NCCCn2cnc(=N)[nH]2)ccc(N2CCOCC2)c(F)c1 89167,N1(C(CSc2n(C)nnn2)=O)CCC(C)(C)C(C(=O)NC2CC(F)(C(=O)OC)C2)C1 89168,c1(C(N2CCN(C(CC=C)=O)CC2CC2CC2)=O)cc2ccc(F)cc2cn1 89169,CCC(CC)(CCNC(=O)Cc1ccon1)NC(=O)C(Cc1ccccc1)SC 89170,C1(N(C(CC(C)c2ccccc2)=O)C)CN(C(c2ccc(O)nc2Cl)=O)CC12CC2 89171,c1(N(CCC(=O)OC)C)ccc(C2CC2c2nnc(C3CC3)n2CC2CC2)cc1 89172,C1(NC(c2c(CC)cco2)=O)(CNC(c2cnc(CC)s2)=O)CC(F)(F)C1 89173,CC(C(=O)N1CC(C(=O)NCC2C(C)C2C)C(F)(F)C1)C(C)(C)C 89174,N1(C(C2CC3(CCC3)C2)=O)CCC2CCN(C(C3CCCCS3(=O)=O)=O)C2C1 89175,c1(OC)cccc(C=CC(N2CC=CC2CNC(=O)C(F)C2CC2)=O)c1OC 89176,C1(NC(c2cc(C)c(C)nc2)=O)CCCN1NC(=O)N(C1CCC1O)C 89177,C(=O)(C(C)(C)c1cccs1)NCC(C)N(C(=O)CSCCN(C)C)CC 89178,C1(C(=O)NCCCCCCN(C(C=NOC)=O)C)CC12C1CC3CC(C1)CC2C3 89179,C1(CC)CN(C(c2cc(O)nc(OC)n2)=O)CCN1C(c1cccc(Cl)c1N)=O 89180,CCC(COC)C(=O)N1CCCC(NC(=O)C(=Cc2cn[nH]c2)C)C1 89181,C1(n2cc(-c3cn(CC)nc3)nn2)CN(c2ccncn2)CCC12CCC2 89182,C(=O)(C(O)CCC(C)C)NCC1C(NC(CC(COC(C)=O)(C)C)=O)C1 89183,c1(C(C)C)cccc(OCc2ncc(-c3nn[nH]n3)o2)c1 89184,c1(CC)ccccc1O.C1(C)(C)CCN(C)C(=O)CC2C(C2)C(=O)N1 89185,c1(N2CC(CNC(C3(C)CCNC3=O)=O)OCC2)cncc(C#N)n1 89186,c1(C(=O)NCC(C)N(C(C2CCCCC2C(N)=O)=O)CC)cc2ccccn2c1 89187,C1(C(C)CO)CCCCN1C(C1CCN(C(=O)C=C(C2CC2)C2CC2)CC1)=O 89188,N1(C(C2(C)CN(C(=O)CC3CCC(O)C3)C2)=O)CCOC(CC2CC2)C1 89189,c1(NC(C)=O)cccc(C(N2CC3(CC3)CC2CNC(=O)C(F)F)=O)c1C 89190,N1(Cc2cnn(Cc3cc(C)no3)c2C)CCCC(NC(=O)CS(N)(=O)=O)C(F)C1 89191,c1(C(=O)NC2C(NC(c3c(C)cccc3)=O)CC2)ccc(N)cc1C(F)(F)F 89192,N1(C(c2ccc(CC)[nH]2)=O)CCCC12CCC2.C12C=CCCC1C(=O)N2 89193,N1(C(C2CSCCN2C(c2cccs2)=O)=O)CCc2ncncc2C1 89194,C(CN=c1cccc(S(=O)(=O)NC(CO)CCC2CC2)[nH]1)c1ccc(C)cc1 89195,Cc1c(C(=O)NC2COCCN(C(c3csc(Cl)c3)=O)C2)c(C(F)(F)F)nn1C 89196,c1(C(N2CC(C)C(NC(c3c(Cl)nsc3Cl)=O)C2)=O)cc(O)cc(O)n1 89197,N1(CCC)C(=O)NC(c2csc(O)n2)C(C(=O)OC(C)(C)C)=C1CC1CC1 89198,C1(CN(C)C(C2CC(CC3CC3)C2)=O)CCCN(C(C2C3CC(=O)CC23)=O)C1 89199,C(=O)(C1CCCc2ncnn21)NC1(C)CN(C(c2ccc[nH]2)=O)C1 89200,C#CCC(C)(CC)C(=O)N1CC(NC(c2ccc(CC(C)C)cc2)=O)C(C)(C)C1 89201,C1(NC(COC2CN(C(C(OC)OC)=O)C2)=O)Cc2ccc(Br)cc2C1 89202,N1(C(C2CC(Cn3cncn3)C2)C(=O)NC(C)C)CCC(C2(C)CC2)C1 89203,Cc1c(C(C)NC(=O)NCCN(C2CCCO2)C)cnn1Cc1ccccc1 89204,C(C(C)N=c1ccc([N+](=O)[O-])c(O)[nH]1)NC(C(C)Cc1ccc(F)cc1)=O 89205,N1(C(C=Cc2n(C)ncc2)=O)CCC2(CCCN2C(=O)C(F)CC2CCC2)C1 89206,C(CN=c1[nH]c(CCSC)cs1)(c1ccccc1F)OCC 89207,O=C1CC(n2cc(CNC(=O)CSc3cccc(Cl)c3)cn2)C(=O)N1 89208,C1(C(=O)NCC(COC)O)CN(C(=O)C(=O)Nc2ccc(C)cc2)CCC1(F)F 89209,N1(C(C2CC3(C(C(=O)OC)C3)C2)=O)CCCC2(CCCNC2=O)C1 89210,c1(C(C)NCC(C)CF)ccc2nonc2c1 89211,c1(C(N(C2CCN(C(C3CC(O)C3)=O)C2)CCC)=O)cnn(C2CCCCC2)c1 89212,c1(C(=O)Nc2c(-c3ccc(C=C)cc3)cncn2)c(C)cc(OCC)cc1C 89213,CC(O)(C(=O)NC1CC2CCN(C(=O)Nc3ccc(F)c(F)c3)CC12)C(F)(F)F 89214,C1(C#N)(C(=O)NC2C(C)N(C(=O)CSc3cccnc3)CC2)CC12CCC2 89215,Cc1nnn(CC(=O)NCC2(O)CN(C(=O)CC(=O)OCCC(C)C)C2)n1 89216,c1(C(N(C)CC2CN(C(C3COC(=O)N3)=O)CCO2)=O)ccc2[nH]ccc2n1 89217,c1(C(=O)NCC2N(C(C(n3cc(C)cn3)OC)=O)C3C(C2)C3)cccc(Cl)c1F 89218,C#Cc1ccccc1CC(=O)NCCC1(CNC(C23CCC(CC2)O3)=O)CCCC1 89219,C(CCCCN(C(=O)CC(=O)NC1CC1)C)NC(C(C1CC1)OC)=O 89220,n1(CC)cc2ccc(C(=O)NC(C3CC(F)(F)C3)C)cc2n1 89221,N1(C(=O)OC(C)(C)C)CCCCC(NC(=O)N(C(COC)N)C2CC2)C1.C1CC1 89222,C(=O)(C1Cc2ccc(Cl)cc21)NCCCN(c1ncnc2c1CCC2)C 89223,C(=O)(C1=CCC(F)(F)CC1)N(C)CC1CC(NC(C2(C(=O)C3CC3)CC2)=O)C1 89224,C=CCC(F)(F)C(=O)N1CCC(CNC(=O)C(CCN(C)C)N(C)C)CC1 89225,c1(C(=O)NCCN(C)C=O)ccccn1.C1(n2ccnc2)(CCOC)CCCC1 89226,C1(OCCNC(C2CC(C(F)F)C2)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 89227,N1(CC(=O)Nc2nc(C(C)(C)C)[nH]c2Cl)CCN(C(=O)CCn2cncn2)CC1 89228,c1(C(N2CCCC(CC(=O)NC(C)CCc3cn[nH]c3)C2)=O)cncn(C)c1=O 89229,C(C)(CNC(=O)CC1CCSCC1)(CO)NC(C(C)=CC)=O 89230,C#Cc1cccc(C(N2CCC(O)(C(C)NC(=O)CC3CCCOCC3)C2)=O)c1 89231,Cn1cnnc1CCC(N1CC(CO)(NC(c2ccc(C3CC3)s2)=O)C1)=O 89232,c1(CN2C3CN(C(c4c(C)nc5sccn54)=O)C(C3)C2)cccc2nc(O)oc12 89233,C(=O)(C1=CCN(C(C2C(C)C2C)=O)C1)Nc1cn(CC#C)nc1 89234,N1(C(c2cc(C)cc(N)c2)=O)CCc2cccc(C(N3C4CCC3CC4)=O)c2C1 89235,N1(C(CS(=O)(=O)N(CC)CC)=O)CCCC2(CNC(=O)Cc3cnco3)CCCC12 89236,C1(CC2NC(=O)N(Cc3nc(C)c(CC(C)C)s3)C2=O)CC2(CCCC2)CO1 89237,c1(SCC)cnccc1C(N1CCCCC1CCCSCCOC)C(=O)NCC 89238,C(=O)(N=c1ccnc(C2CCC2)[nH]1)C1CC(=O)N(C)C1c1ccccc1 89239,C1(C(N2C(C(C)C)(C(=O)NCC3(O)CC(CO)C3)CCC2)=O)C2CCC(C2)C1C 89240,CC(Cc1ccnn1C)C(=O)NC(C)(C)C(C)NC(c1cc(F)c[nH]1)=O 89241,C=CC1(C(N2CC(OCCO)C2)=O)CCN(C(C2CCC2C#N)=O)C1 89242,Nc1cc(C(N2CCCC2(C)CNC(C2CCCC23CCC3)=O)=O)cnc1Cl 89243,Cc1cnn(C)c1CC(=O)NC(CC(F)(F)F)c1nccn1C 89244,c1(C(=O)Nc2c(NC(=O)NCCOC)c(C)cs2)cccc2c[nH]nc12 89245,CCCC(C(O)C(=O)NCC1CCC(F)C1)NC(c1cncn1C1CC1)=O 89246,N1(C(CC2C(C)OCC2)=O)CCC(NC(=O)Cn2cnnn2)C(C)(C)C1 89247,c1(OC)ccc(C(C)C(=O)OCCCCc2cccc(C(N)=O)c2)cc1 89248,c1(CCNC(CC(C)SC)c2nnnn2C2CCOCC2)n[nH]c2ccccc12 89249,C=C(C)c1ccnc(NC(=O)NC2C3CCC2(c2ccco2)C3)n1 89250,n1(CCC)cc(Cl)c(C(=O)NS(=O)(=O)CC)n1.C12COCC1NC(=O)CN2 89251,N1(C(COCC)=O)CCC2(CCC(NC(c3ccnc4ncnn34)=O)C2)C1 89252,c1(C(N2CC(C)C(NC(c3cc(N)c(Cl)cn3)=O)C2)=O)ccc(C2CC2)nc1O 89253,O=C1CCN(CCOC2CCN(c3ccc(Cl)cc3)C2)C(=O)N1c1cccc(Cl)c1 89254,c1(C(N2C(C(C)C)C(C(=O)NCC3CC(F)(F)C3)CC2)=O)ccc2c[nH]nc2c1 89255,C1(CC(N2CCC(CC(C)NC(=O)COCCN(C)C)CC2)=O)CCC(C)(C)CO1 89256,c1(CN(C)C(C2CCCCC2COC)=O)cccc(NC(=O)CCNC(N)=O)c1 89257,CN1C(=O)CSC1=CC(=O)N1CC2CC2(NC(=O)CCn2cnccc2=O)C1 89258,C1(C(N2CC(NC(c3c(Cl)cn(CCC)n3)=O)C2)=O)CC2CCCC(C1)C2 89259,c1(C(N2CCC(O)(C(C)NC(c3c(C)cc(C)o3)=O)C2)=O)c(C)ccc(C)c1O 89260,n1(C(C)C)cc(C(=O)NCC2(F)CN(C(c3ccc(F)s3)=O)C2)c(O)nc1=O 89261,c1(NC(C2CCN(C(c3c(OC)ccs3)=O)C2)C)nc(C)cc(C#N)n1 89262,c1(C(=O)NCCN(C(=O)C(C)(C)C2CCCO2)CC)cccc(S(C)(=O)=NC)c1 89263,C1(C#N)(C(=O)NCC(CNC(CC2(CC)CCC2)=O)(C)F)CC(=O)C1 89264,c1(CC)nc(C(C)C)ccc1C(N1CC(NC(=O)C(C)C2CC2)CC(F)C1)=O 89265,C1(CNC(c2cc(C)n(C3CC3)c2C)=O)CN(C(=O)C(N)=O)CCC12CCC2 89266,n1(CC)cc(S(=O)(=O)NS(=O)(=O)Cc2ccon2)cn1.c12ccn(n1)CC(=O)N2 89267,Cn1nc(C(=O)NC(CNC(c2cc(C(N)=O)cs2)=O)C(C)(C)C)cc1C(F)F 89268,N1(C(C=NOC)=O)CCC(C(N2CCC(F)(CF)C2)=O)C12CCC2 89269,C1(N(C(c2[nH]cc(C(C(C)C)=O)c2)=O)C)CCCN(C(=O)CC2CC=CCC2)C1 89270,C1(C(=O)NC(CCC)C(=O)N(C)C)CN(C(c2ccncc2NC)=O)CCN1C 89271,C=CC1CCCN(C(C23CC(CN2C(c2cc(C)co2)=O)C3)=O)C1 89272,C1(CNC(C2(F)C(C)OCC2)=O)CCCCN(C(=O)C=CCn2cncn2)C1 89273,N1(C(C2CCSCC2)C(=O)NC)CCC(C)CC1 89274,CCCCC(C(=O)NCC(C(N1C2CCCC1COC2)=O)C(C)C)C(C)C 89275,CCCC(C)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CN(C)CCC 89276,CC1C2C(CCN2C(=O)CCC2CCCN2C)CN1C(=O)C=CC1CC1 89277,c1(CN2CCC(CCC(=O)C(=O)CC3CNC(=O)O3)C2)c[nH]c2cccnc12 89278,N1(C(C(CCCC)O)=O)CC2(C1)CN(C(=O)C#CC(C)(C)C)CCO2 89279,CC(O)(CC(=O)N1CC2CC1CC2C(N1CCS(=O)(=O)CC1)=O)CC(=O)O 89280,c1(OC)ccc(C(N2CC(NC(=O)COc3cn[nH]c3)C3(CC3)C2)=O)cc1N 89281,Cc1cc(CNC(C2(C)CCCN2C(=O)CCCCCF)=O)cc(F)c1 89282,C1(CCC)(NC(=O)CC)CCCN(C(C2CCC(OC(F)F)CC2)=O)C1 89283,Cc1cc(Br)ccc1C(C)C(N1CCOC(CNC(=O)C2=C(Cl)CC2)C1)=O 89284,C(=O)(CCCC(=O)N(CC(C)NC(c1ccc(OC)c(Br)n1)=O)C)OC 89285,C1(C(=O)N(C)C)CCCN(C(=O)C(Cn2cncn2)NC(C(CC)SC)=O)C1 89286,c1(C(=O)NC(C2N(CC(=O)OCC3CC3)CC2)=O)ccc2[nH]nc(Cl)c2c1 89287,C(C(C(C)C)NC(=O)Cn1ccc(C(F)F)n1)(c1ccccc1)NC(C=C(C)C)=O 89288,c1(NC(CN2CCC(C(C(=O)OC)C)CC2)(C)C)c(OC)ccc(Br)c1F 89289,C1(C(=O)NC(C)CCNC(=O)C2=CCOC2)CC(C)(C)CCO1 89290,C12(CNC(c3cncc(C)n3)=O)CCC1CN(C(=O)CC1CNC(=O)C1)C2 89291,c1(C(=O)NCC(CNC(=O)C(C)S(C)(=O)=O)OC)cnc2ccc(C)cn12 89292,CCC(C(=O)NC1CN(C(c2nccn2C)=O)CCC1C)C(C)C 89293,C(C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NC(C)CC(=O)OC)C1(C)C)OCC 89294,O(NC(=O)C(C)N(C(=O)Cc1ccccn1)C1CC1)CC(CC)C 89295,c1(C(c2cccnc2)NC(C2CCN2C(C2(O)CC2)=O)=O)cccc(O)c1 89296,N1(C(c2ccc(N)c(N)n2)=O)CCC(NC(C2CCC2)=O)C2(CCC2)C1 89297,N1(C(CCCOC(C)C)=O)CCC(CNC(=O)C=Cc2cccc(O)c2)C(C)C1 89298,CC1(CNC(=O)CC2CCCO2)CC(F)(F)CN1C(c1cn2ccnc2cn1)=O 89299,CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NC(c1cc(F)ccc1C#N)=O 89300,N1(C(CCC2CCCC(=O)N2)=O)CC2CCC(C1)N2C(C1C(Cl)(Cl)C12CC2)=O 89301,CC1=C(C(=O)NCC2COCC2NC(=O)COc2cc(C)on2)CCO1 89302,CC(C)(C)CCC(=O)N1CC(C)(C)CC1CNC(=O)Cn1ccc(C2CC2)n1 89303,N1(C(C(CC)c2ccccc2)=O)CCCN(C(C23CCC(C2)OC3)=O)CC1 89304,N1(C(CCCOC(C)=O)=O)Cc2ccccc2C(NC(=O)COC2CCCOC2)C1 89305,N1(c2ccnc(N(CC)CC3CC4(C3)OCCO4)n2)CCc2c(C)cccc21 89306,N1(C(C2CCCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CCC(C)C(C)(C)C1 89307,c1(OC)ncc(C)cc1-c1ccc(C(=O)Nc2cnnc(C)c2)nn1 89308,CN1CCC(C(=O)NCC=CCNC(=O)CCC(=O)c2ccccc2)CC1=O 89309,c1(C(=O)NC2CC(F)(CNC(C3(C)CC3F)=O)C2)ncn2cccnc12 89310,N1(C(c2cn(CCNC(C(C)(C)CCF)=O)nn2)=O)CC2(CCC2)CC1CO 89311,N1(C(CN(CCOC)C)=O)CC(C)(C(N2CC(F)CC2CO)=O)CC1(C)C 89312,Cc1cncc(C(N2CC(C(C)NC(=O)C(C3CC3)C3CC3)C2)=O)n1 89313,CC1CC2(CO1)CN(C(=O)C(=O)NCc1cncc(-n3cncn3)c1)C2 89314,CCC(CC)=CC(=O)NCC(N)=O.C12(CCC1)CC(=O)N2 89315,C#CC1CCCC(CNC(=O)CC2CN(C(=O)COCC(C)C)C(C)(C)C2)C1 89316,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(NC(c2cnc(OC)s2)=O)CC1 89317,C(CCC(C)(C)C(=O)NOCCC(C)C)NC(CCCC(C(C)C)O)=O 89318,C1(CNC2N(C(=O)O)CCN(C(C)(C)C)C2)C2CCC3C(C2)CC13 89319,Cc1nc(Cl)ncc1CCC1N(C(=O)C(=O)NC(C2CCC(=O)N2C)=O)CCCC1C 89320,N(C1CC2CCC(=O)NC12)S(c1ccc(NC(c2cscn2)C)nc1)(=O)=O 89321,C1(NC(C2(SC)CC2)=O)CC2(CCN(C(C3CCCC34OCCO4)=O)C2)C1 89322,c1(C(=O)NC2CCN(C(C3CCC(=C)CC3)=O)C(C)C2)cnc2ccccc2c1 89323,c1(CNC23CC(C(=O)Nc4c(C)noc4)(C2)C3)cc(C)ccc1O 89324,C1(NC(c2cc(C(=O)OC)sc2)=O)CCCCC1NC(c1n[nH]cc1F)=O 89325,c1(C(=O)NCCCCNC(C2(C3CC3)CCC2)=O)cnc2cc[nH]c2c1 89326,c1(SC)nc(N2CCC(CNS(=O)(=O)c3cccs3)C(F)C2)cc(C)n1 89327,Cc1nscc1CC(N1CC(NC(c2cn(C3CCOCC3)cn2)=O)C1)=O 89328,Cn1ncc2c(N)c(C(N3CC(NC(=O)C=C4CC4)C(F)C3)=O)cnc12 89329,c1(COC)nc(=NC(C)CN(C)C(c2ccc(NC(C)=O)cc2C)=O)s[nH]1 89330,c1(OC)cc(N)ccc1C(N1CC(CCO)(NC(=O)C(C2CC2)OC)C1)=O 89331,C1(CC)CN(C(C2CC(=O)NC2(C)C)=O)CCC1NC(=O)CC1CC2(CCC2)C1 89332,C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)COC(F)(F)F)C(F)C1)NC 89333,c1(C(C)C)ccc(C(N2CCCC2CNC(C2C3(CC3)C23CC3)=O)=O)cn1 89334,c1(-n2c(C(C)CCC(F)F)nc(CC(C)OC)n2)cccc2nc[nH]c12 89335,CC1(CNC(c2ccc(N)cc2Cl)=O)CCN(C(C2(C)CCCO2)=O)CC1 89336,C(=O)(CCCC(C)C)OCC(=O)N(C1CCN(CC(C)C)CC1)CC 89337,c1(C(N2CC(CNC(c3c[nH]cc3Br)=O)OCCC2)=O)cc2n(n1)CCCC2O 89338,CC1CN(C(=O)Cc2cnns2)CC(C)C1NC(=O)CCc1ccncc1 89339,c1(C(=O)NCC(C)N(C(C(C(C)C)NC(=O)OC)=O)C)cc(Cl)cc(Cl)c1 89340,c1(NS(=O)(=O)Cc2cccc(Cl)c2)cnncc1Br 89341,C#CCC(O)C(=O)N1CC(C)(C(=O)N(C)Cc2cc(=O)cc[nH]2)C1 89342,C1(CCNC(c2ccc(C)nc2)=O)CN(C(=O)Cc2occc2C)CCS1(=O)=O 89343,Cc1ncc2n1CCN(C(=O)CC1CCCN(C(=O)CN(C)C(N)=O)C1)C2 89344,Cn1ncc(C(N2CCC(CCF)CC2)C(=O)N(C2CCC2)C2CCC2)c1Br 89345,C1(C(N(CC(F)F)CCC)=O)CCCC2(CCC2)O1 89346,N1(C(=O)CCc2ccc[nH]2)CCC2CC(C(N3C4CCC3CC4)=O)C2C1 89347,C1(C(=O)NCC2CCC(NC(c3c(C)nns3)=O)C2)CC(c2ccncc2)=NO1 89348,c1(C(N2C3CC(NC(C4N(C)CC=C4)=O)C2CC3)=O)cc(Cl)c2[nH]c(O)nc2c1 89349,c1(OC)ncc(CN2CCCC(NC(=O)CNS(C)(=O)=O)CC2)cc1Br 89350,C1(C(=O)NCCCCC2CN(C(=O)CNc3ccccc3)C2)CC1C1CCCC1 89351,Cc1cc(C(=O)NC2(C)CCCN(C(C3CC(CCF)C3)=O)C2)cc(F)c1C 89352,C(=O)(CC(C)CC(C)C)N1CC(C(C(=O)NC(CCC)(C)C)OC)C1 89353,c1(C(=O)NCCN(C2CCCCC2)C(COC(C)C)=O)cccnc1N 89354,CC1CC(NC(C2CSCC(=O)N2)=O)CN(C(=O)CNc2cnn(C)c2)C1 89355,c1(CN(CC)CC)ccc(F)c(CC)c1-c1nc(-c2ccc(=O)n(CC)c2)no1 89356,C#CC1(C(=O)NC2(C(N)=O)CC2)CN(C(c2coc(C3CC3)n2)=O)C1 89357,c1(C(C)C)ccc(CNC(=O)NCC(N2CCCCC2=O)C)cc1Cl 89358,C1(N(C(=O)Cn2ccnn2)CCOC)CCN(C(=O)C(F)C2CCCC2)CC1 89359,C1(C)(CNC(=O)NC2C(c3ccc(C)cc3)OCCC2)CCCS1(=O)=O 89360,C(=O)(CCCCCN(C(=O)CCc1ccco1)C)NCC(CC(C)C)O 89361,c1(C(=O)NCC2CCN(C(C3ON=C(CC)C3)=O)C2)c(Cl)ccc2c[nH]nc12 89362,c1(C(=O)NCCOC2CN(C(=O)C3=C(Cl)CC3)C2)cc2n(n1)CCO2 89363,C1(CNC(C(N)=O)=O)(NC(c2ccc(O)cn2)=O)CCC(F)(F)CC1 89364,c1(CC(=O)NCCCCNC(C2CCN(C(CC)=O)C2)=O)nc(C)c(C)[nH]1 89365,c1(C(=O)NCC2CCN(C(Cc3ncc(C)[nH]3)=O)C2)cn2ccn(C)c(=O)c2n1 89366,N1(C(CNC(N)=O)=O)CCCC2CCN(C(c3cn4c(n3)CCC4)=O)CC12 89367,C1(CC(=O)OC)CCCC2(CN(C(c3c[nH]c(-c4ccc(Cl)cc4)c3)=O)C2)O1 89368,Cc1cc(F)c2cc(C(=O)N(C(C)CNC(C3CC(C)(F)C3)=O)C)[nH]c2c1 89369,C(CN=c1cc[nH]c(C(F)F)n1)(c1ccc(F)cc1)NC(C)=O 89370,c1(C(=O)NCCNC(CCC2N(C)CCCC2)=O)ccc(Br)c(N)n1 89371,c1(C(=O)NCC2CN(C(COCc3n(C)ncc3)=O)C2)ncn2c1CCCCC2 89372,C1(NC(c2c(COC)ncs2)=O)(CO)CCN(C(C2CCCC2)=O)C1 89373,CCCCC(O)C(=O)N1CCOC(C(=O)Nc2cc(I)ccc2Br)C1 89374,C(C(C(C)C)NC(c1cocn1)=O)(c1ccccc1)NC(C1(C)CC(=C)C1)=O 89375,C=CCC(C)(C)CC(=O)N1CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 89376,c1(NC(=O)C(C2CCN(C(=O)Cn3nnc(C4CC4)n3)C2)F)cccc(F)c1 89377,CCCCCC(O)CC(=O)NCC1CC1CNC(c1ccc(Cl)cc1O)=O 89378,CCC(C)CC(C(=O)NCC(C)(O)C(C)C)NC(=O)CCOC1CC1 89379,Cc1cnc(C(=O)NC(CNC(C2COC(=O)O2)=O)C2(c3ccccc3)CC2)nc1 89380,N1(C(C2CC(F)(F)C2)=O)CCCC(C2(NC(C3(c4cc[nH]n4)CC3)=O)CC2)C1 89381,C1(C(=O)NCCCC(=O)OCC)CCN(C(=O)c2c[nH]c(=N)c(C)c2)O1 89382,c1(C(=O)NCc2n(C)ccc2)nc2ccc(O)cc2[nH]1 89383,C1(CNC(c2[nH]cc(CC)c2)=O)CC2CCC(C1)N2c1nnc(CC)o1 89384,c1(C(=O)NCC(CC(C)C)NC(=O)CCc2cnco2)cn2c(n1)CCC2 89385,C1(NCC(=O)Nc2cncnc2)CC2CN(C(=O)Cc3ccnnc3O)CC12 89386,N1(C(COC)=O)CCC2(CC1)CC(NC(C13COCC1C3(F)F)=O)C2 89387,c1(C(=O)OCC)cnc(OC)nc1C.C1(=O)C(C)(C)CN(C)C2CCN1C2 89388,C1(O)(CC#C)CC(C(=O)NCC2CCN(C(c3occc3C3CC3)=O)C2)C1 89389,C1(NC(CCC(=C)C)=O)C(C)CN(C(=O)CCc2cccc([N+](=O)[O-])c2)CC1C 89390,c1(C(=O)NCCCCCN(C(Cc2cnc(C)s2)=O)C)c(C)ccn2ccnc12 89391,N1(C(C(C)NS(C)(=O)=O)=O)CCC(C(C)N(C(=O)Cn2cc(C3CC3)cn2)C2CC2)C1 89392,Cc1nc(C(=O)NC2CN(C(c3ccc(Cl)cn3)=O)CCC2C)c2ccccn12 89393,CCCCCCC(C)CC(=O)NCCN(C(C1CCC2CC2CC1)=O)CC1CC1 89394,C(C(F)(F)C(F)(F)F)OCCC(N1CC(CNC(=O)CCc2cnco2)C1)=O 89395,C=CCC(CC)C(=O)N(C1(C(=O)Nc2c(C)cccc2O)CC1)C 89396,c1(C(=O)NC(C2CN(C(C(C=C=C)C)=O)C2)C)cccc2nc(O)oc12 89397,C1(C(N2CCOC(C(=O)NC3C4CCCC34)C2)=O)(CC)CCCCO1 89398,C1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)CC2C=CC1CCC2 89399,Cc1ccc(C2CCN(C(=O)Nc3ccccc3C(N(C)C)C3CC3)C2)c(C)c1 89400,c1(C(=O)NCC(C2CC2)NC(Cc2cnc(C)[nH]2)=O)ncc([N+](=O)[O-])cc1Br 89401,C1(=O)CC(CC)C(=O)C(CCOC(C)(C)C)C(C)N1CCNC(CCC#CC)=O 89402,N1(C(C(C)=C(CC)C)=O)CC2OCC(NC(c3ccc(Cl)c(OC)c3)=O)C2C1 89403,O=C1CN2C(=O)CCCC1=CC=CC=C2N(C1CC1)Cc1ccc(Cl)c(Cl)c1 89404,n1(CC#C)cc(CNC(=O)C(CC2CCCC2)NC(C2CCOC2C)=O)cn1 89405,c1(C(C2CCCC2)NC(=O)Nc2ccccn2)ccc(Br)c(F)n1 89406,c1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)cccc(N2CCCC2)n1 89407,c1(OC)ccc(N(C(=O)C(CC(C)C)N2CCCC2=O)CC(C)C)c(OC)c1 89408,c1(C(=O)NCC(N2CCCN(C(c3cccs3)=O)CC2)=O)cc2cccnc2o1 89409,C1(N(C)C(C2CC(n3ccnc3)C2)=O)CCCN(C(=O)Cc2ccc(Cl)s2)C1 89410,C1(CCNC(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(=O)CCCC#N)CC1 89411,C(C(C)(C)CN(C)C(=O)NC1CC1C#N)NC(C1C(OC(C)=O)C1)=O 89412,C1(NC(=O)CCCc2cn[nH]c2)CC(F)CN(C(=O)CSc2ccccc2)C1 89413,c1(C(=O)NCCC(C)N(C)C(c2cc(CO)ccn2)=O)cncc(Cl)c1 89414,Cc1cc(CC(=O)NCC(C)(CO)NC(C2(C(F)(F)F)CCCC2)=O)ccc1O 89415,c1(C(=O)NC2CC(N(C(C3C(C(C)C)CCC3)=O)C)C2)cnn(C)c1Br 89416,c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CC(NC(C1C=CCS1)=O)C2 89417,C#CC1(NC(N2CC(CCCCCC)C2)=O)CCN(C(=O)C(=C)CC)CC1 89418,n12cccc1C1(CC1)CN2.c1csc(-c2cnco2)c1 89419,c1(C(CNC(=O)C=C2CCC2)NC(C2(C)CC2(F)Cl)=O)c[nH]c2ccccc12 89420,C(=O)(C(C)(C)CCCNC(N)=O)Nc1cc(OCC)cc(F)c1 89421,c1(C(N2CC3C(C(=O)NC4(C)CC(C)(C)C4)(C3)C2)=O)ccnc2[nH]cnc12 89422,c1(C(C(=O)N(C)CCNC(C2(C)CC2(F)F)=O)(F)F)nc2ccccc2[nH]1 89423,Cn1ccc2sc(C(=O)NC3CC(NC(=O)CSC(F)F)C34CCC4)cc12 89424,N1(C(c2ns[nH]c2=O)=O)CC2(CCN2C(=O)CC2CCC(O)C2)C1 89425,CCCCCCC(CC)NC(C1(OC)CCN(C(=O)CCCNC(N)=O)C1)=O 89426,C(=O)(CCCNC(=O)C1CC1)N(CCC(C)N(C(=O)C(F)=C1CCCC1)C)CCO 89427,C1(C(N2CCC(O)(CNC(c3n(C(C)C)cnc3)=O)C2)=O)COC2CCCCC12 89428,N1(C(C2(C)CCC(C)CC2)=O)CCCC2CN(C(C3CC(=O)C3)=O)CC12 89429,c1(N2CCC3CCN(C)C3C2)nc2c(c(=NCN(C3CC3)C3CC3)[nH]1)CCC2 89430,C(=O)(C1=CC2C=CC1C2)NC(C)C=CC(N1CCN(C)CC1C)=O 89431,C1(C(CNC(C2(CCCC)CCC2)=O)O)CCN(C(C2(OC)CC2)=O)CC1 89432,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)O)C1 89433,c1(CC)nc(C#N)cc(=NCC2C(C)CCCN2C(c2cnnc(Cl)c2)=O)[nH]1 89434,C12CCCN(C1)C2=O.c1(C(=O)NCCOc2cnsc2)nc(C(F)(F)F)cs1 89435,N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 89436,N1(C(=O)NC2CC(CS(C)(=O)=O)C2)CC(O)(Cc2cnccn2)C1 89437,n1(CCOC)ccc(C(N2CCC(NC(=O)C(O)C3CCCC3)C2C)=O)c1C 89438,Cc1cc(C(N2CCC(N(C(=O)C(n3ccnc3C)C)CCO)C2)=O)c(C)o1 89439,CCCCC(CC)CC(=O)NCCCOCCNC(=O)C=Cc1cscn1 89440,c1(OC(C)C)c(F)cccc1C(=O)NCC1CC(CNC(c2cc(F)n[nH]2)=O)C1 89441,C12(CNC(CCC(=C)C)=O)CCC1CN(C(c1cccnc1C)=O)C2 89442,CCCCCCCC(=O)NC1CC(NC(=O)C(C)(C)C2CCCO2)CC1O 89443,CC1CC(=O)NC1C(=O)N(CCCN(C(=O)CC1CCC(C)CC1)C)C 89444,CC(C)C(O)C(C)C(=O)N1CCC(N(C(=O)CCC2(O)CCC2)C)CC1 89445,N1(C(=O)COC2CC(F)(F)C2)CCC2(CCCN(C(C3COC3)=O)C2)CC1 89446,C1(C)(CNC(C2(CCN(C)C)CC2)=O)CN(C(=O)CC2CCCO2)CCO1 89447,c1(CC(N2C(CNC(Cc3c(C)n[nH]c3C)=O)COCC2)=O)ccc(C#N)cc1 89448,CN1CC=C(CC(=O)N2CC3(CCC3NC(c3csc(Cl)c3)=O)C2)CC1 89449,N1(C(C(C(C)C)C)=O)CC2CCC1C1CN(C(c3csc(C4CC4)n3)=O)CC21.CO 89450,N1(C(c2c(CC)con2)=O)CCC2(CC(NC(=O)CS(=O)(=O)CCOC)CO2)C1 89451,n1(CC)cc(C(=O)NC2CC2NC(=O)CC2CC(SC)C2)c(C)n1 89452,C1(NC(c2c(OC)n[nH]c2)=O)CC2CN(C(C34CC(F)(C3)C4)=O)CCN2C1=O 89453,C(C(=O)N(C)Cc1c(C(N2CCCC(CSCC)C2)=O)nco1)(C(C)C)SC 89454,N1(C(CC2CCN(C)C2=O)=O)CCC(NC(c2cc(C3CC3)no2)=O)C(CO)C1 89455,C1(CC)(CC)CC(NC(=O)C(C)C(C)C)CN1C(c1cccc(OC)c1OC)=O 89456,C=CC1(CC(=O)NC(C)(CNC(=O)Cc2cncs2)C2CC2)CC1 89457,N#CC1(C(N2CCN(C(c3ccc(F)s3)=O)C(CC(F)(F)F)C2)=O)CCOCC1 89458,c1(NC(C(CNC(C(CC)(C)CO)=O)OC)=O)ccc2c(c1)OCO2 89459,C(=O)(C1=COCCC1)NC(C)CCNC(=O)CC1CC(O)C1(C)C 89460,c1(SCC(=O)NC(CNC(C2CC3C=CC2O3)=O)CO)ccc2ccccc2c1 89461,C1(CNC(C(=O)N(CC=C(C)C)C2CC2)=O)CC(CO)CO1 89462,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 89463,c1(OC)cnccc1C(=O)NCCc1n[nH]cc1C(=O)NCC(C)(O)CCO 89464,c1(C(N2C(C)CC(NC(c3ccc(=N)[nH]n3)=O)CC2)=O)noc2ccc(Cl)cc12 89465,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(CNC(=O)CSCC(F)(F)F)C1 89466,C12CNCCN1C2.c1ccc(O)cc1.C(CCC)N(C)CC 89467,CC1CC(CNC(=O)CCc2cnoc2)CN(C(C2C3COCC23)=O)C1 89468,N1(C(CCSCC(=O)NC)=O)CC(N(C(=O)CC2CC=CCC2)C)C2(CC2)C1 89469,C1(C(N(CCNC(c2cn(C)cn2)=O)CC)=O)CCn2c(O)nnc2C1 89470,C1(NC(c2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 89471,CC(F)(F)CC(=O)NC(c1ccccc1OC)CNC(C1CSC1)=O 89472,C1(C#CC(=O)N2CCC(NC(c3cn(CC4CC4)nn3)=O)C(O)C2)(CC)CC1 89473,c1(NCC2N(C(CC(CC)C3(C(=O)NC)CC3)=O)CC2)c(Br)c(C)nn1CC#N 89474,C1(CC)CCC(NC(C2CN(C(=O)CC3CCSC3)CC2F)=O)CC1 89475,C#CCC(C)(C(=O)N(C)CCOC1CC1)NC(c1cc(C(F)F)[nH]n1)=O 89476,N1(C(C(C)OC(C)C)=O)CCCC(C2(NC(c3ccc(C(C)C)s3)=O)CC2)C1 89477,S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)N1CC(CC)C(O)C1 89478,c1(C(N2CCC(N(C(CC=C=C)=O)CC3CC3)CC2)=O)cc(C)ncc1C 89479,c1(C(N2CC(COC)(CNC(C3(F)CCOC3C)=O)C2)=O)c(C)ccoc1=N 89480,N1(C(C(c2ccccc2)N)=O)CC(C(=O)NCc2cc(F)cc(Cl)c2)CC(F)C1 89481,CCC(C(=O)N(C)CCC1CCN(C(c2snc(O)c2Cl)=O)CC1)C(C)C 89482,c1(OCCC(=O)NCCC2CCCN2CC2CCCC2)ccccc1Cl 89483,N1(C(c2c(C)nc(CO)s2)=O)CCC2CN(C(=O)Cn3cc(CO)nn3)CCC12 89484,CC1Cn2[nH]c(=NC(=O)NCC3CCC(F)CC3)cc2CO1 89485,c1(CN(C(C)CO)CCC)cccc(-c2ccccc2)c1O.C12CC(C1)C(=O)N2 89486,N1(C(C(CC(=O)OC)(C)C)=O)C2CCC1CC(C(=O)NCc1nnc(O)o1)C2 89487,N1(C(C(c2ccnn2C)C)=O)C2CCC(C2)C1CC(=O)NCC1(F)CCOC1 89488,C(C(C(=O)NC1CC1)N1CCCC(c2ncc(Br)cn2)C1)(c1ccccc1)OC 89489,N1(C(C(c2ccccc2)OCC)=O)CCN(C(C2CC(CC3CC3)C2)=O)CC1 89490,C1(NC(c2c(CC)oc(C)c2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1cc[nH]c1 89491,N1(C(=O)NCc2[nH]cc(C)c2)CCC(C)(C(c2ccccc2)=O)C1 89492,C1(CC(=O)NCc2c(C)nsc2)CC2(C1)CN(C(C1CCCN1C)=O)C2 89493,c1(C(N2CCC(C)(NC(C3CCC(SC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 89494,C1(C(=O)NCCN(C(c2ncc(C(=O)OC)cc2N)=O)CC)Cc2ccccc2N1 89495,c1(C(N2CC(C#N)C(NC(c3ccccc3F)=O)C2)=O)ccc(F)c2ccoc12 89496,C(=O)(C(O)CCCNC(=O)Cn1[nH]cnc1=N)N1CC(C#C)(N(C)C)C1 89497,Cc1cscc1C(=O)NCCC1CCCN1C(c1sccc1F)=O 89498,C1(NC(CC(C)c2ccncc2)=O)CN(C(=O)CSc2nncs2)CC1C 89499,N1(C(COCC)=O)CCN(C(=O)C(O)CC(N)=O)C(C(C)C)C1 89500,c1(C(N2C(=O)CC(COC(CC(C)(C)O)=O)C2)=O)cc(C#N)c(O)nc1N 89501,c1(C(CC)C)ccc(=NCCCOCCc2ccccc2)[nH]n1 89502,C(=O)(CCCCCCNC(=O)C(c1cccn1C)=O)N(C1CC2CCC(C1)N2)C 89503,CN1CCN(C(=O)C(C2(O)CN(C(C3(n4nccn4)CC3)=O)C2)F)C(CO)C1 89504,Cc1cn2cc(C(=O)OCc3ccn4ccnc4c3)nc2s1.C1C(=O)O1.C1CO1 89505,N1(C(Cc2cccc(OC)c2)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 89506,c1(C(=O)OC)nc(NC(C2CSCCN2C(c2cncnc2)=O)=O)cnc1C 89507,N1(C(c2c(C)noc2)=O)CCCC(C(C)(C)O)C1.N12CC=CC1C2=O 89508,c1(OC)nn(C)cc1C(=O)NCCNC(=O)C=C(Cl)Cl 89509,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 89510,C1(C)(CNC(C(C2CC(CF)C2)N(CC)CC2CCOCC2)=O)CCCCCC1 89511,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C(C#C)C1CCC1)C 89512,c1(NC(C)CNC(=O)C(c2cccc(Cl)c2)O)c(F)cccc1[N+](=O)[O-] 89513,Cc1ccc(C(=O)NCC(O)CC(=O)NCc2nn(C)cc2CO)n1C 89514,N1(S(CC)(=O)=O)CCCC(C(N2CC3CC3(NC(=O)CCCCC3CC3)C2)=O)C1 89515,c1(CC(=O)NC2COCC2NC(=O)CN2CC3CC3C2)csc2c(Cl)cccc12 89516,c1(N(C)C)ccc(-c2ccc(Cl)cc2C(N2CCC(F)(CC#N)CC2)=O)cc1F 89517,C(=O)(C1=NOC(C)(C)C1)N1C(C(N(C)C)=O)CC(O)C1 89518,C1(NC(C(CCSC)NC(C(CC#C)O)=O)=O)CCc2n[nH]cc2C1 89519,N1(C(CC2C3CN(C(c4c(COC)ccs4)=O)CC32)=O)CC=CC12CCCCC2 89520,C#CC1CCCCN1C(=O)CC1(NC(=O)C(=O)CC(C)C)CC1 89521,c1(C(=O)NCCC2(C)CCN(C(COCCC=C)=O)C2)cccc2c1OC(C)C2 89522,C(=O)(CCCC(N)=O)N(C)CC1N(C(c2cnc(SC)s2)=O)CCC1 89523,N1(C(CCNC(=O)Nc2ccco2)=O)C(CNC(c2ccoc2)=O)CC2CC12 89524,c1(C(N2C(C(N3CCC(=C)CC3)=O)(CC)CCC2)=O)cnc(O)cc1C 89525,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)C(C)O)nc(C)c(C2CCCC2)c(C)n1 89526,c1(C(=O)NCCOCCNC(c2c(OC)scn2)=O)cccc(N)c1C 89527,N1(C(CSc2cccc(C)c2)=O)CCCC(N(C)C(c2sccc2F)=O)CC1 89528,C=CCCC(C(=O)NCC1CC2(CC2)CO1)NC(C1CN(C)C1)=O 89529,c1(CC(=O)N(CC(CNC(CC2(OC)CC2)=O)C)C)cccc(Cl)c1 89530,C1(CNC(C(=O)N(c2c(C)ccc(F)c2)C)=O)CCC2(CCCOC2)O1 89531,c1(C(=O)NC(C)CCCNC(C2CCCSC2)=O)cnc2c[nH]nc2c1 89532,N1(C(C(C(C)C)OC)=O)CCC(CNC(=O)CCc2ncccc2C)C12CCC2 89533,C(C)(C(C)(C)C(=O)N(C1CC2CCC2C1)C)NC(C(C)=C1CCC1)=O 89534,Cc1cc2ccc1NC(=O)C(=O)N2.C1(C(=O)NC2CC2)CC(=O)N(CC2CCC2)C1 89535,N1(C(c2cnc(Cl)s2)C(=O)NCCCC(=O)OCC)CCN(CCO)C(C)C1 89536,CC(CCN=C(NC1CC1)NC1CCN(c2ccccn2)CC1)C(F)F 89537,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(C1OCC1(C)C)=O)CC2 89538,N1(C(c2c(CCCNC(C3CCN3C3CCCC3)=O)n[nH]c2)=O)CC2CCC1C2 89539,N1(C(c2ccn(CC)n2)=O)CC(CNC(=O)CC2CCCSC2)CC12CCC2 89540,c1(C2CN(C(=O)NCc3c(N)cc(F)cc3F)C2)cc2ccccc2cc1O 89541,CC(C)C(C(C)NC(=O)CCn1cncn1)NC(=O)Cc1ccc(O)cc1 89542,C1(CNC(c2c(C)nccc2)=O)CCCCCN1C(c1coc(C(N)=O)c1)=O 89543,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 89544,CN1CCC(O)C(NC(C2CCC(NC(c3cnn4c3OCC4)=O)CC2)=O)C1 89545,c1(C(N(CCNC(C(C)n2ccnc2)=O)C2CC2)=O)cc(N)c(Cl)c(O)n1 89546,C1(C(=O)NCCN(C(=O)C(O)CC(F)F)C)CC12CCCCCC2 89547,CN1CC(C(=O)NC(C)(C)C(=O)N(C)CCOC(N)=O)CCC1=O 89548,C1(C)(NC(c2c(C)scc2)=O)CCN(C(C2CCC(=O)N(C3CC3)C2)=O)CC1 89549,c1(-c2scc(Nc3nc(C)cc(OC)n3)n2)cc(F)c(Cl)cc1Cl 89550,N1(C(Cc2ccnc(OC)n2)=O)CCN(Cc2ccccc2)C(CCO)C1 89551,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 89552,C1(CNC(=O)CC2CCOC2)COCCN(C(=O)CCOCC2CC2)C1 89553,C1(CCC)CCCCN1S(=O)(=O)N1CCCCC1CC(c1ccccc1)O 89554,c1(C(=O)NC2CCC2NC(C2CC3CCC2C3)=O)cc2c(F)ccc(F)c2[nH]1 89555,CC1(C)CN(C=O)C1C1CCN(C(C2CCOCC2)=O)CC1.C1(N)CCS(=O)(=O)C1 89556,c1(C(=O)NC(CCNC(C(CCC)C)=O)(C)C)cc([N+](=O)[O-])c[nH]1 89557,S(=O)(=O)(c1cc2c(Br)cccc2s1)C(C1CCCC(CC)N1)=O 89558,CC(C)(CS(C)(=O)=O)C(=O)NCC(C1CCC1)NC(c1cnc(N)c(O)c1)=O 89559,Cc1nc(C(=O)NCC(C2CCCCC2)Nc2ncc(I)cn2)c(C)n1C 89560,Cc1cccc(C(O)CNC(c2cc(C#N)no2)c2ccccc2)c1 89561,Cc1cc(=NCCC(C)(O)c2ccccc2)[nH]cc1S(=O)(=O)NCC1CC(F)C1 89562,c1(CN2CC(CC(=O)NOCCF)C2)cccc(Cl)c1 89563,c1(OC)ccc(-c2nccn2-c2ccccc2)cc1C(C)Nc1cnn(C)c1 89564,C=CCC(CC(F)F)NC(=O)COC1CCN(C(C2(O)CCCC2)=O)C1 89565,Cc1ccn2ncc(C(N3CCC4CC3CN4C(c3ccc(Cl)cc3)=O)=O)c2c1 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89656,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 89657,C#CC1CC2(CC2)CN1C(=O)C(C)N(C(c1cc(C(C)=O)c[nH]1)=O)CC 89658,C1(NCCCCCC(CO)NC(=O)OC(C)(C)C)CS(=O)(=O)CC12CC2 89659,c1(C(=O)NCC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(Cl)nnc1Cl 89660,c1(C(=O)NC2CCC(NC(c3ccn(C4CC4(F)F)n3)=O)C2)ccccc1Br 89661,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCc2csc(C)n2)C1 89662,C(C(C)(COC)C(=O)NCCOCCN(C(c1cc(Cl)n[nH]1)=O)CCOC)OC 89663,C=CC(CCC)CC(=O)N1CC(N(C)C(c2ccc(F)cc2F)=O)C(O)C1 89664,c1(C(=O)NCC(CNC(C2C(CC)CC2)=O)O)nccc(C)c1N 89665,c1(C(N2CCCC(NC(c3ccc(F)cc3)=O)C2)C(=O)NC)ccc(Br)cc1F 89666,N12CC(C3(CC3)C1)C(=O)N(CC(C)O)C(=O)C2=O.CC(C(C)C)=C1CCC1 89667,c12ccc(C)c(c1)C(=O)N2.C1(OC)CC(CCSC)N(C(C2CC3CC3C2)=O)C1 89668,C=C(C)CCC(C)NC(=O)CC1CN(C(=O)CN2CCSCC2)CCO1 89669,c1(NC(CCC(n2cc(Br)cn2)CC)=O)cc(NC2CC3CCC2C3)ncn1 89670,CC(CS(C)=O)C(=O)NCC(C1CCCC1)NC(c1cc(CCO)on1)=O 89671,c1c(F)cc(I)cc1F.Cc1ccc(C(C2CCN(C(=O)C(=O)N)C2)C)cc1 89672,c1(NC(c2cccc(OC)c2)C)nc(Cl)c(C)cc1C1CCCCC1 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89691,Cc1c(C(=O)NC(C)C(C)NC(c2ccc(Br)o2)=O)cncc1N 89692,N1(C(c2cc(C)n(C(C)C)c2)=O)CCC(C)C(NC(=O)CCCCC#N)C1 89693,C1(C(N(CCN(C(=O)C(F)(F)c2ncccn2)CC)CC)=O)CCCC(C)C1 89694,C(CCCCOC(=O)CN1CCCC1=O)NC(=O)OCC1(SC)CCC1 89695,C1(CNC(c2c(C)cncc2)=O)N(C(c2nc(Br)c[nH]2)=O)CCC1(C)C 89696,N1(C(Cn2ccc(C)n2)=O)CC2(C1)C(NC(C1C=CCC1)=O)CCS2(=O)=O 89697,c1(C(=O)NCCCCN(C(C(C(C)C)OC)=O)C)ncn2c1COCC2 89698,C1(N(C(C)C(=O)N2CC(N3CCCC3)C2)CC)CCN(C)CC1 89699,C123CCC(C1)(OC2)CNC3=O.CCCCC(=O)NC1(CCN=[N+]=[N-])CC1 89700,C(C1=NOC2OCCC12)NC(C1C=CCN(C(C(CO)OC)=O)C1)=O 89701,C#CCC(C)(C(=O)NCCN(C)C(C)C)NC(=O)Cc1cncnc1 89702,C1(NC(C(CC)N(C)C)=O)CCCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 89703,C1(C(=O)NCCCCCCC2CC2)COCCN(C(c2ccc(C(F)F)o2)=O)C1 89704,c1(CCN2CC(N(C)C(=O)C3CC3)C2)ccc(F)cc1 89705,N1(C(C(c2cnn(C)c2)C)=O)CC2(CCCC(CNC(c3cnsc3C)=O)O2)C1 89706,c1(OC2(C(=O)Nc3ccc(OC)cc3)CC2)ccnc(CO)c1F 89707,c1(CC(C)NC(N2CCN(c3ccc(F)cc3)CC2)=O)ncc(Br)cn1 89708,C1(C(=O)NC2(CNC(=O)CCOC(C)C)CC(OC)C2)C(C)(C)C1(C)C 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89779,C1(c2nc(C(C)OCC)nn2-c2ccc(Br)nc2)CCc2nncn2C1 89780,c1(NC(CC2(OC)CN(C(C(CSC)C)=O)C2)=O)ccc2cncn2c1 89781,c1(SC)cccc(OCC(=O)N(CCCNC(c2ccccc2)=O)C)c1 89782,C1(CCOC)(NC(=O)Cc2csc(COC)n2)CCN(C(=O)C(O)C(C)C)C1 89783,N1(C(C(C)(C)OCC)=O)CCN(C)C(C(=O)N(CC(O)CN(C)C)C)C1 89784,CC#CC1CCN(C(=O)COC2CC(CC)C2)C1.c12cc(sn1)NC2=O 89785,C1(CNC(Cc2cnc(C)s2)=O)CC(C)N(C(=O)C(CO)NC(=O)C(F)(F)F)C1 89786,Cc1cc(C(=O)NC2CC(NC(C3CSCC(=O)N3)=O)C2)c2c(c1)C(C)CCN2 89787,N1(C(C2C(=C)CC2)=O)CCOCC1CCNC(=O)CSc1n[nH]c(O)n1 89788,c1(OC)ccc(C(=O)N(C(C)CNC(c2ccc(C(F)F)cn2)=O)C)c(F)n1 89789,C1(NC(C(C=C)O)=O)CCN(C(=O)C(C)NS(=O)(=O)CC)CC1(C)C 89790,C1(CC(C)C)CCN(C(=O)C(F)n2ccnc2)CC1.C12CC1CNC2=O 89791,c1(C(=O)NCCN(C(C2C(C)CC2C)=O)CC)nc(C)oc1C 89792,C(C(F)C(=O)NCC1CCOC1)C1CN(C(=O)CSC(F)F)C1 89793,C1(NC(C(CC)c2ccccc2)=O)CCCCCN(C(=O)CCC2CCC2)C1 89794,N1(C(C2(NC(CCOC)=O)CCCC2)=O)CCC(NC(=O)CN2CCC2C)CC1 89795,c1(NC2C(NC(C(C)(C)c3nccs3)=O)CCCC2)nc(O)c2cnn(C)c2n1 89796,C1(=O)C(C(C)C)NC(=O)C2(CC2)N1C.C1(C=O)CCC(=O)C1.CO 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89815,C(CC(C)(C)CNC(c1ccc(C2CC2)nc1)=O)NC(c1c(C)csc1)=O 89816,C1(C)(c2cc(C(N(CCCNC(=O)CC3CCCC3)C)=O)on2)NC(=O)NC1=O 89817,C(CC)(CCCC(=O)N(C1CCCN(CC)C1)C)NC(CCCCCOCC)=O 89818,c1(CCC)cc(=NCC2CCCN(C(c3cc(Cl)ccn3)=O)C2)[nH]c(Cl)n1 89819,N1(C(C(CC)OC)=O)CC2CC(O)C1C2NC(=O)CCOc1cccc(Cl)c1Cl 89820,C1(C(N2CCCC(CCC(N3CC(C)C(C)C3)=O)C2)=O)Cc2ccccc2C1 89821,N1(C(CCOC(C)=O)=O)CC(NC(=O)COCC2CCC2)CC1(C)C 89822,CCC(C)(O)C(=O)N1CCC(N2CCN(C(=O)CCc3ncc(C)[nH]3)CC2)C1 89823,N1(C(CCCCCC)=O)CC2(C1)CN(C(=O)CC1CCC1OC)CC2CO 89824,CCC(C)CC(C)C(=O)NCCN(C)C(c1ccc(CN(C)C)nc1)=O 89825,N1(C(COCC=C)=O)CC(NC(C2CC2CC)=O)C(C)C1 89826,N1(C(CSC(C)C)=O)CCC(C)(C)C(CNC(c2ccc(=O)n(C)n2)=O)C1 89827,O=C1CC(=O)NC(C(N2CCC(C=CC(=O)NC(c3ncc[nH]3)CO)CC2)=O)C1 89828,c1(N2CCOCC(CNC(=O)CCN3CCCCC3)C2)ncc([N+](=O)[O-])cc1Br 89829,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C3CN(C4CCC4)C3)=O)C2)C1 89830,c1(C(=O)NCC2(NC(C(CCSC)O)=O)CC2)c(C)ncnc1C 89831,N1(CC(=O)NC2(C)CCN(C(C3CN(COC)C(=O)C3)=O)C2)C(=O)CN(C)C1=O 89832,c1(NC(=O)COc2cccc(F)c2)ccn2c1CSCC2.CN1CC1 89833,C1(C(=O)NC(c2cn(C)cn2)C)(NC(C=C(C)C(F)F)=O)CC1(C)C 89834,C1(C)(COC)CC(NC(=O)CC2CC2)CN1C(c1c(Cl)cccc1Cl)=O 89835,C1(OC)CC(C)(NC(=O)Cc2cncs2)C1.C1(=O)C=CC(=O)N1.C(C)(C)N 89836,n1(CCOC)nnnc1C(c1ccnn1C(C)C)NCCOCCOC 89837,C1(C(=O)Nc2c(CC)cc(C#N)cc2)CCC2(CN(C(C3CC3(F)F)=O)C2)O1 89838,CON(CCC(=O)Nc1nnccc1C)C(=O)Nc1cnn(C2CC2)c1C 89839,N1(C(C(COC)C)=O)CCN(C(=O)CNC(c2nccc(C)n2)=O)CC1 89840,N1(C(CC)=O)CCC(C(=O)NCc2cnn(C)c2)CC1C 89841,C1(OC)CCC2(C(=O)N(CC(O)CNC(c3cccc[n+]3[O-])=O)C)CCC12 89842,c1(N2CC=CC(NC(CCC(C)(C)OCC)=O)C2)ccc(C#N)cn1 89843,C=C1CCN(C(=O)CNC(=O)OC(C)C(F)(F)F)C(C(=O)OC(C)=O)C1 89844,c1(CC(=O)NC2CC(F)(CNC(=O)C3=CCC3)C2)c[nH]c2cccc(F)c12 89845,c1(C(C)NCC2CC(CC(=O)O)C2)ccc(C(F)(F)F)cc1 89846,CC1OC(=O)NC1C(=O)NCC(C1(O)CN(C(c2cnc(O)o2)=O)C1)(C)C 89847,c1(CN2C(C)(C(=O)O)CCC2)nc2cnccc2[nH]1 89848,c1(C(N2CC(N(C(=O)CC3(C#N)CCC3)CC)C2)=O)cncc(C(N)=O)c1 89849,Cc1ncc(Br)cc1C(N1CC2C(CNC(C3(COC(C)C)CC3)=O)C2C1)=O 89850,C12(CC(=O)NCC3CCN(C)C3)CC(CO1)N(C(=O)CC1CCCC1)C2 89851,C1(CC)CCN(C(=O)CCc2ccnn2C)C(C(=O)NCC2CCCCO2)C1 89852,C1(NC(C=CC(=O)N(C)C)=O)CCC(N(C(=O)CC2CCCC2C)C)CC1 89853,COn1cnc(C)c1C(N1CCN(CCNC(=O)Cc2cccnc2C)CC1)=O 89854,c1(C(=O)NC(C)C(=O)NC2CCCCC2NC(=O)C(N)=O)cccc([N+](=O)[O-])c1 89855,C1(C(=O)NC(C2(C(N3C(CCC)CCC3)=O)CC2)C)CCOC(C)(C)C1 89856,c1(C(N2CCC(O)(C(C)CNC(=O)CCC3CC3)C2)=O)c[nH]c2nc(Cl)ccc12 89857,C(C1CCCCCC1)=CC(=O)N(C1CCN(c2nnc(C(N)=O)s2)C1)C 89858,c1(NC(C)CCCC(F)(F)F)cc(=NCc2nc(Cl)cs2)[nH]cn1 89859,C(=O)(CCC1=CCCCC1)N1CCC(C)(NC=O)CC1.C1(CCC=O)CCC(=O)N1 89860,N1(C(C(N(C)C(C2CSCC(=O)N2)=O)C2CC2)=O)CCCC(F)CC1 89861,C1(NC(CCCC#C)=O)CCN(C(=O)Cc2ccc(Br)nc2)C(C)C1 89862,CN1CC2CCC(C1)N2C(C1CC(F)(F)CN1C(=O)CC1CSCCO1)=O 89863,CP(C)(=O)c1cccc(C(=O)NC2CCC(CNC(C3CCC(=O)O3)=O)CC2)c1 89864,C1(NC(CC2N(C(C)C)CCC2)=O)(CO)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 89865,c1(C(=O)NC(C2CN(C(=O)CC3(O)CCOC3)C2)C)nccc2ccccc12 89866,N1(C(C(CC)(C)CO)=O)CC23CCCC2(C1)CN(C(c1c[nH]nc1S(N)(=O)=O)=O)C3 89867,c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cnc(S)nc2)=O)nn1CCO 89868,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2=CC(C)(C)C2)=O)C(C2CC2)CC1 89869,N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C1C(=O)NCc1cnc(C)nc1 89870,C1(=CC(=O)NC2CC(F)(CNC(C3CCC(OC)C3)=O)C2)CCCCCC1(F)F 89871,N1(C(CCc2cc(C)n(C)n2)=O)CC2(CCN(C(=O)C(C)N(C)C)C2)C1 89872,n1(CC(=O)NC2CCC(CNC(CC=C=C)=O)C2)nc(C)cc1C 89873,N1(C(c2c(C)nc(-c3ccccc3F)s2)=O)CC(O)C(O)C1CO 89874,CCCC(C)(C)C(=O)N(CC(=O)NC1(C)CCC(O)CC1)CC(C)C 89875,C(=O)(C(C)(C)CCC#N)N1CC(CNC(C=CC(CC)C)=O)C(C)C1 89876,c1(C(=O)NC(C)CNC(C2CCC2(F)F)=O)ncn2ccccc12 89877,c1(OCC)cnc(N2CCN(C(c3cc(C4CCC5CC5C4)[nH]n3)=O)CC2)cn1 89878,c1(C(N2C(CC)CN(C(=O)CSc3cccs3)CC2)=O)c(Cl)nc2ccccn12 89879,CC1(C)CN(C(C2CC3CC23)=O)CCN1C(c1cc(Cl)c(Cl)c(Cl)c1)=O 89880,N1(C(c2c(C(C)C)scn2)=O)CCC(NC(=O)CCCc2ccccc2)C1C 89881,CC#CCC(C)N=c1[nH]c(=NCC2(C3=CCOCC3)CC2)[nH]c2c1CCCCC2 89882,CC(C(=O)NCC1(F)CC(NC(=O)Cc2cc[nH]c2)C1)C(C)(F)F 89883,c1(CC(=O)NC2CCC(NC(=O)C(O)C3CC3)C2)ccnc(O)c1 89884,C(=O)(C(C)(C)N=[N+]=[N-])N(CC(=O)NCC1(C=C)CCC1)CC#C 89885,CC1CC(NC(=O)CSC(C)(C)C)CN(C(c2nc(-c3ccccc3)n[nH]2)=O)C1 89886,Cn1cc(N)c(C(=O)NCCC2CN(C(C3CC3(C)Cc3ccccc3)=O)C2)n1 89887,C1(NC(c2cc(C(C)=O)on2)=O)CCC2(CCCN2C(=O)C2=CCCSC2)CC1 89888,C1(=O)C(N2CCCC(CC3CC3)C2)C(C2CCCC2)OC(=O)CCN1.CCOC 89889,C(C(C)C(=O)N(CCCNC(c1sccc1Cl)=O)Cc1ccccc1)OC 89890,c1(C(=O)NCC(N(C(=O)Cc2ccccc2)C)C2CC2)ccc(O)cc1O 89891,C(N=c1cc[nH]c(C#N)n1)C1CC(C)N(C(=O)C=CC2CCOC2)C1 89892,c1(C(=O)NC2CN(C(Cc3cc(C)on3)=O)C(CO)C2)cnc(O)cc1O 89893,CC1Cc2cc(Br)ccc2N(C(=O)Cc2cn(C)nc2C(F)(F)F)C1 89894,N1(C(=O)NCc2cc(CC)c(F)cc2)C2(CCCC2)OC2(CCC2)C1 89895,N1(C(c2c(C)cco2)=O)CC(NC(C2(c3cnc[nH]3)CC2)=O)C(C)(C)C1 89896,C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)C(F)C(C)C)OC(C)C 89897,C(=O)(C1=CCC2CCC1N2C(C1CCOC1)=O)Nc1c(C#N)ccc(C)n1 89898,c1(C(=O)NCC2N(C(C3C(=C)C3)=O)CCCC2)cc(O)ccc1[N+](=O)[O-] 89899,C1(C(N(OC)CCO)=O)CCC2(CCCCC2)CC1 89900,CCC(C)CC(C(=O)NCC1(CC(N)=O)CC1)NC(c1cncnc1C)=O 89901,c1(Cc2n(C(COC)C)nc(-c3ccc(O)c(C)c3)n2)cc(F)cc(F)c1F 89902,c1(C(=O)NCC(N(C(C(C)OC)=O)C)C2CC2)nc(C2CC2)ncc1C 89903,N1(C(C(C(C)C)NC(CC)=O)=O)CCCC(C)(CNC(C2C3COCC23)=O)C1 89904,c1(NC(C2(C)N(Cc3ccc(C#C)s3)CC2)=O)ccc(F)c(CO)c1 89905,C(CCC(=O)NCCNC(c1ccnn1CCc1ccccc1)=O)SC(C)(C)C 89906,c1(C(=O)NCC2CC(NC(CCc3ncc(C)[nH]3)=O)C2)cc(Br)c(O)nc1C 89907,C1(CC(=O)NCC(CCNC(c2coc(C(C)C)n2)=O)OC)CCC(C)(C)O1 89908,C(C1=CCCN(C(c2ccsc2C)=O)C1)NC(Cc1cn(CC)nn1)=O 89909,c1(OC)ncccc1C(=O)NCCCCC1CCN(C(c2ccoc2)=O)CC1 89910,C1(NC(CCc2n(C)c(S)nn2)=O)CC2CN(C(=O)CC3CCCC(O)C3)CC12 89911,c1(OC)ccc(CN2CC(CO)(NC(c3cc(C)c(F)cc3Br)=O)C2)c(Br)c1O 89912,CC1=CC2=NCCCNS(=O)(=O)C1=CN2.n1(CC2C(NC)C2)cccn1 89913,c1(C(=O)NCC2(C)CCC(NC(Cc3c(C)con3)=O)C2)cnc(O)n(C)c1=O 89914,C1(C(=O)NC(C#C)CC)C2CCN(C(=O)C(OCC)OCC)CC12 89915,S(=O)(=O)(c1ccc2[nH]c(=NC3C4CCCCCC34)ccc2c1)N1CCC(N(C)C)CC1 89916,N1(C(c2c(C)cns2)=O)CCC(NC(=O)Cn2c(C)ccc2C)CC(O)C1 89917,N1(C(C2C(=C)C2)=O)CCCC(COC)(NC(=O)C(C)NC(C)=O)C1 89918,CC1(C)CCCCC1C(=O)NCC1(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC1 89919,c1(C(=O)OCC(C(c2ccc(F)cc2)=O)=O)cccc2c1OCCO2 89920,c1(C(=O)NC(C)CCNC(=O)Cc2ccc(=N)[nH]c2)cc2ccccc2c(O)n1 89921,N1(C(c2cc(C)sn2)=O)CC(OC2CC2)C(C)(C)C1.C12(CC1)C(=O)NC2 89922,C(N=c1cc(F)nc[nH]1)c1ccc(NC(CCc2cccc(OC)c2)=O)c(F)c1 89923,c1(-c2cccc(OCC)c2Br)ccc2c(C(N3CCC(OC)C3)=O)nn(C)c2c1 89924,Cc1ccc(F)c(N)c1C(N1CC(C(C)NC(C2CC2(F)Cl)=O)C1)=O 89925,CC(CC(N)=O)C(=O)N1CC(O)(CNC(=O)CCc2nc(-c3ccoc3)no2)C1 89926,C1(CN(C(CC)=O)CC)CCN(C(=O)C(O)C(C)c2ccccc2)CC1.C1CC1 89927,C12(CNC(C3(C)CCCO3)=O)CC(CO1)N(C(C1CCCN1C=O)=O)C2 89928,O=S(=O)(C1CCC(C(F)(F)F)C1)Nc1cccc(C2CCC2)c1 89929,S(=O)(=O)(c1ccc(NCCC(C)C)c(F)c1)NCC(CC)(C)CO 89930,C1(C(N(C(C)CNC(=O)CN2CCN(C3CC3)C2=O)CC)=O)CC2(C1)CC2F 89931,C(=O)(CCP(C)(C)=O)N1CC(C)C(CNC(=O)Cc2ccccc2C(F)(F)F)C1 89932,C1(C(=O)NCC(CN(C(=O)CCn2cccn2)C)(C)C)CC2CCCCN2C1 89933,CCCCC(C)CCC(=O)NC1CC1NC(=O)CCc1cncn1C 89934,N1(C(c2cn(CC)nn2)C(=O)NCSc2ccccc2)CC2OC(C)(C)OC2C1 89935,C12(NC(=O)CC3CC34CC4)CC(C1)N(C(C1CC=CCC1)=O)C2 89936,C1(C(N(CCN(C(c2ccc(COC)s2)=O)C)C)=O)CCCCC1F 89937,c1(-c2nc(CCCCC)nn2-c2ccncc2)cccc2nc[nH]c12 89938,c1(C(=O)NCC(CCCC)NC(c2nocc2Br)=O)cc(C)ccc1OC 89939,Cc1cc(Cl)c(C(=O)NC2CCCCN(C(=O)C(C)(C)C)C2)cc1C 89940,C(=O)(C(C(C)C)OC1CCCCC1)NCCCC(C)N(CC(=O)NC)C 89941,C12(C(N3C(CN(C(C(N4CCCCC4)C)=O)C)CC(F)C3)=O)CCC(C1)OC2C 89942,C(C1CCc2ccccc21)n1c(-c2cc(OC)c(N(C)C)cc2)nc(CCC)n1 89943,c1(OCCOC)ncnc(Cl)c1-n1ncc(NC(=O)CCCn2c(O)nnc2O)c1 89944,C1(C(=O)NC2CC(CNC(C(CC=CC)CC)=O)C2)CC2(CCCCO2)C1 89945,c1(C(N2CC(OCCC(=O)NCc3cccc(O)n3)C2)=O)ccc2cccnn12 89946,C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C(C(C)C)C#N)=O)C1)=O 89947,CCCCC(CCC)NC(=O)CC1(NC(c2cnn(C(C)C)c2C)=O)CCC1 89948,C12(CCC(N3C(CNC(=O)CCc4ccncn4)COCC3)=O)CCC(CC1O)C2 89949,N1(C(C(C(CC)C)C)=O)CC(N=c2[nH]c(Cl)nc3ccc(Cl)cc23)CC2(CCC2)C1 89950,CN1CCC2(CCN(C(C3CCCC3CNC(c3cc(CCO)on3)=O)=O)C2)C1 89951,C(=O)(C(O)C(F)(F)F)NCC(C)=CC(=O)NC(CO)C1(C)CC1 89952,c1(C(=O)NC(C2N(C(c3nc(CC)sc3)=O)CCCC2)C)cc(C)nc(C)c1 89953,C1(C(=O)NCC(CNC(=O)C=CSc2ccccc2)O)CCc2nnc(O)n2C1 89954,n1(CCC(C)C)ncc2cc(C(=O)NC(C)CNC(=O)C(O)C(C)(C)C)cnc12 89955,c1(C(N2CC(CCNC(C3N(CC)CC3)=O)OCCC2)=O)cnc2ccnn2c1 89956,N1(C(C)C)CC2(CN(C(=O)OC(C)(C)C)C2)C1.C12(C)CCCC1C(=O)N2 89957,N1(C(CN(C(c2ccc(OC)nc2)=O)CC)=O)CCC2(CCC(C)C2)C1 89958,c1(C(=O)NC2CCC(NC(c3cccc(SC)c3)=O)C2)c[nH]c(=N)c2[nH]ccc12 89959,c1(C(=O)NC2C(NC(c3ccc(C(C)=O)cc3)=O)CC2)nccc2cnn(C)c12 89960,Cc1csc2ncnc(NCC3(CNC(=O)CC4CCCCC4)CC3)c12 89961,C1(C(=O)NC2CCC(N(C(C(CC#C)C)=O)C)CC2)CCC(C)(C)OC1 89962,N1(C(C(C)N(C)C)=O)CC2CCC(N=c3nc[nH]n3C3CCN(C)CC3)CC2C1 89963,CCC(C(=O)NCC(C)(C)CNC(=O)C(C)=CC(C)(C)C)N(C)C 89964,Cc1cnc(SC2CC=CCC2)cc1C(F)(F)F 89965,c1(OC)c(CN2CCC(n3nc(CO)nc3-c3ccc(C)o3)CC2)cccc1Cl 89966,N1(C(C2(CCC)CC(=O)C2)=O)CCN(CCCNC(=O)C=CC(C)C)CC1 89967,C(=O)(CC1=CCCCC1)NC(C)CN(C(=O)CCCCCc1ccccc1)C 89968,c1(C(N2C(C(=O)Nc3c(C)ccc(F)c3)CC2)=O)ccc2n[nH]cc2c1 89969,c1(NS(CC(=O)OC)(=O)=O)cc(CNC(c2cc(CO)[nH]n2)=O)cc(C)c1 89970,C1(CNC(=O)Cn2nnc(C3CC3)n2)CCN(C(c2ccnnc2)=O)CC1 89971,c1(C(=O)NCCC(C)C)ccc(CNC(C2C=CCCC2)=O)o1 89972,C1(NC(c2cc(C(C)C)no2)=O)CCC2(CCCN(C(=O)C3=C(Cl)CC3)C2)C1 89973,c1(OC)ccc(NC(C)=O)cc1C(N1CCCC(N(c2ncccc2Br)C)C1)=O 89974,N1(C(c2c(C)noc2C)=O)CCN(C(C2C3(CC3)C23CC3)=O)CC1CF 89975,C(=O)(C1CCc2c[nH]nc21)NCCCC1CCN(C(C(C)CC2CC2)=O)CC1 89976,CCC(C#N)(CC)C(=O)NCC(C)(C)NC(=O)CN1CCCS1(=O)=O 89977,c1(C(C(N2CC3C(CNC(c4ccc(C)nn4)=O)C3C2)=O)C)ccncc1C 89978,CC1CCN(C(C2CC3CC2C3)=O)CCN1C(C1CC1Cc1ccccc1)=O 89979,C(=O)(C(O)CC(C)C)N1CCCC(C2N(C(c3c(C)sc(O)n3)=O)CCC2)C1.CN 89980,c1(NC(c2c(C)nc(CCCC)nc2C)=O)cccc2cnccc12 89981,CC1c2ccccc2OC1C(N1CCCC(O)(CN(C(=O)CC(C)(C)O)C)C1)=O 89982,c1(C(=O)OC)cnc(C)c(C(=O)NCC2(c3ccccc3)CCCO2)c1 89983,C1(=O)C(C)(C)CCCN1.CC(C)C(C)CCNC(=O)CSCC(N)=O 89984,c1(C(=O)NC2C(C)CN(C(=O)COC3CC(F)(F)C3)CC2)cccc2c1CCC2 89985,c1(C(N2CCC(N(C(C3C(C)CN(C)C3)=O)CCO)C2)=O)cnc2ncccn12 89986,N1(C(C(C=CC)O)=O)CCCCC1C1(NC(c2cc(C(N)=O)nn2C)=O)CC1 89987,c1(C(=O)NCCc2ccc(COC)cc2)cnc(C)c(C#N)c1 89988,Cc1cc(CC(N2CC(C)(NC(c3ncsc3N(C)C)=O)C2)=O)ccc1O 89989,C1(C(N2CC(CCC)C(NC(=O)C(c3ccccc3)C)C2)=O)CC(C(C)C)=NO1 89990,C#CCCCC(C)C(=O)NCCn1ccc(C(=O)NC2CCN(CCO)CC2)c1 89991,CC1CN(C(c2cnc3[nH]nnc3c2)=O)CC(C)CN1C(=O)C1=CS(=O)CCC1 89992,N1(C(c2c(C)c[nH]n2)=O)CCOCC1CNC(C1C=CCCC1)=O 89993,c1(C(C)NC(=O)C(C2CCC2)NC(=O)CCCNC(N)=O)nccc(O)n1 89994,c1(C(=O)NC2CN(C(CSc3ccc(C)cc3)=O)C(C)C2)nc(C)n(C)c1C 89995,c1(C(=O)NC2CCN(Cc3cn(CC4CC4)nn3)C2)ccc2ccncc2c1 89996,c1(C(=O)NC2CCC(NC(CC=CCC)=O)CC2)cnc2c(c1)CCOC2 89997,CC(CCNC(=O)COCc1nc[nH]n1)CCNC(c1c(Cl)nsc1Cl)=O 89998,N1(C(C=CC(=O)OC(C)(C)C)=O)CCCC1CNC(=O)CCC1CCOC1 89999,c1(C(N2CCC(N(C)C(c3cc(CO)ccn3)=O)C2)=O)ccc(CO)c(Cl)c1 90000,C(C(CC(=O)NC1CCC1NC(=O)Cc1cc(F)ccc1Cl)C(F)(F)F)N(C)C 90001,C(=O)(C(F)(F)CCn1cc(Cn2ccc(C(=O)O)c2)nn1)c1n(CC)ccn1 90002,c1(OC)ccc(C(=O)NCC2CC(F)(F)CN2C(c2ccc(SC)s2)=O)c(C)n1 90003,c1(C(C(=O)NC2CC(C)N(C(=O)CN3CCCC3)CC2)(C)C)ccc(F)c(F)c1F 90004,C(=O)(C1=C(Cl)CCC(C)C1)N(CCNC(c1cc(-n2ccnc2)ccn1)=O)CC 90005,Cc1c(C(=O)NCC2COC(C)(C)CN2C(c2ccoc2)=O)sc2ccccc12 90006,C1(c2ccccc2)CN(N(C2CCCN2C)C)CCN1.c1(C)cccc(Cl)c1 90007,c1(C(=O)NC(C(CO)NC(C(C)OCS(C)(=O)=O)=O)C)cncc2nnn(C)c12 90008,C=CCCCC(C(=O)N1CC2COCC2C1)NC(c1[nH]ccc1CC)=O 90009,c1(OC)nc(C)c(C(N2CCOCC2CNC(c2cnc(C)[nH]2)=O)=O)s1 90010,c1(C(=O)NC2(CC(=O)NC(c3c(F)cccc3F)CC)CC2)cccn2nccc12 90011,Cc1nn(C)cc1C(=O)NCC1(C(F)F)CCN(C(=O)Cc2cocn2)C1 90012,CC(C(=O)N(C1CCCCC1NC(C1CC(C#N)C1)=O)C)C(C)(F)F 90013,C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)NCc1c(CN(C)C)cccc1 90014,CC1CCCCC1(C)NC(C1(NC(=O)C=CC2CC2)CCC1)=O 90015,c1(CSC)ccc(C(=O)NCC2CN(C(C3CCCC(C)C3)=O)C2)cc1[N+](=O)[O-] 90016,CC1CC(CNC(=O)CCN2CCCC2)CN1C(c1ccn(C)n1)=O 90017,C1(C(=O)NCC(C)(C)CNC(=O)C(c2cccnc2)O)CC2(C1)CC1(CCC1)C2 90018,C(=O)(C(C)(C)C(=O)N1CCC(CNC(=O)Cn2cnnn2)C1)OC 90019,NC1(CCC2CC(C(=O)Nc3nnnn3-c3ccc(F)cc3)C2)CCCCC1 90020,C1(NC(=O)Cc2cc(C3CC3)on2)CC2CCCC(C1)N2C(c1coc(Br)c1)=O 90021,C1(C(N(C2CCCCN(C(c3cnccn3)=O)C2)C)=O)CCCC(C)(C)CC1 90022,c1(N2CC(OC)C3(C2)CC3)nc2cccnc2c(=NCCSc2nccn2C)[nH]1 90023,C1(NC(C2CN(C(=O)Cc3nc(Cl)cs3)CCC2O)=O)CCc2ccccc2C1 90024,C(CS(=O)(=O)CC(=O)N1CCCCC1c1n[nH]cc1NC(=O)C(O)CSC)OC 90025,C1(O)(CNC(C=Cc2ccc(CCCC)o2)=O)CCN(C(=O)CO)CC1 90026,N1(C(C=C(C)C(C)C)=O)CC2CCOCC2(NC(c2nc(C)oc2C)=O)C1 90027,N1(C(C23CC(c4ccccc4)(C2)C3)=O)CCCC(CNC(C2(CCC)CC2)=O)C1 90028,N1(C(C2CCCN(CC)C2)=O)C2CCCC1CN(C(c1cccc(C)n1)=O)CC2 90029,c1(C(=O)Nc2scnc2C2CC2)n[nH]c2ccc(-c3ccccc3F)cc12 90030,N1(C(=O)OC(C)(C)C)CC(OCC2(C(=O)O)CCC2)CC1c1cccs1.C1CC1 90031,N1(C(c2cc(C)no2)=O)C(C(=O)Nc2oncc2C)CCC1C 90032,C(=O)(C(O)CCC(C)C)NCCN1CCCN(C(c2n(CC)ncn2)=O)CC1 90033,c1(C(N2CCN(C(c3cc(CCCO)on3)=O)CC2)=O)ccc(O)c(Cl)c1 90034,N1(Cc2c(OC(C)C)ccc(Br)c2)CCCC2CN(c3ncncc3F)CC12 90035,c1(OC)ccccc1N(C(=O)CC1CCCN(C(=O)CC2CCCCC2O)C1)C 90036,C1(NC(CCCN(C(C)=O)C)=O)CCCCC1NC(=O)CSC1CCCC(=O)N1 90037,C1(CN(c2cccc(C)c2C)C(=O)NCCOC)CCOC2(CCC2)C1 90038,c1(C(=O)OC)cc(Cl)ccc1NC(=O)CC1CCN(C(c2ccnc(Br)c2C)=O)C1 90039,C(C(C(C)(C)C)NC(=O)CCNC(=O)CO)NC(C(c1cscn1)N(C)C)=O 90040,O=C1CCCCC(C(=O)OCC2CC3(CCC3)CO2)C1 90041,Cc1nc(C(N2CC(F)(CNC(C3CC3(C)C)=O)C2)=O)c(C)s1 90042,N1(C(C(C)=C2CC2)=O)CCC2(CCCC2NC(C2CC(O)C2)=O)C1 90043,c1(N2CC3C(C(=O)NC)C3C2)nc(NCC2CCC(C)(C)O2)c2ncsc2n1 90044,c1(C(=O)NC(C)CC2CN(C(=O)CC3CC3(C)C)C2)ccn2c1CCCC2 90045,C1(COC)(NC(=O)C(C)=CC)CCN(C(C2(C)CC2c2ccccc2C)=O)CC1 90046,CC1CCCCC1C(N1CC(CNC(c2cccc(C(C)(F)F)c2)=O)C1)=O 90047,Cc1n[nH]c(=NCCC2CCC(NC(C34CC(CO)(C3)OC4C)=O)C2)s1 90048,N1(CCN2CCN(CCN(C(CS(CC)=O)=O)C)CC2)C(C)CCCC1C 90049,Cc1ncnc(O)c1C(=O)NC1C2CN(C(c3c(C4CCC4)cnn3C)=O)CC12 90050,N1(CC(=O)NCCC(=O)N(C(CC)CO)C)CCC(C)C1 90051,C1(CCC)(CNC(=O)CCOC)CCN(C(=O)CC2(Oc3ccccc3)CC2)C1 90052,N1(C(C(C2CCOC2)NC(C2(CC(N)=O)CC2)=O)=O)CC2CCC(C1)O2 90053,CCC(O)C(C)C(=O)N(C)CC1CCN(C(=O)Cn2cnnc2O)CC1 90054,c1(CC(=O)N(CCC(C(C)(C)C)NC(C2CCC2)=O)C)ccc(C#N)cc1F 90055,N1(C(C2CC(C)C2)=O)CCc2nc(CNC(=O)CC3CC4CCC3CC4)sc2C1 90056,N1(C(CCCOCC)=O)CCCC(CNC(C2CCCN2C(=O)C(F)(F)F)=O)C1 90057,C1(CNC(C2CC3(CC3)CO2)=O)CC2CN(C(c3cccnc3O)=O)CC12 90058,C1(NC(c2c(C)nco2)=O)CCN(C)C12CCCN(C(=O)C(C)N(C)C)C2 90059,c1(C(=O)NC(C)CNC(c2ccnc(C3CC3)n2)=O)ccc(OC(F)F)cc1F 90060,c1(C(=O)NC(CCCNC(C(C)OCC)=O)(C)C)cccc2nc(S)oc12 90061,c1(C(N2C(C3(NC(C4(OC)CC=CC4)=O)CC3)CCC2)=O)cc(C)cc(F)c1 90062,N1(C(CCN2C(=O)NCC2)=O)CCOC(Cn2cc(-c3csnn3)nn2)C1 90063,N1(C(CC(CC)CC)=O)CCOC2(CCN(C(=O)COC3CCC3)C2)C1 90064,C12(NC(c3cc(Cl)cs3)=O)CCN(C(c3ccn(CC(F)F)c(=O)c3)=O)CC1C2 90065,C1CCN=C2C=CN=C(N2)N1C1CCOCC1.CS(=O)(=O)CC1(CO)CC1 90066,Cc1nc(N2CCOCC2C2CCOC2)c2ccccc2n1 90067,N1(C(c2c(C)ccc(F)c2)=O)CCC2CN(C(=O)C(C)CO)CC2C1 90068,C12CN1CCC2C.c1(C(C)NC(C=NOC)=O)cc(O)nc(SC)n1 90069,c1(C(=O)NCC(C)N(C(=O)CC2CCCN2C)C)cc(C(F)(F)F)ncc1N 90070,c1(C(C)(C)C)cccc2c(NCCCC(C)(C)CO)cnn12 90071,c1(CC)cc(CC)nc(N2CCN(C(=O)CN3CCC(C)CC3)CC2C)n1 90072,c1(C(N(CC(N2CC(=C)C2)=O)CC#C)=O)cc(F)ccc1C 90073,N1(C(C(C(COC)C)C)=O)CC(CO)C2(C1)CN(C(c1cccc(C)n1)=O)C2 90074,C(=O)(CCCN=[N+]=[N-])NC1CCC(C)(CNC(c2c[nH]c(=NC)s2)=O)C1 90075,c1(CC)[nH]nc(Cl)c1C(=O)NC(C)CC1CN(C(C2CCOC2)=O)C1 90076,c1(C(N2C(CNC(C3N(CC)CC3)=O)C(C)CC2)=O)cc2c(s1)CCCC2 90077,CC#CCCCC(=O)N1CCC(C)(NC(c2cnc(C3CCC3)cc2C)=O)C1 90078,CC(C)CCC(=O)NC1CCCC1(C)CNC(=O)CC1CC2CCC1C2 90079,C1(C(=O)NCC2(CCC)CC2)CC2CCC(C1)N2C(=O)CS(=O)(=O)CC 90080,N#Cc1[nH]c(=NCC2(O)CCCN(C(C3(CCF)CCOCC3)=O)C2)sc1Cl 90081,C1(C(=O)NC(CN(C)C)C(=O)NCc2c(CC)c[nH]n2)COCCN1C 90082,CCC1=NOC(C(=O)NCCCN(C(=O)Cc2nc(C(C)(C)C)cs2)CCO)C1 90083,c1(C(N2CCC(C(=O)NC(c3c(C(=O)OCC)n[nH]c3)=O)C2)=O)snc(C)c1N 90084,C1(C(N2CCCC(n3cc(CCCCO)nn3)C2)=O)(OC)CC2CCC1C2 90085,C(=O)(CCS(=O)(=O)C1CCCC1)NCCC(C)N(C)C(C1SCCS1)=O 90086,C12(CC(=O)NCCc3ncc(CNC(C(C)O)=O)[nH]3)COC(C)(C1)C2 90087,C1(C(N(CC)CC)=O)OCCC1NC(=O)CC1(CCCC#C)CC1 90088,C1(NC(C(C)C2(O)CCC2)=O)CN(C(c2ncccc2Br)=O)CC2(CC2)C1 90089,N1(C(C2(C(N)=O)CC2)=O)CCC(CNC(C2(CCN(C)C)CC2)=O)CC1 90090,CCC(C(=O)N1CCCCC(N(C(=O)C(C)(C)OC(C)=O)CC)C1)C(F)(F)F 90091,c1(C(=O)NCC(=O)N(CCCN(C(C(C)N(C)C)=O)C)C)ccc(F)cc1F 90092,N1(C(C(c2cnccn2)C)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)CC1C 90093,Cc1cc(C(N2CC(C(C)(C)O)(CNC(C3CN(C(C)C)C3)=O)C2)=O)nnc1O 90094,N(C(=NCC1CC1)NCc1ccnc(-n2ccnc2)c1)Cc1c(C)nns1 90095,c1(CNc2ccc(-c3ccc(OC(C)C)nc3)cn2)c(F)cncc1F 90096,c1(OC)nsc(OC)c1C(N1CCC(CCNC(=O)CN2CCCC2C)C1)=O 90097,c1(C(=O)NCc2c(CNC(c3cn(C)nc3)=O)nco2)cc(Br)cnc1C(F)F 90098,c1(CC(=O)NCC2C(NC(C3C(C)(C)C3)=O)CC2)c(Cl)cccc1Br 90099,C1(C(N(CC#C)CCO)=O)CCC=CC1NC(C1CCC1C(=O)OC)=O 90100,c1(C2N(C(C(=O)NCCSC)C3CCCC3)CC2)cccc(OCCN)c1 90101,c1(N2CCC(N(C)C(C3CC3C3CC3)=O)C2)nc(Cl)nc2c1ncn2C 90102,c1(CC(C(N2C(c3nc(C)[nH]n3)CCCC2)=O)N)ccc2ncsc2c1 90103,c1(C(N2CCCCC2CO)=O)n[nH]c2cccc(-c3cccc(C(F)F)c3F)c12 90104,C(=O)(CC1=CCCC1)CCC.N1(C2CN(C(C(C)N)=O)C2)CCCCC1=O 90105,C1(n2cc(-c3ncc(C)cn3)nn2)CC2CCC1(NC(=O)C(C1CCC(=O)N1)C)C2 90106,C1(C(=O)NCc2cccs2)CC12CCN(Cc1ccc(Cl)cn1)CC2 90107,N1(C(C(CC(=O)OC)C)=O)CCC(NC(C2(CC3CC3)CC2)=O)C12CCC2 90108,c1(CNC(=O)NCCC(C)N(CCC)C)sccc1OC 90109,C1(C(N2CC(N3CCN(C(C(CC)(C)O)=O)CC3)C2)=O)Cc2cc(F)ccc2O1 90110,C1(C)(CNC(c2cc(CC)no2)=O)CCN(C(C2(C)CCC(OC)CC2)=O)CC1 90111,Cc1nc2c(s1)CCN(C(=O)C(C1CCCCC1)C)C2C 90112,N1(C(c2cncc(C)c2)=O)CCCC(NC(=O)C2=CCC2)C(F)C1 90113,C(c1ccc(Cl)cc1)=CC(=O)N(C(C)CCNC(N1CC2CCC1C2)=O)C 90114,Cc1cc(NC(=O)C(CC(C)C)NC(=O)C(=O)C(C)C)c(C)cc1F 90115,N1(C(c2nc(CC)sc2N)=O)CC(NC(=O)C(c2ccccc2)F)CC1(C)C 90116,N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C)CC1CNC(=O)COCc1ccnn1C 90117,N1(C(CC)C)CCN(C(C2COCC2NC(=O)Cc2cncn2C)=O)CC1 90118,C(=O)(C(F)C(C)(C)O)NC1CN(C(C2(OC(=O)NC)CCC2)=O)C1.CC 90119,CN1CCCC1c1cc(C(=O)NC2CCC2NC(=O)CNc2nccs2)n[nH]1 90120,c1(CNCC)ccc2c(c1)OCCO2.c1(C(N2CCC(N)C2)=O)cc(O)ccn1 90121,C(=O)(C#CC1CCCO1)N(CCC(=O)N1CCC1CNC(=O)OC(C)(C)C)C 90122,n1(CC(=O)NC(C)C(C)(C)NC(=O)CN2CCOCC2)cc(CN(C)C)nn1 90123,CS(=O)(=O)c1csc(C(=O)NC2CC(C)(NC(C3CC3C#N)=O)C2)c1 90124,N1(C(c2c(CC)con2)=O)CC(NC(=O)Cn2ccc(C(F)F)n2)C(F)C1 90125,C(=O)(CC(C)C(C)(C)NC(c1ccc(Cl)cc1)=O)NC(C(=O)OC)CO 90126,CC1(C)CC(NC(N)=O)CCN(C(c2ccccc2CO)=O)C1.C12(CC1)C(=O)N2 90127,C1(CCOC)(NC(C2CCCC2)=O)CCN(C(c2ccccc2SCCO)=O)C1 90128,c1(CC)ccccc1CN1CCN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1 90129,C(C(=O)NOC(=O)C=CCF)=C.CC(C)(C)OC(=O)C=CCF 90130,c1(C(=O)NC(C(=O)NCCn2c(CC)ncc2)C2CCCC2)ccc(F)c(F)c1 90131,c1(CC(N2CCC(NC(C)=O)C2)=O)ncccc1C.C12C(C1(C)C)CNC2=O 90132,C1(NC(c2scc(C)c2)=O)C2CCC1CC(NC(=O)C=CCCC(C)C)C2 90133,C1(C(N(CCCNC(c2cc(Cl)c(F)cc2Cl)=O)C)=O)CCC2C(CC1)C2(F)F 90134,N1(C(c2n(C)ccc2)=O)CCC2CCCC12CNC(c1ccc(N)c(Cl)c1O)=O 90135,c1(C(N(C2(C)CC2)Cc2ccc(Cl)cn2)=O)nc(C(F)(F)F)ccc1C#N 90136,c1(CN(C2C(C)CCNCC2)C(=O)C(F)n2cccn2)cncc2ccccc12 90137,CCCC(C(O)C(=O)NCC1(C)COCCO1)NC(=O)Cc1csnc1C 90138,C1(C(NOC)=O)CCC(C)N(C(=O)NC2C(F)(F)C23CCC3)C1 90139,Nc1cc(C(=O)NCC2(C(F)(F)F)CCNC2)nc(C2CC2)n1 90140,c1(C(N2CC(NC(C3(OC)CCOCC3)=O)C3C2C3)=O)ccn2nccc2c1 90141,N1(C(Cn2cc(C(C)=O)nn2)=O)CCCC(NC(=O)Cc2ccnn2C)C1C 90142,C1(C(N2CCC(CC=C)(NC(=O)CCCN(C)C)C2)=O)CCC(C2CCC2)CC1 90143,c1(OC)ccc(Br)cc1C1(NC(c2coc(C)n2)C(=O)NCSC2CCOC2)CC1 90144,c1(C(N(CCCN(C)C(C2CC(F)C(=O)N2)=O)C)=O)cnc2c(c1)NC(=O)CO2 90145,C1(C(=O)NCC2(CC(N3C(C(C)(C)OC)CCC3)=O)CC2)C(C#N)C1(C)C 90146,N12CCN(CC1)C(=O)C1CCC1C(=O)NC(C)C2.C1(CF)CCCCC1 90147,C1(NC(CCC)=O)COC2(CCN(C(C)=O)C2)C1.c1(C(CO)OC(=O)O)ccccc1 90148,N1(C(C2(C(C)C)CC2)=O)CC(C2CN(C(=O)CCCOC3CCOCC3)C2)C1 90149,Cc1cnc(CNC(C2CCCN(C(C3CCCCC3O)=O)C2)=O)nc1 90150,N12CCN(CC1=O)CCC2.C1(CCOC)(C(=O)NCCOCCF)CC1 90151,C(C(C(C)C)C(C)C)NC(C1(C)CCN(C(C(C)C(F)F)=O)C1)=O 90152,C(=O)(C(CC)C(F)(F)F)NC1C(C(N(CC=C)CC2CC2)=O)C2C1C2CC 90153,C(CC(=O)NCCCOC(C)C)NC(C1CC1)C.C(=O)(C(=O)N)NCCCCC 90154,C(=O)(C1=CCCCC1C)N1CCC(CN(C(c2sc(C)c(Br)c2)=O)C)C1 90155,Cc1nc(C(=O)NCC2CCCN2C(=O)C(F)(F)c2cscn2)c(C)n1C1CC1 90156,C(c1cccnc1C)=CC(=O)NCC(CNC(c1nncc(CCC)c1)=O)OC 90157,C1(C(c2n(C)nnn2)NCc2ncnn2C(F)F)CCC2CC1C2(C)C 90158,N1(C(c2c(CC)nns2)=O)CCN(C(C2CCCN2C(=O)OC)=O)CC1C 90159,N1(C(C(COC)(F)F)=O)CC2COCCC2(NC(c2csc(C)n2)=O)C1 90160,N1(C(C=Cc2cc(OC)ns2)=O)CCC(CNC(C2CCS2(=O)=O)=O)C12CC2 90161,CC1(C)C(=O)NCC1NC(C1CC(F)CN1C(c1ncc(Cl)cc1Cl)=O)=O 90162,CCC(C)C(O)C(C)C(=O)N1CC2CC1C2NC(C1(CC=C)CC(C)=NO1)=O 90163,c1(C(N(CCN(C(C2OCCC2C)=O)CC)CC)=O)snc(Cl)c1Cl 90164,c1(C(=O)NC2C(CNC(COCC)=O)C2)ccc(C)c(F)c1N 90165,c1(OC)cc(C(=O)N(C2C3CN(C(C4CC(CC5CC5)C4)=O)CC23)C)cc(N)c1 90166,Cc1ccc(C(C)C(=O)NCC2CCC2C(=O)N(C2(CO)CCC2)C)o1 90167,c1(C(N2CCC(CN(C(c3cnc(OC)s3)=O)C)C2)=O)sc(C)nc1C 90168,N1(C(c2cn(CCC)nn2)=O)CCC(C(=O)NCC2CCCC(=O)N2)C(C)(C)C1 90169,C=CCC(CNC(c1cnco1)=O)C(=O)NC(c1cnccc1C)C 90170,C(C(O)CC(C)C)NC(C1N(C(CCC)=O)CCC1)=O.c12cn(nn1)CCS2 90171,CC(C(C(F)(F)F)n1cc(CCn2cncn2)nn1)C(C)(C)C 90172,N1(C(c2ncc(NC)nc2)=O)CC(C)(C)CC1C(N1CCC(c2cc[nH]n2)C1)=O 90173,C(=O)(C(O)CC(N)=O)N(C1CCCN(C(=O)CSc2cccnc2)CC1)C 90174,c1(C(C)C)noc2ncc(CNCC3CCCC3C#N)cc12 90175,C(N=c1[nH]c(N2CCC(CF)C2)nc2ccccc12)c1n(C)ccn1 90176,Cc1cc(C(=O)NC2CCC(CNc3ncc(I)cn3)C2)c2ccc(F)cc2n1 90177,C1(C(N2CCCC(NC(c3cccnc3)=O)(CO)C2)=O)CCc2nccn2CC1 90178,c1(C(=O)NC(CC(C)NC(CN2CC(CC)C2)=O)C)c(OC(C)C)ccnc1F 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90301,C(c1cccnc1)=CC(=O)O.C1(=O)CCCc2nnc(o2)CCN1 90302,O=S(=O)(c1ccc(N2Cc3ncsc3C2)c(F)c1)NC1CCc2c1ccc(F)c2Br 90303,c1(C(N(C)CCNC(C2CCC3(CC3)C2)=O)=O)cc2cccc(Br)n2c1 90304,c1(C(N2CC3CC(NC(=O)C(F)(F)CO)C2C3)=O)c[nH]c2cc(F)c(F)cc12 90305,N1(Cc2ccc(-c3cncc(C(=O)OC)c3)nc2)Cc2ccc(Br)cc2CC1C 90306,C1(OC)CC2N(C1)C2=O.c1(CNC(=O)CC2CN(C)C2)snnc1C 90307,C(C(C)(CC(C)C)NC(=O)CC(C)F)NC(c1ccc(C(C)C)s1)=O 90308,N1(C(C(C)(C2(C)CC2)OC)=O)CC(CO)C2(C1)CN(C(c1conc1C)=O)C2 90309,C(CCC(=O)NCC1CCCC1O)NC(COCCOCC)=O 90310,C=CCCC(F)(F)C(=O)NCCCC(C)(C)NC(C1CC(C)=NO1)=O 90311,C1(C(N(CCN(C(c2c(CC)n(CC)nn2)=O)C)C(C)C)=O)SC2C=CC1CC2 90312,c1(C(=O)NC(CNC(C2CC(C)C2(C)C)=O)(CO)CO)c(F)ccc2c1OCO2 90313,c1(C(=O)NCc2ccc(Cl)c(Cl)c2)cc2c(Cl)cc(F)cc2[nH]1 90314,N1(C(CCOCC#C)=O)CC(CNC(=O)C=C(Cl)Cl)(OC)C1 90315,C1(COC(=O)CN(CC(F)F)C(=O)C2CC2)CCCC(F)(F)C1 90316,c1(NC(CC2(NC(C3=C(C)OCC3)=O)CCC2)=O)cc(Cl)nc2ccccc12 90317,CCCCCC(=O)NCC(=O)NC1CC1c1nncn1C.C12CCCN(C1)C2=O 90318,N1(C(C(C(CC)C)O)=O)CCOCC(F)(CNC(C2(F)CC=CC2)=O)C1 90319,c1(C(=O)NCCC(C)(C)NC(C(CC=C)CC)=O)cnn2c1OCC(OC)C2 90320,C(=O)(CS(=O)(=O)C1CC1)NC1C2CC(CNC(C(c3ccncc3)C)=O)(C2)OC1 90321,C1(C(N(C)C2CC2)=O)C2CN(C(c3ccc(-c4cnc[nH]4)cc3)=O)CC12 90322,C1(C(=O)NCC(C)NC(c2ccnn2C2CC2(F)F)=O)(CC)CNC(=O)C1 90323,c1(C(=O)NCC(CC)NC(c2nonc2CC)=O)ncc(F)cc1F 90324,c1(C(=O)OCC(CC(CC)C)=O)cc2cc([N+](=O)[O-])ccc2[nH]1 90325,c1(C(=O)NCC(CNC(C2CN(C(N)=O)C2)=O)F)cc(Cl)c[nH]1 90326,CC1C(NC(=O)COc2ccc(Cn3cc(Cl)cn3)cc2)C2CCN1CC2 90327,C1(CNC(c2cc(CNC(C=CC(C)C)=O)[nH]n2)=O)CCCC(C)O1 90328,C#CCC(CC(F)F)C(=O)NCC1(CN(C(=O)C(CO)C(F)(F)F)C)CC1 90329,c1(N)nccc(OC)n1.c1(CCC(=O)NC(CN(CC)CC)C)ccsc1Cl 90330,CCC(C(=O)NC1(CC2C=CCC2)CCC1)NC(C)=O.C12(CC1(F)F)C(=O)NC2 90331,C1(NC(c2c(C)cnn2C(C)C)=O)CC(C)CN(C(=O)COC2(C)CCCC2)C1 90332,c1(CCNC(C2CC(F)(CN)C2)=O)cc(Br)ccc1C 90333,c1(CC(=O)N(C(C)(C)C(=O)C2CCOC2)C2CC2)ccnc(Cl)c1F 90334,N1(C(C2(C)N(C)CC(OC)C2)=O)C2CCC1CN(C(C1CN(C)C1)=O)C2 90335,c1(CCC)ccc(C(=O)N(CC(C)N(C)C(c2cc(C3CC3)nn2C)=O)C)cc1 90336,c1(NC(C2C=CCN2C(=O)CC(O)c2ccccc2)=O)nc(Cl)c(Cl)cc1Cl 90337,CCS(=O)(=O)CC(=O)NC1CCC(CCNC(=O)CCc2ncc(C)[nH]2)C1 90338,C1(CN(C)C(C2CCNC2=O)=O)COCCN1C(c1ccc(C(F)F)s1)=O 90339,c1(C(CC)CN(C(=O)C(=O)N(C)CC2CC(C)(C)C2)CC)ccccc1 90340,c1(C(=O)NC2CC(C)(NC(CC)=O)C2)cccc(C(C)=O)c1 90341,C(=O)(C#CC1CCCCC1)N(C)CC1CCCN1c1cc(C(C)(C)C)ncn1 90342,N1(C(C2C(C#N)CC2)=O)CCOCC1CNC(C1CCC(F)CC1)=O 90343,c1(C(=O)NCC(CN(C(CCCC=C)=O)CC)(C)C)cc(C)nc2c1cnn2C 90344,CCCCC(C(=O)NCC=CC(=O)NC1CC2OC(=O)CC12)C(C)C 90345,C1(C(N(C(CO)C2CC2)C)=O)CC(C)(C)CCN1C(c1csc(O)n1)=O 90346,CCCC(C)(O)CC(=O)NC(CCF)C(=O)N1CC(C)(C)C1C(C)C 90347,Cc1cc(-c2cnn(C3CCOC3)c2)ccc1C(=O)Nc1cccc(Cl)c1F 90348,c1(SCC2(CC(=O)NCc3c(C(=O)NCC(F)F)c[nH]n3)CC2)ccccc1 90349,C1(CC(=O)OCC)CCC2(CCC2)N(C(=O)C(C2CC(C)(C)NC2=O)(C)C)C1 90350,c1(C(N2CCN(C(=O)C(F)C3CC3)CC2)=O)ccc2nc(O)[nH]c2n1 90351,C1(CNC(C(C)(C)C(N)=O)=O)C(C2CC2)CCN1C(C12CCCCC1C2(F)F)=O 90352,CCCC(C(=O)NCC1=CCN(C(c2ccc(OC(C)C)cn2)=O)CC1)C(C)C 90353,c1(C(=O)NC2CN(C(CC(CC)O)=O)C2)cnc2c(c1)NCC2 90354,Cc1ccc(C(CNC(=O)CC(C)CF)NC(C2CCN2C2CCCC2)=O)cc1 90355,c1(-c2scc(C)n2)cccc(C(C)NCc2cn(Cc3ccno3)nn2)c1 90356,n1(CC(=O)NC2C=CC(CNC(C3CC(O)C3)=O)C2)nnnc1-c1ccsc1 90357,N1(C(C(CC=C)(C)C)=O)CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC(C)(F)C1 90358,CS(=O)(=O)C1CN(C(c2ccc(F)s2)=O)CC1NC(c1cc2sccc2s1)=O 90359,c1(C(=O)NCC(C2CC2)NC(C(N2CCOCC2)C)=O)cc(C(F)(F)F)no1 90360,Cn1ccnc1CCC(=O)NCCC(O)CNC(=O)COC1CC(F)(F)C1 90361,c1(COC)cncc(C(=O)NC2CC(C)(NC(=O)CC3CCC3)C2)c1 90362,C(=O)(CC(C(F)(F)F)n1cccn1)NCCN(c1cc(C)c(C)nn1)CCC 90363,c1(OCC)ccc(C(N2CC(N(C)C(c3coc(C)n3)=O)C3(CC3)C2)=O)cc1O 90364,c1(C(=O)OC)cnc(NCC2CC2CNC(=O)C(c2ccccc2C)(F)F)nc1 90365,c1(C(=O)NC2CCN(C(C(C(=O)OCC)F)=O)CC2)cnc2[nH]nc(O)c2c1 90366,c1(OC)ccccc1CCC(N1CCCCC1C(C)NC(=O)CCNC(N)=O)=O 90367,N1(C(C23CCC(NC(CC4CC(N(C)C)C4)=O)(CC2)C3)=O)Cc2cnn(C)c2C1 90368,C1(N(C)C(c2ccn(CC(F)(F)F)n2)=O)CCCC(NC(c2ccsn2)=O)C1 90369,N1(C(C(=O)N(CCN(C(=O)C(C)c2ccsc2)CC)CC)C)CCOCC1=O 90370,C=CCC(C)C(=O)NCCn1cc(C(=O)NCCc2cn(C)nn2)nn1 90371,C1(CNC(CCC=C)=O)CN(C(C2CCCCN2C(C2CCCC2)=O)=O)CCN1C 90372,c1(C(c2nn[nH]n2)NC(C2CCN(S(CCC)(=O)=O)C2)=O)ccc(Br)cc1 90373,C(CCC(O)C(=O)NCc1ccncc1F)NC(c1cc(OC)ncc1)=O 90374,c1(C(N(C(CCC)C(=O)NC(c2ncccc2F)C)C)=O)cccn2cncc12 90375,C(C)(C)(C(=O)N1CC(OCCC(=O)N(CC(C)C2CC2)C)C1)SC 90376,C1(C(=O)Nc2c(CC)cccc2)CC(C)(C)CCN1C(=O)CCn1ccnn1 90377,CCCC(CC)CC(=O)N1CCC(NC(=O)C(C(C)C)OCC)CC1C 90378,N1(C(=O)OC(C)(C)C)CCC(C(N2CC3C(NC(=O)C(C)C)C3C2)=O)C(F)(F)C1 90379,c1(CC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)C(C)C2=CCCC2)c1F 90380,c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CC2)=O)nc2ncccn2n1 90381,C1(C(=O)NCC(CCC=C)O)N(C(=O)CN(CC(C)(C)C)C)CC12CCCC2 90382,N1(C(c2c(C)cns2)=O)CC(O)(C2(CNC(c3cc(F)cc(C)c3N)=O)CC2)C1 90383,CCCCC(CC)C(=O)NCCCCCCC(=O)NC1CCCC1 90384,C1(C(=O)NC(CCOCC)C)COCCN1C(c1ccc(-c2cnn(C)c2)o1)=O 90385,CN1CC2C(C(=O)NCC3CN(C(C45CCC(CC4)O5)=O)CC3O)C2C1 90386,N1(C(C=C(CC)C)=O)CCC(O)(CCNC(=O)CN2CCCC(N(C)C)C2)CC1 90387,C1(NC(=O)CC2CSCCS2)CN(C(=O)CN2CC=CC2)C2(CCC2)C1 90388,C(=O)(CC(C(F)(F)F)NC(=O)C(O)C(F)(F)F)NC(c1cnn[nH]1)C 90389,N1(C(C(C2CCN(C(=O)C(F)OC(F)(F)F)CC2)C)=O)CCc2cc(C#N)ccc21 90390,N(C1CCc2cc(CNC(=O)Cc3nc(C)sc3C)ccc21)C(C1(SC)CC1)=O 90391,CC(C)C(O)CCN.c1(C2(C(c3nnnn3C3CC3)C3CC3)CC2)ccc(OCC)cc1 90392,C1(c2cccnc2)(C(=O)NC(CC(C)NC(C(CC)(C)C)=O)C)CC2(CCC2)C1 90393,C(=O)(CCC(C)(C)NC(=O)CP(C)(C)=O)N1CC(CC)SCC1 90394,C(CC(C(=O)N1CCCC1CN(C(=O)C=C(Cl)Cl)C)NC(=O)C(C)C)SC 90395,C1(C(=O)NC(CC=C)CNC(=O)C(C)CN(C)C)Cc2ccccc2C1 90396,c1(C(=O)NC2CCC(NC(c3cnc(=NC)[nH]c3)=O)C2)c2c(c[nH]c1=N)CCC2 90397,c1(C(N2C(C)(c3cn(-c4cc5c(s4)CCC5)nn3)CCC2)=O)n[nH]cc1[N+](=O)[O-] 90398,Cc1nc(C(=O)N(C(C)CCNC(c2sc(C3CCCO3)nc2C)=O)C)c(C)o1 90399,N1(C(C(CCC)C)=O)CCC(C(F)(F)F)C(NC(c2ccc(Cl)c(O)c2)=O)C1 90400,CCS(=O)(=O)CC(=O)NC1CN(C(=O)CC2CC2C(F)(F)F)CC1OC 90401,C1(O)(CCNC(c2n(C)ncc2)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 90402,N1(C(COCCOCC#C)=O)CCN(C(C2(C)CCCS2)=O)CC1CC1CC1 90403,N1(C(C(C)N(CC)CC)=O)CCCC(NC(=O)CC2(C)CCCC2)C(F)C1 90404,c1(C(N2C(CNC(C(C)SCCCC)=O)CN(C)CC2)=O)ccc(S(N)(=O)=O)cc1 90405,C(=O)(C1=C(Cl)CCC1)N1C(C(C)C)C(C(=O)NCC2(C3CC3)CCCO2)CC1 90406,N1(CC(=O)NCC2CC(F)(CNC(CC(C)c3ccco3)=O)C2)C(=O)CN(C)C1=O 90407,c1(C(=O)NCC(C2(C(N(C)Cc3ncc(C)o3)=O)CC2)C)ccc(C#N)cn1 90408,CC1CC(NC(=O)COCCN2CCCC2)CN1C(=O)CC(=O)NCCO 90409,c1(C2c3n(nnn3)C(CSC)N2)cccc(C#N)c1.C(C)(C)(C)OC(=N)O 90410,C1(C(=O)OCC)CCc2cnc(C)n2C1.C12CC3CC(CC13)NC(=O)C(=O)NC2 90411,C(CCSC)(C(=O)N1CC(CC2CC2)C1)NC(c1c(CC)nns1)=O 90412,C1(NC(C2(CC(C)C)CCC2)=O)CC2(C1)CC2NC(C12CCC(CC1)C2)=O.COC 90413,N1(C(C2CCC(C)C2)=O)CCC2(CC1)CCN(C(c1ccc(C(F)F)nc1)=O)C2 90414,C1(NC(CC2N(C(C(C)OC(C)C)=O)CCC2)=O)CCC(SCC(F)(F)F)CC1 90415,N1(C(C(CCC2CC2)OC)=O)CC(C)(C)OCC1CNC(=O)C#CC(C)(C)C 90416,c1(C(CNC)NC(=O)CCC2(O)CCC2)cccs1 90417,n1(CCNC(c2nnnn2CCC2(C)CC2)C(C2CC2)OC)ccc(O)nc1=O 90418,N1(C(C(C)N(C)C2CC2)=O)CCC(C)(C)CC1C(=O)NCCCN1CCOCC1 90419,N1(C(CC=C=C)=O)CCC(N(C)C(c2cnn(-c3cccnc3)c2)=O)CC1 90420,C=CCC(F)(F)C(=O)NCCC1CCCN(C(C2CN(C(=O)OCC)C2)=O)C1 90421,C1(C)(CNC(CCC=C(C)C)=O)CN(C(C2C3CCCCC23)=O)C(C)(C)C1 90422,C(=O)(CC(C(C)C)OCC)N(CC(CN(C(c1ccc(C#C)o1)=O)C)O)C 90423,n1(CC(N2CC(C)(C)C2C2CCN(C(=O)NC3CC3)CC2)=O)cccc(O)c1=O 90424,c1(C(=O)NC(C(C)OC)Cc2ccccc2)ccc(CCN)cc1 90425,CCCC(C)(O)CC(=O)NC1CCC(CCNC(c2nc(C)ccc2F)=O)C1 90426,Cc1ccc(NCCC(=O)NC2CN(C(C3CC(O)C3)=O)C3CC23)cc1 90427,Cc1ccc(CC(=O)NCC(C)(C)CN(C)C(c2ncccc2N)=O)c(F)c1F 90428,C(=O)(C(C)(C)C(=O)N(C)C)NCN1CCCC(C(=O)NCCc2c(C)con2)C1 90429,N1(C(=O)C2=COCC2)CCCC(F)(CNC(=O)CC2COCC2O)C1 90430,c1(C(=O)NC2CN(C(c3c(C)ncc(C)c3)=O)CC2(C)C)cnc2[nH]cncc1-2 90431,CC(C)C(F)C(=O)NCC1CCC(C(=O)NCC2COCC(C)O2)CC1 90432,c1(CC)c(C(=O)N(CCCN(C(=O)C=Cc2ccsc2)C)C)oc2ccccc12 90433,CC1CC(CN(C2CCN(NC(C=O)=O)C2)CCO)CCS1.C12(C)CC3CC1C2C3 90434,c1(C(N2CCC3C(NC(c4n(C)ccn4)=O)C32)=O)cccc2c1CCC(=O)N2 90435,c1(C2C(CC(C)C)C2)ccc(OC(F)(F)F)cc1.C12CN(C1)C2=O 90436,c1(C(N2C3CCN(C(CSC)=O)CC3CC2)=O)c[nH]c2c(F)c(F)ccc2c1=O 90437,S(=O)(=O)(c1cn(C)cn1)NC(c1nc(C(C)C)[nH]n1)C 90438,c1(NC(CN(CC(C)C)C(C2(C)CCCOC2)=O)=O)ccc2ccncc2c1 90439,N1(C(CSCCCC)=O)CCC2CN(C(c3cc(C)cc(Br)c3)=O)C2C1 90440,C(=O)(C#CC1CCC1)N(c1nncn1C)CC(=O)NC(C1(C)CC1)C 90441,C(=O)(C1=CCCCC1C)N(CCCNC(c1cc(OC)c(Cl)cc1)=O)C1CC1 90442,c1(C(N2CCC(N(C(=O)Cn3cncc3C)CC#C)C2)=O)nccnc1CC 90443,N1(C(=O)OC(C)(C)C)CCOCC(C)(CNC(=O)CN2CCCC(C)C2=O)C1 90444,C1(C(=O)NCC(CCC)NC(c2coc(C(C)OC)n2)=O)CN(C)C(=O)N1 90445,c1(C(=O)NCCn2cc(-c3cccc(F)n3)nn2)cnc2ncc(Br)cc2c1 90446,C1(C#CC(=O)N2CC(CNC(c3cc(O)cc(Cl)c3)=O)C(C)(C)C2)(CC)COC1 90447,C(C(C)(C)CC(=O)NC1CCCC1NC(c1cncc(N2CCCC2)c1)=O)OC 90448,C12(C(=O)NC3C(NC(c4nc(C)sc4)=O)C3)CCC(CO)(CC1)CC2 90449,C(=O)(C1=CCC(C(F)(F)F)OC1)Nc1ncc(C(C)SC)cn1 90450,N(C1CCOc2c(Br)cccc21)C(c1c(F)ccc(F)c1)C1CCOC1 90451,c1(C(=O)NCC(CNC(=O)C2=CCCC2)F)cc2ccccc2n1CC1CC1 90452,C1(OCCNC(CC2CC(OC)C2)=O)CCN(C(=O)Cc2ccnc(O)c2)CC1 90453,c1(CN)cnn(-c2ccccc2)c(=O)c1.c1(C2C3(C2)C(=O)N3)ccc(Cl)cc1Cl 90454,N1(C(C(CC=C)C)=O)CC(C(C)(C)C)CC(CNC(C2(n3cccn3)CCC2)=O)C1 90455,CC1CN(C(C23CC2C3)=O)C(C)CN1C(=O)C=CC1CCOCC1 90456,c1(C(=O)NC2C(CNC(C(=Cc3ccccn3)C)=O)CCC2)cc2cccnc2s1 90457,CC1CCC(C)C1NC(=O)CC1CN(C(C2CC(C(C)C)C2)=O)CC1C 90458,c1(C(=O)NCCC(C)NC(c2ccn(C3CC3)n2)=O)ccc(P(C)(C)=O)o1 90459,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCCN(C(C2=CC(Cl)=C2C)=O)CC1C 90460,C1(CC(=O)NC)CN(C(=O)C=C(C)Cl)CCN1C(=O)Cc1ccc(O)cn1 90461,N1(C(CCC(C)NC(=O)C(C)(C)C2(O)CCC2)=O)C2CCC1CC(O)C2 90462,C1(O)(CCNC(C2CC2F)=O)CCN(C(c2ncnn2C2CCOCC2)=O)CC1 90463,CCCC(CNC(C1CN(C)CCO1)=O)C(=O)Nc1cnc(Cl)cc1C 90464,CCC(C)(C(=O)N1CCN(C(=O)CCCOC(C)C)C(C2CCCC2)C1)C(N)=O 90465,N1(C(C2C(C)CC2C)=O)CCCC(O)(CCNC(=O)C=C2CN3CCC2CC3)C1 90466,c1(CN2CC(C(=O)OC)C3(C2)COC3)ccc2nc(O)cn2c1 90467,c1(OC)ccc(CN2CC3(CCN3C(c3cc(C)ns3)=O)C2)cc1O 90468,C1(C(=O)NCC2CC(C)C2)CCC2(CCN(CCn3cccc3)CC2)O1 90469,Cc1c(CCC(=O)NC(CNC(=O)CN(C)C)C(C)C)c(O)nc2[nH]nc(O)c12 90470,c1(C(C(=O)NC(C)(C)C)N(C)CC2(CCl)CCC2)cnc2c(c1)CCC2 90471,c1(C2(C(N(C(CNC(c3nc(CCC)sc3)=O)C)C)=O)CC2)ccc(C)cc1 90472,C1(C)(C(N2CCC(OCC#C)C2)=O)C=CCN1C(c1cn(C(C)C)nn1)=O 90473,C1(C(=O)NC2CN(C(=O)NC(C)C)C2)CCCCC1NC(C1(N(C)C)CCC1)=O 90474,C1(C(C(=O)NC(C)(CNC(c2ccncc2O)=O)C2CCC2)O)CCCCCC1 90475,CC(C)C(CCN(C)C(C1CC2CCC2C1)=O)NC(=O)C(N1CCNC1=O)C 90476,C=CCC(C)(C)C(=O)NC1CCCN(C(c2ccc(CC)c(Br)c2)=O)C1 90477,C(=O)(CCN(OC)C(=O)C(C)CC(C)(C)C)NCC(C)N(C(C)=O)C 90478,C(=O)(CC(C)CCc1ccccc1)NC(CNC(C1CN(C(C)=O)C1)=O)(C)CO 90479,N1(C(c2csc(Cc3nn[nH]n3)n2)=O)CC2CCC(C1CO)N2C(=O)CO 90480,C(CCC(CO)NC(=O)CC(C)(C)C)NC(c1c(C)occ1)=O 90481,c1(CC)onc(C)c1C(=O)NCCC1CC(C(=O)NCC2CCCC(C)O2)C1 90482,CCCCC(CNC(c1ccnn1C)=O)NC(c1ncccc1F)=O 90483,N1(C(CC(=O)OCC)=O)CCC2(CC1)CC(NC(=O)CC1CC1(Cl)Cl)C2 90484,N#Cc1ccc(C2CC2C(=O)NCC(C2CC2)NC(=O)CO)c(F)c1 90485,c1(C(N(C)CCNC(=O)CC2CC3CCC2O3)=O)cc(S(=O)(=O)NCCO)c[nH]1 90486,CN(C)S(=O)(=O)N1CC(C(=O)NCC2CCN2C(C2CCC2)=O)C1 90487,c1(C(N2C3C(NC(COC(CC)(C)C)=O)CC(C3)C2)=O)nc(C)n2ccccc12 90488,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(O)C2)=O)ncc(Cl)cc1Cl 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90593,C1(C(C)C)CCC(C(=O)N(C)CC2CCCCC2O)N1C(=O)CCc1ccsc1 90594,N1(C(C(C2CCCOC2)OC)=O)CCCC(C)(C)C1CNC(=O)C1=NOCC1 90595,C1(C(=O)NCC(CC=C)(C)C)CCN(C(=O)C(CSC)OC(C)=O)CC1O 90596,C1(C(=O)NCC2(C)CCCN2C(C2(C)CCC(=O)NC2)=O)SC2C=CC1CC2 90597,c1(C(C)C)conc1C(=O)NCCC(C)NC(C1CCOC1C1CC1)=O 90598,c1(C(C)NC(Cc2cccc(Cl)c2)CO)nc2cccc(Br)c2[nH]1 90599,C(=O)(CCCC(C)CC)NC(CC)C(=O)NCC1(C)CCC(C)CC1 90600,Cc1[nH]nc(C(F)F)c1C(=O)NCC1(CN(C(=O)CSc2nncs2)C)CC1 90601,C(c1ccc2occc2c1)=NC(N1CC(C)N(C(=O)OC(C)(C)C)CC1C)=O 90602,c1(NC(C=CC(=O)OCC)=O)ccc(C(=O)Nc2ccc(O)cc2I)c(Cl)c1 90603,c1(OC)cncc(C=CC(N2CCC(NC(=O)Cc3ccn(C)n3)C2(C)C)=O)c1 90604,c12ccc(c(O)c1)C(=O)N(C(=O)C=CS(C)=O)CCn1cc-2nn1.C(C)(C)OC 90605,c1(C(=O)NCCc2c[nH]c(=NCC3CC3)s2)[nH]nc2ccncc12 90606,N1(C(CC2CCN(C)C2=O)=O)CC2(CNC(=O)CN3CC=CC3)CCC1C2 90607,CC(C)(CCC#N)C(=O)NCC1(CNC(=O)CC2CCCN2C)CCC1 90608,Cc1coc(C)c1C(N1CC(CNC(=O)CCOCC(F)(F)F)C2CC12)=O 90609,c1(C(N2C(CNC(C(C)C#N)=O)CC2)=O)cc(Cl)ccc1O 90610,N#Cc1ccc(C2CC2NC(=O)COc2ccccc2F)cc1 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90749,c1(OC)ccc2c(c1)CCCC2C(=O)NCC1C=CCN1C(=O)CCC1CC1 90750,N1(C(C(CO)NC(C(C)C)=O)=O)CC(NC(c2nnc(S)n2C)=O)CC2(CC2)C1 90751,C(c1ccccc1)=C(CC)C(=O)NCCC1(NC(C2CC(C)CO2)=O)CCCC1 90752,Cn1cnc(C=CC(=O)NC2CC(NC(C3CCCC(F)C3)=O)C2)c1 90753,C(=O)(C1CCCn2ccnc21)N1C2CN(C(c3cc(C)c(Cl)cc3F)=O)C(C2)C1 90754,CCCCCC(C)(C)C(=O)NCC(C)CN(C(=O)CC1CC(O)C1(C)C)C 90755,N1(C(=O)COC2CCCCC2)CC(F)(F)CC1CNC(c1ccn2c1CCC2)=O 90756,N12CCC(C)(C1)CNC(=O)CN(C)CCSCC2=O.c1(C(C)=O)ccccc1 90757,c1(C(=O)NC(C2CCCCN2C(=O)CC2CCCC23CC3)C)cn(C)c(O)n1 90758,C#Cc1ccc(C(=O)NC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CCCC)cc1 90759,N1(C(c2cc(CC)no2)=O)CCC(NC(=O)CCCF)C(C(N)=O)C1 90760,C(Cn1cncn1)(C(=O)NOCCC(C)O)NC(C1C(C(C)C)CCC1)=O 90761,C1(CC)CN(C(=O)C(CO)NC(=O)CSC(F)(F)F)C(C)CO1 90762,c1(-c2n(C(COC)C)nc(CSC)n2)nc2ccccc2cc1Cl 90763,C(CC(C(=O)N(C)CC1CCN(C)CC1)NC(=O)CC1OCCC1(C)C)OC 90764,N1(C(C(CCC)N(C)C)=O)CCN(C(c2n[nH]cc2CC)=O)C2(CCC2)C1 90765,C(=O)(CCCCCF)NCCNC(C1(SC)CCC1)=O 90766,c1(OC(C)C)cnc(C(N2CC(CC(C)NC(C3C=CCCC3)=O)C2)=O)cn1 90767,N1(C(c2nc(CCC)oc2)=O)CCN(C(C2CCOC2C)=O)C2(CCC2)C1 90768,C1(C2C(C(N3CCC(NC(C)=O)C3)C(=O)NC)C2)COc2ccccc2O1 90769,C1(C(=O)NC(c2nc(C)[nH]n2)CO)CCCCN(C(c2cc(=O)c(O)c[nH]2)=O)C1 90770,c1(SC)cc(C(=O)NC(CCNC(C2(C(F)F)CC(O)C2)=O)C(C)C)ccc1N 90771,N1(C(C2(C(=O)OCC)CCC2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C(C2CC2)C1 90772,c1(CCC(=O)NC2CC3(C(N(CC)CC)C3)C2)c(C)nc(Br)nc1O 90773,c1(CC)cnc(Nc2c[nH]nc2C(N2CCCC(NC3CC3)C2)=O)nc1 90774,N1(C(C2(C(C=C)=O)CC2)=O)CC=CC1OC1CCN(C(=O)C2CC2)C1 90775,C1(C(=O)OC)CCN(C(c2ccc(OC)c(OCC(C)C(F)(F)F)c2)=O)CC1O 90776,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCC(C)(NC(=O)CCC2CCCO2)C1 90777,CC(C)C1=CCC(C(N2C3CCC2(CNC(c2ccccn2)=O)CC3)=O)CC1 90778,N1(C(CC=C)=O)CCC2(CCC2NC(=O)C=C2CCSCC2)CC1 90779,Cc1nccn1C(C)C(=O)NC1CCCC1NC(=O)CCN(C1CCCCC1)C 90780,CN1CC(C(=O)NCC2COCC2NC(c2cn(CC(N)=O)nn2)=O)CCC1=O 90781,c1(C(N2C(CC(=O)NCC3(C#C)CCC3)CCC2)=O)ccc(OC)cc1Cl 90782,c1(C(N(C(C(=O)NCC2(C=C)CCC2)C)CC2CC2)=O)c(C)[nH]c(C)c1C 90783,S(=O)(=O)(c1cncc(Br)c1)N1C(C(=O)Nc2cc(Br)nc(Br)c2)COCC1 90784,C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(C2CC(O)C2)=O)C1 90785,Cn1nc(C(=O)NC2CCCN(C(C3(C(=O)OC(C)(C)C)CC3(C)C)=O)C2)cc1Cl 90786,c1(C(=O)NC(CCC2(NC(=O)OCC=C)CCCCC2)=O)cnnc(C)c1C 90787,C1(C(=O)N2CC(c3ncccn3)C2)CC(F)CCN1C(c1cncc(Cl)c1)=O 90788,n1(CCC)cnc(N(C)Cc2cc(C)no2)c1 90789,c1(CC(N2CCN3CCCCC3C2)=O)cc(C(F)(F)F)n2ncnc2n1 90790,c1(C(=O)NC(C(=O)NCCC(C)O)C2CCOC2)c[nH]c2ccccc12 90791,c1(NC(COC2CCCN(C(C(CCC)NC(C)=O)=O)C2)=O)ccc(Cl)c(Cl)c1 90792,C(=O)(C(C)C(C)NC(=O)C=CC(C)C)NCC(=O)NCCOCCOC 90793,CC(C)C(CC(=O)NC1(C(N)=O)CCCCC1)NC(C1CCC2(CCC2)C1)=O 90794,N1(C(COCC(=C)C)=O)CCC(N(C(=O)CSCCC(C)C)C)C(C)C1 90795,c1(C(=O)NC2CN(C(=O)C(F)C3CCOC3)CC2O)ccc(F)cc1[N+](=O)[O-] 90796,N1(C(C(C)CC(N)=O)=O)CCC2CN(C(c3cc(CO)on3)=O)CC2CC1 90797,CC1CN(C(C23CCC(CC2)OC3)=O)CCC1NC(=O)C(C)(C)c1nncn1C 90798,C1(C(=O)Nc2ccnc(Cl)c2Br)Cc2cc(O)ccc2CN1Cc1cnc(Br)s1 90799,C(=O)(C#CC1CCCCC1)N1CCC(C)(NC(C(CCCC)ON=C(C)C)=O)CC1 90800,C1(NC(COCC(N2CCCC2)C)=O)C2CN(C(C3(F)CC=CC3)=O)CC12 90801,N1(C(C2(N(C)C)CCC2)=O)CCCC(C)(C(=O)NCc2ccccn2)C1 90802,N1(C(c2cc(C)c(C)s2)=O)C(C(=O)N(C2CCCCCC2)CCO)CC2CCCCC12 90803,N1(C(C2C(C)C2C)=O)CCC(CC(=O)N(C2(CO)CC2)C)C1 90804,c1(C(N2C(CNC(c3c(C)cno3)=O)CCCC2)=O)c(O)nnc2c1CCCC2 90805,Cc1ccc(CCC(=O)NC2CC2NC(c2c(C)noc2N)=O)cc1C 90806,C1(CNC(CNC=O)=O)CN(C(c2cnc3ccnn3c2)=O)C2CCCCC12 90807,N1(C(C2C(C)CCCC2)=O)CC2CCN(C(c3cn(C)[nH]c3=N)=O)CC2C1 90808,Cc1cc(=O)n(C)cc1C(=O)NCC1C(CNC(=O)C=CC2CCCN2C)C1(F)F 90809,c1(NC(C2C(NC(C3C(C)(C)C3(C)C)=O)COCC2)=O)ccc(O)cc1F 90810,c1(NCC(N2CCN(CC)CC2)(C)C)ccc(S(=O)(=O)NC)cc1C#N 90811,c1(C(=O)NC(CNC(c2c(C)nc(CC(C)C)s2)=O)C2CC2)cn2c(n1)CCC2 90812,c1(S)nnc2n1CC(CC)CC2.c12ccc-1cc2F.N1(CC)CCSCC1 90813,Cn1ncc(C(=O)NCc2occc2C(N2C(CO)CC2C)=O)c1N 90814,c1(C(N2CC(NC(C(CC=C)OC)=O)C(O)C2)=O)cccc(OC)c1F 90815,C(=O)(C(C)CCCC(C)=O)NC(CCCNC(c1c(C)nn(CC)c1Cl)=O)C 90816,c1(C(N2C3CN(C(c4nc(C)n(C)n4)=O)C(C3)C2)=O)nc2nccc(C)n2n1 90817,C(=O)(C1=CCCCC1C)NCc1ccc(C(N2CC=C(C)C2)=O)cn1 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90835,c1(OC(C(C)(O)C2CCCCC2)=O)cc[n+]([O-])cc1 90836,O=C1CCc2cc(CSc3nccc(O)n3)sc21 90837,C1(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccc2O)C12CCC2 90838,N1(C(CS(CC)=O)=O)CC2(CCC(NC(=O)C(c3cccs3)SC)CC2)C1 90839,C1(NC(c2c(C)cco2)=O)CCC2(CCCN2C(c2cccc(Cl)c2F)=O)CC1 90840,N1(C(CCCSCCC)=O)CCCCC1c1cn(-c2cnccc2C(=O)O)nn1 90841,C1(N(C(=O)CC2CCS(=O)(=O)C2)CC)CCCN(C(c2cc(C)[nH]n2)=O)CC1 90842,Cc1cc(NC(C(C)NC(c2cnn3cnccc23)=O)C(C)C)ncc1[N+](=O)[O-] 90843,C(=O)(C1=C(Cl)CCCC1)N(CC(CC)NC(c1cc(Cl)ccc1C(C)C)=O)CC 90844,c1(OCCN(NC)C)cccc(Cl)c1.C1(C=O)CC1 90845,c1(C(c2nnnn2C)NCC2(OC)CCCSC2)cnc(N(C)C)cc1Cl 90846,N1(C(c2c(C)nn[nH]2)=O)CCNC(C(N2CCCC(C(=O)N(C)C)C2)=O)C1 90847,CCCCCC(O)CN(C(=O)COC1(C)CN(C(=O)CC2CCCC(O)C2)C1)CC 90848,C1(C(N(CCC)CCNC(C2C3CCCC23)=O)=O)CCCCC12OCCO2 90849,c1(C(=O)NC2CN(C(c3cnc(Cl)[nH]3)=O)CC2F)cc2cc(F)cc(F)c2[nH]1 90850,C1(NC(C(C)Cc2cnc[nH]2)=O)CCCCCN(C(c2ccc(CO)nc2)=O)C1 90851,c1(C(N2CCC(NC(c3ccn(C)c3)=O)C(F)C2)=O)cn2c(n1)COCC2 90852,CN(C)N=Nc1ccccc1C(=O)NCC1CC(C)(C)CN1C(C1CC(O)C1)=O 90853,c1(C(=O)NC(C(CO)NC(c2c(CC)scc2)=O)C)cc(F)cc2cc[nH]c12 90854,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NC1CC(SC)C1)CCN(C)C 90855,c1(C(=O)NC2(CN3CCN(C(C(N)=O)=O)CC3)CC2)cnn2cccc(Cl)c12 90856,C(=O)(CCCCCF)N(CC)CC1CCN(C(C2CCCS2)=O)CC1 90857,N1(C(c2c(CC)n3c(n2)CCCC3)=O)CCC(C2CCCN(C(=O)OC)C2)CC1 90858,c1(C(=O)NC(CC=C)CNC(=O)C(C)CC2CC2)cnn2ccnc(C)c12 90859,C12(C(N(CC(C)(C)C)C(C#C)C3CCC3)=O)CCCC1N(C(=O)CC1CSC1)CC2 90860,C12(C(=O)NC(c3ccsc3)(C)C)CC(CO1)N(C(=O)CCn1ccnc1)C2 90861,c1(OCC)cccc(C)c1CC(=O)NC(C)CN(CC(c1ccccc1)OC)C 90862,CCN=C(NCCN1CCOC(CF)C1)NC1CCOC1 90863,C1(CNC(CCC=CCC=C)=O)CCN(C(c2cnc(CC)s2)=O)CC1C 90864,N1(C(c2cc(C(=O)OCC)sc2C)=O)CCC2C(C1)CN2C(c1cnsc1C)=O 90865,Cc1ccc(Cl)c(NC(=O)C(C2(N3CCCC3)CCC2)C2CC2)c1 90866,c1(C(N2CCC(NC(C(CC)O)=O)CC2)=O)c(Br)sc(C)c1C 90867,c1(-c2n(C(CC)C)nc(-c3ccnn3C)n2)cc(Cl)cc(C#N)c1 90868,N1(C(COCCCC)=O)CCCC(NC(=O)C(C)N2CCC2)C1 90869,C1(CC(=O)NC(C2CCOC2)C#C)CCCN(C(=O)Cn2ccc(C)n2)CC1 90870,C(CCC(C)C)(C(=O)N(C1CCCN(C(=O)CC2(C)CC2)C1)C)NC(C)=O 90871,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)CC2(C)C)ccc2c(c1)CCC2 90872,C(=O)(C(CC(C)C)ONC(=O)CC1CC(F)C1)NC1C(CCOC)C1 90873,C123CCCC1CC2(CC)CC(COCCO)C(=O)N(C)CCCNC3=O 90874,CCC(C)(C(=O)NC(c1ncn(C)n1)C)N(C(=O)Cc1cnn(CC)c1)C 90875,c1(NC(C2CC(C)CN2C(=O)CCc2ccc[nH]2)=O)ccc2c(c1)OC(F)(F)O2 90876,C(c1ccc(-c2nn[nH]n2)cc1)=CC(=O)Nc1ccc(I)cc1Cl 90877,N1(C(c2c(SC)cccn2)=O)CC(NC(c2csc(C)c2)=O)CCC1C 90878,c1(CNC(=O)C(F)CC2CC2)cc(C)c(C(=O)NCc2scc(C)c2)o1 90879,c1(C(=O)NC2CCC23CN(C(C2CCC(C(N)=O)CC2)=O)C3)cnc2[nH]nnc2c1 90880,CCCCCCC(CC)C(=O)NCC1CN(C(C2(CCO)CC2)=O)CCC1(F)F 90881,c1(NCCOC2CN(C(c3c(OCC)nc(C)cc3)=O)C2)c([N+](=O)[O-])cnn1C 90882,CCCC(CNC(C1(NC(=O)COCC(=O)NC)CCOC1)=O)CCO 90883,C1(C2CC2)(CNC(c2nn(C)c(C3CC3)c2)=O)CN(C(=O)C(F)F)C1 90884,Cc1ccc(Br)cc1C(N1CCC(F)(C(N2CCC(F)C2)=O)C1)=O 90885,c1(C(N2C(C(N(CC#C)CCO)=O)CC2C)=O)coc2c1COC2 90886,C1(NC(=O)CC2CCC2)CC2CC1CN(C(c1coc(Sc3nncs3)n1)=O)C2 90887,c1(C(=O)NCC2C3CN(C(c4c(C)cc(C)[nH]4)=O)CC32)cc2c(ccn2C)s1 90888,N1(C(C(C)S(C)(=O)=O)=O)C(C(=O)NC(c2ccccc2)CF)C2CC(O)C1C2 90889,CCC(CC1CCCC1)C(=O)N(CC(O)CNC(c1c(C)[nH][nH]c1=N)=O)C 90890,c1(C(N2CC(C)N(C(c3ccc(Cl)o3)=O)CC2)=O)ccc2c(c1)NC(=O)C2 90891,N1(c2c(C)non2)CC(C(N2CC(NC(=O)COCC(C)(C)C)C(C)C2)=O)CC1=O 90892,N1(C(c2cc(-c3cccnc3)[nH]n2)=O)CCC2C1CCCN2C(C1CC1F)=O 90893,c1(CNC(c2n(CCOC)ncc2Br)=O)ccc(Br)c(OCCO)c1 90894,CC(C)CCC(=O)N1CC(CCNC(=O)Cn2cc(C(C)=O)nn2)C(C)C1 90895,N1(C(C(C)NC(C2CCCC2)=O)=O)CCN(C(=O)Cn2nccn2)CC(O)C1 90896,c1(C(N2CCN(C(CC3(C=C)CC3)=O)C(CF)C2)=O)csc2cccnc12 90897,C1(NC(c2c(C)cno2)=O)CCC2(C1)CN(C(=O)Cc1cccs1)C2 90898,C1(NC(=O)Cc2ccsc2)CC12CCN(C(=O)CC1(c3ccon3)CCC1)CC2 90899,N1(C(CC2C(C)(C)C2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCCCC2 90900,CS(=O)c1ccc(CC(=O)NC23CC2CN(C(c2ccc(C4CC4)o2)=O)C3)cc1 90901,CC(C)CC(CNC(=O)CC(C)(C)C(F)F)C(=O)NCC(C)(O)CN(C)C 90902,c1(C(=O)NCCC(C)C)n[nH]c2ccc(-c3ccc(-c4cncs4)cc3)cc12 90903,N1(C(C(=O)NC(C)C)=O)CC2(CCC2NC(C2CCOCC2(C)C)=O)C1 90904,c1(C(C)NC(=O)COC2CCN(C(=O)C(C)(C)CF)C2)ccc(C#N)cc1 90905,CCCCCC(O)C(=O)NC(C(=O)NCc1cc(C)ns1)C1(O)CCC1 90906,N1(C(C2(CC#C)CCOCC2)=O)CCC(CNC(c2cn(C)cc2C)=O)C(C)C1 90907,Cc1nc(C)c(C(N2CCC(C)(CNC(C3CCC3(C)C)=O)C2)=O)nc1C 90908,C1(C(N(CCCOC)C2CC2)=O)(NC(c2cc(C)cc(C)c2)=O)CCC(C)(C)C1 90909,Cc1nn(C)cc1C(O)C(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1C 90910,c1(NC(C(c2ccc(OCC)nc2)N(C2CCC2)C)=O)cc(C(F)(F)F)cc(F)c1 90911,c1(CCC(=O)NC(CNC(=O)COC2CCCOC2)C2CC2)ccc(F)c(F)c1 90912,C1(F)(CNC(C2(N(C)C)CCC2)=O)CCC(NC(=O)C(=O)NC2CC2)C1 90913,C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1c(OC)c(Cl)ccc1)C 90914,c1(CNC(C2C(C(=O)NCC(C(C)C)(C)F)CCO2)=O)cc(O)cc(F)c1 90915,Cc1cc(C)n(CC(=O)N(CC(CO)(CO)NC(c2cn[nH]c2)=O)C)n1 90916,Cc1cc(C(=O)Nc2cnc(Cl)c(C)n2)ncc1C1=CC(C)(C)CC(C)(C)C1 90917,CN1CCN(CC(=O)NCC(C)(C)NC(=O)C(F)=C(C)C)CC1.c12ccc(cc1)o2 90918,C1(OC)CC(NC(N2CCN(c3cccc(C(F)(F)F)c3)C(=O)C2)=O)C12CCC2 90919,C1(NC(=O)COc2ccc(Cl)cc2)CCN(C(C2CCOCC2)=O)CCC1CO 90920,C(=O)(C1=CCCSC1)NC(C(C(=O)NCCN1CC=C(C)CC1)C)C 90921,C1(C)(SC(SC(C(=O)OC)C2CC(c3cccnc3)C2)=S)CC=CCC1 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90939,c1(C(=O)NC2C(C)CN(C(C3(n4ccnn4)CC3)=O)CC2)cnc2ccc(F)cn12 90940,N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC#N)CC1C(C)C 90941,C=CCCCC(=O)N1CC(CNC(c2cncn2C(C)C)=O)CC1C 90942,N1(C(C2(CC)CCC2)=O)CCC(CNC(c2ccnc(Cl)c2Cl)=O)C(C)C1 90943,C=CCC(CC(=O)N1CCCCC1CC)NC(c1cnc(C)nc1)=O 90944,c1cnc2ccc(-n3nc(-c4ccsc4)nc3Cc3cccnc3)cc2c1 90945,N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(C2(CC(F)F)CCC2)=O)C2CC12 90946,C1(C(N(C)CC2CCN(C(=O)CN(S(C)(=O)=O)C)C2)=O)CCCC(F)(F)C1 90947,N1(C(=O)Cc2cnsc2)CC2CCC1CN2C(=O)Cc1cc(C2CC2)no1 90948,c1(C(N2CCCC(N(C(=O)C(O)CC(N)=O)C)C2)=O)cc2cnccc2[nH]1 90949,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cncnc2)ccc(C)c(C)c1F 90950,C(CC(C(=O)NC1(C)CCN(C(=O)CN2CCC(NC=O)CC2)C1)N(C)C)SC 90951,C12(C(N(C)CCNC(=O)CSc3cccc(F)c3)=O)CC3CC1C2C3O 90952,C#CCC(C)(C)C(=O)N(CCC(C)NC(c1ccccc1OC(C)CC)=O)C 90953,c1(C(=O)NC2CN(C(c3cc(C)nn3C)=O)CC2(C)C)nn2c(c1C)CCCC2 90954,C(=O)(C(C)(C)CNC(=O)C(C)CO)NCc1nc(OC)oc1 90955,CC1(C)CN(C(=O)C=CI)CC1C(=O)NCC1(F)CCCCCC1 90956,N1(C(c2cc(C)n(CCO)n2)=O)CC(NC(C2COC(=O)C2)=O)CC12CCC2 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90974,C1(C)(CC)CC(NC(=O)Cc2ccsc2Br)CN1C(=O)CC(C)C 90975,N1(C(CCOCCCOC)=O)CCCC2(CCC(NC(C3CC4(CSC4)C3)=O)C2)C1 90976,c1(CNC(C2(NC(C(C3CCOC3)C)=O)CC(O)C2)=O)ccc(C#N)o1 90977,CCCCS(=O)(=O)CC(=O)N1CCCC2CN(C(c3cc[nH]c3C3CC3)=O)CC12 90978,CC(CC(=O)N1CCC(CCNC(c2conc2C2CCCO2)=O)CC1)C(F)F 90979,c1(Cc2cc(C(=O)NCC(C)(CO)NC(CC=CC=C)=O)on2)ccccc1Cl 90980,C1(CC(N2CC(CCN(C)C)C2)=O)C2CCCC2N1C(c1ccc(C(F)F)o1)=O 90981,N1(C(C=CC)=O)CCCC2CCN(C(c3cn4c(n3)COCC4)=O)CC12 90982,C1(CNC(C2(CC#C)CCOCC2)=O)CC(C)(C)CN1C(c1cnnc(C)c1)=O 90983,c1(NC(=O)NCC2COC3(CO)CC2C3)c(C(F)(F)F)nc2n1CCCC2 90984,N1(C(c2c(C)nncc2)=O)CCC(C2CC(NC(c3cnc(Cl)s3)=O)C2)C1 90985,C#CC1(C(=O)NCCCN(C)CC)CN(C(=O)C(C(C)C)OCCOCC)C1 90986,Cc1cc(C)c(C(=O)NCCCC2CCCCN2C(=O)C(c2ccnn2C)O)o1 90987,C(=O)(C(CC(C)(C)C#N)N1CCN(C)C(=O)C1C)NCCCCC 90988,CC(C)(C)CCC(=O)OCCCOC1CCN(C(=O)Cc2cccc(F)c2)CC1 90989,C1(C(=O)NC(C=C)C2CC2)C2CCC(C2)C1NC(c1cnc(C)o1)=O 90990,c1(NC(C(C)C)CCNC(C2CCCC2C(C)C)=O)cc(C#N)cc(Cl)n1 90991,C1(C(CNC(CC2N(CCC)CCC2)=O)(C)C)CCCCN1C(=O)COC 90992,CC1CCN(C(c2cc3ccsc3[nH]2)=O)CCN1C(=O)Cn1cncn1 90993,c1(C(=O)NCC2C(C)CCCN2C(=O)CC23CC(C2)C3)cc(F)cc(N)c1F 90994,c1(C(N(C2CCN(C(=O)COCC3CCOC3)CC2)C)=O)cccc2sccc12 90995,c1(NC)c(C(=O)NC2CC(NC(C3CCCC3O)=O)C2)cc([N+](=O)[O-])cc1Cl 90996,c1(OC)ccccc1C=CC(=O)NC1CCCCC1NC(=O)CSC(F)F 90997,CCC(CC)C(C)C(=O)NC12CCOC(CNC(c3cc(Cl)cnc3O)=O)(C1)C2 90998,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 90999,C1(OC)CCCC(C(=O)NCc2cc(C(=O)NCCC(C)(C)N(C)C)no2)C1 91000,CCCC(CCCNC(C1CCC(=O)O1)=O)NC(c1sc(C)cc1C)=O 91001,Cc1ccc2[nH]c(=NC(CNC(=O)CSc3ccc(O)cc3)CC(C)C)sc2n1 91002,C(=O)(CC(O)CC(C)(C)C)NC1C(C)N(C(c2ccc3nn[nH]c3n2)=O)CC1 91003,N1(c2cc(C)nc(CO)n2)C2CCC1CC(CNC(c1cc3c([nH]1)CCC3)=O)C2 91004,CCCC(C(=O)NC1CCCC(NC(c2ccc(N)c(SC)c2)=O)C1)S(N)(=O)=O 91005,C=C=CC(C)C(=O)N(CCCN(C)C(c1ccn(-c2ccc(F)cc2)n1)=O)C 91006,C1(NC(C(C2CCCCCC2)C)=O)C2CC1N(C(=O)COCc1nc[nH]n1)C2 91007,CCCCCCC(F)C(=O)N1CCC(N(C(=O)CC2(O)CCOC2)CCC)CC1 91008,N1(C(c2cn(-c3cnn(C)c3)nn2)C(=O)NC(C(=O)OC)C)CCCCCC1 91009,c1(SCC(=O)NC2(C)CC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)ccc(C#N)cc1 91010,c1(C(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91011,c1(NC(C2CC(=C)CN2Cc2cc(C)[nH]c2C)=O)ccc(Br)cc1OC 91012,CCC(C)CCC(O)CC(=O)N1CCC(C)(C)C(CNC(C2(F)CCCC2)=O)C1 91013,C12(CNC(Cc3cccc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91014,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C4)=O)C3)cn12 91015,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2ccc(CC)[nH]2)=O)C1C 91016,c1(OC)ccc(C(=O)NC2CCC(NC(=O)C=Cc3ccco3)C2)nc1Br 91017,c1(NC(CCC)C2CCC2)[nH]c(=NCC23CCC(CC2)CC3)nc2c1ncn2C 91018,CS(=O)(=O)CCC(O)C(=O)NC(CNC(=O)CCOCC(F)F)CC(F)(F)F 91019,N1(C(C2CC(C)OC2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91020,CN=c1[nH]c(=NCc2cc(SC)ccn2)[nH]c(=NC2CC(n3ccnc3C)C2)[nH]1 91021,C(CNC(=O)NC1C2CC(C(=O)OC(C)(C)C)CC12)(C(F)(F)F)N(C)C 91022,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(Cc2c(CC)con2)=O)C1(C)C 91023,N1(C(c2c(CN(C)C)cco2)=O)CCCC2(CCCN2C(=O)Cc2ccon2)C1 91024,C(=O)(CCCCCn1ccnn1)N1CC2C(C1)CN2.N1(CC)CCC(C(N)=O)C1 91025,N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC12CCN(C(=O)C=C1CCOCC1)C2 91026,N1(C(C2CC(C)(C)OCC2)=O)C(C(=O)N(CCO)CCO)C2CC(O)C1C2 91027,C(=O)(C1=CC2CCCCCCC12)NC1C(C)(C)CN(C(=O)C=CC2CCCO2)C1 91028,N1(C(c2ncc(NC)nc2)=O)CCN(C(=O)CNC(=O)C(C)CC)C2COCC12 91029,c1(C(=O)NCC(CC=C)NC(c2ncn(C)c2C)=O)cnc2ncnn2c1C 91030,c1(CCCC(=O)NCCN(C(C2(F)CCOCC2)=O)CC)ccccc1F 91031,C1(CC(=O)NC2CC3CN(C(C(CC)C)=O)CC32)CCCC2(CCC2)O1 91032,c1(CC)c(C(=O)NC2CCN(C(C3CC34CCCCC4)=O)C2)cnc2ncnn12 91033,C=CCN=C(NCC1CCN(CC)C1)N(C)CC1CCCS1(=O)=O 91034,c1(C(=O)NC(C)C(C)NC(c2cnc3sccn23)=O)ccc(S(=O)(=O)CF)nc1 91035,Cc1nc(C=CC(=O)NCC(CO)NC(=O)C=Cc2nnn(C)n2)cs1 91036,Cc1cnn(C(C)C(=O)NCC2CC(F)(CNC(c3cnn(CCO)c3)=O)C2)c1 91037,N1(C(C2(C#N)CC2)=O)CCC(N(CCO)Cc2ccccc2)CC1 91038,C1(C(=O)Nc2c(OC)c(C)sc2)CN(C(=O)OC(C)(C)C)CC12CC2.C12CN1C2 91039,c1(OC)ccccc1CCNC(=O)COC(C1CC(c2ccc(Cl)cc2)C1)=O 91040,c1(OC)ccn2ncc(C(=O)NC(C)C(CO)NC(c3ccccc3F)=O)c2c1 91041,CCC(CC)(CCNC(=O)C(C)(CC)OC)NC(=O)CSC(F)(F)F 91042,C(=O)C(CC(C)C)N(CCCCCOC(F)F)CC1CCN1C.CS 91043,C(=O)(CCCCCC(C)O)NCC1N(C(c2ccc(C=C)cc2)=O)CCC(C)C1 91044,C1(C)(NC(C=C(CC)CC)=O)CCCN(C(C2CC2c2cnnn2C)=O)C1 91045,N1(C(c2cc(OCC)ncc2)=O)CCN(C(=O)CN2CCS(=O)CC2)CC1CO 91046,CC1CN(C(C2(C)CCCN2C(c2ccc(C(F)F)o2)=O)=O)CC1N=[N+]=[N-] 91047,C12CCN(C(C3CC3)C1)Cc1cnc(s1)C(=O)N2.c1(OC)ccccc1C(C)C 91048,Cc1nn(CC(=O)NC(C2(O)CN(C(C3CC(=C4CCC4)C3)=O)C2)C)c(=O)n1C 91049,C1(c2nnnn2C)(NCCOC)CC(C)CCO1 91050,C12CCC(CC1)N2CC.N1(CC)CCOCC1C1CCC1 91051,N1(C(c2cccc(C)c2Cl)C(=O)NC)CCCC2(CC1)CNC(=O)C2 91052,N1(C(CCC#CC)=O)CCN(C(=O)COc2cccc(C)c2)C(C2CCCC2)C1 91053,Cn1nc(C(F)F)cc1C(=O)NC(c1ccccc1)CNC(C1CC2CC1CO2)=O 91054,C(=O)(CCC[N+](=O)[O-])N1CCC(C)C1CNC(=O)Cc1csc(C2CC2)n1 91055,c1(C(N(CCN(C(CN(CCC#C)C)=O)C)C)=O)cnn(C)c1CCC 91056,c1(CN(C)Cc2cn(C)nc2-c2cnn(-c3ccccc3)c2)ncc2ccccn12 91057,c1(N2C(CNC(C(C)C3CC3)=O)CCCC2)ncnc2sccc12 91058,N1(C(C(C(CC)CC)F)=O)CCC2(CCN(C(c3cccc(F)c3)=O)C2)C1 91059,c1(N(C)CCC2CSCCO2)ccc(S(=O)(=O)N2CC(SC(F)F)C2)cc1Cl 91060,C(=O)(C1=CCCSC1)NC(c1c(CC)cccc1)CNC(=O)C(F)OC 91061,c1(NC(C2NCCN(c3nc(C)c(F)cn3)C2)=O)cc(F)c(C)c(Br)c1 91062,c1(CN(C2C3(CN(C(CN(C(C)=O)C)=O)C3)CC2)C)cccc2c1OC(F)(F)O2 91063,CC1CCN(C(=O)CN2CCNC(=O)C2)C(CNC(=O)CC(O)C2CCCC2)C1 91064,N1(C(C(C)=C(CC)C)=O)CCC(NC(c2ncnc(OC)c2OC)=O)CC1C1CC1 91065,C(=O)(C(C)(C)C(C)NC(c1sccc1C)=O)N(CCCCCOC)C 91066,c1(CCN2C(CNC(CNC(C(C)(C)C)=O)=O)CCCC2)ccc([N+](=O)[O-])cc1 91067,C1(C(=O)NCc2cnc(C)nc2)C2CC3C(C2NC(=O)CCCF)C13 91068,C=CC(C)(O)CC(=O)NC1CCN(C(=O)C(F)(F)CC2CC2)CC1C 91069,c1(-n2cc(NCCSC3CC3)nn2)ccc(NS(CC)(=O)=O)cc1 91070,c1(CN(CCC(=O)NCc2cc(C(N)=O)sc2)CC2CCCO2)nccnc1N 91071,c1(-c2nn(-c3cscc3)c3c2CCC3)ccc2cn(-c3ccncc3)nc2c1 91072,CC(C)(C)C1=NOC(C(N2CC(C)(C)OCC2CNC(=O)C2=CCCCC2)=O)C1 91073,CCCCC(CNC(c1ccc(OC(F)F)cc1)=O)NC(=O)CC(CC)OC 91074,N1(C(C(CCN(C)C)O)=O)CC(F)(F)CC1C(=O)Nc1cccc(O)c1 91075,C(CCCCC(=O)N1CCCC(N(C)C(C2(C)CCCNC2)=O)C1)OC 91076,C1(C)(C(N2CC(CNC(C3(CCCC)CC3)=O)C2)=O)CCOC(C)C1 91077,C1(NC(C(C)SC(C)C)=O)CCCCN(C(=O)COCc2ccccc2O)C1 91078,C1(O)(CC)CCCN(C(C2(OC)CCN(C(=O)C#CC(C)(C)O)C2)=O)CC1 91079,c1(C(=O)NCC2CCN(C(CC(C)(C)OC)=O)CC2)cccc(C)c1C#N 91080,C1(CC(=O)N(CC(CNC(C2C(CC(C)C)C2)=O)C)C)CCC(=O)C1 91081,C1(C(=O)NC(C2CCCC2)CC)CCN1C(=O)CNC(N)=O 91082,C1(CC=C)(NC(c2nccn2CCOC)=O)CCN(c2nnc(C#N)s2)C1 91083,C(CCC(=O)NC(C(C)C)C1(c2ccccc2)CCC1)OCCC 91084,c1(CN2CCOCC(NC(CC(=O)OC)=O)C2)cc(C)c(OC)cc1C 91085,N12CC(CC(C)(C)C1)Nc1ccccc1OCC2=O.CCS(=O)(=O)OC(C)C 91086,c1(N2CCC(N3C(CC)CCCC3)C2)nc(COC)nc(C)c1Br 91087,C1(NC(C2C=CCC2)=O)CC1C1CCCN(C(c2ccc3occc3n2)=O)C1 91088,c1(N2C(CN3CCN(C)C(=O)C3)CCC2)nc(=NC2CC2F)[nH]c2cccc(F)c12 91089,C1(NC(C(N2C(=O)CCC2=O)C)=O)C2CC1N(C(N)=O)C2.C12(CC1)C(=O)N2 91090,C1(C(=O)NC(C(=O)NCCCN(OC)C)(C)CO)CC(C2CC2)=NO1 91091,N1(C(C)C)CCN(C(=NCc2nncn2C)NCc2ccc(F)cc2F)CC1=O 91092,N1(C(C2N(CC)CC2)=O)Cc2n[nH]cc2C1C(=O)N(CCC=O)OC 91093,N1(C(COCCOC)=O)CC(O)CCC1C(=O)NCCCS(C)=O 91094,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(c2ccccc2Cl)=O)CC(C)C1 91095,CCC(O)CC(=O)NCCCCCN(C(=O)C(c1ncccc1C)(F)F)C 91096,c1(C(=O)NCC2CCN(C(=O)COC3CCOCC3)C2)cnc2[nH]cnc2c1 91097,C(C(CNC(=O)Cn1ccc(C)cc1=O)S(C)(=O)=O)NC(C1(OC)CCC1)=O 91098,C1(=O)CCCC(=O)N1.C1(C(=O)NC)CC(F)(CCCN(C)C(=O)OC(C)(C)C)C1 91099,c1(N(C)C)ccc(C(=O)NCC2(CO)CCN(C(C3(C)C=CCCC3)=O)C2)cn1 91100,c1(C(=O)NC2CC(NC(=O)CC3CC3)C2)cc2cc(F)ccc2[nH]1 91101,Cc1cc(C(=O)NC2CC(CCNC(C3(CO)COC3)=O)C2)c(C)c(C)c1 91102,C12(C(=O)NCC(C)(C)NC(c3c(C)c(O)ccc3)=O)CCCN1CC(O)C2 91103,N1(C(C2CCC(NC(C(CC)C(=O)OC)=O)C2)=O)CCC(F)(F)C(C)C1 91104,c1(OC)c(C#N)ccnc1CNCc1cccnc1NS(=O)(=O)CCCl 91105,N1(Cc2c(OC)cccc2Br)CCOC2(CCS(=O)(=O)C2)C1 91106,Cc1cc(C(=O)N(C)CC2CCCN(C(C3CCC3C)=O)C2)cc(O)c1 91107,c1(C(N2CC(CCCCNC(COC(C)C)=O)C2)=O)ccc2ncnc(O)c2c1 91108,Cc1cc(=O)c(C(=O)NC2(C3CCCN3C(C3CCCC34CCC4)=O)CC2)c[nH]1 91109,N1(C(C(C)O)=O)CCC(C2(O)CN(C(C3CCC4(CCC4)CC3)=O)C2)CC1 91110,C1(NC(C(CN(C)C)O)=O)CN(C(c2ncc[nH]2)=O)CC(C)(C)C1 91111,N1(C(C=C(C)C(F)F)=O)CCCC2CN(C(c3cc(Cl)ccc3F)=O)CCC12 91112,c1(N(C)C)ccccc1C(=O)C(N1CCCC(CCNC(=O)OC(C)(C)C)C1)=O 91113,c1(C(N2CC(NC(C(CCC)OC)=O)C3(C2)CC3)=O)[nH]c2ccccc2c1OC 91114,N1(C(CN(C2CC(C#N)C2)C(c2cnn[nH]2)=O)=O)CCc2cnccc2C1 91115,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(=O)CC2(C(F)(F)F)CCC2)CC1 91116,C1(NC(c2cc(CC)on2)=O)CCN(C(c2cc3sccc3[nH]2)=O)CC1F 91117,c1(C(=O)NC2CN(C(C=C(CCN(C)C)Cl)=O)CC23CC3)cc2sc(C)cc2[nH]1 91118,C(=O)(C(F)C(C)(F)F)NC(C(C)C)CCNC(c1ocnc1C1CC1)=O 91119,C(=O)(C1=CC2C=CC1C2)N1CCC(CCOC)(NC(c2cnc(OC)cn2)=O)C1 91120,N1(C(c2nc(-c3ccn(C)n3)sc2)=O)CCCC(NC(=O)C(F)CC2CC2)C1 91121,c1(C(=O)NC2CCC(NC(C3(F)CCCC=C3F)=O)C2)cc2n(n1)CCO2 91122,C1(NC(C(CC#C)O)=O)COC2(CCN(C(c3ccc(Cl)nc3O)=O)CC2)C1 91123,c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C(O)CC2)=O)nccn2ccnc12 91124,N1(C(CCNC(C)=O)=O)CC23CCCC2(C1)CN(C(=O)CCC(C)O)C3 91125,N1(C(C(C)=C2CCC2)=O)CCC(N(C(=O)CSC2CC2)CC2CCCN2C)C1 91126,C(C)(C(CC(=O)N1CCC(C)(F)CC1)NC(=O)CC1CC(SC)C1)OC 91127,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(C3CCC4CCC(=O)N34)=O)C2C1 91128,Cc1ncnc(C)c1C(=O)NCC=CCNC(C1CC(c2ccccc2)CO1)=O 91129,N#Cc1c(F)cc(C(=O)NCc2ccc(CNC(=O)CCC(F)F)cc2)cc1F 91130,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91131,N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCN(C(=O)C(O)c2ccsc2)CCC1C 91132,C1(C#N)(OC)CC(C(=O)NC2(C(=O)NCCC#CCO)CCC2)C1 91133,C(=O)(C(F)CCC(C)(C)C)N1CCCC(C)C1CNC(C12CCCN1CCC2)=O 91134,N1(C(CN(C)C2CC2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91135,N1(C(CN)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91136,CC1(C)CC(CNC(=O)COCCCF)CN1C(=O)C1=NNC(C(F)(F)F)C1 91137,N1(C(Cc2c(C)cccc2)=O)CC2CCCC(CNC(c3cn(C)cn3)=O)C2C1 91138,CC(C)(C)C(=O)N1CCCC1CN1CCC(NC(c2cscc2C(F)(F)F)=O)C1 91139,C(C(=O)N1CC(F)(CNC(c2ccc(C3OCCO3)cc2)=O)C1)(C(C)C)OCC 91140,c1(NC(=O)CNc2cccnc2)ccc2nonc2c1.C12CC1CNC2=O 91141,c1(C(N2CCOCC(NC(C(Br)=C(C)C)=O)C2)=O)nc2cnccc2s1 91142,CC1(C(=O)NCC2CCN(Cc3nn[nH]n3)CC2)COc2ccccc2O1 91143,O(NC(=O)C(CC1CC1)NC(C1CC(=O)N(OC)C1)=O)CCOC 91144,O=C1CCN(C2CCN(C(c3cc(C(F)F)n(C(C)(C)C)n3)=O)CC2)C(=O)N1 91145,C1(O)(CNC(Cc2cccc(OC)c2)=O)CCCN(C(C2CC2C(N)=O)=O)CC1 91146,c1(NC(=O)NC2C(C)(C(F)F)C2)ccc(C#N)c(C#N)c1 91147,C=CC(C)(CC)C(=O)N1CC(COC)(NC(=O)C=CC(C)(C)SC)C1 91148,N1(C(c2c(C)coc2)=O)CCC(C(C)NC(=O)CC2CCC3CC23)CC1 91149,c1(NC(C23CCC(c4ccccc4)C2C3)=O)cccnc1Br 91150,N1(C(c2c(C(C)(C)C)cns2)=O)CC(C2CN(C(=O)CC3CCSC3)C2)C1 91151,N1(C(C(c2cccc(C)c2)C2CCN(C)CC2)=O)CCC=C(C(=O)O)C1 91152,c1(C(=O)NC2CCC(NC(CNC(C)=O)=O)C2)ccc(C=CC(C)C)cc1 91153,C12(c3n(Cc4ccc(C(C)=O)cc4)nnn3)CCC1CN(Cc1cnc3n1CCC3)C2 91154,c1(OC)cc(OC)c(CN2CCN(C(c3ccnc(F)c3C)=O)C3CC23)c(Br)c1 91155,CC1(C)C(NC(c2cncnc2)=O)C(C)(C)C1NC(c1ccc(F)s1)=O 91156,c1(CNC(c2nnnn2C2(C)CC2)CC)nccn1-c1ccccc1 91157,c1(CC)cc(N)ccc1C(=O)N(C1CCCCC1N(C(=O)C(N)=O)C)C 91158,N1(C(C(CC)C)=O)CCC(CNC(C2CCCN2C=O)=O)CC1 91159,N1(C(C(=O)N(C)C2CC2)=O)CCCC1CCCNC(=O)CCc1ccncn1 91160,C1(NC(CC2C(C)(C)N(C(=O)Cn3cncn3)CC2)=O)CCC(C2CC2)CC1 91161,C1(C(=O)NCc2onc(COC)n2)CC1C1CN(C(c2cn(C(C)C)cn2)=O)C1 91162,c1(-c2nc(C3CN(C(=O)NCc4ncc(F)nn4)C3)on2)ccc(F)c(F)c1 91163,c1(CN(CC(c2ccccc2Cl)(C)O)C)cc(Cl)cc(Cl)c1 91164,c1(C(=O)NCCCNC(CCSc2n(C)nnn2)=O)cc(=O)c(O)c[nH]1 91165,C(C)(CNC(=O)Cn1cc(C(C)O)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91166,CC1CC(NC(c2ccsc2C(F)(F)F)=O)CCN1C(C1CCC(C#N)CC1)=O 91167,C1(C)(CNC(C(CC=C)C)=O)CCN(C(c2ccc3c(c2)CC3)=O)CC1 91168,Cc1cc(O)nc(C)c1C(N1CCN(C(c2onc(C)c2C)=O)CC(C)C1)=O 91169,C=C(CC)CN=c1nc(N2CCN(CC(c3cccs3)O)CC2)c2c([nH]1)CCC2 91170,CC1CCc2[nH]nc(C(N3CCC(NC(=O)Cc4cccs4)C3C(C)C)=O)c2C1 91171,C1(NC(c2cccc(C3CC3)n2)=O)CCOC(C2CCCC2)C1.C1C=CCS1 91172,c1(C2C(NC(=O)NCCCNCC)CCO2)ccccc1Cl 91173,C1(N(C(CC(CC)C)=O)C)CN(C(=O)CN2CCC(NC(C)=O)CC2)CCC1O 91174,CCS(=O)(=O)c1ccc(NC(=O)NCc2cnc(N3CCOCC3)nc2)cc1 91175,c1(NC(CN(CC)CC)=O)cccc(CNC(C2CC2C(C)C)=O)c1 91176,c1(C(c2n(CCOC)nnn2)NC2COC(=O)C2)ccc(F)c(Cl)c1Cl 91177,C1(NC(CCCSC)=O)CCCC(NC(c2ncccc2C(C)(C)O)=O)CC1 91178,C(c1ccncc1)=CC(=O)NCC1(O)CC(NC(CSC)=O)C1 91179,Cc1cnc(C=CC(=O)N(C)CC2CCN(C(C3CCN3C3CCCC3)=O)C2)[nH]1 91180,C12(NC(C(C(C)C)SCC)=O)CCCC(NC(c3ccc(C)nc3N)=O)(C1)C2 91181,C(CC(C)(C)C(=O)NCC(CC)NC(c1ccccc1NC(=O)CC#N)=O)OC 91182,N1(C(C(C(C)NC(C(=O)NC)=O)C)=O)CCCC2CN(C)CC12 91183,C1(NCC)CCCN(C(=O)C(C2(O)CCC2)NC(=O)CC2CC(C)(C)CO2)C1 91184,N1(C(CNC(=O)NC)=O)CCCC(c2cn(CCNC(C3CCCO3)=O)nn2)C1 91185,C1(NC(c2ncn(CC)n2)=O)COC2CN(C(c3c(C)cc(C)cc3N)=O)CC12 91186,N1(C(C=CCC)=O)CCC2(CCCC2NC(=O)Cc2c[nH]c3cc(Cl)ccc23)C1 91187,N(C(=NCCCn1cccn1)NC(c1ccc(F)c(F)c1)C)C(C#C)CC 91188,N1(CC)CCN(C(C2CCN(C(C3CNC(=O)N3)=O)CC2)=O)CC1(C)C 91189,C1(NC(C(C)O)=O)CCCC1NC(=O)Cc1cnc[nH]1 91190,c1(C(=O)NCC23OCCC(NC(CC=C)=O)(C2)C3)nnn2c1CCCCC2 91191,c1(OC)ccc(Br)cc1S(=O)(=O)Nc1cc(C(=O)O)ccc1F 91192,c1(-c2onc(-c3ccc(-c4ccc(C)cc4)cc3)n2)ccc2ncccc2c1 91193,C1(C(C)C(=O)N(C)Cc2cn[nH]c2)CCN(C(=O)C(C)(C)N(C)C)C1 91194,C(C)(CO)(C(=O)NCCC1CN(C(c2cncc(Cl)n2)=O)C1)NC(C)=O 91195,CC1CN(C(C2CCN(CCF)CC2)=O)CCN1C(=O)Cc1ccncc1Cl 91196,CCCCCC(O)C(=O)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2C)CC1CO 91197,C(=O)(C1=CCCOCC1)N1CC(C)CC(NC(c2c(CC)occ2)=O)C1 91198,N1(C(C(C2CC2)OCC)=O)CC(C)(OCC(=O)N(CCCF)C)C1 91199,CC(C)C(C)CC(=O)N1CC(C(=O)NC(CC2CCC2)CO)CC(C)C1 91200,N1(C(C(CC(=O)OC)C)=O)CC(NC(c2c[nH]c(C)c(Cl)c2=O)=O)C2(CCC2)C1 91201,N1(C(C(C(=O)OCC)CC)=O)CCC2(CC(C(N3CC(O)C(O)C3)=O)C2)C1 91202,C=CC(C)(O)CC(=O)N1CCC(c2cn(CC(=O)NCC)nn2)CC1 91203,C1(NC(COc2ccc(C(C)C)cc2)=O)CCN(C(c2nncn2C)=O)C1(C)C 91204,c1(C(=O)OC)ccc(NC(=O)C(CC2CCCC2)N2CCC(CNC(C)=O)C2)s1 91205,N1(C(c2c(C)cc[nH]2)=O)CCC(C2(NC(=O)CC3C(C4CC4)C3(F)F)CC2)CC1 91206,C=CCCCCCCC(=O)NCCNC(=O)CC1CCCCC12NC(=O)NC2=O 91207,c1(C(CNC(C(C)C2CCOC2)=O)NC(c2ccc(CO)s2)=O)ccc(Cl)nc1 91208,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91209,N1(C(c2c(C)cc(O)nc2)=O)CCCC2(CCCN2C(C23CC(C2)C3)=O)C1 91210,c1(CCC)ccc(S(=O)(=O)N2CC3CCC(C2)N(C(c2nnc(C)o2)=O)C3)cc1 91211,c1(C(=O)NCCN(C2CCCC2)C(C=Cc2ncc(C)[nH]2)=O)ccc(Cl)cc1O 91212,c1(C(N(CCN(C(CNc2nccc(OC)n2)=O)C)C)=O)ccc(C)c(C)c1O 91213,C(=O)(C1CCCc2scnc21)N1CCC(N(C(=O)CC2C=CCCC2)CC)CC1 91214,c1(C(C(=O)NC2CCCO2)N(C(c2cccnc2)C)CC2CC2)ccc(Cl)s1 91215,C1(C(=O)NCCNC(C(CC)c2ccccc2)=O)CCC2(CCOCC2)CO1 91216,C1(COC)CN(C(c2ccc(Br)nc2F)=O)CCN1Cc1scnc1C 91217,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91218,C(c1cccc(O)c1)=CC(=O)NCC1CN(C(CCCOC(C)C)=O)CC1C 91219,Cn1ncc(C#N)c1C(=O)NCCc1ocnc1CNC(=O)CCn1cnnn1 91220,S(=O)(=O)(c1cccc(Cl)n1)NC1C2CN(C(c3ccc(NC(C)=O)c(F)c3)=O)CC21 91221,N1(C(C2CN(C(N)=O)C2)=O)CC2CCC2(NC(c2ns[nH]c2=O)=O)C1 91222,Nc1cc(C(=O)NCc2cc(O)nc(C3CC(C)C3)n2)cc(O)c1Cl.C1CC1 91223,C1(C(=O)NCC(C)(CO)NC(c2cc(F)n[nH]2)=O)CC2CCCC(C1)C2 91224,C(=O)(C1=CC2(CCOC2)C1)N1CC(C(C(=O)NCC2(C)CCN(C)CC2)OC)C1 91225,CC1(C)CCCC(C(=O)NCC23CC(NC(C4CCS(=O)(=O)C4)=O)(C2)C3)O1 91226,C1(C(=O)OC)CCCC(Cn2ccnc2-c2cccc(C(C)C)c2)C1 91227,c1(NC(C2(F)CN(C(C(n3ncc(C)c3)C)=O)C2)=O)cccc(Cl)c1C 91228,C=C(Br)CC(C)(C)C(=O)NCC1CCC(NC(c2cnn(CC(C)C)c2)=O)C1 91229,CC(C)(O)C(C)(C)CNC(C1COCCN(C(C2CCCCCO2)=O)C1)=O 91230,N1(C(CCC=C=C)=O)CCC2(CC1)CC(NC(=O)COCCCOC)CCO2 91231,C1(OC)(CNC(=NCc2ccco2)NCC2CCCCC2C)CCSCC1 91232,C(=O)(CCCCC(C)CC)NCC(CCC)C(=O)NCc1nnsc1C 91233,c1(C(=O)NCC)ccc(N(C)CC2CCCCC2CNC(=O)C(N)=O)cc1 91234,CCCCC(O)C(=O)N1CCC(CNc2ncc(Br)c(O)n2)C1 91235,c1(C(N2CCC(NC(CC3(OC)CCC3)=O)C(F)C2)=O)cc2nc(Cl)ccc2o1 91236,C1(CNC(c2nc(COC)sc2)=O)C2CCC(C2)N1C(=O)CC1C=CCCC1 91237,C(C)(C)(CC(=O)NCc1ccc(Cl)nc1)N(C(CCSCC)=O)C 91238,c1(C(=O)NCC2CN(C(c3[nH]cc(C)c3)=O)CC2(C)C)cnc2ncnn2c1O 91239,N1(C(c2n(C)ncc2)=O)CC2CC2C1CNC(=O)CC1CC(F)C1 91240,Cc1nc2ncc(C(=O)NCC3CCN3c3ncnc4c3ncn4C)c(=O)n2[nH]1 91241,N1(C(=O)NCCc2cccc3[nH]ccc23)CCc2nc(O)cc(Br)c2C1 91242,C1(CN)CCCC2(CCC2)O1.C12(CCCC1)C(=O)N2 91243,c1(C(CC)NC(C2C=CC(NC(c3nnsc3C)=O)C2)=O)cccc(O)c1 91244,C=C1CON(C(=O)CC2(N(C(=O)CC3CCC(C)C3)C3CC3)CCC2)C1 91245,c1(CC(N2C(C3(NC(C(CSC)C)=O)CC3)CCC2)=O)ccc(C)nc1Cl 91246,C=CCC(C)C(=O)NOC1CCCN(C(C2CC(CC3CC3)C2)=O)C1 91247,CC1(NC(=O)CC2CC23CC3)CCCN(C(c2cscc2Cl)=O)C1 91248,C12(C(=O)NCCC(O)CNC(C3(c4ccccc4CO)CC3)=O)CCN(CC1)C2 91249,C=CCCC(F)(F)C(=O)N1CC(C(=O)N(CC(C)O)C2CC2)C2(CC2)C1 91250,CC1(C)C(C(=O)NC(C2CC=CCC2)C(N2CCC(F)(F)C2)=O)C1(C)C 91251,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(C2CC2)cn1)NC(CC)C(C)O 91252,N1(C(CCC=CCC=C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91253,N1(C(CCC=C)=O)CCOCC(CNC(=O)C(F)(F)CN(C)C)C1 91254,Cc1ccc(F)c(CNC(C2CCC(CNC(C3CC4CCC4C3)=O)C2)=O)c1 91255,c1(C(C)C)ccc(NC(C2CN(C(=O)COCC3CCCCO3)CC2C)=O)nc1 91256,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91257,N1(C(C(C)=CC2CC2)=O)CCC2(NC(=O)Cc3ccn(C(F)F)n3)CCCC12 91258,C(=O)(C(CC(F)F)C1CCC1)NCC=CCNC(C(C=C)(F)F)=O 91259,N1(C(C(C)=C2CC2)=O)CCC(C)(C)C1C(=O)NCc1nc(C(N)=O)co1 91260,CC(C)C(F)C(=O)NC1CCCC(NC(c2cccc(C3(N(C)C)CC3)c2)=O)C1 91261,C1(C(=O)NCc2c(C(=O)NC(C)(C)CO)scc2)CC(=O)CCO1 91262,C1(N(C(=O)CC2CSCCS2)CC)CC2CCC(C1)N2C(=O)Cc1ccsc1 91263,N1(C(C2C=CC(NC(C(C)OCCOC)=O)C2)=O)CCOCC2(CC2)C1 91264,c1(C(c2n(CCCSCC)nnn2)NCC2OCCC2C)nc(Br)c(C)cc1Cl 91265,C#CCCN=C(NCC(C)C(F)(F)F)NCCOC(C1(c2ccccc2)CC1)=O 91266,C1(C(=O)NCC2(NC(C3CCN(C4CCCCC4)C3)=O)CCC2)CCCOCC1 91267,Cc1cc(-c2ccccn2)cc(C)c1CC(=O)Nc1c(Cl)cc(Cl)cc1Cl 91268,c1(C(C)C)ccc(C#N)c(N(c2nn[nH]c2C(F)(F)F)C)n1.C12CCN(CC1)C2 91269,CCN=c1[nH]c(C)c(C(N2CCCCC2CNC(C2CCN(C)C2)=O)=O)s1 91270,c1(C(N2CC(C)N(C(c3cnn4ccsc34)=O)CC2)=O)cccc2ccsc12 91271,CC1CC(CC(=O)NCC=Cc2ccccc2)CN1C(c1cc(C(N)=O)c[nH]1)=O 91272,Cc1cc(=NC(=O)C2CCCC(NC(=O)N(C3CN(C)C3)C)C2)[nH]o1 91273,Cc1ncsc1C(N1CC(OCCNC(c2sccc2COC(C)C)=O)C1)=O 91274,Cc1cn(C)cc1C(=O)N(CC(=O)N(CCCC(C)(F)F)C)C1CCC1 91275,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91276,N1(C(CCC)=O)CCC(NC(c2cc(CC)ccc2F)=O)CC1C 91277,C=CC(CCC)CC(=O)N1CCN(C(=O)COCCNC(=O)C(C)OC)CC1 91278,n1(C(CC)C)ncc2c(N(CCCNC(c3cc(=O)c(Br)c[nH]3)=O)C)ncnc12 91279,c1(CC)nc(C)ncc1C(N1CCCC(NC(=O)CN(C)CCOC)CC1)=O 91280,N1(C(Cc2cc(C)no2)=O)CC2CN(C(c3ccc4ncnn4c3)=O)CC2C1 91281,c1(C(=O)NCCC2CC(NC(C3CC(O)C(F)C3)=O)C2)cncc2c1CCCC2 91282,c1(C(=O)NC(CNC(C=CCC)=O)(C)C)c[nH]cc(Br)c1=N 91283,N12CC(C(CC(F)F)C1)C2=O.c1(C2CN(C(=O)OC(C)(C)C)C2)nc[nH]n1 91284,C(CCCS(=O)(=O)c1ccc(F)cc1)Nc1ccncc1.CC 91285,Cc1ccccc1CCNC(C1CN1C(C1CCOCC1)=O)=O 91286,C(=O)(C1CC=Cc2ccccc21)NCC1C(C(N=c2nnn(C)[nH]2)=O)C1 91287,N1(C(C(CC)=CC)=O)CCCCC(CNC(=O)C(c2ccc(Cl)cc2)CO)C1 91288,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91289,C1(N(C(C(C)OCC)=O)CC)CCCN(C(c2n[nH]c(=N)s2)=O)C1 91290,C1(CNC(C(CC)SC)=O)CCCN(C(=O)CSc2nncs2)CC1 91291,N1(C(=O)Nc2c(C(=O)OC)n(C)nc2)CCC2NC(=O)NCC2C1 91292,N1(C(C(CC)C(C)O)=O)C2CCCC1CN(C(=O)C(C)CC1CCCCC1)CC2 91293,C1(CNC(=O)COCC2CC2(Cl)Cl)CC2COCC2N1C(c1ccc(O)cc1)=O 91294,c1(C(N2CC3CC2(c2nc(C)no2)C3)C(=O)NC(CC)C)ccc(C)c(Cl)c1 91295,C(=O)(C(O)C1=CCCCC1)NC1(C)CCN(C(N2C(CO)CC(CC)C2)=O)C1 91296,C1(NC(C2(CC)CCCCC2)=O)CN(C(=O)CC2CCN(C)C2)CC1N=[N+]=[N-] 91297,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91298,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1(C2CCCO2)CCC1 91299,CC(O)(CC(=O)NC(C1CCCC1NCc1cc(F)c(Cl)cc1Cl)=O)CC(=O)O 91300,C(=O)(CC(C(C)CC)NC(=O)CCCC)NCC1(CC=C)CCOC1 91301,C12(CNC(=O)Cc3cccs3)CCN(CC1)C(=O)CO2.c1(CO)ccncc1 91302,CCC(C(O)C)C(=O)NC(c1ccc(CNC(=O)CNC(C)=O)cc1)C 91303,c1(CCC(=O)Nc2cccc(OC3CCOC3)c2)cc(F)c(F)c(F)c1 91304,C1(OC)(OC)CCC1C(=O)NC1CCCC1NC(=O)CNC(c1ccccc1)=O 91305,c1cc2[nH]c(=NCc3ccc(C(F)(F)F)s3)[nH]c(=NCC3CCCSC3)c2[nH]1 91306,CN(CC(=O)NC1CCOCC1)N1CCC(N(C)C)C1 91307,C12COCCN(C1)C(=O)NC2=O.C1(N2CC(C(C3CC(C)C3)=O)C2)CCOCC1 91308,CC(C)(C)CC(O)C(=O)NCC(=O)NCC1(CC(=O)NCCO)CC1 91309,C1(O)(C(=O)NCC(C)N(C)C(c2ccc(C(F)(F)F)cc2)=O)CC(C)(C)C1 91310,CCC(C)(CC)C(=O)NCCC(CNC(c1coc(C(F)(F)F)n1)=O)OC 91311,CCCC(O)C(CO)NC(=O)CCN(C(=O)Cc1cnn(CC)c1)CCOC 91312,c1(CNC(C(CO)OC)=O)ccc(C(C)NC(c2[nH]nnc2C2CC2)=O)cc1 91313,N1(NC(C2(NC(c3cc(C)ns3)=O)CC2C)=O)CCNC(=O)C1 91314,Cc1ccc(C#N)c(NC(C2C=CC(NS(=O)(=O)c3ccccc3)C2)=O)c1 91315,c1(C(=O)NCc2cc(F)ccc2-c2ccc(Cl)c(Cl)c2)n[nH]c2c1COCC2 91316,Cc1nc(C(N2CCC3(CNC(=O)Cc4cn[nH]c4)CCCC23)=O)c2ccccn12 91317,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CCC1C 91318,n1(C(C)C)c(CC(=O)Nc2ccc(N3CCCOCC3)cc2)nnc1S 91319,c1(NC(C2C=CCN(C(CCC=C)=O)C2)=O)sc2ccccc2c1CS(C)(=O)=O 91320,C1(C(NC)=O)CCCCC1C.C(C)(CCNC(=O)CC1(C(=O)N)CC1)N(CCC)C 91321,c1(C(N2CCC(NC(CCOCC)=O)C23CC3)=O)coc(S(C)(=O)=O)c1 91322,C=CC(C)(CC)C(=O)N1CCC(C2CCCN2C(=O)C2=NNC(=O)C2)C1 91323,c1(CNC(C2(CC)CCN(C(C(C(CC)O)C)=O)CC2)=O)nn(C)c2c1CCC2 91324,C(=O)(C(O)CC(C)(C)C)NC(CC)CC(=O)NC1CC2COCC(C1)C2 91325,N1(C(C(=O)N(CCCC2CCCC2)C)CCCCC2CC2)CCCN(C)C(=O)C1 91326,c1(CN2CC(C)(NS(CCC)(=O)=O)C2)ccc(OC)c(F)c1 91327,CCC(CC)CCCC(=O)NC1(COC)CCN(C(c2cnc(C(C)C)[nH]2)=O)C1 91328,c1(NC(CC)=O)cc(C(=O)NC2CCCC2CNC(c2nc(C)cs2)=O)ccn1 91329,C1(C(=O)NCc2occ(C(=O)Nc3c(OC)nccc3)n2)C2CCC(C2)C1C 91330,C#CC1CN(C(=O)C(CNC(C2CC(=C3CC3)C2)=O)C(F)(F)F)CCN1C 91331,C1(OCC)CC2(C1)CC2C(=O)NCC(C)NC(c1cncnc1)=O 91332,C(=O)(C(CC)CCCC)NCC(=C1CN(C(c2cccc(SCC)c2C)=O)C1)F 91333,C12(CNC(c3c(C)coc3)=O)CCC(CC1)N2C(c1cc2scnc2[nH]1)=O 91334,Cn1[nH]cc(C(=O)NCCN2CCN(C(C3CN(C(N)=O)C3)=O)CC2)c1=O 91335,C1(OC)CC2CC1CN(C(=O)CC1(NC(c3cnncc3C)=O)CC1)C2 91336,c1(C(N(CCCOCCNC(C2CCC(C)S2)=O)C)=O)cccc(Cl)c1 91337,C(C(=O)N=c1c(Cl)c[nH]cc1I)C(c1cc2cc(F)ccc2[nH]1)C#N 91338,c1(NCCC(=O)NC)[nH]c(=NC(C)c2ccoc2)nc2ncn(C)c12 91339,c1(C(N2CC(C(=O)Nc3c(Br)ccnc3Cl)C2)=O)cn2cccc(Br)c2n1 91340,c1(-n2c(C(=O)NC(C)(C)CNC(=O)CC3CCCCC3)cnn2)ccccc1F 91341,C1(NCc2ncn(C)c2)CN(C(=O)Cc2ccccc2O)CC1C#N 91342,C1(C2C(C)C2)C(=O)NCC(O)CN1C.C(=O)(CO)NC1CCC1 91343,c1(C(=O)NC(CC)CNC(c2n[nH]cc2C2CC2)=O)n[nH]c(C)c1C 91344,Cc1cc(O)ncc1C(=O)NC1CC(C)(CNC(c2ccc(O)c(Cl)n2)=O)C1 91345,C1(NC(CCC2(NC(c3c(OC)nsc3)=O)CCCC2)=O)CC12CCCCC2 91346,N1(C(c2cc(C)sc2)=O)C2CCC1CN(C(=O)CN1CCC(N(C)C)CC1)C2 91347,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91348,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCO3)=O)C4)=O)cc12 91349,c1(C(C)=O)cc(Cl)c(N2CCN(C3CCN(C(C4CCC(=O)N4)=O)C3)CC2)nc1C 91350,CC1CCC(C)(C(=O)NC2CC(CNC(c3cnc(S)[nH]3)=O)C2)C1 91351,c1(NC(C2N(S(CC=C)(=O)=O)CCSC2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91352,c1(OC)ccc(N)cc1-c1cn(C(C)CC(=O)NC2(C3CCCO3)CCC2)nn1 91353,c1(C(=O)NC2C(NC(c3cc(OC)ns3)=O)CCC2)sc2cccnc2c1Cl 91354,C(CC(=O)NC12CC1CN(C(c1nc(Cl)sc1C)=O)C2)(C(C)C)OCC 91355,C(CCCCCSC)SC1CC(NC(=O)NCC#C)C1 91356,c1(NC(C2CCN2S(=O)(=O)CCCCl)=O)cc2ccoc2cn1 91357,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CF)(C2)C3)=O)C1)=O 91358,c1(CNC(c2n(-c3c(C)cccc3)nnn2)C2(CF)CC2)c(F)cnc(Cl)c1C 91359,N1(C(c2cc(C)c(C)s2)=O)CC23CCCCC2(C1)CN(C(C1CC2CC2C1)=O)C3 91360,C(CN=c1cc[nH]cc1C(=O)OCC)C1CC(NC(C2CCC(=C)CC2)=O)C1 91361,c1(CN2CC(F)(C(=O)NCC)C2)csc2ccccc12 91362,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91363,c1(OC)ncnc(N2CCC(O)C(C(=O)OCCC(F)(F)F)C2)c1C 91364,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91365,N1(C(C2CCN(CCF)C2=O)=O)CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O 91366,c1(C(N(CC(c2ccccc2)CC)CC)=O)ccc(C(F)(F)F)s1 91367,N1(C(C(C)=C2CC2)=O)CCOCC1C(=O)NC(C)(CO)C(C)C 91368,CCC(C(=O)NC(CC(=O)N1CCC(NC(=O)OC)C1)C(C)OC)C(F)(F)F 91369,C1(N(C(=O)CCN2CCC2)C)CC2CCC(C1)N2C(c1cc(S(N)(=O)=O)c[nH]1)=O 91370,C1(CNC(Cc2cc(C)[nH]n2)=O)CC(O)CN(C(=O)CCc2ccccc2)C1 91371,c1(CN2CCC(NC(C=CC)=O)C2)cc(C(=O)O)c(O)cc1F 91372,C1(CNC(C(C2CN(C(C(N3CCOC3=O)C)=O)C2)O)=O)CCC(N(C)C)C1 91373,c1(C(=O)NC2(n3ccnc3C=C3CCC(N(C)C)C3)CC2)c(Cl)ccc(F)c1F 91374,c1(OC)c(C(=O)NCC(C)NC(=O)COC2CCOC2)cc(Br)cc1F 91375,CN1CCOCC1CNC(C12CC1CCN2C(C1CCC(CO)CC1)=O)=O 91376,C1(C(=O)NCC)CC(F)(CCN(C)C)C1.N1(C(C)=O)CC(NC)C1.C1C(=O)O1 91377,c1(C(=O)NC(CCNC(c2cc(C(C)C)no2)=O)(C)C)cc2c(ccn2C)[nH]1 91378,C1(C(N2CCCC(N(C(Cc3c(C)cco3)=O)CCF)C2)=O)CCCCC1(F)F 91379,C1(C(=O)NCC(CC)(C)Cl)COCCN1C(c1cc(=O)cc[nH]1)=O 91380,C=CCC(C)(C)CC(=O)NCC1CCCN1C(c1cc(C)c(C)nc1O)=O 91381,C1(COC(=O)COC2CCCCC2)CN(C(=O)C=CC2CCOCC2)CC2CC12 91382,N1(C(=O)CN2CCN(C)CC2)CCN(C(C)CNC(C2(SC)CC2)=O)CC1 91383,CC1=NOC2(C1)CC(C(N1CCCCC(CNC(C3CCS(=O)(=O)C3)=O)C1)=O)C2 91384,C1(C(=O)NC(C(C)C)C2CCC2)(CC)CCN(C(c2c[nH]nc2C)=O)CC1 91385,N1(C(C(CCC)O)=O)CC2(C1)SCCC2NC(c1cncc(OC)n1)=O 91386,c1(C(=O)NCC(C2CC2)Nc2cc(OC(C)C)ncn2)ccc(C)c(Cl)c1F 91387,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)(NC(c2cc(Cl)ncc2O)=O)CC1 91388,Cc1noc(C)c1CCC(=O)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 91389,N1(CC2CCN(C(CNC(C)=O)=O)CC2)CCC2(CC1)OCCc1ccccc12 91390,c1(NC(CCC)CNC(=O)C(C)c2ccco2)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 91391,C1(C(=O)NC2(CO)CN(C(c3sccc3CO)=O)C2)CCc2ccnn2C1 91392,Cc1ccc2[nH]c(C(N3CC(CCNC(=O)C#CC4CC4)C3)=O)cc2c1 91393,n1(C(C)C)cc(Br)c(C(=O)NCC2CC(NC(=O)Cc3cn[nH]c3)C2)n1 91394,C1(SCn2c(C(C3(C)CC3)NC3CC(CC#N)C3)nnn2)(N)CCCC1 91395,CC(CF)N=c1[nH]c2c(c(=NC(C)c3ccn(CC(F)(F)F)n3)[nH]1)CCC2 91396,C1(F)(CNC(c2c(C)nc(O)s2)=O)COCCN(C(c2cncc(O)c2Cl)=O)C1 91397,N1(C(Cc2ccn(C)n2)=O)CCN(C(=O)C(F)(F)CC2CCCC2)C(C(F)F)C1 91398,C1(NC(C2CCCNS2(=O)=O)=O)CCN(C(C2CCCCC2)=O)CC12CCC2 91399,CC(C(F)C(=O)NC1C2CC3CN(C(c4ccc(F)cc4F)=O)C1C3C2)C(F)(F)F 91400,C=CCC(CNC(c1c[nH]c(C(=O)OC)c1)=O)NC(=O)CCCOC1CCOCC1 91401,C1(CC(=O)NC(CCC)CCO)CN(C(C2CCOCC2)=O)CCC1C 91402,c1(C(=O)NC2(C)CCCN(C(C3C(=C)C3)=O)C2)c[nH]c2ccccc12 91403,c1(NC(C2CC(SC)CC(C)(C)O2)=O)cc(Cl)cc2c1OCC(=O)N2 91404,N1(CCC)CCc2nc(C(=O)N(CCO)Cc3ccccc3)cn2CC1 91405,N1(C(c2nc(CC)sc2)=O)CCC2C(C(=O)NCC(F)(CC)CC)C2C1 91406,CCCCCCCC(O)C(=O)NCCCN1CCCS1(=O)=O 91407,c1(N2CC(C)(CC)OCC2)ccc(S(=O)(=O)NCC2CCCCS2)cc1Br 91408,c1(C(C)=O)c(Cl)nc[nH]c1=NCC1CC(C)N(C(=O)CC2CSC2)C1 91409,c1(C2(F)CC(C(=O)NCC(C)CNC(C3CC(O)C3)=O)C2)cccc(F)c1 91410,C1(NC(CC2(C(=C)F)CCC2)=O)CC2(C1)CN(C(c1scnc1Cl)=O)C2 91411,N1(C(C(CSC)O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CSCC3)=O)CCO2 91412,C(=O)(C(C)(CNC(=O)CC1OCCCO1)CC)N1C(C)(CCC)CC1 91413,c1(OC)cccc2cc(C(=O)NC3CCN(C(=O)C(F)=CCCF)C3)oc12 91414,C1(C(=O)Nc2cc(NC(c3ncn(C(C)C)n3)=O)ncn2)CCN(CC)C12CC2 91415,N1(C(CCN(C(=O)CC2C=CCC2)C)=O)CCCCC1CF 91416,c1(C(=O)NCC(C(C)C)NC(c2ccsc2Br)=O)ccnc(C2CC2)n1 91417,c1(OC)cccc(C)c1NC(C1(CNC(c2ccc(C(F)F)o2)=O)CCCO1)=O 91418,C12(OC)CCN(CC1)N1CC(C1)NC2=O.C12CC3(CCC3)N1C2=O.C(C)(=O)OC 91419,CC1CN(C(c2csc(Cl)c2F)=O)CC1NC(C1(C)CC1(F)Cl)=O 91420,c1(C(=O)NC(C(=O)NC2(C)CC(O)(CO)C2)C2CC2)cccc2occc12 91421,C(=O)(C(=O)CC(C)C)NCCC(C(=O)NCC(C(C)C)OC)O 91422,C12(CC3(CN(C(=O)CNC(=O)Cc4ccnn4C)C)CC3)CCC(CC1)C2 91423,N1(C(CC#CC)=O)CCCC(C(=O)NCc2cc(C)sc2C)C1 91424,C1(C(C(=O)NC(C(=O)NCC)C)(C)C)CCCN(C(c2cn(C)nc2C)=O)C1 91425,c1(CNC(=NCNCC(=C)C)NCCC2CCC2)coc2ccc(C)cc12 91426,Cc1cc(NCc2cn(Cc3cccnc3Br)nn2)cnc1Cl 91427,c1(O)ccc(C)c2c1CCC2.C1(OC(C)=O)(CNC(=O)C=CC(=O)NC)CCOCC1 91428,c1(CC(=O)N2CCNCC2)c(C)nc(O)nc1O.c1(C=O)nncn1C.CSC 91429,C1(C(=O)NCC(CC(F)(F)F)NC(c2cnco2)=O)CCc2c[nH]nc2C1 91430,C1(C(=O)NCC(C(=O)OC)OC)CCCN(C(=O)COC(C)C)CC1 91431,N1(C(C(SC)SC)=O)CCCC(O)(CCNC(=O)CCC2CC2(F)F)C1 91432,N1(C(C2N(CCCC)CCCC2)=O)CCCCC(NC(C2(CC(C)C)CC2)=O)C1 91433,C(=O)(C(C(C)(C)O)NC(c1ccc(F)c(O)c1)=O)N(C1CC(F)(F)C1)C 91434,c1(SC)ccc(C(=O)NCC(CO)NC(=O)CS(C)(=O)=O)cc1.c1(S)ccc(Cl)cc1 91435,C1(NC(C2(CC=C)CC2)=O)CN(C(=O)CCc2ncnn2C)C2CCCC12 91436,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 91437,c1(SC)cc(C(=O)N(C(C)CCNC(=O)CN2CCC(C)(O)C2)C)ccc1F 91438,C(=O)(C(C)NC(C)=O)N(C1CCCC1)CCNC(CSCC#C)=O 91439,CCC1=C(C(=O)N2CC(C)N(C(c3ncc(C)cc3F)=O)CC2C)SCCO1 91440,c1(CN(C)C(C2C3COCC23)=O)ccc(CNC(c2cccc(O)c2)=O)cc1 91441,c1(C(=O)NC2CN(C(CSCC=C)=O)CC2N=[N+]=[N-])cnc2c(c1)ncn2C 91442,Nc1cccc(C(=O)NCC(c2ccccc2)NC(c2cc[nH]c2C(F)F)=O)n1 91443,c1(NC(C2N(C(CCCN(C)C)=O)CC(O)C2)=O)c(Cl)nc(Cl)nc1CO 91444,Cc1ccc(C(CNC(=O)CC(C)(F)F)N(C(=O)Cc2ccncn2)CCO)cc1 91445,C1(CNC(C(c2c(C)onc2)N(CCC2CC2)C)=O)CCC(C)(C)CC1 91446,N1(C(C(CCOC)C)=O)CCN(C(c2ccc(C(C)=O)c(C)c2)=O)CCC1C 91447,C1(CNC(CN2C(C)CCC2)=O)CCCCN(C(C2(C)C=CCCC2)=O)C1 91448,C(CCCCC(=O)N(CC(O)C(F)(F)F)C)N(C(c1c(C)snn1)=O)C 91449,C1(C(=O)NCCC2(O)CN(C(CC(CCC)C)=O)C2)Cc2nn(C)cc2C(=O)N1 91450,CC(C)C(C(=O)NC(C1(O)CN(C(=O)COc2ccc(F)cc2O)C1)C)C(C)C 91451,c1(C(C(=O)NC2(CC=C)CCN(C(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 91452,N1(C(C(=O)N(C)CC2CC2c2ccccc2)=O)CC2CC1CN2 91453,n1(CC)nc(Cl)c(C#N)c1NC1CCCCCC1.N12CCC(C1)CC2=O 91454,Cc1ccc2cc(C(=O)NC3CC3NC(=O)C(F)n3ccnc3)c(C)nc2c1 91455,N1(C(COCCC)=O)CCN(C(=O)CCC(=O)NCC)C2CCCCC2C1 91456,C#Cc1cccc(CC)c1F.c12cccc(c1)CNC(=O)C1CC(C1)NC(=O)C2 91457,C(=O)(CC(C)C(C)C)NC1CN(C(C2(CC#C)CCCCC2)=O)CC1CO 91458,Cn1cc(C#N)cc1C(=O)NC(CC1CCOCC1)C(=O)NCc1nnc(O)o1 91459,C1(C(=O)NCC2(C(=O)NCC3CC4CC(=O)C3O4)CC(=C)C2)CCCC2(CC2)C1 91460,CC(CC(F)(F)F)N(C)C(C1C2CC1N(C(=O)C#CC1CC1)C2)=O 91461,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 91462,c1(C(C)NC(CC(CC)CC)=O)ccc(CN2CCCCC2)cc1 91463,c1(CC(=O)NC(CC2(C(=O)OCC)CC2)CO)c(C)nc(C)nc1O 91464,c1(OC)ccc2c(NC(C3(C(C)C)CNC(=O)C3)=O)cccc2c1 91465,C1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)C(C)C)CC2CCC(C1)S2(=O)=O 91466,N1(C(Cc2cn(C)nc2)=O)CCOCC(NCc2cccc(O)c2Cl)C1 91467,c1(C(=O)NC(CNC(C(c2ccccc2)C)=O)C2CC2)ccc2n[nH]cc2c1Cl 91468,n1(CC(=O)N(C2CCN(C(=O)CCc3cn(C)nc3C)C2)CC)ncn(C)c1=O 91469,c1(-c2nc(C)c(C(=O)NCC3(C)CC3(F)F)s2)ccc2ccccc2n1 91470,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 91471,C(CC(C(=O)N1CC2COCC2O1)NC(=O)CC1COCC(C)O1)OC 91472,N1(Cc2c(C)onc2)CCC2(CC1)CC2C(N1CCC(CO)C(O)C1)=O 91473,Cc1c(NC)ncnc1N1CCC(CNCCC2(C)CC2(F)F)CC1 91474,CC1C(C)N(C(=O)Cc2cnccn2)CCN1C(c1cnc(F)c(F)c1)=O 91475,N1(C(C2N(C(c3ccc(OCC(C)C)cc3)=O)CCSC2)=O)CCOC(C#N)C1 91476,C=C(C)C1OCCC1C(=O)NC(C12CCC(CC1)C2)CNC(=O)Cc1cnc(C)s1 91477,N1(C(CCC(C)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 91478,C(CNC(C1CCNC(=O)C1)=O)(CC(F)(F)F)NC(Cn1nc(C)c(Cl)c1)=O 91479,c1(C(=O)NC2CCCN(C(C=CC)=O)CC2)cc(S(=O)(=O)N(C)C)cn1C 91480,c1(C(=O)NCC2CN(C(CN(c3ccnn3C)C)=O)C2)cc2n(n1)CCO2 91481,C1(C)(CC)CC(C(=O)NCC2CC3(C2)CN(C(=O)CN=S(C)(C)=O)C3)CCO1 91482,C1(CCNC(C)(C)C)CCCN(C(C2CC(NC(CSCC(=O)OC)=O)C2)=O)C1 91483,C1(NC(=O)C(F)C2CCOC2)(CNC(C23CCC(C2)C3)=O)CCCC1 91484,C1(CNC(=O)CC2CC3(CCO2)CC3)CCC2CN(C(c3ccsn3)=O)CC12 91485,S(=O)(=O)(CCCN=C1NS(=O)(=O)c2ccccc21)COC1CC(OCC)C1 91486,C1(C(N2CCCC(N(C(=O)CC3CCCS3(=O)=O)C)C2)=O)CCCCC1(F)F 91487,c1(C(=O)NCC2(CNC(C(c3ccc(C)s3)C)=O)CCC2)cc2cn[nH]c2cn1 91488,c1(CC)ncnc(N2CCC(C(C)(C)C)(CNC(=O)CC(F)F)C2)c1F 91489,c1(Nc2scc(CNC(CCCCC)=O)n2)ccn2cc(C(=O)OCC)nc2c1 91490,N1(C(=O)OC(C)(C)C)CCN(C(=O)Nc2cccnc2)C(c2cccnc2)C1 91491,c1(CC)cnc(N2CCC(N3CCCC3)C2)nc1 91492,C1(C(=O)NCCCOC2CCC2)(CC)CCCN1C(=O)C(C)SC(C)C 91493,N1(C(C(CN(CC)CC)F)=O)CCN(C(=O)CCCSC)C2CCCC12 91494,c1(CC(=O)NCC2(F)CC(NC(C3CC3F)=O)C2)cc(Cl)ccc1Cl 91495,N1(C(=O)COCC2CCC2)CCC2(CC2C(N2CC(N3CC(F)C3)C2)=O)C1 91496,c1(C(=O)NC2(CNC(C3(S(N)(=O)=O)CC3)=O)CCC2)ccc(=O)n(CC(F)(F)F)n1 91497,C1(NC(c2cc(COC)on2)=O)CCCN(CCn2nc(C)nc2C)C1C 91498,Nc1nn(CC(N2CCCCC(NC(C3CCCCC3O)=O)C2)=O)cc1[N+](=O)[O-] 91499,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NCCC3CC(C)=NO3)on2)C1 91500,C(=O)(CC(C)CC(C)(C)C)NC(CC1CC2N(C(CC=CC=C)=O)C(CC2)C1)C 91501,c1(C(C)=O)c(C)[nH]c(C(N2CC=CC(NC(c3cscc3Br)=O)C2)=O)c1C(C)C 91502,CN1CCC(CC(=O)NC2CCCC2CNC(=O)CC23CC(N(C)C)(C2)C3)C1 91503,Cc1cc(N)c(F)c(C(N2CCCC(F)(CNC(C3(O)CC3)=O)C2)=O)c1F 91504,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 91505,C1(C(=O)Nc2c(C)cc(Cl)cc2)COC2CN(C(c3cnccn3)=O)CC12 91506,c1(C(=O)NCCN(C(=O)C(C)n2cccn2)CCC)ccc2sccc2c1 91507,C(c1ccc(F)c(F)c1)=C(C)C(N1CCC(C(=O)N(C)C2CC2)C(O)C1)=O 91508,C1(CNC(C(CC)C(C)O)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1CO 91509,C12(NC(C3CCC(C(N)=O)CC3)=O)CCC1CN(C(=O)CC1CCCS1(=O)=O)C2 91510,Cc1cc(=O)n(CC(N2CC(NC(c3cn(C4CC4)nn3)=O)C(O)C2)=O)cn1 91511,Cc1ccc(C(N2CCN(C(=O)C(C)n3cncn3)CC2C2CCC2)=O)c(N)n1 91512,c1(C(=O)NCCC2CC(NC(c3c(C)cc(SC)o3)=O)C2)ccnc2c1CCC2 91513,C(c1csc(Br)c1)=CC(=O)NC1CCCC(NC(=O)CC2CCC2)C1 91514,N1(C(C2(C#N)C(C)C2)=O)CC(CO)C2(C1)CN(C(c1cccnn1)=O)C2 91515,c1(OCC2(CN(C)C)CC2)cc(C(F)(F)F)ccn1.N12CCCC(C1)CNC2=O 91516,c1(C(=O)NC2(C(=O)NC3C(C)(C(F)F)C3)CSC2)cncc(CO)c1 91517,c1(C(=O)NC(c2[nH]nc(C(C)O)n2)C)ncn2c1COc1ccccc1-2 91518,c1(C(C)C)ccc(CC(=O)N(CC(F)(F)F)C)cc1Cl.c12nccn1C2 91519,CC1CC(NC(C2(C(F)(F)F)CC(F)C2)=O)CN1C(c1ccoc1)=O 91520,N1(C(CNC(=O)C=Cc2nccs2)=O)CCN(C(C2CCCC2)=O)CC1C1CC1 91521,C(=O)(CC(C)(C)CC)N1C(C(C)C)C(C(=O)N(C)Cc2nnc(O)o2)CC1 91522,CC1CCC(C)(C(=O)NCCN(C2CCCCCC2)C(C23CCC2C3)=O)CC1 91523,C1(C(=O)NCC2(NC(=O)COc3ccc(Cl)cc3)CCC2)OC2CCC1CC2 91524,N1(C(c2cn(C)c(O)n2)=O)CCN(CCNC(C2C(COC)(COC)C2)=O)CC1 91525,Cc1nc(N(C)C)sc1C(=O)N(C1CN(C(=O)CCC2CCCN2C)C1)C 91526,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCCC1(C)CNC(c1cnccn1)=O 91527,Cc1cc(C(N2CCCC2CNC(C2CCCC(N(C)C)C2)=O)=O)ncc1F 91528,c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCN(C)C2)cc2sccc2n1C 91529,CC1COCC(CNC(=O)CC2CCCN2C(=O)CO)O1 91530,c1(C(=O)NCC(CC)NC(c2cnc(OCC)s2)=O)noc(C)c1[N+](=O)[O-] 91531,C=CCCCCCCCC(=O)NC(C)CCN(C(=O)Cc1nccn1C)C 91532,N1(C(C(C)N(C(CC(C=C)CCC)=O)C2CC2)=O)CC2(CCOC(=O)N2)C1 91533,N#CC1CN(C(=O)CCN2CCCCC2)CCN1C(=O)CC1CCCCC1 91534,C1(C2CN(C(=O)CCN3CCC3)C2)(NC(C2C(C(C)(F)F)C2)=O)CC1 91535,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCN(C(=O)CC(O)c3ccccc3)CC2C1 91536,c1(CCC(=O)OC(C)C)cncc(Oc2ccc(NC(=O)OC)cc2)c1 91537,CC(C(=O)NC1(N(C(=O)CC2(O)CCCC2)C)CC1)C(C)n1cccn1 91538,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 91539,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CCC(C(F)F)C2)C1 91540,c1(C(=O)NCC2CCCN(C(C3(C4CCCO4)CC3)=O)C2)cc2ncccc2[nH]1 91541,C12(C(N3CC(NC(c4cc5n(n4)CCO5)=O)C(O)C3)=O)CCC(CO)(CC1)C2 91542,c1(CN(C)C(C2(C3CCCN3C(C3CCCSC3)=O)CCC2)=O)ccc(O)nn1 91543,C1(COC)CN(N2CC(C)(NS(C)(=O)=O)C2)CCO1 91544,C1(C(=O)NCC2N(C(C=Cc3ncn(C)c3)=O)CC2)CC2(CCOC2)C1 91545,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 91546,c1(C(N(C)C)=O)ccc2c(c1)CCC2NC(=O)C(c1ccccc1)Nc1nccs1 91547,N1(C(Cc2cc(C)no2)=O)CCc2ccccc2C(NC(=O)CCCF)C1 91548,c1(CNc2c(OC)ccnc2)cnn2cccc(-c3c[nH]c4nccc-4c3)c12 91549,C=CCC(CC=C)NC(C1CCCC1NC(=O)CN(C)CCC)=O 91550,Cc1nc(N2CC(C)(NC(=O)CNC(c3cccs3)=O)C2)cc(O)n1 91551,C1(C)(CCNC(C(C)C)=O)CCN(C(=O)COC2CCN(C)CC2)C1 91552,C1(=O)CC(c2cccnc2)N1.N12CC(C1)CC2=O.C1(N(CCOC)C)CCCC1 91553,C1(NC(C23CC(C)(OCC2)C3)=O)CN(C(c2cccc(=O)o2)=O)CC12CCCC2 91554,C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1OCCN(C(c2cccs2)=O)C1 91555,Cn1cc2ccc(NC(C3CC34CCN(C(=O)CCc3cccs3)CC4)=O)cc2n1 91556,c1(C(C)NC(=O)Nc2cncc(-c3csc(=N)[nH]3)c2)c[nH]c2ccc(F)cc12 91557,c1(NC(C2CCN2c2ncncc2I)=O)ccc2ncccc2c1 91558,CC1CCC(NC(c2coc(Cl)n2)=O)CN1C(C1CCCN(C(=O)C2CC2)C1)=O 91559,c1(C2(C(=O)NCC3(F)CC(NC(c4c[nH]cc4Br)=O)C3)CC2)ccc(Cl)nc1 91560,N1(C(CC(c2ccc(C)cc2)C)=O)CC(NC(c2ccnnc2O)=O)C2(CC2)C1 91561,C(CC(C(C)C)(c1nnnn1CCCOC(C)C)NC1COCCN1C)OCC 91562,C(N=c1ccc(C#N)n[nH]1)C1C(NC(c2c(C)ccc(C(C)C)c2)=O)CCC1 91563,C1(CCCNC(C2(C(C)C)CC2)=O)CCCCN1C(c1cncc(N)c1)=O 91564,C1(NC(COCCOC)=O)CC(NC(c2coc(C(F)F)c2)=O)CC1O 91565,N1(C(c2[nH]cc(C)c2)=O)CCC(C(C)OCCNC(=O)C(F)F)CC1 91566,Cc1nc(O)nc(C)c1CC(=O)NCC1CC1NC(c1ccc(C(C)C)s1)=O 91567,CCC(CCOC)C(=O)N1CC(C)(C)CC1C(=O)NCCCO 91568,CC1CC=C(C(=O)NC(C(=O)NC2CC2(C)C(F)F)C(C)(C)O)CC1 91569,C1(NC(C2CN(C)C(=O)N2)=O)C2CC3CN(C(=O)Cc4ccc(Cl)s4)C1C3C2 91570,C1(C(=O)NCCC#N)CCC(C2CC2)N1C(=O)CC1CCSC1 91571,Cc1cccc(C2(C(N3CCC(CC(=O)N(C)C)C3)=O)CC2)c1 91572,c1(CC)ccc(Br)cc1NC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1O)=O 91573,c1(C(N2C(CNC(c3cnsn3)=O)CC(F)C2)=O)cn2c(n1)CCCC2 91574,CC1(C)C2CCC1(C)C2C(N1CCC(O)(CNC(=O)C=CC2CC2)CC1)=O 91575,CCC(F)(F)C(=O)NC1CCC(NC(=O)Cn2cc(C3CC3)cn2)C1 91576,C(=O)(C(O)C(C)C)NCCN(C(=O)C(C)n1cccc1)CC 91577,c1(C(N2CCC(N(C(CN(c3ccccc3)C)=O)C)C2)=O)cc(O)c(F)cc1N 91578,c1(C(=O)NC2CN(C(C3C(OC)(OC)CC3)=O)CC2C)c(C)cccc1Cl 91579,C(CC1=CCN(C)CC1)NC(C(CC(F)F)NC(CCCNC(C)=O)=O)=O 91580,CN=c1ccc(CCC(=O)N(C2CN(C(=O)CNS(=O)(=O)NC)C2)C)c[nH]1 91581,C(C(C)CC(F)(F)F)NC(C(CCN(C)C)NC(c1ccc(C)nc1)=O)=O 91582,CON(Cc1ccccc1)C(=O)CC(C(C)C)NC(=O)C(O)Cn1cncn1 91583,N1(C(C(CSC)OC)=O)CCC(C(=O)NCC2CCSC2)=C(F)C1 91584,CCCC(C)(CC)C(=O)NCCN1CCCN(C(C2(C3CC3)CC2)=O)CC1=O 91585,N1(C(=O)OC(C)(C)C)CC2CNC(=O)CCC2(NC(C)CC2CCC2)C1 91586,c1(C(N2CC(CNC(C(CCOC)C)=O)(OC)C2)=O)ccc(Cl)c2occc12 91587,C(CO)(CCCCNC(=O)CNC=O)NC(C(C(C)C)N(S(C)(=O)=O)C)=O 91588,C1(Cn2cc(C3(N(C)C)CCC3)nn2)CCN(C(=O)CO)CC1 91589,c1(CC(=O)NCCNC(=O)CCSC2C(C)(C)C2)c(F)cccc1F 91590,c1(C(=O)NC2(CC=C)CN(C(c3cc(Cl)c(C)cn3)=O)C2)ccc(C)c(F)c1N 91591,c1(C2(NC(C3(CNC(CN(C)CCO)=O)CC3)=O)CC2)ccnc(Cl)c1 91592,Cc1cccc2c(C(=O)NCC(CC(F)(F)F)NC(=O)C#CC3CC3)nccc12 91593,c1(CN(C(CC(=O)O)CC2CCCCC2)C2CC2)cc(O)nc(C2CCC2)n1 91594,N1(C(C(C)=CC)=O)CC(C)OC2(CCN(C(=O)CCNS(=O)(=O)CC)C2)C1 91595,C1(C(N(C2CN(C(=O)CC34CC(CN3)C4)C2)C)=O)CC(=O)CC(c2ccccc2)O1 91596,C1(C2CN(C(C)=O)C2)CN(C(C2CC(Cc3ccccc3)=NO2)=O)CCO1 91597,C1(C)(CC)CC(NC(c2cc(OC)cc(Cl)c2)=O)CN1C(c1cc(Cl)c[nH]1)=O 91598,C1(C)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)(C)C)CC(C)OC(C)C1 91599,c1(CC)nnc(C)cc1C(N1CCCC1C1(NC(=O)C(CSC)OC)CC1)=O 91600,c1(C(N2CC(N(C(=O)C(CCO)N(C)C)CC)C2)=O)ccc2c(C)cc(O)nc2c1 91601,C(=O)(C(C(C)(C)OC)NCC1CC=CCC1)OC 91602,CC(C)CC(O)C(C)C(=O)NCCn1cc(C(=O)NCCc2nncn2C)nn1 91603,C1(NC(COCCC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1 91604,C(=O)(C1=CCCOC1)NC(C(CO)NC(c1c(C)sc(Cl)n1)=O)C 91605,c1(CC(=O)NCC(CNC(c2cc(CC)ncc2)=O)(C)O)cc(C)cc(C)c1 91606,C(CCCC(C)NC(N1C(NC(C)=O)CCC1)=O)NC(=O)CCOCC(F)(F)F 91607,c1(OCC)ccc(C(=O)NC2CCC(NC(=O)CS(C)(=O)=O)CC2)cc1 91608,C(=O)(C1CCc2c(Cl)cccc21)NCC1(C(F)F)CCN(C(C=COCC)=O)C1 91609,c1(CNC(CC2(C)CCN2C(=O)CC2CCOC2=O)=O)cncc(O)c1 91610,C#CC1(NC(=O)CC2CCSC2C)CN(C(=O)C(C)COC)C1 91611,C1(N(CCN(C(C(C)C2(O)CCC2)=O)C2CC2)C)CCN(C2CCCC2)CC1 91612,c1(C(=O)NC(C)CCNC(C2(C)CC2Br)=O)cn(C(F)F)cn1 91613,c1(CNC(C2CCCN(C)CC2)=O)cnc2ccc(Cl)cn12 91614,Cc1csc2ccc(C(=O)NC3CC(CNC(C4CC5CC4C5)=O)C3)cc12 91615,c1(CC)cc(CC)ccc1C(N1CC2C(CNC(=O)OCC(C)(C)C)C2C1)=O 91616,C1(NC(CNS(N)(=O)=O)=O)CCCN(C(c2sccc2-n2cnnn2)=O)CC1 91617,Cn1c(CCC(=O)NC2(C)CCCCC2(C)C)nc2cc(Cl)ccc12 91618,C1(CNC(c2cc(F)cc(F)c2Br)=O)CCN(C(c2cnnc(Cl)c2)=O)CC1(F)F 91619,N1(C(C(C(=C)C)(C)C)=O)CC(=O)Nc2c(Br)cccc21 91620,N1(C(CC(C=C)CC)=O)CC2CCC1C(CNC(=O)C=Cc1csc(C)n1)C2 91621,CC1(CNC(C23CCC2C3)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 91622,N1(c2nccc(N3CCCC(C4CCN(C)C4)C3)n2)CCc2nnnn2CC1 91623,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)cn(CC(C)C)nc1C1CC1 91624,C1(C)(C(=O)NC(CC(C)NC(C(CC)F)=O)C)CNC(=O)C1 91625,C1(O)(CN(c2nnnn2CC(=O)NC2CC2)C)CCN(C(=O)CCCF)CC1 91626,Cn1nnc2cc(C(=O)NC3CN(C(=O)Cc4ccns4)CC4(CC4)C3)ccc12 91627,CC1(C)CCC(NC(C2(C)CN(C(c3cnc(C4CC4)o3)=O)C2)=O)C1 91628,N1(CC#CCC(=O)O)CCCC(C(=O)NCC(c2ccccc2)NC(C)=O)C1 91629,N#Cc1ccc2c(c1)N(C(C1(F)CCCN(C(c3ncccc3F)=O)C1)=O)CC2 91630,c1(OC)cccc(C(=O)NCC(C)N(C2CCOC2)C)c1OCCO 91631,N1(C(C2=NNC(=O)C2)=O)CC2CC(C1)CN(C(=O)CN1CCCCCC1)C2 91632,c1(CC)ncncc1C(N1CCCC1CCNC(=O)C(C)Cn1ccnc1)=O 91633,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 91634,c1(C(N(C(C(C)NC(COCCCCCC)=O)C)CC)=O)cnc(OC)nc1 91635,CC1(CNC(c2c[nH]c(=N)o2)=O)CCCN(C(=O)CCc2ccsc2Br)C1 91636,N1(C(C2(C)CC2)=O)CCN(C(c2ccncn2)=O)CC1c1ncc[nH]1 91637,Cc1cc(CN2CCN(c3ccc(C4CC4)c(C)n3)CC2)ccc1F 91638,C1(CNC(CCNC(CCC#C)=O)=O)CCOC1C=C 91639,N1(C(C2C(C)(C)CO2)=O)CC2(C(=O)NCCCC(F)(F)F)CC1CO2 91640,C(C)(C)(S(C)(=O)=O)c1cn(NC(=O)CCC2COC(CCC(=O)C3(C)CC3)C2)nn1 91641,C(=O)(C(O)CCCn1cncn1)N1CC(C)C(NC(=O)Cc2ccc(Cl)cc2)C1 91642,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(CO)N(C)C)=O)CC12CCC2 91643,C=CC(C)(C)CC(=O)NCCOC1CN(C(C2CCC(C)S2)=O)C1 91644,C(C)(C)(CC(F)C(=O)N(C)CC1COC(=O)N1)NC(c1c(C)c[nH]n1)=O 91645,C(=O)(C(C)(C)C(C)O)NC1(CC(N2CCC(C)(N(C)C)C2)=O)CC1 91646,C(N=c1nnc(C)c(C)[nH]1)C1(C)CCN(C(c2ccc(C(=O)OCC)[nH]2)=O)C1 91647,c1(NCC(C2CCCCC2)OC)[nH]c(=NCc2cc(C)cs2)nc2scnc12 91648,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C(=O)NC)C2C)c[nH]c(=N)c(C)c1 91649,N1(Cc2cc(OC)ns2)CCCOC(c2cn(CC(O)CO)nn2)C1 91650,CC(C)C(C(=O)NC1CC(CO)C12CCC2)C(C)NC(c1cocc1C(N)=O)=O 91651,C1(C(=O)Nc2cn(CCC)nc2)CC(C)CN(C(=O)CC2CSC2)C1 91652,N(C(=NCC1CC1)NC1CC2CCC1O2)CC(N1CCCC1)C 91653,c1(-c2ncc(C(N3C(CNC(c4cc(C)no4)=O)CC3)=O)s2)ccccc1Cl 91654,c1(C(=O)NC2(CC)CCN(C(C3CCCC(O)C3)=O)CC2)cc(C#N)ccc1N 91655,C1(C(N(C2CCN(C(CCC#CC)=O)C2)C)=O)CC2(CCCC2)C1 91656,c1(OCC(=O)N(C(CN(C(c2c(C(C)C)nco2)=O)C)C)C)ccccc1C#N 91657,Cc1cccc(CC(N2CCC(c3ocnc3C(=O)N(C)C)C2)=O)c1 91658,C1(CC(=O)N(C2CC(NC(c3c(C)nc(C4CC4)s3)=O)C2)C)CC2(CCC2)CO1 91659,C1(NC(c2nc(CNC(C(C)N(C)C)=O)oc2)=O)C(O)C2CCCC12 91660,C(C(O)C(C)(C)C)N(C(C(C)N(C(Cc1c(C)ocn1)=O)C)=O)C 91661,N1(CC=CC(=O)NCC2C(NC(CNS(CC)(=O)=O)=O)C2)CCOCC1 91662,C=C=CCCC(=O)N1CCC(N(CCO)C(c2ccn(CCC)n2)=O)C1 91663,CC1CC(NC(c2ccsc2)=O)CN1C(=O)CC12COCC(C1)C2 91664,Fc1cc(Cl)cc(Br)c1C(C1CC1)Nc1ncc2ccnc-2[nH]1 91665,C1(CC(=O)NC2CN(C(C34CC(C3)C4)=O)CC23CC3)CC2(CCC2)CO1 91666,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 91667,C(=O)(CC1=CCCCC1)NC1C(C)(CNC(CC2(OCC)CCC2)=O)CCC1 91668,C1(NC(c2nc(CC)oc2)=O)CC2(CCCN(c3ncc4ncn(C)c4n3)C2)C1 91669,C#Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CC2(C)C)ccc1Cl 91670,C1(CCCNC(C(C2CC(C)(C)C2)OC)=O)CCCCN1C(C1CSC1)=O 91671,c1(NC2CCC3CN(C(c4c(C(C)C)ccs4)=O)CC32)ccc([N+](=O)[O-])cc1F 91672,c1(C(N(CCCC(=O)NCCc2nccs2)C)=O)c[nH]c(C#N)c1 91673,N1(C(C2N(C(c3cc(OC)nn3C)=O)CCC2)=O)CCc2ccc(C#N)cc2C1 91674,C(=O)(C(COCC)CC)NCCC1CCC(CNC(C(CC)OCC)=O)CC1 91675,C(=O)(C(C)S(N)(=O)=O)NCCn1ncc(C(N(CC(CC)C)C)=O)c1 91676,N1(C(C(n2nnnc2C2CC2)C)=O)CCCC1(C1CC1)C(=O)O 91677,C1(C)(COC)CN(C(C2(n3cccn3)CCN(C(=O)OC(C)(C)C)CC2)=O)CCO1 91678,Cc1nc(C(N2CC(F)CC2CN(C)C(C2CNC(=O)C2)=O)=O)cn1C 91679,CC(C)(C)C(CC(=O)O)NC(=O)C(c1cc(Br)co1)=O 91680,N1(C(C2(CC=C)CC2)=O)CCN(C(=O)CCc2ccsc2)CC1C 91681,N1(C(CC(C)c2ccco2)=O)CC(O)CC1C(=O)Nc1nc[nH]n1 91682,C#CC1(O)CN(C(=O)CCOCCN(C)C(C2CCC(CC)CC2)=O)C1 91683,CC#CCCC(=O)N1CC2C(C1)SCCO2.C(=O)(CCCS)NC.OC 91684,C1(O)(CN(C(=O)CC2CCC(=O)N2)C)CN(C(=O)CCc2cnoc2)C1 91685,c1(-c2cn(C3CC(C(=O)NCCCC(C)(C)OC)C3)nn2)ccc(C(C)C)cn1 91686,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCC2)=O)COC(C)(C)C1 91687,N1(C(CNC(C(C)(C)C)=O)=O)CCOC(C)(CNC(C2CC2(Cl)Cl)=O)C1 91688,C1(C(=O)NC(CNC(c2ccc(C)[nH]2)=O)C(C)(C)C)COC2(CO)CC1C2 91689,C#CCC(CC(F)F)C(=O)OCc1ccc(C)cc1 91690,CCC(CC)CC(F)C(=O)NCC1CC(CNC(c2cnc(C)cc2C)=O)C1 91691,N1(C(c2ccc(C(C)C)o2)=O)CC2(C)CC1(C(N1CC3(CCC3)C1)=O)C2 91692,c1(C(=O)NCC2(F)CC(CNC(COC)=O)C2)ccc(N2CCCC(O)C2)cc1 91693,C(C1=CCN(Cc2cc(Cl)cc(Cl)c2)CC1)NC(c1c(CC(C)C)cccc1)=O 91694,C1(OC)CC(CC(=O)N(CCCCN(C(=O)C(C)(C)CO)C)C)C1(C)C 91695,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 91696,N12CC3(CC(CO3)C(C)n3ccc(n3)C1=O)C2.C1(OCCNC=O)CC1(F)F 91697,C=CCCCCCCC(=O)N1CCN(C)C(CNC(C2CCCC2CC)=O)C1 91698,c1(OC)cccc(OC)c1C(=O)NC1CCC(NC(=O)CCC(C)C#N)C1 91699,C1(NC(c2c(OC)nsc2)=O)CCN(C(c2nn(C)nc2Br)=O)CC1F 91700,c1(C(=O)NCC2C(NC(C3(OC)CCC34CCC4)=O)CC2)cc(F)c(F)c(F)c1 91701,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCn2cc(Cl)cn2)C1)OC 91702,Cc1nc(C2CC2)ncc1C(=O)NCC1(C)CC(NC(c2cc(Cl)c[nH]2)=O)C1 91703,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 91704,C1(CCCNC(CC2(OC)CCCC2)=O)CCCCN1C(C1CC(C)(C)C1)=O 91705,C=C(Cl)CN=c1[nH]c(=NCc2ccc(C)nc2)[nH]c2cc(SC)ccc12 91706,Cc1ccc(C(N2CC(NC(=O)CN(CC(C)(C)C)C)C(O)C2CO)=O)c(F)c1 91707,CCC(CCC(=O)N(CC(=O)OC)C1CC1)NC(=O)CCF 91708,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 91709,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC(C)C)CNC(=O)CCc1cnn[nH]1 91710,N1(C(c2c(C#C)c[nH]n2)=O)CC(CNC(=O)CCC(CC)CC)OC2(CCC2)C1 91711,c1(N(C)Cc2ccccc2[N+](=O)[O-])ccc(S(=O)(=O)NCC2CCCCS2)cn1 91712,C(CCCC(=O)N(C)Cc1nnnn1C)NC(C1C(CC)OCC1)=O 91713,C1(CC)COC(C)(C)CN1C(C1C(C)CCN1C(c1cnc2ccnn2c1)=O)=O 91714,N1(C(C2C(=O)NCC2)=O)CCOC2CN(C(c3csc(C4CCCO4)n3)=O)CC12 91715,C1(N(C(c2c(C)nns2)=O)C)CCC(NC(=O)C(C)Cc2cccc(Cl)c2)CC1 91716,O(NC(=O)C(=O)C(C)(C)C)CC(N1CC(C)CC(C(=O)NC)C1)=O 91717,CC1CN(C(C2(CO)CCCC2)=O)CCN1C(C1CCC(=O)NC1)=O 91718,N1(CC(N2CCC(N(C(=O)CCC3CCC3)C)CC2)=O)C(=O)NC(C)(CCO)C1=O 91719,C1(CC(=O)NCC2(CNC(C3N(C(C)=O)CCOC3)=O)CCC2)COCC(C)(C)O1 91720,N1(C(COCCCC)=O)CCN(C(C2(C)CCC(OC)C2)=O)CC12CCC2 91721,C1(CC#C)(C(=O)O)CCN(C(=O)Cc2cc(C)sc2C)C1 91722,C1(C(C)O)CCCN(C(c2c(CNC3CCC(=O)C3)cnn2C)=O)C1 91723,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 91724,c1(C(=O)NCc2c(SC)cccc2)cnn2ccc(-c3ccnc(O)c3)cc12 91725,O=C(C=CC(F)F)NN1CCCC1NCc1nc[nH]n1 91726,C1(NC(C2C(SC)CCC2)=O)CC2COCC(C1)C2NC(=O)Cc1nccn1C 91727,C1(C(N2CCN(CCNC(=O)CC3=CCCC3)CC2)=O)CC2CCCCN2C1 91728,c1(-c2cn(C(C(=O)Nc3c(CC)sc(C)c3)C)nn2)c[nH]c2ccccc12 91729,Cc1nc(C(=O)N(C)C)ncc1NC(=O)C=Cc1ccsc1 91730,C1(C(=O)NC(C)C(=O)NCC(=O)N(CC(F)F)C)(CSCC)CCC1 91731,C1(C(C)NC(C(c2cccc(O)c2)C)=O)CCN(C(=O)C=CC2CCCC2)CC1 91732,CCC(C)(CC)C(=O)N1CCC(CNC(=O)C(C)Oc2cccnc2)C1 91733,c1(C(N2CCC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)=O)c(Cl)cnn1C 91734,c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C2CC2)ccc(F)cc1F 91735,c1(CC(C(=O)NC(C)(CNC(c2ncccc2Cl)=O)C2CC2)O)c(F)cccc1F 91736,C(=O)(C#CC1CC1)NCC1CC(C(=O)NCC#CCOC)C1 91737,c1(C(=O)OC)coc(C=CC(=O)N(CC(C)N(C(=O)Cc2ccon2)C)C)c1 91738,N1(C(c2scc(CC)c2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)CC(C)(C)C1 91739,c1(C(=O)NC2CC(NC(C3(SC)CCC3)=O)C2)ccc2nc(CO)[nH]c2c1 91740,C1(C(N(CCCNC(=O)Cc2cc(CF)on2)CC)=O)CCC(OC)CC1 91741,C1(CNC(C2CCCC3CC23)=O)CCCC12CCN(C(C1CCCC1O)=O)CC2 91742,c1(OC)n[nH]c(C(=O)NCC2(CNC(=O)Cc3cnc(C)s3)CC23CCC3)c1Cl 91743,N1(C(C(=O)NC(CC)COCP(C)(C)=O)=O)CCc2ccccc21 91744,C1(CNC(C(C=C)O)=O)CC(F)CN1C(C1CCC(C)O1)=O 91745,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 91746,c1(C(N2CC=CC(NC(C3(C(C)C)CCOCC3)=O)C2)=O)onc2ccccc12 91747,c1(C(C)NC(=O)C(C)(C2CC2)N(C(=O)CSC2CC2)C)ccccn1 91748,N12CC(C(C(C)C)C1)C2=O.n1(C(C)C)cnc(C(=O)NOCC(C)O)c1 91749,C(=O)(CCCCC(N)=O)N(C1CC1)CC1N(C(CCOC(CC(C)C)C)=O)CCC1 91750,C1(N(C(c2onc(COC)n2)=O)C)CCC2CN(C(=O)C=CI)CC12 91751,CON(C)C(=O)CNC(=O)CCOCCCNC(C12CCCCC1C2)=O 91752,Cc1nn(CC(N2CCN(C(=O)CN(C3CCSC3)C)CC2)=O)c(C)c1C 91753,C1(C(N(CCN(C(C)C)C(C2CC2(C)C)=O)C)=O)COCCO1 91754,c1(NC(C2(COC)CC3CC2C3)=O)ncnc(N(C)C)c1C 91755,c1(CC(=O)NCCCCN(C)C(C2CCCS2(=O)=O)=O)c[nH]c2ccccc12 91756,Cc1ccc(Cl)c(N)c1C(=O)NC12CCN(C(c3ncccc3O)=O)CC1C2 91757,CCCC(C(=O)NCC1CCC(NC(=O)CCc2ccc(O)c(F)c2)C1)C(C)C 91758,c1(C(=O)NCCC(=O)NCC2C(C)CCO2)ccc(CC#N)cc1 91759,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 91760,CC1(C)CC(NC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(C2(C)CC=CCC2)=O)C1 91761,C1(C(C(=O)NCCN(C)C)O)CCN(C(C2CNC(=O)C2)=O)CC1 91762,c1(NCC(CNC(C2(C=C)CCC2)=O)C)ncnc2c1nnn2CC 91763,Cc1c[nH]c(C(=O)N(C)CC2(CNC(c3cc(N)c(F)cn3)=O)CC2)cc1=O 91764,C(CCC(C)C)(C(=O)NC1CCCC1(C(=O)OC)OC)N(C)CC.c12nccn1C2 91765,c12cccc(c1C)NC(=O)C2.c1(C(N2CCCC2C)=O)sc(Br)nc1C.CO 91766,C1(C(N(CC(=O)N(C)C)CCC)=O)CCCN(C(=O)C2=C(Cl)CC2)C1 91767,c1(NC(COCCCNC(C(c2n(C)ncc2)O)=O)=O)ccc2c(c1)COC2 91768,c1(C(N(CC(C)(C)NC(C2CCCC2(F)F)=O)C)=O)ccc([N+](=O)[O-])o1 91769,C=CC1CN(C(c2ccno2)=O)CC1NC(c1ccc(C2CC2)c(F)c1)=O 91770,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C)c(F)cccc1F 91771,C1(CCC(=O)NCC(C2CC2)SC)CCCN1C(=O)CCn1cccn1 91772,c1(C(N2CCN(C3(S(C)=O)CC3)CC2)C)ccc(Cl)cc1 91773,CCC(CO)C(=O)NCCc1nc(-c2ccc(Cl)cc2)cs1 91774,C1(c2occc2)CCCC(c2nc(-c3ccc(Br)s3)no2)O1 91775,c1(NC(C2CCN2Cc2cnn(-c3ccccc3)c2)=O)cccc(Br)c1I 91776,c1(C(N(CCC(C)(C)NC(CC(CC)C)=O)C)=O)cn2ccc(C)cc2n1 91777,c1(NC(C)CN(C(C(C(C)C)SC)=O)C2CC2)c(F)cccc1[N+](=O)[O-] 91778,c1(C(=O)NCC(C2CCCCC2)NC(C(C)N(CC)CC)=O)ncc(Cl)cc1Cl 91779,c1(OC)ccc(Cl)c(F)c1-c1cccc(C(=O)NCC2CC(O)C2)n1 91780,c1(OC)ccnc(NCC(=O)NC(C)C(C)(C)NC(=O)CC2(C)CCCCC2)n1 91781,C1(C(F)F)(OC)CCCN(C(c2nc(Cl)oc2C)C(=O)NC(C)C)C1 91782,N1(C(=O)NCC(c2cc(C)c(F)cc2)=O)CCc2ccncc2C1 91783,Cc1c(C(CCN(C(c2c[nH]nn2)=O)CCO)C(=O)O)cccc1Cl 91784,C1(NC(Cc2ccc(C)s2)=O)CN(C(=O)C(F)n2ccnc2)C2CCCC12 91785,c1(-c2onc(-c3ccc(-n4c(C)cc(C)n4)cc3)n2)cc(F)c2nc(C)cn2c1 91786,CCCCC(O)C(=O)NCc1cn(C2CCCN(C(=O)CCCOC)C2)nn1 91787,c1(CCC)ccc(F)cc1C.C1C(CC(C)C)N1 91788,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 91789,C1(C(=O)NCC2(C=C)CCC2)C2CCCC2CN1C(C1CCC2(CCC2)C1)=O 91790,C(C(CNC(C1CCS(=O)(=O)C1)=O)S(C)(=O)=O)NC(C1(CC#C)CC1)=O 91791,c1(C(=O)NC2CC(C(C)NC(c3c(CC)nccn3)=O)C2)cc(Cl)c(Cl)n1C 91792,C=C=CCC(=O)N1CCC(N(C(c2cn(C(F)(F)CO)nn2)=O)CC)C1 91793,C(C(CC1CC1)C(=O)NCC1CC12CC2(F)F)NC(c1n(CCC)ccc1)=O 91794,N1(C(c2coc3c2COC3)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 91795,CC(C)CCC(=O)C(=O)N1CC(C2CC2C(N2CCC(CCCO)C2)=O)C1 91796,C1(O)(CNC(c2cc(CNC(CCC=CCC=C)=O)no2)=O)CCC(C)C1 91797,C#CCC(C)C(=O)N(CC(C)NC(c1ccc(-c2cn[nH]c2)cc1)=O)CC 91798,c1(OCCCC(=O)NC(CNC(C(C)OCOC)=O)(C)CO)ccccc1Cl 91799,CC(CC(F)(F)F)C(=O)N1CCC(O)(CN(C(=O)C(F)CC2CCCCC2)C)C1 91800,c1(CC)cc(C(N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)=O)ccc1F 91801,C(C1CCCO1)=CC(=O)NCCC(C)N(C(=O)CCC1CCC1)C 91802,C(=O)(CCP(C)(C)=O)N(CC)CC1CCCN1C(=O)Cc1sc(O)nc1O 91803,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 91804,CC(C)(C#N)CCCC(=O)NCC1C=CC(NC(c2c(F)cccc2F)=O)C1 91805,C1(NC(C(C=C)CC)=O)(CNC(c2csc3cncn23)=O)CC2CCC1CC2 91806,C12(C(N(C(C)CNC(=O)OC(C)(C)C)C)=O)CCC1CN(C(CCS(C)(=O)=O)=O)C2 91807,c1(C(=O)NC2(C)CN(C(COC(C)C)=O)C2)cc(C2CC2)ccn1 91808,C1(CNC(C(C2CC2)OC)=O)C(C)CCCN1C(c1cn(CCCF)nn1)=O 91809,Cc1cc(C(N2CCC2C(=O)NCC2CCOC2)=O)oc1C 91810,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 91811,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN2C(=O)CC2CCCCC2O)C1 91812,c1(C(N2CCC(C(CO)NC(c3c(C)onc3)=O)CC2)=O)ccc2nonc2c1 91813,C1(C(=O)Nc2ccc(OC(C)C)cc2)CN(Cc2cnc(Br)c(F)c2)CCC1O 91814,C1(NC(CC(C)OC)=O)CCS(=O)(=O)C12CN(C(C1CCN(C(C)C)CC1)=O)C2 91815,c1(C(C(=O)NCCC)N(C)Cc2cccnc2)cnn(CCF)c1 91816,C1(C(=O)NCc2ccc(C)c(Cl)c2)CCN(C(=O)CC2CCCCC2)C(C)(C)C1 91817,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)cc1Cl)=O 91818,C(c1c(F)cccc1F)=CC(=O)NC(CC)CNC(c1ccc(C(N)=O)[nH]1)=O 91819,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 91820,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2CC1 91821,n1(C(C)C)cnc2c(N(C)Cc3nc[nH]n3)[nH]c(=NCc3nncs3)nc12 91822,N1(C(c2c(COC)cco2)=O)CCCOC(CNC(c2ncsc2C)=O)C1 91823,c1(C(=O)NCCCN(C(C2CC(C)(F)C2)=O)CC)cc2n(n1)CCCNC2=O 91824,C1(O)(CNC(COCC)=O)CN(C(c2cnc(OC)s2)=O)C1 91825,N1(C(c2c(C)cccn2)=O)C2CCC1CN(C(C1CC3C=CC1C31CC1)=O)C2 91826,C1(NC(CC)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 91827,c1(NC(CN2CCC(CSC)CC2)=O)cc(-c2nn[nH]n2)c(F)cc1F 91828,c1(C(=O)NC2C(OC)CN(C(c3cccnn3)=O)C2)ccc(F)c(SC)c1 91829,C1(O)(C(N(CCNC(Cc2ccn(CC)n2)=O)CC)=O)CCC(C)(C)CC1 91830,Cc1ncc(CC(=O)NCCCN(C(=O)C=CC2CCCO2)CCO)[nH]1 91831,N1(C(C(CC)(F)F)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)CCC2C1 91832,c1(C(N2C(C)(CNC(C(C)OCC#C)=O)CCC2)=O)ccc(Cl)cc1O 91833,c1(C(N2CCCOCC(CNC(C(C)C3CC3)=O)C2)=O)coc2ccc(O)cc12 91834,c1(NC(C2N(C(C3CCC(=C)CC3)=O)CC2)=O)cc(F)c(C)cc1F 91835,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 91836,c1(C(=O)NC2(CN(C(C3C(OC)C3)=O)C)CC2)cnc2[nH]c(C)nc2c1 91837,c1(C(=O)NCC2CN(C(C3(CCC=C)CC3)=O)CC2O)nc2n(c1Cl)CCCC2 91838,c1(C(N(CCNC(=O)Cc2ccsc2)CC2CC2)=O)cccnc1-n1ccnc1 91839,N1(C(CCOC(C)C)=O)CCCC2(C1)C(NC(c1cc(F)n[nH]1)=O)CCN2C 91840,c1(C(=O)NCC(CC)(C)NC(c2csc(COC)c2)=O)nc(O)sc1C 91841,N1(C(CN(C)CC2C(C(=O)NCCC#C)C2)=O)CCCC(SC(C)=O)C1 91842,c1(C(N2CC3(N(C(C(C(C)C)SC)=O)CC3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 91843,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(c2ccc(NC)s2)=O)C12CCC2 91844,C1(CC)COC(C)(C)CN1C(C1(F)CCN(C(=O)CN2CCC(F)CC2)C1)=O 91845,Cc1cccn2c(C(=O)OC(c3ccccc3)CN)cnc12.C1(C)C(=O)N1 91846,c1(OC)cc(Cl)ccc1C(N1CCC(CNC(c2ncc[nH]2)=O)C(C)C1)=O 91847,CCCCCC(C)NC(=O)C(c1cn(C)nn1)NC(c1ccc(F)s1)=O 91848,C1(C(=O)OCC2(OCC)COC2)CSC(CCC(F)(F)F)C(=O)N1 91849,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)Cn2cccn2)CC1 91850,N1(CC(=O)OC)CCN(Cc2ccc3c(c2)CC3)CC1=O.c12cc(cs1)NC(=O)C2 91851,c1(C(N2CCN(CCCNC(C3(C)COCCO3)=O)CC2)=O)cnn2c1OCC2 91852,C1(CNC(=O)COCC(F)(F)F)CCCN1C(C1(c2cc[nH]n2)CC1)=O 91853,Cc1cc(C(=O)NCC2CC2C(=O)NCCn2ccc(CO)n2)ccn1 91854,c1(C(N(C)CC2N(C(c3c(C)nns3)=O)CCC2)=O)cnc2nc(O)ccc2c1 91855,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1coc(CO)c1)=O)C3 91856,c1(CNC(C2CSCN2C(c2ncon2)=O)=O)cc(F)c(F)cc1F 91857,C1(C(=O)Nc2n(CCCSC)nnn2)CCCC(NC(C2(C)CCC2)=O)C1 91858,c1(CCC(=O)N(C(C(C)=CC)=O)C2(CC(=O)OC)CC2)ccn(C)n1 91859,CN1CCN(C(=O)CC2CCC2)CC1CNC(C1(C)CC=CCO1)=O 91860,c1(CNC(C(=O)NCc2ccc(SC)cc2)=O)ccc2c(c1)CCO2 91861,Cc1cc(C(=O)NCCC2CC(NC(=O)Cc3ccsn3)C2)n2nc(C)cc2n1 91862,N1(C(C=CSC)=O)CC(NC(C2(n3cnnn3)CC2)=O)CC12CCCCC2 91863,CC1(C#CC(=O)NC2CCCC(NC(c3cc[nH]n3)=O)CC2)CC1 91864,Cc1onc(C)c1C(=O)NC1C2CC(NC(C3CCCC3C)=O)CC12 91865,CN1CCC(C2CCCN2C(C2CC2C(=O)NC(C)(C)CNC(N)=O)=O)CC1 91866,N1(C(C2N(C(C)=O)CCCC2)=O)CCCC(O)(CN(C(=O)C(F)(F)C2CC2)C)C1 91867,C1(NC(Cn2c(C)ncc2)=O)CN(C(C2(C)CCCO2)=O)CC(C)(C)C1 91868,N1(CC)CCCC2CC(O)CCC12.c12cc(OC)cc(c1)N2.N12CCC(C1)C2 91869,N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NOCCCN3CCC3)CO2)C1 91870,C1(NC(C)CCc2ccccc2)CCC2CC1C2(C)C 91871,c1(C(=O)NCCN(CCC)C(c2cc(C(C)(C)C)nn2C)=O)cc(C)nc(N)c1 91872,C1(CC(N2CC(O)(C(C)NC(c3ccc(OC)o3)=O)C2)=O)CCCOCC1 91873,C1(C(N2CC(=C(C(=O)NC3(C)CCN(C)C3)F)C2)=O)CC2(CC(OC(C)=O)C2)C1 91874,CON1CCC(C(=O)NCc2nc(CNC(c3cc(=O)n(C)o3)=O)cs2)CC1 91875,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 91876,N1(C(C23N(C(Cc4nn(C)c(Cl)c4)=O)CC(C)(C2)C3)=O)C2CCC1CC(C(N)=O)C2 91877,c1(NC(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C(C)C)ccc([N+](=O)[O-])cc1Cl 91878,N=c1nc2c(c[nH]1)CC(C(=O)NCC13CC(CN1C(C1COCCO1)=O)C3)CC2 91879,C1(CNC(C2(COC)CN(C(CCC=C=C)=O)C2)=O)CCC2(CCC2)O1 91880,C1(NCCN(C(=O)CCC#Cc2ccccc2)CC)CC(c2ccc(C)cc2)=NO1 91881,C1(NC(C(N2C(CC)CCC2)=O)=O)CCCCN(CCCSc2ccccc2)C1 91882,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 91883,C1(CNC(=O)C(=O)Nc2nnc(-c3ccccn3)s2)CCCN2CCCC12 91884,c1(NC(c2scc(-c3ccc(CNC)cc3)n2)=O)cc2n[nH]cc2cc1C 91885,c1(C(=O)NCC(CC(C)C)NC(=O)C(C)OCC2CCC2)cnn2c1NCCC2 91886,C1(NC(Cc2c(C)con2)=O)CCCCN(C(=O)C(F)C(C)(F)F)C1 91887,c1(NC)cnn(C)c1S(=O)(=O)NC(=O)C(=O)NCC1OC(=O)CC1(C)C 91888,Cn1ncc(Cl)c1C(=O)NCC1CCCN1C(c1cncn1C1CC1)=O 91889,N#Cc1c(NC(=O)NCC(=O)NCc2ccc(Br)o2)cccc1Br 91890,C1(OC)CCC2CN(C(=O)CC=CCNC(C3(CO)CCC3)=O)CC12 91891,C#CC1(C(=O)NC2CN(CC)CC2C)CCN(C(c2ccc(O)nc2)=O)C1 91892,C1(CN(C(=O)C(=O)NCC(C2CC(F)(F)C2)OCC(F)(F)F)C)C2CCCC12 91893,C(C(C)(C)C(=O)NC1CCC(C(N2CCCC2)=O)C1)NC(CC(=O)OC(C)(C)C)=O 91894,Cc1cc(F)cnc1C(=O)NC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1 91895,N1(C(C=C(C)C)=O)CCC(N(C(c2cnco2)=O)CC2CC2)C1 91896,C1(C(N2CC(CNC(c3ccc(OC)nn3)=O)C(O)C2)=O)Cc2cccnc2C1 91897,C(N=c1cc(C)nc(C)[nH]1)C1N(C(CCCCCN(C(C)=O)CCO)=O)CCC1 91898,C1(C(=O)NCC(C2CCC2)NC(C(c2cccnc2)C)=O)CCC2CC1C2(C)C 91899,C(CC1CCc2ccccc21)OC(c1c(C#C)cn(C)n1)=O.C12CC(F)CN1C2=O 91900,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)CCCC(F)F)C1(C)C 91901,c1(C(=O)NC(C)CNC(=O)CC(C)N(C)C)cc(Cl)cc(F)c1N 91902,C1(CNC(CCCOC)=O)CC(C)CN(C(C2CCC(CO)CC2)=O)C1 91903,C=C=CC(C)C(=O)N(C)CC1CCCN1C(=O)C(C)CCc1cccc(F)c1 91904,c1(NC(COCC(n2cc(CCO)nn2)C)=O)ccc(-n2cc(Br)cn2)cc1 91905,C=CCC(Cc1ccccc1)C(=O)N(C(C)CNC(C1CC(F)C1)=O)C 91906,c1(C(=O)NCC2(CCNC(C3CC3(F)F)=O)CC2)ccc2c(c1)B(O)OC2 91907,c1(C(=O)NC2C(NC(CC(CC(C)C)C)=O)CCCC2)cc2nn[nH]c2cc1F 91908,N1(C(C(C2CCOC2)OC)=O)CC2(CCN(C(c3cc(N)c(F)cc3C)=O)C2)C1 91909,N1(C(C(c2cncnc2)C)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(C2CC2)C1 91910,c1(C(=O)NCC#CCNC(c2nc(C(=O)NCC=C)sc2)=O)nccn2nccc12 91911,C(=O)(CC1OCCc2ccccc21)N1CCC(C)(NC(=O)CC2(O)CCC2)CC1 91912,C1(=O)C(C(F)(F)F)CN1.CCCCC(=O)NC1(CNC(=O)OC)CCCC1 91913,Cn1ncc(C(=O)NC2CCC(n3cc(-c4ccccc4)nn3)CC2)c1C1CC1 91914,N1(C(CC2(N(C)C(C3C4CCC(=O)C34)=O)CC2)=O)CCC2(CCO2)C1 91915,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(C2CSC2)=O)CC1 91916,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 91917,N1(C(C2CN(CC(C)C)C(=O)C2)=O)CC2(CCN(C(c3ccon3)=O)CC2)C1 91918,N1(C(C2(C(N)=O)CCC2)=O)CCC2(C=C(C(=O)NC3CC(n4cncn4)C3)C2)C1 91919,c1(NC(CC2(C)CCN2C(=O)C(C2CCCCC2)F)=O)ccc2c(c1)OCC2 91920,c1(NC(N2CCSCC(C)C2)=O)ccc(S(=O)(=O)CF)cc1 91921,CC1C2CC(C2NC(=O)CC(C)(C)C)N1C(=O)N1CCC(CC(=O)NOCCO)C1 91922,C1(CC(=O)N(CCCCCO)CC)CN(C(=O)Cc2cccc(O)c2)CCO1 91923,c1(C(N2C(C(=O)NC(c3ccccc3)C#C)CC2)=O)cc(F)c2cc[nH]c2c1 91924,c1(C(C(N2CC(COC)(CNC(=O)C(O)CC3CC3)C2)=O)CO)ccc(F)cc1 91925,N1(C(C(CC)F)=O)CCN(C2CCN(C(=O)CCNC(C3CCCO3)=O)C2)CC1 91926,C(=O)(C1CNCc2n[nH]cc21)N1CCC2(CC(C(=O)NCC(N)=O)OC2)C1 91927,C(=O)(CC(C)(O)COC)NC(CC)CNC(c1ccccc1OC(F)(F)F)=O 91928,N1(C(CO)=O)CCC(OCCOCCCCC)CC1.C(=O)(C(O)C(C)C)NC 91929,C1(NC(CCC(C)N(C)C)=O)CCN(C(c2cnc(N)c(N)c2)=O)CC1C 91930,C1(CNC(CN(C2CCCC2)C)=O)(NC(C2(C)CC2C)=O)CC2CCC1CC2 91931,c1(CCC)cc(C(N2CC(CCNC(=O)CSc3nccn3C)C2)=O)n(C)n1 91932,c1(CCNC(C=C(C)CNC(C2CC(C#N)C2)=O)=O)csnc1C 91933,c1(OC)cc(Cl)ncc1NC(C1C=CC(NCc2nccnc2Cl)C1)=O 91934,N1(C(CCC=CC)=O)CCC2CN(C(C3CC34CCCC4)=O)CCC12 91935,C#Cc1cn(C)nc1C(=O)NC1CCCCC1CC(=O)NCC(F)(F)CO 91936,c1(CNC(C2N(C(C)=O)CCC2)=O)ccc(O)c(C)c1.C12C=CC(C1)NC2=O 91937,c1(CNC(=O)NC2CC(C)(COC)C2)cccc(CO)c1 91938,C1(NC(N2C(c3ccc(C)cc3)CCCC2)=O)CCc2ncc(Br)n2C1 91939,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 91940,C(c1cnc[nH]1)=C(C)C(=O)NCC(CNC(=O)CCCNC(N)=O)CO 91941,N1(C(C(CC)(C)C)=O)CCC(C2(NC(=O)CC3CCOC(C)(C)C3)CC2)C1 91942,CCC(C)C(O)C(=O)Nc1cccc(NC(=O)CC23CCCC2C3)c1 91943,CC1(CC(=O)NCC2COCC2NC(c2cc(Br)no2)=O)CCOCC1 91944,c1(C(=O)NC2CC(F)(CNC(C=CCC)=O)C2)cccc(COC)c1OC 91945,c1(OC)cc(C)ccc1OCCCn1nnnc1C(C)(CC1CCC1)NCCF 91946,NC1CCN(C(c2csc(-c3ccco3)n2)=O)C(CO)C1 91947,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CCO)C1 91948,N1(C(C(C(C)C)SCC)=O)CCOC2(CCN(C(C3COC(=O)O3)=O)C2)C1 91949,C(C(C(=O)N1CCC(NC2CC2)C1)NC(=O)C=CC(=O)N(C)C)SCC 91950,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 91951,Cc1cn(C2CCC2)[nH]c1=NC(=O)c1cc(-c2nc3ccccc3o2)ccc1F 91952,C1(CNC(CN(C2(C)CCC2)C)=O)CCN(C(c2csc(CC3CC3)n2)=O)C1 91953,CC1Oc2c(C(=O)NC(CNC(=O)C(C)(F)F)C3CC3)cccc2NC1=O 91954,CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN(C(C2CCOCC2)=O)C1(C)C 91955,N1(C(=O)CC2CCS(=O)(=O)CC2)CCN(C(=O)C2=CCCOC2)CC(O)C1 91956,C1(C(=O)NC(CC)CNC(c2cnc(O)c(OC)c2)=O)CCc2nc(C)cn2C1 91957,c12ccc(cc1)n2C.c1(C(C(=O)NC2CC2)NCCCC2CC2)ccc(Br)cn1 91958,CN1CC2C(CNC(=O)NCC3(NC(=O)CNC(=O)C4CC4)CCC3)C2C1 91959,Cc1cc(CNCC(=O)NC(c2cccc(Br)c2)C(F)(F)F)ncn1 91960,C(C(C)(C)C(=O)NOCCN(C)C)NC(C(C)CSC(F)(F)F)=O 91961,c1(C(=O)NC(C2CCN(C(C3(OC)CCCOC3)=O)CC2)C)cnc(Cl)cc1N 91962,c1(CNCCC(=O)Nc2c(C)nn(C)c2C)cc(C#N)ccc1Cl 91963,C1(C(C)C)CCC(CC(N)C(N2CCCC(C(C)C)C2)=O)CC1 91964,C=C(C)C(C)(O)C(=O)NC1CCN(C(=O)COc2cccc(Cl)c2Cl)CC1CC 91965,Cc1ncnc(C(=O)NCC(C)(C)NC(=O)CCCN2CCCCC2)c1C 91966,c1(N2C(C)CN(C(=O)CC3CCC(C)CO3)CC2)ccc(Cl)cc1[N+](=O)[O-] 91967,C(=O)(C(CC(C)C)N(C1CC1)Cc1ccccc1Br)OC.C1(=O)C(c2cccs2)O1 91968,CC1CN(C(C2C3CCN(C(C4CC(=O)OC4(C)C)=O)CC23)=O)C12CCOCC2 91969,N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCCN(C(c3cc(O)no3)=O)C2C1 91970,N12CCC(O)(CC1)CC2=O.C(C(F)F)(C(C)(C)C)NCc1cccc(CSC)n1 91971,c1(C(N2CC(CNC(C(CCC)C)=O)C(O)C2)=O)ccc2cc[nH]c2n1 91972,c1(C(=O)NC2(C)CCN(C(C(C)(C)CC3CC3)=O)C2)nccc2[nH]ccc12 91973,c1(CC(=O)NCc2nccc(N3C(CC)CN(C)CC3)n2)ccc2c(c1)COC2 91974,Cc1cccc(C(=O)C(=O)Nc2cccc(CNC(=O)CC(C)C)c2)c1 91975,c1(CC(O)COCCOC)cn(C(C)CNC)nn1.C(C)(C(=O)NC)SCC 91976,CP(C)(=O)c1ccc(C(=O)NCC23CCCC(CN2C(=O)COC2CC2)C3)nc1 91977,N1(C(c2c(CC)ccs2)=O)CCC2(CC(C(N3CCCCCCC3)=O)C2)C1 91978,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)COCC(F)(F)F)C2)C1 91979,c1(C(N2CCC(CN(C(C(F)OC)=O)C)C2)=O)cccc2ccc(O)nc12 91980,C1(C(N(c2nnc(COC)s2)C)=O)CCCN1CC(C1CCCC1)O 91981,C1(C(CO)N(C)C(c2cc(C(=O)NCC3(F)CC3)[nH]n2)=O)CCCCC1 91982,c1(C(N2CCC(NC(c3c(C(=O)OCC)cco3)=O)C2)=O)c(C)noc1Cl 91983,Nc1ncnc2c1ncn2CCCCC(=O)Oc1cccc2c1ncn2C 91984,c1(CNC(Cc2nnc(C)o2)=O)nc(C)c(C(=O)NC(C2(C)CC2)C)o1 91985,c1(C(=O)NC(C)CCCNC(C2(C)CC2(Cl)Cl)=O)ccccc1Br 91986,c1(C(N(CC(C)(C)NC(C2CCS2(=O)=O)=O)C)=O)cn2c(n1)C(=O)N(C)CC2 91987,C(=O)(C(C)C(C)NC(=O)CCN(CCCO)C(c1cnns1)=O)OC 91988,CC(C(=O)NC(C)CCN(C)C(c1ccc(C2CCOC2)cc1)=O)C(C)(F)F 91989,c1(C(N2CCOC(COC(c3ccc(Cl)cc3)=O)C2)C)ccc(F)cc1 91990,C12(C)CCCN1C(=O)CNC2.C1(C(C)=O)CCCCC1C.C12(CCCC1)CC(=O)N2 91991,n1(CC)ccc(C(=O)NCC2(CNC(=O)CC=CC(C)(C)C)CCCCC2)c1C 91992,C1(C(=O)NCC2C(NC(CSCCC#N)=O)CCCC2)CCC2CCCCN12 91993,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 91994,C(CC(CC)C(=O)NCC1CCN1C(C1CCCC(C(C)C)C1)=O)=CC 91995,S(=O)(=O)(c1c[nH]ccc1=NC1CC(C)(C(N)=O)C1)NCc1c(C)nn(CC(F)F)c1 91996,N1(C(C(CC)(C)CO)=O)CC(NC(c2cn(C(F)F)cn2)=O)C(N=[N+]=[N-])C1 91997,C1(C(=O)NC2CC(C)CN(C(C3CC(=O)CS3)=O)C2)(OC)CCC(C)(C)C1 91998,Cc1cc(C(=O)NC(C2CCCC2)CNC(=O)CSc2nc[nH]n2)cc2nc[nH]c12 91999,N1(C(C(CC)=CC)=O)CCCC(C(C)(C)NC(C2CCCCC2O)=O)C1 92000,C(=O)(C1=CC2(CCN(C(C3(N(C)Cc4ccc(CC)cc4)COC3)=O)C2)C1)OC 92001,c1(NC)cncc(C(N2CCCC(CN(C(=O)Cc3cc[nH]c3)C)C2)=O)c1 92002,c1(C(=O)NCC2(OC)CN(C(C3CCC(CC)C3)=O)C2)cc(OC)cc[n+]1[O-] 92003,C1(NC(C(C2CCC2)OCC)=O)COCC1NC(=O)CN(c1ccccc1)C 92004,C1(NC(c2c(C)snc2)=O)CCCC(C(=O)N(C(C)C)Cc2ccncc2)CC1 92005,c1(CC)nn(C)c(OC)c1C(c1nnnn1C)NCCc1nnc(C)n1C 92006,N1(C(c2ccn(-c3ccccc3)n2)C(=O)NC(CC)C)CCCCC1C 92007,c1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)cccc2nccnc12 92008,c1(OC)ncccc1C(=O)Nc1cccc(CNC(=O)Cc2c[nH]nc2C)c1 92009,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COC)CCCC2)=O)C(COC)C1 92010,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92011,N1(C(C=CC=CC)=O)CCC(CC(=O)NC(CN2CCCC2)CC)C1 92012,N1(C(C(CC)CO)=O)CC2CCCC2(NC(c2cc(C)no2)=O)C1 92013,CCC(C)C(C(=O)NC(c1ccccc1)CC)NC(=O)C(C)OC 92014,c1(C(N(C2CCCN(C(C)=O)C2)CC)=O)ccc2[nH]ccc2c1.c12cnn(c1)C2 92015,C=CCCN=C(NCC(C)C(F)(F)F)NCc1ccc(C2CC2(F)F)cc1 92016,C1(C(N2CCCC(C(C)NC(=O)C3=CCCO3)C2)=O)CC2CCC(C1)N2C 92017,CCC(CCC(=O)N(C1CCC(C)CC1)C)NC(c1cc(C)c(CC)o1)=O 92018,c1(C(N2CCC(C(C)C(N3CCNC(=O)C3)=O)CC2)=O)cc(C#N)ccc1Cl 92019,C1(C(=O)NC(CCN(C(=O)Cc2cccnc2)C)(C)C)OCCOC12CCC2 92020,Cc1ncc(C(F)(F)F)cc1C(=O)NC1(C)CN(C(=O)CC2CCC2C2CC2)C1 92021,CCC(CC(=O)NC1CCC(CC(=O)Nc2conc2CC)CC1)SC 92022,c1(Nc2c(OC)ccc(OC)c2)cnc2c(Br)cc(Br)cc2c1 92023,N1(Cc2cn(CC)nc2C)CCOCC(C(N2CCOCC2c2ccc(Br)s2)=O)C1 92024,C(=O)(CCC(=O)NCCCNC(=O)C(C)CF)NC.C12CCN(C1)C2=O 92025,c1(-c2cn(CCC3CN(C(c4cc(Br)cs4)=O)C3)nn2)cc(F)cc2c1OCC2 92026,N1(CC(=O)NCC2CCC(NC(C=C(C)Cl)=O)CC2)CCCCC(O)C1=O 92027,N1(C(Cc2c(C)cnn2C)=O)CC(NC(c2cnc(C)nc2C)=O)CC(O)C1 92028,C1(CC(=O)NCCN(C(C)C)C(C23CC4CC2C3C4)=O)CCCN(C)C1 92029,CCC(C)(C)NCCN(C(CNC(C1CC1C)=O)=O)CC(C)NC(=O)N(C)C 92030,C1(CC)C(C(=O)NCC(C)(O)C2CCC2)CCCN1C(C1CCC(C)(C)OC1)=O 92031,n1(C(C)C(N2CCCC2C(C2CC2)NC(=O)CN(C)C)=O)ccc2ccccc12 92032,Cn1cnc2c1CCC(C(=O)NC1CCCN(C(=O)COc3ccsc3)C1)C2 92033,N1(C(C=CS(C)=O)=O)C2CCC1CC(NC(c1cc(Cl)cc(Cl)c1)=O)C2 92034,C1(CNC(C(C)N(C)C2CC2)=O)C2CCC(C2)N1C(C1CC(=O)N(C2CC2)C1)=O 92035,C1(C(=O)NC2(C(N3CCCC3)=O)C(OC)C2)C(C)(C)C1(C)C.C12(O)CN(C1)C2=O 92036,N1(C(C(C)OCCCC)=O)CC2C(CNC(C3(CCOC)CC3)=O)C2C1 92037,C1(C(N2CCN(C(c3coc(Cl)n3)=O)CC2CC(F)F)=O)CCCN2CCCC12 92038,Cc1ccccc1C(C)CC(=O)N1CC(O)(C(C)NC(c2nncn2C)=O)C1 92039,C1(NC2CCC(CN3CC(C(C(N)=O)=O)OCC3)CC2)SC2C=CC1CC2 92040,CC1CC(CNC(=O)CCC2CC2C)CN(C(=O)C=Cc2ncc[nH]2)C1 92041,CC(CF)CC(=O)N1CCC(C(C)CNC(c2ccn(C3CCC3)n2)=O)CC1 92042,c1(Nc2c(C(N(C3CCCN(C(C)(C)C)C3=O)C)=O)nccc2)nccc(C#N)n1 92043,CC(CCCCN=c1c(C#N)c[nH]c2ccccc12)NC(C1CC1C)=O 92044,C1(N(CC(F)F)C(=O)C2CC2)CCN(CC2CCCN(c3ncccn3)C2)CC1 92045,C1(C(=O)NCc2c(C(N(C)CC3CCN(C)C3)=O)scc2)CCC(=O)NC1 92046,Cc1nc(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)[nH]c1C 92047,C(C(C)(CC(C)C)NC(C1CCOC1(C)C)=O)NC(c1nc(CCC)oc1)=O 92048,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92049,C(C)(C)(CC(=O)N1CCC(c2ccon2)C1)N(C(=O)C(C1CCCCC1)O)C 92050,S(=O)(=O)(c1c[nH]ccc1=NCCc1ccc(Br)c(F)c1)NCCC(C)(C)OC 92051,N1(C(C2C(C)CC=CC2)=O)CCN(C(=O)CCn2ccccc2=O)CC1CCO 92052,n1(CC(C)C)ccc(=NC(=O)C2CCCN(C(C3CCCC(O)C3)=O)C2)[nH]1 92053,N1(C(CCN(C(c2c(CC)cco2)=O)C)=O)Cc2n[nH]cc2C1CO 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92071,N1(C(CCN(CC)CC)=O)CC2(CCCC2)C1C(=O)NC1CCCC(C)C1 92072,CC(CC(F)(F)F)C(=O)N1CCN(C(C23C4C5C2C2C3C4C52C(N)=O)=O)CC1C 92073,C1(NC(c2cc(C)sn2)=O)CC(NC(c2ccsc2C)=O)C12CCC2 92074,CC1(C)CN(C(=O)Cc2cc(Br)ccc2F)CCC1Nc1cnc(Cl)c(I)c1 92075,c1(-c2cn(C(C)C(=O)NC(CO)C(C)(C)CO)nn2)cc(Br)ccc1Cl 92076,C(=O)(C(C1CCC1)C1CCC1)N(C)CC1CCN1c1nncs1 92077,C1(C(=O)NC2C(SC)CCC2)CCC(O)CN1C(=O)Cc1nonc1C 92078,C1(CNC(CC2(NC(C3CC3C3CCC3)=O)CCC2)=O)CNC(=O)CO1 92079,CC1CCCC(=CC(NC[Si](C)(C)C)=O)C1.C(CC=O)NCCO 92080,N1(C(c2ccn(C)n2)=O)CC2COCC(C1)C2NC(C1CCC2(CCOCC2)O1)=O 92081,N1(Cc2ccc(C)o2)CC2(CN(C(=O)CN3CCC(N(C)C)CC3)C2)C1.[SH](C)=CF.C(O)CC.C.CCC 92082,C12(C(=O)NC(CC#C)C)CC1CCN2C(=O)CC1(O)CCC1 92083,C(=O)(CCC(CC)CCC)NC1(C(N2CCN(C(C#C)C)CC2)=O)CCN(C)C1 92084,C1(C)(C(N(CC=C)CCC)=O)CCN(C(C2CCC2COC)=O)C1 92085,c1(CNC(c2ncc(Cl)c(Cl)c2F)C(=O)OCCCCCC)c(C)cc(C)cc1C 92086,C(c1ccccc1F)=CCC(N1C(CN(C(C(CCOC)C)=O)C)CCCC1)=O 92087,CN1CCC(CC(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)C1=O 92088,N1(CCOC)CC(C(N2CCC(NC(=O)CCSCC(C)C)C2)=O)CCC1=O 92089,CC1OCCOC1C(=O)NCc1ccsc1C(=O)NCC1CC(O)(C2CC2)C1 92090,C1(C(=O)NCCC(CNC(C(C)Oc2ccccc2)=O)O)CCCC(=O)N1 92091,C1(CCCC)CCN(C(N2C(C)(CC(=O)NC)CC2)=O)CC1.C(C)(C)(C)O 92092,c1(C(N2CC(CNC(c3c(CC)scn3)=O)C2)=O)cnc2ncnn2c1C 92093,C1(C(=O)NC2CCN(C(=O)OC)C2)CN(C(c2ncoc2C)=O)CCO1 92094,N1(CCC=C)CCCC(c2nc(-c3ccc(CC)nc3)nn2CC)C1 92095,CC(C)(C#N)CCC(=O)NC1CN(C(c2cc(F)c(F)c(F)c2)=O)CC12CC2 92096,C1(O)(CNC(=O)C(F)c2cnoc2)CCN(C(c2cc(F)cc(F)c2)=O)CC1 92097,N1(C(CC(=O)OCC)=O)CCCN(C(=O)CNC(=O)CC2CCCC2)C(CO)C1 92098,c1(NC(c2cccc(NC(C3(F)CCCNC3)=O)c2)=O)cc2cnccc2[nH]1 92099,C1(C2(N(C(C3CCCS3)=O)CC)CC2)CCCCN1C(=O)CCNC(C)=O 92100,Cc1ccc(Cl)c([N+](=O)[O-])c1C(=O)NC(C)CCNC(C1C(C)C1C)=O 92101,N1(C(c2cccc(CC)n2)=O)CCC(C2(NC(=O)C(C)CC3CC3)CC2)C1 92102,c1(-c2cn(CC(=O)N(CC(C)C)C)nn2)cncc(-c2cn(C)nn2)c1 92103,CC1CC(NC(=O)NCCCCc2nccn2C)CC(C)S1(=O)=O 92104,C=Cc1ccc(C(=O)NC23C(CN(CCC(=O)NC4CC4)C)CC(CC2)C3)cc1 92105,C1(C(=O)NCC(CC)NC(=O)C=CCN2CCCC2)(CF)CC1(F)F 92106,CCCCCS(=O)(=O)NCc1cncc(-c2nn[nH]n2)c1 92107,N1(C(c2c(C)c[nH]n2)=O)CCN(C2CCCN(c3nnco3)C2)CC1 92108,Cc1cc(C(=O)NCCC(C)NC(C2COCCN2CC2CCC2)=O)ncc1F 92109,C1(C(N(CCC(=O)NC2C3(C)C(C2)CN3)CCCO)=O)CCC(=O)NC1 92110,c1(OC(C(N2CCN(C(C3(CC)CCCC3)=O)CC2C)=O)C)ccc(F)c(F)c1 92111,C(=O)(C#CC1CCC1)NC1C=CC(CC(=O)NCC(=O)N(C)C2CC2)C1 92112,C1(NCC2(CNC(COC)=O)CCC2)CCC(C(N)=O)C1 92113,N1(C(c2cc(CC)on2)=O)CCC(O)C1C(=O)NC(c1cnn[nH]1)C 92114,c12ccc(nc1C)NC(C(=O)O)C2.C1(C(C)OC)CCOCC1 92115,c1(C(=O)NCC2N(C(CCCCC(N)=O)=O)CCOC2)ccc2ncccc2n1 92116,Nc1ccc2ccccc2c1S(=O)(=O)NC1CC2CC2CC1C 92117,c1(OC)cc(C)cc(-c2nc(C)c(NCc3cc(F)cc(C#N)c3)s2)c1O 92118,c1(Cc2ccccc2S(=O)(=O)C(F)F)n[nH]c2c1CCCCC2.Cc1nc2n(C)c1[nH]2 92119,N1(C(CN(C(C=C)=O)CC)=O)CCN(CCN2CCC(OC)CC2)C(=O)C1 92120,CC1CN(C(=O)CSc2nncs2)CC(C)C1NC(c1cccc(=O)o1)=O 92121,c1(C(C)NC(=O)NCc2cc[nH]c2C2CC2)cc(C(C)(C)C)ccn1 92122,C(=O)(CC(C)CC(=O)N1CCC1CC(C)(C)COC)OC.C12(CCCO1)C(=O)NC2 92123,C1(CNC(C(C)(Cl)Cl)=O)C(C2CC2)CCN1C(=O)Cc1ccc(C2CC2)cc1 92124,N1(C(C(C)C)=O)CCOC(CNC(C2CCOC(=O)N2)=O)C1 92125,CCCC(O)C(=O)N1CCOCC1CCNC(=O)CCC1CCOC1 92126,c1(OCC)cc(=NC(=O)c2ccn(-c3ccccc3)n2)[nH]o1 92127,Cc1cc(C(=O)NC2CN(CC(=O)NC3COCC3N(C)C)C2)cs1.C1(=O)CN1 92128,C(=O)(CCC(C)NCC1C(C=C)C1)NC1(c2ccccc2)CC(C(C)(C)C)C1 92129,N1(C(C=NOC)=O)CC2(NC(=O)COCC3CCCCO3)CCCC2(F)C1 92130,C(=O)(C(C)(C)n1cc(Cl)cn1)C(CC(CN)O)(C)C.C1(CC(=O)N(C)C2CC2)(CC)CC1 92131,C(CN=C(NC1CCS(=O)(=O)C1)N1CCN(C)C(=O)C1)(C1CCOCC1)OC 92132,c1(OC)ccc(C(N2CC(c3cc(NC(C)=O)ccc3O)C2)=O)cc1Cl 92133,C1(OC)CC(NC(c2ccccc2C2CCOC2)=O)CN(C(C2(Br)CC2)=O)C1 92134,CCCC1CCCNC(=O)c2cc(n[nH]2)N1.c1(C(=O)OC)cccc(Cl)c1 92135,CCCC(C(O)C(=O)NC(c1nnc(O)n1C)C)NC(c1cc(C)co1)=O 92136,O(NC(=O)CC(C)C(C)(C)C)C(CC(C)C)C(=O)NCCC(C)O 92137,C(N=c1cc(C(F)(F)F)nc[nH]1)C1CC(NC(c2ccc(Cl)nn2)=O)C12CCC2 92138,c1(CC(N2C(CNC(=O)C3=CCC3)COCC2)=O)cn2ccsc2n1 92139,C=Cn1nncc1C(N1CCCC1(C)CNC(C1CC1c1ccccn1)=O)=O 92140,c1(OC)ccc(N2CCN(Cc3ccc(-c4ccsc4)nc3)CC2)c(F)c1 92141,N1(C(CNC(c2cc(C)no2)=O)=O)CC2CCCCC2(NC(=O)CCCCO)C1 92142,N1(C(CN(C(C)=O)C)=O)CCCC(CNC(=O)C(CO)NC(N)=O)C1 92143,Cc1sc(C(F)(F)F)nc1C(=O)NC1CN(C(C2CCCOC2)=O)CC1C 92144,c1(C(N(C)CC2(NC(C3CCC4(CC4)C3)=O)CC2)=O)c[nH]c(=N)cc1Br 92145,C1(CNC(C2CN(CC)C(=O)C2)=O)CC2CN(C(=O)C(F)(F)C3CC3)CC12 92146,N1(CC(=O)Nc2c(C)ccc(S(=O)(=O)NC)c2)CCCc2c1ccc(C)c2Br 92147,C1(NC(C2CCCN(CCC)C2)=O)CCCCN(C(c2ccco2)=O)CC1 92148,C1(NC(C(CC=C)c2ccccc2)=O)CCCN(C(C2(C)CC=CCC2)=O)C1C 92149,Cc1ccc(CC(=O)NCC2(CCNC(c3ccc(C)nn3)=O)CC2)c(Cl)n1 92150,CC1(C(N2CCOC(CCNC(=O)CN3CC=CC3)C2)=O)CNC(=O)C1 92151,C(=O)(CN=c1cc[nH]cc1)NCC12N(C(C=CSC)=O)CCC1CCC2 92152,CC1CN(C(c2n[nH]c(C3CC3)c2Cl)=O)CC1CCNC(c1n[nH]cc1Cl)=O 92153,CCC(CC)CCC(=O)N1CC(C)(NC(=O)CC2CCCC2O)C1 92154,CCCCCC(C)(C)C(=O)NCC1CC(C(N2CCC23CCN(C)C3)=O)C1 92155,c1(C(=O)NCC23C(CN(c4ccnc(N(C)C)n4)C2)C3)c(Cl)cccc1[N+](=O)[O-] 92156,CCC(CNC(=O)C(Cc1ccoc1)NC(c1cc(CO)on1)=O)CC 92157,C1(CNC(CC)=O)CCCCN1C(c1cn(C2CC2)nn1)=O 92158,c1(COC)ccc(O)cc1.c1(CNCC2N(C(C(C3CC3)=O)=O)CC2)nnnn1C 92159,C1(CC(=O)OCC)CC(NC(=O)CCc2nc(-c3ccco3)no2)C12CCC2 92160,CC(CC(=O)N1CC(CNC(=O)CCNC(=O)CO)C(F)(CO)C1)C(C)(C)C 92161,CCC(CC)(C(=O)N1CC2CC1CN(C(c1ncc(F)cc1F)=O)C2)C(=O)O 92162,CC(CCCC(=O)NC(C)(CO)C(C)(C)C)NC(c1nnc(S)n1C)=O 92163,c1(N(C)C)cc(C(=O)NC2CCC2CNC(=O)CCCc2ccsc2)ccc1Cl 92164,C1(NC(Cc2c(C)occ2)=O)CCN(C)C12CCCN(C(C1CC(=O)NC1=O)=O)C2 92165,c1(C(=O)NCC2(NC(c3c(C)nn(C)c3C)=O)CC(OC)C2)c(C)nc(C)nc1C 92166,C1(C(N(C2C3CN(C(c4ncc[nH]c4=O)=O)CC23)C)=O)CN=C2N=CNN2C1 92167,N1(C(Cc2cn(CC)nn2)=O)CCCC(CCNC(=O)C(=O)Nc2ncc[nH]2)C1 92168,c1(C(=O)NC2CCCCC2NC(=O)C(C2(O)CCCC2)F)cnc2[nH]cncc1-2 92169,C1(C#CO)(NC(C(C)Sc2ccccc2)=O)CCCCC1 92170,c1(C(=O)NC2(C(=O)NC(C(=O)OC)C3CCC3)CCCC2C)cncc(C=C)c1 92171,CC(C)C(CNC(=O)C(C)(C)C1(C)CC1(F)F)NC(=O)COC1CCC1 92172,c1(OC)cccc(NC(=O)C(c2ccc(Br)nc2)N(CCC#N)C2CC2)c1 92173,CC(CC(C)(C)C)C(=O)NC1CCN(C(=O)CC2NC(=O)NC2=O)C1 92174,C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(=O)COCC2CCCOC2)CC1(F)F 92175,Cc1nn(C)cc1CC(N1CCC(CNC(c2ccc(C(C)(C)OC)o2)=O)C1)=O 92176,N1(C(CCc2cc(C)[nH]n2)=O)CC2CCC(NC(=O)CSC(F)(F)F)CC2C1 92177,C1(N(CCN(C(C(C)CC2CCC2)=O)C(N)=O)CC=CC2CCC2)CCS(=O)(=O)C1 92178,C1(CNC(C2(CC(C)C)CCNC2=O)=O)COCCN(C(C2(F)CC2)=O)C1 92179,C1(NC(c2[nH]cc(CC(C)C)c2)=O)C(C)CCN(C(C2CCCC(C)C2)=O)C1C 92180,c1(C(C(=O)NCCN(CCOC)C(c2cccnc2)=O)(C)C)ccc(F)c(F)c1 92181,N1(C(CC2C(C)(C)OCC2)=O)CC2(CCC(NC(=O)CC3CCC4CC34)CC2)C1 92182,c1(C(C)CNC(C2CC3CCC2O3)c2nnnn2C)ccc(OC(F)F)cc1 92183,Cc1ncncc1C(N1CC(O)(C(C)(C)CNC(C2(C)CCN(C)C2)=O)C1)=O 92184,c1(CC(=O)OC)cccc(NC(C2CCC2C(=O)NCCCNC(N)=O)=O)c1 92185,Cc1cc(NC(=O)C(N)Cc2ccc(C(C)C)nc2)cc(C)c1 92186,Cc1nnc2n1CCCC2C(=O)N1CC(O)(CNC(=O)CCc2cncnc2)C1 92187,C1(NC(C=CCOC)=O)CC2CCC1(C(=O)NCC1=C(C)CCC1)C2 92188,N1(C(C2CC(O)(CC#C)C2)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 92189,C1(C(=O)NCCn2ccnc2)CCC(n2cc(-c3cnccn3)nn2)CC1 92190,N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(=O)CC1CCCOC1)C2 92191,C1(C(=O)NC2CC(C(N)=O)C2)(COC)CCCN(C(=O)C(=O)NC(C)C)C1 92192,N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(C2(NC(=O)C(F)C(C)C)CC2)C1 92193,c1(C(=O)NCC2(F)CCC(NC(C3(CC)CCOC3)=O)C2)nccc(OC)c1O 92194,CC(C)C(O)CCN=c1nc2c(cnn2C)c(NCc2cccnc2Cl)[nH]1 92195,C1(CC(=O)NCc2c(C(N(CC(C)O)C3CC3)=O)[nH]cc2)CCC2(CC1)CC2 92196,Nc1c(F)ccc(Cl)c1C(=O)NC1CN(C(C2CCCN(C(=O)C3CC3)C2)=O)C1 92197,C=CCCC(C1CC1)NC(=O)C(c1cccs1)NC(=O)CCc1nccn1C 92198,C1(N(C(=O)CCN(S(C)(=O)=O)C)C)CCCN(C(C2CCCC2O)=O)CC1 92199,N1(C(c2c(OC)cccn2)=O)CCc2cc(-c3cc(F)ncc3C)ccc2C1 92200,C#Cc1ccc(C2CC2C(N2CCC(F)(CNC(=O)C(C)CCC)C2)=O)cc1 92201,C(c1ccccc1)=CCC(=O)NCC1N(C(CN(C)C(C2CCO2)=O)=O)CCC1 92202,C1(CC(=O)NC(CC)C(F)(F)F)CCCCN(C(=O)Cc2csnc2C)C1 92203,C#CC1(C(N2CCCN(C)CC2)=O)CCN(C(=O)CC2CCCCO2)C1 92204,C(CCC(=O)NC1CC(O)C1)(c1n(C)nnn1)NCCC1CC1 92205,C1(NC(c2c(C)nccn2)=O)CC2(NC(c3ccc(CCF)cc3)=O)COC1C2 92206,CC(CC(=O)NCCCCC(C)(C)NC(c1ccnn1CC(F)F)=O)P(C)(C)=O 92207,CCCC(C(O)C(=O)NCC(C)(C)CC)NC(=O)CCS(N)(=O)=O 92208,N1(C(CCc2ccc(C)nc2)=O)CC(O)CC1(C)C(=O)NCC(C)CN(C)C 92209,C1(C)(C(N2CCN(CC(C)C)CC2)=O)CC12CCN(C(C1CCCN1C)=O)CC2 92210,N1(C(C(C)(CO)OC)=O)CC(NC(c2cnc(CC3CC3)nc2O)=O)CC(O)C1 92211,O=S1(=O)CC2(CCN(CC3CC4(C3)CC(F)C4)C2)CC12CCCCCC2 92212,C(=O)(C1=NOC2COCC12)NCC(C(=O)N(CC)Cc1cn(C)nn1)(F)C(C)C 92213,C1(C2(O)CN(C(C3CC(=C4CCC4)C3)=O)C2)(COC2CN(C)C(=O)CC2)CC1 92214,CCC(C)C(C)(O)CNC(c1c[nH]nc1CNC(c1ccnc(O)c1)=O)=O 92215,c1(C(=O)NCC(CNC(C(C(C)C)SC)=O)C)cc(Br)ccc1N 92216,C1(CC(N2CCc3sccc3C2C)C(=O)NC)Cc2ccccc2CN1 92217,N1(C(CC2C(C)(C)C2)=O)CCN2CCN(C(=O)C(F)C(F)(F)F)CC2C1 92218,c1(CC)cncc(C(=O)NC2CCN(C(=O)CN(C)C3CC3)C2C)c1 92219,CC(CCNC(c1ccc(F)c(F)c1)=O)N1C(=O)Cn2cccc2C12CCOCC2 92220,c1(C(N2C(C)(C(=O)NCCc3cc(C)cc(F)c3)CC2)=O)cnn2c1OCCC2 92221,c1(NC(CC)CSC)ccc(S(=O)(=O)NCC2CCN(C)CC2)cn1 92222,Cc1cc(NC(=O)CC(C(C)C)c2ccc(Cl)cc2)ccc1OC(F)F 92223,Cc1c(C(=O)NCC2CN(C(C3NC(=O)CC3C)=O)CCO2)cnn1C 92224,C12(NC(c3c(C)cc(C)[nH]3)=O)CCN(C(=O)Cc3cncnc3O)CC1C2 92225,C(CCCC(C)C)N(C(c1ccccc1)C(=O)N(c1ccn(C)n1)CC)C 92226,c1(CS(=O)(=O)NC)ccc(OCC(NOCC)=O)cc1 92227,C1(C(N2CCC(=CBr)CC2)=O)CCCOC12CCOCC2 92228,Cc1ncncc1NC(=O)NCC1CN(C(C2CC23CCCC3)=O)CC1O 92229,C(=O)(CC(C)(C)C(=O)NCC(O)CNC(c1c(C(F)(F)F)cccc1F)=O)OC 92230,C1(CNC(c2c(CC)cccn2)=O)CCN(C(c2nc(Cl)ccc2F)=O)CC1C 92231,c1(C(=O)CC2CCCN2C(C2(C(F)(F)F)CC2)=O)cc2c(C3CC3)cccc2[nH]1 92232,C(=O)(C1CCCc2c(O)cccc21)N1CC(C)(C)C(CNC(c2ccsc2)=O)C1 92233,C1(C(=O)NCC(C)(C2CC2)NC(C2(C(F)F)CCCO2)=O)CC12CC(O)C2 92234,c1(NCC)scnc1C(N1CCC(C(C)C(=O)NCC(CC2CC2)OC)C1)=O 92235,CC(C(=O)N(C)CC1CN(C(c2cn(C)nc2Br)=O)CCO1)C(F)F 92236,N1(C(C2(F)CCCN(C(=O)Cc3ccoc3)C2)=O)CCC([N+](=O)[O-])CC1 92237,c1(N(CC)CC)nc2cc(Br)ccc2cc1NC(C)=O.CC(CC1CCCCC1)CO 92238,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92239,N1(CCOC)CCCC(NC(=O)CC2CCN2C(=O)Cn2cnc(C#N)n2)C1 92240,c1(C(=O)NCC2C(NC(c3cc(CCC)on3)=O)CC2)c(Cl)cc(C)cc1Cl 92241,N1(Cc2ccc(C#C)s2)CCC2CN(C(c3cc4c(Cl)nccc4o3)=O)CC2C1 92242,CN=c1nc(N2CCCC(C)(F)C2)[nH]c(=NCCS(=O)(=O)C(C)C)[nH]1 92243,c1(OC)ccc(Br)c(C(=O)NCC2CCN(C(C3CNC(=O)C3)=O)CC2)c1 92244,c1(OCC)nnc(C2CCCN2S(=O)(=O)Cc2noc(C)n2)nc1C(=O)OC 92245,C1(N(C(=O)C(=O)NC2CCCCC2)C)CCCCC1CNC(=O)C(CCO)N(C)C 92246,C(=O)(C(=O)CC(C)C)N1CC(C(C(=O)NC(CCC)c2ccco2)O)C1 92247,CCC(C)C(C(=O)N1CC=CC1(C)C(=O)NCCc1cn[nH]c1)OC 92248,C(=O)(CCCCCCNC(=O)Cc1csc2nc(C)cn12)N1CC(C(=O)NC)C1 92249,c1(C(=O)NCCN(C(=O)Cc2csc(Cl)c2)C2CC2)ccc(-c2cc[nH]n2)s1 92250,N1(C(=O)CCOc2cc(F)ccc2F)CCC2(CCN(c3cnc(F)cn3)C2)C1 92251,c1(C(N(C)CC2CN(C(CC3C(C)CCO3)=O)C2)=O)cccc(=O)n1O 92252,N1(C(c2cc(Br)n[nH]2)=O)CCC(C2CCN(C(c3cncc(Cl)c3)=O)CC2)CC1 92253,N1(C(C2(c3c(C)cccc3)CC2)=O)CCC2CCC12CNC(=O)CCCNC(N)=O 92254,C1(NC(=O)C=Cc2ccc[nH]2)COC2(CNC(C3CCS(=O)(=O)CC3)=O)CC1C2 92255,C1(C)(NC(c2scc(OC)c2)=O)CCN(CC(=O)NCC(C)C)C1 92256,c1(C(=O)NC2(CNC(c3csc(Cl)n3)=O)CCOC2)cccc(F)c1O 92257,C1(C(=O)NCC=CCNC(c2cnc(O)s2)=O)(C(F)F)CC(F)(F)C1 92258,Cn1cccc1C(=O)NCCCCCNC(=O)CC1(C)CC1(F)Cl 92259,C(=O)(C(C)(C)C(C)C)NCC(C1CCC1)CNC(CC(=O)NCC)=O 92260,CC1(C)C(C(c2nnnn2C2CCCC2)NCCn2ccnn2)C1(C)C 92261,CCN=C(NCC1(C2CC2)CCCO1)NC(c1ccc(Br)cc1)C 92262,c1(C(=O)NCCCC(C)NC(=O)C(C)OC2COC2)ccc(C(F)F)c(F)c1 92263,C1(C2CC2)(C(N2C(CC(N)=O)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92264,c1(C(N2CC(CNC(C3(F)C(C)OCC3)=O)(CO)C2)=O)scc2c1CCCC2 92265,O=S(=O)(c1c[nH]ccc1=NC1CCC12CCC2)NCCCC1CCCO1 92266,c1(C(=O)NC(C)CC2(O)CCC2)[nH]ccc1CNC(C1COC(=O)N1)=O 92267,C1(NC(Cn2cc(C(C)O)nn2)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92268,c1(C(=O)NC2C(NC(c3nn(C)c(Br)c3)=O)C2)ccn2ccsc12 92269,C12(C(=O)NCC(CC3CN(C(C4C(C)C4)=O)C3)(C)C)CCCN1S(=O)(=O)CC2 92270,c1(CC)nc2c(C)csc2c(=NCc2ccc3ncsc3c2)[nH]1 92271,C(CNC(C1(C)CC1(C)C)=O)(CC(F)(F)F)NC(CC(=O)NCC)=O 92272,N1(CCCN(c2ccccc2)C)CC2CN(C(=O)Cc3ccccn3)CC2C1 92273,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92274,C1(NC(c2n(C)ncc2)=O)CCN(Cc2c(F)cccc2Cl)CC1F 92275,c1(NC(N2C(C)(C(=O)OCC)CCC2)=O)cc2occc2n1C 92276,N1(C(=O)Cc2csnn2)CCCC(c2cn(Cc3ccccc3)nn2)C1 92277,C=C1CC2CCCC(C1)N2C(=O)C(CNC(=O)CCc1cscn1)CC(C)C 92278,C12(CNC(=O)CC3CCCCC3)CCC1CN(C(c1occc1F)=O)C2 92279,c1(NC2CCN(C(C3CCCC(C)O3)=O)C(C)C2)ncnc2c1ncn2C1CC1 92280,N1(C(C(=O)NCC)=O)C2CCC1CC(C(=O)NCCC13CCCN1CCC3)C2 92281,Cc1[nH]nc(C(N2CCCC(CCCCNC(c3ccnc(O)c3)=O)C2)=O)c1Cl 92282,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92283,CC1=CCSC1C(=O)N(C1CCN(C(c2cnc(Cl)[nH]2)=O)C1)C 92284,CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCCCc3nccs3)C2)=O)C1 92285,c12nc(cs1)C(=O)N(CCNc1cc(Cl)c[nH]1)C2.C1(C(COCC)C)CCCC1 92286,N1(C(C(C)N2CCCC2)=O)CC2C=CC1C(C(=O)NCCc1cn(C)cn1)C2 92287,O=C(C1=CCCOCC1)NC(CO)C(=O)NCCc1cnn[nH]1 92288,N1(C(C(C2CC2)OC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92289,C1(=O)CC(C)CCN1.C(=O)(C(C)(C)CC1CCOC1)Cc1ncc(C)o1 92290,N1(C(C2(Cl)C(OC(C)=O)C2)=O)C2CCC1CC(CSc1ccc3c(c1)CCC3)C2 92291,C1(C)(NC(c2cccc(OC)c2)=O)CCN(CC2CCC(F)(F)CO2)CC1 92292,N1(C(CCCCCC#C)=O)CC2CCCC(NC(=O)CC3CCN(C)C3=O)C2C1 92293,c1(CCNC(=O)C(=O)NCc2cc3c(s2)CCC3)cccc(F)c1Cl 92294,c1(-c2cn(CCNC(COCc3cc(C)no3)=O)nn2)ccccc1S(C)=O 92295,c1(C(C(F)(F)F)OC(C(c2n(C)cnc2)O)=O)cccc(C(F)(F)F)c1 92296,c1(OC)c(NC2C3CN(C(c4ccc(Cl)cc4)=O)CC23)ncnc1Cl 92297,c1(N(C2CN(C(c3cc[nH]c3C3CC3)=O)C2)C)cc(O)nc(O)n1 92298,c1(COCC(=O)NCC(CCCC)NC(=O)C(CC)CCC)ccc2c(c1)CCC2 92299,c1(OC)ncc(C(F)(F)F)cc1NC(C1CC1NC(c1ccc(Br)cc1Cl)=O)=O 92300,C(=O)(CCC(C)C#N)N1CCN(CCNC(c2c(SC)nn(C)c2)=O)CC1 92301,C1(C)(C(N(CC(CNC(C2CC(CC)(CC)C2)=O)C)C)=O)CCC(C)C1 92302,C(=O)(CCC(C)(C)NC(=O)C(C)CC#N)N(C1(C(=O)NC)CCC1)C 92303,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C(C)C)=O 92304,C(C(C)C(F)C(=O)N(CCC1=CCCCC1)C)NC(c1c(C)ncnc1)=O 92305,CC(C)C(C(=O)NCCC1CCN(c2ccc(F)cc2)CC1)Sc1ccncc1 92306,Cc1cc(C)c(C(N2CCCCCC2CNC(c2nccnc2N)=O)=O)cc1N 92307,c1(C2(C(c3nnnn3C)NCC3C(OC)COCC3)CC2)cc(Cl)cc([N+](=O)[O-])c1 92308,c1(CNC(c2ccc(C)cc2)c2n(CCSC)nnn2)cc(C)cc(C)c1 92309,c1(OC)cc(N)c(F)cc1C(=O)NCC=CCNC(C1CCC2(CCC2)CC1)=O 92310,C(=O)(C(C)(C(C)C)OC)N1CCC(CC)C1C(=O)Cc1cn(CCCO)nn1 92311,c1(OCC)cc(N)ccc1OC.C1(C(=O)OC(C)(C)C)CCCC(C(=O)NC(C)=O)O1 92312,C1(NC(C(CC)CO)=O)CC2(CCN(C(C3C=C3C)=O)C2)C1 92313,C1(CNC(C=CC)=O)CCN(C(C2CC2(C)C(F)(F)F)=O)C12CC2 92314,c1(C(=O)NCC2(O)CCN(C(Cc3nc(C)[nH]n3)=O)C2)cccc2cnccc12 92315,C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)CN(C)C(c1cc2n(n1)CCCC2O)=O 92316,c1(N2CCCC(N(C(C(c3cnn(C)c3)C)=O)C)C2)ccnc2cc(Br)ccc12 92317,Cn1nc(-c2cccs2)cc1NC(C1(F)CCN(C(C2CC(O)CN2)=O)C1)=O 92318,CC1CN(C(C2(CO)CCOCC2)=O)CC(C)N(C(=O)CCc2cc(Cl)no2)C1 92319,c1(CC(=O)NCC2(COC)CCCN2c2cc(O)ncn2)cccc(F)c1F 92320,C=CCCCCC(=O)NC1(CCNC(c2cc(CC(C)(C)O)oc2C)=O)CCC1 92321,c1(OC)ccccc1SCC(=O)NCCC(C)(C)NC(C1C(Cl)(Cl)C12CC2)=O 92322,N1(C(C(CC)F)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1c1cnn(C)c1 92323,c1(CC(N2C(CNC(C3CC(O)C3)=O)CCC(C)C2)=O)nnc2n1CCCC2 92324,Cc1cc(CNC(=O)C(C)N2CCCC2)oc1C(=O)NC1CCCCC1 92325,C1(CC)N(C(C2(C(C)C)CCN(C(c3cccnc3O)=O)C2)=O)CC1(C)C 92326,N1(CCS(C)(=O)=O)CCCN(C(C2C3CN(CC(=O)NC)CC23)=O)CC1 92327,C(=O)(C(CCCCC(C)C)NC(C1CC1CO)=O)NC(=O)OCC=C.C1CC1 92328,C1(CC(=O)OC)CC(C(N2CC(c3ccccc3)C2(C)C)=O)CCO1 92329,C1(CC(N2CCC(OCCC)C2c2cccc(Br)c2)=O)CC2(CCC2)CO1 92330,c1(C(C)C)cccc(C(=O)NC2CC2)c1.C1(C)CCCNC(=O)C(=O)N1 92331,N1(C(c2n(C)ncc2)=O)CCC(C2(NC(c3coc(CO)c3)=O)CC2)CC1 92332,CC1=CCN(C(c2cc(CCNC(C3(N(C)C)CC3)=O)on2)=O)C1 92333,c1(C(=O)NCC2(C(=O)NC3(CC)CCCCC3)CCCCO2)n[nH]c2c1CCC2 92334,c1(C(=O)NCC(CC)(CC)NC(CN(C(=O)OCC)C)=O)csc2nnsc12 92335,Cc1cnc(F)c(CNC(=O)C(CCCF)NC(=O)C2=CCCCC2)c1 92336,N1(C(c2cc(CC)sn2)=O)CCCCC1C(C)NC(c1csc(C2CC2)n1)=O 92337,c1(N(C(C)=O)C)cnc(Cl)cc1C(=O)ON(C1CCCC(C)C1)C(C)(C)C 92338,C12=Nc3nc(C)c(o3)C(CCCO)C=CC1=CC=C2NCCOC 92339,C1(C(=O)NCC2C(NC(c3cc(C(F)F)[nH]n3)=O)C2)C2CC3CC(C2)CC1C3 92340,N1(C(C(C)OCC)=O)CCc2ccccc2C1CNC(=O)Cc1ccsc1Cl 92341,c1(C(N(C2CC(c3cccc(C#C)c3)C2)C(N(C)C)=O)=O)cc(N(C)C)c(Br)cn1 92342,c1(CNCCCC2CN(C(=O)N(C(C)(C)C)C3(C4CCCO4)CC3)C2)cccnc1 92343,Cc1cc(CC(N2CCC(NC(c3cc(-c4ccccc4)co3)=O)C2)=O)cs1 92344,N1(C(CC2(C(=O)SC)CC2)=O)CC(O)C(N)C1.c1(OC2(N(C)C)CC2)ccccc1 92345,N1(C(COc2cc(C)cc(C)c2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 92346,C=CCCCCC(=O)N1CCCOC(CNC(=O)CC(C)(C)C#N)C1 92347,c1(C(=O)NC2CCC(NC)C2)cnc2ccsc2c1 92348,C1(O)(CNC(C(CO)N(C)C)=O)CCN(C(c2nn(C)cc2C(F)(F)F)=O)C1 92349,C1(C(C)NC(CCN(CCCC(C)C)C)=O)CN(C(C2CCCCS2)=O)CCO1 92350,C(C(C)(CC(C)C)NC(c1ncccc1O)=O)NC(C(C)(C)OCC)=O 92351,c1(SC)cncc(C(=O)N(C)CCN(C(=O)C(C)n2ccnc2)CCOCCO)c1 92352,c1(C(=O)NC2CN(C3CN(C(C(CC)=CC)=O)C3)C(=O)C2)ccc(F)c(C)c1Cl 92353,c1(C(c2nnnn2C2CCOC2)NCC2(COC)CC2)cc(Br)c[nH]1 92354,CC1CCN(CC(=O)NCc2ccccc2)CC1NC(=O)CC1CC2CCC1O2 92355,c1(N2CCN(C(COC)=O)CC2)nc(N2CCC(C(F)(F)F)CC2)cc(C)n1 92356,Cc1ccc(C(N2CC(CC(F)C(=O)N3CC(O)(c4cc[nH]n4)C3)C2)=O)[nH]1 92357,C1(CC2CN(C(=O)NC3CCCC3C(F)(F)F)C2)CC(O)C12CCC2 92358,C1(C2CCN(C)CC2)(C(N(C(CC)CNC(=O)CCC2CC2(F)F)C)=O)CC1 92359,C(=O)(C1=C(Cl)CCCC1)NCC1C2CN(C(CCNC(=O)NC)=O)C1C2 92360,O=S(=O)(c1cccc(=NCc2ccoc2C2CC2)[nH]1)N1CCC(C2CC2)C1 92361,CC(C)CC(C)C(=O)N1CCOC(CNC(c2ccnc(Cl)c2O)=O)C1 92362,c1(C(=O)NC(CC=C)CNC(=O)CCc2cnc[nH]2)c(Cl)cccc1Cl 92363,C(=O)(C(C)(O)C(C)(C)C)NCC(CN(C(=O)CSc1ccccc1[N+](=O)[O-])C)O 92364,Cc1cc(C(=O)NC2CN(C(c3cncnc3C(C)C)=O)CC2O)c(C)s1 92365,C1(CCNC(c2cnc(OC)s2)=O)CSCCN1C(c1csc(C)n1)=O 92366,N1(C(C(=O)NCC)c2nccs2)CCC(C)(N(C)Cc2ccccc2)CC1 92367,N1(C(C2(CC)CCNC2=O)=O)CCC(CO)(CNC(=O)C(CC)NC(N)=O)CC1 92368,c1(C(N(C)CCN2CCN(C(C3C4CNC(=O)C34)=O)CC2)=O)cccc(F)c1O 92369,c1(C(N2C(C(=O)NC(C3CN(C)CCO3)C)CCC2)=O)cnn2c1CCC2 92370,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)CC1CCC2CC12 92371,c1(NC(=O)NCC(=O)NCC(CC2CC2)OC)ccn(CC)c1C 92372,C12CN(CCC1O)C2=O.c1(NC(CCc2nnc(N(C)C)o2)=O)ncncc1Br 92373,C12(C(N3CC(C(C)NC(=O)CCCN(C)C)C3)=O)CCCCC1C2 92374,Cc1c(C(=O)NC2CCC(C(C)NC(c3cccnc3O)=O)C2)nnn1C 92375,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 92376,N1(CCN2CCC(C)CC2)CC(NC(C2(c3ccccc3Cl)CCC2)=O)CCC1C 92377,N1(C(CC(C)OC)=O)CC2(CC2)CC1C(N1CCC(CC(=O)OC)C1)=O 92378,N#Cc1cncc(NC(C23CCC(NC(=O)C(=O)NCC(F)F)(CC2)C3)=O)c1 92379,c1(CNC(=O)Nc2ccc(Cl)cc2)ccc(-c2cc(C(N)=O)ccn2)cc1F 92380,C1(CNC(C(c2ccncc2)C)=O)CCC(C(=O)NCc2ccncc2)CC1 92381,c1(CNC(CN(CC)CC)=O)csc(C(=O)NC(CO)CCOC)c1 92382,C1(CC(C)(C)C)CN(C(c2ccsc2C#N)=O)CC1NC(=O)CC1(C#N)CC1 92383,C1(C(=O)NCC(C)(C)NC(c2nnc(C)s2)=O)CCCC(F)(F)CC1 92384,C(=O)(C(C)(F)C(F)(F)F)NCC(C)CN(C)C(c1cc(N)cc(O)n1)=O 92385,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 92386,C1(CC)CN(C(C23CCC(F)(CO2)C3)=O)CCN1C(c1ccc(NC=O)cc1)=O 92387,c1(OC)cc(O)c(C(=O)OCCC(O)CC(C)C)cc1I 92388,C1(CC)CCCN(C(C2COCC2(C)C)=O)C1C(=O)N(C1CC(CO)C1)C 92389,c1(N2CC(COC)(CNC(=O)C3=CCCCC3)C2)nc[nH]c2ncnc1-2 92390,c12ccc3c(ncnc3c1)NC(=O)C1CN(CCS1)C2=O.CN(C)CCO 92391,c1(C(=O)NCCCN(C(C(C)OC)=O)C)c2c(c[nH]c1=N)CCC2 92392,C1(NCCc2c(C)cncc2)Cc2ccc(Cl)cc2C1(C)C 92393,c1(C(N2CCC(C(F)F)(CNC(=O)C3=COCCC3)C2)=O)cncc2ccsc12 92394,C=CCC(C(=O)NCC(=O)NC(C)CC)NC(=O)Cc1cnn(C)c1 92395,C1(C(=O)NCCN(C(=O)OC)C)(NC(C2CC(F)C2)=O)CCOCC1 92396,C12(C(=O)NC(CC)CNC(=O)CNC(C3CCCC3)=O)CCCC1C2Br 92397,C1(C(=O)NCC(CO)NC(c2cnc(Cl)n2C)=O)(OCC)CCCCCC1 92398,C(CCCCC(=O)N1CCC(NC(c2cn(C)[nH]c2=N)=O)CC1C1CC1)N(C)C 92399,N1(C(C(C)C(C)O)=O)CCC2(CC1)CC(CNC(=O)Cn1cnnc1O)C2 92400,c1(C(N2CCN(C(CCC)=O)CC23CC3)=O)nccc2ncccc12 92401,c1(NC)c(C(=O)NC2CC2CNC(c2cc(C3CC3)no2)=O)sc2nccnc12 92402,C1(C(=O)NC(CNC(COc2cc(C)cc(F)c2)=O)C)CCCC(F)(F)CC1 92403,c1(C(N(CCN(C(CN2CC(C)C2)=O)C)C)=O)cc(=O)c(Br)c[nH]1 92404,C1(N(CCCc2c(C)cccc2)C(=O)NC(C)C)CS(=O)(=O)CC1O 92405,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 92406,CC12CCCCC1C(=O)N2.C(=O)(C(Cl)Cl)NCCNC(=O)C1CC1 92407,c1(CCC(=O)NCC(CC)N(C)C(C2CC2)=O)cccc(OCC)c1 92408,N#Cc1ccc(CC2CCN(C(=O)Sc3cccnc3C(F)F)C2)cc1 92409,Cn1ncc([N+](=O)[O-])c1C(=O)NCCCNC(C1(C(F)(F)F)CC1)=O 92410,N1(C(c2c(C)ccnc2)=O)CC2CCC1CC2NC(C1(O)CCSCC1)=O 92411,C1(C(C(c2nc(C)[nH]n2)O)C)CCN(C(=O)COC2CCCC2)CC1 92412,c1(SCC)ccc(C(N2CC(NC(c3nc(C4CC4)cs3)=O)C(CC)C2)=O)cc1 92413,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)C(C)c3ccsc3)C2)c(O)n1 92414,N1(C(Cc2ccc(C)o2)=O)Cc2occ(C(=O)NC(CCO)C(F)F)c2C1 92415,C1(C(=O)NCCCN(C(COC)=O)C)(C(=O)OC(C)(C)C)CC(CNCO)CO1 92416,C1(C(=O)NC(CCCC)CNC(=O)Cn2nccc2C)CNc2ccccc2O1 92417,CCCCC(CC(=O)NC(C)CCF)NC(C1CC2CCC1O2)=O 92418,C(=O)(C(C)(C)CCCNC(C1CCCN(C(C2CCOC2(C)C)=O)C1)=O)OC 92419,c1cc(-c2ccc3c(c2)OCO3)c2c(c1)C(c1nc(CC3CCOC3)n[nH]1)CC2 92420,c1(CC)cccc2c(CC(=O)NC3CC3CNC(=O)C3=CCOCC3)c[nH]c12 92421,CON1CCC(C(=O)NCC2CC3CN(C(C4CCCC4OC)=O)CC23)CC1 92422,C1(NC(c2cnc(OC)c(C)c2)=O)CCCCCN(C(C2CC3(CC3)CO2)=O)C1 92423,c1(C(=O)NC2CC(CNC(CC3(C=C)CCOCC3)=O)C2)ccc2cnoc2c1 92424,c1(C(=O)NCCCNC(C2(OC)CCCOC2)=O)cnc(C(F)(F)F)c(C)c1 92425,Cn1cnc2c1CN(C(=O)COC(C)(C)CNC(c1ccc(N)c(F)n1)=O)CC2 92426,c1(-c2scc(CC(=O)N(CCCCNC(CC=C)=O)C)n2)ccccc1OCC 92427,N1(Cc2ccn(CC)n2)CC2CC(CN(C(c3ccccc3C(C)(C)C)=O)C2)C1 92428,c1(C(C(F)F)NCCNC(=O)NC2CCCC3CC23)ccc(F)cc1F 92429,N1(C(C(C)OCC)=O)CCC2C(NC(c3ccc(C(N)=O)cn3)=O)C12 92430,c1(NC(c2cc(Nc3cc(N(C)C)ncn3)n(C)n2)=O)cccc(O)c1Cl 92431,C(c1cnn(C)c1)=CC(=O)NC(C1CN(C(CN(C)C(N)=O)=O)C1)C 92432,c1(C(=O)NCCC2CCN(C(C3CCC(=O)N3)=O)C2)cc2n(c1)CCC2 92433,CC(C)(C(=O)NCC1CCN1C(=O)Cc1cc(C(F)(F)F)co1)C1CC1 92434,c1(CN2CC(C(=O)Nc3cnccn3)C2)cccc(Oc2ncc(Br)cn2)c1 92435,c1(C(N2CCC3(C(=O)NCC(=O)OCC)C(C2)C3)=O)cccc2c(Br)ccnc12 92436,CC(CF)CC(=O)NC1(NC(=O)C(COC(C)(C)C)N(C)C)CCOCC1 92437,CCC(CC)C(=O)N1CCC(C)(CNC(=O)C(c2ccccc2F)OC)C1 92438,C(CC(C(C)(C)C)NC(C1CC(=O)CC(=O)N1)=O)N(C(C(C)=C(C)C)=O)C 92439,C(=O)(C#CC1CCOCC1)N1C(CNC(C=Cc2cn(C)nn2)=O)CC(F)(F)C1 92440,c1(C(=O)OC)ccc(S(=O)(=O)NC2CCC(O)C(C)CC2)c(Cl)c1 92441,C1(C(N(C(C)C2CC2)C)=O)CC12CCN(C(c1cn3cccnc3n1)=O)CC2 92442,C(N=c1[nH]c(C)cc(=NCC23CCCN2CCC3)[nH]1)C1CC(OC)C1(C)C 92443,CC1C(C(=O)Nc2cccc(-c3ccncc3)c2)CCCCC1C=O 92444,C12(C(=O)NC3C(C(C)(C)C)CN(C(=O)CC4=CCCC4)C3)CCCC(C)(C1)OC2 92445,N1(CCCO)CCCC(CCNC(c2cc(OC3CCOCC3)ccn2)=O)C1 92446,C(=O)(CCCC(=O)N(C)C)NCC(C1CCCC1)NC(c1[nH]c(CC)c(Cl)n1)=O 92447,CC1CCC(NC(C2CC(C)(C)C2C(F)(F)F)=O)CN1C(c1cc2c([nH]1)CCC2)=O 92448,C(=O)(C(CC(F)F)C1CCC1)NC(CNC(=O)COc1cccc(F)c1F)CO 92449,C1(NC(C2N(C(N)=O)CCC2)=O)C2CC1N(C(C1CC3CCCC13)=O)C2 92450,C12(C(N3CC(C#C)N(C(c4cncc(F)c4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 92451,N#Cc1ccc(C(O)C(=O)NCCc2cccc3sccc23)c(F)c1 92452,CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CN(C(C2(O)CCOC2)=O)C1 92453,N12CCC3(CC1)OCCCC3C2=O.Cc1[nH]nc2ccc(-c3nn[nH]n3)cc12 92454,C=CCCC(F)(F)C(=O)NC(C)CCC(=O)NCCOC(C)C 92455,c1(C(N2C3(CNC(C(C=C)(C)C)=O)CCCC(C2)C3)=O)ccc2oc(C)nc2c1 92456,C(=O)(CS(=O)(=O)CC(C)C)NCCC1(O)CCN(C(C(CC)(C)OC)=O)CC1 92457,S(=O)(=O)(c1cnc2nccn2c1)NCc1[nH]nc(C2OCC(C)C2)n1 92458,N1(C(c2cnc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc3ccccc23)CC1C 92459,Cc1noc(C)c1CC(=O)N(C1(F)CN(C(=O)CSCCC(C)C)C1)CC1CC1 92460,N1(C(c2n(C(C)C)cnc2)=O)C2COCC1CC(NC(=O)C(C)CC(N)=O)C2 92461,c1(C(=O)NCCCN(C(=O)COc2ccc(C(N)=O)cc2)C)csc(C#N)c1 92462,C1(NC(C=CC)=O)CS(=O)(=O)C2CN(C(c3nnn(C4CCOC4)c3C)=O)CC12 92463,C(=O)(C(C)NC(C1CN(C(=O)C(C)n2ccnc2)C1)C)NC(=O)OCC 92464,C(CN=c1[nH]cnc(Cl)c1CO)C1CCC(NC(C2CC(C(=O)O)C2)=O)C1 92465,N1(C(C(CC)c2cccnc2)=O)C2CCC1CN(C(=O)C#CC1CCCOC1)CC2 92466,CCCC(O)C(=O)NC(C(N1CCC(CN(C)C)C1)=O)C1(C)CC1 92467,N1(C(C(C=C)OC)=O)CCN(C(c2c(OCC)cccc2CC)=O)CC1CO 92468,c1(OC)ccc(CN2CCC(CC(N3CCCC3C(N)=O)=O)C2)c(Br)c1 92469,C1(CNC(c2n(CC)cnn2)=O)CCN(C(=O)CC23CCCC2C3)C1(C)C 92470,c1(CC(=O)NC2CN(C(=O)C(F)=CC3CC3)C3CC23)cc(F)cc(Br)c1 92471,CCC(O)C(C)(C)C(=O)N1CCC(c2n[nH]c(C[N+](C(=O)CCCN=[N+]=[N-])([O-])OC)n2)C1 92472,S(=O)(=O)(CC(=O)N1CCCC(C(=O)NCC2CCCCN2C(N)=O)C1)NC 92473,CC1(C(=O)NCC2(C(=O)Nc3ccsc3Cl)CCOCC2)CC=CCO1 92474,c1(CC(=O)NCC2CN(C(CN(C)C)=O)C2)csc(NC=O)n1 92475,Cc1ncc(Br)cc1NC(C1CN(C(=O)C(C)S)CCC1C(F)(F)F)=O 92476,c1(C(=O)NCCCNC(CN2CCN(CC(C)C)CC2)=O)cccc2nc[nH]c12 92477,Cc1cc(N)cc(C(=O)N(CCCNC(=O)C(c2ccccc2F)C)C)c1F 92478,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 92479,C(CN=c1[nH]c(=NCC23CCCC2OCC3)[nH]c2cccc(F)c12)N(S(C)(=O)=O)C 92480,c1(C(N2CC(CCNC(c3n(CC)ncn3)=O)C2)=O)cccc(OC(C)CC)c1 92481,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 92482,c1(C(c2n(C(CC)C)nnn2)NCC(C)OCCO)ccc(Cl)c(C)c1Cl 92483,N1(C(CCSC)=O)CC(CNC(=O)Cc2ccc(C)c(OC(C)C)c2)C(F)(F)C1 92484,C1(C(=O)NC(c2ccccc2F)CNC(C(C)(C)O)=O)CCC2(CCCCC2)CC1 92485,c1(OC)ccc(O)c(C(=O)NC2CC(CNC(C3CCO3)=O)C2)c1 92486,c1(C(=O)NC2C3CN(c4c(C)c(Cl)ncn4)CC32)c(C)cc(O)nc1C 92487,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)NC(N)=O)C2 92488,O(NC(=O)CC(C)N(C(=O)C(c1ccnn1C)O)C1CC1)CCOCC#C 92489,N1(C(c2c(CC)c(C)sc2)=O)CCCN(C(=O)CSc2ccncc2)C(C)C1 92490,C1(NC(c2csc(C)c2N)=O)CC2(C1)CC(NC(=O)CCNC(=O)C(C)(C)C)C2 92491,C=C(C)C(CC(=O)N1CCCC(C(=O)N(CC(C)OC)CC)C1)OCC1CC1 92492,c1(C(=O)NC(C(C)NC(=O)CCOc2ccc(F)cc2)C)c[nH]c2cccnc12 92493,CCC(CCOC)C(=O)N1CCOC(C)(CNC(=O)CCNC(=O)CCCOC)C1 92494,c1(NC(=O)NCc2cc(OC)ns2)nc(C)ccc1SC(C)(C)C 92495,Nc1nonc1C(=O)NN1CCCC1.N12CC(C1)CC=CC2=O.n1(CC)ccnn1 92496,N1(C(c2cc(C)cc(C)c2)=O)CCCC2(NC(c3ccnnc3C)=O)CC2C1 92497,CC1OCCN(C(=O)C(c2cnn(C)c2)C)C1C(N1CC2(CCC2O)C1)=O 92498,N1(C(CCSCCCC)=O)CC2CCCN(C(c3ncoc3C)=O)C2C1 92499,C1(NC(CC2C(C)OCC2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 92500,c1(NC)ccc(C(=O)N(CCC(=O)N2CCC2C2CCCOC2)C2CC2)cn1 92501,c1(C(=O)NC2CCC(NC(c3nn(C)c(F)c3)=O)C2)ccn2c(O)nnc2c1 92502,Cc1cccc2[nH]cc(C(N3CC(N(C)C(C4CCC(C5CC5)C4)=O)C3)=O)c12 92503,N1(C(C(CCC)NC(C)=O)=O)CCCC(F)(CNC(C2SCCCS2)=O)C1 92504,c1(C2C(CC(=O)NC3(CO)CN(C(C(CC)(F)F)=O)C3)C2)ccc(F)c(F)c1 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92662,CC(C)C(O)CC(=O)NCC1CC(O)CN1C(c1ccc(F)c(F)c1)=O 92663,C1(C(N(C2CCN(C(C3CN4CCC3CC4)=O)CC2)C)=O)CN(CP(C)(C)=O)C1 92664,c1(C(C)C)ccc(C(C)CC(=O)N(CCNS(C)(=O)=O)CC2CC2)cc1 92665,c1(OC)ncc(C=CC(=O)NC2CCCN(C(c3cncc(OC)c3)=O)C2)cn1 92666,Cc1cccc(C(CNC(C2C3CCCC23)=O)N(C)Cc2ccccc2)c1 92667,C(=O)(C(C)CN(C(=O)CCc1ccn(C)c1)C)NCC(=O)NC(C)C 92668,C1(Cn2cc(C(CC)O)nn2)(NC(=O)CC2CCC(C)C2)CCCCC1 92669,C1(CNC(=O)CCc2cn[nH]c2)(CNC(C2CC3CCCC23)=O)CC2(CC2)C1 92670,n1(CCC(=O)NC2CN(C(=O)CCCC(F)F)CCC2F)cnc([N+](=O)[O-])c1 92671,C1(C(=O)NCC2OCCN(C)C2)COC2(C1)CN(C(=O)CC(F)(F)Cl)C2 92672,C12(CNC(C(C=C=C)C)=O)CCC(CC1)CN2C(=O)C(C)=CC1CC1 92673,C1(C(=O)NC2CCCCCN(C(c3cc(C)[nH]n3)=O)C2)CCC(C2CCCO2)O1 92674,N1(C(C(C)OCCOCC)=O)CC(NC(C2CC2C(C)(C)C)=O)C(F)C1 92675,C1(OC)COC(CC)CN1C(=O)CC(COC)OC 92676,C1(C(=O)NC(=Cc2cn[nH]c2)CNC(CCC(C)(F)F)=O)CCS(=O)(=O)C12CCC2 92677,c1(CO)cc(NC2CC(CC(=O)NC(c3cc(C(=O)OC)[nH]n3)=O)C2)ccn1 92678,C1(CNC(=O)NCc2cccnc2Cl)CCCCN1Cc1c(CC)cccc1 92679,CN(C)C1CCCc2ccc(NC(c3nc(-c4ccc(F)cc4)no3)=O)cc21 92680,c1(CC(=O)NC2CCN(C(C3(SC(C)C)CC3)=O)C2)ccccc1C(F)(F)F 92681,C1(O)(CNC(C=CC(=O)N(C)C)=O)CN(C(c2ncoc2C2CCC2)=O)C1 92682,c1(-c2cn(C(C)CCO)nn2)ccc(Cl)cc1.C1CCC1 92683,C1(COC)CC12CCN(C(c1cc(C3CCNCC3)sc1I)=O)C2 92684,C(=O)(C(C(C)C)NC(C)=O)NCC1C(NC(=O)Cn2cc(C(=O)NC)nn2)C1 92685,C1(NC(C2(OC)CN(C(C(CC)F)=O)C2)=O)CC(=O)N(CC)C1 92686,C(=O)(C(C)(O)CCC)NCC(C)(C1CCC1)NC(c1c(CC)n(CC)nc1)=O 92687,Cc1nc(C)n(CCC(=O)N(CCCNC(c2nncn2C2CC2)=O)C2CC2)n1 92688,c1(C(N2CCN(C(CC3(C#N)CCC3)=O)CC2)=O)cnn2c1OCCC2 92689,C1(C(=O)NCC2(NC(C=CC3(C)COC3)=O)CCC2)CC2C(C1)C2(C)C 92690,c1(CN2CC(CC(=O)Nc3cc(CC)c(Cl)cc3)C2)cn2cccnc2n1 92691,N1(C(c2cccc(C(CC)=O)c2)=O)CCN(C)C(=O)C1 92692,c1(C(=O)NCC2C(NC(c3c(COC)cccc3)=O)CC2)cc2n(n1)CCC2 92693,Cc1ccc(C(C)NC(c2nc(-c3ccoc3)no2)=O)nc1 92694,c1(CCN(CCC(C)C)C(=O)CC2COCCOC2)ccc2c(c1)CC2 92695,N1(C(c2cnc(C)s2)=O)CC2CCC1C1CN(C(C3CCC34CCC4)=O)CC21 92696,c1(C(N(CCNC(CC(C)OC)=O)C2CC2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 92697,c1(CC(C)C(=O)NC23COC(CN2c2ccncn2)C3)c[nH]c2ccccc12 92698,c1(C(c2n(CCC)nnn2)NCc2ccc(CC)s2)ccccc1NC(C)=O 92699,CC1COCC(CNC(=O)CCCCN(C(=O)C(=C2CCCCC2)F)C)O1 92700,CCCC(C(O)C(=O)NCCC(=O)NCC(C)C)NC(c1c[nH]nc1C)=O 92701,N1(C(C(=O)N(CC(C)O)CCNC(c2cnsc2)=O)C)CCCCC1=O 92702,Cc1ccccc1OCCC(=O)NCC(C)(C1CCC1)NC(C12CCN(CC1)C2)=O 92703,c1(OC)c(C(=O)N(CC(C)NC(c2csc(C)c2C)=O)C)sc(Cl)c1Cl 92704,N1(C(CCCOC(C)C)=O)C(C(=O)NC2(C(N)=O)CCC2)CCC12CC2 92705,c1(NC(COC(c2cc(CC)ncc2)=O)=O)cc(C)cc(Br)c1C 92706,C1(CNC(=O)CC2CCC(=O)N2)CCN(C(=O)CC2(CO)CCC2)CC1 92707,CC1(C)CN(C(=O)CC(c2cccs2)NC(N)=O)CC1C(=O)NC1(C)CNC(=O)C1 92708,N1(C(N2CCC(OC)C2)=O)CCC2C1CCN2C(c1cccc(C2CC2)c1)=O 92709,c1(CN2CC3(N(C(c4ccc(C=C)cc4)=O)CC3)C2)ccc(C#N)cc1O 92710,N1(C(c2ccn(C)n2)=O)CC2CC1CN(C(=O)Cc1c[nH]c(=N)nc1O)C2 92711,c1(C(=O)NCC(C)CNC(=O)C(C)(O)c2ccccc2)cc2c[nH]nc2s1 92712,CCCCC(C(=O)NCC1CCC(C(=O)NCC(C)(C)CC)C1)C(C)C 92713,N1(C(C(C)NC(CC)=O)=O)CC2CCC1(CNC(C1CCCS(=O)(=O)C1)=O)CC2 92714,Cc1c(C(=O)NC(C)CCNC(=O)C(CCO)N(C)C)cnn1C(C)C 92715,c1(OC)ccc(NC(C2(CNC(=O)CC3CC4(CC4)C3)CCC2)=O)c(Br)n1 92716,N1(C(CC(COC)C)=O)CC2COCC(C1)C2NC(c1cncc(F)c1C)=O 92717,CCCCCCOC(C)C(=O)NCCC1(O)CN(C(C2CCN(C(C)C)C2)=O)C1 92718,c1(C(N2C(CNC(C(N(C)C)C3CC3)=O)CCC2)=O)ccc2nc(O)n(C)c2c1 92719,C1(NC(C=C(C)C)=O)CN(C(c2sc(-n3cccc3)nc2C)=O)CC1C 92720,Cc1cnccc1C=CC(=O)N(CCNC(c1c(O)cccc1F)=O)C(C)C 92721,C1(NC(c2c(C)ccs2)=O)CCC(C(=O)NCCCC(C)O)CC1 92722,C1(C(=O)NCC(CNC(C=Cc2c(C)ccs2)=O)C)CCc2nnc(O)cc2C1 92723,C=C1c2ccccc2C(=O)N1CC(=O)NC1CC(C)N(C(c2cc(OC)n[nH]2)=O)C1 92724,Cc1cc2[nH]c(C(N3CCN(C(C4CC5CCC(C4)O5)=O)C4CC34)=O)cc2o1 92725,C1(C)(C(=O)NC(CC)COC)CCCN1C(=O)CC1CCOC1=O 92726,C(CCC(=O)NOCCSC)N(C(C(C1CCCO1)SC)=O)C 92727,C1(O)(C(=O)NCCCN(C(c2c(CCC)n(C)nn2)=O)CC)CC2CCC1C2 92728,C(CC(C(C)C)NC(=O)C(C)(C)NC(=O)C(F)(F)F)NC(CCSC)=O 92729,C=CCC(CNC(=O)CCn1cc(C)cn1)NC(c1n[nH]cc1Br)=O 92730,CC(C)(C)S(=O)(=O)CC(=O)N1CCCC1CCNC(c1cc(O)nc(O)c1)=O 92731,C(=O)(C(O)CC(F)(F)F)Nc1cc(C(=O)O)ccc1C(=O)NC1N(CC)CCC1O 92732,N1(C(C(COC)COC)=O)CC(NC(c2cc(OC)nc(C)c2)=O)CCC1C 92733,C(=O)(C(C)S(N)(=O)=O)N1CCC(N(CC#C)C(C2OCCC2(C)C)=O)CC1 92734,c1(C(N2CCC(CNC(c3cncnc3C3CC3)=O)C2)=O)cc2nc[nH]c2cn1 92735,c1(CC(=O)NCCN(C(=O)CC(C)OC)CC)cccc(OC(C)C)c1F 92736,N1(C(C2CCC(NC)C2)=O)CCC=C(C(=O)NC(c2ccc(C)o2)(C)C)C1 92737,c1(N2CC(C(C)C)OCC2)nc(N(C)CC2(CN(C)C)CC2)nc2ccc(Cl)cc12 92738,C=CC1OCCC1NC(C1CCN(C(c2ns[nH]c2=O)=O)C1C(C)C)=O 92739,CCC(CC)CCCN(C(=O)C(C1CCCN(C(=O)C(C)OC(C)=O)C1)(C)C)C 92740,O=C1CC2C(C(=O)NC3CC(C(F)C(=O)NC4CCCC5(C4)N=N5)C3)C2C1 92741,CC(C)(C#N)CCC(=O)NC1CC(C)(NC(c2ccn3cccc3c2)=O)C1 92742,c1(-c2c(OC)cc(C(=O)Nc3c(Cl)n[nH]c3C)nc2)ccc2c(O)ncccc1-2 92743,C1(F)(CNC(C(C)OCC=C)=O)CCC(CNC(=O)C(C)SC)CC1 92744,c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)Cc3csc(C(C)(C)C)n3)C2)no1 92745,c12cccc(c1)NCCCC(=O)N1CCC(CC1)N(CC)C2=O.C(N)(=O)NC 92746,C(C1CCC(C)CC1)=C(C)C(N1CCN(C(C23CCC(C2)OC3)=O)CC1)=O 92747,O=C1CCC2(c3ccccc3)SCC(C3=CCC(F)(F)CC3)N12 92748,c1(CC(C(=O)NCC2N(C(CC3CC(=C)C3)=O)CC2)C)ccccc1F 92749,C1(NC(CN(C(C)C(=O)OC)CCC)=O)CCCN(CCCc2ccccc2)C1C 92750,C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(c2ccc(N(C)C)c(Cl)c2)=O)CCOC1 92751,C12(CC)CCC(NC(=O)CC(C)(C)OC)(CC1)CO2.C123CCC(CO1)(C2)C(=O)NC3 92752,c1(C(=O)NCCC2C(C)CN(C(=O)C3=CCS(=O)(=O)C3)C2)cc2ccnn2cn1 92753,C1(NC(COC)=O)CCCN(C(=O)C(=O)NCCOCC(F)F)C1C 92754,c1(C(c2n(CCCC)nnn2)NC(C)C(=O)NC)ccc(Br)c2cccnc12 92755,N1(C(C(CC)C)=O)CCOC(C#N)C1.c12csc(n1)C(=O)N2 92756,CC(C)CC(CN(C)C)N(C(=O)CS(N)(=O)=O)C(c1cnc(C2CC2)nc1)=O 92757,N1(C(C(CSC)(C)C)=O)CCC(F)(F)C(CNC(=O)CC2CC=CCC2)C1 92758,N1(C(CSCC)=O)CCCC12CCN(C(c1nccn3cnnc13)=O)CC2 92759,c1(N2CCC(S(N)(=O)=O)C2)ncc(S(=O)(=O)NCCc2c[nH]c(=N)s2)cc1Cl 92760,N1(C(CCC=CC)=O)CCC(C)(C)C1CNC(=O)CC1CCC1C1CC1 92761,c1(C(=O)NC2C(CC(=O)NCC3(CC)CCOC3)C(O)C2)cc(Cl)cn1C 92762,CN(C)NC(=O)CCC(=O)NC1(CCNC(c2csnc2C(F)F)=O)CC1 92763,c1(NC)ccc(CNCC23CC2CN(C(=O)OC(C)(C)C)C3)c(Br)c1 92764,c1(CC)[nH]ccc1C(=O)NCC=CCNC(=O)C(C)Cn1cccn1 92765,C1(CC)CN(C(=O)NCc2cc3cc(Cl)ccc3s2)CC2(CCOC2)O1 92766,c1(OCC)cccc(C(=O)NCC2CC(NC(=O)CCOCC(C)(C)C)C2)c1N 92767,N1(C(c2cc(C(C)C)[nH]n2)=O)CCC2(CCN(C(=O)CSC(C)C)CC2)C1 92768,C(=O)(CCCCC(=O)NCC(C)(C)CN(C)C(C1(C(N)=O)CCC1)=O)NC 92769,N1(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC2(CC1)CC2NC(=O)C(N)=O 92770,C1(C(N2CC(C)(C(=O)OCC)C2)=O)C(C)CCN1C(C1CC2CCC2C1)=O 92771,C1(C(N(CC(=O)OCC)C)=O)CN(C(=O)CCCn2cncn2)CCC1C 92772,CC(C(O)C(F)F)NC(=O)CCCC1(NC(c2ccc(CF)cc2)=O)CCC1 92773,C(=O)(C(c1nccs1)N(C)CCC1OCCO1)NCC 92774,C1(C2CN(Cc3ccoc3)C2)(NC(c2c(CC)n(CC(C)C)nc2)=O)CC1 92775,c1(NC(=O)OCC)nccc(NCC23CC(c4ccccc4)C(C2)C3)n1 92776,C1(C(=O)NC(C(=O)N(C)CC2CCCC2O)CC2CCCC2)CCCNC1=O 92777,C1(C)(C(C)C)CC(N=c2cc(Cl)nc(C(C)(C)C)[nH]2)CN1C(c1cccs1)=O 92778,CS(=O)(=O)c1nccc(NCC23CCC(NC(=O)CCNC(=O)CO)(CC2)CO3)n1 92779,c1(OC)cccc(CC(C)C(=O)N2CC(CO)(NC(c3nc(O)sc3C)=O)C2)c1 92780,c1(OC)c(Cl)ccc(C(=O)NC(CNC(=O)CCc2cnn[nH]2)C(C)(C)C)c1F 92781,C1(C(=O)NCC(C)C#N)CCC(NC(=O)C=Cc2cocn2)CC1 92782,N1(C(c2cc(NC(C)=O)on2)=O)CC2(CCN(C(=O)OC(C)(C)C)CC2)CC1C 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92974,C=CC1(C)COCCN1c1nnc(-c2cc(C)cc(F)c2)n1CCOC(C)C 92975,CCC(CCCC(=O)NC(C)CCC(C)(C)C)NC(c1n[nH]cc1C)=O 92976,c1(OC(C)C)nc(C(=O)NCCSC(C)C)ncc1F.N12CC3C(C3C1)C2=O 92977,CC1(C)CC1(C(=O)NCC1CC(=C2CC2)C1)NC(=O)C=CCO 92978,C1(C2C(C(C)(F)F)C2)CN(C(C2CCSCC2)=O)CC1NC(C1CCC(=O)N1)=O 92979,c1(CNC(Cc2c(C)nc[nH]2)=O)ncc(C(N2CCC(CC(F)F)C2)=O)cn1 92980,n1(C(C)C)ccc(CC(=O)NC(CNC(c2csnc2Br)=O)C2CC2)n1 92981,C1(N2C(=O)C3(F)CN(C3)C2=O)CCCC(C)(C)O1.c1(C(C)=O)ccccc1Cl 92982,C1(F)(CNC(CCC#CC)=O)CCN(C(C2CCC2C)=O)CC1 92983,C1(C(=O)NCC2(COC)N(C(CCCCOCC)=O)CCC2)CC(=O)NC1(C)C 92984,N1(C(COCC#C)=O)CCN(C(=O)C(n2nnnc2C(C)C)C)C(C)C1 92985,c1(OCc2nn(C)cc2Br)cc(Br)ccc1C(N1CC(C)C1)=O 92986,c1(CC(=O)NCC2OCCN(C(CCSCC)=O)C2)ccc(C)cc1Cl 92987,c1(C(C)=O)ccc(C(=O)N(CC(C)CNC(=O)C(F)C(C)C)C)nn1 92988,c1(C(=O)NCC2C(NC(=O)CN3CCOCC3)C2)ccc2cccnc2c1 92989,c1(C(=O)NC2C3CN(C(C=CC=CC)=O)CC2C3)cccc(C#CC2CC2)c1 92990,N12CCN(C(c3ccccc3)C1)C(=O)NC2=O.C1(C(F)(F)F)C2CCCC12 92991,c1(C(=O)NCC2N(C(C(c3cnccn3)C)=O)CCCC2)cccc2c1CNC2=O 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93113,CCCCCCC(=O)NCC(c1ccccc1F)NC(=O)CC(C)C(C)C 93114,N1(C(CCOCC#C)=O)CCC2(CCC(CNC(c3cccc(F)n3)=O)C2)CC1 93115,c1(C(N(C)Cc2cn(-c3ccccc3C#N)nn2)=O)ccc2nnnn2c1 93116,Cc1coc(C=CC(=O)NCC(CNC(=O)Cn2cccnc2=O)CO)n1 93117,N1(C(C(CO)SC)=O)C(C(N2CC(O)CC2CN(C)C)=O)C2CC(O)C1C2 93118,c1(C(=O)NCC(CNC(=O)CCCc2ccccc2)OC)ccc2ncsc2c1 93119,C1(CCNC(C(CC)OCC)=O)CN(C(=O)C(C)NC(=O)C=C(Cl)Cl)CCO1 93120,N1(CC(=O)NCC(CNC(C2(C)CC(F)C2)=O)CO)CC(=O)NC1=O 93121,c1(OC)cc(OC)cc(C(=O)NC2CN(C(=O)C=Cc3cncs3)C2)c1 93122,C1(C(=O)NC(CNC(CCn2ncc(C)c2)=O)C)CCC(O)CN1C 93123,c1(CCN(C)C(C2CSCN2C(C2CCCC2)=O)=O)cccc(O)c1 93124,C1(CC(=O)NC2C(NC(Cn3cc(C(C)=O)nn3)=O)C2)NC(=O)NC1=O 93125,c1(NC(C2(CNC(CC(C)O)=O)CC2)=O)ccc(Cl)c(Cl)c1 93126,c1(OC)ncc(NCC2(Cc3cccc(Br)c3)CC2)c(C)n1 93127,c1(N(CC(C)CNC(=O)CC(C)C(F)F)C)ccc2c(n1)CC(C)(C)CC2=O 93128,N1(C(Cn2nnc(C)n2)=O)CC(C(=O)NC(c2cn(C)nn2)(C)C)CCC1(C)C 93129,C1(CNC(C=CC(CC)C)=O)CCCC2CN(C(c3nc(C)nn3C)=O)CC12 93130,CC1(C)CC(CNC(C2(C)CCC(=O)N2)=O)CN(C(=O)CCCc2ccsc2)C1 93131,CC(C)(CC(=O)NC(CO)C(C)NC(=O)CN1CCCNC1=O)c1ccccc1 93132,C(C)(CN=[N+]=[N-])NC(N(C(COC)C)C1CC1)=O 93133,C1(NC(C)Cc2ccc(Cl)cc2Cl)CC2CCC1(C)C2(C)C 93134,C=CCC(C(=O)NCC(C(C)(C)C)NC(c1cnn2c1CCC2)=O)C(C)(C)C 93135,C12CC(F)(F)CN1C2=O.c1(NC(CC(=O)OC)=O)oc(SC(C)(C)C)nc1C 93136,CCCCC(C(=O)NC1CCCCN(CCc2nnc(C)o2)C1)NS(C)(=O)=O 93137,Cc1ccc(F)cc1C(N1CCN(C)CC1C(=O)N(C1CCOC(C)(C)C1)CC)=O 93138,c1(C(N2CC3C(NC(=O)CCC4CC(F)(F)C4)(C3)C2)=O)cc2c(o1)CCCC2 93139,C(c1cc(C)c(C)cc1C)=CC(=O)NCC(CNC(C(CC=C)N(C)C)=O)(C)O 93140,CCC(C)(C)C(C)NC(=O)C(C)CNC(=O)CN1CCOC1=O 93141,N1(C(c2nc(C(N)=O)sc2)=O)C2CCC1C(NC(=O)C(O)Cc1cnc[nH]1)C2 93142,C12(C(=O)NCC(CC=C)NC(=O)CCOc3ccc(Cl)cc3)CC1COC2(C)C 93143,N1(C(C(C)O)=O)CCC(CO)(CNC(c2cc(-c3cccc(Cl)c3)on2)=O)C1 93144,N1(C(c2snc(C)c2Br)=O)CCN(C(=O)C(C)C2CC2)C(C)C1 93145,C12(NC(CCC=C=C)=O)CCN(C(=O)C=C(C)CN3CCOCC3)CC1C2 93146,N1(C(C(=CC2CCCC2)C)=O)CC2OCC(NC(=O)CSc3cccs3)C2C1 93147,N#Cc1cc(S(=O)(=O)N2CC(F)CC(F)C2)ccc1NCCOc1ccccc1Cl 93148,N1(C(=O)OC)CC(C(C(=O)N(C)CC2CC2Cl)OC)C1 93149,c1(N(CCCN(C(Cn2nnc(C)n2)=O)C)C)ncnc2cc(Br)ccc12 93150,C1(NC(c2cnn(CCC)c2C)=O)CCC12CN(C(=O)CCC(C)OC)C2 93151,C(=O)(N=c1ccc(C2CC2)n[nH]1)NCC1OCC(C)(C)C1 93152,c1(C(=O)NC2C3CN(Cc4ccc(C)cc4F)CC32)ccc2oncc2c1 93153,CC1(C)CC(CNC(C2CCCCNC2=O)=O)CN1C(=O)Cn1nnc(=N)[nH]1 93154,N1(C(C(CC)C)=O)CCC2(CCN(C(c3cnc(OC)cc3C)=O)CC2)C1 93155,C1(C(N(CCCO)C)=O)COC(CNC(=O)CSCC(N)=O)C1 93156,N1(CC(=O)NCCc2c(-n3cccn3)ncnc2Cl)CCC(CO)C(F)C1 93157,c1(C(=O)NC2C(C(=O)NCCC(C)C)C2)cc(C(=O)OC)cc(C(F)(F)F)c1 93158,CC(CC(C)(C)C)C(=O)NC(C)CCCCNC(C1CCCC(=O)N1)=O 93159,Cc1ccc(C)c(OCC(C)(C)NC(=O)Cc2nnnn2C2CC(F)(F)C2)c1 93160,c1(C(C2(F)CC(COCOCC)C2)=O)cnn(C)c1C(=O)O.C(CCCO)OC 93161,C(CCC(=O)N(C1CCC(NC(=O)Cn2nccn2)C1)C)=CC(C)C 93162,c1(CNC(C(C)C)(C)c2nnnn2C2CC2)ccccc1-c1cccc(CSC)c1 93163,c1(CNC(CC2C3CN(C(C4(C)CC(=C)C4)=O)CC32)=O)nnc2n1CCC2 93164,c1(C(N(CCC(=O)NCc2c(OCC)scc2)C)=O)cc(C)ncc1C 93165,c1(C(N2C3C(NC(C(CC)C)=O)C(C3)C2)=O)cnc2ncnn2c1O 93166,C=C(CNC(C1CC1C(F)(F)F)=O)CCNC(C1(C)CC1(F)F)=O 93167,CC1(C)OCCC1C(=O)NCCCN1CCN(C(c2[nH]ncc2C#N)=O)CC1 93168,C(=O)(C(CC(C)(C)C)OC)N1CCN(C(CNC(C2C(CCC)C2)=O)(C)C)CC1 93169,C=Cn1nccc1C(N1CC(OCC(=O)NCCC(C)N(N2CCCC2)C)C1)=O 93170,C1(C(=O)NC2CC(Nc3ccnc(C(CC)C)n3)C2)CC2CCCC2C1 93171,C1(C(=O)NCC(C)NC(C2CCS(=O)(=O)CC2)=O)CCc2nc(O)[nH]c2C1 93172,C1(NC(CCC)(C)c2nnnn2CCCC2CC2)CCCS(=O)(=O)C1 93173,C1(CC=C)(NC(=O)CCCc2ccccc2)CC2CCC(C1)N2c1nnc(C)o1 93174,Cc1nc(C2CC2)ncc1C(=O)NC1CC1CNC(C1(Br)CC1)=O 93175,C(CCN=c1[nH]cncc1I)CCC(N1CCCCC1)=O 93176,C(=O)(N1CCCc2nccn21)c1cc(CNC(=O)C2CC2)[nH]n1 93177,CC(CCc1ccccc1)C(=O)N(C)C(c1cncn1C)C 93178,C1(C(N(CC(=O)NC2COCC2Cc2c[nH]nc2C)CC)=O)CN(C)CCO1 93179,C(CC(=O)NCC(C)(O)CCO)(C(C)C)NC(COCC)=O 93180,c1(CNC(CNC(C(CC)N(C)CC2CC2)=O)=O)c(F)cccc1F 93181,c1(C(=O)NC(CCNC(C(C2CC(F)(F)C2)OCC)=O)C)ccsc1CC 93182,Cc1cc(C(c2nnnn2C)NCc2nc(C(C)(C)C)no2)cc(Br)c1 93183,C(C(CCS(C)(=O)=O)OC)NC(c1ccc(Br)o1)COC 93184,c1(C(=O)NC(C)C(C)NC(c2cn(C)c(O)n2)=O)cc2c(Br)ccc(F)c2[nH]1 93185,N1(CC(C)NC(c2onc(CC)n2)C)CCN(C(=O)C(C)(C)CF)CC1 93186,N1(C(C(C2CCN(C(C3CCC(CC)CC3)=O)C2)C)=O)CC2CC(C)C2C1 93187,CCCCCC(O)CNC(=O)C(C1CN(C(c2cc[nH]n2)=O)C1)OC 93188,C1(C(=O)NC2(CNC(C(CC(=C)C)C)=O)CCCC2)CC(c2ccccc2)=NO1 93189,N1(C(c2cnc(C)[nH]2)=O)CCc2nc[nH]c2C12CCN(C(C1(C)CCCO1)=O)C2 93190,c1(C(=O)NCC(CCOC)NC(C=C(CCC)CCC)=O)ccc2ncsc2c1 93191,c1(C(=O)NCC23CC(CO2)N(C(C2CCCCC2)=O)C3)cnnc2ccccc12 93192,c1(NC2(c3ccccc3)CCN(C(=O)OC(C)(C)C)C2)nsc2ccccc12 93193,N1(C(CCCNC(C)=O)=O)CCCC1C=CC(=O)N(C(C)CC1CC1)C 93194,C(CN=C(NCc1cnccc1N(C)C)NCC1CC2C(C1)C2(F)F)OC 93195,c1(C(N(CCCCCCNC(C2CC2(F)F)=O)C)=O)ccc2c(n1)COCC2 93196,c1(OC)ccc(SCC(=O)NCCC(C)CCNC(=O)C=CC2CCC2)cc1 93197,C1(C(C)C)C(C(=O)NC2COCC2C(F)(F)F)CCN1C(c1ccncc1F)=O 93198,C1(CNC(c2cnn(C3CC3)c2)=O)CCCCN(C(C2(F)CCCCCC2)=O)C1 93199,CCCCCCN(C(=O)C(F)OC(F)(F)F)CCNC(C1CCC1n1ccnc1)=O 93200,Cc1cc(C(=O)NCC2(F)CN(C(=O)CN3CCC(F)(F)C3)C2)cc2nn[nH]c12 93201,N1(CC)CCOC(Cn2cc(-c3cncn3C)nn2)C1c1cnn(C)c1 93202,c1(-c2cn(CCC(=O)N(C3CCC(OC)CC3)C)nn2)c(C)nc(O)nc1C 93203,CC1=C(C(=O)N(CC(C)C(=O)NCC2(CO)CC=CC2)C)CCO1 93204,C1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)CC(C)(C)OC(C)(C)C1 93205,c1(OC)ccc(C(=O)NC2CC(NC(=O)C=Cc3cccs3)C2)cc1F 93206,c1(OC)ccc([N+](=O)[O-])cc1NNC(=O)C1CCSCC1 93207,N1(C(CC(=O)NCCCCCC)=O)CCC(NC(=O)C(O)C2(CO)CC2)C(CC)C1 93208,c1(C(c2nnnn2CCC2CC2)NC(CCC(=C)C)C)ccc(C)cc1[N+](=O)[O-] 93209,CC12CC(CC(=O)N(CCCNC(C3CCCC(C(N)=O)C3)=O)CCO)(CO1)C2 93210,c1(OC)ccc(C(C)NC(=O)C(=O)NCC(O)CC(F)(F)F)cc1OC 93211,c1(COC)ccc(CNC2C(C(N3CC(CF)C3)=O)CCC2)cc1 93212,C(CCNC(C1(n2cncn2)CC1)=O)(C(C)C)NC(c1c(CC)n[nH]c1)=O 93213,CCCCCCCC(=O)NC1CCN(C(C2(CCC)CC(=O)C2)=O)CC1C 93214,N1(C(C2(OC)CCCCC2)=O)CC(CNC(=O)C(C)SC)C(C)(C)C1 93215,CC(C)C(CC1(C(=O)O)CC1)N=c1nc(O)c2cnn(C(C)(C)C)c2[nH]1 93216,c1(C(N2CCC(O)(CN(C)C(C3CCS(=O)CC3)=O)C2)=O)ccccc1S(C)=O 93217,c1(C(N2CC(C)N(C(=O)CC3CCCCN3C)CC2)=O)cnc2ccnn2c1O 93218,Cn1nc(C(N2CC(O)CCC2C(N2CC(N3CCOCC3=O)C2)=O)=O)cc1C#N 93219,c1(C(=O)NCc2occ(C(=O)NCCC3(O)CCC3)c2)cccc2ccoc12 93220,C1(CNC(C2N(C(C)C)CCC2)=O)CCN(C(C2CSCC(=O)N2)=O)CC1C 93221,N1(C(C=CCNC(c2nn(C)c(Cl)c2)=O)=O)CCNC(=O)CC1 93222,C1(NC(c2cc(C)sn2)=O)CCN(C(c2cscn2)=O)CC1(C)C 93223,CCC(COC)S(=O)(=O)NC(=O)CCc1nc(C(C)C)no1 93224,C1(C(N2C(CNC(C(C)OC)=O)COCC2)=O)CCc2ccc(F)cc2C1 93225,Cc1cc(C(=O)NC(CO)C(=O)NCCn2cncn2)nnc1O 93226,c1(OC)cc(C#N)ccc1C(=O)Nc1cc(-c2cn(-c3ccccc3C)nn2)cs1 93227,c1(C(=O)NCCNC(c2c(CC)nc[nH]2)=O)cc(C)nn1C1CCC1 93228,C1(C(=O)NCCCC)CC12CCN(Cc1ccc(Br)cc1F)C2 93229,N1(c2nc(C)nc(C#N)c2)CCCC(C2(NC(C3C4CC5C(C4)C35)=O)CC2)C1 93230,C1(CC(N2C(CNC(C(N3C(=O)CCC3=O)CC)=O)CCC2)=O)CCCC(=O)N1 93231,C=CCC(C(=O)NCC1CC2(CC2)CN1C(c1cnn(C2CC2)c1)=O)C(C)C 93232,c1(C2CCN(C(C(C)(C)NC(C3CCCC(C)C3)=O)=O)C2)cc2scc(Cl)c2[nH]1 93233,C(N=c1[nH]cnc2cc(Br)ccc12)C1(C(=O)NCC(C2CCS(=O)(=O)C2)O)CC1 93234,n1(CC)c(C)cc(C(N2CCN(C(C3CCC(C)O3)=O)CC2COC)=O)c1C 93235,c1(C(=O)NC(C2CCN(C(C(C)O)=O)CC2)C)cc(P(C)(C)=O)ccn1 93236,C1(O)(CN(C)C(c2ncccc2Br)=O)CCN(C(C2CCC(=O)NC2)=O)C1 93237,c1(C(N2CC(O)CC(NC(c3c(C)ncs3)=O)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 93238,c1(OC)cc(C)c(CCNC(C2(F)CCOC2C)=O)cc1C 93239,CC1CC(N=c2[nH]c(C3CCCC3)nc(=N)[nH]2)CCN1C(c1ccc(CO)s1)=O 93240,C1(C(=O)NC2CCN(C(C3(c4ccsc4)CC3)=O)C2)CCC(CO)CC1 93241,CN1CC2(CC2)CC1C(=O)NC1CN(C(=O)Cc2ccoc2)CC1F 93242,CCC(C)C(C(=O)NCC1(C)CN(Cc2ccccc2OC(C)C)CCO1)OC 93243,CC(C)CC(CC(=O)NCC(F)C1CCC1)NC(c1ccc(O)cc1)=O 93244,Cc1oc(C(N2CC(NC(=O)C(O)Cc3cn(C)cn3)C2)=O)cc1S(C)(=O)=O 93245,C(C(C)(C)CC(=O)NCC1(CO)CC2CC2C1)NC(c1c(CCC)[nH]cc1)=O 93246,N1(C(C(C2CCCCC2)OC)=O)CCC2C(C1)CN2C(c1cn2ccsc2n1)=O 93247,c1(NC(C)=O)ccc(N)c(C(=O)N(C)CCN(C)C(C2CC2C)=O)c1 93248,C(C(=O)NOC1CC1)(c1ccoc1)NC(C1C(C#C)C1)=O 93249,c1(NC(=O)C(N2CCC(c3ccc(Br)cc3)C2)=O)ccc2c(c1)CCO2 93250,N1(C(COCCC=C)=O)CC2CCC1C(NC(c1ccc(Cl)c(F)c1O)=O)C2 93251,N1(Cc2cn(CCN(C(C3(C)CCCOC3)=O)CC)nn2)CC2CS(=O)(=O)CC2C1 93252,C12(COC)CC(CNC(=O)CC)(CN1C(=O)CCCCF)C2 93253,C1(=O)CS(=O)(=O)CCO1.C#Cc1ccc(OCC)cc1.C12CCC1OCC(=O)N2 93254,c1(C(N2CCCC(C(C)(C)C)C2)=O)ncn2c1CCC2 93255,Nc1c(C(N2CCN(C(c3cc(O)cs3)=O)CC2CF)=O)nnc2ccccc12 93256,c1(CC)cc(OC)nc(N2CCCCC2c2cncnc2)n1 93257,c1(CC)nc(C(=O)NC2(CNC(c3nc(C)oc3OC)=O)CC2)c2ccccn12 93258,CCCC(C)(O)C(=O)NCC1(F)CCN(C(=O)CCc2ccc(Cl)nc2)C1 93259,CC1(C)CCCC(C)(NC(=O)C(C2(O)CN(C(=O)C(C)n3ccnn3)C2)F)C1 93260,c1(CC(=O)NC(CSCC)C(=O)NC2CC(n3ccnn3)C2)ccccc1O 93261,c1(C(=O)NC(C(C)(C)C)CNC(C2(CO)CCCC2)=O)ccc2cccnn12 93262,CCC(CCOC)C(=O)N1CCCC(CCNC(C2(O)CCSC2)=O)C1 93263,C(=O)(C(CCF)NC(c1cccnc1)=O)N(c1c(C)nsc1)C 93264,C1(CNC(=O)C2=CCOC2)CC2(CCC2)CN1C(=O)COc1ccc(F)cc1 93265,C1(O)(CCNC(c2n(C(C)C)ccn2)=O)CCN(C(c2cc(F)c[nH]2)=O)C1 93266,N1(C(c2c(C)cnn2C)=O)CC2(CCCC2NC(=O)C(F)=CC2CC2)C1 93267,C1(C(=O)NC(CCCCC)C)CC2(CCC2)CN1C(C1CCCCC(=O)C1)=O 93268,CC1CCn2ncc(C(=O)NCC(C)(C)NC(c3ccc(N)cc3O)=O)c2C1 93269,C(c1cccc(Cl)c1Cl)=CC(=O)NCC1CCN1C(C1CC2(CC2)C1)=O 93270,Cc1c(Cl)c(C(=O)NCC2CN(C(c3nc4c(s3)CCC4)=O)CCC2C)nn1C 93271,N1(C(C2CCN(C(c3cncc(C)c3)=O)CC2)=O)CCc2c(C#N)cccc2C1 93272,CC(CS(C)=O)C(=O)NC1(CNC(=O)CN(C2CCC2)C)CCC1 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93362,C12CCCCN(C1)C2=O.C=CC(C)(C)C(=O)NCC1(F)CCN1C(=O)OC(C)(C)C 93363,c1(CC(=O)NCC(CCOC)NC(=O)C=C(C)c2ccsc2)cc[nH]c(=N)c1 93364,c1(OC)cc(C2CC2)cc(OC)c1O.C1(C(CNC)=O)C2CC3C(C2)C13 93365,Cc1ccc(C=CC(=O)N(CC(=O)NCC2CCC2)CC(C)O)o1 93366,N1(C(c2c(OC)nccn2)=O)CC(C2CC2)(C(N2CC3CCC=CC23)=O)C1 93367,N1(C(c2ncc(CC)s2)C(=O)NCCCCCC)Cc2ncsc2C1 93368,CC(CC(=O)N(CCCNC(=O)Cc1csc(-c2ncccn2)n1)C)C(C)(C)C 93369,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cnc4[nH]ncc4n3)=O)CC1C2)OC 93370,N=c1[nH]nc(CC(=O)NC2CCC(CCNC(c3cc(Cl)c[nH]3)=O)C2)s1 93371,C1(CCNC(=O)C(F)n2cccn2)(NC(c2ccc(F)cn2)=O)CCOCC1 93372,C(CCCCCC=C)NC(C(CN(C(c1c(C#C)c[nH]n1)=O)C)C)=O 93373,N1(C(CC(c2c(C)cccc2)C)=O)CCOC2(C1)CN(c1ccc(C#N)cn1)C2 93374,C1(NC(CC(CC)SC)=O)CCN(C(=O)COc2cccc(F)c2F)C(C)C1 93375,C(C1c2ccsc2CCN1C(c1ccc(F)cc1)=O)NC(C(COC)O)=O 93376,C1(CNC(Cc2c(C)noc2C)=O)C2CCC(C2)N1C(c1[nH]ccc1C1CC1)=O 93377,C1(NC(c2nn(C)c(O)c2)=O)CCCC(C(=O)NOCC2CC2)CC1 93378,c12ccc(cc1)CC(c1n(CCCC)nnn1)(C)N2.C(C)(C)(C)OC(=O)NC 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93415,c12sc(cc1C)N(C1CCCCC1)C(C)C(=O)N(C)C1CCN(C1)C2=O.CC 93416,c1(C(N(CC(=O)NCC2CCSC2)CCOC)=O)cnn(C(C)(C)C)c1 93417,CCS(=O)(=O)CC(=O)N(C(C)CCCc1ccccc1)C(C1CC1)C1CC1 93418,N1(C(=O)OCC)CCC(CNC(=O)C(C)Oc2ccccc2OC(F)F)C(O)C1 93419,C1(CCCCCNC(CCC#C)=O)CCN(C(c2ncn(C)c2C)=O)CC1 93420,N1(C(c2cc(OCC)no2)=O)CC(C(=O)NCC2CCN(CC)C2)CCC1C 93421,c1(SC)ccccc1C(N1CCC(N(C)C(C2CCCC2(F)F)=O)C1)=O.C(C)(C)(C)N 93422,n1(C(C(C(CC)(C)C)O)C)cnc2c(N(c3ccc(F)cc3C)CC)ncnc12 93423,C12(C(=O)OC)CCCC1N(C(c1csc3ccccc13)C(=O)NCC(C)C)CC2 93424,C1(NC(C(C)=CC2CC2)=O)CC1C1CCN(C(c2nccc3n[nH]cc23)=O)CC1 93425,c1(SC)ccc(C(N2CCC(C(=O)NC3(C)CCN(C(C)=O)C3)C2)=O)cc1 93426,C1(NCC(C)(O)Cn2cc(Br)cn2)CC12CCN(S(=O)(=O)CC1CCC1)CC2 93427,Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)(NC(=O)CC2CC=CCC2)C1 93428,c1(CC(=O)NCC2N(C(CCC=C=C)=O)CCC2)c(C)nc2ccccc2c1C 93429,S(=O)(=O)(c1cccs1)CCCCN1CCC(N(c2c[nH]nc2C2CC2)C)CC1 93430,C1(C)CCC2(C1)COCCO2.C1(c2nnn[nH]2)(CC(F)(F)F)CCN(C2CC2)C1 93431,C1(C(=O)NC2N(C(C)=O)CC2)CCC2(CN(c3cc(Cl)nc(C4CCCO4)n3)C2)O1 93432,CC1CCN(C(=O)CC2(C)CCOC2)CC1CNC(C1(C)CCC1)=O 93433,C1C(C)CN=C2C=CN=C(N2)N1C.c1(C(CC)SCCCC)nnc(C)s1 93434,C1(C)(C(N2CCC(NC(C3(CCOC)CC3)=O)CC2)=O)CCN(C)C1=O 93435,CCC(CNC(c1cncs1)=O)(CC)NC(C12CCCC1(C(N)=O)C2)=O 93436,c1(C(=O)OC)sccc1S(=O)(=O)Nc1cc(C(F)F)cc(C(F)F)c1 93437,C1(NC(C=NOC)=O)(CNC(=O)C(C2CC2)OCC)CCCCC1 93438,CCC(C)(C#N)C(=O)N1CC(NC(c2oncc2C)=O)C(C)C1 93439,Cc1ncc(C(N2CCC(CCNC(=O)Cc3cncnc3)C2)=O)c(C)n1 93440,c1(CC(N2C(CNC(C(CC)C(C)C)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 93441,c1(C(C)C)cc(C(=O)NCC2CC(CF)C2)cs1.N12CC(C1)C2=O 93442,c1(NC(C2(OC)CCN(C(=O)CC(CC)SC)C2)=O)cnc2ncnn2c1 93443,C(=O)(C(CCC(C)(C)C)OC(=O)CCc1c(C)cccc1Cl)OC 93444,N1(C(CSCC)=O)CC(C)CCC1CNC(c1nc(-c2ccncc2)no1)=O 93445,C1(C(C)(C)O)C2CN(C(C3CCO3)=O)CC12.C1(C(=O)O)CCC1 93446,C1(CCC)CN(C(=O)C(CC)Oc2ccccc2)CCN1C(c1cc[nH]c1)=O 93447,C(=O)(C(O)CCCSC)C(C#C)CN(CC(=O)OC)C 93448,N1(C(c2c(CC)cc(N)cc2)=O)CCCC2(NC(c3ccc(OC)s3)=O)CC2C1 93449,c1(NC(C)=O)ccc(CC(=O)NCC2CCC(NC(c3ccsc3C)=O)C2)cc1 93450,C1(CCC(=O)NCC(C(C)C)=O)CCCCN(C(C2CC(=C3CC3)C2)=O)C1 93451,CCCC(O)CN(C)C(=O)NCCCc1cn(C2CCOCC2)nn1 93452,C1(NC(C2(C)CC(F)C2)=O)CCCCC1NC(=O)CSc1ccccc1Cl 93453,C1(C(=O)NC(C)C(CO)NC(=O)C(O)C2CCC2)CC(C(C)(C)C)=NO1 93454,c1(C(=O)NCCc2ccc(CNC(CC=C(C)C)=O)cc2)ccc(O)c(C)c1 93455,N1(C(C2(N(C)C)CCCC2)=O)CCOC(C)(CNC(c2cncc(Cl)n2)=O)C1 93456,CN1CCC(NC(=O)N(C(c2ccccc2)Cc2ccccc2)C)C1 93457,CC1(C)CC(NC(=O)CCNC(=O)C2CC2)CCN1 93458,c1(CC)cc(N)ccc1C(=O)NCC1CCCN1C(=O)CCc1cnc(O)[nH]1 93459,c1(C(N2CCCC(NC(=O)CCCF)CC2)=O)cc2cccc(F)c2cn1 93460,c1(COC(c2cnn(Cc3cccc(Br)c3F)c2)=O)ccc([N+](=O)[O-])cc1 93461,c1(C(=O)OC)cnc(C)[nH]c1=NCC(C)NC(=O)C1CCCc2n[nH]cc21 93462,CCCC(CNC(=O)C(=O)C(C)(C)C)C(=O)N1CCC2(CSC2)C1 93463,C1(NC(C2N(C(C)=O)CCOC2)=O)CC2(C1)CN(C(=O)C(=O)NC1CC1)C2 93464,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 93465,N1(CC)CC(CN(C(=O)COC(C)=O)C)C1.C12(CC1)C(=O)NC2 93466,Cc1cc(F)c(C(N2CCCCC2CNC(C2CCCN2C=O)=O)=O)cc1F 93467,n1(CCC)cc(-c2cn(CC(=O)OC(C)C)nn2)c(C)n1.C12CN(CCO1)C2=O 93468,c1(OC)ccc(NC(=O)NC(=O)NC2CC2)cc1CO.c1(SC)ccccc1 93469,c1(C(=O)NC(C)CCCCNC(=O)Cn2cncn2)ccc(C2CC2)nc1O 93470,N1(CCN(C)C)CCC(=O)N(CCC(=O)SC2CCCO2)C1=O 93471,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 93472,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 93473,N1(C(c2nc(C)sc2)=O)C2CCC1C(NC(c1cnc(C3CC3)[nH]c1=N)=O)C2 93474,C(CCNC(C1C(SC)C1)=O)(C(N)=O)NC(C(CC)N(CC)CC)=O 93475,c1(C(=O)NCc2cn(CC(=O)N(CC(=O)OC)CC#C)nn2)ncc(F)cc1F 93476,Cc1oc(C2CCOCC2)nc1C(=O)NCC(C)CN(C(=O)CC1CC1(C)C)C 93477,Cc1sccc1C(N1CCC(CCNC(C2(c3ccccc3)CC2(C)C)=O)C1)=O 93478,CC1CSc2ccc(C(=O)NC3(CNC(=O)CNc4nccs4)CCOC3)cc2N1 93479,c1(C(=O)OC)cccc(CC(=O)NCC(C)N(C)C(c2ccc(Br)cn2)=O)n1 93480,N(C(=NCc1ncn(CC)n1)NCCNC(C)=O)C(c1cnc(COC)[nH]1)C 93481,CC(CCc1ccccc1)CC(=O)NCC1(O)CN(C(=O)CC2CCCOC2)C1 93482,n1(CC(=O)N(CC(CNC(C2(OCC)CC2)=O)C)C)ncc(Br)c1C 93483,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(C(C)C)noc2)=O)C1(C)C 93484,c1(CC(N2C(CNC(c3ccsn3)=O)CC3CC32)=O)cc2ccccc2o1 93485,c1(COCCCC(=O)OC)csc2cccnc12.C12CCC(C1)C(=O)N2 93486,C1(C(N2CC3C(NC(CCc4nc(C)sc4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 93487,N1(C(C2CC(NCC3CCCC3c3ccccc3)C2)=O)CC2CC23CC13 93488,CC(C)(O)CC(=O)NC1CCN(C(=O)COCc2ccc(Cl)nc2)C1 93489,c1(CC)ccc(C(=O)NCC2CCCCCN2C(C2CCC(=O)C2)=O)cc1Cl 93490,Cc1snnc1C(N1CC(CO)(NC(=O)Cn2cnc(C(N)=O)n2)C1)=O 93491,C(C(=O)N=c1cc(C)[nH][nH]1)C1N(C(c2c(C)cccc2I)=O)CCNC1 93492,CCC(CCC(=O)NCCCC(C(C)C)NC(=O)CCS(=O)(=O)CC)OC 93493,N1(Cc2cccc(C(C)NC(=O)NC3CC3)c2F)c2ccccc2SCC1C 93494,Cc1nc(O)nc(C)c1CC(=O)NCC(C)(O)CNC(=O)CN1CCOCC1 93495,C1(OOC(=O)COC(c2c(Cl)ccc(C)c2N)=O)CCc2cc(Br)ccc2O1 93496,Nc1ccc(C(=O)NC2CC(CCC(=O)NCC(F)Cl)C2)nc1F 93497,C1(CNC(CSCC=C)=O)CC2CCC1N(C(c1cc(C)nc(N(C)C)n1)=O)C2 93498,N1(C(C(C)SC)=O)C2CCC1CC(NC(c1ccc(O)c(C)c1C)=O)C2 93499,c12ccc3c(c1)COC31CN(C1)C(C(=O)NCC)c1cccc-2c1.CCCOCC 93500,N1(C(c2cc(C)cc(F)c2)=O)CC(NC(c2cccc(C)n2)=O)C2CCCC12 93501,C1(NC(C(C)OCC2CCCO2)=O)C2CC(NC(=O)CC3(O)CCOCC3)CC12 93502,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CC2)nccc2n[nH]cc12 93503,c1(CC(C)(O)c2cccs2)cn(CCN2CCC(NC(=O)Cc3ccns3)C2)nn1 93504,N1(C(c2ccc(C)c(O)c2)=O)CC2CC1CCC2NC(c1n[nH]cc1C(C)C)=O 93505,CCC(C)(C)C(=O)N1CCCC(CC(=O)NCCCNC(=O)OC)C1 93506,c1(C(=O)NC2CCCN(C(C(C)N(C(C)=O)C)=O)CC2)cc2cnccc2[nH]1 93507,C(C(C)(C)C(C)(F)F)N(C(=O)CP(C)(C)=O)C(C1CC(C(C)C)C1)=O 93508,C1(NC(c2cc(OCC)n[nH]2)=O)CN(C(C2(C)CC(F)(F)C2)=O)CC1F 93509,c1(C(C)C)cccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cnnn2)n1 93510,c1(CNC(CC(c2ccc(O)cc2)N)=O)c(F)ccc(Cl)c1F 93511,C(=O)(C#CC1(C)CC1)N(C)CC1N(C(CCC(=O)N(C(C)C)C)=O)CCCC1 93512,C1(C)(CNC(C2C(C(=O)OC)CCO2)=O)CCN(C(=O)CN2CCOCC2=O)C1 93513,C(=O)(C(C)(O)C(C)OC)NC1CC2(C(NC(CC(=C)C)=O)C2)C1 93514,C(=O)(C(C)(C)C(=O)N1CC(CNC(c2cccc(F)c2C)=O)C(O)C1)OCC 93515,C#Cc1cccc(CC(=O)NC2CCOCC2C(N2CCOCC2C(C)O)=O)c1 93516,CC(C)C(C)C(CNC(=O)C(c1cnn(C)c1)O)NC(=O)C=Cc1cncn1C 93517,N1(C(CC2C(NC(C(C)CC3CCCC3)=O)CCC2)=O)CC2CCC(C1)C2O 93518,N1(C(c2c(F)ccc(C)c2)=O)CC2CCN(C(C3CC4CC3CC4O)=O)C(C2)C1 93519,C(CC(=O)NCC(C)CNC(=O)CCNC(C1CCC1)=O)N(C(C)=O)C 93520,c1(-c2scc(C(=O)NCC(C3CCCCC3)NC(C)=O)n2)cccc(Cl)c1 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93750,c1(CNC(CCCCNC(c2c(CCOC)n[nH]c2)=O)=O)cc(C)cnc1F 93751,C(CC(O)C(F)(F)F)NC(C)(C)C.C1C(C)(C2CC2)NC(=O)O1 93752,C1(C)(CNC(C(C)SC)=O)CCN(C(c2cncc(CO)c2)=O)C1.C(N)=O 93753,CC(=O)CCCCC(=O)N1CC2CCC(Nc3cc(-n4ccnc4)ncn3)C2C1 93754,C1(C2(OC)CCC2)(NC(CC2CC(CNC(C(CCC)=CCC)=O)C2)=O)CC1 93755,N1(C(C)C(=O)NCC(c2ccccc2)NC(=O)CC2CC2)CCC(O)CC1 93756,c1(NC(=O)NC2CCN(C(=O)C=Cc3ccccc3)C2)ccc2cccnc2n1 93757,N1(C2(C)CC2)CCCC1CN(C(C1CC(C(=O)OC)C1)=O)C1CC1 93758,c1(C(COCCN(C)Cc2ccc(F)c(F)c2)O)ccc(Cl)c(F)c1 93759,c1(CN2CCN(CC(=O)Nc3cccc(O)c3)C(=O)C2)cnc2[nH]ccc2c1 93760,N1(C(C=COCC)=O)CC(NC(c2nc3ncccn3n2)=O)CC12CCOCC2 93761,c1(OC)ccc(C(F)F)cc1NC(=O)C(=O)NCC1CC(=O)C12CCC2 93762,c1(OC)nn(C)cc1C(=O)NC(C)C(C)C(=O)NCCCCC1CCCC1 93763,C1(C(N(C(C)C)CCO)=O)CC(NC(C2CC(F)(CF)C2)=O)CCO1 93764,Cc1nc(C(=O)NC(C)(C)C(C)NC(=O)CNC(C2CCCCC2)=O)n[nH]1 93765,C(C(O)CC(C)(C)C)NC(C(C1CCCO1)NC(c1n(CC#C)cnn1)=O)=O 93766,c1(C(=O)NC2(C)CC(NC(Cc3c(C)nsc3)=O)C2)cnn(C)c1Cl 93767,C(=O)(CC(C)C(C)C)NC1C(NC(C(C)(C)SC)=O)C1 93768,C=CCCC(O)CNC(C12CC1CN(C(=O)CCC(=O)NC)C2)=O 93769,C(CCCCC(=O)NC1(CO)CCN(C(=O)CC2CN(C(C)=O)C2)C1)SC 93770,Cc1cn2cccc(C(N3CC(CNC(C4(C)CCCC4)=O)C(C)C3)=O)c2n1 93771,CC1CCN(c2cncc(C(N3CC(N(C)C(C45CCC4C5)=O)C3)=O)c2)CC1 93772,N1(C(c2n(C)ccn2)=O)CC2CC(C(=O)NCCC(F)=C(F)F)C(C2)C1 93773,N1(C(=O)N(C(c2nc(C3CCOC3)n[nH]2)C)C2CC2)CCCC(C)(F)C1 93774,C(C(COC)C(=O)N(CC(C)(C)CNC(=O)CC1C=CCCC1)C)OC 93775,CC(C)C#CC(=O)NC1COCCC1NC(=O)CC1CC2CC2C1 93776,C(=O)(C(C)(C)C(=O)N1CCC(C)C(NC(=O)Cc2ccccc2Cl)C1)OCC 93777,N1(C(C)CNC(=O)CC2C=CCC2)CCN(C(=O)CN2CCCCC2=O)CC1 93778,C1(COC)(CNC(=O)CCn2ccnc2)CCN(C(=O)Cn2cccn2)CC1 93779,C=CCCCC(=O)N1CCC(N(C(=O)C(C)Cc2cnn(C)c2)C)C1 93780,N1(C(C23N(C(C(C4CCC4)OCC)=O)CCC2C3)=O)CC(C)(C)OC(C)(C)C1 93781,C(=O)(CCC1=CCCCC1)N1CCC(C2N(C(c3n(C)nnc3)=O)CCC2)CC1 93782,c1(OC)cccc(C(=O)NC(C)CCNC(=O)C(C)(C)C2CCCC2)n1 93783,CCCC(CC)C(=O)N(C)CC1CCCN(C(c2ccnc(O)c2)=O)C1 93784,C#Cc1ccc(C(=O)NCC2CCCN2C(=O)C(C)CN2CCOCC2)cc1F 93785,CC1CNC(=O)CC(NC(=O)Cc2ccc(Cl)c(Cl)c2)C1 93786,c1(C(N2CCCC(CCNC(CNC(C)=O)=O)C2)=O)cccc2c1CCN2 93787,C1(NC(C(CO)N(C)C)=O)CCCC(CNC(=O)CC2(c3ccccc3)CC2)C1 93788,Cc1cc(C(=O)NCCN(C(=O)CN2CCC(C)C2)C)cc([N+](=O)[O-])c1O 93789,C(=O)(C(C)CN1CCOCC1)N(CCNC(CCOCC(C)(C)C)=O)CC1CC1 93790,Cc1ccc(SC(C)C(N2CC(CNC(=O)C=C3CCN(C)C3)C(C)C2)=O)cc1 93791,C1(OC)CCC2(C(N3CC(NC(=O)C(C)OC4CCCC4)C(C)C3)=O)CC12 93792,C12(NC(c3cncc(OC)c3)=O)CCCN(C(c3ccsc3)=O)CC1C2 93793,c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)CC)ccc(Cl)c(N)c1 93794,N1(C(c2ccc(SC)cc2)=O)CC2CC1CCN2C(=O)C=Cc1nc(C)cs1 93795,C#Cc1cncc(NC(=O)C=CC2CCN(C(=O)C(C)C(C)(C)C)CC2)c1 93796,C(c1ccc(F)cc1)=C(C)C(N1CC2CC1CN2C(c1cc(O)cc(=O)o1)=O)=O 93797,N1(C(c2cn(CC)nc2C2CC2)=O)CC2(CC(NC(C3CCNC3=O)=O)CO2)C1 93798,C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NCC(C)N(C)C)C1 93799,C(=O)(C(C)(C)CC(F)(F)F)NCC1(C(N)=O)CN(C(CCCc2n(C)cnn2)=O)C1 93800,c1(C(N2C(C(=O)NCC(=O)OCC)CC2)=O)cc2cc(Cl)ccc2[nH]1 93801,Cc1cc(F)cc(C(=O)NC2CCC(NC(=O)C(O)C3CCC3)CC2)c1C 93802,Cc1nn(C)c(C)c1NC(=O)CN1CC=CCC1 93803,CC(C)(O)CCNC(=O)NCC(C1CCN(C2CCC2)C1)c1ccccc1 93804,N1(C(CNC(CC)=O)=O)CC2(CCC2)CC1C(N1CC2CC(CO)C(C2)C1)=O 93805,N1(C(C=C(C)C(C)(C)C)=O)CC2CC1C2C(=O)N(C1CCCC(O)C1)C 93806,C1(C)(CNC(C=NOC)=O)CN(C(C2(OC)CC2)=O)C(C)(C)C1 93807,C1(CC(N2CC(C)(NCC)C2)=O)CN(C(=O)C(C)(CC2CCC2)OC)CC12CC2 93808,N1(C(C2(OC)CS(=O)(=O)C2)=O)CC(NC(C2CCCC2C(C)C)=O)CCC1C 93809,C12CC3CCC(C1)N3C(=O)Cn1cc(nn1)C(O)C1(CCCC1)N2.C=CCC1CC1 93810,C#Cc1ccc(NC(C2(C)CCN2C(c2ccc(OC(F)F)cc2)=O)=O)cn1 93811,C(C(C)(C)C(=O)NCC(CCO)c1cncn1C)N(C(C)=O)C 93812,S(=O)(=O)(c1ccccc1C(F)(F)F)N1CCC(NC(C2(F)CCCC=C2F)=O)C1 93813,C1(NC(c2c(C)cc(F)s2)=O)CC2CCC(C1C)N2C(c1ccc(CF)cc1)=O 93814,C1(CC(=O)NC(C2CCN(C(=O)CCOC3CC3)C2)C)COCCN1CC1CC1 93815,C1(NC(c2n(CC(C)C)ncc2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C(C)C1 93816,c1(C(=O)NCC2(C)CCC(NC(c3cccc(C)n3)=O)C2)cc(F)c(F)cc1F 93817,C12(C(=O)OC)CCCC1(C(=O)NCCNCC1CC1CO)CC2 93818,CC1(C)CCC(O)(CNC(C2CN(C(C3(n4cncn4)CC3)=O)C2)=O)C1 93819,c1(C(=O)NCC(CC(C)C)NC(=O)C(C#N)=CC2CC2)cccc([N+](=O)[O-])c1 93820,C1(NC(C)=O)CCCC(NCCn2nnnc2C)C1 93821,c1(C(N(C)CC2(NC(C34CCCC3C4(F)F)=O)CC2)=O)c[nH]c2ccc(Cl)cc12 93822,CC1CCCN(CCNC(c2csc(-c3cccc(Cl)c3)n2)=O)C1CO 93823,c1(NC2CC(C)N(C(=O)CCCCF)C2)nc2c(cc1C#N)CCC2 93824,c1(C(N(CCC(C)NC(c2cnc(OC)s2)=O)C)=O)cccc2c1CCO2 93825,c1(C(=O)NC)c(C)o[nH]c1=NC(=O)c1nn(C)cc1NC(=O)NCc1ccncc1.O 93826,c1(C(=O)NCC2C(C)CN(C(=O)Cc3cccc(Cl)c3)C2)ccnc2[nH]cnc12 93827,N1(C(COCCCCC)=O)CC(CCNC(=O)Cc2ccco2)C(C)C1 93828,C1(C(=O)NCC2CCC2)(NC(CC2CCN(C)C2)=O)CCCCC1 93829,N1(C(c2cn(CCC3CC3)nn2)=O)CCCN(C(C2CC23CC(O)C3)=O)C(CO)C1 93830,C1(NC(Cc2onc(C)n2)=O)CCN(C(C2(N3CCCC3)CC2)=O)CC1F 93831,c1(C(N2CC(F)(CNC(=O)CC3CCC(=O)N3)C2)=O)cccc2c1CCCC2=O 93832,c1(C(C)NC(C2(F)CN(C(C(C)SC)=O)C2)=O)cncc(F)c1 93833,C(=O)(C1=COCCC1)N(C(C(=O)NCCC(C)O)C1CC1)C 93834,C1(C(N2CC(C)C(NC(=O)C(c3ccc(Cl)cc3)(C)O)C2)=O)CN2CCC1CC2 93835,c1(CC)nc(=N)[nH]c(=NC2CC2NC(=O)CCCCCCBr)[nH]1 93836,CC1(C)CCOC1C(N1CCC(N(CCO)C(c2coc(Cl)n2)=O)C1)=O 93837,C(=O)(C(CO)C(C)(C)C)N(C)CC1CCN(C(=O)CC(O)C2CC2)C1 93838,c1(C(N2C(CNC(C(C)(O)C3CC3)=O)CCCC2)=O)cnc(Cl)cc1Cl 93839,C1(NC(c2nc(C(C)OC)oc2)=O)CCC(NC(C2CC2F)=O)CC1 93840,c1(C(=O)NC2CC2NC(C2CC(=O)N(C3CCCC3)C2)=O)csc2c1CCCC2 93841,c1(N2CC3CC(O)CC3C2)nc2c(c(=NCCOC(F)(F)F)[nH]1)CCC2 93842,N1(C(C(C)SC)=O)CCC(N=c2nc(C(C)(C)C)[nH]s2)C2(CCC2)C1 93843,CC#CCC(C(=O)NCCC(C)CC)NC(=O)C=C(C)C(=O)N(C)C 93844,N1(C(CNS(CC)(=O)=O)=O)CCCC(CCNC(C2CCCO2)=O)CC1 93845,c1(C(=O)Nc2ccc(C#C)cc2)ccc2cccc(Br)c2n1 93846,c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cc2ncccc2C)C(C#N)C1)=O 93847,CN1C=NC2=CNC(=NC3CC(CN(C(=O)C4CC4)C4(CCCCC4)C3)CCC2)C1=O 93848,N12CC3CN(CC3C1)NC2=O.C1(N2CCC(CCc3cn[nH]c3)C2)CCCCC1.[SH4] 93849,C(=O)(CCCCCCCc1ccccc1)N1C(C(=O)NCc2c(C)n[nH]c2)CC1 93850,N1(C(c2c(C#C)cn(C)n2)=O)CCCC2(C1)C(NC(c1ccsc1)=O)CCN2C 93851,C1(CC)CCCN(C(=O)CCc2cn(C)nn2)C1C(=O)NC1CN(C)NC1=O 93852,CC1CCCC=C1c1cnc2[nH]cc(C(=O)Nc3csc(Br)c3)c2c1 93853,CC(C)(C(=O)NCC1CC(F)(F)CN1C(c1ccoc1Br)=O)C(F)F 93854,CCC1=C(C(=O)NCC2CN(C(=O)C(C)C3CCOC3)CCO2)CCCO1 93855,Cc1cc(SCC(=O)NCC(C)(CO)NC(C2CC(C)CCO2)=O)cc(C)c1 93856,c1(C(=O)OC)cc(OC)cc(OC)c1CN1CC(CC#N)C2(CC2)C1 93857,CCC(CC(=O)NCC=CCNC(=O)C(C1CCC(=O)CC1)F)C(C)C 93858,c1(C(N2C(CNC(c3c(C)[nH]c(C(F)(F)F)c3)=O)CC2)=O)cc(S(N)(=O)=O)co1 93859,C(=O)(C(C)CCCN(C)C)N1CC(C)C(n2cc(S(=O)(=O)C3CC3)nn2)C1 93860,c1(CC(=O)NCC(CNC(C(CC)(C)C(N)=O)=O)OC)c(C)cc(C#N)cc1C 93861,n1(CC)nc(C)c(C(=O)NC(CNC(c2sc(C)cc2Cl)=O)CC)c1C(F)F 93862,c1(OC)cc[n+]([O-])c(C(=O)NCCC(C(C)C)NC(C2CC2C)=O)c1 93863,c1(C(=O)NCCCCNC(=O)CO)ccc(C(C)C)cc1.c1(SC)cscc1C1CC1 93864,C1(C(=O)NC2(C(N3C(C(C)C)COCC3)=O)CC2(C)C)Cc2ccccc2C1 93865,[N-]=[N+]=NC1CC(C(=O)NCC2CC2)N(C(=O)C#CC2CCC2)C1 93866,N1(C(C(C)N(CCC)C(c2csc(Cl)c2)=O)=O)CC(=O)N(C)CC1C 93867,CC1CN(S(=O)(=O)c2ccc(NC(C)CCO)cc2Br)Cc2ccc(Br)cc2O1 93868,c1(C(=O)NC(C(C)C)Cc2ccc(F)cc2)ccc(N2CCCC2=O)c(Cl)c1 93869,Cc1ccc(OCCC(=O)N(C)CCN(C)C(c2cc(N)ccc2O)=O)c(C)c1 93870,CC1(C(=O)NCC2OCCC2NC(C2CC(OC3CC3)C2)=O)CC(C#N)C1 93871,Cc1cccc(Br)c1C(C(=O)N(C)Cc1ccco1)NC(=O)CCc1nccs1 93872,C=CC(CC)CC(=O)NC12CC(C1)N(C(=O)C(C1CC1)OC)C2 93873,C=CCCCCCC(C)(c1nnnn1CCOC)NC(C)CCCC(C)C 93874,C(C)(C)(CN=c1[nH]cnc(NCC(C)(C)OC2C=C2)c1C)SC.CCO 93875,C1(C(N2CC(C)C(NC(c3cncc(Cl)c3)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 93876,C12(C(=O)NC(C)(CNC(C34COCC3C4)=O)C3CC3)CC(C)(C1)OC21CCC1 93877,CCC1=NOC(C(=O)NC(CNC(c2cnn(CC)c2CC)=O)CC)C1 93878,C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2c[nH]nc2C1 93879,Cc1cc(C(F)F)oc1C(N1CC(NC(C2CCC(F)(F)C2)=O)C(O)C1)=O 93880,CN1CCN(C(C2(O)COC2)=O)C(CNC(=O)CC2CCC(=O)N2)C1 93881,C1(C(=O)NC(C)(C)C)CN(C(C)=O)CCN1C.C12CCCN1C(=O)NC(CC)C2 93882,Cc1csc(C(=O)NCC2CCCCN2C(c2ccc(C(F)F)o2)=O)c1Cl 93883,C1(C(N(CCCNC(C=CC=CCC)=O)C)=O)CCOC(C)C1 93884,c1(OC)ccc(C(C)(C)C(=O)N(O)Cc2c[nH]nn2)cc1Cn1nnc(=N)[nH]1 93885,C1(C(=O)NC(=O)C2CC2)CC2(CC2)CN1CC1(C)CC(C)(C)C1 93886,C1(C(=O)NC(C#C)CC(C)(C)C)CC(N=[N+]=[N-])CN1C(c1ccc(O)nc1)=O 93887,C1(CC=C)(NC(=O)CCC2CC2(F)F)CCN(C(C2CC3CCC3C2)=O)CC1 93888,c1(C(=O)NCCCCCN(C(C2CCCN(CC)C2)=O)C)cc(OC)nc(Cl)c1 93889,N1(C(C2CC(C(F)F)C2)=O)CCC(Cn2cc(C3COCC3O)nn2)C(F)(F)C1 93890,CCCC(CC)C(=O)NC1(CCC)CCCN(C(c2cc(CC)no2)=O)C1 93891,N1(C(c2cc(C)n(C)c2)=O)CCCC2(CC(NC(=O)CCc3nccs3)C2)C1 93892,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 93893,C1(C(=O)NC(C)(C)CNC(c2ccccc2)=O)CC1CCS(C)(=O)=O 93894,C(=O)(CC(C(F)F)C(C)(C)C)NC(CNC(c1ncc(C)cc1C)=O)(C)C 93895,c1(CC)ccccc1-c1cn(C(C)C)nn1.C1(C(=O)N)CC2CC2C1 93896,C1(NC(c2cnc(C)nc2O)=O)CC2CC(C1)N(C(=O)CN(C1CCCC1)C)C2 93897,n12cccc(c1=O)NC(=O)c1cccc-2c1.CC(CC(N)=O)N(C)C 93898,c1(C(N2CC3CC2CCC3NC(C2(C(F)F)CCC2)=O)=O)cccn2ccnc12 93899,N1(C(C(=O)NCCNC(C)=O)=O)CCC(C2CC2)(CNC(=O)CC(F)(F)F)C1 93900,C1(CCNC(c2[nH]cc(C(C)=O)c2)=O)CN(C(c2sccc2CC#N)=O)CC1C 93901,O(P(C)(=O)CNC(C1OCCC1CNC(c1c[nH]c(=O)cn1)=O)=O)CC 93902,c1(CNC(c2c(C)cnn2C)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 93903,N1(C(CCSCCCC)=O)CC2CC2(NC(c2oncc2C)=O)C1 93904,C1(C(=O)Nc2cncnc2I)CCN(C(=O)CC2CCCC2)CC1O 93905,N1(CCC(N2CCCC(CC(=O)N(CC(F)F)C3CC3)C2)=O)CCCCCC1 93906,c1(OCC)nc(N(C2CN(C(c3ccc(C)cc3)=O)C2)C)ncc1OC 93907,C1(OC)CCC(F)(C(=O)OC(C23CC4CC2C3C4)C)C1 93908,c1(C(=O)NC2(c3ccccc3)CN(C(c3cnn(C4CC4)c3)=O)C2)n[nH]c(O)n1 93909,c1(C(=O)NC2CC3(C(NC(CN4C(C)CCC4)=O)C3)C2)ccnc2[nH]c(O)nc12 93910,n1(CC(=O)NC2CCCCC2CO)[nH]cc2c(=O)ncnc1-2.C12(CCC1)CC(=O)N2 93911,C1(C(=O)NCC(CNC(CC(C)OC)=O)O)CC(=O)N(c2nccs2)C1 93912,CCCCC(CC)C(=O)NCCNC(c1sccc1C(C)(C)C)=O 93913,Cc1cc(C(N2CCNC(C(=O)NC3CC(O)C3)C2)=O)cc(C#N)c1 93914,c1(C(=O)NCCC2(O)CN(C(CSCC)=O)C2)sc2cncn2c1C 93915,c1(-c2cn(CC3CCN(CC(C)(C)C(=O)O)C3)nn2)ccc(F)c2[nH]ncc12 93916,N1(C(C(CCF)NC(c2cc(C)ns2)=O)=O)CCCC(C)(O)C1 93917,C1(CNC(CCC2N(C(C(C)NC(N)=O)=O)CCC2)=O)CCCC12CC2 93918,c1(CN(C)C)cccc(F)c1-c1cnc(NC(=O)CCC2CCCC2)nc1 93919,c1(C(=O)NC(c2cccc(N)c2)C)cnc2n1CCOCC2 93920,C(=O)(C(C)(C)CC(F)(F)F)NCC(CNC(c1c(OC)c(F)ccc1)=O)C 93921,CCC(C)(O)C(=O)NC1C=CCN(C(c2cn(C)nc2C)=O)C1 93922,c1(N(C(CCOCCCN(C(CCCOC)=O)C2CC2)=O)C)ccc(O)cc1 93923,CCC(CC)C(F)C(=O)NCCN(CCOCCSC)C(C1CCCC(F)C1)=O 93924,C1(C(N2CC(OCCC(=O)N(C)CC3CCC3)C2)=O)COCCN1C 93925,C12(C(=O)NCCN(C(CCc3nc(C)sc3)=O)C)CC(C)(CO1)C2 93926,C(CN=c1c(C)c[nH]c2ccccc12)NC(CN1C(c2ccc(C)cc2)CCC1)=O 93927,Cc1cc2ncc(CNCC(C)NC(=O)CN3CCCC3C)cc2[nH]1 93928,N1(C(CCC=C)=O)CCC(CO)(NC(c2csc(-c3ncccn3)n2)=O)C1 93929,C1(CCNC(=O)C(O)CN2CCCC2)CCN(C(=O)CNc2ccccn2)CC1 93930,N1(C(CNC(CCC)=O)=O)CCC(C(=O)NC2CC(O)(CCO)C2)(CC)C1 93931,c1(CNC(c2ccc(CC)cc2I)=O)cnc2c(c1)c(C)nn2C 93932,C(=O)(C(C1CN(C(=O)OC(C)(C)C)C1)SCCOCCF)NCCSC(C)=O 93933,C1(CNC(c2cc(C)cc(Cl)c2)=O)CC2COCC2N1c1nccc(CO)n1 93934,c1(CNCCCN(C(=O)NCC)C)cccn1Cc1ccccc1 93935,c1(C(=O)NCC(CC=C)NC(=O)C(C)CO)cccc(CN2CCN(C)CC2)c1 93936,C1(NC(COC)=O)COC2(C1)CN(C(=O)CCc1cnc(C3CCC3)o1)C2 93937,N1(C(C2(C)CCC2)=O)CCCC1CCCNC(=O)Cc1nnc(O)s1 93938,c1(C(=O)NC(C)CNC(=O)Cn2cccn2)nn(C)cc1N.c1(CC)nncn1C 93939,c1(OCC)ncc(C(N2CC(N(C(c3cccnc3)=O)Cc3cnn(C)c3)C2)=O)s1 93940,c1(CNC2C(C(=O)Nc3c(C)n(C(C)C)nc3)CCC2)ccc(F)cc1[N+](=O)[O-] 93941,c1(NC(CC(C)NC(C2CCC3CC3CC2)=O)C)c([N+](=O)[O-])cnn1C 93942,c1(CN2C3(CC3)C2=O)ccc(F)c(F)c1.c1(CCCC)ncc(C(F)(F)F)[nH]1 93943,n1(CCOC)nnnc1C(CNCCc1cccs1)NCCOC(C)(C)C 93944,C1(CNC(C(COC)C)=O)CN(C(=O)C(F)=CCCF)CCCO1 93945,c1(NC(c2cccc[n+]2[O-])=O)cccn2ncc(C(=O)NC3C(OC)CC3)c12 93946,c1(OC)cc(CC(=O)NCC2(C(C)NC(=O)CC(C)(F)F)CC2)cc(F)c1 93947,c1(C2(NC(=O)NCC(CCCC(C)O)O)CCC2)ccc2c(c1)OCCO2 93948,c1(C(=O)NCCN(C(=O)C(c2ccc(F)cc2)C)CC)ccc(F)c2c1OCC2 93949,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 93950,C1(NC(C2N(C(C3N(C(=O)OC(C)(C)C)CC3)=O)CC2)=O)CCc2nc(O)[nH]c2C1 93951,Cc1c(C(=O)NCC23CC(CNC(=O)C(C)(C)CN(C)C)(CO2)C3)cccc1N 93952,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 93953,c1(C(CC2N(Cc3c(C)nc(C)[nH]3)CCCC2)=O)ncc(Br)c(C)n1 93954,CC1(CCS(=O)(=O)NC2C=CCC2)OCCO1 93955,N1(C(C)C(=O)Nc2cc(O)nc(O)c2)CC2C3CCC(C2C1)N(C(C1CCC1)=O)C3 93956,c1(C(CNC(CN(CC)CC)=O)OCCNC(=O)COC)cc(F)ccc1Br 93957,N(C1CCCn2cnnc21)C(=O)CC1CCCN(C(c2c[nH]nc2Cl)=O)CC1 93958,C1(CNC(C(C)OC)=O)(NC(C2(C)CCNC2=O)=O)CC2CCC1CC2 93959,C1(CCC(=O)N(C2C3CCC2CC3)CC)CCCC2CC12.C12CCCN(C1)C2=O 93960,C1(C(=O)NC2C(N(C(Cc3c(C)cco3)=O)C)CCCC2)CN2CCN1C(C)C2 93961,C1(CN(C)C(C2CCNC2=O)=O)CN(C(=O)COCc2cccnc2)CCO1 93962,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 93963,c1(NC2CC3CC(OC)CC3C2)cc2cc(Br)ccc2s1 93964,c1(-n2cc(C(CCC)N(C(=O)CC(C)C)CC)nn2)ccc(F)c(F)c1 93965,c1(NCC(=O)NCC(=C)CCNC(c2occc2Cl)=O)ccccc1CC 93966,C1(C(NOC(C(C)C)CC)=O)(CNC(C2CSCC(=O)N2)=O)CC(C)(C)C1 93967,Nc1ccc(C(N2CC3(CCCC(CNC(=O)C4CC4)O3)C2)=O)c2c1CCCC2 93968,C(=O)(C(C)(C)C(=O)N1CCOC(C2CC2)C1)OCCc1c(OC)cccc1 93969,c1(C(C)NC(=O)C(Cc2ncccn2)NC(=O)OC(C)(C)C)ncc(Cl)n1C 93970,c1(COC)ccc(C(=O)NC2CN(C(=O)CCCNC(=O)OC)CC2O)cn1 93971,c1(C(=O)NC(CC)(CNC(=O)C(F)(F)COC)CC)ccc2cccnc2n1 93972,c1(OC)nc(C(=O)NC2CN(C(c3snnc3C3CC3)=O)C2)ncc1F 93973,C(C)(C)(C(C)CC(=O)N1CC(OCCO)C1)N(C(C1CCC(C(N)=O)C1)=O)C 93974,CCCC1=NOC(C(=O)N(C2(C(=O)N(CC(O)CO)C)CC2)C)C1 93975,CC(=O)CCC(=O)NCC1CC(NC(C2CC2(F)F)=O)C1 93976,C1(N(C(=O)CNC(N)=O)C)CN(C(c2cc(C3CCCC3)cn2C)=O)C2CC12 93977,c1(C(=O)NCC(CC)NC(COCCC)=O)cc2n(n1)CC(C)(C)CO2 93978,C(C(C(=O)NOCCF)NC(c1ccc[n+]([O-])c1)=O)SCC 93979,c1(C(=O)NC2C(NC(C(C)=C3CC3)=O)CC(F)(F)C2)cnc2c(F)cccc2c1 93980,N1(C(CC(CCC)(C)O)=O)CC2(C1)CN(C(c1cc(CC)cs1)=O)CC2CO 93981,C(=O)(CCCCCCNC(=O)CC1CCC(C)O1)NCc1scc(CSCC)n1 93982,c1(CC)ccc(C2CCCC2)cc1.c1cn(CC(=O)NCCC2CCC2)nn1 93983,Cc1cc(F)ccc1COC.CC(CO)OC(CCONC)=O.C1C(C2CC2)C(=O)N1 93984,c1(C(N2CCC(CC3CC3)C2)C(=O)NCCSC)cccc(C(F)(F)F)n1 93985,C1(C)(C(=O)NCC2(CNC(CCC(C)C)=O)CC2)CC2CCC1C2 93986,c1(C(=O)OC)cc(NCCC2=CCCCC2)cc(Cl)c1C 93987,c1(C(N2CCCC(C3N(C(CC=C)=O)CCC3)C2)=O)ccc(CC)cc1Cl 93988,CCCCC(O)CC(=O)NC(CCSC)C(N1CCC2(CCCO2)C1)=O 93989,c1(C(N2CC(NC(CCC#C)=O)C(C)C2)=O)ccc(OCC=C)cc1Cl 93990,c1(C(=O)NC23CCN(C(c4ccn(CC)n4)=O)CC2C3)ccc2occ(C)c2c1 93991,N1(C(CSCCOC)=O)CCCC2C1CCN2c1ncc(Br)c(C)n1 93992,C(=O)(C1=CCSC1)NC(C1CCCN1C(C1CCCCN1C)=O)C 93993,C1(C(=O)NC(C)Cn2cc(CC3CCNC3=O)nn2)C2Cc3cc(Cl)ccc3C12 93994,c1(NCCCN(C(c2cccc(C)n2)=O)C)ncccc1S(=O)(=O)NCC(C)C 93995,N1(C(C(=O)N(C)CCN2CC(C)OC(C)C2)=O)CCCC(C)(c2ccc(O)cc2)C1 93996,C1(NC(CCOCC(C)C)=O)CCCC(NC(=O)CCc2nc(N(C)C)no2)C1 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94278,n1(CC)ccnc1C=CC(=O)N(CCCCCCNC(C1(F)CCC1)=O)C 94279,c1(OC)nc(C)ccc1C(=O)NC(CNC(=O)CC1C(=O)NN=C1C)CO 94280,N1(C(C(CC)OC)=O)CCC(C)C(CNC(C23CCC(CC2F)C3)=O)C1.c1(C)ccccc1 94281,N(C1c2ccc(Br)cc2CC1(C)C)C(=O)Nc1cc(OCC)cc(F)c1 94282,c1(C(=O)NCC(CNC(C(C=C)(C)O)=O)CO)cc(OC)cnc1F 94283,C(=O)(C1=CCCCC1C)NCC(CC)(CC)NC(=O)C(C)OCCC(C)C 94284,CCC(C)(COC)C(=O)NCCCOCCNC(c1ccnc(N(C)C)n1)=O 94285,CC1CCN(C(c2ocnc2C2CC2)=O)CC1CNC(C1(C)CCCS1)=O 94286,c1(C(=O)OC)oc(C(=O)N(CC(O)CNC(=O)Cc2ccco2)C(C)C)cc1C 94287,C1(C(=O)NCC(CC)OC)CCN(C(C)Cn2cc(C)cn2)C1 94288,C(=O)(C(CC(=C)C)NC(=O)CCCCSC)NC(CC#C)C(=O)O 94289,O=C(O)CC(Cc1cn(CC2CCOC2)nn1)NC(=O)CC1CCC(O)C1 94290,C1(C(N2CC(c3ccc(F)nc3)C2)=O)(NC(CC=O)=O)CCOCC1 94291,C1(O)(CC(=O)N(C)CCOCCNC(C2CC2c2ccn(C)n2)=O)CCCCC1 94292,C12(C(=O)NCC3CCCN(CC)C3)CCCC1CCN2C(=O)C(O)CCC(C)C 94293,C(=O)(C1=NOC2(CCC2)C1)NC1CCCC(C(=O)NCC2(C#C)CCCC2)CC1 94294,c1(OC)cccc(N(C(C2CCC(N)C2)=O)C(C2(C)COC(=O)C2)=O)c1 94295,C1(CCNC(=O)C2=NOCC2)CCC2CN(C(=O)C3=C(Cl)CCC3)CC12 94296,N1(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)CC(C2CCOCC2)C1 94297,C#Cc1cc(C(N2CC(C)(C)C(NC(=O)C#CC3CC3)C2)=O)ccc1C 94298,C1(NC(CSC)=O)CCCC(NC2CN(C(C3(OC(C)C)CC3)=O)C2)C1 94299,CCC(CC(=O)N(CCNC(c1cc(Br)ncc1OC)=O)CC)C(C)(C)C 94300,CCC(COC)(CC)C(=O)N1CC(=O)CC1C(=O)N(C)CCc1nccs1 94301,C(=O)(CCC1=CCCCC1)NCC1(CO)CCN(C(C2(C)C(C)CCC2)=O)CC1 94302,C1(C2(O)CCOCC2)(C(N2C(C(C)(C)NC(=O)Cc3ccoc3)CCC2)=O)CC1 94303,CC1CC(C(=O)NCCCS(C)=O)CC(=O)N1.c12nocc1C(=O)NOC2 94304,N1(C(C(C(C)C)C2CCC2)=O)CCC2(CCOCC2)C(NC(=O)CN=S(C)(C)=O)C1 94305,CN1N=C(CC(=O)N2CCCC(n3cc(CNS(N)(=O)=O)nn3)CC2)CC1=O 94306,C(=O)(C1CCc2ccc(Cl)nc21)N(CCN(C(CC1(OC)CCC1)=O)C)C 94307,N1(C(CNC(C)=O)=O)CC(NC(=O)C2=NNC(=O)CC2)C2(CCCC2)C1 94308,C1(NC(CCC(C)OC)=O)(CNC(C2CC(OC)C2)=O)CCC(F)(F)CC1 94309,C1(CC=C)(NC(=O)C(C)(C)Oc2ccccn2)CN(C(C2CCC2=C)=O)C1 94310,c1(CC(C)C)ncc(C(N2CCC(NC(C3CC=CC3)=O)C(O)C2)=O)c(O)n1 94311,Cc1cc(=NCC(CO)CC(C)C)[nH]c(NCCN=S(C)(C)=O)n1 94312,C12(C(=O)NCC(=C)CCNC(c3nn(C)cc3C)=O)CCC(C)(CO1)C2 94313,N1(C(C(COC)(C)O)=O)CCC(NC(c2cccc(COC(F)(F)F)c2)=O)C(C)C1 94314,c1(CNC2CCCC(C(=O)OCC)C2)c[nH]c2ccncc12 94315,C1(C(=O)Nc2ccc(F)nc2F)CCC2(CN(C(c3csc(Br)c3)=O)C2)O1 94316,C(CC(C(=O)N(c1ccc(OC)cc1)C)OC(=O)CCC(=O)C1CC1)SC 94317,C1(C(N2CC(C(C(=O)NC(C3CC3C(=O)OC)C)OC)C2)=O)(CC)CCCO1 94318,C1(CNC(c2cc(C(C)C)[nH]n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1C 94319,c1(OCC(=O)NC2CC(NC(CC(C)OC)=O)C2(C)C)cc(Br)ccc1F 94320,C1(C(C)(C)O)(NC(c2cc[nH]c2)=O)CCN(Cc2cccc(Br)c2F)CC1 94321,C(=O)(C1=CC2(CCOC2)C1)NCCC1CCCN(C(C(n2ncc(C)c2)C)=O)C1 94322,N1(C(C2(C(N)=O)CC2)=O)CCC(CNC(C2C3CC4C(C3)C24)=O)CC1 94323,N1(CCC)CC(C(=O)NC(C)(CNC(c2occ3c2CC3)=O)C(C)C)CC1=O 94324,Cc1cc([N+](=O)[O-])c2ccccc2c1N(CC(C)(C)CO)CC(C)O 94325,CC1CN(Cc2ccc3c(c2)CC3)CCN1C(c1c(Br)nnn1C)=O 94326,C1(C(=O)NCCc2cncc(C)n2)CCC(C)(C)CN1C(=O)COCC(F)F 94327,CN1CCC(O)C(NC(c2occc2CNC(C2(C)CCCC2O)=O)=O)C1 94328,C1(C(N2CC(NC(c3cnc(S)[nH]3)=O)C3(C2)CC3)=O)Cc2n[nH]cc2C(=O)N1 94329,N1(C(=O)C(O)c2cnc[nH]2)CC2CCCC(C1)N2C(=O)C(O)C1CCCC1 94330,C1(C)(C(=O)OC)C=CCN1C(=O)C(F)C1CC(NC(C2CC(O)C(F)C2)=O)C1 94331,CC1CCN(C(=O)OC(C)(C)C)CCN1C(=O)Cn1cc(C(C)(C)CO)nn1 94332,N1(CC(=O)NC2CC(C(C)NC(=O)CCc3ccccc3)C2)CCCOC1=O 94333,C1(F)(CNC(c2csc(C(F)F)c2)=O)CCCN(C(=O)CCOC2CC2)C1 94334,c1(CCC)ccc(CN(C2COCCC2CO)CC)cc1C 94335,C(c1ccc(O)c(O)c1)=CC(=O)NCC(C)NC(c1c(C#C)cnn1C)=O 94336,C1(NC(C(CCCC)C)=O)CCCCCN(C(=O)CCc2cnccn2)C1 94337,C1(CNC(C(C)C2CCCO2)=O)CC2(CCN(C(c3cc[nH]c3)=O)CC2)C1 94338,C12(C(=O)NC3(CCNC(c4c(C)nccc4)=O)CCOCC3)CC1COC21CCC1 94339,c1(OC)c(Cl)cc(C(=O)NCC(C)(C2CC2)NC(=O)C=C(C)C(F)F)nc1Cl 94340,N1(C(c2c(CC)cccc2F)=O)CCN(C(=O)C(F)=C(C)C)CC12CCC2 94341,c1(C(C)C)cccc(C(=O)NC(C)(CNC(=O)CSc2ccccc2)CO)c1N 94342,C(C(C)(C)C(=O)N1CCCC(C(C(=O)NC(C)CSC)OC(C)=O)C1)SC 94343,C1(CCN(C)C(c2ncccc2F)=O)CCN(C(c2ccnn2CC2CC2)=O)CC1 94344,c1(NC)ccc2[nH]nc(I)c2c1.c12c(cccc1F)c1ncsc1c(=O)[nH]2 94345,N1(C(c2cc(C)[nH]c2)=O)CCCC1(C)C(N1CCC1CCO)=O 94346,C1(NC(c2cnc(OCC)nc2)=O)CC2CC1N(C(c1cccc(=S)n1O)=O)C2 94347,C1(CN(C2(C)CNC2)C)CN(C(=O)OC(C)(C)C)CC1CN(C)C 94348,c1(C(N2CC(F)(CNC(C3C(C=C)C3)=O)C2)=O)oc(C2CCC2)nc1C 94349,c1(OC)ncc(C(N2CCCCC2CNC(=O)C(O)c2ccco2)=O)cc1F 94350,c1(C(N(CC(CN(CCC(=O)NCCOC)C)O)C)=O)cc(C(F)F)ncc1F 94351,c1(CC(=O)NC2CCN(C(=O)CCCc3cccs3)C2)ccc(O)nc1 94352,c1(CNc2cc(N3CCN(CC=C)CC3)ncn2)sc2ccccc2c1C 94353,c1(C(N(C2CC(NC(C3C(C)CCC3)=O)C2)C)=O)ccnc2c1ccn2C 94354,c1(CC)c(C)nc2ncnn2c1N1CCC(CCNC(=O)C=C(C)C(C)C)C1 94355,N1(C(C(C)SCC)=O)CCN(C(c2nc3ncccn3n2)=O)CCC1C 94356,c1(COC)nc(C(=O)NC(C)CCCNC(CC2C(C(=O)OC)(CF)C2)=O)cs1 94357,Cn1cc(C(O)C(=O)NC(C(=O)NC2(c3ccncc3)CC2)C2CCC2)cn1 94358,C(=O)(C(O)C(F)(F)F)N(C)CCOCCN(C)C(C1CCC1C(C)(C)C)=O 94359,N1(C2CCN(CC=C)C2=O)CCN(C(c2cn(C)nn2)=O)CC1C 94360,c1(C(=O)NC2C(NC(c3onc(CC)c3C)=O)CCC2)ccc(Br)nc1N 94361,C1(CCOC)(NC(c2nn(C)nc2Br)=O)CCN(C(=O)CCS(N)(=O)=O)CC1 94362,N1(c2ncc(OC)cn2)C2CCC(C2)C1C(=O)Nc1ccc(F)c(I)c1 94363,CCCC(O)CC(=O)N(C)CC1(O)CCN(C(=O)C(C)=C(C)C)C1 94364,c1(-c2cn(C(CC)SC)nn2)ccccc1F 94365,C1(C(N(CCCNC(=O)CC(C)c2ccncc2)CC)=O)CCC(=O)N1C 94366,c1(C(=O)NCC(C23CCC(CC2)C3)NC(=O)CC(F)F)nccc2nn[nH]c12 94367,C(=O)(CS(C)(=O)=O)NC1CCN(CCNC(C(C)NC(=O)NC)=O)C1 94368,N1(C(C(F)=CCC)=O)CCC(C2CC2)C1C(N1CC(C)C(C)C1C)=O 94369,N(C1CCCc2c[nH]nc21)C(N1CCC(Cc2ccc(C)c(Cl)c2)C1)=O 94370,c1(OC)c(Cl)ccc(C(=O)NC2CN(S(=O)(=O)c3cn(C)cn3)CC2F)c1F 94371,N1(C(CC(CC)C)=O)CC2(CCCC2NC(c2cc(F)c(F)cc2N)=O)C1 94372,CC1CC2(CCN(C(C3(C(F)(F)F)CC3)=O)CC2)CN1C(C1CC12CCCC2)=O 94373,c1(-n2c(C3CCC(F)C3)nc(C(n3cncn3)CO)n2)cccc2c1CCCC2 94374,C1(C(=O)NC2CC(CF)C2)CN(C(=O)COc2cccc(O)c2)C2CC12 94375,Cc1ncc(CC(N2CC(NC(=O)OC(C)(C)C)C2)=O)o1.C=O 94376,N1(C(Cc2cnc(C)nc2O)=O)CCOC2(CCN(C(=O)C=CCF)CC2)C1 94377,CC(C(=O)NC1CCC12CN(C(c1ccc(-n3cccn3)nc1)=O)C2)S(C)(=O)=O 94378,N1(C(C(CCCC=C)NC(C2C=CC2C(=O)OC)=O)=O)CCC(C2=NOCC2)C1 94379,N1(C(c2ccc(C(N)=O)o2)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)C2C1 94380,C(=O)(CS(=O)(=O)CCC)NC1CCN(C(c2ccc(CC)nc2C)=O)C1C(C)C 94381,c1(C(=O)NCCCN(C(c2c(SC)cnn2C)=O)C)c(Cl)ccnc1C 94382,C1(NC(=O)C(C2(O)CCCC2)F)CCCN(C(=O)CC2CCCC(C3CC3)O2)C1 94383,c1(CC2C(C(N(CC(C)(C)NC(C3CC4CC4C3)=O)C)=O)C2)ccc(Cl)cc1 94384,c1(C(N(CC(O)CN(C)C(C2OCC2(C)C)=O)C)=O)cnncc1O 94385,CC1(C)OC(C)(C)C1C(=O)NC1(CN2CCN(C(=O)C(O)P(C)(C)=O)CC2)CC1 94386,C1(C#N)(C(=O)NCC(CC)N(C(=O)C=CC(=O)OC(C)(C)C)C2CC2)CCC1 94387,Cc1ccc(C(N2CCC(C(C)NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)cn1 94388,CCCCC(CNCc1cccc(F)c1)NCc1cc(CO)on1 94389,N1(C(c2c(CC)nc[nH]2)=O)CC(C)(C)CC1CNC(=O)Cc1c[nH]ccc1=O 94390,c1(C(=O)NC(CC(C)C)CNC(=O)Cc2nnc(S)n2C)cc2sccc2[nH]1 94391,c12cncc(c1)C(=O)NC(C)CCCOC2=O.C1(Cl)(C(=O)NCC)CC1 94392,c1(C(=O)NC(CNC(CNC(C(CC)C)=O)=O)(C)C2CC2)cc(S(N)(=O)=O)co1 94393,c1(C(=O)NCC2(OCC)CCC2)c(NC(c2nc(C)ccc2F)=O)cccc1F 94394,N1(C(C(CC)C)=O)CC(OC(=N)O)C(CCn2cc(CNC(N)=O)nn2)C1 94395,c1(CCN(C(C2CCC(=O)N2)=O)SC)ncccn1.n12cc(nn1)SCC2 94396,c1(CCC(=O)N(CC(C)NC(C(C2CC2)OCC)=O)C)ccncc1 94397,Cc1csc(=O)n1CC(=O)NCC1COC(CNC(C2C3COCC23)=O)C1 94398,Cc1cc(C(N2CCCC2CN(C)C(C2CC(F)C2)=O)=O)c2scnc2c1C 94399,c1(CN2CC(C)(CC(N3CCN4CCC3CC4)=O)C2)ccc(S(C)(=O)=O)cc1F 94400,c1(C(=O)NCCC(=O)NC(c2ccsc2)CC)cocc1C 94401,C1(C(=O)NC2CC(O)(C(N3CCC(CC(=O)OC)CC3)=O)C2)CC2(CCC2)CO1 94402,N1(C(c2cc(OC)c(C(F)(F)F)cc2Br)=O)CCCN(C(=O)C(C)C)C(CO)C1 94403,C(CC(=O)N1CC(NC(N)=O)C1)(C(F)(F)F)NC(c1c(CC)ocn1)=O 94404,C1(NC(COCCC#C)=O)CCN(C(C2(CC=C)CCCC2)=O)CC1CC 94405,c1(C(=O)NC2CC(NCc3ncccc3O)C2)cc(O)c(O)c(Cl)c1 94406,C1(CNC(CC)=O)CN(C(C2CCN(CC)C2)=O)CCCO1 94407,c1(C(=O)NCCCNC(CNC(CN(C)CC)=O)=O)c[nH]nc1S(N)(=O)=O 94408,C1(C(=O)NC2C(NC(c3c(CCC)nns3)=O)COCC2)CCCCC(=O)N1 94409,CC(C)(CCNC(=O)Cc1csc(C2CC2)n1)NC(=O)C(C)(O)c1ccccc1 94410,N1(C(C2(C(N(C)C)=O)CC2)=O)CCC2(CCCC2Nc2ncc(Cl)c(O)n2)CC1 94411,Cc1cc(O)c(Cl)cc1C(=O)NCc1ccccc1CN(C)C 94412,CC1CC2CN(C(=O)CC(C)(C)N(C)C(C3COCC3(C)C)=O)CCN2C1 94413,N1(C(C2N(C(c3c(NC)cnnc3)=O)CCCCC2)=O)CCc2c[nH]nc2C1 94414,N1(C(C(C)=C(C)C)=O)CCCC(N(C(=O)Cn2cc(Br)c(C)n2)C)C1 94415,C1(N(C(CN(C(=O)Cn2c(C)csc2=O)CC)=O)C)CCCCCC1 94416,O=C(CCCC1(NC(C2C(c3ccccc3)C2(F)F)=O)CCC1)OC 94417,N1(C(C(CC)OC)=O)CCC2(CC1)COCC(CNC(c1ncc[nH]c1=O)=O)O2 94418,N1(C(c2cc(CC)[nH]n2)=O)CC2CC2(NC(=O)CCOC2CCCOC2)C1 94419,C1(C(N(CC(=O)OC)C)=O)COCCN(C(=O)CC=C(Cl)Cl)C1 94420,C1(C(=O)NC(c2c(F)cccc2F)C)CN(C(=O)C(=O)C2CCCC2)CCC1O 94421,Cc1ccc(NC(C2CCC(CNC(=O)C(N3CCSCC3)C)O2)=O)cc1 94422,N1(C(C2OCCC(C)(C)C2)=O)CC(NC(c2cn(CCO)nn2)=O)C2(CCC2)C1 94423,C1(NC(=O)Nc2nn(C3CC3)ccc2=O)COc2ccc3ccccc3c2C1 94424,CC1CN(CC2=COCCO2)CCN1CCO.C1C(C)N1 94425,n1(CC)ncc(C(N2CC(C(C(=O)NC3CC4CC4C3)OC)C2)=O)n1 94426,C1(c2cn(CC(C)O)nn2)CCCN(C(=O)CS(=O)(=O)NCC(=O)O)CC1 94427,C(N=c1[nH]c2cc(F)c(F)cc2s1)C1CCCN(C(C2C(C)CCC2)=O)C1 94428,CN1CCCC(F)(C(=O)NCC(C2CCCC2)NC(c2cscc2Cl)=O)C1 94429,C(CCCCC(=O)NCCc1csc(C)n1)N(C(CNC(=O)OCC)=O)C 94430,C1(C(=O)NCC2(C(=O)NC(C)COCC)CC(=C)C2)CCS(=O)CC1 94431,C1(C(N(C)CC2(NCc3c(C)cccc3)CC2)=O)CC12CCOCC2 94432,N1(c2cc(NCc3cc(C#N)cs3)nc(C)n2)CCC2(CCOC2=O)C1 94433,S(=O)(=O)(c1ccc(NCc2ccco2)c(F)c1)N1CCC(C(C)O)CC1 94434,c1(SCC(=O)NCC(CNC(Cc2n(C)cnn2)=O)(C)O)cc(F)ccc1F 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94629,c1(C(=O)NC(C(=O)NC(CN2CCCC2)CO)C2(O)CCC2)sccc1Cl 94630,C1(CNC(C(C=CC)O)=O)CCN(C(c2csnc2C2CC2)=O)CC1O 94631,Cc1coc(C(N2CCC(C(C)NC(=O)CC3CC(=O)C3)C2)=O)c1C 94632,n1(Cc2c(C(C)C)cccc2Br)c(-c2cn(C)nn2)csc1=Nc1ccc(O)cc1 94633,C(c1cncnc1O)=CC(=O)NC1CCC1NC(=O)C(F)(F)CC1CC1 94634,C(CCCCCO)c1cn(C2CC(NC(C3C(C)C3C3CC3)=O)C2)nn1 94635,N1(C(c2cc(C)sc2C)=O)CCCC(NC(=O)C=Cc2cccnc2)C1C 94636,C1(N(C(=O)C(C2CCCCC2)O)C)C2CN(C(=O)CC(F)F)CC12 94637,O=C(C1CCCc2n[nH]cc21)NCC(C1CCC1)Nc1nc(Cl)nc2sccc12 94638,c1(C(N(C)CC2CCN(C(CC3(OC)CCC3)=O)C2)=O)cc(C)ccc1C 94639,c1(N(CC#C)C)nc2cc(Br)ccc2c(=NCC2(CO)CCCCO2)[nH]1 94640,c1(C2(C(=O)NC3C(NC(=O)CO)CCC3)CCC2)ccc(Br)cc1 94641,c1(C(C2CC2)NC(CCN(C)C(=O)N(C)C)=O)nn(C)cc1Cl 94642,C1(CNC(c2c(OC)csc2)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1C 94643,C(=O)(C1OCCn2ccnc21)NCCN(C(c1cc(OC)c(O)cc1F)=O)CC 94644,N1(C(CCN(CC)CC)=O)CCCC(CC(=O)NC2CC2O)CC1 94645,Cn1ncc(C(=O)NC(C2CCN(C(C3CCC3(C)C)=O)CC2)(C)C)c1Cl 94646,N1(C(c2c(CC)cc(C)cc2)=O)CC(C2CN(C(C3CC3(C)CC)=O)C2)C1 94647,N1(C(CCc2nc(C)c(C)o2)=O)CC(CO)C2(C1)CN(C(C1CC(F)(F)C1)=O)C2 94648,c1(C(N2CCC(NC(c3cc(OC)no3)=O)CC2C)=O)ccc(C#N)c(OC)c1 94649,c1(C(N(CCNC(=O)C(C)(CC)OC)CC)=O)ccc([N+](=O)[O-])cc1Br 94650,Cc1ccc(C2CCN(C(C3CCSCC3)C(=O)NC3CC3)C2)cc1 94651,C(=O)(C(=O)CCCC(C)C)N1CC(CCNC(c2ncc(C)nc2)=O)C1 94652,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3c[nH]nc3C)C2)nc1Br 94653,C1(C(N2CC(F)(CNC(c3[nH]n(C)c(=O)n3)=O)C2)=O)CCCC12NC(=O)NC2=O 94654,N1(C(C2CCC(CC)C2)=O)CC2(CCN(C(=O)COc3cc(C)on3)C2)C1 94655,C1(C(N2CC3C(C(=O)NC4CCN(S(C)(=O)=O)CC4)C3C2)=O)CCCCC1(F)F 94656,C1(NC(C(C)NC(=O)CC(F)(F)F)=O)C2CC1CN(C(=O)CN1CCCC1)C2 94657,C1(C(=O)NCC2CCN(C(C34CCCCC3C4)=O)C23CC3)Cc2nccnc2C1 94658,N1(C(c2ccn3cnnc3c2)=O)CCCC(C2CN(C(=O)CSC(F)(F)F)C2)C1 94659,C(N=c1ccnc(N2CCC(NC(=O)N(C)C)CC2)[nH]1)C1N(C)CC(O)C1 94660,N1(C(C(C(C)OC)NC(c2c[nH]c(=S)cn2)=O)=O)CC2(C1)CC2(F)F 94661,C1(C(=O)NCC2(F)CCC(NC(CCC#CC)=O)C2)CN2CCN1CC2C 94662,C(c1cnn(C)c1)=CC(=O)NC1(CNC(C(CC)O)=O)CCOC1 94663,c1(CNC(C2(CNC(C3(C)CCC3)=O)CCC2)=O)cccc(CS(N)(=O)=O)c1 94664,C(=O)(C1CCc2snnc21)NCCN(CCC)C(C1OCCOC1(C)C)=O 94665,C1(CN(C(c2nscc2Br)C(=O)NCC(F)F)C)CC2CCC1O2 94666,C=CCN=C(NCc1ccsc1)NCC1C(C)(C)C1(F)F 94667,C1(NC(COCCC)=O)CCSC12CN(C(=O)C(C(C)C)n1cncn1)C2 94668,C(=O)(CC1=CCCCC1)NC1CN(C(C2CC3(CC(C)C3)C2)=O)CC12CC2 94669,C1(NC(C2(SC)CN(C(C3CC34CC4)=O)C2)=O)CC2(CCCO2)C1 94670,c1(C(=O)NCCC2N(C(CSCCC)=O)CCOC2)c(C)nc(O)nc1C 94671,C=CCC(C)C(=O)NC1COCCC1C(=O)NCC(F)C1CCC1 94672,Cc1ccc(OC2(C(=O)NC34CC3CN(C(c3ccc(C)nc3)=O)C4)CC2)cc1 94673,C1(C)(CNC(C2(C(=O)NC)CCC2)=O)CC(NC(=O)CCc2ccon2)C1 94674,CC1(C)CCC(NC(=O)CCNC(=O)C=CC2(C)COC2)C(CNC2CC2)C1 94675,N1(C(c2ccccn2)=O)CC2(C1)CN(C(C1CC(OCC)C1)=O)CCO2.OCC 94676,Nc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)C(F)C2CCOC2)c1 94677,C1(NC(CCCC(=O)OC(C)(C)C)=O)COC2(CCN(S(=O)(=O)CCCCl)C2)C1 94678,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NC1(CC(N)=O)CC1 94679,CN=C(NCC(c1ccc(OC)c(Br)c1)O)NC1CCCn2nccc21 94680,c1(C(=O)NCC2(C(N)=O)CN(C(c3nccnc3Cl)=O)C2)cnc2[nH]nnc2c1 94681,C1(C(N2C(CCNC(=O)CC(=O)N(C)C)CC(OC)C2)=O)CC2(C1)CC21CC1 94682,CC1(C)CCN(CC(=O)NC2C=CCC(C(=O)NCC3(C)CCCC3O)C2)C1 94683,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 94684,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 94685,c1(C(=O)NCCCOCCCNC(C2CN(C)C2)=O)c[nH]c2ccncc12 94686,Cc1cc(NCC2CCN2C(=O)CC(C)c2cnn(C)c2)c(Br)cc1[N+](=O)[O-] 94687,Nc1cc(C(N2CC(O)CC2CNC(=O)C(F)n2cccn2)=O)c(F)c(F)c1 94688,c1(C(=O)NC2C(CC)N(C(=O)Cc3conc3C)CCC2)ccc(CO)cc1F 94689,N1(C(c2c(CC)cc(F)cc2)=O)CC2CCN(C(c3cc(Cl)cnc3C)=O)C2C1 94690,c1(C(=O)NCc2nc(C(=O)NCC3CC3)co2)cnc(O)c(F)c1 94691,C(=O)(C(F)C(CC)CC)N1C(C(=O)NCC(C)N(CC)CC)C(CC)C1 94692,Cc1cnc(C(=O)NCCNC(=O)C=CC2C(C)C2(Cl)Cl)cc1Br 94693,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 94694,C1(NC(CSCC#C)=O)C2CC3CN(C(=O)CC(n4nc(C)cc4C)C)C1C3C2 94695,c1(C(=O)NCC2(CNC(c3cnc(C(F)F)cn3)=O)CCC2)c(F)cccc1F 94696,c1(C(N(C)CCOCCCNC(C2CC23CCOC3)=O)=O)cn2cccnc2n1 94697,c1(C(C(=O)NCCOCC)N(CC(Cl)Cl)CC)ccc(C(F)F)c(F)c1 94698,CCCC(C(O)C(=O)N1CC(N(C)CC)C1)NC(=O)Cn1cnc(=N)[nH]1 94699,CC(C)(CNC(=O)CC1CCC(O)C1)CO 94700,C(=O)(CC1COCc2ccccc21)NC(C1CN(C(C2CCC(C)CC2)=O)C1)C 94701,CC1CCC(CC(=O)NCCC2(CNC(=O)CCc3cncs3)CC2)OC1 94702,CC1C(c2ccccc2)NCCN1Cc1cc(-c2cccc(F)n2)on1 94703,C12(C(N3C4C(OC5(COC)CC5)CC(C4)C3)=O)CCC(CC(=O)OC)(CC1)CC2 94704,n1(C(C)(C)C)c(O)nc2cc(C(=O)NCC3CCC3NC(C3CC3Cl)=O)ccc12 94705,N1(C(C2(NC(C(CC)O)=O)CCCCC2)=O)CCN(CCO)C(C)C1 94706,C12(C(=O)OC)CCCCC1N(C(=O)Cc1csc(N3CCCC3)n1)CC2 94707,N1(CC(=O)NCC(CNC(CCOC(=O)CO)=O)C)CCCCC1C 94708,CC1OCCCC1C(=O)NC1CCC(NC(c2csc(Cl)c2Cl)=O)C1 94709,C1(C(C)NC(=O)C(F)C2CCC2)CN(C(c2cc[nH]c(=N)n2)=O)CCO1 94710,C(=O)(C(O)C(F)(F)F)N1CC(CC=C)(NC(=O)C(c2ccccc2)OC)C1 94711,c1(OC)ccc2c(ccn2CC(=O)N(CC(C)NC(=O)CCC(C)O)C)c1 94712,c1(C(=O)NCC2N(C(C3CCOC3)=O)CCN(C)C2)nnc(O)c(Br)c1O 94713,C1(NC(CSC)=O)CC2(C1)CC(CNC(c1cc(Cc3ccccc3)on1)=O)C2 94714,CC1CC(C(N2CC(NC(C3(C)CC3(F)Cl)=O)C2)=O)CCS1 94715,N1(C(CN(C(C)C)C)=O)CCC2CN(C(c3ccc(O)nn3)=O)CC2C1 94716,C(=O)(C(=O)N=S(C)(C)=O)N1CC2(CC(NC(c3c(C)sc(Cl)n3)=O)C2)C1 94717,C1(CC)CCN(C(=O)C(O)CC2CC2)C(C(=O)NCC(C)(C)C2CC2)C1 94718,c1(CC(=O)N(C2CN(C(c3n[nH]cc3C(F)(F)F)=O)C2)C)c[nH]c2ccccc12 94719,C1(CC(=O)NCCN2CCCC2)CCCC1NC1CCN(C(C23CC(CO2)C3)=O)C1 94720,C1(NC(C2(NC(C3CNC(=O)N3)=O)CC(F)C2)=O)CC2CC(O)C1C2 94721,C1(COC)(NC(=O)CC2CC3C=CC2CC3)CCCN(C(=O)CCC(C)(C)F)C1 94722,N1(C(CCc2n(CC)ccn2)=O)CC(N(C(=O)C(C)C(C)(F)F)C)C(C)(C)C1 94723,CC(C)CCC(C(=O)N(CC(C)CO)C)NC(=O)CCc1cnco1 94724,C(CC(N)=O)(C(=O)NC(c1ccccc1O)C)NC(C(F)OC)=O 94725,CC1(C)Cc2ccc(S(=O)(=O)NC(C(=O)O)C(F)(F)CC3CC3)cc2C1=O 94726,C1(OC)CN(C(c2conc2C(C)C)=O)CC1NC(C12CC1CNC2=O)=O 94727,c1(NC(C2CC(C(N)=O)C2)=O)cccc(CNC(=O)Cc2cnsc2)n1 94728,c1(C(=O)NCCC2CC(NC(C3N(CC)CCC3)=O)C2)cccc2sccc12 94729,C(C)(CCC(=O)NC1C(C(=O)NC2(CCOC)CC2)CCC1)SC 94730,c1(C(=O)NCC2(C)CC(NC(c3cnn(CC)c3Cl)=O)C2)sc2cncn2c1C 94731,c1(-c2ccc(C)cc2)cn2cnc(C(=O)Nc3nc(C)ccc3C#N)c2s1 94732,C1C(C(NOC)=O)CCCN1 94733,C1(CC(N2CC3CC2(C)C3)C(=O)NC(C)(C)C)CCOC2(CCC2)C1 94734,c1(COC)cccnc1C(=O)NCCC1CCCN(C(c2cc(C)co2)=O)C1 94735,N#Cc1[nH]c(=NCCCNCC2CCC(n3ccnn3)CC2)sc1Cl 94736,c1(C(=O)NCCNC(c2cc(C(C)(F)F)n[nH]2)=O)cccc2c1CCC2 94737,C1(NC(C(CC)N(C)C)=O)CC2CCC(C1)N2C(c1cnc(-c2ccoc2)s1)=O 94738,N1(C(C(C)OCOC)=O)CC2(CC(C(=O)NCC3CC=CC3)CO2)C1 94739,C1(CC(=O)NC(C)CCOC(C)C)(OC)CN(C(C2CCC2)=O)C1 94740,C1(C(=O)NC2(CF)CCN(C(C(CC)CO)=O)C2)CCn2c(O)nnc2C1 94741,N1(C(C2(OC)CCSC2)=O)CC2C(CNC(C3CN(C(C)C)CCO3)=O)C2C1 94742,CCCCCCC(C)C(=O)NC1CCCCN(C(=O)COCCOCC)C1 94743,C=C=CCCC(=O)N1CC(O)(CN(C)C(c2sccc2SC)=O)C1 94744,N1(C(c2ccc(C(N)=O)cc2)=O)CCCC2(CCN(C(=O)CNS(N)(=O)=O)C2)C1 94745,c1(NC(=O)NC(c2cccc(C)c2)C)cccc2c1CC(=O)N2 94746,C1(NC(C2(SC)CC2)=O)CN(C(=O)CC(C)F)CCC1F 94747,c1(OCC)cc(C)nc(N2CCOC(c3cc(C)cc(C)c3)C2)n1 94748,C(=O)(C1CCc2ccccc21)N1CCN(C(c2c(C)nn(CCO)c2C)=O)CC1 94749,C12(NC(C3(C=C)CCC3)=O)CCC(NC(c3c(C)coc3C(C)C)=O)(CC1)C2 94750,N1(C(C(C(=O)OC)F)=O)CC2(CCN(C(=O)COc3ccc(F)cc3O)C2)C1 94751,c1(C(N2CCC(O)(Cc3cn(C(CC)C)nn3)CC2)=O)cnc2[nH]c(C)nc2c1 94752,N1(C(C(CCC)O)=O)CCC2(CCN(C(c3cc4c(C)nn(C)c4s3)=O)CC2)C1 94753,C#CCC(O)C(=O)N(C)CC1CCCN(C(=O)C(F)(F)CC2CC2)C1 94754,c1(C(N(CCCCNC(C2CC2(C)C)=O)C)=O)ccc(OCC(F)(F)F)nc1 94755,C1(C(=O)NC2(CC=C)CN(C(c3ccc(=O)oc3)=O)C2)CCN(C)C1=O 94756,C(=O)(C(O)CC(F)(F)F)NC1CCC(C(=O)NCc2ccc(C)cc2F)C1 94757,CC(CF)CC(=O)NC1(COC)CCN(C(C2CCN(C(=O)OC(C)(C)C)C2)=O)C1 94758,C1(CNC(=O)CCF)CN(C(c2ccc3[nH]ccc3c2)=O)CC12CCC2 94759,C(CC(C)C(=O)N1CCC(OC(F)F)C1)=CC.C(C(C)(C)C)N1C(=O)C1 94760,N1(C(C(c2cnn(C)c2)C)=O)CC(C(N)=O)OC(C)(C)C1 94761,C(=O)(CCCNC(c1coc(CC2CC2)n1)=O)NCC(C)OCC#C 94762,C1(C(=O)NCCOCCCO)CCC2CN(C(=O)COc3ccsn3)CC12 94763,C1(NC(c2ccsc2-c2ccccc2)=O)CC(O)CN(C(=O)C2=C(Cl)CC2)C1 94764,C1(CCNC(CN(CC)CC)=O)CCC(NC(c2ccc(C)o2)=O)C1 94765,C(=O)(C1CCc2c[nH]nc21)N(C1CN(C(CC(CC)OC)=O)C1)C 94766,c1(OCC)ccc(F)c(C(=O)NC(C2CCN(C(=O)CC3CC3(Cl)Cl)C2)C)c1F 94767,Cc1ccc(C(=O)NC2CCC(CNC(=O)CCC(=O)N(C)C(C)C)C2)nc1C 94768,c1(CC(=O)NC2CCCC(NC(=O)NN3CC4CCC3C4)C2)c(F)cccc1F 94769,CC1(C)CC(CNC(c2ccc(O)c(F)c2F)=O)CN(C(C2C3CCC23)=O)C1 94770,c1(C(N2CCC(O)(CN(C(=O)C(=O)NCC3CC3)C)C2)=O)ccn2nccc2c1 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94842,Cn1nc(C(=O)NCC2(NC(c3cc[nH]n3)=O)CCC2)cc1C(F)F 94843,C(=O)(C1=C(C#N)CCC1)N1CC(COC)N(C(C2(S(C)(=O)=O)CCCC2)=O)CC1 94844,C1(C(=O)NC)(NC(c2ccc(C(=O)NCCC(=C)COC)s2)=O)CCC(C)(C)CC1 94845,CC1CN(C(=O)CCC(F)(F)F)CCC1C(=O)N(CCCO)C 94846,C(=O)(CC(O)C(C)(C)C)N(CCN(C(c1ccnc(OC)c1F)=O)C)C 94847,Cn1cnnc1CCC(=O)NCc1ocnc1Cc1cn(CCCSC)nn1 94848,CC1Oc2ccccc2N(CC(=O)N2CCN(Cc3ccc(N)cn3)CC2)C1=O 94849,N1(C(C2(CC)CCCN2C(=O)Cn2ccnc2)=O)CCC2CN(C)CC2C1 94850,C(CCC(C)(C)NC(=O)Cc1cnc(C2CC2)[nH]1)NC(C(C)OCCCC)=O 94851,CCC(CCC(=O)NCc1cccc(C#N)n1)NC(C1CCCN1N=O)=O 94852,c1(C(=O)NCC2C3CN(C(=O)CCC4CCCC4)CC23)cnc2[nH]cnc2c1 94853,Cc1cnc2n1CCC(C(N1CCN(C(=O)C#CC3CC3)C(CO)C1)=O)C2 94854,c1(CC)c(C(=O)NCC2CCCCN2C(=O)C(F)F)cnn1-c1cccc(C#N)c1 94855,C(CCCCC(=O)NC1(CC(=O)OC)CC1)N(C(C1CCCCC1F)=O)C 94856,c1(OC)coc(C(=O)NC2CCC2NC(c2cc(C#N)no2)=O)cc1=O 94857,c1(C(N2CC(CCNC(CC(C(C)C)C)=O)OCC2)=O)ccc2nnc(O)n2c1 94858,N1(C(c2ncn(CC)c2)=O)CC(NC(c2occc2C(C)C)=O)C(C(F)(F)F)C1 94859,C#CCCCCC(=O)N1CCC(C(C)C(=O)N(C(C)C(=O)OC)C)CC1 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94878,c1(C(N(C(CCNC(C=C(C)C(C)C)=O)C)C)=O)cc2ccc(O)cc2[nH]1 94879,C(CCCCCNC(=O)CC1CCNC1=O)NC(c1n(CC=C)ccc1)=O 94880,C1(c2cccc(O)c2)CCN1N1CC2CCC(O)CC2C1 94881,CC12CCC1CN(C(c1cn(CCNC(C3(C)CCC(=O)C3)=O)nn1)=O)C2 94882,C1(C(N(CC(C)N(C(CCC=CC)=O)C)C)=O)CCCC(OC)C1 94883,c1(C(N2CCC(O)(C(C)NC(=O)CN(C)S(N)(=O)=O)C2)=O)cc(Cl)cc(Cl)c1 94884,c1(C(=O)NCC(CC)NC(=O)Cn2ncc(Br)c2C)cnc(Cl)n1C 94885,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NC1CC(CNC(=O)Cn2cncn2)C1 94886,C(=O)(CC(F)(F)C(C)C)N1CC(N(C(C(C)N)=O)C)C1.C(c1c[nH]cn1)=CC 94887,N1(C(c2n(CC)nnc2)=O)CC2(CCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 94888,c1(OC)cc(O)c(CNC2CC2C(=O)Nc2ccc(Br)nc2F)c(Br)c1 94889,N1(C(C=C(CCC)C)=O)CCC(NC(c2cnn3cc[nH]c23)=O)C12CCCC2 94890,CCC(CNC(=O)C(=O)NCC(C)OC)OC 94891,c1(OC)cc(C(N2CCCC2CNC(=O)C(C)C(C)C)=O)cc(Br)c1 94892,Cc1nc(O)nc(C)c1C(=O)NC(C1CN(c2ncc(C#N)cc2F)C1)C 94893,O=C(N=c1[nH][nH]cc1I)C1CCCN1Cc1cc(Br)cc(Br)c1F 94894,c1(CNC(C(CC)C)c2nnnn2CC(F)F)ccc(F)c(F)c1C 94895,CC1(CCNC(C2(C)CN(C(=O)CC34CC(C3)C4)C2)=O)CCOCC1 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94913,C1(OC)CC(O)CN(C(=O)CCOC2CN(C(=O)CCNC(=O)CO)C2)C1 94914,N1(C(Cn2c(C)ccn2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC12CCC2 94915,CCCC(C)(O)C(=O)N1C2CCC(C2)C1C(=O)NCC(CC)C1CC1 94916,N1(C(C(CC)C)=O)CC2CC(C1)CN(C(c1c(C)cc(Br)cc1Cl)=O)C2 94917,C(=O)(C1=CCCCC1P(C)(C)=O)N1C(C(C)NC(CCOC)=O)CCC1 94918,N1(C(C2(C#C)CN(C(C3CC4OC3C3CC43)=O)C2)=O)CC2CC(C)C2C1 94919,C#Cc1ccc(C(=O)NC(C)(CNC(c2ccc(F)nc2F)=O)C(C)C)cc1 94920,c1(NCc2scc(C)c2)cc(N(C)Cc2ccc(N3CC=CC3)cc2)ncn1 94921,C1(C(=O)OCC(C(C)C)(C)C)Sc2ccccc2NC1=O 94922,C1(COC)(NC(C2CCCCS2(=O)=O)=O)CCCN(C(C2(CF)CC2)=O)C1 94923,CC1CCN(C(C2CN(C)CCN2C)=O)CCN1C(=O)CNC(=O)CN(C)C 94924,CCCCCC(O)C(=O)NC1CC(CC(=O)NCC2(C)CC(C)=NO2)C1 94925,CC1=C(C(=O)N(CCCCCNC(=O)Cn2cnc(C(N)=O)n2)C)CCC1 94926,c1(C(N2CC(CN(C(=O)C(O)C3CCCC3)C)C2)=O)ccsc1Cl 94927,c1(-c2cncc(CN(C(CC(C)C)=O)CC(=O)O)c2)ccc(CO)c(Br)c1 94928,N1(C(C2(C)CCN(S(=O)(=O)C3CC3)C2)=O)CCC2(CCNC(=O)O2)CC1 94929,O=C1CCCCC(C(N2CCCCC2CNC(C2CC3CC2CC3O)=O)=O)N1 94930,CCC(O)C(C)C(=O)N(CCNC(c1cc[nH]c1C(C)C)=O)C(C)C 94931,C1(C(=O)NC2(C#C)COC2)CC(F)(F)CN1C(c1cc(C)on1)=O 94932,C1(COC)(CNC(=O)CC=CCc2ccccc2)CCN(C(c2cnns2)=O)C1 94933,C12(C(N(C3CCCC3)CCCNC(c3nccnc3N)=O)=O)COCC1C2(F)F 94934,C12(Cc3ccccc3)CCC(CO)(CC1)OC2CN1C(=O)NCCC1.O=[N+]([O-])CCCl 94935,C1(C(=O)NCC(C2CCN(C(C3C(C(C)O)C3)=O)CC2)O)CC2(CCOC2)C1 94936,c1(NC(CN(CCNC(CC)=O)C)=O)cccnc1OC 94937,N1(C(C2CC(OC)C2)=O)CCC2CCC(NC(c3cc(F)ccc3F)=O)C1C2 94938,Cc1ccc(C#N)c(N2CCN(CC(=O)NCc3cccc(Cl)c3)CC(O)C2)n1 94939,N12CC(C(C)(C)C1)NC(Cc1ccccc1)C2=O.C1(C=O)(CF)CC1.CO 94940,C(=O)(CC(C)(C)C(C)(F)F)NC(CNC(C1(C)CCN(C)C1)=O)(C)C(C)C 94941,C(CCC(C(=O)NCC(C)C)N1CCCC(OC2CCOCC2)C1)OCC 94942,N1(C(C(C)(C)C#N)=O)Cc2ccccc2CC1CNC(=O)Cc1ccc(Cl)cc1 94943,CCCCCC(C)(C)CNC(=O)C(C1CCN(C(c2sc(F)cc2C)=O)C1)F 94944,c1(C(N2CCC(C(C)NC(=O)CC(=O)NC3CC3)C2)=O)cnc2sccc2c1 94945,N1(C(C2(CC#C)CC2)=O)CCc2sc(CNC(=O)C=CC3C(C)C3(Cl)Cl)nc2C1 94946,CCCCC(O)C(=O)N(C)CCOCCNc1cncc(N(C)C)n1 94947,CN1CCCC(O)(CNC(C2CC(=O)CN2Cc2ccccc2)=O)C1 94948,C(=O)(CC(C(C)(C)C)NC(=O)CC1=CCOCC1)NCc1c(C)noc1C 94949,c1(C(N2CC(N(C(CC(n3ccc(C)n3)C)=O)C)C2)=O)n[nH]c2c1CN(C)CC2 94950,c1(CC(=O)NCC(C2CCOC2)NC(CCC#C)=O)cccnc1OC 94951,n1(CC(CC)O)cc(C(=O)NCC#CCNC(C2CCCOC2)=O)nn1 94952,C1(NC(C2OCCN(CC)C2)=O)CC2CC1CC2C(=O)NC1CN(C)C1 94953,C1(C)(CC)CC(NC(C2CC(F)(CO)C2)=O)CN1C(c1cnc(C2CC2)s1)=O 94954,C1(CC=C)(Nn2cc(C)nn2)CCN(C(=O)Cn2nc(C)cc2C)C1.C1CC1 94955,N(S(=O)(=O)N1Cc2ccccc2C1)Cc1ccccc1.C12COCC1CNC2=O 94956,c1(C(=O)NCC(CNC(C(CN(CC)CC)F)=O)C)cnc2c(c1)NCC2 94957,N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)C=CS(C)(=O)=O)C(CF)C1 94958,S(=O)(=O)(c1cc(Br)c(OC(F)(F)F)cc1Br)NC(C(C)C)C(=O)O 94959,N#CC1CCC(C(=O)NCC(C2CC2)NC(C2CCS2(=O)=O)=O)CC1 94960,C1(N(C(=O)Cc2cc(C3CC3)on2)C)CCC2CN(C(=O)C#CC3CCOC3)CC12 94961,C1(C(c2cccc(Cl)n2)NC(c2n(CC)ncn2)C)CC12CCC(F)(F)CC2 94962,N1(C(CC)=O)C(C)C2CC1C2NC(=O)CCc1ccc(Cl)c(C)c1 94963,c1(NC(C2CCN(C(=O)C=C3CC3)CC2)C)ncnc(Cl)c1C 94964,c1(C(N2C(CNC(CCc3cc(C)sc3C)=O)COCC2)=O)ccc(C#N)n1C 94965,c1(CNC(C(C)N(C)C(C2CCC(=O)N2)=O)=O)cccc(COC(=O)C(C)(C)C)c1 94966,Cc1cccc(C(=O)NC2(C)CC(NC(=O)C(C3CC(F)(F)C3)O)C2)c1 94967,C1(CNC(c2cncn(C)c2=O)=O)CN(C(=O)Cc2cnn(C)c2)CC12CCC2 94968,N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(C2CCCN(C)C2)C1.C12(C=O)CC3CC1C2C3 94969,c1(C(=O)NCC(CN(C(C2(CC#C)CC2)=O)C2CC2)O)cn(C)cc1C(F)(F)F 94970,c1(NC(=O)C(C)C(C)(C)C)c(C)cccc1F.C12(CC=C)CCN(C1)CC(=O)N2 94971,N(C1CCC(NC(c2cc(CO)[nH]n2)=O)c2ccccc21)C(=O)Cc1cn[nH]c1 94972,N12CCN(CC1C)CC2=O.CCC(C)CC(=O)NCCNc1cnn(CC)c1 94973,c1(N(CCCNC(c2ncoc2C2CCC2)=O)CC)ncnc(Cl)c1C(C)=O 94974,N1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)CC2)C(=O)CC(C)(C)C1=O 94975,c12cc(sc1CC)C(=O)NC(C)c1ncc(s1)C2.C(=O)OC 94976,N1(C(CNC(=O)OCC)=O)CCOCC(C)(CNC(=O)C(C)C2CCCO2)C1 94977,C1(C(N2CC(OC)(CNC(C3(C4CCC4)CC3)=O)C2)=O)CC(c2ccccn2)=NO1 94978,C=CCC(C)(C)C(=O)NCC1(OC)CC1.c12cnc(s1)CNC2=O 94979,CCC(C(=O)NCC(C)NC(c1ccc2nccn2c1)=O)C(C)(F)F 94980,c1(CCC(N2CC(OCCC(=O)NC3C(OC)C(O)C3)C2)=O)cncnc1O 94981,c1(C(N(C2CCN(C(=O)CCCNC(N)=O)C2)C)=O)cncc(OCC(F)(F)F)c1 94982,C1(C(=O)Nc2cccc(C3(C)CC(=O)C3)c2)CC2CCCCN2C1=O 94983,C(C1=CCN(C(=O)C=Cc2cn(C)cn2)CC1)NC(CN(C)C(=O)C1CC1)=O 94984,c1(C(=O)OC)ccccc1-c1nc(Cn2cc(CCS(=O)(=O)N(C)C)nn2)n[nH]1 94985,C(=O)(C(F)(F)c1ccccn1)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 94986,CCCCCC(F)C(=O)N1CC(C(=O)NCCN2CCOCC2)C2(CCC2)C1 94987,Nc1ccccc1-c1cn(CCCC(=O)NCc2csc(O)n2)nn1 94988,c1(CC)cccc(C(=O)NCC(C)(O)CNC(=O)COc2ccc(O)cc2)c1 94989,C(CCSC)(C(=O)NC1CCN(CC(=O)NCCC#N)CC1)OC 94990,c1(OC)cc(N2CCCC(N(C(=O)NCC3CN(C(=O)N(C)C)C3)C)C2)ncn1 94991,O=S(=O)(c1ccc(N2CCC3(CCC3)C2)cc1Br)NCC1C2CCCCC12 94992,N1CCc2c(O)ncnc2C1.c12ncc(F)c(n1)N1CC3C(C1)N23.CN 94993,c1(C(C(=O)Nc2cnccc2Cl)N(CCN(CC)CC)C)ccc(F)c(OC)c1 94994,C1(NC(C(COC)NC(C(CCC)O)=O)=O)CNC(=O)C12CC2.c12cnn(C)c1C2 94995,C1(C(N(CCC)CCNC(=O)C(C2CCC2)OC)=O)CCCCO1 94996,C1(C(N(C)CC2CCCN2C(=O)Cc2cccc(O)c2)=O)OCCN(C)C1=O 94997,N1(CCOC2CCC(Oc3ccc(OC)cc3)CC2)CCC(F)(F)C(C)C1 94998,c1(N(CCCC)C(c2ccc(C(=O)O)o2)c2ccccc2)cc(C)cc(C)c1O 94999,CCC(CC(=O)N1CCC(C2CC2)(CNC(c2cnc(C)s2)=O)C1)C(F)F 95000,C=CCC(F)(F)C(=O)NCC(C1CCC1)NC(c1ccc(F)c(C(F)F)n1)=O 95001,C1(C(N2CC(C(N(C(C=C)C)C)=O)C(OC)C2)=O)OCCCC1(C)C 95002,N1(C(c2ccc(NC(CCC(C)C#N)=O)cc2)=O)CCN(C)C(=O)C1C 95003,c1(C(N(C)CCOCCNC(=O)CC2CCCC2O)=O)nn(C)c2c1COCC2 95004,C(=O)(C(O)CC(N)=O)NC(C(=O)NC(C)Cn1cncn1)CCC1CCC1 95005,Cc1cc(C)c(C(N2CCC(C)(NC(=O)CC3NC(=O)NC3=O)C2)=O)[nH]1 95006,Cc1nc(N2CCOCC2)ccc1N(N1CCCC1)C(=O)NC1CC(=C2CCC2)C1 95007,CC(CCN=c1nc(-c2cccs2)cc[nH]1)NC(=O)CC1CCN(C)C1 95008,N1(C(c2ccc(CN(CCC)C)o2)=O)CCCC2C1CCN2C(C1CC1C#N)=O 95009,Cc1cn2ccc(C(=O)NCC(C)(C(C)C)NC(c3cnnc(O)c3)=O)cc2n1 95010,C1(C(N2CC(CN(C(C3C(C)OC(=O)N3)=O)C)C2)=O)CCc2nncn2C1 95011,N1(C(C(C)OC)=O)CC2C(C(=O)NC3CC(C(C)(C)C)C3)C2C1 95012,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CC2(CCC2)CCC1C 95013,c1(C(N2C(CCNC(CC(C)OC)=O)CSCC2)=O)c(F)cc(OC)cc1F 95014,c1(C(N2CC(NC(C(COC(C)C)(C)C)=O)C(O)C2)=O)ncc(OC)cc1F 95015,c1cccc(CNC(c2cc(COC)on2)=O)n1.C123CC(CO1)(C2)CC3=O.CF 95016,C12(C(=O)NCc3cc(CC)on3)CC1CCN2C(c1ccc(Br)o1)=O 95017,C1(C(=O)NCCN(C(C(CC)=CC)=O)CCOCCO)CCCC2(CCC2)O1 95018,c1(OC)ccccc1SC(C)C(=O)NCc1cc(C(=O)NC(C)C(C)(C)O)co1 95019,c1(OC)ccc(-n2nnnc2SC(C2COC(=O)N2)CCO)cc1 95020,c1(C(=O)NCC(CNC(C(C=CC)O)=O)C(F)(F)F)cncc(P(C)(C)=O)c1 95021,c1(OC(=O)NCCC2CCC(CC)O2)ccc2c(c1)NC(=O)C2=O 95022,C#CCCCCCCC(=O)NCCNC(=O)CCn1cc([N+](=O)[O-])cn1 95023,Cc1nn(C)c(Cl)c1C(c1nnnn1CCC1(C)CC1)NCc1cccs1 95024,Cc1nn(C)c(C)c1CCC(=O)NCC1CC(F)(CNC(=O)CC2(O)CCC2)C1 95025,Cc1nn(C)c(C)c1OCC(=O)NC1CCC(CNC(C2(CO)CC2)=O)C1 95026,C(=O)(C(F)(F)C(F)(F)F)NC1C(NC(CSCCC(C)C)=O)CC1 95027,C(=O)(CC(O)CC(C)(C)C)NCC(C)CC(=O)NCC1(C#N)CCCCC1 95028,N1(C(c2cc(C)c(O)nn2)=O)CC(C(=O)Nc2cncc(C)c2C)CCC1(C)C 95029,C(=O)(CC(C)(C)C1CCC1)Nc1c(N(C(=O)Nc2cc(C)on2)C)cccc1 95030,C1(C(C)(C)NC(C(C)N(C(C=C(C)C)=O)C)=O)C(=O)NN=C1C 95031,CCC(C)C(CNC(C1CC=CCN1C(=O)C(F)CC1CCC1)=O)CO 95032,C1(NC(C(CC)Oc2ccccc2)=O)CCCC(CNC(=O)C(F)=CCCF)C1 95033,c1(C(=O)NC(CC)CN(C(=O)CC(O)CC)C)cnn2ccn(C)c12 95034,CCCC(C(=O)N1CC(CNC(c2[nH]cc3c2CCCC3)=O)CC1(C)C)C(C)C 95035,N1(C(CC2CC(OCC)C2)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)CCO2 95036,C1(CNC(c2ccc(C#C)o2)=O)CC(C)(C)CCC1NC(c1occ(C)c1C)=O 95037,C1(CNC(COc2cc(C)on2)=O)CN(c2nc(C)nc(C)c2C)CCC1(F)F 95038,CC1(CNC(C2CN3CCN2CC3)=O)CCN(C(C23COCC(C2)C3)=O)CC1 95039,c1(N2C(CNC(C3(CC#C)CCCO3)=O)CN(C)CC2)nc(CC)nc(C)c1Br 95040,Cc1cnc2nccc(C(=O)NCC(C)NC(=O)C(C(C)C)n3cccc3)c2c1 95041,N1(C(C)=O)CCc2c(C)nc(O)nc2C1.C1(=O)C(C)(C)C(=O)NC(CC)CN1 95042,c1(C(=O)NCC(CCOC)NC(c2ccc(C)c(F)c2)=O)ncc(Cl)cc1F 95043,C(=O)(C(C)CC(C)(F)F)N1CC(CNC(C(C(CC)C)O)=O)(OC)C1 95044,c1(C(=O)NCCC(C)NC(C(C2CCC2)OCC)=O)c(C)ccc(Cl)c1O 95045,N1(C(c2csc(-c3ccccc3)n2)C(=O)NCCOCC)CC(C)C(C)C1 95046,N1(C(CCSc2n(C)nnn2)=O)CCN(C(=O)CCNC(=O)CO)CC12CCC2 95047,C1(C(N2CC(C)(CCC(N3CC(OC(C)C)C3)=O)C2)=O)CCCCNC1=O 95048,N#Cc1cccc(-c2ccc(Sc3ccccn3)cc2)c1Br 95049,CC1CCC(O)(C(=O)NCC2CC(C(=O)NCCN3CCCCC3=O)=NO2)CC1 95050,C(CC)(C(=O)N1CC(CC(F)C(=O)N2CCCC2C(C)(C)COC)C1)OCC 95051,c1(C(N2C(C(C)NC(c3n(CC)ncn3)=O)CCC2)=O)n[nH]c2c1CC(C)CC2 95052,C1(CNC(C2CCCN(C)C2)=O)CN(C(=O)COCCF)CCC12CCC2 95053,C1(CCCNC(CC2(OC)CCCC2)=O)CCCCN1C(c1ccccc1O)=O 95054,c1(C(N2CCN(C(C)C(N)=O)CC2)C(=O)NC)c[nH]c2c(Br)cccc12 95055,c1(OC)cnc(C=O)c(F)c1.C1(=O)C(C)(C)C(=O)N2CCC3C(C23)N1.OC 95056,C1(C(N2C(C(=O)N(C3CC3)CC3CCCOC3)CCC2)=O)C2(CC2)C12CC2 95057,C1(NC(c2cc(NC(c3c(C)cc(Br)cc3)C)ncn2)=O)CC2CCCCN2C1 95058,C(=O)(CC(C)(C)C1CC1)NC(CNC(C(NC(=O)OC(C)(C)C)SC1CC1)=O)=O 95059,Cc1nc(O)ccc1C(N1CCC(CCNC(=O)CC2(C(F)F)CC2)C1)=O 95060,C1(C(=O)NCC(C)(C2CC2)NC(C2(C(=O)OC(C)(C)C)CC2)=O)CC(CC)CCO1 95061,C(c1ccccc1F)=CC(N1CCC(C(C)NC(=O)CC2(C)CC2F)CC1)=O 95062,N=c1[nH]nc(CCCC(=O)NCCC(O)CNC(=O)CC2COCCO2)s1 95063,c1(C(=O)NCCCNC(C(C(CC)O)C)=O)ccc2sccc2c1 95064,N1(C(C(CC(=C)C)C)=O)CCC2C1CCCN2C(c1cc2c(Cl)cncc2o1)=O 95065,N1(C(c2c(CCC)occ2)=O)CC2(CCC(NC(=O)CC3C=CCC3)CC2)C1 95066,CCCCCC(=O)NC1CCN(C(=O)C(C)Cc2ccncc2)C1C(C)(C)C 95067,CN1CCC(C(=O)NC2(CNC(c3cnc(C(F)F)s3)=O)CCOC2)C1=O 95068,C1(C(=O)NC(C)CNC(c2cnc(S)n2C2CC2)=O)COC2(CO)CC1C2 95069,c1(CNC(C2N(C(C=CC(C)C)=O)CCC2)(C)C)ccc(NS(C)(=O)=O)cc1 95070,C(=O)(C(C)(C)C1=CCSCC1)N1C(CNC(c2cc(C)c(C)o2)=O)CN(C)CC1 95071,C(=O)(CC1OCCc2ccsc21)NC1CCN(C(C=CC)=O)CC1(C)C 95072,Cc1c(C(=O)NCCC2CCCN(C(=O)CC(O)CN(C)C)C2)ccn1C(C)C 95073,C1(OC)CC(NC(=O)C(=O)NC2CC(CN)C23CCC3)C12CCC2 95074,CCCC(CC(C)C)C(=O)N1CCC(CNC(=O)CCCn2cncn2)(OC)C1 95075,C1(NC(CN(C)C(=O)C2CC2)=O)CC2CCC1CC2NC(c1n[nH]c2c1COC2)=O 95076,C1(NC(C(C)NC(c2ccoc2)=O)=O)CC2CC1CN2C(c1ccc(O)cn1)=O 95077,C1(C(C)NC(N(C(C2CCCO2)C)C)=O)CCC(C(F)(F)F)CC1 95078,CC1CC(C(=O)NC2CC(CNC(C3(CN(C)C)CCCCC3)=O)C2)C1(C)C 95079,CC1=C2CC(Nc3cc(NC4CCCN(c5nccs5)C4)ncn3)CN=C2NN1 95080,C12(NC(C(CCCC)NC(N)=O)=O)CCC(CC1)N(C(=O)COc1cccnc1)C2 95081,C1(NC(COCCSC)=O)CCN(C(C2COC3(CCC3)CO2)=O)CC(C)(C)C1 95082,C1(C(N(C)CC2CCN(C(C(CC)F)=O)C2)=O)CCCN(C(C)=O)C1 95083,C1(C(N(C)Cc2nn(C)c(=O)o2)=O)CCN(C(=O)C(F)OC(F)(F)F)C1(C)C 95084,C1(C(N2CC3CC2CN3Cc2cncc(F)c2)=O)CCCC2CCCCC12 95085,C1(NC(C=CCN(CC)CC)=O)CC(O)CN(C(c2cnc(-n3ccnc3)s2)=O)C1 95086,C(CC(C)(C)C(=O)NCCC1(O)CCN(C(=O)CC(C)CN(C)C)C1)OC 95087,c1(CN(C)CC2CCCN2C(c2cncc(C3CC3)c2)=O)cc(C(=O)OC)ccn1 95088,C1(C)(C(=O)NC2CCN(C(c3cnc(OC)c(C)n3)=O)C2)CCCCCCC1 95089,C12(NC(c3ccc(C)cn3)=O)COCCC1CN(C(=O)CCc1ccn(C)c1)C2 95090,N1(C(C=C(C)CNC(=O)Cc2[nH]cnc2C)=O)CCCC(OCCO)C1 95091,Nc1ccc(C(=O)NCC2CCN2C(c2cccnc2O)=O)c(F)c1F 95092,C1(CNC(CSCCCC)=O)CC(F)CN1C(=O)COCC(C)C 95093,C(=O)(CCCC(C)(C)NC(c1ncn(C(C)C)n1)=O)Nc1cc(C)cc(F)c1 95094,N1(C(CCCC#C)=O)CC2CCOC2(CNC(=O)C(C)CC(N)=O)C1 95095,C(CCCCCN(C)C(C1CCCN1C1CCCC1)=O)NC(c1c(C)con1)=O 95096,c1(C(=O)NCCC(C)NC(c2coc(C(F)F)c2)=O)cn2ccnc2s1 95097,N1(C(c2c(C)sc(C(F)(F)F)n2)=O)CCOCC(CNC(c2ccco2)=O)C1 95098,N1(C(C(C=C)O)=O)CCCCC(C2CN(C(c3cnc4sc(C)nc4c3)=O)C2)C1 95099,C(C(CC(F)(F)F)NC(C1CCCOC1)=O)NC(=O)CCc1ncc[nH]1 95100,C(=O)(C#CC1(C)COC1)N1CCC(C(=O)NC2CCC(CC)CC2)(CF)C1.CC 95101,c1(C(=O)NCCC2(O)CN(C(C(C)NC(N)=O)=O)C2)cnc(O)c(C(F)(F)F)c1 95102,C(=O)(C1=CC(O)C(NC(=O)Cn2cccn2)C1)NC1CCN(C(C)C)C1 95103,C1(C(=O)NC(C(=O)N(C(C)C)C2CC2)CC2CCOCC2)CCCCC(=O)N1 95104,N1(C(C(C2CCCC2)OC)=O)CCOC(n2cc(C3CC3CO)nn2)C1 95105,c1(C(=O)NC2CC(CC(=O)NC3CCC3CSC)C2)ccnc2c1CCO2 95106,c1(C(=O)NC2CCCC(NC(c3c(C)scn3)=O)C2)cccc(C(F)F)c1Cl 95107,Cc1cc(C(N2CC(C(=O)NCC3CC4C=CC3C4)CC(F)C2)=O)ccc1I 95108,c1(C(=O)NCC(CNC(c2cc(C)nc(C)c2)=O)OC)cnn2ccn(C)c12 95109,C1(NC(=O)Cn2ccnn2)CCCC(C(N2Cc3c[nH]nc3C2)=O)CC1 95110,n1(CC(=O)NCCN(C(c2ncc[nH]2)=O)CC)cc(CC2CCCO2)nn1 95111,CCCS(=O)(=O)C(C)C(=O)NCCCCNC(=O)CC1CCCC(=O)N1 95112,CCC(CNC(c1ccc(Cl)o1)=O)(CC)C(=O)NC1CCCC12CC2 95113,c1(C(=O)NC(CN(C)C(C2CCC=CCC2)=O)(C)C)ncccc1C(F)F 95114,c1(NC(c2n(C(CC)(C)C)nnn2)C2CC2)cc(SC)cc(C)c1 95115,c1(C(=O)Nc2ccco2)cc(O)nn1C.C=CCC1CNC(=O)CNC(=O)N1 95116,c1(C(C(=O)NCC(=C)C)NC(=O)C(c2ccccc2)C)n[nH]c2ccccc12 95117,c1(-c2cc(C(c3n(C(CC)C)nnn3)NCC(=O)N(C)C)n[nH]2)ccc(Cl)cc1 95118,c1(OC)cccc(COCCC(N2CCC(CNC(=O)C(C)(O)CC)C2)=O)c1 95119,C1(C(N2CC(C)(NC(c3c(F)ccc(N)c3F)=O)C2)=O)CCOC2(CCCC2)C1 95120,Cc1cc(N)ccc1C(=O)NCC1CCC(NC(c2ccsc2C)=O)C1 95121,C1(C(=O)NC(CC#CC)CO)CC2(CCN1C(c1ccn3ccccc13)=O)CC2 95122,c1(C(C)OC)cccc(Cl)c1NC(N(CC(CC)(O)CC)C)=O 95123,C(=O)(C1CCCc2nn[nH]c21)NC1C(NC(=O)COc2cccnc2)CCCC1 95124,Cc1ccc(C)c(CNC(C2(C)CCCN2C(=O)CCC(C)C)=O)c1O 95125,N1(C(C(C)OCC)=O)CC(OC)CC1CNC(C1C=CCC1)=O 95126,C1(C(N(CCNC(=O)Cc2cncn2C)CC)=O)CCCCC1(C)C 95127,C=CCCCCCCNC(=O)C(C1CCCCN1C(=O)CCC(C)(F)F)NC(C)=O 95128,N1(C(C=CC)=O)CCCC(C)(C)C1CNC(c1cc(S(C)(=O)=O)co1)=O 95129,C(=O)(CC(C)C=C)NC(C(=O)NCC(=O)OCC#C)CC1CCCCC1 95130,CCCCC(C(=O)NCCN(C1CCCC1)C(c1ccc(Cl)cc1C)=O)C(C)C 95131,C1(CCCNC(C2N(CCC)CCC2)=O)CCN(C(=O)CC(C)N(C)C)CC1 95132,N1(C(c2cc(C)n(C)c2)=O)CCC(NC(=O)CCCC(=O)N(C)C)C(F)(F)CC1 95133,CC(C)(C)C(CO)C(=O)NCC(C1CCCC1)NC(=O)C(C)(C)n1cc(Cl)cn1 95134,c1(NC(c2c(C)cc(Cl)cc2)=O)cccc(NC(C23CC(CO)(C2)OC32CC2)=O)c1 95135,N1(C(C)=O)CCN(C(=O)CC2CCCN(C(c3cncc(F)c3)=O)C2)C(CO)C1 95136,N1(C(C(C)Cc2cnc[nH]2)=O)C2CCC1(CNC(=O)CC1CNC(=O)C1)CC2 95137,C1(C(=O)NCCCCC2CN(C(C3CC(=O)NCC3)=O)C2)CC(=O)CC(=O)N1 95138,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCN(C(Cc2cc(OC)c(F)cc2)=O)CC1 95139,c1(C(=O)NC23CCN(C(c4cccc(C)n4)=O)CC2C3)cnc2ccnn2c1C 95140,N1(N2C(C=O)CCC2)CC(NC(=O)CCCCCF)CC(O)C1.Cc1ccccc1C 95141,C1(C)(C(=O)NCC(CC)NC(=O)CC2CC2(C)C)CCCCNC1=O 95142,C1(COC)CCOCC1C12CCCN1C(=O)N2.c1(SC(C)C)n[nH]c(C)c1O 95143,Cc1noc(C)c1CN(C)C(C1CC(NC(c2cccc(CO)n2)=O)C1(C)C)=O 95144,N1(C(CCOCCN(C)C(C2CC3CCC3C2)=O)=O)CCOC2C(O)CC12 95145,C1(CCC#N)CN(C(=O)CCF)CC1NC(c1ccccc1-n1cccc1)=O 95146,c1(N(C(COC(C(CC2CC2)OC)=O)=O)CC(C)C)ccccc1C 95147,C1(C(N2C(C(=O)NC(c3cn(C)nn3)C)C=CC2)=O)C2CCC(F)C12 95148,c1(-c2cccc(C(=O)Nc3ncc(C(C)OC)cn3)c2)cc(C(C)=O)ccc1F 95149,C1(N(C2CCC2)C)CSC(C(F)(F)F)C1.CC(C)(C)OC(=O)O 95150,CCCC(O)CC(=O)N1CCN(CC(C)(C)NC(=O)CC2CCN(C)C2=O)CC1 95151,c1(CC(=O)NC2CC3(CC(NC(c4c(C)nn[nH]4)=O)C3)C2)ccc2ccncc2c1 95152,C(CCCC(=O)NC(C1CCCN1C(C1CSCCS1)=O)(C)C)SC 95153,Cc1cccc(C(F)C(=O)N2CCC2CNC(c2cc(CO)n(C)n2)=O)c1 95154,C1(NC(CC(CC)O)=O)CC(C(=O)N2CCC(CN=[N+]=[N-])C2)=CC1O 95155,C1(C(N2CC(C(C(=O)NCC3CCN(C(C)=O)C3)OC)C2)=O)CCCSC1C 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95173,CC1c2nccn2CCN1C(=O)CC1CC(NC(C2Cc3nccn3C2)=O)C1 95174,Cc1cc(C(=O)NC2CCCCC2N(C)C(c2c[nH]nc2F)=O)cn1C 95175,c1(C(=O)NC2CC(NC(c3cccc(C#C)c3)=O)C2)cn2cc(Br)sc2n1 95176,C=CCC(C)(CNC(=O)C=CC1CCCN1C(c1ccc(OC)nn1)=O)CO 95177,N1(C(CSC(C)(C)C)=O)CCC2(NC(C3COCC3(C)C)=O)CC2C1 95178,c1(C(N(S(CC(=O)OC)(=O)=O)CC2CCNCC2)=O)cnc2ccccc2c1 95179,N1(Cc2onc(C)n2)CCC(F)(F)C12CCC2 95180,N1(C(C(CC)F)=O)CCC2CN(C(c3ccnc(N4CCCC4)n3)=O)CCC12 95181,c1(C(N2CC3CN(C(CCCCC)=O)C3CC2)=O)cc(=O)c2cc(O)ccc2o1 95182,Cc1nc2cc(CC(=O)NCCN(C(=O)CC(C)CC(C)(C)C)C)ccc2o1 95183,CC(C)CC(O)C(=O)OC1CN(C(C2(CSc3ccccc3)CC2)=O)C1 95184,C12(Nc3ccnc(NC(CCC=C(C)C)C)n3)CC(C)(C1)OC21CCC1 95185,N1(C(c2c(OC)csc2)=O)CCC(NC(=O)C(C)P(C)(C)=O)C2(CCC2)C1 95186,Cc1cc2cc(-c3ccncc3C(=O)c3ccccc3C)ncc2cc1Cl 95187,C1(NC(C2(C)N(C)CCC2)=O)CC2(CCC(NC(C3CCN3C3COC3)=O)CC2)C1 95188,C(CCC(C)CC(=O)NC1CCN(C(C2CCN2S(C)(=O)=O)=O)CC1)=C(C)C 95189,C#CC1CCCC(NC(C2CCCC(NC(=O)CCN(CC)CC)CC2)=O)C1 95190,c1(C2CN(C(=O)CC3(OC(F)(F)F)CC3)C2)cccnc1 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95296,C(=O)(C(CC(F)F)c1ccccc1)N(CCNC(C1(C)ON=C(C)C1)=O)C 95297,CC(C)(C(=O)NCC(CO)NC(C1CCOC1)=O)C1CCC1 95298,C1(NC(N2CC(C(CC)C)C2)=O)C2CC3CC1CC(O)(C3)C2 95299,CNS(=O)(=O)N1CCC(C(=O)NCCNC(C2CN3CCC2(C)CC3)=O)CC1 95300,C1(c2ccccc2)(NC(C(C)=CC)=O)CCN(C(=O)C=Cc2nccs2)C1 95301,CC1CCC(Cl)=C(C(=O)N2CCN(C(=O)C(C)(C)CS(N)(=O)=O)CC(C)(C)C2)C1 95302,N1(C(C(C)OCCC)=O)CC2CC(C1)C(C(=O)O)C2N(C)C 95303,c1(C(N2CCOCC(NC(C(COC)(F)F)=O)C2)=O)cc2ccc(F)cc2cn1 95304,c1(SC(C)C(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)C2)ccc(F)c(F)c1 95305,C1(N(C(c2cc(C(C)C)no2)=O)C)CCCC(NC(C2CN(C(C)C)C2)=O)C1 95306,c1(CC(N2CCC(NC(CC3CC(SC)C3)=O)C(C)C2)=O)nc2ncccn2n1 95307,C(=O)(C(F)CCC(C)(C)C)NC(CCC=C)C(=O)NCC(C)CC1CCC1 95308,N=c1cc[nH]cc1C(=O)NCC1CCC1NC(=O)CCCNC(N)=O.c1(S)ccccc1 95309,C1(C(=O)NCC(C)N(C(COc2cccc(C(C)C)c2)=O)C)CN2CCC1CC2 95310,c1(CC)cccc(C(=O)NC2CN(C(c3cccnc3O)=O)CC2C)c1O 95311,O=C1CCC(C(=O)N2CC3(NC(=O)CCC4CCCC(O)C4)CCC2CC3)=NN1 95312,Cc1onc(C(N2CCCC(NC(=O)Cc3cc[nH]n3)C2C)=O)c1[N+](=O)[O-] 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95364,c1(-c2cn(-c3c(C(N(C)C)=O)cccc3)nn2)ccc(S(C)(=O)=O)c(F)c1 95365,Cc1c(C(N2CC3CC3(CNC(=O)CCOC3CC3)C2)=O)cccc1C(F)(F)F 95366,N1(C(C(C)(C)OCCC)=O)CCCC(N(C(c2nc[nH]c2C(F)(F)F)=O)CC)C1 95367,C(C)(CNC(c1ccc(C(c2ccco2)=O)o1)=O)(CO)NC(CCC)=O 95368,c1(OC(C)C)cc(CN(CCCNC(C2CCN(C(C)=O)C2)=O)C)ccn1 95369,c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)ccc(-c2cccnc2)s1 95370,c1(C(=O)NCC2CCN(C(c3cc(C(C)=O)on3)=O)C2)cncc(C)n1 95371,c1(NC(C(C)n2ccnn2)=O)cccc(CNC(c2ccoc2Br)=O)c1 95372,c1(OC)c(F)c(C(C(=O)NCCCSC)N(CCCO)C)cc(F)c1F 95373,C1(NC(COCC)=O)CC1C1CCCN(C(=O)CC2CN3CCC2CC3)C1 95374,N1(C(c2c(C)ccs2)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC2(CC2)C1 95375,C1(C(=O)N)CCC(C)(C)C1.C1(OC(C)C)(CN(C(C2(C)CC2)=O)C)CCC1 95376,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CC(N(C)C)C2)=O)C1 95377,Cc1cccc(C(=O)NCC2(C)CCC(NC(c3cnccn3)=O)C2)c1 95378,C1(C#N)(C(=O)NCC2CC(OC)CN2C(C2CCC2(C)C)=O)CCOCC1 95379,C1(C(=O)NC2C(OC)CCC2)CCC(O)CN1C(c1cccc(NC(C)=O)n1)=O 95380,C123CC(C1)(OC21CCC1)CN(C(=O)CCCOC)CC(=O)N3.CCCCCC 95381,N#Cc1cc(Br)ccc1N1CCN(C(C2CC(c3cccnc3)CN2)=O)CC1 95382,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 95383,n1(C(C)C)ccc(CCN2CCCC2c2cncn2C)n1 95384,N1(C(C(=O)NC(CC)CN(C(=O)C=C2CCC2)C)C)C(=O)NC2(CCCC2)C1=O 95385,N1(C(Cc2nc(C)oc2)=O)CC2C3CCC(C2C1)N(C(c1ccc(F)o1)=O)C3 95386,C(C(=O)N=c1ccn(CCF)[nH]1)(C1CC1)NC(c1c(C)cns1)=O 95387,c1(C(=O)Nc2cccc(CO)c2)ccc2nccn2n1 95388,CN=c1[nH]c(=NCCCC2CC(C)CO2)[nH]c(N(C)C)c1[N+](=O)[O-] 95389,C#CC(C(C)(C)C)N(C(=O)Nc1cccc(C2CC2)c1)C(=O)OC(C)(C)C 95390,C(=O)(C(C)Cc1cccnc1)NC(c1cn(Cc2cnc(CN(C)C)s2)nn1)C 95391,C(CC1C(=O)Nc2ccccc21)NC(=NCC(C)C)NCC1(C)C=CCCC1 95392,C1(C(=O)NC2(C(N(OC)C)=O)CC2)COC2(C1)CN(C(C1CCCN1C=O)=O)C2 95393,C1(C(C)C)CN(C(C2CCCCCC2)=O)CCN1C(c1cccn1C)=O 95394,C(=O)(C1C(=O)NCCn2ccc(c2)C(=O)N1)OC.C1(COC)CCC2CC12 95395,c1(N2C3C(CNC(C4(C)CC4Br)=O)C(CCC3)C2)nc(O)c2ccc(Cl)cc2n1 95396,c1(OC(C)C)cnccc1C(=O)NCC1(NC(=O)Cn2ncnn2)CCCCC1 95397,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(c2ccon2)=O)ccccc1 95398,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CC1CCCCC(=O)N1)C2 95399,c1(C(=O)NC(CN(C(=O)CC2CCC(C)(C)CO2)CC)C)[nH]c(=N)ccc1C 95400,C=CCN(OC)C(=O)C(C)C1CCCN(C(=O)CCC(F)(F)F)C1 95401,c1(C(C(=O)NC2CC2)N(c2ccccc2)C)cnc(OCCC#N)cc1F 95402,C(=O)(C#Cc1ccccc1)C(=O)C(N1CCCC(C2CCCC2)C1)=O.NC 95403,C1(NC(c2cccc(C)n2)=O)CC2CC1CC2C(=O)N(C(C)CO)C1CC1 95404,N1(C(C2(F)C(C)C2)=O)CCC(C2(NC(c3ccc(CO)nc3)=O)CC2)CC1 95405,C#CCCCCCNC(C1CCCCN1C(=O)CC1(OCC)CC1)=O 95406,C1(C2CCCC2)(CC(=O)NCCNC(C(c2cccs2)N(C)C)=O)CCOCC1 95407,c1(NC(CNC(C(C)N(CCC)CCOC)=O)=O)cc(O)cc(=O)o1 95408,C(=O)(CCOCSC)N(C(CN(C(COCCC)=O)C)C)C 95409,c1(C(C2(F)CCOC2)n2cc(C3CN(C(N(C)C)=O)CCO3)nn2)ccc(F)cc1 95410,CC1CCN(C(C2CC=CCO2)=O)CCN1C(C1CCCC(=O)CC1)=O 95411,N1(C(C2(CC)CC2(F)F)=O)CC(NC(c2cc(C)c(C)o2)=O)CC2(CCC2)C1 95412,c1(C(=O)Nc2nc(C)c(Cl)nc2)cn2c(n1)CN(C(c1ccc(F)nc1)=O)CC2 95413,CC(=O)CCCCC(=O)NC1CC(C(F)C(N2CCCC(CCF)C2)=O)C1 95414,C1(C(N2CC(NC(=O)CCCCCO)C(C(F)(F)F)C2)=O)Cc2ccncc2C1 95415,Cc1nc2c(s1)CCCC2C(=O)NCCOCCCNC(c1ncsc1C1CC1)=O 95416,c1(C(=O)NCCCN(C)C(c2nccnc2N)=O)c(F)ccc2c1OCC2 95417,N1(C(C(c2ccccc2F)C)=O)CCC2C(NC(=O)CSc3ccc(Cl)cc3)C12 95418,c1(C(=O)NC(CNC(c2cc(C)c(F)cn2)=O)C2CC2)c(Cl)ccc(C)c1O 95419,C1(CC(=O)NC2C=CCN(C(c3c(C)nco3)=O)C2)CC(=O)CC(=O)N1 95420,c1(NC(C)=O)ccc(C(=O)N(CC(C)O)CCNC(c2ccn(C(C)C)n2)=O)s1 95421,N1(C(c2c(C)c[nH]n2)C(=O)NCCC#N)CCN(c2cccnn2)CC1 95422,C1(O)(CN(C(C2COC3COCC23)=O)Cc2ccco2)CCN(C(C)CCOC)CC1 95423,c1(C(=O)NC2CCN(C(C(CSC)C)=O)C(C)C2)cn2cnnc2cn1 95424,C1(CNC(C=CCC)=O)CCCC1NC(c1cc(CCOCC)on1)=O 95425,CC(C(C)(C)C(N)=O)NCC(C)CCC1CCNCC1 95426,N1(C(C(C)CC(N)=O)=O)C2CCC1CC(N(C)C(c1cccc(C(N)=O)c1)=O)C2 95427,c1(C(=O)NC2CCN(C(C(C)(C)CF)=O)CC(O)C2)ccc2c(c1)C(=O)OC2 95428,N1(C(C(F)OC)=O)CCN(C(=O)CN2CCOCC2)C(CO)C1 95429,C1(N(C(=O)CC(C)=C(C)C)OCC)CCSC(C)C1.c1(C)nnc(S)o1 95430,N1(C(C(C)SC)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC2C1 95431,C1(C(=O)Nc2cc(C(=O)OCC)n[nH]2)CCN(C(c2cc[nH]c2)=O)CCC1(F)F 95432,c1(CNC(C2CCC(NC(c3c(CC)non3)=O)C2)=O)nc(Cl)ccc1F 95433,c1(CNC(CNC(=O)OC)(C)CO)ccc(C(C)CC(=O)N(C)CCO)cc1 95434,c1(C(=O)NCCN(C)C(C2CCCC2)=O)cc(-c2ccoc2)on1 95435,Cc1cnc(C(=O)NCC2CC(C)N(C(c3c(O)cccc3F)=O)C2)c(C)c1 95436,c1(CC(=O)NCC(CO)NC(CNC(=O)OC)=O)ccc(F)cn1 95437,CC(C)C(C(C)NC(c1cscc1Br)=O)NC(c1ccc(C(C)(C)C)o1)=O 95438,C=CCCC(C)NC(=O)C(C)N(C(=O)C(=O)NC(C)C)C1CC1 95439,c1(NC)ccc(Cl)c(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2ccoc2)c1 95440,C1(NC(C2CC(=O)NCC2)=O)CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1(F)F 95441,CCCS(=O)(=O)c1ccccc1C(=O)NC1CC(NC(=O)CC(CC)CCC)C1 95442,C1(CNC(CC=C)=O)C2CCC(C2)N1C(C1CCOC1C)=O 95443,C1(NC(C2CCC(F)CC2)=O)CCCC2CN(C(C3CCS(=O)(=O)CC3)=O)CC12 95444,C=CCC(C)(C(=O)NC1CN(C(=O)CCc2cccnc2)CCC1F)N(C)C 95445,N#Cc1cc(NC(C2CSCCN2C(C2CC2C2CC2)=O)=O)cc(Cl)c1 95446,C=CCC(C)(C)CC(=O)NC(C)CCN(C(=O)CCC(C)(C)OC)C 95447,c1(OC)cc(OC)c(C(N2CC(NC(=O)Cc3scnc3C)CC2C)=O)c(N)c1 95448,c1(C(=O)NC(C)CNC(=O)CSC(F)F)cc2cccc(Cl)c2cn1 95449,C1(C(=O)NC(C(=O)N(CC)Cc2ccoc2)C2CCC2)CC2CC2C1 95450,N1(S(C(CC)C)(=O)=O)CC2(CN(C(=O)COc3ccccc3)C2)C1 95451,C1(C(C)(C)C)(CO)CCN(C(=O)C(C)(C)C(=O)NC(c2cc(Cl)no2)CC)C1 95452,C=CC(C)(CCOC)C(=O)N1CC(C(=O)NCC2CC3CCC3C2)CC12CCC2 95453,Cc1cc(C(=O)N(CC(=O)NC(CC2CCCC2)CO)CC2CC2)cn1C 95454,c1(OC)ccc2[nH]nc(C(=O)NC(C)CNC(c3c(F)cc(C)cc3F)=O)c2c1 95455,C=Cc1cccc(-c2cnc(N3CCN(C4CCOCC4)CC3C)nc2)c1 95456,CC1CN(C(c2ccc(F)c(C#N)c2)=O)C(C)CN1C(c1ccc(C2CC2)cc1)=O 95457,CCCC(CCC)CC(=O)NC1(C(F)F)CC(NC(=O)CC(CC)OC)C1 95458,C(CO)(CCCCNC(C1(CF)CCC1)=O)NC(=O)COc1ccccc1 95459,c1(C(=O)NC2CC3CN(C(c4ccc(F)cc4F)=O)CC23)cccc2nc[nH]c12 95460,C(=O)(C(C)CS(C)=O)N(CCNC(c1cc(-c2cccc(C)c2)no1)=O)CC1CC1 95461,c1(CN2C(C(=O)Nc3cccc(C(=O)OC)c3Cl)CCC2)cc2cccnc2[nH]1 95462,c1(C(=O)NCC2N(C(CNC(C)=O)=O)CC3CCC2C3)ccc2ncccc2c1F 95463,c1(-c2n(CC(n3ccc4cc(Cl)ccc34)C)ccn2)cc(S(C)(=O)=O)ccc1F 95464,C1(NC(CSS(C)(=O)=O)=O)COCCC1Nc1ccco1 95465,C1(N(C(C=CCC)=O)C)CCCN(Cc2c(C(F)(F)F)nn(C)c2Cl)CC1 95466,C1(C(=O)NC2CC(NC(C=CC3C(C)C3(Cl)Cl)=O)C2)C2CC3CC(C2)CC1C3 95467,C(CC(=O)NC1CC(C)CCC1O)(C(C)(C)C)NC(c1ccc(C)[nH]1)=O 95468,c1(-c2c(C)occ2)nc(Cc2c[nH]nc2-c2ccsc2)n(-c2cccnc2)n1 95469,c1(C(=O)NCC(CNC(CC=CC)=O)F)cnc2ccccn12 95470,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)CC2C=CCCC2)C1 95471,N1(C(=O)C=Cc2ccco2)CC2CCC(C1CO)N2C(=O)CSC1CC1 95472,CC1COCC(CC(=O)NC(c2cccnc2)C(=O)N2CC=CC2)O1 95473,c1(N(C(c2ccccc2)CC)CC(C)C)nccc(=NC(C)c2cccnc2)[nH]1 95474,c1(N2CCCC(C(=O)NC)C2)ccc(C(N2CC(NC)C3CC3C2)=O)cc1[N+](=O)[O-] 95475,c1(CCC(=O)NC2CC3CCC2N3C(C2CC3(CC3)CO2)=O)ccc(O)c(F)c1 95476,CC(C)C(C(=O)N(CC(C)O)C1CCC1)n1cncn1 95477,C1(NC(CCc2cc(C)sc2C)=O)CCCCN(C(C2(C(F)F)CCC2)=O)C1 95478,N1(CCC2CCN(C(=O)Cc3cscc3Br)C2)CCC(O)(c2ccccc2)CC1 95479,CCC(CN(C)C)CC(=O)NCCC(C)NC(c1cnn(C2CCCCC2)c1)=O 95480,c1(C(=O)NCc2cccc3c2CCN3)ccc2c(F)cc(F)cc2n1 95481,C(=O)(CC(C)P(C)(C)=O)NCC(CNC=O)OC.C(C)(C)(C)OOC 95482,C1(CCC(=O)OC(C)C)(C(N2C(C)(C)COCC2=O)C)CC(F)C1.C1(CO)CC1 95483,C1(CNC(C2CCSC2)C)CCC(C2COCCN2C(=O)OC(C)(C)C)O1 95484,N12Cc3ccccc3CC1CCNC(CC)C2=O.c1(N)ccc(Br)s1.OC 95485,c1(C(=O)NCC2CN(C(CS(CC)=O)=O)CC2O)cc(F)cc(C)c1C 95486,C1(CC)CN(C(=O)C(C)n2ccnn2)CCC1CNC(=O)Cc1cc(C)ns1 95487,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NCc1cc[nH]n1 95488,C1(CNC(C(F)=CCC)=O)CN(C(c2ccc(N3CCCCC3)nc2)=O)CCO1 95489,CC(C)(C#N)CC(=O)NCC1CCN(C(c2cn(CCCC#N)nn2)=O)CC1 95490,C(=O)(CC(C)c1ccco1)NCCCN(C(CSC)=O)CC1CCCCC1 95491,Cc1sc(Cl)c(C(=O)NC(C)(CNC(c2ccnc(C3CC3)n2)=O)C(C)C)c1C 95492,C(=O)(C(C(C)C)C(C)C)N(CCNC(N1CC(COC)C1C(=O)OC)=O)C 95493,C1(CC#C)CCCN1C(=O)C(=O)NCCCCC1CN(C(C2CCCCO2)=O)C1 95494,N1(C(COCC)=O)CCCN(C2CCN(C(c3cc(N)cc(F)c3)=O)C2)CC1 95495,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 95496,C1(CC(N2CCC(OCCC)C2)=O)CN(C(c2sccc2C#N)=O)CCO1 95497,c1(C(=O)NCC(C)CNC(=O)CSCc2nnnn2C)cccc2nsnc12 95498,c1(OC(C(=O)NCC2C(NC(CC=C)=O)C2)(C)CO)ccc([N+](=O)[O-])cc1 95499,c1(-c2ccc(NCCN(C(c3cc(C)c(O)nn3)=O)CC)s2)ccc(Cl)c(Cl)c1 95500,C1(NC(C=C(C)C(C)C)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 95501,c1(C(=O)NC(c2ccc(F)c(F)c2)C)ccc(OC(F)(F)F)cc1[N+](=O)[O-] 95502,C1N(C(C)C=O)CC1N=c1[nH]nco1.C1CCCC1 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95539,C1(N(C(=O)CC2CCC(F)(F)C2)C)CCCN(C(=O)C#CC2CCC2)CC1 95540,c1(C(=O)NC(CSCC)C(=O)NC2CC(=O)N(C)C2)cc(C#N)ccc1N 95541,C1(C(=O)NC(c2nccs2)CC)CC(O)CN1C(C1CN(C(C)=O)C1)=O 95542,C1(C(=O)NC2C(CC(=O)Nc3c(C)nsc3)C(O)C2)CC2(CCC2)C1 95543,c1(CC)ccc(CC(=O)NC2CCC(C)N(C(c3[nH]ccc3C)=O)C2)cc1F 95544,C(=O)(C1=NOCC1)NC1(CC=C)CN(C(c2c[nH]nc2C)=O)C1 95545,C(=O)(C#CC1CCCO1)N1CC(CCC)(NC(=O)CN2C(=O)CN(C)C2=O)C1 95546,c1(NC(CNC(CNC(CN(CCC#C)C)=O)=O)=O)c(C)[nH]c(C)cc1=O 95547,c1(CC)cc(C(=O)NC2CN(C(=O)CC(O)CN(C)C)CC23CC3)cc(F)c1 95548,C1(NC(CCSC)=O)CN(C(=O)Cc2cncn2C2CC2)CC1O 95549,c1(C(=O)NCC2(C(=O)NC3C(C)(C(C)C)C3)CCOCC2)cc(C#N)ccc1F 95550,c1(C(N2CCCCC(CNC(C3CC3F)=O)C2)=O)ccc2c3c(cccc13)CC2 95551,N1(C(C(F)OC)=O)CC2CCC(CNC(c3sccc3S(C)(=O)=O)=O)(C2)C1 95552,C1(C(=O)NC2CC3CC(NC(CCSCC)=O)CC32)CC(C(C)(C)C)=NO1 95553,CCC(F)(C(=O)OC)C(=O)NC(CCN(C)C(C1CCCC2CC12)=O)C(C)C 95554,CC1CN(C(=O)C=Cc2cnccn2)CC(C)CN1C(C1COC1)=O 95555,Cn1ccc(C(=O)NC2CC2C(=O)Nc2ccc(C(F)F)cc2F)cc1=O 95556,C1(OC)CCCN(C(=O)C(CNC(=O)C(C)=CC(C)(C)C)N=[N+]=[N-])CC1 95557,C12(CNC(CC3(COC)CC3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 95558,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 95559,c1(OC)ccc(OC)c(OC(C2CCCN2C(c2sccc2Cl)=O)=O)c1.C1CN1 95560,C1(CNC(C(N2CCCCC2)C)=O)CCN(C(C2CC23CCC3)=O)C12CC2 95561,C1(C(=O)N(C)CCC2CCCO2)(CC)CN(C(=O)CN2CCOCC2)C1 95562,C1(CNC(C(N2CCN(C(=O)NCC(=O)OC)CC2)=O)=O)CCCC(C)CC1 95563,C(CC(C)C)(C(=O)NCC(O)CNC(C1(CF)CCC1)=O)NC(C)=O 95564,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CCC)n(C)n2)=O)CC1OC 95565,N1(C(C2CC(OCC)C2)=O)CCCCC(NC(c2cccnc2CO)=O)C1 95566,CC1CN2CCC1=CC2=O.C1(NC(C2CCC2)=O)CC2(CCC2)C1N(C)C=O 95567,CC1CN(CC(=O)NCc2cn(C3CC3)nn2)CCC1C(=O)N(C)C 95568,Cn1ccc2ccc(C(=O)NC(C)(CNC(=O)CCN3CCCCC3)CO)cc12 95569,c1(-c2ccc(CCC3(CC)CCCCO3)s2)ccc(C)c(C(=O)OC)n1 95570,c1(CN2CCC(NC(c3cccc(Br)c3Br)=O)C2)cc(F)c(Br)c(F)c1 95571,N1(C(CN2CCN(CC)CC2)=O)CCCC(O)(CNC(=O)CC(C)N(C)C)C1 95572,Cc1nn(-c2ccccc2)nc1Cn1cc(C(C)C2CC2)nn1 95573,C(C(C(C)(C)C)NC(=O)CC1CSC1)NC(C1C(C(C(C)C)O)C1)=O 95574,c1(NC(CCN2CCC(C(C)N)CC2)=O)ccc(C#N)c(Cl)c1.C12CCN(C1)C2 95575,C(CCC(C)CC(=O)NCCCCN(C)C(c1ncn(C)c1C)=O)=C(C)C 95576,n1(CC(N2CC(NC(C3(C=C)CCC3)=O)C3(C2)CC3)=O)nc2n(c1=O)CCCC2 95577,CC(C)CCC(=O)N(CC(O)CN(C)CS(=O)(=O)CC1CN(CC(F)(F)F)C1)C 95578,c1(C(=O)NCC2C3CN(C(C4C(C)CC=CC4)=O)CC32)ccc2cn(C)nc2c1 95579,N1(C(C(c2cncnc2)C)=O)C2CCC1C1CC1(NC(=O)C(F)=CC1CC1)C2 95580,C(=O)(C(C)(C)C(=O)N1CCCCC1C1CN(C(=O)CC2(NC(C)=O)CC2)C1)OC 95581,Cc1ccc(C2C(C(=O)N(C(CNC(c3cocn3)=O)C3CC3)C)C2)o1 95582,C(=O)(CC(F)(F)F)Oc1nnc(C(C)(C)CCCC=O)s1.C12CC(F)(C1)CN2CC(=O)OC 95583,c1(C(N2CCCCC(NC(C(=O)NC(C)C)=O)C2)=O)ccc2nn[nH]c2c1 95584,Cc1ncc(Br)c(CN2CCSCC2C(=O)NCc2ccccc2Br)n1 95585,CC(C)(CCNC(c1csc(-c2ccccc2)c1)=O)C1CC1 95586,C(=O)(C1=C(C#N)CCC1)NCCCC(C)(C)NC(C1C(C)(CC)C1)=O 95587,CC1SCCCN1C(=O)C(=O)NCCCNC.C(C(F)(F)F)S 95588,C1(C(N(CCC(=O)NCC2C3COCC23)C)=O)OC2CCC1C2 95589,CC1CC(NC(c2ncccc2Cl)=O)CN1c1cc(C(N)=O)ncn1 95590,N1(C(CCOCC#C)=O)CCCC(NC(c2ccn(C)n2)=O)C(F)C1 95591,N1(C(CC2(C=C)CN(C(=O)C(C)Oc3ccccc3)C2)=O)CC2(C1)CC2(F)F 95592,c1(C(=O)NC2(C(=O)O)CC(C#C)C2)cc2ccc(Br)cn2n1 95593,C1(CC)(NC(N2CCN(Cc3cccc(F)c3)CC2)=O)CCCNC1=O 95594,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 95595,c1(NC(C2C3CCN(C(C4CCCCO4)=O)CC23)=O)cnc2[nH]ncc2c1 95596,C1(C)(C(=O)NCCCN(C(C)=O)C)CCN(C(C2CC(=C3CC3)C2)=O)CC1 95597,c1(C(N(CCn2c(CC)ncc2)CC)=O)nc(C2CC2)sc1Br.c12cn(nn1)C2 95598,C1(C(N(C(C(N)=O)C2CCCC2)CC)=O)CCC1NC(C1CCC1)=O 95599,N1(C(c2nc(CC)oc2)=O)CCCC(C2(NC(c3cnc(Cl)c(F)c3)=O)CC2)C1 95600,c1(C(N2CCC(C3NCC34CCC4)CC2)=O)nc(C2CC2)ccc1I 95601,c1(OC)ccncc1C(=O)NCc1nocc1C(N1CCC1(C)C(N)=O)=O 95602,CC(C)CC(C)CC(=O)N1CCC1(C)CC(=O)NOCC(O)C(F)(F)F 95603,N1(C(c2nncc(C)c2)=O)CCC2(NC(c3cc(=O)n(C)cn3)=O)CCCCC12 95604,c1(OCC)cc(C=CCN2CCC(O)CC2C(N)=O)c(OC)cc1Cl 95605,N1(C(CC(COC)(C)O)=O)CCC(N=[N+]=[N-])(C(=O)NOCCF)C1 95606,Cn1ccc2[nH]c(C(N3CCC(NC(C4(n5cccn5)CC4)=O)C3)=O)cc12 95607,c1(C(=O)NCC2(CNC(C3N(C)CCC3)=O)CC2)ccc(N2CCCC2)nc1 95608,C(C(=O)N=c1cc(C)n(CCO)[nH]1)=CCOC1C(C(=O)OCCC)CCCC1 95609,N1(C(C(CCO)N(C)C)=O)CCC2(CN(C)C2)C(C(=O)NCCSC)C1.C(C)(C)(C)O 95610,Cc1nscc1C(=O)N(C)Cc1cn(Cc2nc(C(C)(F)F)n[nH]2)nn1 95611,c1(C(N2CC3C(CNC(C=COCC)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1OC 95612,CC1(C(=O)NCC2CN(C(C3C=CCS3)=O)CC2O)CCCC1O 95613,c1(C(N(C(CNC(=O)C=CCn2cncn2)C2CC2)C)=O)ccc(CO)nc1 95614,CN1CCC(C(=O)NC(C)(C)CCCCNC(=O)C(F)CC2CCC2)C1=O 95615,c1(OC)cc(C(=O)OC(C)C(=O)NC(C2CCOC2)=O)c(F)cc1F 95616,Cc1nc(NCc2cc(CC3CC3)on2)cc(=NC(C)c2ccc(Cl)c(C#N)c2)[nH]1 95617,c1(NC2(c3n(C(CC)(C)C)nnn3)CC(c3n[nH]cc3C)C2)cccc(Cl)c1 95618,c1(CCCNC(C2CC2C2CCNCC2)=O)nc2c(s1)C(CCCN)CCC2 95619,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 95620,c1(NC2CN(C(c3nc(COC)sc3)=O)CC(C)C2)ncnc(N(C)C)c1[N+](=O)[O-] 95621,c1(C(N2CCCC(NC(Cc3c(CC)noc3CC)=O)C2)=O)cnc(Cl)cc1Cl 95622,c1(NC(=O)CN(C2CCC2)C(C2(Cl)CC2)=O)cccc(OC2CCOC2)c1 95623,Cc1cccc(O)c1C(N1CCOC(CNC(=O)C2=NNC(C(F)(F)F)C2)C1)=O 95624,c1(C(=O)NC(C)C(N2CC(CNC(n3cnnn3)=O)C(C)C2)=O)cccc(Cl)c1F 95625,N1(C(CC2(C=C)CCC2)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 95626,c1(C(=O)Cn2cccn2)cc(-c2ccc(Cl)cc2)ccc1O 95627,c1(SC)nn(C)cc1C(N1CCC(C)C1CNC(C1(C(C)C)CCC1)=O)=O 95628,N1(C(c2cnn(C)c2C(F)(F)F)=O)CCC2(CCN(C(=O)C(F)C3CCC3)C2)C1 95629,c1(C(N(CC(CNC(c2c(O)ccc(CC)c2)=O)C)C)=O)cc(S(N)(=O)=O)co1 95630,c1(OC)cc(NC(c2cccc(F)c2)C2CCC2)cc(Br)c1OC 95631,C1(OC)CCC(C(=O)NCC2CCCCC2NC(=O)CSC2CC2)CC1 95632,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)CS(C)(=O)=O)C(O)C1)=O 95633,C=CCCC(C(=O)N(CC)CC1(CNC(=O)CC(=C)Br)CC1)c1ccccc1 95634,C1(C(N2CCC(CN(C)C)C2)=O)CCCCN1C(C1CC(=C2CC2)C1)=O 95635,c1(NCCNC(C2CC(Cc3n(CC)cnn3)OCC2)=O)ccccc1[N+](=O)[O-] 95636,C1(C(=O)NCC2(C(N(CCC#C)CCO)=O)CC2)CC1C#N 95637,CCC(C)(C#N)C(=O)NC1CCCN(C(=O)CCC(=O)c2ccc(F)cc2)C1 95638,C1(NC(c2cnn(C)c2F)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 95639,c1(C(=O)NCC(=O)NCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 95640,Cc1cc(NC(C2CCCCCN2C(c2cccs2)=O)=O)ccc1O 95641,CCCCCCCCN(C(=O)C(CC1CCC1)OCC)CCO.C1(=O)C(C)O1 95642,C1(NC(C(C2(O)CN(C(C=C(COC)C)=O)C2)F)=O)CCC2(CCC2)C1 95643,N1(C(c2c(OC)c(Cl)cc(Br)c2)=O)CCn2cnc(C3=CCSCC3)c2C1 95644,Cc1cc(C(=O)NCCN2CCN(C(C3CCNC3=O)=O)CC2)cnc1O 95645,N1(C(C(C=CC)O)=O)CCCC2(CCN(C(=O)C=CSc3ccccc3)CC2)C1 95646,C1(CNC(C2C3CNC(=O)C23)=O)CCN(C(c2cccc(O)n2)=O)CC1 95647,C(=O)(C(F)(F)C(F)(F)F)NCC(CC=C)C(=O)NCC(C1CCC1)OCC 95648,C1(CNC(N2CC3CC(C(=O)OC(C)(C)C)C3C2)=O)CN2CCCN1CC2 95649,CC(C)CN=C(NCc1sccc1Cl)N1CC(C)N(C(c2ccccc2)C)C(C)C1 95650,CCC(CC(C)C)C(=O)NCC1CC2(CC2)CN1C(=O)CCCOCCOC 95651,C(CC(C)C)(C(=O)N)NC(=O)NCC(=O)NC.c1(CC2CCC2)ccc(Cl)c(Br)c1 95652,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 95653,CCCC(C(C(=O)NCC)N1CC(O)C2(CC2)C1)OC 95654,c1(CC(N2CC(=C(CNC(C(CC)SC)=O)F)C2)=O)ccc(F)cc1C 95655,C(CCCCCO)NC(C(c1nnnn1C1CCCC1)OC)(C)C1CCCO1 95656,N1(C(CCCN(CC(CC)C)C(=O)OC(C)(C)C)=O)CC(O)(C(F)(F)CF)C1 95657,N1(C(c2ncn(C(C)C)n2)=O)CC2(CCCC2NC(C2(C3CCC3)CCC2)=O)C1 95658,c1(NC(=O)CN2CCC23CN(C(C2CCCCC2)=O)C3)c(F)cc(F)cc1Cl 95659,C1(NC(C(c2ccccc2)N(C)C)=O)CCN(C(=O)NCCSC(F)F)CC1 95660,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2cnc(C)o2)=O)C(c2cn[nH]c2)C1 95661,CC(C(=O)N1CCC(n2cc(-c3ccc(Br)cc3)nn2)CC1)C(F)F 95662,N1(C(C(CCC)O)=O)CC2(CCN(C(=O)Cc3ccc(Br)cc3F)CC2)C1 95663,N1(C(c2c(Cl)ccc(C)c2)=O)CC2CN(C(c3ccc([N+](=O)[O-])s3)=O)CCC12 95664,N1(C(c2c(OC)scc2)=O)CCCC2(NC(c3cc(Cl)ccc3N)=O)CCCC12 95665,c1(C(N2CC(N(C(=O)COCCCF)C)C2)=O)cn2ccncc2n1 95666,N1(C(c2ccc(-n3cc(C4(C(C)C)CC4)nn3)cc2)=O)CCC2(CCSC2)C1 95667,c1(OC(C(=O)NC(CN(C(C(C)O)=O)C)C)C)ccc(Cl)cc1 95668,c1(C(N2CC(CC(C(=O)NCC(C(C)(F)F)F)F)C2)=O)ccc([N+](=O)[O-])[nH]1 95669,c1(C(=O)NC(CN2CC(C)CC(C)C2)C)nc(Cl)c(Br)cc1[N+](=O)[O-] 95670,c1(NC(c2ccc(N(C)C)cc2F)=O)n[nH]c2cc(-c3ccco3)ccc12 95671,NC1CCCCN(CC(N2CCN(c3cccc(Cl)c3)CC2)=O)C1=O 95672,CC1C(NC(=O)CC2=CCCC2)CC2CCC1N2C(=O)CC1CCC2CC12 95673,c1(C(=O)NCC2N(C(c3cccc(C)c3)=O)CC(O)C2)c(C)cc(O)nc1C 95674,c12cc(Cl)ccc1S(=O)(=O)N1CC2C1.n1(CCC=O)cc(Br)cn1.C(=O)O 95675,C(N=c1[nH]c(Cl)nc2c1S(=O)(=O)CC2)c1cc(CNC(c2ccsn2)=O)c(F)cc1 95676,c1(OC)ccccc1C(F)(F)C(=O)N(C)CCN(C)C(c1cc(Cl)ncn1)=O 95677,CCCS(=O)(=O)CC(=O)NC1CCC(NC(=O)CC2OCCC2(C)C)CC1 95678,C1(N(C)C(c2cc(C(C)(C)C)on2)=O)CCC(NC(=O)CCCC#N)CC1 95679,c1(-c2ccccn2)ccc2c(c1)CC2.n1(CCC)nnnc1CNCC(F)C1CCC1 95680,C1(CNC(c2cn(CC)nn2)=O)CC12CCN(C(c1c(C)nnn1CC)=O)CC2 95681,CN1CCOCC1CC(=O)NC1CCN(C2CCN(C(C3CC=CC3)=O)C2)CC1 95682,C1(C(N(C(C)CNC(c2cnoc2C2CC2)=O)C)=O)CCCCC1O 95683,c1(NC(CN(C(c2c(OC)cccc2)=O)C2CC2)=O)c([N+](=O)[O-])cnn1C 95684,c1(C(=O)NNC(=O)C2CC(n3ccnc3)C2)cc(F)cnc1Br 95685,C1(C(=O)NCCCN(C)C(C2CC3(CCO2)CC3)=O)CC12CCC1(CC1)O2 95686,Cc1cc(C(=O)NC2(c3cc(Br)ccc3Cl)CC2)cc(C)c1N 95687,c1(C(=O)NCC(C2CCCC2)NC(C(CCOC)NC(C)=O)=O)ccc(N)c(F)c1 95688,CC(F)(CC1CCCC1)C(=O)NCC1CCCN1C(c1nc(=N)cc[nH]1)=O 95689,C1(CNC(c2c(C)ccnc2)=O)CC2CC(C1)N(C(c1ccc(F)cc1F)=O)C2 95690,C1(CNC(C(c2cnc(OC)nc2)N2CCOCC2CO)=O)C2CCCCCC12 95691,C1(C(N(C2CCN(C(C(n3ccc(C)n3)C)=O)C2)C)=O)CCC(CO)CC1 95692,CC(CC(N)=O)C(=O)N(C(CCF)C(=O)NC(C)CCO)C 95693,N1(C(CC=C=C)=O)CCN(C(=O)C=Cc2ccc(SC)s2)C(CC)C1 95694,c1(N2CCC(C)(C(=O)Nc3n(C)nc(O)c3)C2)nccc(C#N)n1 95695,C1(C(=O)NC2(CO)CN(C(c3cn(C)nc3)=O)C2)CC2C=CC1C2 95696,C1(CNC(c2c(CC)nn(C)c2)=O)N(C(=O)CC2CC(C)=NO2)CCC1(C)C 95697,N1(C(c2c(C)cnnc2O)=O)CCC2(CCN(C(C3(C)CC3C)=O)CC2)C(C)C1 95698,c1(C(=O)NCC(O)CNC(c2ccc(F)cc2Cl)=O)cnc2sccc2c1 95699,c1(C(N(C)CC2N(c3ncc(C)cn3)CCC2)=O)cc(Br)cc(Cl)c1C 95700,C1(C(=O)NCCC(=O)NCCOC)CCCN1C(c1ccccn1)=O 95701,c1(OCC2CCOC2)cccc(Br)c1.C12COCCN1C(=O)N2C 95702,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(c2ncccc2Cl)=O)C(C(F)(F)F)C1 95703,c1c(F)cccc1Cl.C1(NC(C)=O)COCC1NC(=O)C(F)(F)c1csc(=N)[nH]1 95704,C1(C(=O)NC2C(NC(C3=C(C)OCC3)=O)COCC2)CN2CCN1CC2C 95705,N1(C(CCC(=O)NCC)=O)CC(C)CN(C(c2cc(C)ccn2)=O)C(C)C1 95706,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 95707,c1(OC)cncc(C(C(=O)NN(C)C(c2cccnc2)C)OC)c1.C1(C)CCOC1 95708,c1(C(C(=O)NC2(C(C)NC(C(C)OCCOCC)=O)CC2)(F)F)cc(Cl)sc1Cl 95709,c1(NC(CN(C(CCCNC(CSC)=O)=O)C(C)C)=O)cccnc1C 95710,N1(C(c2c(C)[nH]cc2)=O)CC(N=[N+]=[N-])CC1C(N1CCC12CC(O)C2)=O 95711,C1(CCNC(c2c(CC)con2)=O)CN(C(C2CC(F)CN2C)=O)CC1C 95712,c1(C(=O)NC2CCCN(C(c3cc(CCC)[nH]n3)=O)C2C)c(C)ccc(C)c1N 95713,c1(C(N(CC(C)(C)CNC(=O)CSC(C)C)CC)=O)cnc2c(C)cccc2c1 95714,CC(CCNCC1CCCC1O)CCN 95715,N1(C(CN(C)CC)=O)CC(C)(C)OC2(C1)CN(C(C1COCCO1)=O)C2 95716,C1(C)(C(=O)NC2CC(C(C)NC(=O)CCc3ccnn3C)C2)CCC(=O)CC1 95717,c1(COC(C2C(NC3CC(C)C3)CCC2)=O)nc(-c2ccccc2)n[nH]1 95718,N1(C(=O)CCNc2ccccc2C(F)(F)F)CC2(CCN2C(C2CC2Cl)=O)C1 95719,C(c1scnc1C)=CC(=O)N(CC(C)(C)NC(c1c(CC)occ1)=O)C 95720,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 95721,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 95722,Nc1ccc(C(=O)NC2(CNC(=O)CN3C(=O)CNC3=O)CCCC2)cc1F 95723,C1(C(=O)Nc2cccc(NC(C3(C)CC3)=O)c2)SC2C=CC1CC2 95724,C(=O)(C(C)CCCC(C)C)NC(C(=O)NC(C#C)CC)CCOCCO 95725,CC1CC=C(C(=O)NC2CCCC(CNC(=O)CN(CCO)CCO)C2)CC1 95726,Cc1ncc2cc(C(N3CCC(n4cc(CC(O)C5CC5)nn4)C3)=O)nn2n1 95727,c1(COC)nn[nH]c1C(=O)N(CCC(C)NC(=O)C=CCF)CCO 95728,CCC(C)CCC(O)CC(=O)N1CCC(O)(Cc2cn(CCCCO)nn2)CC1 95729,N1(c2snc(COC)n2)CCOC(CN(C(=O)C=CCN(C)C)C)C1 95730,c1(COC)nc(=NCC(C)N(C(=O)C(c2ccc(F)cc2)CO)C)s[nH]1 95731,C1(C(N(CC(CC)NC(=O)CCOCCCCCO)C)=O)OCC2COCCC12 95732,c1(C(=O)Nc2cc(C(=O)OC)sc2)ccccc1-n1cc(C(O)C(C)C)nn1 95733,C1(CNC(COCCN(C)C)=O)CN(C(=O)Cc2cncnc2)CCO1 95734,C1(NC(c2ccc(C(=O)OC)cc2C)=O)CCC2CCCCC2C1 95735,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CCO4)=O)C3)OCC2)=O)CCOCC1 95736,CC1CC(C(=O)N2CC(O)(C(C)(C)CNC(C3(C)CCCCCC3)=O)C2)=NO1 95737,C(C(N=c1ccnc(NC2CC2)[nH]1)C(C)CO)c1ccc(C(C)C)cc1.C1CO1 95738,c1(CN(C(CC)=O)C)cncc(-c2ccc(N(CCC#N)CC)cc2)c1 95739,C=CCCC(O)CN1C(=O)C(NC(=O)C=C(C)C(F)F)CC1.C(C)(=O)NC 95740,C#CCC(C)(C)C(=O)N1CC(N(C(=O)Cc2ccn(C(C)C)n2)C)C2(CC2)C1 95741,C1(NC(CC=C)=O)(COCCCC)CN(C(=O)Cc2cc(Br)cs2)C1 95742,C(CCCN=c1ccnc[nH]1)NC(c1c(C)occ1)=O 95743,O(N=c1ncnc2[nH][nH]c(I)c1-2)N1C2CN(C(c3ccc(C)c(F)c3F)=O)CC21 95744,c12ccc(F)c(c1F)C(=O)NC2.C1(C(=O)N)CC(N(C)C)C1.C1(OCC)CC1COC 95745,c1(N(C(C)CCNC(C2CC2(C)Br)=O)C)nnccc1C#N 95746,N1(C(CCCOCC)=O)CC(C)C(C)(CNC(c2ncc(CC)o2)=O)C1 95747,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 95748,N1(C(C(C)(C)OCC)=O)CC2CCCC2(CNC(=O)Cn2cnc([N+](=O)[O-])c2)C1 95749,N1(C(C2C3(CC(NC(C(C(C(C)C)OC)O)=O)C3)C2)=O)CCCC2(CCCC2)C1 95750,C1(N(C(c2ncn(C(C)C)c2)=O)C)CN(C(=O)C(CC2CCC2)N(C)C)CC1F 95751,C1(C(=O)NCC23OCC(NC(C(C)n4cccn4)=O)(C2)C3)CN2CCN1CC2 95752,Cc1nc2ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)C)cc2c(=O)n1C 95753,C1(C(N2CCC(C)(C(N3CC(C(C)C)OCC3)=O)C2)=O)CC2CC(=O)C1O2 95754,O=C(NNC(=O)C12CC(CO)(C1)C2)C1CC(SC(F)F)C1 95755,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(SC)o2)=O)CCCO1 95756,N1(C(c2c(CC)csc2)=O)CC2CN(C(c3cnc(OCC)nc3)=O)CC12 95757,N1(Cc2cc(OC)cc(O)c2)CCCCC(C)(F)C1.c12cc(nc(C)n1)S2 95758,C12(NC(c3ccc(F)o3)=O)CCCN(C(c3cc4ccsc4[nH]3)=O)CC1C2 95759,c1(C(N(CCC(C)NC(C(CC=C)C)=O)C)=O)nc2ccccn2c1F 95760,C1(NC(C2(COC)CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 95761,CCCC(C(=O)NCC(C)(CC)NC(c1cnc(COC)s1)=O)S(N)(=O)=O 95762,C(=O)(CC(C)C(C)C)N1C(C(C)NC(c2cnc(C)nc2)=O)CCC1 95763,C(CC(C)C)(C(N)=O)NC(c1n(CC(=C)C)nnn1)c1cnc(-c2ccsc2)s1 95764,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 95765,C(=O)(CCC(=O)c1cccnc1)NCCCC(C)NC(=O)C(F)n1cccn1 95766,CC(C)(C#N)C(=O)NCCCOCCCNC(C1CC(O)(c2ccccc2)C1)=O 95767,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 95768,C1(F)(CNC(c2ccc(Oc3cccnc3)cc2)=O)CCN(C(=O)NC2CCC2)C1 95769,C1(O)(C(CNC(CCCOC)=O)C)CCN(C(=O)CC2(C3CC3)CC2)C1 95770,N1(C(c2nc(COC)oc2)=O)CCOC(CN(C)C(C2COCCN2C)=O)C1 95771,C1(C(=O)NCCCC(C)C)CN(C(C2(NC(N)=O)CC2)=O)CCC1C 95772,c1(C(=O)NCC2(NC(=O)C=CI)CCCCC2)ccc2nc(O)[nH]c2c1 95773,c1(C(=O)NCC(C)(O)CNC(c2ccc(C3CCC3)nc2)=O)ccc(N)c(O)c1 95774,C1(N)CCCC(NC(=O)CNC(C(C(C2CC2)OCC)=O)=O)C1.c1(N)ccsn1 95775,C(CNC(=O)CCC1CCOC1)(CC(C)C)NC(c1cc(C)[nH]n1)=O 95776,CCN=C1NC2CCCCCCC2N1.CCCC[SH](=O)=O 95777,N1(C(c2nccc(C)c2N)=O)C2CCC1CN(C(C1(C)CCC(=O)NC1)=O)C2 95778,N1(C(c2n(COC)ncc2)=O)CC(CCNC(=O)COCC(C)C)OC(C)C1 95779,C1(N(C(=O)CCC2CCC(=O)C2)C)CCCN(C(=O)CN2C(=O)CNC2=O)CC1 95780,C1(CNC(c2ccc(O)nc2)=O)CCCCN(C(=O)CCc2cnoc2)C1 95781,C1(C2CCC2)(NCCc2ccc(NC(=O)NC)nc2)CC1(F)F 95782,c1(C(=O)NC2CC(NC(C(C=C)(C)C)=O)C2)sc2ccc(C(F)(F)F)cc2c1C 95783,C1(C(N(C)CC2CN(C(C=CCC)=O)C2)=O)(CO)CCCC1.c12cnc(s1)[nH]2 95784,c1(OC)ccc(F)cc1SCC(=O)NC1CC(C)N(C(c2cnncc2O)=O)C1 95785,Cc1cccc2[nH]c(C(N3CC4CN(C(C5(C)CC5C)=O)CC4C3)=O)cc12 95786,C1(NC(c2n(CC)ccc2)=O)CC2CC(C1)N(C(=O)C(Br)=C(C)C)C2 95787,C(C(=O)NNc1cccc(C(F)(F)F)c1)Nc1cn(CC2OCCN(C)C2)nc1 95788,C1(NC(C(CCCC)O)=O)CCN(C(=O)CN2CCC(C)(C)C2)CC(O)C1 95789,N1(C(c2cnc(CC)nc2O)=O)CCOC2CN(C(c3n[nH]c(C4CC4)n3)=O)CC12 95790,Cc1nn2c(c1CNC(C1(n3nccn3)CC1)=O)CN(C(c1ccco1)=O)CC2 95791,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCOC2)CCC2(CC(=O)N(C)C2)C1 95792,c1(OC)ccc(CC(=O)O)c(C(=O)OC(C)C(N2CCCC2C(F)(F)F)=O)c1 95793,Cc1cc(C(=O)NC2CCN(C(c3cncc(C(F)F)c3)=O)C2)c(F)c(Br)c1 95794,N1(C(c2c(C)c[nH]n2)=O)CC(NC(C2CC23CC3)=O)CC1(C)C 95795,CC1CCC(C(C)C(=O)NCCN(CCCN(C)C)C(=O)Cc2cnnn2C)CC1 95796,c1(C(N2CCC(NC(c3cc(Cl)cc(F)c3F)=O)C2)=O)cccc2cc[nH]c12 95797,CC1=C(C(=O)N(C(CNC(=O)C(CO)N(C)C)C2CC2)C)S(=O)(=O)CCO1 95798,C1(CN(C)C(C2C3CNC(=O)C23)=O)CCCN(C(=O)COc2cnn(C)c2)C1 95799,C1(OC)CCC2(C(=O)NCC(C3CCCC3)NC(c3scnc3C)=O)CCC12 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95887,C1(NC(C)=O)CC(NC(c2ccc(OC(F)F)cn2)=O)C1(C)C 95888,c1(C(=O)NC2C(NC(C3(C#N)CCCO3)=O)COC2)cc2ccncc2s1 95889,S(=O)(=O)(CCCCF)N1CC2C(N)(CC(=O)OC(F)F)C2C1 95890,CC#CCC(C(=O)NC(C)(C)CCCO)NC(=O)OC.C(C)(C)(C)O 95891,c1(NC2(CC)CC2)cc2cccnc2c(Br)n1.S1(=O)(=O)c2cccnc2N1 95892,N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(C1CC2(CCCC2)C1)=O 95893,C1(C(N(CCF)CC)=O)C2CCCC2CN1C(c1cnn2cccc2c1)=O 95894,N1(CCC(=O)NC(CC(C)NC(Cc2ccn(CC)n2)=O)C)CCN(C)CC1 95895,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C(C)=C3CC3)C2)C1 95896,Cc1coc(C(C)C)c1C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1 95897,N1(C(C2C(OC)C2)=O)C2CCC1C(F)C(NC(=O)CCc1cnccn1)C2 95898,CC1C(=O)CCC(C(=O)NCC(N2CCN(C(c3ccnnc3O)=O)CC2)=O)C1 95899,c1(NC(=O)COc2cc(F)ccc2F)ccc2c(c1)OCO2 95900,CC1(C)C(NC(=O)C2=CCSC2)CCN1C(=O)CCc1ccc(F)nc1 95901,Cc1ccc(C(C(=O)NCc2conc2C)N(C)Cc2ccccc2F)c(F)c1F 95902,c1(C(C)CNC(=O)Nc2sncc2Br)cccc(C(F)(F)F)c1 95903,C(c1ccc2c(c1)OCO2)=CC(=O)NC12CC(CNC(=O)CC3(CO)CC3)(C1)C2 95904,C(C(C)C(=O)NC1CCC1NC(=O)C(C)(C)C)OCC 95905,N1(C(CC2CN(C(C)=O)C2)=O)CC(O)(CNC(=O)COC2CCOC2)C1 95906,Cc1ccc(C)n1CCN(C(=O)Cc1cscn1)Cc1ccc(F)cc1 95907,c1(C(=O)NC(CC(C)C)CNC(C2CC2C#N)=O)c[nH]c2c(F)cccc12 95908,N1(CCc2ccc(=N)[nH]n2)Cc2cccnc2N2CC(O)CC2C1 95909,N1(C(Cn2cc(CNC(C(C)CN(C)C)=O)nn2)=O)CCn2nccc21 95910,C#CCCCC(=O)NC1CCC(CCNC(c2ccc(Cl)cc2)=O)C1 95911,c1(C(=O)NCCC2CCN(C(C3CCC(F)C3)=O)C2)cc(-n2ccnc2)ncn1 95912,C1(NC(C(CC)N(C)C)=O)CN(C(c2nc(C)c(C)s2)=O)CC(F)(F)C1 95913,C1(OC)CC(NC(=O)C=CC(C)C)CN(C(=O)CN2CC=CC2)C1 95914,C(=O)(C1CCc2cc(Cl)ccc21)NC1OCCN(C(C(C)OCCN(C)C)=O)C1 95915,CS(=O)(=O)C(CNC(=O)Cc1cc[nH]c1)CNC(C1(F)CCCOC1)=O 95916,O=C(CCCn1cccc1)NC(C1CCCC1)CNC(=O)C(F)n1cccn1 95917,c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)C)cccc2[nH]cc(Cl)c12 95918,CC1(C)CC(CC(=O)NCC(N2CC(N)C2)=O)CO1.C1(C2CC2)(C)CC1 95919,Cc1cc(C(=O)NC2(C)CN(C(c3cc(C4CC4)nnc3O)=O)C2)cc(O)n1 95920,N1(C(c2c(C)cns2)=O)CCN(C(=O)CCCCC#N)CC1C 95921,C1(CNC(C2C(C(C)C)OCC2)=O)C2CN(C(c3c(N)cnn3C)=O)CC12 95922,c1(C(N2CCC(NC(C3CC(CCC)OCC3)=O)C2C)=O)c(F)cc(O)cc1F 95923,C(=O)(C(C)(C)CSC)NCC1C(C(N(C(CC)CC)C2CC2)=O)CC1 95924,N1(CC)CCC(C2(NC(=O)CCC(C)(C)F)CC2)CC1 95925,C1(C(N(CCCOCCNC(c2ccc(C)cc2)=O)C)=O)CCC2(CCC2)C1 95926,n1(CC)[nH]c(C(=O)NCCOCCCN(C)C(C2CC2C(C)C)=O)nc1=O 95927,C1(C(N(C2(COC)CC2)C)=O)CN(C(=O)C(=O)NOC)CCN1C 95928,C12(CNC(C(c3ccccc3)OCC)=O)CC1CN(C(=O)Cn1cc(N)cn1)C2 95929,Cn1ncc(C(=O)O)c1CNCc1c[nH]nc1-c1cccc(Br)c1 95930,C(=O)(C(C)CC(F)(F)F)N1CC(C)(C(=O)NCCCc2cc(C)no2)C(C)C1 95931,CC1(C)CC(C(N2CC3CCC3(CCNC(=O)CN(C)C3CC3)C2)=O)C(C)(C)O1 95932,CCCC(C)CC(=O)NC(C)(C)CNC(C1SCCS1)=O 95933,c1(C(=O)NC2C(CC(=O)NC(C)CO)CC2)ccnnc1O 95934,C1(C(=O)NC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)CO)CC2(CCCCC2)CO1 95935,n1(CC)cnc(C(N2CC(O)(C(C)NC(=O)C(O)CN3CCCC3)C2)=O)c1 95936,c1(C(N2C3(CNC(C4(CC)CCCC4)=O)CC(C2)C3)=O)ccc2nc(C)cn2c1 95937,N1(C(COCCCCC)=O)CC(NC(=O)CN(C(=O)COC)C)CCC1C 95938,C1(C(C)NC(=O)Cc2cscn2)CCCN(C(c2cn(C)nc2C(F)F)=O)C1 95939,N1(C(CC2(COC)CCC2)=O)CC2CC1CN2C(c1cc(OC)cs1)=O 95940,CC1CC(CNC(c2ccn(C)n2)=O)CN(C(=O)CCOC2CCCOC2)C1 95941,C(C(=O)N(OC)C(C)CC)N(C(=O)NC1CCC(C)(COC)C1)C 95942,C1(CNC(C2(CCC)CC2)=O)(OC)CCN(C(c2ccc(CC)cc2O)=O)CC1 95943,c1(SC(C(=O)NCCCCCN(C(c2cc(C)no2)=O)CC)C)ccccn1 95944,c1(C(N2C(CNC(C(C)(C)CF)=O)CC2)=O)ccc(Cl)c2ccccc12 95945,C(=O)(C(C(C)C)c1cnc(C)s1)NC(CC(C)NC(C=CC)=O)C 95946,Cc1c[nH]cc(C(=O)NCCC2(O)CCN(C(c3ccc(Cl)cc3N)=O)C2)c1=O 95947,c1(SC)c(C(=O)N(C)CCN(C(C2CC2C2CCC2)=O)C(C)C)cccc1F 95948,CC1(C)C(CO)CN1C(=O)C(c1ccoc1)NC(=O)C(O)CN1CCCC1 95949,CCCCC(C(=O)NC)NC(C1CCOC1C(=O)NC1(CC)CCOCC1)=O 95950,N1(C(CCCC(C)=O)=O)CCCC2(C1)C(NC(c1ccc(CO)o1)=O)CCN2C 95951,CCCCN=C(NC(C)CC)N1CCC(OCC)C1.C12CC3(CC3)CN1S(=O)(=O)C2 95952,c1(C(=O)NC2CC(F)(CNC(c3cc(CC)nn3C)=O)C2)cc2ccccc2o1 95953,CC(C)CC(C)(CNC(C1CC(CCO)C1)=O)NC(=O)C(N1CCCCCC1)C 95954,C12CC(C1)C(=O)N2.C(=O)(CCn1ccnc1)NCCNS(C)(=O)=O 95955,N1(C(c2nc(OC)c(F)cn2)=O)CCN(C(=O)Cc2ccsc2C)C(C)CC1C 95956,c1(C(=O)NC(CNC(c2cc(OC)ns2)=O)C2CC2)[nH]c2ccc(F)cc2c1C 95957,c1(CNC(=O)CC(C)NC(=O)C(F)C2CCCC2)ccccc1O 95958,C1(C(N2CC(CN(C)C)C2)=O)CCC2CCC1N2C(=O)CCc1cn(C)cn1 95959,C#CCC(CC#C)C(=O)NC(C)(CC)CCNC(c1ccc(Br)c(C)n1)=O 95960,C(CCC(=O)NCCCCn1cc(CC2CC2)nn1)C1C(C)C1 95961,CCCC(C)(C)C(=O)NCC1CCCN1C(c1cnn(C2CCOCC2)c1)=O 95962,C(=O)(C(O)C(F)(F)c1ccccc1)N1CCCC(CCNC(=O)CC(F)(F)F)C1 95963,C(CO)(CCCCNC(c1ccc(F)c(SC)c1)=O)NC(C(CCOC)C)=O 95964,N1(C(CC(CNC)C(F)(F)F)=O)CCC(C2CC(NC(=O)C(C)OC)C2)CC1 95965,C1(CNC(C2CCN(C(c3ccc(C)s3)=O)C2)=O)COCCN1C 95966,c1(COc2ccc(C(CO)C(=O)O)cc2)c(F)ccc(Cl)c1F 95967,C1(CC)(NC(C2CNC(=O)O2)=O)CCN(C(=O)COc2ccc(C)c(C)c2)CC1 95968,C=CCC(C)(C(=O)NCc1csc(CNC(C2CCCCC2(F)F)=O)n1)N(C)C 95969,C1(F)(C(=O)NCC2C3CN(C(c4cc(C)n(C)n4)=O)CC32)CCN(C)CC1 95970,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(F)C2)c[nH]c2cc(C)ccc12 95971,N1(C(C2CC(=O)CC(=O)C2)=O)CC(NC(=O)CNC(=O)NC2CC2)C2CCCC12 95972,c1(OC)ncc(Br)cc1C(=O)NCC1(C)CN(Cc2csc(C)c2)C1 95973,Cc1ccccc1C(C)C(=O)NCCOCCN(C1CC2CC2C1)C 95974,C1(NC(C(CC)N(C)C)=O)CCN(CCC2CCOCC2)CC1O 95975,c1(SC)nc(C(=O)N(C)CCOCCNC(=O)C(C)C(C)C)cc(O)n1 95976,c1(C(N(CC(C)NC(=O)C(C)Cc2cnco2)C)=O)ncccc1N 95977,C12(NC(CS(=O)(=O)NC)=O)CCCCCC1N(C(c1ccc(C)o1)=O)CC2 95978,C1(CC(N2CC(CC(C)NC(c3cc(Br)c[nH]3)=O)C2)=O)CNC(=O)C1 95979,C1(CNC(c2ccc(C3COC3)cc2)=O)CCN(CCNC(N)=O)CC1 95980,c1(NCC2CC(C(C)C)C2)ccc(S(=O)(=O)NCC2CCCC(C)(C)O2)cc1Br 95981,C(C(C)(F)C(C)(C)F)NC(CC1CC(C)N(C(=O)CNC(N)=O)C1)=O 95982,CC1CC(CC(=O)Nc2cc(CC#N)cc(Cl)c2)CCCC1 95983,N1(CC(C)(C)F)CCN(c2cc(N3CC(OCC4CC4)C3)ncn2)CC1 95984,N1(C(=O)NC2C(C)NCCC2)CCOC2(CCS(=O)(=O)C2)C1 95985,CCC(CC)CC(=O)NCCC1CC(F)(F)CN1C(=O)C1=C(Cl)CCC1 95986,c1(C(N2C(CNC(CC=C)=O)CC2)=O)cn(CCCCc2ccccc2)nn1 95987,C1(CNC(Cc2cc(C)sc2)=O)(NC(=O)CC2CCCN(C)C2)CCN(C)C1 95988,c1(CC)cnc(C(C)(C)CCCNC(=O)CCOCCOC)[nH]1.N12CC(C1)CC2=O 95989,C1(COCC(=O)N(CCCNC(=O)COC2CCOC2)CCO)CCCCO1 95990,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)cnc2ncnn2c1C 95991,N1(C(COCCOC)=O)CCCCC1CC(=O)NC(C)C 95992,N1(C(Cc2ncn(C)c2)=O)CC=C(C(=O)NCCC2CCCC3CC23)C1 95993,CC(CC(=O)N1CCCCC1C1(NC(=O)C(=Cc2c[nH]cn2)F)CC1)C(C)(C)C 95994,c1(N2CCC(C)C(F)(F)CC2)nc(=NCC2COCC2(C)C)[nH]c2c1CCCC2 95995,C(Cc1ccoc1)(C(=O)NCCC(O)C1CC1)NC(=O)Cn1cncn1 95996,CC(C)CC(=O)NC(C)CC(C)NC(=O)Cn1cncn1.C1(=O)CN1 95997,NC(=O)CC(O)C(=O)NC1CCCCC1CNC(c1ccc(-c2ccco2)[nH]1)=O 95998,CC1CCn2ncc(C(N3CCC(C)C3CNC(=O)C(O)c3ccsc3)=O)c2C1 95999,C(=O)(C(F)(F)C1(O)CCC1)NCCCCN(C(C(N1CC(C)C1)C)=O)C 96000,c1(C(N2C(CNC(C3COCCO3)=O)CC2)=O)cnc2[nH]cnc2c1 96001,CCCCC(O)C(C)C(=O)NC1CC(N(C)C(c2c[nH]nc2Cl)=O)C1 96002,N1(C(CC(CC)C)=O)CC2CC(NC(=O)C(C)Cc3c(C)noc3C)CC2C1 96003,c1(C(N2CC(C(C)NC(CCC(=O)NCC)=O)OCC2)=O)cc(Cl)c(N)c(Cl)c1 96004,C1N=C2N=c3c(cnn3C)=C(N2)NN(C)CC1.C1CCC(OCC(F)(F)F)C1 96005,N1(C(CC2C(C)OC(C)C2)=O)CC2(CCCCN(C(C3CCCS3=O)=O)C2)C1 96006,c1(N2CC3(C(CO)CN(C(C(CC)OCC)=O)C3)C2)cc(C)c([N+](=O)[O-])cc1F.C(C)C 96007,CC(CN=c1[nH]c(N2CC3CC=CCC3C2)nc(=N)[nH]1)N1CCCCC1 96008,c1(C(=O)NCC2CC(CNC(C=COCC)=O)OC2)ccc2ncnc(C)c2c1 96009,c1(CN(CCC)C(=O)NC2(CC(F)F)CCCO2)c(C)noc1C 96010,c1(C(=O)NCCC(CNC(c2ccc(CC)cc2)=O)OC)ccc2nccn2c1 96011,Cc1cnc2ccc(C(N3CCC(C)C(CNC(C4CCCO4)=O)C3)=O)cn12 96012,C1(NC(C2(C(=O)OC)CC2)=O)CN(C(=O)CNC2CC2)C2(CCOC2)C1 96013,N1(C(C(CCC)(C)O)=O)CCCN(C(c2cnc3sccc3c2)=O)CC1 96014,C(=O)(C#CC1CCOCC1)N1CC(NC(C2C(OCC)C2)=O)C(CN(C)C)C1 96015,C1(NC(CC(C)=CC)=O)CC2CN(C(=O)Cn3cncn3)CC2C1 96016,N#Cc1ccc(Cl)c(C(=O)NC2C=CC(CNC(c3coc(Cl)n3)=O)C2)c1 96017,Cc1[nH]cc(C(N2CCC(C(C)NC(=O)C(C)OC(C)(C)C)CC2)=O)c(=O)c1Cl 96018,C12(NC(C(C)(F)F)=O)CC3CC(C1)CC(CNC(c1cc(O)nn1C)=O)(C3)C2 96019,Cc1ccc(C(C)(C)C(=O)NCC2(c3ccc(Cl)cc3)CCCC2)cn1 96020,CC1CCCCN1CC(c1ccc(F)cc1)C1CC(F)(F)C1.c1(=O)c(=O)[nH]1 96021,C(CN=c1nc(Cl)[nH]c(C)c1C#N)C1CCCN(C(c2cc3n(c2)CCOC3)C)C1 96022,N1(C(=O)CC2CC2)CCCCC1C1CCN(Cc2nc(C(C)(C)C)ns2)CC1 96023,Cc1cn2cc(C(=O)N(CCNC(C3CC3(C)C(F)F)=O)C3CC3)nc2s1 96024,C(=O)(C(C)(C)CC(=O)NC1CCCCC1CNC(=O)C(C(C)C)N(C)C)OC 96025,CCC(CC)(CO)C(=O)NCCOCCCN(C)C(c1cn(C)ccc1=O)=O 96026,C1(CSC)COC(C)CN1C(C1CCS(=O)(=O)CC1)C(=O)Nc1cccc(OC)c1 96027,c1(COCC(=O)N(CC(C)N(C)C(c2cnn(CCF)c2)=O)C)ccccc1F 96028,N12CCCC(C1C)C2.C(=O)(CS(C)(=O)=O)NCc1nnc(OCC)s1 96029,c1(C(=O)NC2(CNC(=O)CC3(O)CCOCC3)CC2)cnc2[nH]nc(O)c2c1 96030,N1(C(CSC)=O)CC2CCCN(C(c3c(C)nn(C)c3-n3ccccc3=O)=O)C2C1 96031,N1(C(C2(C=C)CCN(C(=O)CC(=O)OC)C2)=O)CCc2nc(O)[nH]c2C1 96032,C(=O)(C1=CCCOC1)N1C(CCNC(C2CC2(Cl)Cl)=O)CSCC1 96033,S(=O)(=O)(c1cccc(F)c1)NCC(=O)N(C)CCc1ccc(F)cn1 96034,c1(C(C)C)nc(NCCN(C)C)cc(N2CCC(OCc3nc[nH]n3)CC2)n1 96035,N1(C(C2=C(C)CCCC2)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C2COCC12 96036,Cc1cc(=NCC2(C)CC2(F)F)[nH]c(=NCCN2CCCC2)[nH]1 96037,c1(C(C)NC(N2CCN(C(C(=O)OC)c3ccco3)CC2)=O)cc(F)ccc1F 96038,CN1CCC(C(=O)N(C)CCN2CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)C1=O 96039,C1(CCC)CCCCC1CC.C12CC(C1)NC(=O)CSCC(=O)N2 96040,N1(C(CCOCC#C)=O)CC2CCCC(NC(=O)CNC(=O)OC)C2C1 96041,N1(C(CCNC(=O)NC)=O)CCC(CNC(c2ccc(C(N)=O)cc2)=O)C(C)C1 96042,C1(NC(CNC(C(C)SCCCC)=O)=O)CCCN(N2CC(O)C2)C1 96043,c1(CCC(=O)NCC(CC)NC(=O)C(C2CCCC2)SC)cccc2c1OCO2 96044,C(=O)(C1=CCCC1C)NC1CCC(CC(N2CC(CC(=O)OCC)C2)=O)C1 96045,c1(C(N2CCC(CCNC(C=COCC)=O)CC2)=O)oc2c(c1C)C(=O)CCC2 96046,n1(CC=C)c(N2CCC(C)(C(=O)OCC)C2)nnc1C1CC1(F)F 96047,C1(CNC(C2CC(=C)C2)C)(Cc2ccccc2)CCOCC1 96048,c1(C(=O)NCc2cc(N(C)C(C3CC(O)C(O)C3)=O)ncc2)cnn2c1CCC2 96049,c1(C(=O)NCC(CNC(C2(OC)CCOC2)=O)(C)C)cc(Br)ccc1C1CC1 96050,C1(NC(C(=O)NCCC(N)=O)=O)CCCCN(C(=O)CSC2CCS(=O)(=O)C2)C1 96051,N1(C(CCCN(C(C)C)C)=O)CC(C)(C)CC1CNC(c1[nH]nnc1C1CC1)=O 96052,N1(C(c2cn(CC)nn2)=O)CCCCC1C(C)NC(c1cnc(S)n1C1CC1)=O 96053,N1(N2CCCC(C=O)C2)CCC(C)(CNC(=O)COC2(C)CCOC2)CC1.CC=O 96054,c1(C(N2CCC3(NC(Cc4c(C)noc4C)=O)C(C2)C3)=O)ccc2nn[nH]c2n1 96055,c1(CCC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96056,C1(OCC)CC2CC(c3nc(-c4cccc(-c5onc(CC)n5)c4)no3)CC12 96057,c1(C(N2CCC(OCCNC(C(CC#C)C)=O)C2)=O)n[nH]c2c(C)cccc12 96058,c1(-c2ccc(CNCC(=O)NC3CN(C(C=NOC)=O)C3)s2)cccc(F)c1 96059,c1(C(=O)NCC2N(C(C(CC)C)=O)CC(F)C2)ccc2ccc(C#N)cn12 96060,C(c1cccnc1)=CC(=O)N(C(C)CNC(c1cnc(C2CCCO2)s1)=O)C 96061,C(=O)(C1=CC2C=CC1C2)N1CC(COC)(NC(=O)C(C2CCC(=O)N2C)C)C1 96062,c1(-n2c(Cc3onc(C)n3)nc(C3CCC(C)CC3)n2)cccc2ccccc12 96063,c1(C(=O)NCC2CC(NC(C3=C(C)OCC3)=O)C2)cccc2c1CCCC2 96064,n1(CCC)cc(C(=O)N(CCN(C(=O)C(C)n2cccc2)CC)CC)c(C)n1 96065,C1(C(=O)NCC2CCCC(NC(c3nn(C)cc3C)=O)C2)(SC)CC(F)(F)C1 96066,CCCC(CCC)CC(=O)N(CCNC(=O)C(C)NC(=O)C(C)(C)C)C1CC1 96067,CP(C)(=O)CCC(=O)N1CCCCC(C(=O)NC2CC3(CC3)C2)C1 96068,CCC(C)(F)C(=O)NC1CC(CO)N(C(=O)CCc2ccc(O)nn2)C1 96069,N1(C(CSCC(C)C)=O)CCC(CC(=O)NCC2CCC2)C1(C)C 96070,c1(CCC(=O)NC2C(CNC(Cc3cc(C)sc3)=O)C2)cnc2ccccc2c1 96071,N1(C(C#CC2(CC)CC2)=O)CCOCC(CNC(c2c(CC)cccc2C)=O)C1 96072,C(=O)(C1CC(=O)Nc2ncn(C)c21)N(CCNC(COC(CC)CC)=O)C1CC1 96073,c1(N(C)C)cc(Cl)cc(CNC(=O)C(=O)NC2CCOC(C(F)(F)F)C2)n1 96074,C1(C(=O)NCCOC2CCN(C(=O)C(F)(F)c3ccccn3)C2)CCNC(=O)C1 96075,c1(SC)ncc(C(=O)NC(C2CC(NC(=O)C(F)C(C)(C)O)C2)C)c(O)n1 96076,c1(SC)ccc(C(N2CCC(C(C)NC(=O)C=C3CCOCC3)C2)=O)cc1 96077,N1(C(C2(OCC)CCCC2)=O)CCCCC(Nc2ncc(C)c(C)n2)C1 96078,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96079,C=CCCC(C(=O)NC1CC(CO)(CO)C1)NC(c1ccc(C)nn1)=O 96080,c1(C(N2CC(NC(C3CCN(C(CC)=O)C3)=O)C(C)C2)=O)cc2ncccn2n1 96081,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C=CC3CCCO3)C(CCO)C2)=O)cs1 96082,c1(C(=O)NC2CC(NC(C3C(C)OCCC3)=O)C2)ccc(P(C)(C)=O)nc1 96083,N1(C(CC(C(C)=O)(C)C)=O)CC2CC(C1)N(C(=O)CCn1cnc3ccccc13)C2 96084,c1(C(N2CC(C)C(NC(c3ccc(CC4CC4)s3)=O)C2)=O)coc2c1CSC2 96085,N12CCCCC1C(=O)N2.C(C)(C(=O)NC(C(=O)OC(C)C)C1=CC=C1)NC 96086,C=CC(C)(CC)C(=O)N1CCC(N(CCO)C(c2ccc(=O)oc2)=O)CC1 96087,c1(C(N(C2CN(C(=O)CC3CC(F)(F)C3)C2)C)=O)ncsc1C(F)(F)F 96088,c1(N2CC(NC(Cc3ccc(OC)nc3)=O)C(C)C2)cc(C)ncc1C#N 96089,C12(C(=O)NC3C(NC(c4ccnc(S)c4)=O)CC3)CC(C1)C(C(F)(F)F)O2 96090,c1(C(N2CC(NC(CC=CCC)=O)CC2(C)C)=O)cnn2c1CC(C)CC2 96091,C#CCCCC(=O)NC1(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 96092,CCC(C(=O)NC(c1ccccc1)C(=O)Nc1ccsc1)NC(C)=O 96093,C1(CNC(c2cc(C(C)(C)C)no2)=O)CCN(C(C23CCC(CC2)C3)=O)CC1(F)F 96094,c1(OC)cc(CC(=O)N(C)CC2CN(C(C3CC34CC4)=O)CC23CC3)ccc1C 96095,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96096,C(=O)(C(Cc1ccccc1)C1CC1)NCC(C)(C1CCC1)NC(c1cocn1)=O 96097,C(=O)(CC1OCc2ccccc21)NCCCCNC(C(c1n(C)cnc1)O)=O 96098,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 96099,N1(C(=O)C=C2CCOCC2)CCC2CN(C(C3(C4CCCOC4)CC3)=O)CC2C1 96100,CC(C)C(C)C(=O)N1CCN(CCN(C(=O)CC2CCCC2)C)CC1 96101,C(=O)(C1CCc2nnc(C)n21)NCc1scc(CNC(C(CC=C)(C)C)=O)n1 96102,C1(C(N2CCC(Cn3ccnn3)C2)C(=O)NC(CC)(C)C)CC12CCCCC2 96103,Cc1cccnc1CNC(c1c[nH]nc1CCNC(C1OCCC1C)=O)=O 96104,N1(C(=O)OC(C)(C)C)CC(F)(NC(c2ccc(F)cc2)CO)C2(CCC2)C1 96105,CCCCCC(O)CC(=O)OCC(N1Cc2ccccc2C1)=O 96106,C1(CCC)CN(C(=O)Cn2cc(Br)c(C)n2)CCN1C(=O)Cn1cnnn1 96107,C(=O)(C(O)CC(F)(F)F)NC1CC(C)(C(=O)NC(C)Cc2ccnn2C)C1 96108,C(=O)(CCCCC(OC)OC)NCC(C)(C1CC1)NC(CS(CC)(=O)=O)=O 96109,c1(C2C(C(=O)NC(CC)CNC(c3nc(Cl)sc3C)=O)C2)ccc2c(c1)OCO2 96110,C(=O)(C1CCCc2nncn21)NC(CC)(CC)CCNC(=O)CC(C)SC 96111,CC1(C)CCCC(C(N2CCCC2CNC(C2(C(N)=O)CC2)=O)=O)C1 96112,CON(C(=O)C=CC1CCN(C(=O)CC2COCC(C)O2)CC1)C1CCCC1 96113,C(=O)(C(C)(CC)C(=O)OCC(=O)C1CC1)OCC.C12(c3ccccc3)CN(C1)C2 96114,C(=O)(C(CCNC1(c2ccccc2)CCC1)C(C)(C)C)OCC 96115,n1(CCCC)nnnc1C(c1n[nH]cc1CC)NCc1cc(Br)cs1 96116,C(=O)(CCC(C(C)C)NC(=O)C1=COCC1)N1CC=C(COC)CC1 96117,CCS(=O)(=O)CC(C)NC(=O)C(N1CCCC(N(C)C)CC1)=O 96118,C1(CC(=O)NC2(CO)CN(C(C(c3n(C)ncc3)O)=O)C2)CC2(CCC2)CCO1 96119,c1(C(=O)NC(C(C)NC(CCCCOC)=O)CO)c2ccc(F)cc2nn1C 96120,c1(C(=O)NC(C(=O)NCC(COC)(C)C)C2CC2)cc(=O)cc[nH]1 96121,c1(OC)cccc(C(F)(F)C(=O)NCC(O)CN(C(=O)CC2CC(CF)C2)C)n1 96122,Cc1noc(C(F)(F)Cl)c1C(=O)N(CCCCNC(=O)CCC1CCN(C)C1)C 96123,c1(C(=O)NC(C2CCOC2)CNC(=O)CCn2cccn2)cccnc1O 96124,N1(C(CC2(OCC)CCC2)=O)CCOC(CNC(c2nnc(S)n2C)=O)C1 96125,C12(OC)CCCCC(C(=O)N(C(CNC(C3CCS(=O)(=O)N3)=O)C3CC3)C)(C1)C2 96126,c1(OC)cc(C(=O)O)ccc1CNc1ccc(-c2nncs2)cc1 96127,C1(CC(=O)NCC2CC2F)CCC(O)C1.C1CCC(=O)N1 96128,C1(C(=O)NCCc2nncs2)(CNC(=O)Cc2sccc2Cl)CCCO1 96129,c1(CCC(=O)N(C)CCOCCNC(C2CC2C(F)F)=O)ccccc1Br 96130,CCCCCCCC(F)C(=O)NC(C1CCCN1C(C1CC(F)(CF)C1)=O)(C)C 96131,n1(CC)[nH]nnc1=NCC(COC)NC(=O)CC1CC(O)C12CCC2 96132,N1(C(CC)C(=O)NCCC(C)NC(=O)Cn2nnc(=N)[nH]2)CCN(C(C)C)CC1 96133,C1(C(=O)NC2C=CCN(C(c3cc(F)ccc3Cl)=O)C2)CCn2c(O)nnc2C1 96134,c1(C(=O)NCC)cccc(NC(c2ccc(-n3nc(C)cc3C)nc2)=O)c1 96135,Cc1cc([N+](=O)[O-])c(S(=O)(=O)N2CCC(c3c(C)noc3C)CC2)cc1F 96136,C1(CCC)CN(C(C2(n3cnnn3)CC2)=O)CCN1C(C12CC(C#N)(C1)C2)=O 96137,c1(C(N(C2CCN(C(c3ccc(OCC)cc3)=O)C2)CCC)=O)c[nH]ccc1=N 96138,N1(C(c2cc(CC)on2)=O)CCC(NC(C2(C)CCCOC2)=O)C(F)C1 96139,C(=O)(CC(C(F)(F)F)N1CCOCC1)NCC(C)NC(c1cc(Cl)ns1)=O 96140,CC1CCN(CC(=O)NCCC(C)(C)NC(=O)C(F)CC2CCC2)C1 96141,C=CC(C)(C)CC(=O)NC(C)CCN(C)C(c1cc(Cl)ncc1NC)=O 96142,C(CCC(=O)c1c(C(=O)NCC2CCC(N)C2)scc1)OCCC.C(C)(=O)OC 96143,N1(C(CCc2cc(C)[nH]n2)=O)CCOCC1CCNC(=O)CCOC1COC1 96144,Cn1ccnc1C(=O)NC(C(=O)NCC1(O)CCSC1)C1(C)CC1 96145,C(CCCC(=O)NCC#CCNC(=O)C(c1ccccc1)SC)SC 96146,CC(O)C(C(=O)NCC(c1cccs1)O)NC(C1CC(=O)C1)=O 96147,Cc1nc(C(=O)NCC2(CNC(=O)CC(C)(C)C)CCCC2)c(C)c(C)n1 96148,N1(C(COCC(=O)OC)=O)CCC2(CC1)CC2(C)C(N1CCC(O)(CO)CC1)=O 96149,CC(C)(CN1CCCC(C(=O)NCCSc2ccccc2Cl)C1)C(F)F 96150,C1(CNC(CCC(C)(F)F)=O)CN(C(c2cnc3c[nH]nc3c2)=O)CCC1(C)C 96151,c12ncc-1[nH]2.n1(CCCNC(C2C(CC)C2)=O)cc(C(C)=O)nn1 96152,c1(CC)ccc(C=CC(=O)NC2CCCN(C(=O)CN3CCCCC3)C2)cc1 96153,C(=O)(CC(C)(C)C(=O)N1CC(NC(C2CCC(OC)CC2)=O)C(CO)C1)OCC 96154,C1(CNC(COCCC=C)=O)CCC(C)(C)CN1C(C1CCCCS1)=O 96155,CCCCN=C(Nc1c(CC2CC2C)cc(OC(F)F)cc1)NC1CC1 96156,C1(c2cn(CCOC)nn2)CCCN(C(C2CC3(CO)CC2C3)=O)CC1 96157,C(C)(C)(CCC(=O)N1CCCC(CCC(=O)NC2(CSC)CC2)C1)OC 96158,N12CCC(F)CC1C(=O)NCC(CC)C2=O.c1(CN(C)C)ccnn1C(C)C 96159,C(=O)(C(C)CC(F)(F)F)NCC(CCC)NC(=O)C(COCC)N=[N+]=[N-].C(C)=O 96160,C=C(C)CCCC(=O)NCC(C)(C(C)C)NC(c1coc(C(C)OCC)n1)=O 96161,CC1CN(C)CCC1(c1nnnn1C)NCc1ccc(Br)cc1Cl 96162,C(=O)(CC(C)CC(F)(F)F)NCC1N(C(c2cnc(SC)s2)=O)CC(O)C1O 96163,N1(C(C2C(CC)C2)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(C(F)F)n1)=O 96164,C1(C)(CN(CCN2CCN(C(CCC)=O)CC2)C)C2Cc3ccccc3C12 96165,N1(C(CCNC(=O)OCC)=O)CCC(OC)C(SCC(C)(C)C)C1.C1(=O)CN1 96166,N1(C(c2cccc(C)c2C)=O)CC2CCC1(CNC(c1[nH]cnc1C)=O)CC2 96167,c1(NC(CCCCOCCCCSC)=O)ccc(Oc2ccc(F)cc2)c(F)c1 96168,CC1(C)C2CC(C(=O)NC3(C)CN(C(=O)CNS(=O)(=O)C4CC4)C3)CC12 96169,c1(OCC)nc(C(N2CC3CC2CCN3C(=O)C=NOC)=O)cc2ccccc12 96170,N1(C(c2nccc(N)c2Cl)=O)CCC(NC(c2ncc(F)cn2)=O)C(CO)CC1 96171,C(C#CC#CCO)NC(C1CCC(NC(N2CCCC2)=O)C1)=O 96172,C1(NC(CC2N(C(C)=O)CCC2)=O)(CN(C)C)CCN(C(=O)CNC=O)CC1 96173,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCN(C(=O)C(O)CC(C)C)C(C(C)C)C1 96174,c1(N2CCN(CCCC)CC2)nc(N(CCC(C)F)C)nc2c1CCC2 96175,CCC(C)(C)C(C(=O)NCC1(CNC(c2nccn3nccc23)=O)CCCC1)OC 96176,Cc1ccc2nc(C)c(C(=O)NC3CCN(C(c4ncccc4Cl)=O)C3)cc2c1 96177,c1(NC)c(C(=O)NCCC(C)NC(c2c[nH]c(Br)c2)=O)sc2nccnc12 96178,N1(C(c2ncccc2Cl)=O)CCC(C2CC2)C1C(N1CC2(CCC2)CC1CO)=O 96179,C1(CNC(C(CNC(=O)C(c2ccnn2C)OC)OC)=O)CCCCCN1C 96180,C1(C)(CNC(C(C)(C2CC2)OC)=O)CCCN1C(C1CC2(CCC2)C1)=O 96181,C1(NC(C=C(CCC)C)=O)CC2CC1N(C(=O)CC1(O)CCCCC1)C2 96182,c1(C(CC(=O)N2CCC(C(N)=O)C2)NC(c2cnc(C)[nH]2)=O)cccc(Br)c1 96183,c1(NCCNC(CC)=O)ncc(S(=O)(=O)NC2CS(=O)(=O)CC2C)cc1Cl 96184,C#CC1CCN(C(C2CC(O)CN2C(=O)CC2CCC(=O)NC2)=O)C1 96185,C(=O)(C1=COCCC1)N1C(C(=O)Nc2cccc(C3CC3)c2)CSCC1 96186,CCC1=NOC(C(=O)NC2CC(CCNC(=O)C(C)NC(=O)CC)C2)C1 96187,Cc1cc(-c2cn(CC3(O)CN(C(C4CC(n5cnnc5)C4)=O)C3)nn2)n(C)n1 96188,CC1(C(N2CCN(C3CCCN(C(C4CCC(=O)N4)=O)C3)CC2)=O)CCNC1=O 96189,c1(C(=O)NC(C2CCOC2)CNC(c2n(C(C)C)nnc2)=O)cnc2n1CCC2 96190,N1(C(CCOC)=O)CC(C2(CO)CC2)C1.c12ccc(cc1)NC(=O)CC2C 96191,C1(NC(c2c(C)ccc(Cl)c2)=O)CCN(C)C12CCCN(C(C1(C)CC1Br)=O)C2 96192,c1(C(=O)NCC(C)(C)NC(c2ccoc2Br)=O)cnc(O)n(C2CC2)c1=O 96193,C1(C)(NC(c2n(CCC)nnn2)C2CC2(Br)Br)CCC(=O)N(C)C1 96194,CC1(C(=O)NCCCN(C(=O)CC2(CO)CCCC2)CCO)CCCNS1(=O)=O 96195,c1(C(=O)NCCN(C(C2(OCC)CC2)=O)CC)nccc(Br)c1O 96196,c1(C(=O)NCC(=C)CCNC(C23CCCCC2C3)=O)cc2c(cc1Cl)NC(=O)C2 96197,O(NC(=O)OC(=O)Cc1nc[nH]n1)CC(=O)OCC 96198,C1(C(=O)NCC2(C)CCN(C(CC(C(C)C)O)=O)C2)CC12C1CC3CC(C1)CC2C3 96199,C(=O)(C(C)(O)CCN(C)C)NCC(CC)NC(c1cccc(C(F)F)c1)=O 96200,c1(OC)cccc(C(N2CCOC(C3CC3)C2)C(=O)NC2CC2)c1C1CC1 96201,N1(C(Cc2c(C)noc2C)=O)C2CCC1(CNC(c1cccc(F)c1)=O)CC2 96202,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96203,c1(C(C(=O)NC(CNC(C(C)Cc2ccccc2)=O)CO)C)nc(F)ccc1Cl 96204,C1(C(N(CCCC)CCCC)=O)C2CCCC2CN1C(=O)C(C)n1cncn1 96205,N1(CC(=O)NC(C2CCN(C(c3cc(C(F)F)no3)=O)C2)CCC)CCC(C)C1 96206,c1(NC(C2C3CC(N)C(C3)C2)=O)c(Br)cc(Br)c2cccnc12 96207,Cc1cc(C(F)(F)F)nn1CC(=O)NC1CCCCC1NC(c1ccc[nH]1)=O 96208,N1(C(CCCOCC)=O)CC2(CCN(C(=O)C(C)CCO)CC2)C1C(C)C 96209,CC1=C(C(=O)N2CC(NC(c3ccsc3CO)=O)C(C)C2)CCO1 96210,CCC(C(=O)NC1CC(CNC(=O)C=CCN(C)CC)C1)n1ccnc1 96211,N1(C(C(C(CC)O)C)=O)CCC(NC(C2CCCN2C)=O)C12CCCC2 96212,c1(CN(C2CCCC2)C(=O)CC2CCCCCC2)ccc(Br)cc1Br 96213,N1(C(CC(CCC)C)=O)CC(CNC(c2ccnc(C)c2C)=O)OC(C)(C)C1 96214,Cc1ccc(C(N2CC(C(F)C(=O)NOc3nc[nH]n3)C2)=O)c2c1CCCC2 96215,c1(CCCC(=O)NC2(CCNC(=O)Cc3ccncc3Cl)CC2)ccc(Cl)cn1 96216,CC(C)C(CCNC(C1CCSC1)=O)NC(C1CCC(=O)N1)=O 96217,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)NC1CC2(CCC2)C1 96218,C(=O)(C1=CC2CCCC12)NCC1N(C(CSC(C)C)=O)CCN(C)C1 96219,c1(C(=O)NC2C(NC(c3cc(OC)no3)=O)C2)ccc(CCF)cc1 96220,CC1CCC(C(N2CCC(Cc3cn(CC(=O)N(C)C)nn3)C2)=O)OC1 96221,Cc1nn(C)c2nc(C(=O)N(CC(F)F)CCNC(=O)C(=O)NC(C)C)ccc12 96222,C1(C(=O)NC2C(O)C3CCCC23)CCN(C(=O)CCC2CC2)O1 96223,CCC(CCC(=O)NC(CC(=O)NC)C1CC1)NC(C1CCCS1)=O 96224,C(=O)(C(F)(F)C(O)C1CC1)NCC(C)(C)CNC(=O)C(N1CCC(C(N)=O)CC1)=O 96225,N1(C(C23CC(C)C2C3)=O)CCC2(CCC(NC(=O)C(C)(Cl)Cl)CC2)C1 96226,CCCCCC(CC)C(=O)NCC(C)(C1CC1)NC(=O)C(C)Cc1ccccc1 96227,c1(CNC(=O)NC(c2ccccc2F)C2CC(N)C2)ccnc(Cl)c1 96228,N1(CCN2CCC(CNC(c3ccc(OC)cn3)=O)C2)CCC(O)C(O)C1 96229,c1(NCc2cccc(CNC(CCCC#C)=O)c2)ncnc(C(=O)OC)c1F 96230,N1(C(c2c(OC)cnn2C)=O)CCN(C(=O)CCCNC(=O)OC)C(C)C1C 96231,c1(NC(c2n(CCCC)nnn2)c2nncn2C2CCCC2)cc(F)cc(F)c1 96232,N1(C(c2ccc(C(=O)OCC)cn2)=O)CCC(F)(C(=O)OC(C)(C)C)CC1 96233,c1(-n2c(C(c3cscc3CC)NC(C=C)(C)C)nnn2)ccccc1Cl 96234,Cc1ccc(CCC(=O)NC2C=CCN(C(C3(C(N)=O)CC3)=O)C2)cn1 96235,C1(NC(c2c(Cl)cn(CC)n2)=O)(CC)CCN(C(=O)CSc2nccn2C)CC1 96236,C1(NC(C=CC)=O)CCOC12CCN(C(C1(C)CCS(=O)(=O)CC1)=O)CC2 96237,C1(=O)CCC(CC)OCCN1C.n1(CCC)nccc1C(=O)OCC 96238,c1(OCC)ccc(NC(=S)NCCN(C)C(C2CCC23CCCO3)=O)cc1OC 96239,c1(NC(C(C)C2CC2)=O)ccccc1-n1cnnn1 96240,C(N=c1[nH]c(C(C)C)nc(C)c1Br)C1CC(NC(c2c(CC)noc2C)=O)C1 96241,c1(CC(=O)NCCn2cc(-c3c(OC)c(F)ccc3)nn2)c(F)ccc(F)c1Cl 96242,C1(C)(CC)CC(NC(=O)C(c2cnn(C)c2)NC(=O)CC(C)=C(C)C)C1 96243,c1(CN=c2scc(CC(=O)Nc3cc(Br)cnc3I)[nH]2)c(Cl)ccc2c1OCO2 96244,N1(C(CCSC)=O)CC(NC(c2cc(-c3ccncc3)no2)=O)CC12CCOC2 96245,C1(NC(CC2CCC(C)(C)CO2)=O)CC2CN(C(=O)C3=CCCOC3)CC2C1 96246,c1(CC)cc2c(N3CCC(CF)(NC(c4cnsn4)=O)C3)nc(C)nc2s1 96247,c1(OC)nsc(C(N2CCCCC2Cc2ccccc2OCC2CC2)C)c1Cl 96248,c1(OC)cc(C(N2CC(C(O)C(=O)NCCC(C)(O)C3CCC3)C2)=O)n(C)n1 96249,c1(C(N2CCN(C(c3cncc(N(C)C)c3)=O)C3C2C3)=O)cncc2sccc12 96250,C(=O)(C1CCCc2ncnn21)NC12CC(CNC(=O)COCC(F)(F)F)(OC1)C2 96251,C1(C)(NC(C2C(CC)C2)=O)CCN(C(=O)CCn2c(C)c(C)sc2=O)CC1 96252,C(CO)(CCCCNC(=O)CCC1OCCO1)NC(C(C)CN1CCCCC1)=O 96253,C(=O)(C1CCOc2ccccc21)NCCCCCCN(C(C(CC(C)C)=O)=O)C 96254,c1(C(N(C2CN(C(c3ccccc3S(C)=O)=O)C2)C)=O)cccc(C#CCO)c1 96255,CC1(C)OC2(C(=O)NCC(C3CCCC3)NC(C3CCOCC3)=O)CCC1CC2 96256,N1(C(CNC2CCC(C3CC3)C2)=O)CC2(CCC1CN1CC1=O)CC2.CS.CO 96257,S(=O)(=O)(C1CN(C(=O)NC2CCC(C)(C)CC2)C1)NC(C)C 96258,N#Cc1[nH]c(=NCC(C2CCCC2)NC(C2(O)CCSCC2)=O)sc1Cl 96259,c1(CC(C)NCCOc2ccccn2)ccncc1S(=O)(=O)NC1CC1(F)F 96260,C1(C(N(C)Cc2c(C)cnn2C)=O)CN(C(c2nccs2)=O)CCC1C 96261,C1(NC(c2cnc(C)nc2)=O)CCCN(C(C2CCCC(F)(F)C2)=O)C1C 96262,c1(C(=O)NCCCN(CCCNC(COCCCC)=O)C)cnc(C(F)(F)F)cn1 96263,N1(C(c2cc(C#N)no2)=O)CCN(C(c2c[nH]nc2C(F)(F)F)=O)CC1C1CC1 96264,CC(C)C(C(=O)NC1CCCN1)N1CCCCC1.C1C(=O)N1 96265,C(CCN=C(NNS(CC)(=O)=O)NC1CCC(=O)N(C)C1)C1OCCO1 96266,C=C1CCCN(C(C2CCOC2CNC(=O)C=CC2CCCN2C)=O)C1 96267,O=C(C#CC1CCOC1)NCC1(F)CC(NC(c2nccnc2C(N)=O)=O)C1 96268,c1(C(N2CCCC(C(C)NC(=O)CSc3ccncc3)C2)=O)cnc(Cl)cc1Cl 96269,c1(N(C)C)cc(NC2C3CN(C(C4(C(F)(F)F)CCOCC4)=O)CC23)ncn1 96270,c1(C(=O)NCC2(NC(c3ccc(F)s3)=O)CC2)cccc2cccnc12 96271,N1(C(COC2CCN(C(c3cc(C)c(=N)[nH]c3)=O)C2)=O)CC(C2CCCC2)C1 96272,C1(O)(CC#C)CC(C(=O)NC(C2CCN(C(=O)CC=C=C)C2)C)C1 96273,CC1CCN(C(=O)CCc2ccc(Cl)cc2F)CC1CNC(=O)CN(C)C(N)=O 96274,C1(NC(=O)CSc2ccccc2)CCN(C(c2ccccc2Br)=O)CC1 96275,C(=O)(CS(=O)(=O)CCO)NC1C(C)CN(C(=O)CCc2cccc(Cl)c2)C1 96276,C(CC(C)(C)CC(=O)NC1CC=CCC1C(=O)OCc1ccoc1)OC 96277,C(N=c1[nH]c(=N)[nH]c(=NC2CCCCC2n2cccn2)[nH]1)C1C(C)C1C 96278,CC(CC(=O)N1CC(O)(CNC(C2COC(=O)N2)=O)C1)CC(F)(F)F 96279,CC1OCCCC1(c1nnnn1C1CCOCC1)NC1CCCC1 96280,c1(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)cc2c(s1)CCS(=O)(=O)C2 96281,C(CN(C)C)(C(=O)N1CCCC1C(C)=O)N(C(CC)C)C(=O)OCC 96282,C1(C(=O)NCc2nncs2)CN(C(C2CC2Cl)=O)CC12CCC2 96283,c1(C(=O)NCCCNC2CCCN(CCCOC)C2)nnc2ccccn12 96284,c1(C(CC)O)ccc(C(C(=O)NCCC2CC2)N(C2CCCCCC2)C)cc1 96285,N1(C(C(C)(C)OCC)=O)CCC(N(CCO)C(c2sccc2F)=O)CC1 96286,Cc1cc(C#N)sc1C(=O)NCCC(=O)NCC1CCCCC1O 96287,C1(N2C(C)CN(C(=O)CC3CCNCC3)CC2)CCc2ccccc2N1 96288,c1(N2CCCC(CCNC(CC(C)OC)=O)C2)nc(C)nc2ccccc12 96289,C1(CNC(C(C)=CC)=O)COCCN1C(c1coc(O)n1)=O 96290,Cc1ccc(O)c(C(=O)N(C)CC2CC(F)CN2C(C2CN3CCC2CC3)=O)c1 96291,N1(C(C(N2CCCCCC2)C)=O)C2CCC1CN(C(=O)C(N)=O)C2 96292,C1(NC(CCc2n(C)ccn2)=O)CN(c2nccc(C(F)F)n2)CC(F)(F)C1 96293,C1(NC(CCc2n(C)cnn2)=O)CCN(C(C2CCCC2)=O)CCC1CO 96294,c1(C(=O)NCCN(C(C(C)=C2CCC2)=O)C(C)C)cccc2c(C)ccnc12 96295,C(CC(=O)N(C)CC1CN(C)CCO1)(C(F)(F)F)NC(c1c(C(C)C)ocn1)=O 96296,C(=O)(C1=C(Cl)CC1)N.C(C(=O)NC)(C1CCOC1)OC.C12CCC1NC(=O)C2 96297,N1(C(CCCCN(C)C)=O)CCC2C(C1)CN2C(c1cnn2cccnc12)=O 96298,C1(OC)CCC(C(=O)N(C)CCN(C(C2(Br)C(C)C2C)=O)C(C)C)CC1 96299,Cn1ncc2c(C(N3CCN(Cc4cc5ccoc5cn4)C4CC34)=O)cccc12 96300,c1(C(N2CCC(NC(C(CC)O)=O)(CF)C2)=O)c(F)ccc(F)c1N 96301,N1(C(c2cnc(O)o2)=O)CCC2CCN(C(C3CCCC(F)C3)=O)C2C1 96302,N1(C(c2n(CC)ncc2Cl)=O)CCOC(C)(CNC(C2(F)CCCCC2)=O)C1 96303,CCCC(C(=O)NC(CN(C)C)CC(=O)NCCC1=CCOCC1)C(C)C 96304,C1(N(C(=O)C(c2ccnn2C)N(C)C2CC2)C)CN(C(=O)C#CC2CC2)CC12CC2 96305,CCCS(=O)(=O)CC(=O)NC1CC(CNC(c2cn(C)nc2OCC(F)F)=O)C1 96306,N1(C(c2ccc(C)nn2)=O)CCC2CCN(C(=O)C(C)CCO)CC2C1 96307,C1(C(C)C)CN(C(=O)C(C(C)C)OC(N)=O)CCN1C(c1cccc(Cl)c1)=O 96308,c12cc(no1)NC2=O.C(=O)(C(C)OCCN(C)C)NC1C(C(=O)OC)C1 96309,Cc1ccnc(C(=O)N(CC(O)CNC(=O)C(C)OCC2CCOCC2)C)c1N 96310,N1(C(C(CSC)O)=O)CCCC(NC(=O)C(O)CCc2ccccc2)C1C 96311,Cc1cc(Br)cc(NC(C)CC2(C#N)CC2)c1 96312,C1(C(N2C(CNC(c3c(Cl)cnc(CC)n3)=O)CC2)=O)C2CCCCCCC12 96313,c1(C(N(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)CC)=O)cc2sccc2s1 96314,O=C1CCCCCN1CCOc1nc(CCc2nc(-c3ccccc3)no2)no1 96315,N1(c2nccc(C#N)n2)CC2CCN(C(=O)CCCCCl)C2C1 96316,CCC(C)C(O)CC(=O)NC(CO)C(=O)NC1CCCC1(C)N(C)C 96317,C1(C(=O)NCCCNC(=O)COCC2CCCC2)Cc2ccncc2N1 96318,N1(C(c2c(CCC)occ2)=O)CCC2C(C1)NC(=O)CN2C(C1CNC(=O)N1)=O 96319,N1(c2nccc(OCC)n2)Cc2[nH][nH]c(=NC(=O)c3cc(F)nc(F)c3)c2C1 96320,Cc1c(NC(C2C3CCC(C3)N2C(=O)C(C)c2cccs2)=O)ccnc1Cl 96321,C(C)(C)(CNC(=O)C=CC(F)F)N(C(=O)CC1CC1)C.CC1CC1C 96322,C1(CC)CC(F)CN1C(=O)CC1CCCC(NC(c2cnn[nH]2)=O)C1 96323,c1(CN)nc(-c2cnc(C3CC3)[nH]2)n(C)n1.C(C)(C)(C)OC(N(C)C)=O 96324,C1(COC(C2CCC(C(F)F)CC2)=O)CC2(C1)CCOC2 96325,c1(C(=O)NC(C)CNC(c2cccc(OC3CCC3)c2)=O)ncc2ccccn12 96326,CCC(C)(C(=O)NCCN(C(=O)C(C(C)C)c1ccc(NC)cc1)CC)C(F)F 96327,C(=O)(C(F)CC(C)(C)NC(=O)CC(C(=C)C)OCC)N(CC=C)CCO.C(C)=O 96328,Cc1ccc(O)c(CNC(=O)CC(C)NC(c2cnsn2)=O)n1 96329,C(=O)(CC(F)(F)CC(F)(F)F)N(CC(O)CNC(c1cn(C(C)(C)C)nn1)=O)C 96330,c1(CCC(=O)NCC2(C)CN(Cc3cnc(C(=O)OC)[nH]3)C2)ccc(F)cc1 96331,N1(C(c2n(C)ncn2)=O)CC(NC(=O)Cc2ccc(Br)cc2Cl)CC(F)(F)C1 96332,C1(CCC(=O)NC2(C)CC(NC(c3ocnc3C(F)(F)F)=O)C2)NC(=O)NC1=O 96333,C=CC(C)CC(=O)NCC1CCN(C(=O)CCCc2cc(C)no2)C1 96334,C1(C(NOCCC(C)C)=O)CCCCN1C(=O)C(C)SC(C)C 96335,C#Cc1ccc(C(=O)NCC2(C)CN(C(=O)CNC(=O)CC(C)(C)C)CCO2)cn1 96336,N1(C(C=CC(C)NC(c2ccc(CC)[nH]2)=O)=O)CCCC1(C)C(C)C 96337,c1(N(C(C(C)O)=O)C(C2CC2)=O)ccc2ccsc2c1.N1(C(CN)=O)CCCC1 96338,CC(C)(C)CCC(F)C(=O)N1CCC2(CC(C(=O)NOC3CC3)C2)C1 96339,CN(C)S(=O)(=O)NCC(=O)NC1CCN(C(=O)C=CCOCc2ccccc2)C1 96340,C1(NC(c2ccc(C(F)F)nc2)=O)CCCC(CNC(C2CCCC23CC3)=O)C1 96341,CC1CCN(C(=O)C(F)(F)F)CC1C(=O)Oc1c(C(=O)OC(C)(C)C)cccc1 96342,c1(C(=O)NCCCC(C)NC(C2CCC(=O)N2)=O)ccnc(C(F)(F)F)c1F 96343,CCCCCC(O)C(=O)N1CCCC(CC(=O)NC(C)C(C2CC2)OC)C1 96344,C1(CC(=O)OC)C2CN(C(=O)NCc3nc(-c4cccc(C)c4)no3)CC12 96345,N12CC(C3CC13)COCCOC(C)C2=O.c1(COCC)cn(CC(O)CC)nn1 96346,C12(NC(c3cccc(OCCF)c3)C)CCC1CCN2 96347,c1(-n2ccc(C(=O)NC(C(C)NC(C3(O)CCC3)=O)CO)n2)cccc(C#N)c1 96348,C1(C(=O)NCC(CNC(CSCC=C)=O)(C)O)CC2OC1C1CC21 96349,c1(NC(C2CCCN(Cc3cc(=O)[nH][nH]3)CC2)=O)cccc2c(O)ncnc12 96350,C=C(C)CC(C(=O)NCc1cn(CC(=O)N(c2cnn(C)c2)CC)nn1)OC 96351,C(=O)(C(C)(C)CCC(=O)N1CC=CC(NC(=O)C(O)CC(C)(C)C)C1)OC 96352,c1(CNC(c2c(C(C)C)c[nH]n2)=O)ccc2c(c1)CCN(C(=O)CCN(C)C)C2 96353,O=C1NCc2ccc(OCO)cc2N1.N12CC3(CCSCC3)C1CCNC2=O 96354,c1(OC)nscc1C(N1CC(OCC(=O)N(C)Cc2cnoc2C)C1)=O 96355,C1(NC(C(C)N(C)C)=O)C2CCN(C(=O)CCC(=O)N3CCOCC3)CC12 96356,S(=O)(=O)(c1ccc(NCc2nc(Cl)ccc2Br)cc1Br)NC(CC)CO 96357,Cc1[nH]nc(C(=O)N(CC(O)CN(C(=O)CC2(C)CCCCC2)C)C)c1C 96358,c1(-n2ccc(C(=O)NCCNC(C(C)C)=O)n2)ccc(F)cc1F 96359,Cn1cnn(CC(N2CCC(OCCNC(C3CCC4(CC4)C3)=O)C2)=O)c1=O 96360,c1(OCC)ccc(NC(=O)NC2CCCC(CC(F)(F)F)C2)cc1OC 96361,C(C(C(=O)N(CCC(C)NC(C1(C(C)(C)O)CCC1)=O)C)OC)OC 96362,c1(C(C)(C)O)cc(C(=O)N(CCNC(c2nnc(C3CCCC3)s2)=O)C2CC2)no1 96363,S(=O)(=O)(c1cccs1)NC(C)CCNC(=O)CCNC(C1(CF)CCC1)=O 96364,c1(CC)n[nH]cc1C(=O)N(C(C)C(=O)NCC#CC1CC1)C 96365,C(C(C#N)NC(C1CC1C(C)NC(=O)CNC(C)=O)=O)OC 96366,c1(C(=O)NCC2N(C(C(C)C(F)F)=O)CCC2)csc2ccc(F)cc12 96367,N1(C(c2c(CC)noc2)=O)CC(C2CCN(C(c3nc(C)no3)=O)CC2)C1 96368,N1(C(C(N2CCOCC2)C)=O)CCC(OCCNC(C2CC(C)(F)C2)=O)C1 96369,Cn1cnnc1CNCCN(C1CCN(C(=O)CCOCC2CCCO2)C1)C 96370,C(=O)(C(=O)NNC(=O)C(C)OCCOCC#N)OC(C)C 96371,C1(C)(C(=O)NCC2(CCNC(C3(CCCC)CCC3)=O)CC2)CCOC1 96372,N1(C(C(CC)N(C)C(c2ccc(O)cc2)=O)=O)CC2(CCC(=O)O2)C1 96373,c1(OC)ncccc1C(=O)NC(C)CNC(c1[nH]c(C2CC2)nc1C)=O 96374,CCC(C)C(C(=O)N(CCC(=O)N(CC(C)(C)O)C)CC)N(C)C 96375,C1(NC(C2(F)CN(C(CCCOCCC=C)=O)C2)=O)CCCN(CC)C1 96376,Nc1cccc(C(=O)NCC2CCCN2C(c2csc(C3CCCO3)n2)=O)c1F 96377,n1(CC)cccc1C(=O)NC1(CNC(c2ccc(CC(C)(C)C)s2)=O)CCC1 96378,N1(C(CN2CC(C)C2)=O)CCC(CCNC(c2ccncc2O)=O)CC1C 96379,c1(N2CCC(C(c3nc(CC)on3)NC(=O)NC)C2)cccc(F)c1F 96380,c1(C(N)=O)cc(C(N2CC(n3cnnc3)C2)=O)on1.C12CCC1C(=O)NC2 96381,Cc1ccc(=O)n(CC(=O)NC2CC(C)(NC(C3CCCC3CF)=O)C2)n1 96382,c1(C(N2CCCC(CN(C(=O)C3=CCCSC3)C)C2)=O)cc2c(Cl)c(F)ccc2[nH]1 96383,C=CCC(CC=C)C(=O)N1CCN(C(=O)CC2CC(=O)NC2=O)CC1CCC 96384,Cc1cc(Br)cnc1NC(=O)N(C)C.c12cncnc1N2.C12CCCC1C(=O)OC2 96385,C1(C(=O)OCC)CN(C(=O)C(C(C)C)NC(=O)NC(C)C)CC1C 96386,C1(C)(C(=O)NCC23CN(C(CCC)=O)CC(F)(C2)C3)CCc2ccccc2O1 96387,CC(C#N)CCC(=O)N1CCC(CNC(=O)CCC2CCCCC2)CC1 96388,C(=O)(C1=CCCCC1)NCCC1CN(C(C2(OCC)CCC2)=O)C1 96389,C(=O)(C(CC)C(F)(F)F)NCCC(=O)NC(C#C)C(C)OC 96390,N1(S(Cc2c(C)non2)(=O)=O)CCCC12CCOCC2 96391,N1(C(C2(C)CC(F)C2)=O)CC2C(NC(=O)COc3cccc(F)c3)C2C1 96392,N1(C(c2c(C)oc(CNC(=O)COC(C)C)n2)=O)CC2(CO)CC2(CO)C1 96393,C1(NCC)CCCN(C(=O)C(CC)NC(c2cnc(NC)cn2)=O)C1 96394,C(C(COC)C(=O)NC1CCC(NC(=O)C(C)(C)C2CCCO2)CC1)OC 96395,C1(CN(C(COCCC#C)=O)C)CCC(CNC(N)=O)CC1.C1(=O)CCN1 96396,c1(C(=O)NCC(CC(F)(F)F)NC(C(C)=CC)=O)cc(Br)c2[nH]nnc2c1 96397,C1CCC(O)C(=O)N1.c1(C(=O)NC2(C)CCCOC2)cnn2c1OCC2 96398,c1(SCCC)ccc(C(N2CC3(NC(=O)C(C(=O)OC)OC)CC2C3)=O)cc1 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96416,c1(C(N2CCN(C(COCCOC)=O)CC2C(F)F)=O)onc2cc(C)ccc12 96417,N#CCCCC(=O)NCC(C1CC1)NC(c1cnc(-c2ccccc2)o1)=O 96418,C1(C)(N(C)C(C2CCN2C2CCCC2)=O)CCN(CC2CCCN(C(=O)CO)C2)C1 96419,c1(C(=O)NC2CC=C(C(=O)N3C(C4(C)CC4)CCC3)C2)cc2cccnc2[nH]1 96420,Cn1cc(C(=O)NCC2CC(F)CN2Cc2ccc(CC(=O)O)s2)c(C(F)(F)F)n1 96421,CCCCC(O)CC(=O)NC1CN(C(c2ccccc2CC)=O)CC2(CC2)C1 96422,N1(C(=O)C=Cc2ccoc2)CC2CCC(C1)N(C(c1cc3cnccc3[nH]1)=O)C2 96423,NC12CCC1CN(C(c1cnn(-c3ccc(Br)cc3)c1)C(=O)NC1CCC1)C2 96424,C1(CNC(=O)Cc2cscn2)CC(O)CN1C(C1CC(=O)N(c2nccs2)C1)=O 96425,C(=O)(CC(C)(C)C=C)N1CCCC(N(C(c2cccc(F)c2O)=O)CC)C1 96426,c1(C(N2CCC(N(C)C(c3nccnc3N)=O)C2)=O)n[nH]c2c1COCC2 96427,O=C1Nc2cccc(-c3ccc(F)c4ccncc34)c2C1=O 96428,C(=O)(C1=CCC(NC(=O)CC2CC3C=CC2C3)C1)NC(C(=O)OC)CO 96429,N1(C(c2c[nH]c(=NC)o2)=O)CCC(NC(=O)C=C2CCN(C)CC2)C(C)C1 96430,c1(C(N2C(C(=O)NC(CCCC)CO)C=CC2)=O)cc(C)n(C)c1C 96431,C(CC(C)C)(C(=O)NC1C=CC(CO)C1)N(C(C(C)SC)=O)C 96432,Cc1cc(-c2cn(C(C)C(=O)N3CC(C4CCCOC4)C3)nn2)cnc1C#N 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96609,Cc1cc(C)c(NC(=O)CC2(NCc3cccc(C(=O)O)c3F)CCC2)cn1 96610,c1(C(N(C2CCN(C(c3cnnn3C3CC3)=O)C2)CC)=O)cc(F)c(O)c(F)c1 96611,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C)C1CC1 96612,c1(NCC2(O)CCCC(C)C2)cnc2ccc([N+](=O)[O-])cc2n1 96613,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(=O)C=CC2CCCO2)C1 96614,N1(C(CCC(N)=O)=O)CC2CCCCN2CC1CNC(=O)CC1CCOCC1 96615,N1(C(COCCOCC#C)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)C2C1 96616,C1(NC(c2ccno2)=O)(CO)CCN(C(=O)C(c2ccc(F)c(F)c2)O)CC1 96617,N1(C(CC2ON=C(CC)C2)=O)CC(F)(F)CC1CCNC(c1cc(OC)n[nH]1)=O 96618,C1(NC(C(=O)Nc2cc(C(C)C)sn2)=O)CCCN=C(I)CC1 96619,CC1(C)CC1(C#N)C(N1CCC(O)(CNC(=O)CC(=O)NCC2CC2)C1)=O 96620,CC(C)C(O)CC(=O)NCC1(NC(c2ccc(-c3nccs3)cc2)=O)CCOC1 96621,N1(C(c2c(OC)nccc2)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 96622,c1(C(=O)NCC2CC(NC(c3c(OC)cccc3)=O)C2)cnnc2ccccc12 96623,c1(C(=O)NCC(C)NC(=O)C(F)(F)C2(O)CCC2)cccc(C(F)C(F)(F)F)c1 96624,c1(OCC(=O)NCC(C)(C)NC(C2CCCC2)=O)ccc(CC2C=CCC2)nc1 96625,C#Cc1ccc(C(=O)NC2CCCC2NC(C2(CCCC)CCNC2=O)=O)cc1 96626,CCC(C)(COC)C(=O)N(C)CCN1CCN(C(=O)CCC(C)OC)CC1 96627,Cc1cccnc1SCC(=O)NC1CCCC1n1cc(C(O)CC)nn1 96628,C1(n2cc(CC(C)C)nn2)CCCN(C(=O)C2CC2)C1.C12CC(C1)C2 96629,N1(C(Cc2c(C)nn(C)c2C)=O)C2CCC1CN(C(C1CC(=C3CC3)C1)=O)C2 96630,c1(CNC(CN(C(C)=O)C)=O)ncccc1CNC(C1CN(C)C1)=O 96631,C1(NC(C(CC2CC2)NC(Cc2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 96632,C1(CNC(C(C=CC(=O)OCCOC)=CC)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 96633,c1(N(C(c2ccnn2CC)C(=O)NCCC)C)ccc(C)c(F)c1 96634,C1(C2CCN(C(=O)CNC(=O)OCC)CC2)(NC(C=CCCC)=O)CC1 96635,CC1(C)CCC(F)(F)CC1C(=O)NC1CCN(CCn2cccn2)CC1F 96636,C1(C(=O)NC2CCCC(NC(C3CCC(N(C)C)CC3)=O)C2)(OC)CCCCC1 96637,C(=O)(C1=COCCO1)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)CCCC1 96638,N1(C(c2n(C=C)nnc2)=O)CCCC2CN(C(c3cccc(F)c3Cl)=O)CCC12 96639,CS(=O)(=O)c1ccc(OCC(=O)NC23CC(C(=O)Nc4cncnc4)(C2)C3)cc1 96640,c12ccc(cc1)N(C)C(c1n(CCC)cnc1)C(=O)NCS2.C(CC#N)SC 96641,CON(C(=O)C=CC1CCN(C(=O)CC2CCCC2O)CC1)C(C)F 96642,C1(C=O)C(C)(C)C12CC2.c1(CSCC(=O)N(CCCN)C)nc[nH]n1 96643,N#CC1CCC(CC(=O)NCCNC(C2CCCCCC2)=O)C1 96644,C1(NC(C2C(C)C2C)=O)CC(NC(c2cncc(-c3ccnn3C)c2)=O)CC1O 96645,C1(C)(CN(C(=O)C=C(Cl)Cl)C)CCCC1NC(c1sccc1C(F)F)=O 96646,Cn1ncc2c(C(=O)NC3CCC3NC(c3cnc4c(c3)CCC4)=O)ccnc12 96647,N1(c2ccn(C)n2)Cc2ccc(CNc3cc(O)n(C)n3)cc2C1=O 96648,c1(OC)ccc(C(N2CC(N(C(=O)C(c3ccc(C)s3)C)C)C(F)C2)=O)cc1F 96649,c1(CN(CC(=O)N(C2CCN(C(C)=O)C2)C)C)c(I)ccnc1F 96650,N1(C(C=C2CCC(C)CC2)=O)CC2CCC(CNC(C3CCCCN3C)=O)C2C1 96651,N(C(=S)NNC(=O)c1cc(N)cc(F)c1)C1(c2nnnn2C)CCOCC1.CC(C)C 96652,c1(OCCOC)ccccc1CC(=O)NCC(O)CNC(=O)CC1CC1CSC 96653,c1(C(N2CCCC(C)(NC(C(C)n3cccc3)=O)C2)=O)ccc2[nH]ccc2c1 96654,N1(C(CC(C)NC(C(N2CCOCC2)C)=O)=O)CCC(NCCC(O)C(F)F)CC1 96655,C1(CNC(CCOCCNC(C2C(C)C2)=O)=O)CCC2(CC1)CC2 96656,c1(C(N2CCCCC2C)C(=O)NCC(C)C)cc(OC(F)F)ccc1Cl 96657,C(c1cncn1C)=CC(=O)NC(C(CO)NC(c1n(CCOC)ncc1)=O)C 96658,C(=O)(C(F)(F)C1=CCOCC1)N1C2C(NC(c3cc(C)c(C)[nH]3)=O)C(C2)C1 96659,N1(C(COCC(=O)OC)=O)CCCC1C(C)(C)C(=O)NCc1nc(C)co1 96660,C(=O)(C(C)(C)n1cc(N(CC(C)Sc2ccccc2)C)cn1)OCC 96661,c1(C(=O)NCCC2CCN(C(C(COC)N(C)C)=O)C2)ccc(OC)c(SC)c1 96662,c1(C(=O)NCCN(C(C(C)CC(N)=O)=O)C)cn2ccc(Br)cc2n1 96663,C1(C(=O)NC2CC(=C)C2)CC2(CCN(C(c3cc(C)sc3C)=O)C2)CO1 96664,C1(C(COC)C2CC2)CCCN(C(=O)Nc2cc(OC(C)(C)C)ccn2)C1 96665,N1(C(CC(CC)SC)=O)CC2(CC(NC(c3cccc(OC(F)F)c3)=O)C2)C1 96666,c1(C(C(=O)NCc2cccc(Cl)c2)N(CCSC)C)ccnc(S(C)(=O)=O)c1 96667,c1(CNC(C(C)OCC)C)ccccc1-n1cc(CC(=O)O)nn1 96668,C(=O)(CC(C1CC1)NC(=O)C(C)(C1CC1)N(C)C(C1CCCO1)=O)NC 96669,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 96670,N1(C(C)=O)CCOCC1C(N(C1CCN(C)C1=O)c1cncn1C)=O 96671,c1(CNC(c2n(CC)nc(C3CC3)c2)=O)cc(OC)ccc1OCC1CC1 96672,C=CCC(C(=O)NC(COC)CNC(=O)CCCCC(C)C)C(C)(C)C 96673,N1(C(CS(CC)=O)=O)CCN(C(C2CCN(C)C(=O)C2)=O)C(C)C1 96674,C(=O)(CC1=NN(C)C(=O)C1)NCCCCC(C)NC(c1ncnc(C)c1C)=O 96675,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)CCc3nncs3)CC21 96676,N1(Cc2nc(SC)nc(O)c2)CCC(O)C12CCSC2 96677,C(=O)(C1CCCc2nnn(C)c21)NC(C1CN(C(c2nccc(C)n2)=O)C1)C 96678,N1(C(C2CC(C(C)(C)C)C2)=O)CC(NC(C2(OCC)CC2)=O)C(F)(F)C1 96679,N1(C(CC(CC)C2CC2)=O)CCC2(CC1)CCN(C(C1CC(=O)N(C(C)C)C1)=O)C2 96680,C1(C(N2CCCC(CN(C(=O)CC(C)(C)N(C)C)C)C2)=O)CCC2(CCC2)CO1 96681,c1(C(=O)NC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2s1 96682,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OC1)C2 96683,S(=O)(=O)(c1ccc(SC(C)CN2CCOC2=O)c(Br)c1)NCCCOC(C)C 96684,N1(C(C2C(=C)C2)=O)CC2CCCC(CNC(c3c(CC)noc3C)=O)C2C1 96685,Cc1cccc(C(O)CN(C=O)C(c2nc(COCc3ccccc3)no2)=O)c1 96686,C1(CNC(CCCC=C)=O)CCC(C)CN1C(c1ccc(-c2cnc[nH]2)cc1)=O 96687,CCC(CC(C)C)C(=O)NC(C1CN(C(=O)CCOC2CCOCC2)CC1C)CC 96688,N1(C(c2[nH]cc(C)c2)=O)CCCC(C2CC(C(N3CCC3)=O)C2)C1 96689,C1(CNC(C(CC)OC)=O)CN(C)CCN1C(=O)CCOCC(C)C 96690,c1(OCCC)ccc(NC(c2cnc(C)o2)C(=O)OC)cc1OCC 96691,Cc1ccc(F)c(C(N2CCC(CC(=O)NCCC3(C)CCCCC3)C2)=O)n1 96692,Nc1cc(C(N2CCN(C(=O)C(F)C3CCC3)CC2C2CC2)=O)c(F)c(F)c1F 96693,C1(C(=O)NCC(CO)NC(=O)CCc2cncnc2O)CCC12CCOCC2 96694,C1(CNC(C2C=CCC2)=O)C2CN(C(c3cc(CC(F)(F)F)[nH]n3)=O)CC12 96695,N1CCC2CN(C(=O)CC)C(C)C12.CON1CCC(N(C)C)CC1 96696,C1(C(N2CC(F)(F)C2)=O)(OC)CCN(C(C2CCCN2C(C)C)=O)C1 96697,N1(C(CCc2cc(C)on2)=O)CC(NC(=O)C(F)(F)CN2CCCC2)C(C)C1 96698,C1(OC)(CNC(C2CCO2)=O)CN(C(C2(c3ccccc3)CC2(F)F)=O)C1 96699,CCC(CC)C(=O)NC(CNC(c1c[nH]nc1OC)=O)CO 96700,c1(N2CCc3c(cc(C)s3)C2)nc(N2CCSC(C)C2)c2c(n1)c(C)nn2C 96701,c1(C(=O)NC2C(CNC(C(CC)(C)OC)=O)C2)cnc2ncccn12 96702,C1(CCNC(CN(CC)CC)=O)CCCCN(Cc2ccccc2C)C1 96703,C(C(N)CC(F)(F)F)NC(C1CCCN(c2snc(CC)n2)C1)=O 96704,c1(C(=O)OCCC(C)C)ccn2nc(-c3ccccc3)nc2c1 96705,c1(CN2CC3C(CC(=O)OC)C3C2)ccc(C(=O)NCCC#C)c(F)c1 96706,c1(N2C(=O)CN2CC)ccc(F)cc1F.C1(=O)CCCC2(CCC2)N1.C(C)(=O)OC 96707,CCCCC(CC)C(=O)N(CC(C)NC(c1c(CC)nn(C)c1CC)=O)CC 96708,CC(CC(C)(C)C)C(=O)N1CC(NC(=O)C(C)(C)Cc2ccc(O)cc2)C(C)C1 96709,c1(OCC)ccc(N(C)CC=Cc2ccccc2OC)cc1O 96710,c1(COC2CC(NC(CCNC(=O)OC(C)(C)C)=O)C2)c(F)cccc1F 96711,C1(C(=O)NC2(CSC)CCC2)CCCCN1C(=O)C=C(C)C 96712,c1(CCC(=O)N(CC(C)NC(C2CC2C)=O)CC)c(F)c(F)ccc1F 96713,CC(C)P(C)(=O)CC(=O)NCCNC(=O)CC(F)(F)Cl 96714,C1(CC(=O)N(CC(=O)OC)CCC)CC(NC(C2CCOC2C(C)C)=O)C1(C)C 96715,C1(CNC(=O)OC(C)(C)C)COCCN1C=O.c1(C2CN2C)ccccc1Cl 96716,C1(O)(CNC(C(C2CC2)OCC)=O)CCCN(C(=O)COc2ccccc2O)C1 96717,Cc1ccccc1OCCCC(=O)NC1CCCC1NC(C1(O)CC(CF)C1)=O 96718,N1(C(c2cnn(CC)c2C)=O)CC(n2cc(C3CCCN3C)nn2)CCC1(C)C 96719,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)C(N=c2[nH]c(CC(C)C)nc(Cl)c2C)C(C)C1 96720,C(C(CNC(=O)CC1CCSCC1)C(F)(F)F)NC(CCc1nnc(C)n1C)=O 96721,Cc1cccc(CCNC(=O)CC2CCCN(C(C3CC=CC3)=O)C2)c1 96722,c1(C(N2CCC(N(C(C(CC=C)OCC)=O)CC)C2)=O)cc2n(n1)CCCN2 96723,CCCC(CNC(C1CCN(C(c2cccc(O)c2C)=O)C1(C)C)=O)CCO 96724,Cc1ccc(C(C)C(=O)NCCSCc2cn(CCO)nn2)cc1 96725,N1(C(c2onc(CC)n2)=O)CC2CCCC(N(C)C(C3CCC4CC4C3)=O)C2C1 96726,C#CCC(C(=O)NCC1CCN(C(C)=O)C1)NC(c1coc(CCC)n1)=O 96727,c1(C(=O)NC2(C(=O)Nc3ncc(F)cc3Cl)CC2)cc(Cl)cc(Cl)c1 96728,N1(C(CC=CC=C)=O)CC2(CCN(C(c3sccc3Cl)=O)CC2)CC1C 96729,C1(CCNC(CCNC(=O)C=CCl)=O)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 96730,Cc1cn(C)nc1C(N1CC(n2cc(Cn3cc(C)cn3)nn2)C(O)C1)=O 96731,C1(CNC(c2ccco2)=O)CN(C(=O)CC2(C#N)CC2)CCN1C(c1ncc[nH]1)=O 96732,c1(CC)ccc(C(N2CCOCC2CN(C(=O)CC(C)CF)CC)=O)nc1 96733,C1(CC(=O)N(CC(C)NC(c2cccc(C(F)(F)F)c2)=O)C)CCC(=O)N1C 96734,N1(C(c2nccc(C)c2N)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C2CCC12 96735,CC(C)(CO)CCCNC(C1(C)CCN(C(c2cncc(OC(F)F)c2)=O)C1)=O 96736,c1(C(N(C2CC2)CC2CCN(C(C(C)C)=O)C2)=O)cnc(OC(C)C)cn1 96737,N#Cc1cc(F)c(NC(C2CCCN2C(=O)CN2CCCCC2)=O)cc1F 96738,c1(C(N2CCC(C(C)(C)NC(C(C(C)C)C#N)=O)CC2)=O)ccn2cncc2c1 96739,C1(CC(=O)NCCOC2CCN(C(c3c(C)cno3)=O)C2)CCC(C)(C)CC1 96740,c1(C(=O)NC(C)CN(C(=O)C(CO)NC(N)=O)C)cccc2cnnn12 96741,c1(C(N2C(C(=O)O)C3CC3C2)=O)cnn2ccsc12 96742,O=C(C1CCCc2nn[nH]c21)NC1CC1NC(c1c(C(F)(F)F)cncc1F)=O 96743,N1(C(C(C=C)(C)C)=O)CC2CCCC(N(C)C(c3nn(C)cc3Cl)=O)C2C1 96744,N1(C(C(CC)COC)=O)CCCC(F)(CNC(=O)Cc2ccccc2OCC)C1 96745,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 96746,c1(N2CC(=C(CNC(c3c(OC)cccc3)=O)F)C2)ncc2ncn(C)c2n1 96747,c1(CCNCCN(C(=O)CN2CCC2C)CC)nccn1C(F)F 96748,C1(C(N2CC(COC)OCC2)=O)CCC2(CCC2)CO1.C12CC(CO)CC1OC2 96749,C(=O)(CCCCCF)NCC(C1CCCCC1)OC(=O)C(C(C)O)NC(C)=O 96750,c1(CSC(C(=O)NC(COC)CNC(=O)COCCCF)C)ccccn1 96751,CC(C(=O)N1CCN(C(c2ccc(C(N)=O)nc2)=O)C(CC2CC2)C1)C(C)(C)C 96752,C(C(C)C(=O)N(CC(F)(F)F)CC)NC(CCN(CCC)C)=O 96753,c1(C2CC(NC(c3cccc(SC(C4CSCCS4)=O)n3)=O)C2)ncccc1F 96754,c1(C(C(=O)NCCNC(CC2CC(OCC)C2)=O)C)ccc([N+](=O)[O-])cc1 96755,c1(NC(C(CC)n2ccnc2)=O)ccc(Br)c2c1CCO2 96756,C=C(C)C1OCCCC1C(=O)NCC1CN(C(C2CN(C)C2)=O)CC12CCC2 96757,c1(OC)cc(OC)nc(N2CC(CO)(NC(=O)C(O)C(C)C)C2)n1 96758,C(CC(C)C)(C(=O)NCCC(F)(F)C(C)C)ONC(C1CC(SC)C1(C)C)=O 96759,c1(CCC(N2C(c3c(OC)cccc3)CCCC2)=O)ccc(C=NO)cc1 96760,CC1CCCC1(C)C(N1CCOC(CNC(c2ccoc2Br)=O)C1)=O 96761,c1(OC)ncc(C(=O)NCCCNC2CC2)s1.C1(C(=O)N)CCCN1C1CC1 96762,C1(CNC(CCn2c(C)ncc2)=O)CCN(C(=O)C(c2ccncc2)C)CC1O 96763,CCCCC(O)C(=O)N1CCN(Cc2cnc(OC)c(Cl)c2)C2CC12 96764,C1(NC(C(C)OCC)=O)CCN(Cc2cnc(CC3CCCC3)s2)CC1C 96765,CC(Cn1cccn1)C(=O)NCc1n[nH]cc1C(=O)N(C1CCCC1C)C 96766,C1(N(C(c2c(OC)csc2)=O)C)CCCCC1NC(c1cncc(CO)c1)=O 96767,C1(NC(c2ccc(O)cc2)=O)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 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96785,CC(C)CC(C)(O)C(=O)N1CCC(n2cc(C)nn2)C2(CC2)C1.C(N)(=O)N 96786,C1(NC(c2cnc(C(C)C)[nH]2)=O)CCN(C(C23CSCC2C3)=O)CC1O 96787,C(C)(C)(CCCCC(=O)NCC1CC(NC(c2cnc(C3CC3)o2)=O)C1)N(C)C 96788,N1(C(c2cnc(C3CCCCC3)s2)C(=O)NCC)CCC(O)CC(C)(C)C1 96789,Cc1nc(NCC2CCC(F)C2)cc(N2CCN(c3ccncc3Cl)CC2)n1 96790,c1ncc(C)cc1[N+](=O)[O-].C1CCC(=O)N2CC1(O)C2.C(CCN)SC 96791,C=C(C(=O)N1C(C(=O)Nc2ccc(C(=O)OC(C)(C)C)cc2)CC2CC12)C(F)(F)F 96792,C(C(=O)Nc1noc(C)c1Br)(C(C)C)NC(C)=O 96793,N1(C(C2CC(C)CN2C(=O)Cn2c(O)nnc2O)=O)CCCC(C2(C)CC2)C1 96794,C(Cc1cc[nH]n1)(C(=O)N(CCCSC)C)OC.C1=CCNC1=O 96795,Cc1cc(Br)ccc1CC(=O)NC1CC1NC(C1(C)CC(C)(C)C1)=O 96796,CCCC(C)(O)CC(=O)NCCN(C(=O)Cc1ccc(SC)cc1)C 96797,Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N1C2CCCC1CN(C(=O)CN(C)C)CC2 96798,CC(C)C(C)CC(=O)N1CC(CC(N2CCN(C(=O)CCC3CCC3)CC2)C)C1 96799,c1(OC)cncc(-c2cn(C)nn2)c1.C12CC(C1(C)C)OC(=O)C(=O)N2 96800,c1(-c2n3nc(n2)CC3C)cc2c(cc1F)NC(=O)CC2.C1(CO)CC1 96801,c1(C(C)(O)CNC(=O)C(O)C2CC2)cccc(I)c1 96802,CCC(C)CC(C(=O)NCC1CCCN1C(C)=O)NC(c1cnn(C2CC2)c1)=O 96803,c1(C(=O)Nc2cnccc2[N+](=O)[O-])cc(-c2ccc(CCO)s2)cc2c[nH]nc12 96804,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 96805,c1(C(N2CC(CNC(C3CCc4nn[nH]c4C3)=O)C2)=O)cc2n(n1)CC1(CC1)C2 96806,Cc1ccc(-c2cnc(-c3nccn3CCN3CCOC(C#N)C3)nc2)cc1Cl 96807,CC(CN(C)C)CCC(=O)NCCN(C)C(C1CCC(F)(F)C1O)=O 96808,C(CC(C)(C)C)(C(=O)NC(C)(CNC(c1ccnc(C(N)=O)c1)=O)CC(C)C)OC 96809,C1(C)(C(N(C(CC(CC)C)C)C)=O)CCCN(C(=O)C=C(C)C2CC2)C1 96810,C(C)(CC(C)(C)C)(C1CCSCC1)NC(C1CCC(F)(F)C1)c1n(C)nnn1 96811,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 96812,c1(-c2cccc(CC(=O)NC(C)=O)c2)nc2c(s1)CCN(CC1C=CCC1)C2 96813,C1(c2cn(CC3CN(C(=O)CSCc4cccnc4)C3)nn2)CCOCC1.CS 96814,Cc1cc(=NC2CCCn3cc(N4CCOCC4)nc32)[nH]c(C2CCC2)n1 96815,N1(C(C2C(c3c(C)cccc3)C2)=O)CCN(C(c2nc(O)c(C)s2)=O)CCC1C 96816,C1(CNC(C(COCC)NC(=O)C(Cl)Cl)=O)CCCC2(CC2)C1 96817,C#Cc1cccc(C(N2CC=CCC2C(N2CCCC(CCCC)C2)=O)=O)c1C 96818,Cc1cnn(C)c1C(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 96819,c1(C(N2CC(C3C(C(=O)NCCS(CC)=O)C3)C2)=O)cc(C)cc(C#N)c1 96820,c1(C(=O)NC(C(C)NC(C2CN(C3COC3)C2)=O)CO)ccc2ncccc2c1 96821,c1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)snc(Cl)c1Cl 96822,N1(C(C2(CC)CC2)=O)CCC(CNC(c2ccc(C)s2)=O)C(F)(F)C1 96823,C1(NC(c2cc(C)nc(O)n2)=O)C2CCCCN(C(=O)Cc3c[nH]nc3C)C12 96824,C(=O)(C1=C2CCN=C2NC=C1)NCC(CNC(C1N(C)CC(C)(C)C1)=O)O 96825,C(=O)(C1=COCCC1)N1C(C)CC(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 96826,C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCCN(C(C2(C)CCN(C(C)=O)C2)=O)C1 96827,C1(CNC(C(n2c(C)ccn2)C)=O)CCC2CN(C(=O)CCc3ncccn3)CC12 96828,c1(-c2onc(-c3cccc(N(C)C)c3)n2)cccc2cc(N(C)C)ccc12 96829,N1(C(CCc2ccc(N(C)C)s2)=O)CCCN(C(=O)OC(C)(C)C)C(C)C1 96830,CC(F)(F)CCCC(=O)NC1CC(F)CN(C(c2cc(C(F)(F)F)ns2)=O)C1 96831,CC1=C(C(=O)C(NOCC(N2CCN(CCCNC(C(C)N)=O)CC2)=O)=O)CCO1 96832,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 96833,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 96834,C1(C(=O)NC(CCCNC(c2c(Cl)cc(C)s2)=O)C)CCCC2(CCC2)O1 96835,C1(C)(C(=O)NC23CC(NC(CCN(C)C)=O)(C2)C3)C2CCC(C2)C1(C)C 96836,N(C1C(=O)Nc2ccc(F)cc21)C(C1=C(C)OCC1)=O 96837,N1(C(C(N2C(C)CN(c3ccncc3)CC2)=O)=O)CCC(C2(O)CCC2)CC1 96838,CN1CCC1C(N1CC(CNC(=O)C=CC(F)(F)F)C1)=O 96839,CCC(C(=O)OC)C(=O)NCCOC1CN(C(=O)C=Cc2nccs2)C1 96840,C12(CCN(C(=O)C(C)(C)C#N)C1)C(=O)N2.C(C(=O)N(C)C1CC1)OCC 96841,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(CN(C(C(C)OCC=C)=O)C)C1 96842,N1(C(c2cccn(C)c2=O)C(=O)NC2CCCC2)CCc2c(ncn(C)c2=O)C1 96843,O=C(C1CCCc2nn[nH]c21)N(CC(=O)NCc1noc(CSC)n1)C1CCC1 96844,N1(C(C2(COC(C)C)CC2)=O)CC(N(C(=O)C(C)CN2CCOCC2)C)C(O)C1 96845,Cc1ccc(C(=O)NC23CC2CN(C(c2ncn(C(C)C)n2)=O)C3)c2ccccc12 96846,c1(C(=O)NC(c2ccc(F)cc2)CNC(CC(C)CF)=O)cnn2ccccc12 96847,c1(C(=O)NCC2COCCN2C(c2ccnnc2O)=O)c[nH]c2ncnc(O)c12 96848,Cc1ccc([N+](=O)[O-])cc1C(=O)Nc1cnc(Br)c(Cl)c1.c12cccnc1NC2=O 96849,C1(C(=O)NCC2(F)CC(NC(CCOCC#C)=O)C2)CCC(CC2CC2)CC1 96850,c1(C(=O)NCC(CC)(C)NC(C2CCC23CCC3)=O)nsc2ccccc12 96851,Cc1[nH]nc(C(=O)NC2COCC2n2cc(-c3ccnn3CC(F)F)nn2)c1C 96852,N1(C(C(C(=O)NC)(C)C)=O)CCc2ccccc2C(NC(=O)CCNC(N)=O)C1 96853,CON(C(=O)C=CC(C)NC(=O)C(CO)N(C)C)C1CCC1 96854,CC1(C)CCOC1C(N1CCCCC1C1CCN(C(=O)C(O)C2CCCC2)C1)=O 96855,C(=O)(CC(O)CC(C)C)NC(CC)(CNC(C1C=CCS1)=O)CC 96856,N1(C(CC(C=C)C)=O)CCC2CCCC12C(=O)NCCCC(C)CO 96857,C(=O)(C1=NOC(C)(C)C1)NCC1C(CNC(c2c(OC)ncc(F)c2)=O)C1 96858,Cc1cc(C(N2CCN(C(=O)CCCN3CCCC3)CC2C)=O)cc2c1CCC2 96859,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)=CC2CC2)CC1)C)C(N)=O 96860,Cc1noc(C)c1CC(C)NCc1cnc(-c2ccccc2F)s1 96861,c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C)cc(C)c(C)c(Br)c1 96862,c1(NCC(C)N(C)C(C2CC(F)(CO)C2)=O)cc2nn[nH]c2cc1[N+](=O)[O-] 96863,N1(CCNC(C2CCC2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1 96864,C1(C(N(C2CCSCC2)C)=O)CCCC(NC(c2ccc(Cl)s2)=O)CC1 96865,c1(NC(C(C)N(C2CCC(N(C)C)C2)C(c2ccnn2C)=O)=O)ccccc1 96866,C1(NC(C2(N3CCOCC3)CC2)=O)CC2CCC(C1)N2C(C1CCC=CO1)=O 96867,c1(CC)c(C(=O)NCC(C)N(C)C(c2cnn(CCO)c2)=O)cnn1CC 96868,c1(C(C(=O)NCCC(CNC(C(C)(C)OCC)=O)O)CC)c(C)noc1C 96869,C(C)(CO)(CC(C)C)NC(CN(C(C(COCC)C)=O)C1CCC1)=O 96870,Cc1cc(Cl)c(C(N2CCC(CO)C(NC(=O)CCc3ccsc3)C2)=O)cn1 96871,C(=O)(CS(N)(=O)=O)NCC.C(CC(=O)N1CC(CC)C1)NC(=O)OCC 96872,N1(C(c2ccc(OC)s2)=O)CCC2CN(C(C3CCCC3C(C)C)=O)CC12 96873,N1(C(C2(C)CC2C(F)(F)F)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 96874,c1(C(C(=O)NCC2CCOC2)N(CC=C)C(C)C)ncc(CC)[nH]1 96875,CCC(C)(O)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)CCO 96876,C12(C(=O)NCCC(C=C)C)CC(CN1C(=O)CC1C=CCCC1)C2 96877,C(=O)(C1CCCc2nncn21)N1C(C(C)(C)NC(C(C)S(N)(=O)=O)=O)CCC1 96878,n1(CCOC)cc(C(=O)NCCC2(O)CN(C(=O)Cc3cnnn3C)C2)cn1 96879,c1(OC(c2nc(CN3CCC(O)C(C)C3)cs2)C)c(Cl)cc(Cl)cc1Cl 96880,c1(CC(N2CC(C)C(NC(c3cnc(N(C)C)nc3)=O)C2)=O)cc(O)nc(O)n1 96881,c1(C(=O)NOCc2ccccc2)ncn(Cc2cc(C(F)F)no2)n1 96882,C1(C(N(C)CCNC(=O)COC(F)(F)F)=O)CC2(C1)CC(O)C2 96883,CCCCC(CNC(=O)CC1OCCC1(C)C)NC(C1CCC(=O)N1)=O 96884,CC1=C(C(=O)N2CCC(NC(=O)C=Cc3scnc3C)C(F)C2)C(=O)OC1(C)C 96885,N=c1[nH]c(=NCC2CCCCS2(=O)=O)[nH]c(=NCCC2(n3ccnn3)CC2)[nH]1 96886,c1(CNC(N2CCCC(c3n(C)ncc3)C2)=O)ccc2c(O)nnc(O)c2c1 96887,CC(C(=O)NCC1(F)CN(C(c2ccc(Cl)cc2O)=O)C1)C1=CCCC1 96888,Cc1cc(C(=O)N(CC(C)N(C)C(C2(O)CCCC2)=O)C)ccn1 96889,CCC(CCC(=O)NC1CCC(C(=O)NCCSC(C)(C)C)CC1)OC 96890,Cc1nc(C(C)NC(=O)CC2CCN(C(c3c[nH]c(C(N)=O)c3)=O)CC2)c(C)o1 96891,S(=O)(=O)(c1ccc(C(N2CCCC(F)C2)=O)cc1)NC1CC(CN)C1 96892,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 96893,N1(C(C2(CC)CC2)=O)CC(C)OC2(CCN(C(c3cccc(C)c3)=O)CC2)C1 96894,N1(C(C(C=C)(C)C)=O)CC2CC(C1)CN(C(C1CC(n3cnnc3)C1)=O)C2 96895,C1(C(=O)NC(CCO)C2CCCC2)C2CCC(C2)N1C(=O)CC1CSCCO1 96896,N12CCCC(C)(C1)C2=O.c1(OC(CC)CSN2CCCC2=O)ccccc1C 96897,N1(C(CC2CC(NC(C(C)Cn3ccnc3)=O)C2)=O)CCC2(CCCCC2)C1 96898,c1(C(N2CCN(C(=O)C=CI)CC2CF)=O)cnc2n1CCOC2 96899,C(CC(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)C(C)NC(C)=O)OC 96900,c1(C(=O)OC(C)(C)C)cc2c(s1)CCC2C(=O)OC(C(N1CC(OC)C1)=O)=O 96901,C(=O)(C1=CCN(C(=O)C(c2ccccc2)F)CC1)NC(C#C)CC 96902,c1(C(N2CCCC(NC(C(CC)(C)F)=O)C2)=O)cc(OC)c(OC)c(F)c1 96903,C(=O)(CCCCC(F)(F)F)NCC1CCCC(CNC(C2C(CC)C2)=O)C1 96904,C1(NC(C(CC)CC(C)C)=O)CCCC2CN(C(c3csc(C(C)=O)c3)=O)CC12 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97059,c1(C(=O)NCCCN(C)C(c2nc(O)nc(O)c2F)=O)nnn2c1C(=O)NCC2 97060,Cc1ccc(Cl)cc1C(=O)NC1CN(C(=O)COC2CCN(C)CC2)CC1C 97061,c1(C(=O)NCCCNC(CC2C(C)=NOC2=O)=O)nccc2[nH]nc(C(C)C)c12 97062,N1(C(C(CCCC)O)=O)CCC2(CCC(CNC(c3ncoc3C)=O)OC2)CC1 97063,C(=O)(CCCC(=O)NCCCCNC(c1cc(OCC2CC2)n[nH]1)=O)OC 97064,CCCCC(O)CC(=O)NCCCC(C)NC(c1cc(OC)nc(C)c1)=O 97065,C1(COCCOCC)(Cc2cccnc2)CCCCC1.N12CCC(C1)OCC2=O 97066,C(CC(=O)NN1C(=O)CCC1c1ccccc1)(C1CCOCC1)OCC 97067,N1(C(C(=O)NC2CCN(C(c3c(C)onc3)=O)C2)(C)C)CCS(=O)(=O)CC1 97068,CC1CCC(=CC(N2CC(CC(F)F)C(C)C2)=O)CC1 97069,CC1CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1CNC(=O)CCc1cnco1 97070,c1(C(C(=O)NCCOCCNC(c2c(C)cncc2)=O)C)c(C)nn(C)c1C 97071,c1(C(c2nnnn2C2CC(F)(F)C2)NCCCCCCSC)ccc(C)nc1C 97072,n1(CC(CC)O)cc(C(=O)N(C)CCNC(=O)CCC2CCC(C)O2)nn1 97073,CC(C)C(C(=O)N1CC(CC(C)(C)CNC(c2coc(CO)c2)=O)C1)n1cnnn1 97074,c1(C(=O)NCC2CCC(NC(c3cc(C(C)C)[nH]n3)=O)C2)ccc(Cl)c(Cl)c1 97075,N1(C(C2CCN(Cc3cccc(CC)n3)C2=O)=O)Cc2ccncc2C1 97076,c1(C(N2CCCC(CNC(C)=O)C2)=O)ccc(NC(=O)CC2CCC(=O)N2)cc1 97077,N1(C(c2ccc(C)nc2C)=O)CC2CCN(C(=O)C(O)CN(C)C)CC2C1 97078,Cn1c(CNC(N2CCCC2c2ccc3c(c2)OCO3)=O)nc2ccccc12 97079,C1(C(N)=O)(CNC(C2(CC)CCCN2C(=O)C(C)SC)=O)CC(F)(F)C1 97080,c1(CC(=O)NCC(CC(F)(F)F)NC(C2CCCSC2)=O)c[nH]c2ccccc12 97081,N1(C(c2cn(C(C)C)nn2)C(=O)NCCC2(C)CC2)CCCC(C)(C#N)C1 97082,C(CC(=O)N1CC=C(CCNC(=O)C(C)(C)C)CC1)(C(F)(F)F)OC 97083,CC(O)(C(=O)N1CCN(C(c2cnc(C3OCCO3)s2)=O)C(CO)C1)C(F)(F)F 97084,C(=O)(C(CC(F)F)NC(=O)COC1CC1)N1CC(C)(COC)C1 97085,C1(CNC(=O)COCC2CC2)CN(C(c2cnn3c2CCC3)=O)CC12CC2 97086,C(CN=c1[nH]ccnc1F)C1CCC(NC(c2nc(CC)sc2)=O)C1 97087,Cc1ccc(C(C(=O)N2CC(CCNC(C3CC3C(F)(F)F)=O)C2)N(C)C)cc1 97088,N1(C(C2(C(C)=O)CC2)=O)CCCC1c1ccccc1.C12CN(C1)C(=O)N2 97089,c1(OC)ccc(C(=O)Nc2nc(C(=O)Nc3ccccc3C(N)=O)cs2)c(Cl)n1 97090,N1(C(CCC(=C)C)=O)CC2(CC(NC(=O)Cc3cccc(OC)c3)CO2)C1 97091,C(C(C)(COC)CN=c1[nH]c(=NCC(CSC)CO)[nH]c2c(F)cc(F)cc12)OC 97092,C(CC1=CCN(C(=O)Cc2cnccn2)CC1)NC(CN(C)C1CC1)=O 97093,C1(C(=O)Nc2ccc(O)nc2)CC2CCC(C1)N2C(C1CC(O)C1)=O 97094,C1(NC(c2c(C)sc(-c3nc[nH]n3)n2)=O)CC2CCC(C1)N2C(C1CC1CF)=O 97095,C(=O)(C(C(C)C)SC)N1CC(CCO)(NC(CC(=C)Br)=O)C1 97096,N1(C(COC(C)C)=O)CCC2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 97097,C(c1c(Cl)cccc1Cl)=CC(N1CCN(C(=O)CSC2CC2)C(CCO)C1)=O 97098,N1(C(CC2(CC=C)CCCC2)=O)CCCCC1C(=O)NCC(CSC)OC 97099,c12c(ncnc1Cl)NCCCCC(C)NC2=O.c1(CC)ccc(C)cn1 97100,c1(OC)ccn2c(C(=O)NCC3CCC(n4cc(C(O)C5CC5)nn4)C3)cnc2c1 97101,c1(C(=O)NCC(CNC(CC2(C)CC(F)(F)C2)=O)F)cnc2c(c1)NCC(=O)N2 97102,c1(OCC)c(C(=O)NC2CCN(C(C3(CF)CC(F)(F)C3)=O)C2)cccc1F 97103,C12(C(=O)NCCCC(C)(C)NC(CC(CC)C)=O)CCC(=O)N1CCS2 97104,CN1CCCCC1C(=O)N(c1cc(-n2cncn2)ncn1)C1CCNCC1 97105,Cc1ccc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)C(C)(C)C2)=O)cc1C#N 97106,C1(CC(=O)NCC23C(CN(C(Cc4ccc(C)cc4)=O)C2)C3)CCOCC1(C)C 97107,C12(NC(c3n(CC=C)ccn3)=O)CCC1CN(C(=O)CNS(=O)(=O)NC)C2 97108,C1(C(C)C)N(C(=O)NCC(c2ccc(F)cc2)N(C)C)CC12CCCCC2 97109,c1(C(N2c3c(cccc3)C(C)C2)C(=O)NC2CCC2)c[nH]c2ncc(Cl)cc12 97110,C(=O)(CC(F)(F)CC)N(CCNC(CCSCCC)=O)C 97111,c1(NCCNC(CC2(C)CCN(C(C(C)S)=O)C2)=O)cccc(C#N)c1 97112,c1(CC(=O)NC(CC)CNC(c2cc(COC)c[nH]2)=O)cncnc1O 97113,C1(C(=O)NCCN(C(c2[nH]cc(OC)c2)=O)C2CC2)(CF)CC2(CCC2)C1 97114,c1(C(=O)NCC2CCC2)cnc(O)cc1C(=O)O.C1CCNC(=O)O1 97115,C(=O)(CCCC(C)(C)C)N1CC(C)C(CNC(c2cnc(CCN(C)C)s2)=O)C1 97116,N1(C(C(C(C)O)(F)F)=O)CC2CCC1CN2C(c1cc2c(s1)CCCC2)=O 97117,Cc1ccccc1-c1ccc(C(=O)NCC(=O)Nc2cn(C)nc2C(N)=O)cc1 97118,c1(C(=O)NCC(C)N(C(c2cc(C)ns2)=O)C)ccccc1SC(C)C 97119,C1(CNC(C2(C)CCCCC2)=O)CC2(CCC2)CN1C(=O)CCSCC(N)=O 97120,CC1=C(C(=O)N2CC(F)(F)CC2(C)CNC(C2CN3CCN2CC3)=O)SCCO1 97121,N1(C(c2cc(C)oc2)=O)CCC(C(=O)NCC(C)(O)C(C)C)C1(C)C 97122,Cc1cc(Cl)ccc1OC(C)C(=O)N(C1CC(NC(C2(F)CCCC2)=O)C1)C 97123,c1(C(=O)OC)cccn(CC(=O)NCCc2cc(C)[nH]n2)c1=O 97124,N1(C(CCC#CC)=O)CCc2ccccc2C1CNC(=O)CCN(C)C(C)=O 97125,N1(C(C(c2ccccc2)OC)=O)CCCC(C(C)NC(C2(C(N)=O)CC2)=O)C1 97126,c1(C(=O)NC2CC(C)(C(=O)NCC3(CCC)CCC3)C2)ccc(C)nn1 97127,C1(C(N2CCC(CNC(C3(CC(C)C)CCC3)=O)C2)=O)C2CCCCC12 97128,C1(CC)C(C(N2CC(C#N)C2)=O)CCN1C(c1cc(C)ncn1)=O 97129,C1(CC)C(NC(c2csc(O)n2)=O)CCN1C(C1CCCN1C)=O 97130,C(=O)(C#CC1CCCCO1)NCC1C(NC(CCNC(COC)=O)=O)C1 97131,CCC(CC(F)F)C(=O)N1CCC(C2(NC(c3ccc(CC4CC4)s3)=O)CC2)C1 97132,c1(-c2cn(C3C=CC(C(N(CCC=C)C)=O)C3)nn2)cc(C(=O)OC)ccn1 97133,c1(C(N(CCCNC(C2CCCC23CC3)=O)CC)=O)ccc(F)c(C(F)F)c1 97134,Cc1coc(C)c1C(=O)NCC1CCN1C(C1(c2ccc(Cl)cc2)CCCCC1)=O 97135,c1(C(=O)NC(CN(C(C(C(=C)Cl)(C)C)=O)C)(C)C)cccc2[nH]ncc12 97136,C1(C(=O)NCc2c(CNC(COC)=O)cccn2)Cc2ccc(C)cc2S1.C(C)C 97137,Cc1cncc(CCNC(C2(NC(=O)C=CC3CCOC3)CSC2)=O)n1 97138,c1(N(CC)CC)ccc(C(=O)NC2CCCCC2NC(c2cocc2C)=O)cc1 97139,c1(C(=O)NCc2cc(C(=O)NCc3c(C)cccn3)no2)ccc2c[nH]nc2c1 97140,N1(C(C(CC)OCC)=O)CC2CC(NC(c3cc(C(C)C)n(C)c3C)=O)C1C2 97141,c1(NC(c2n(CC(=C)C)nnn2)CCSC)cc(OCC)ccc1C 97142,C=CCC(CNC(C1CCCC(C#N)C1)=O)C(=O)N1CCC(C)(CO)C1 97143,Nc1cncc(C(N2CC(CO)(NC(C3CC3c3cn[nH]c3)=O)C2)=O)c1 97144,C1(NC(c2n(C)ccc2)=O)CCN(C(=O)CC2CCC2)CC1O 97145,C(=O)(CC(C)COC)NC(C(N1CC(F)(CC)C1)=O)COC 97146,CCCCC(C(=O)N1C2CCCC1CN(C(C1(C3CCCCO3)CC1)=O)C2)C(C)C 97147,Cc1c(C(=O)NCC(C2CC2)NC(=O)CC2(CO)CCC2)oc2ccccc2c1=O 97148,C1(C(=O)NCC=CC)CCN(C(=O)C2=CCCC2C)CCO1 97149,C(=O)(CCCN(C)C)NC(CC)CN(CCC(C)(C)C)C(=O)C=CC(C)CC 97150,C(c1cccc(F)c1Cl)=CC(=O)N(C1CC(NC(C(C2CC2)OC)=O)C1)C 97151,CCC(CNC(c1cc(NC(C2CCCN2C(N)=O)=O)n[nH]1)=O)(CC)NCC 97152,C#CC1CCC(C(N2CCCC(NC(=O)CCOC(C)C)C2)=O)CC1 97153,C1(NC(C(C=CC)O)=O)CC2CC(C1)N(C(=O)CCOCC(F)F)C2 97154,N1(C(C(CCC)=CCC)=O)CCC2CN(C(=O)C(CC)C3CCCCC3)CC2C1 97155,CC(C(=O)NC(CCNC(c1ccc(C(C)(C)C)c(Cl)c1)=O)CO)P(C)(C)=O 97156,C1(C(=O)OC)CC(OC)CN1C(=O)Cc1cccc(C)c1 97157,CC1CC(NC(c2cc(C(F)F)on2)=O)CN(C(=O)C2=CCCCO2)C1 97158,c1(CC)oc(C)cc1C(=O)NCC(CO)NC(c1ccn(CC#N)n1)=O 97159,CC1CN(C)CCN1C(C1CC(O)CN1C(c1ccc(F)cc1I)=O)=O 97160,c1ccc2c(c1)COC2.c1(C(n2nnnc2C2(C)CCN2)C)ccccc1Cl 97161,c1(OC)cc(-c2cnc(Cl)c(C(=O)N(CC#N)CC#N)c2)c(F)cn1 97162,O=c1[nH]ccn2c(N3CCC(CC(=O)O)C(F)(F)CC3)nnc12 97163,C1(CC)CC1C1CC1C(N1CCCC1CN(C)C(c1c(C)coc1C)=O)=O 97164,n1(CC(=O)NCC2CN(C(CN(C(COC)=O)C)=O)CC2O)nc(O)ccc1=O 97165,C1(CNC(Cn2c(C(C)C)nnn2)=O)CCCCN(C(=O)C(F)CC2CC2)C1 97166,CN1CCOC(CN(C)C(C2CCC(C3CC3)N2C(c2cncc(O)c2)=O)=O)C1 97167,C1(NC(CN(CC(C)(F)F)C)=O)CC=CCC1C(=O)NC(CC(C)C)C 97168,c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)o2)=O)ccc(F)cc1OC 97169,c1(C(N2C(CC(=O)NC3CC4(CCC4)C3)CCC2)=O)ccc2cnccc2n1 97170,Cc1ccc(C(=O)NCCn2ccc(C(=O)N(C3COCC3(C)C)C)c2)n1C 97171,C12(CC(F)(F)C1)C(=O)N2.Cc1scc(C(N2CCC(CC3CC3)CC2)=O)c1N 97172,c1(OC)cnc(Cl)[nH]c1=NC1CC2CN(C(c3ccc(F)c(F)c3F)=O)CC2C1 97173,Cc1cnccc1N1CCC(C(N2CCC(c3ccncn3)CC2)=O)CC1 97174,C#CCC(C)(C)C(=O)NCC(CNC(c1ccnn1C1CCC1)=O)C(F)(F)F 97175,S(=O)(=O)(c1cccc(Cl)c1)N1CCC2(C(C(=O)NCC(C)OC)C2)C1 97176,C12(NC(C(CC)C(=O)OC)=O)CCCN(C(=O)C(C)COC(C)=O)CC1C2 97177,C1(NC(c2[nH]cc(CC)n2)=O)CC2CC1N(C(=O)Cc1cccc(C)c1Cl)C2 97178,N1(C(C(C)SC)=O)CC(C2CN(C(=O)COc3ccsc3)C2)C1 97179,N1(C(c2cc(OC)cc(C)n2)=O)CC2CC(C)N(C(=O)CC3CNC(=O)C3)C2C1 97180,O(NC(=O)CC(C(F)(F)F)NC(=O)CSC1CC1)CCC=C 97181,C1(CC)CN(C(=O)CN(c2ccccc2)C)CC12OCCO2 97182,N1(C(c2c(CC(C)C)cccc2)=O)CC(NC(c2cnn(CO)c2)=O)CC(O)C1 97183,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97184,N1(C(c2c(C)nc(Br)s2)=O)CCC(C)(NC(=O)CC2CCC(=O)N2)CC1 97185,c1(C(C)OC)nc(CC(=O)N(C(C)CNC(c2c[nH]nc2C)=O)C)cs1 97186,N1(C(C=C(CCC)C)=O)CCN(C(c2cncc(-n3cnnn3)c2)=O)C(CF)C1 97187,N1(C(CCNC(=O)OC)=O)C(CNC(=O)Cn2nc(C)nc2C)CC2COCC12 97188,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCCC2NC(=O)C=CI)CC1 97189,Cc1nn(C)c(C(=O)NCC2(C)CC(NC(c3cnco3)=O)C2)c1Cl 97190,c1(C(N(CC(C)NC(CCOCC)=O)C)=O)cc2cc(Cl)ccc2o1 97191,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97192,C(=O)(C1CCc2c[nH]nc21)NCCC(C(F)(F)F)NC(=O)COCCOCCO 97193,C(=O)(C(C)C(C)C)N(CCC(C)(C)NC(c1n(CC)ncn1)=O)C 97194,C(CCC(C)(C)C(=O)NCC(O)CC(C)C)NC(C=C(CCC)C)=O 97195,CCCCCCCCC(=O)NC(CC)CCCC(=O)N1CCOC2CCC12 97196,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97197,Cc1cccc(Cl)c1C(N1CCC(C)C1CNC(=O)CCOCCN(C)C)=O 97198,C(=O)(C#CC1CCCCC1)N(C)CC1CCCCN1C(C1CC(O)CN1C)=O 97199,CCC(C)C(C(=O)NCCCCNC(=O)CC(F)(F)F)NC(C)=O 97200,C1(C(=O)NC2(C(N(C3CCCC3)C)=O)CC2)CCCN1C1CC1 97201,n1(CC(=O)NCC2(F)CC(NC(Cc3cn(CC)nc3)=O)C2)nc(O)ccc1=O 97202,C1(C(N2CC(O)(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)CCCCN1N=O 97203,c1(NC(c2ccc(C(=O)OCC)cn2)=O)c(Oc2cccc(Cl)n2)cccc1Cl 97204,c1(C(C)C)ccc(C(N2CCCC(CO)(NC(=O)CCC3CCC3)C2)=O)c(O)n1 97205,CCCCCC(=O)NC(C(=O)NC(c1ncc(C)o1)C)C(C)C 97206,c1(OC)cc(N)c(Cl)cc1C(=O)NC1CCN(C(C2(C)C(C)(C)C2(C)C)=O)CC1C 97207,C=C1CON(C(=O)C2(NC(=O)CC34CCCC3C4)CCC2)C1 97208,C(N=c1nc2sccc2c(NCC2CC(=O)NC(C)C2)[nH]1)c1ccn(C)n1 97209,N1(C(CN(C(=O)OC)C)=O)CCC(C(C)C(=O)NC(c2ccccc2)(C)C)C1 97210,CCS(=O)(=O)CCCCCN1CC2C(CNC(=O)CCN3C(=O)CCC3=O)C2C1 97211,CON(CCC(=O)N(C(CO)CC(C)(C)C)C)C(=O)NC(C)CC(N)=O 97212,C(CC(F)(F)Cl)NC(CNC(=O)NCCC1(OC)CCC1)=O 97213,C1(N)CC(CNC(c2cc(CO)c(C)o2)=O)C1(C)C.CC(C1CC1)=CC1CC1 97214,N1(C(CC=C=C)=O)CC2CC(NC(=O)CS(=O)(=O)CCC)C(C2)C1 97215,CCCC(C(O)C(=O)NCCC1CCC(C)(C)C1)NC(c1cc(C)nnc1C)=O 97216,CCC(C)(C(=O)NCC1(C)CC(F)(F)CN1C(c1ccc(F)c(F)c1)=O)C(N)=O 97217,C12(C(=O)NCC(CNC(CCCOC(C)(C)C)=O)O)CCC(C)(CC1)C2 97218,N1(C(C(C)Br)=O)CCCC(C2CN(C(=O)C(F)(F)C(C)O)C2)C1 97219,O=C(NN1CCOCC1)N1CC2CCCC2C1.C12CCC(CC1)C(=O)O2 97220,c1(NC(CNC(CCC)=O)=O)ccc(Oc2ccc(C(=O)N(C)C)cn2)cc1F 97221,C(=O)(CC(CC)C(F)F)N(CC(=O)NCc1cccnc1)CCC 97222,N1(C(C(CO)OC)=O)CC2(CNC(c3sccc3OCC(F)F)=O)CCC1CC2 97223,C1(C(=O)NCC(C)(C2CC2)NC(c2cnc(COC)s2)=O)CN2CCN1CC2 97224,c1(C(=O)NC2C3CC2CN(C(C2CN(C4CCOC4)C2)=O)C3)cc(Cl)ccc1Cl 97225,C1(NC(C2N(CCC)CCC2)=O)CCCN(C(C2(CC)COC2)=O)C1 97226,c1(C(Cn2nc(-c3cccc(OC(C)C)n3)nc2C(C)CF)OC)cccc(Cl)c1 97227,Cc1cc(=NCCCCC2(C)OCCO2)[nH]cc1S(=O)(=O)NCC1CCC1C 97228,CCS(=O)(=O)CC(=O)N1CCCC1CN(C)C(C12CCC(CO1)C2)=O 97229,C1(NC(CCN(CC)CC)=O)CN(C(c2snc3ccccc23)=O)CC1C1CC1 97230,C(=O)(CC(C)(C)C#N)NCC1CN(C(c2ccc(CC=C)cc2)=O)CC1C 97231,c1(-n2c(C(C3(C(C)C)CC3)NCC(c3cccs3)C)nnn2)ccc(F)cc1 97232,Cc1ncc(C2CCCC(NC(=O)CCc3cccc(Cl)n3)C2)n1C 97233,N1(c2c(C)nc(C)nn2)CC(C)(C)CCC1C(=O)Nc1nc(Cl)nc(Cl)n1 97234,C1(C2(O)CN(C(=O)C(C(C)C)n3cnnn3)C2)(CNC(CCC#CC)=O)CC1 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97394,N1(C(=O)NC(c2nocc2N(C)C)C)CCOC2(CCc3ccccc32)C1 97395,C1(C(=O)OC)CCC(O)CN1C(C1CC(C)(NC(C2CCSCC2)=O)C1)=O 97396,C(C)(C)(CCC(=O)N1CSCC1C(=O)NCc1snnc1C)OC 97397,CC(C)C(F)(F)CC(=O)N1CC(CNC(C2(C)CCSCC2)=O)OC(C)(C)C1 97398,N1(C(CCCC(C)=O)=O)CCC(C(=O)N(C(C)CO)C2CC2)C(C)(C)C1 97399,C1(CC(=O)NCC2C(C(=O)NC3C(C#N)CCC3)CCO2)Cc2ccccc2C1 97400,CC(=O)CCC(=O)NCCCC1(c2cc[nH]n2)CC1.C12(CC1)C(=O)N2 97401,c1(C(N(C2CC(NC(C3(F)CCCC3)=O)C2)C)=O)cncc(-c2cnccn2)c1 97402,C1(C(=O)NCCOCCN(C(C(C)C(F)(F)F)=O)C)CN2CCCC2CO1 97403,C1(CNC(Cc2c(C)cc(F)cc2)=O)CCC2CN(C(=O)CCc3ncc[nH]3)CC12 97404,N1(C(C(CC)C2CC2)=O)CCC(N(C(=O)C=Cc2ncc[nH]2)CC2CC2)CC1 97405,C(=O)(C1CCCn2nccc21)N1CC(CN(C)C(c2ccc(=O)n(CCO)c2)=O)C1 97406,N1(C(CC=CC=C)=O)CC(CC=C)(NC(C2(C3CCCCO3)CC2)=O)C1 97407,C1(NC(C(=O)NCc2ncc(C(C)C)[nH]2)=O)CNC(=O)C1(C)C 97408,N1(C(C(C)OCCCCCC)=O)CCC(C(=O)Nc2cncc(Cl)c2C)CC1C 97409,CC(CCNC(=O)Cc1ccccn1)CCNC(=O)C(O)CCn1cncn1 97410,c1(CC)cc(N2CCCC(CCNC(C3(C)CC=CCC3)=O)C2)ncn1 97411,N1(C(C(CSC)C)=O)CCN(CCNC(=O)CCc2cncn2C)CC1 97412,Cc1noc2ncc(C(N3CC(NC(c4cc(F)cc(Br)c4)=O)C3)=O)cc12 97413,C12(C(=O)NCCC3CN(C(COCC=C)=O)CC3C)CCC(N(C)C)(CC1)CC2 97414,C1(NC(C(=O)NCC)=O)CN(C(c2ccc(F)cc2N)=O)CC(C)(C)C1 97415,C1(CC(=O)NCCC(C)NC(C2CCN(c3ccncc3)C2)=O)CC(C)OC1C 97416,N1(C(c2c(C)cc(C(F)(F)F)s2)=O)CC2(CNC(=O)CC3(C)CC3(F)Cl)CCC1C2 97417,c1(CC)nc(NC(C2C(C)CN2C(=O)COCCSC)=O)co1 97418,N1(C(CC(C)(C)F)=O)CCC2(CCOC2)C(CNC(C23CCC(CC2)OC3)=O)C1 97419,N1(C(C2C(C)(C)C(O)C2)=O)Cc2cc(Cl)ccc2CC1C(=O)O 97420,C1(CC)(CO)CCCN(C(C2CCCCCC2NC(=O)CC(C)SC)=O)C1 97421,c1(C(=O)NC2(CF)CCN(C(C(C)(C)c3cc[nH]n3)=O)C2)cc2c(s1)CCC2 97422,O=C1OC(CNC(=NCCF)NCCc2ccc(C#N)cc2)CCC1(F)F 97423,c1(N2CC(N(C(C)=O)C)C2)cccc(CCC(=O)NC2C3COCC23)c1 97424,C1(NC(C(C)n2cncn2)=O)(CO)CCN(C(=O)CC2(CN(C)C)CCC2)C1 97425,C(=O)(CCC(F)(F)Cn1cc(CC(c2ccc(C)cc2)O)nn1)N(CC(=C)C)C 97426,C12(CNC(c3nn(CC)c(C4CC4)c3)=O)CCCC1N(C(=O)CS)CCC2.C1CC1 97427,C1(C(=O)NCCC(=O)N(C(CC)CC)CC)CCCN(C(=O)C=CC=CC)CC1 97428,C=CC1(C(N2CCC(O)(C(C)C)C2)=O)CCN(C(C2C=C(C)CS2)=O)C1 97429,c1(C(=O)NC(C)(CNC(C2(O)CC2)=O)C2CC2)c(Cl)csc1Cl 97430,CC1(C)CC(CO)N(C(C2(NC(=O)Cc3cncs3)CC(F)C2)=O)C1 97431,C1(C(=O)NC2CCN(c3nnc(-c4ccon4)s3)C2)CCOC2(CCC2)C1 97432,C(CCNC(=O)Cn1[nH]cnc1=N)(C(=O)NC1CCCCC1C(N)=O)OC 97433,CCCC(CCCNC(c1cc(C)[nH]c1C)=O)NC(=O)Cn1nc(C)n(C)c1=O 97434,c1(C(N2CCCC(CCN(C)CCO)C2)=O)cc([N+](=O)[O-])n[nH]1 97435,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 97436,c1(C(=O)NCCC(C)NC(Cc2nc(CC)sc2)=O)ccc(O)c2c1CCCC2 97437,c1(NCCC(CC)O)ccc(S(=O)(=O)N2CCOC(CC(OC)OC)C2)cc1Br 97438,N1(C(C(c2cn(C)nn2)NC(c2cc(CC)no2)=O)=O)CC2CCC(CC2)C1 97439,N1(Cc2ccc(NC(c3n(CC)nnn3)Cc3ccccc3)s2)CCCCCC1 97440,C1(C(=O)NC2C(CNC(c3cccc(Br)c3)=O)C2)CC2CCC1C21CC1 97441,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(F)C1 97442,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 97443,CC(C)(CN=c1ccnc(-c2cccc(Cl)c2)[nH]1)NC(c1cc(C(F)F)[nH]n1)=O 97444,c1(OCc2ccc(CNC(=O)C(=O)NC3C(C)CSC3)cc2)ccc(Cl)c(Cl)c1 97445,O(S(=O)(=O)c1cc(Br)ccc1Br)c1cccc(C(=O)N(C2CC2)CCO)c1.C1CC1 97446,N1(C(C(c2ccnn2C)C)=O)CC2CCCCC2(CNC(c2csc(C#N)c2)=O)C1 97447,N1(C(C(C2CCCCC2)SC)=O)CCCC1C1(NC(=O)C=Cc2cc[nH]n2)CC1 97448,Cc1c(Br)noc1C(N1CCC(O)(CNC(=O)Cc2cncnc2)C1)=O 97449,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)N(C)CCn1ccnn1 97450,C1(C(=O)NC(C)CF)C2CCC(C2)N1C(c1ncccc1Cl)=O 97451,c1(C(=O)NC23CC(NC(c4cncc(Cl)c4)=O)C(OC2)C3)ccc2oncc2c1 97452,C1(C(=O)Nc2cnc(I)cn2)CN(Cc2cccc(C(F)F)c2)CCC1O 97453,C1(C(C)(C)NC(CN(C(C)=O)C)=O)CCCN1C(=O)Cc1ccccn1 97454,c1(C(N2CCOCC(C(C)C)C2)C(=O)NC)ccc(Cl)c(Cl)c1F 97455,c1(C(=O)NCC(C)CNC(C2CC(F)(CO)C2)=O)c(C#N)ncn1C 97456,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 97457,c1(C(=O)NCCCC2(NC(c3cccnc3O)=O)CC2)ncccc1Br 97458,C(C(C)NC(=O)Cn1nc(C)cc1C)(C(C)C)NC(CCC#C)=O 97459,c1(C2N(C(CCC)=O)CCC2)cccc(Br)c1.c1(S2=CC=C2)cn(C2CC2)nn1 97460,C1(CC(=O)NC2CCCC(NC(=O)CN3CCCNC3=O)C2)CC2C=CC1CC2 97461,N1(C(CCSCCC)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 97462,Cc1nc(C(C)C)sc1C(C)N(c1nccc(-c2ccccc2)n1)C 97463,C=CC1(CC(N2CC(C(N)=O)(CNC(=O)CNS(=O)(=O)CC)C2)=O)CCCCC1 97464,C1(NC(C)=O)CCCN1C(=O)NCCn1cccc1 97465,C#CCCCC(=O)NCC1CCC1C(=O)NC1CC=C(C)CC1 97466,c1(C(=O)NC2C(C)N(C(=O)Cc3cnn(C)c3)CC2)cc2cccnc2nc1N 97467,c1(CC(=O)NCC(CC=C)NC(c2nccn2CC)=O)ccc(CO)c(F)c1 97468,Cc1cc(C(=O)NC2CC3(C2)CC(C(=O)Nc2cc(I)ncn2)C3)cc(O)n1 97469,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2ncoc2C2CCC2)=O)CC1 97470,C1(CNC(c2c(OC)ncc(Cl)c2)=O)CCC2(CN(Cc3csc(Br)c3)C2)O1 97471,N(C(=NCCC12CCC(CC1)OC2)NCC(F)(F)CO)C(C)C 97472,C1(CNC(c2nn(C)c(CO)c2)=O)CC2(CO1)CN(C(c1ccc(Cl)s1)=O)C2 97473,C1(NC(C2CC(N=[N+]=[N-])C2)=O)CCC2(CCN(C(=O)CNC(=O)NC3CC3)CC2)C1 97474,N1(CC(=O)NC(CNC(CCN(C(CC)CC)C)=O)CO)CCC(C)C1 97475,N1(C(CC(=O)NCC#C)=O)CC(NC(=O)Cc2csc(Cl)n2)C2(CCOCC2)C1 97476,C1(CNC(C2C(C)(C)C2)=O)CCCCCN1C(=O)C=Cc1cc(Cl)sc1Cl 97477,C1(C(N2CC(F)(CNC(CC3C(C)C3(F)F)=O)C2)=O)CC(O)CN1C 97478,c1(OC)ccc(C)c(C)c1-c1ncccc1C(=O)NC(c1cn(C)nn1)=O 97479,CC1CCN(C(c2coc(CNC(C3CCC4CC4C3)=O)c2)=O)C(CO)C1 97480,C1(C(=O)NC(C2CN(Cc3nc(CCC)on3)C2)C)CC12CCCCC2 97481,c1(C(=O)NCC23C(CN(C(C(CCCC)O)=O)C2)CC3)c(C)nn2ncccc12 97482,c1(NC(=O)NC2CCc3c[nH]nc3C2)nc2ccccc2cc1[N+](=O)[O-] 97483,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 97484,c1(CC(=O)Oc2ccc(C(CC)OC)cc2)c(F)cccc1F 97485,c1(C(=O)NCCC2(CNC(c3ccc(SC)cc3)=O)CC2)cc(SC)nc(Cl)c1 97486,C1(NC(C(CCCCC)O)=O)CCCCC12CCN(C(=O)CC1(O)CCCC1)C2 97487,C(=O)(CC(C)C(C)(C)C)N1CCC(CNC(c2nc(COC)oc2)=O)C1 97488,c1(OC)cc(C(=O)NCCC2(O)CN(C(c3cc(Cl)ccc3O)=O)C2)cc(Cl)n1 97489,C1(C(=O)OCC)C(NCC(c2ccccc2)(C)F)C1(C)C 97490,CC1CC(C(=O)NCCCN(CCO)C(c2cncc(F)c2)=O)C(=O)O1 97491,N(C1CC(C)n2ncnc21)C(N1CCN(CCOCC=C)CC1)=O 97492,C1(NC(c2cnn(C(C)(C)C)c2Cl)=O)CC(F)CN(C(c2ccc(F)cc2)=O)C1 97493,c1(-c2ccc(CC(C)C)cc2)cnc2ccc(C(=O)Nc3ccnc(O)c3)cn12 97494,N1(C(C(C)=CC2CC2)=O)CC(C(=O)NCC(O)C(C)C)CCC1C 97495,CC1CNCC2(CC2)C(=O)NC2CC(C2)NC(=O)C1.c1(CCC2CC2)ccc(F)cn1 97496,N1(C(CCC#CC)=O)CCC(CCNC(=O)CSS(C)(=O)=O)C(F)(F)CC1 97497,C(CCCCC(=O)N1CC(N(C)C)C(C)(C)C1)N(C)C(c1ccnn1C)=O 97498,c1(CC(=O)NC2CCCN(C(CC3(C)CCCO3)=O)C2)ncn2c1COCC2 97499,c1(-n2c(C(=O)NCC3C(C(=O)NCC(C)CO)CCC3)cnc2)ccc(Cl)cc1 97500,C(CCCC(=O)NC(C)(C)CN=[N+]=[N-])N(C)C(c1c[nH]nc1Cl)=O 97501,C(C(=O)Nn1cnn(C)c1=S)N(CCC)C(C1(C(C)(C)O)CCC1)=O 97502,N1(C(c2cc(C)c(=N)[nH]c2)=O)Cc2ccccc2C1C(=O)NC(C)C(F)(F)F 97503,CC1CN(C(C2(O)CC3CCC2C3)=O)CCC1CNC(=O)CC(C)c1cnn(C)c1 97504,C1(C(=O)NC2(C)CCN(C(C3N(C)CCC3)=O)C2)CC2(CCCCC2)CO1 97505,C1(CC(=O)N(CCC(=O)NC(c2nocc2C(N)=O)C)CC)NC(=O)NC1=O 97506,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 97507,N1(C(C(CCC2CCC2)NC(C(C(CC)C)N(C)C)=O)=O)CCOC(C)(C)CC1 97508,C(C)(CO)(C(=O)NCC1CN(C(C2CCN(C(C)(C)C)C2)=O)C1)OC 97509,C1(O)(C(N2CC(NC(c3cnc(SC)s3)=O)C2)=O)CCCCCC1 97510,CC1(C#N)CC2CCC1N(C(C1COCCC1NC(=O)CN1CC3CC3C1)=O)C2 97511,C1(C(=O)NCCCC(=O)NC)CCN(C(=O)CCC2OCCO2)C12CCC2 97512,CCOC1CC2CC(C)=NOC(CCC)(CCC(=O)NC1)NC2=O 97513,N1(C(C(C)CC2CCC2)=O)CCOC2(CCN(C(=O)C(=O)NC3CC3)C2)C1 97514,C=CCCC(C)(C)C(=O)NC1CCCC1CNC(=O)C(CC)N(C)C 97515,c1(-c2cn(C)nc2)cc(C(=O)NCCC2(NC(N)=O)CC2)ncn1 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97691,C(=O)(C(C(C)CC)N(C)Cc1ccccc1Br)NCCCC=C 97692,N1(C(C2CC3CC3C2)=O)CCC2CN(C(=O)CC3CC3Cc3ccccc3)C2C1 97693,C(CC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccc(C)cc1)OC 97694,C1(C#N)(C(=O)NCC2C(NC(c3nc(N(C)C)oc3)=O)CCC2)CC12CCC2 97695,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C(C2CCC2)OC)C(C)C1 97696,C1(NC(c2cc(OC)ns2)=O)C2CCN(C(c3cc(F)c(F)cc3Cl)=O)CCC12 97697,c1(C(N2CCN(C(c3ccn(CC)n3)=O)C(C)C2)=O)ccc2[nH]c(=N)sc2c1 97698,c1(C(=O)NCC2CCCC3(CN(C(C(C)Br)=O)C3)O2)c(O)cccc1[N+](=O)[O-] 97699,c1(C(C)C)ccc(-c2cn(CCC(=O)N(C3(C)CCOC3)C3CC3)nn2)cc1 97700,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 97701,C(=O)(C(CC)C(C)O)NC1(CC)CCN(C(c2ccc(O)nn2)=O)C1 97702,CCCC(C(=O)N1CC(F)(CNC(c2nccnc2N)=O)C1)NC(N)=O 97703,C1(NC(C(CC)C)=O)CCCCCC1NC(=O)CCSc1ccc(Cl)cc1 97704,N1(C(c2cccc(OCC#C)c2)=O)CCC2CN(C(=O)C=CC(C)C)CCC2C1 97705,C1(C(N2CC3CC3(C(=O)NC3CCC3)C2)=O)CCC(C(F)(F)F)CC1 97706,C(=O)(CC1OB(O)c2ccccc21)N1CCC(NC(C(CC)(F)F)=O)CC1 97707,C1(C)(C(=O)NCC2(F)CN(C(C3CCCC(C)(C)O3)=O)C2)CCCCNC1=O 97708,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 97709,C(=O)(C(F)(F)C(F)(F)F)NC(CCCC)CNC(c1ccccc1Br)=O 97710,c1(OC)ccc(F)nc1NC(C1CCCC1NC(c1c(O)cccc1F)=O)=O 97711,C1(CC(=O)NCC2(CO)C(C=C)C2)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 97712,N1(C(COCCCC)=O)CCN(C(=O)CC2COC(C)(C)CO2)C(C2CCC2)C1 97713,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CCCc2ncc(C)o2)CC1(F)F 97714,c1(C(=O)NC2C(NC(C(C)C(F)(F)F)=O)COC2)cc2cc(Cl)ccc2[nH]1 97715,c1(N2CC(C)(C(F)(F)F)C2)ncc(C(F)(F)F)cc1Cl.C12(CC1)C(=O)N2 97716,c1(C(N(CC(CC)NC(=O)C(C)n2cnnn2)C)=O)ocnc1C1CC1 97717,c1(CCN(C(=O)CC2CCN(CC3CCOCC3)C2)CC)c(F)cccc1F 97718,C1(C(=O)NCC2N(C(CCCCCC=C)=O)CCC2)CCC2(CC1)CCC2O 97719,c1(C(=O)NC2CN(C(c3c(N)ncc(C)c3)=O)CC2F)cn2ccncc2n1 97720,CCC1=C(C(=O)NC2C=CC(CC(=O)NCCC(C)(O)C3CC3)C2)CCCO1 97721,c1(C(N(C)CCNC(=O)CCCc2cnn[nH]2)=O)ccc2oc(O)nc2n1 97722,N1(C(c2ccc(C(C)C)nc2)=O)CCCN(C(c2cccc(F)c2)=O)CC1CO 97723,C1(CCOC)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)CSC 97724,c1(NC(CC2(NC(C3N(C)CCCC3)=O)CCC2)=O)c(C#N)ccc2ccccc12 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97742,Cc1cc(NC(=O)CC(C#N)c2nc(C3CC3)nn2CCCN(C)C)ccn1 97743,c1(CC(N2CCN(C(=O)C(F)(F)C(F)F)CC(O)C2)=O)cncc2ccccc12 97744,CCC(CC)CCCC(=O)NCC=CC(=O)NCCCN1CCOC1=O 97745,C1(C(=O)NC2CCC(CNC(c3cccc(C4CC4)c3)=O)C2)CC2CCC1C2 97746,C12(NC(C3N(CC)CC3)=O)CCCN(C(=O)CCCCOC)CC1C2 97747,Cc1cc(=NC2CC3(COC(C)(C)C3)C2)[nH]c(=NCc2[nH]c(=N)ccc2C)[nH]1 97748,C(C(C)(C)CC(=O)NCCN1CCC1)NC(CSCC)=O 97749,c1(N2Cc3c(C)cccc3CC2)nc(=NCC(C)CCO)[nH]c2ccccc12 97750,C1(NC(=O)C(C)n2cccc2)CCCC1.N(CCOC)(C(=O)C1CC1)CC 97751,c1(C(C)C)ncc(NC(=O)NCCCN(C)C(C)C)cn1.C1C(=O)N1 97752,C12(CC(C(F)(F)F)(NC(C3(C)CC3C)=O)C1)CNC(C)C(=O)N2.C(CC#N)OC 97753,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(C)C(C(=O)NCc2ccc(F)cc2C2CC2)C1 97754,Cc1cc(C)c(C(=O)NCCCCC(C)NC(=O)C(C)(C)C2CCCO2)cn1 97755,N1(C(C(C(C)C)N2CCCC2=O)=O)CCc2sccc2C1CC 97756,c1(CC(N2CC(NC(C(C)(C)C)=O)C2)=O)cncc(F)c1 97757,C1(C)(COC(C(C)C(C)c2ccccc2F)=O)CCCCC1(C)C 97758,c1(OC)cc(C(N2CCCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)cc(C)n1 97759,n1(CC)cc(Cl)c(C(N2CCC(N(C(=O)CC3CCS(=O)(=O)C3)CCO)C2)=O)n1 97760,C1(C)(CC(=O)NCCOC2CCN(C(C3(C(C)C)CC3)=O)C2)CCS(=O)(=O)N1 97761,N=c1[nH]c2c(s1)CN(C(=O)C1=NOC(c3ccccc3)C1)CC2.C12CC(C1)O2 97762,CCCC(C(=O)N1CC2CC1(CNC(c1c(C)ncn1O)=O)C2)S(N)(=O)=O 97763,C1(CCNC(C(C)NC(C2CCCC2)=O)=O)CCCCN1C(=O)Cn1cnnn1 97764,C(C)(C(C)C(=O)NC1C(C)CCC1C)NC(C1(OCC)CC1)=O 97765,CCCCC(C(=O)NCC(C)(C)NC(c1cnnc(O)c1)=O)C(C)C 97766,C(=O)(C1CCCc2c[nH]nc21)N(CC(C)NC(=O)CC1COC(=O)C1)C 97767,c1(SC)cc(C(=O)NCC2CC(NC(C3CC=CCO3)=O)C2)nn1C 97768,c1(C(=O)NCC2CC(NC(c3cc[nH]n3)=O)C23CCC3)c[nH]c2cnccc12 97769,N1(C(C(C(=O)OCC)F)=O)CC2CCC1C1CN(C(=O)C(C)(F)C(C)(C)F)CC21 97770,C(C(C(C)C(C)C)Nc1cncc(F)n1)NC(c1cncc(OC)c1)=O 97771,C1(c2n(C)nnn2)(NCc2ocnc2C)CC2CC1CC2F.c1nn[nH]n1 97772,n1(CC(N2CC(O)(CCNC(C(C(C)C)OCC)=O)C2)=O)cnc2ccccc12 97773,c1(OC)ccncc1C(=O)NC(C1CCN(C(=O)CNS(N)(=O)=O)C1)(C)C 97774,c1(NC(C2C(C(=O)NC(CC#C)C)C2)=O)ccc(O)nn1 97775,N1(CC(N2CCN(c3cccnn3)CC2)=O)CC2COCC(CO)(C1)C2O 97776,CC(O)(Cn1ccccc1=O)C(=O)NCC1CC(NC(c2cnc[nH]2)=O)C1 97777,Cc1ccc2c(=NCc3ncc(C)s3)[nH]c(=NC3CCCSC3)[nH]c2c1 97778,c1(NCC(COC)(C)CO)[nH]c(=NCCc2ncccc2C)nc2scnc12 97779,N1(C(C2CCC(C)O2)=O)CCC(C)(CNC(C2C=CS(=O)(=O)C2)=O)CC1 97780,c1(C(N2CC3C(C(=O)NC(COCCC)(C)C)(C3)C2)=O)ccc2c(c1)C(=O)CC2 97781,N1(C(CCC(=O)NC)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 97782,N1(C(C(CC)OC)=O)CC2(C1)CN(C(=O)C(CC(C)C)OC)CC2COC 97783,N1(C(C2C(C)CC(=O)C2)=O)CCN(C(c2cnn3ncccc23)=O)C2(CCC2)C1 97784,C1(C(=O)NC(=O)CSC2CCCCO2)(NC(CSCCOC)=O)CCCCC1 97785,CC(C)C(C)C(CN(C)C)NC(C1(c2ccc(OC(F)(F)F)cc2)CCCC1)=O 97786,C(C(=O)N(C(C(=O)N(C)Cc1ncc[nH]1)C1CC1)C)(SC)SC 97787,c1(C(=O)NC2CN(C(=O)C(F)CC3CCCCC3)CC2F)ncc(Cl)cc1O 97788,N1(C(C(CC#C)(C)NC(c2ccncc2OC)=O)=O)CCN2CCCC2C1 97789,c1(C(=O)NCC(CNC(=O)C(C)=CC(C)(C)C)OC)ccc(Cl)s1 97790,C1(N(C(Cc2cc(CC)no2)=O)C)CCCC(NC(c2cc(OC)n(C)n2)=O)C1 97791,C1(C(N)=O)CCCN(CCC(=O)NC2CN(C(C3CCN(C)CC3)=O)CC2O)C1 97792,n1(CC)ncc(C(=O)NC2CCCCC2CNC(c2cn(C)cn2)=O)c1C 97793,C1(C(C(=O)NC(CC)C)NC(C)C)C2CCCC12.C(C)(CC)N 97794,N1(C(C#CC(OCC)OCC)=O)CCC(F)(CNC(c2cnnc(O)c2)=O)C1 97795,C(CCN=c1nc(N2CCC(C)C3(CCCCC3)C2)cc(C)[nH]1)OCC 97796,C#Cc1ccc(F)c(C(=O)NC2CCN(C(=O)C(C)(CO)OC)CC2)c1 97797,c1(C(N2CC(CNC(C3(c4ccno4)CC3)=O)OCC2)=O)cc(F)ccc1CO 97798,CCC(CNCC1CCN(C2CC2)C1)(CC)C(=O)Nc1ccc2cc[nH]c2n1 97799,CC1CN(C(C2CN(C(c3csnc3Cl)=O)CCN2C)=O)CC(=O)N1C 97800,C1(NC(c2c(OC)csc2)=O)CCN(Cc2c(C)noc2C)CC1(C)C 97801,CCC(CC(=O)N(CCC(C)NC(c1ccn(C(C)C)c1C)=O)C)C(F)F 97802,c1(C(C)C)nc(C(=O)NCCCNC(C2CCCC2C(F)F)=O)co1 97803,c1(C(=O)NC2(CCCNC(=O)Cc3cncs3)CC2)cc2nc(Cl)ccc2s1 97804,c1(C(=O)NC(C(=O)N(CCC(O)CO)C)Cc2ccoc2)nnn(C)c1N 97805,C1(C(N(CC(CNC(C(C)=C(CC)C)=O)O)C)=O)C2Cc3cc(Cl)ccc3C12 97806,N1(C(C(C)SCC)=O)CCOC(CCNC(C2(c3cccnc3)CCCC2)=O)C1 97807,C1(C(=O)Nc2ccc(OCC(=O)OC)cc2)CCCCC1(OC)OC 97808,N1(C(Cn2c(C)nc(C)n2)=O)CCC(C(=O)NC(c2nncn2C)C)CC1(C)C 97809,N1(C(C2ON=C(C)C2)=O)CC2CN(C(c3cc4cnccc4o3)=O)CC2(C)C1 97810,C1(NC(CC=C)=O)CCN(C(=O)Cc2occc2C)C1C1CC1 97811,C1(C(=O)NC2C(CNC(c3nc(C)c(C)s3)=O)COC2)CCC(=O)N(C(C)C)C1 97812,c1(N(C(C)=O)C)cccc(C(=O)NC2CCC(NC(c3cncs3)=O)CC2)c1 97813,CC(CC(=O)N1OCC(F)(F)C(=O)NCC(C)C1)C(C)(C)C 97814,CC(CC(=O)NC1CN(C(=O)C(c2cccc(Cl)c2)=O)C1)C(=O)c1ccccc1 97815,c1(NC(C(CCC)NC(c2cn3ccsc3n2)=O)=O)cnc(C)c(C#N)c1 97816,CCCCCCCCCCCC(=O)NCC1CCCN(C(=O)C=CC2CCC2)C1 97817,c1(C(N2CCC(C(=O)NCCC(C)(C)OC)C2)=O)c(C)nsc1N 97818,c1(C(N(C(CC)CNC(=O)C(C)OC(C)(C)C)C)=O)nc(C)n(C2CC2)c1C 97819,C1(NC(c2cnc[nH]2)=O)CN(C(=O)CC2CC3(CC3)C2)C2(CCCCCC2)C1 97820,C1(NC(C(C)OCCC=C)=O)CCCC12CCN(C(c1cc(Cl)sc1Cl)=O)CC2 97821,c1(Nc2ccc(-c3c(OC)nccc3)cn2)ccn2nccc2n1 97822,N1(C(c2ccc(-c3ccccc3)s2)C(=O)NN2CCOCC2)CC(F)(C2CC2)C1 97823,N1(C(C(=O)NCC)=O)CCOCC1CCNC(=O)C(F)(F)C1CC1 97824,C1(C(=O)NCC(C)N(C(c2ccc(C)o2)=O)CC)CC2(CCOC2)C1 97825,N1(C(=O)NC(C)C=O)CCC2(CCC(C)O2)CC1.Cc1csc(CNC(C)C)n1 97826,c1(C(=O)NCC(CC=C)NC(=O)CC2CC2C(F)(F)F)ncccc1Cl 97827,C(=O)(N=c1nc(C2CCC3(CC3)C2)[nH]s1)c1c(C)n[nH]c1.C1CCC1 97828,Cc1cc(N2CCCC2C2(NC(=O)C(C)C(C)C)CC2)ncc1[N+](=O)[O-] 97829,c1(OC)c(NC(=O)CC2CCN(Cc3c(F)ccc(C)c3F)C2)ccc(F)c1F 97830,N1(C(c2ccc(O)nc2)=O)CC2(C=C(C(=O)NC3COCCC3(F)F)CO2)C1 97831,N1C(CC(=O)NCC2(C(=O)NCCc3cc[nH]n3)CCC2)CCOCC1=O 97832,C1(C)(CC=CCOC)CN2CCC1(N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)CC2 97833,c1(N(c2n(C)nnc2)C(C2CNC2)C2CCC2)ccn2ncc(Br)c2n1 97834,C1(C(N(CCC(=O)NCC(CCC)OCC)CC2CC2)=O)CC(C)(C)CCO1 97835,C(=O)(C1=CCCCC1P(C)(C)=O)NC1CCC(NC(c2ccc(OC)s2)=O)C1 97836,c1(C(N2CC(C)(C)C(NC(C3CC(O)C3)=O)C2)=O)cncc2[nH]c(=N)sc12 97837,N1(C(c2c(C)cco2)=O)CCC(C(=O)NC(c2ccncn2)C)C12CCC2 97838,C1(NC(=O)COc2ccsn2)CCCC(N(C(=O)Cc2nnc(O)s2)C2CC2)C1 97839,N1(C(C2(C)CCN(C(c3ccc(COC)o3)=O)C2)=O)CCC2CCCC2C1 97840,N1(C(CCCCOC)=O)C2CCC1CC(NC(=O)C(C(C)(C)C)NC(N)=O)C2 97841,CCC(CC)CC(=O)N1CC=CC(OCCOCC=CC(=O)OC)C1 97842,N1(C(c2n(C)nc(C3CC3)c2)=O)CCC(NC(C2CCC(O)C2)=O)C12CCC2 97843,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 97844,c1(C(=O)NCCCn2cc(C3CCCC3O)nn2)cnn2cccc(Cl)c12 97845,c1(NC(=O)OCC)ccc(NC2(c3ccccc3Cl)CCOCC2)cc1 97846,c1(C(=O)Nc2cn(CCC)nc2)c(C)sc2ccc(Cl)cc12 97847,CC1CCCN(C(c2cnc(C(N)=O)s2)=O)C1CNC(C1CC(O)C1)=O 97848,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(C(C)SCCOC)=O)=O 97849,c1(CC(C(=O)NC2(C)CC(NC(C=CC)=O)C2)C)ccc(F)cc1Cl 97850,Cc1cc(Br)cc(C(N2CCC(O)(C(=O)NCc3cncnc3)C2)C(=O)N(C)C)n1 97851,c1(CC)cncc(-c2cn(C(C)C(=O)NC3CC3OC(C)C)nn2)c1 97852,c1(CN(C(=O)CC2(NC(=O)Cc3ccc(F)nc3)CCC2)CC)cccnc1F 97853,O(N1CCC(CC(=O)NCC(C)(C)CCNC(=O)CC(C)COC)CC1)CC 97854,C1(NC(C2(CC(=O)OC)CC2)=O)CCOCC1NC(=O)Cn1cnc(C(N)=O)c1 97855,C1(C(C)CNC(=O)C(C)n2cccn2)CCN(C(c2ccnnc2Cl)=O)CC1 97856,c1(C(C)C)ccc(F)cc1C(N1CCC(NC(=O)C(O)C2CC2)C(O)C1)=O 97857,C#Cc1cccc(CC(=O)NCC2(NC(c3ncccn3)=O)CCCCC2C)c1 97858,C1(C(=O)NC(CNC(C=CCC(=O)N(C)C)=O)(C)C2CC2)CCSCC1 97859,OCC1N=C2NC(=NC3CCCCC23)Nc2ccc(Cl)cc2C1CCCC 97860,c1(OC)ccc2c(c1)OCC(C(=O)N1CCN(C)C3(CC3)C1)=C2 97861,N1(C(c2cnc(SC)s2)C(=O)NCC)CCN(CC)CC1C 97862,c1(C(N(C2CCN(C(c3cc(C)on3)=O)C2)CCO)=O)cc(N)cnc1C 97863,O=C1NC(=O)C2(CCN(C(=O)C(=O)NC3CCC4CC34)CC2)N1 97864,O=C(C1=CCCC1)NC1CN(c2cc(-n3ccnc3)ncn2)CC1F 97865,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 97866,c1(C2(C(=O)NCCC(=C)CNC(c3cnc(O)o3)=O)CC2)ccc(SC)cc1 97867,Cc1cc(C(N2CCCC(CNC(=O)C(C)CF)C2)=O)cc(I)c1 97868,c1(C(C2CCCOC2)(F)F)nccnc1-c1nc(-c2ccoc2)n[nH]1.C1CCCC1 97869,N1(C(c2cc(O)cs2)=O)CCC2CN(C(c3cc(=O)cc[nH]3)=O)CC2C1 97870,C1(C(=O)NCC2C(C)CN(C(=O)COC3CC=CC3)CC2)OCCOC12CCC2 97871,c1(C(=O)NC2CCC(NC(c3c(N)cc(Cl)nc3)=O)CC2)n[nH]c2c1CCSC2 97872,C1(NC(CCNC(COC)=O)=O)CCCCN(C(=O)C(c2ccc(F)cc2)C)C1 97873,c1(C(N2CC(N(C)C(C3CCC(C(F)F)CC3)=O)C2)=O)cc(C#N)ccc1F 97874,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(=O)CC1CC2CCC1O2 97875,CCCCC(C)CCC(=O)NCC1(NC(c2ccc(O)cn2)=O)CCOCC1 97876,n1(C)c(N2CCOC(C(=O)OC)C2)nnc1C(C)C.c1(OCC)ccccc1.C1CO1 97877,C(N=C(NC1CC1)NC1CC(C)(C)Oc2cc(F)ccc21)c1c(C)ncs1 97878,C1(CNC(C2CN(C(C)C)C2)=O)CC(CNC(c2occc2C2CC2)=O)CO1 97879,n1(Cc2cn(-c3c(OCC)scc3)nn2)nc(C)c(Cl)c1C.N12C(CC1C)C2=O 97880,C(=O)(CCC(C)(C)F)N(C)CCNC(C1CCOC1C(F)(F)F)=O 97881,CC1(C)CN(C(C2COCCO2)=O)CC1NC(=O)COc1ccccc1F 97882,CC(C)(C)CC(C)(C)C(=O)N(CC(C(F)(F)F)C(F)(F)F)C.C1CO1 97883,Cc1ccc(C(=O)N(CC2CC2)CC2CC2)c([N+](=O)[O-])c1 97884,Cc1cccc(OCCCC(=O)NC2CCN(C(=O)CCOCC3CC3)C2)c1 97885,CCC(C)CCC(=O)NC1CCCCC1NC(=O)Cn1ccc(C(=O)OC)n1 97886,C1(CNCCCCSC)CCCCC(C)(C)C1 97887,c1(C=O)c(Cl)nc2ccccn12.C(=O)(C(COC)OC)N(CC(CC)OC)C 97888,c1(C(=O)N(C2CC2)CC2CCCN2C(c2csnn2)=O)coc2c1CS(=O)(=O)C2 97889,C1(C(N2C3C(NC(COCCOC)=O)C(C3)C2)=O)CCCC2(CCOC2)O1 97890,N(C(=NCCN1CCOCC1(C)C)NCC(OC)SC)C(c1cccc(C)c1)C#C 97891,C(=O)(CC#Cc1ccccc1)N(CCC(C)NC(C1(F)CC=CCC1)=O)C 97892,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 97893,C=CCC(C)C(=O)NC(C)Cn1cc(CNC(c2ccnn2C(C)(C)C)=O)nn1 97894,Cc1nn(C(C)C)c(C)c1C(=O)NCC(C1CC1)NC(=O)Cc1ccn(C)n1 97895,C1(NC(c2ccc(OCC(F)(F)F)o2)=O)(CO)CCCN(C(C2CCC(=O)O2)=O)C1 97896,c1(C(N2C(CNC(C(CCC)C)=O)CCCC2)=O)c(C)cccc1C 97897,C(=O)(C(O)CC(C)C)NCC(CNC(c1c(C)nc(COC)s1)=O)(C)OC 97898,C12(NC(c3nc(COC)oc3)=O)CCN(C(=O)CN(C)C(N)=O)CCC1C2 97899,c1(OC)nccc(NC(C2CCCN2Cc2cccc(O)c2)=O)c1F 97900,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 97901,C=CCCC(C(=O)NCCCC(N)=O)NC(=O)CC1C=CCC1 97902,N1(C(CCC2C(C)(C)C2)=O)CC2CC(C1)N(C(c1occc1Br)=O)C2 97903,C(C)(C)(C(=O)N(C)CCOCCCNC(c1ccn(-c2ccncc2)n1)=O)SC 97904,N1(C(=O)COCC2CCCCO2)CCN(C(=O)C(F)C2CC2)CC2(CC2)C1 97905,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(Cn1c(C(C)C)nnc1)=O 97906,C(=O)(CCCC(F)(F)CO)N1CCC(C(C)NC(c2nc(C#C)sc2)=O)CC1 97907,C1(C(C)(C)CNC(=O)NC2CCCCO2)CCCOC1c1ccccc1 97908,N1(C(C=C(C)C(C)C)=O)CCCCC1CCNC(=O)CC1CC(C)=NO1 97909,C1(C(N2C(CCC)C(=O)NCC2)=O)CC2CCN(Cc3n[nH]c(C)c3C)CC12 97910,c1(C(=O)NC2CCCN(C(c3cccc(CC)c3)=O)C2C)cc2cccnn2c1 97911,C1(SC)CN(C(C2(O)CC(F)(F)C2)=O)CC1NS(=O)(=O)CC1(C)CC1(F)F 97912,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1C(=O)O 97913,Cc1oc(C)c(C(N2CCC(NC(=O)CCCN3CCCCC3=O)CC2)=O)c1C 97914,C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2c[nH]c(=N)s2)=O)CC1O 97915,Cc1cccc(C)c1NC(=O)C(c1ccccc1Cl)N1CCC(CCC#N)CC1 97916,c1(CN(C)C(=O)Nc2cc(C(C)(C)C)ccn2)cc(C2CC2)ncc1Br 97917,c12cccc(c1)C(=O)C(=O)NCC(=O)N(C)CC(C)CNC2=O.CCOSC 97918,CCCC(C)(O)C(=O)NC1CC(CC(=O)Nc2ccc(CO)nc2)C1(C)C 97919,N1(C(CNC(=O)CCC2CC2(F)F)=O)CCOCC1C(=O)NCC1(Cl)CC1(F)F 97920,N1(C(C(C2CCCO2)NC(CCCCOC)=O)=O)CCC2(C1)CN(C)C2 97921,CC(F)(F)CC(=O)NCC(N1CCN(C(C2CCC2)=O)CC1)=O 97922,C1(NC(CC2(C(=O)OC)CCC2)=O)CCC(n2cc(-c3csc(C)n3)nn2)C1 97923,c1(C(=O)NC2COCCN(C(C3CC4(CCC4)CO3)=O)C2)ccc2ccnn2c1 97924,N1(C(CC(C)OCCC)=O)CCCC(CC(=O)NCC2(C3CCC3)CC2)C1 97925,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)C=Cc2cncs2)nc1 97926,CC(C)C1CCNC(=O)C(=O)N1.c1(C(=O)Nc2cn(C)nn2)cnn(C(F)F)c1 97927,c1(OC)cc(OC)cc(N(CCO)Cc2n[nH]c(Br)n2)c1 97928,c1(OC)ccccc1CC(=O)NC1CC12CC(NC(C1(C)CCCOC1)=O)C2 97929,N1(CC)CC(C(=O)N(C)CCNC(c2ncn(C(C)C)n2)=O)NC1=O 97930,CN1CCN(C(=O)Cc2cnn(C)n2)CC1CNC(=O)Cc1ccc(F)cc1Cl 97931,N1(C(C(CC#C)O)=O)CCCN(C(c2nc(C)n(C)c2C)=O)C(C)C1 97932,c1(C(N2CC(N(C(=O)C3=COCCO3)C)C(C)(C)C2)=O)ccnc2ccncc12 97933,c1(C(N2CC(NC(CN(C3CCC3)C)=O)C3C2C3)=O)ncc(Cl)cc1F 97934,CS(=O)(=O)c1cccc(S(=O)(=O)N2CCC3C(CCN3C(=O)CCNC(N)=O)C2)c1 97935,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)C(C)C#N)C)nc2C1 97936,N1(C(C(C(C)C)OC)=O)C(C)CN(Cc2ncc[nH]2)CC1C 97937,O(C=CC(=O)N1CCC(N(C)C(C2CC(O)C2)=O)C1)CC 97938,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 97939,N1(C(C2(OC)CC(F)C2)=O)CCCC(C)C1c1cn(-c2cc(C)cc(F)c2)nn1 97940,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(c4ccccc4)CC3)=O)C2)C1 97941,C(=O)(C(C)CS(C)=O)N1CC(c2cn(CCN3CC(=C(C)C(C)(C)C)C3)nn2)C1 97942,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)cn1 97943,C(CC(=O)NC(C)CN(C(=O)C=C(C)C(C)C)C)N(CCC)C 97944,Cc1nc(C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)cn1C 97945,C1(CC)(CC)CC(C(=O)N(C2CC=CC2)C)CN1C(=O)C(n1nccc1C)C 97946,C(=O)(C(O)CC(F)(F)F)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O 97947,Cn1ncc2c(-c3csc(NC(c4ccc5c(n4)CCO5)=O)n3)cccc12 97948,CC12CC(C(c3nnnn3C3CCC3)Nc3cnnn3-c3ccccc3)(C1)C2 97949,Cc1cc(C(=O)NCC2CN(C(=O)CCc3cc(OC(F)F)no3)C2)no1 97950,C(C)(CO)C(O)c1cccnc1.Cn1nccc1C1(CC(N)Cc2ccsc2)CC1 97951,C12CCCC(C1)C(=O)N2C.C(C(F)F)NC(=O)CO 97952,CCCC(C)CC(=O)N1CC=CC(NC(=O)Cc2ccc(OC)cc2F)C1 97953,C(CC(C(=O)N1CCCC1C(C)C)NC(C1CC=CCC1)=O)OCC 97954,CCCCCCC(F)C(=O)NC1CCN(C(=O)Cc2cnc(C)nc2O)C1 97955,c1(C(=O)NC(CC=C)CNC(=O)COc2ccsn2)ccn2ncc(Br)c2c1 97956,N1(C(c2ccc(C)o2)=O)CCC(O)CC1C(=O)NOCC1CCC1 97957,N1(C(=O)OC(C)(C)C)CC2CCCC(C(=O)Nc3ncccc3F)(C2)C1 97958,c1(CC(=O)NCCCCCN(C(C(C)C)=O)C(C)C)cc(C(F)(F)F)nn1C 97959,c1(-c2cc(C(N3C(CNC(C(C)N4CCC4)=O)CC3)=O)no2)cccc(Cl)c1 97960,c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)CC2CCN(C)C2=O)c1 97961,c1(CCC(=O)NC(CC)CC(N)=O)ncccc1C.c1(C(=O)N)cn(CC(=O)OC)nn1 97962,CC1CC(C(=O)NCC=CCNC(=O)Cc2ccn(C(F)F)n2)CCS1 97963,c1(COC)cc(N2CCC(OC)(C)C2)nc(C(C)(C)C)n1.C1(=O)CN1 97964,CCC(O)CC(=O)N1CCC1CNC(C1CC1Cc1ccc(Cl)cc1)=O 97965,N1(C(CN2CCC(OC)CC2)=O)CC2CN(C(=O)CCC=C(C)C)CCC2(CO)C1 97966,N1(C(C(C)(C2CC2)OC)=O)CCC(NC(c2nc(C3CC3)ncc2Cl)=O)C(F)C1 97967,Cc1ccn(CC(=O)NCC#CCNC(c2sc(C(C)C)nc2C)=O)c(=O)c1 97968,C1(C2(C(=O)NCC(C3CCOCC3)C)CC2)CCCCN1C(c1csnc1Cl)=O 97969,CCCCS(=O)(=O)NC(C)C(=O)NC1(CNC(c2nnn(C)c2C)=O)CCC1 97970,N1(C(=O)COCC2CC2)CCN(C2CCOCC2)C(=O)C1 97971,C1(CN(C(C)=O)CC2CCCCN2C(=O)CCc2nncs2)CC(C)(C)CN1C 97972,C1(C(=O)NC2(CO)CCN(C(=O)CCc3nncs3)CC2)CCC2(CCOC2)O1 97973,N1(C(c2cnc(CC)s2)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)NC 97974,C1(CCNC(=O)C(F)CC2CCCC2)CN(C(=O)C=Cc2cc[nH]c2)CCCO1 97975,C(CN=c1[nH]cnc(Cl)c1CO)N(C(C1(C)CCC(OC)CC1)=O)C 97976,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 97977,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 97978,C1(CNC(COC(C)C)=O)COC(C(F)(F)F)CN1C(=O)CC1CCC(C)CC1 97979,CCC(C)C(C(=O)N(CC(O)CNC(=O)C(c1cccc(O)c1)C)C)OC 97980,C(=O)(C(CC(C)C)NC(C)=O)NC1C(NC(C2CCC(=C)CC2)=O)COC1 97981,c1(C(N2CCC(O)(C(N3CCOCC3)=O)C2)=O)c(F)cncc1F 97982,C#CCC(CC#C)C(=O)NCC1CCN(C(C2(C)CCN(C)CC2)=O)C1 97983,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 97984,CCC(O)CC(=O)N1CC(CC(C)NC(=O)Cc2cc(-c3cccs3)on2)C1 97985,C1(C(N2CCC(CN(C)C(N)=O)C2)=O)CCC2(CCC2)OC1.C12CN(C1)C2=O 97986,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 97987,N1(C(c2oc(C)c(CO)c2)=O)CCN(C(c2cc(CC3CC3)on2)=O)CC1C 97988,CN1CCOC2(CN(C(=O)CC3(NC(C4CC=CCC4)=O)CC3)C2)C1 97989,CC1CC(C(=O)NCc2ccc(Cl)cc2)N(CC2(O)CCOCC2)C1 97990,C(CC(F)F)(C(=O)NC1C2CCCC12)N(C(=O)CC1CC(F)(F)C1)C 97991,N12CCC(C1(C)C)NC2=O.N1(C(=O)OC)CC(NS(=O)(=O)C(F)(F)F)CC1=O 97992,C1(c2cn(CC3CC(F)(F)C3)nn2)(NC(=O)CC2CCCO2)CCCOC1 97993,C(=O)(CCCC(C)(C)NC(=O)C=Cc1cnn(C)c1C)N1CC(CC)(CC)C1 97994,C1(NC(=O)CCN2CCOCC2=O)CN(C(c2conc2C2CC2)=O)CCC1O 97995,N1(C(C2C(C)C2C)=O)CCOC(CCC(N2CCCC(C(=O)NC3CC3)C2)=O)C1 97996,C(=O)(C(CNC(c1cccc(F)c1)=O)C(C)(C)C)NC(C)CCO 97997,C1(CN)CN(C(=O)CSC(=O)NC(C)C(C(=O)C(C)(C)C)=O)CC1CO.C(C)(C)C 97998,c1(CNC2CCCC2)cc(Br)ccc1OC(F)(F)F.c12cc(c[nH]1)C(=O)NC2C 97999,C1(NC(C2N(C(CC)=O)CCCC2)=O)CCC(C)N(C(=O)C=Cc2ccoc2)C1 98000,N1(C(=O)CCCc2ccccc2)CCN(C(=O)C(O)c2ccco2)C(CCO)C1 98001,N1(C(CC2CCC(C#N)C2)=O)C2CC1CN(C(=O)COc1cccc(F)c1)C2 98002,O=C(CCCC(F)(F)F)NCC1CC(O)CN1C(=O)C(O)C1CCC1 98003,C(CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1SCC2)SC(C)(C)C 98004,CCCC(C)(O)CC(=O)NC(C)CNC(c1ncccc1-n1cccn1)=O 98005,c1(C(=O)NCC2N(C(CCCC(C)C)=O)CC2)ccc2c(c1)C(C)CO2 98006,C1(C(N(C2CCN(C(c3cc(C(F)(F)F)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98007,C1(n2cc(-c3c(OC)n[nH]c3)nn2)CC(C(=O)NCC2(C)CC(F)(F)C2)C(O)C1 98008,c1(C(=O)NC(CCCNC(c2nc(C)[nH]n2)=O)C)cn2cc(Cl)cnc2n1 98009,c1(CSc2c(NC(N3CCC(C)(NC(C)=O)C3)=O)cccc2)cc(C)cc(F)c1 98010,Cc1cc(C(F)F)n(CC(=O)NC(CNC(=O)C(C)CC2CCC2)C2CCC2)n1 98011,C1(C2(NC(=O)CN(C(=O)CCn3cncn3)CC3CC3)CC2)(OC)CCC1 98012,c1(CC(=O)NC23N(C(COCCCOC)=O)CC(C2)C3)c[nH]c2ncccc12 98013,CCCCCC(CC)C(=O)NC1CC(F)CN(C(c2ccc(C)nn2)=O)C1 98014,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98015,C(CC(F)F)(C(=O)NCc1cc(O)cc(F)c1)N(C)C(c1ccnc(CO)c1)=O 98016,C1(CN(C(Cc2nnc(C)s2)=O)C)CCC(CNC(=O)C(C)C(C)O)CC1 98017,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98018,N1(C(C=C(C)C(=O)O)=O)CCC2CN(C(c3cn4cccc(C)c4n3)=O)C(C)C12 98019,C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CCC1CCOC1 98020,C1(c2n(C)ccn2)CN(C(=O)CCC2(C)CC2)CCN1C(=O)CC=CCO 98021,c1(CNC(=O)NCCc2ccc(OC(F)(F)F)cc2)ccc2ncccc2n1 98022,N1(C(c2cc(F)c(C(F)(F)F)c(F)c2)=O)CCN(C2CCNC2=O)CC(O)C1 98023,c12nc(ncc1Cl)SC1CN(C1)C2=O.Cc1cccc(C(=O)NN2CCCC2)c1 98024,N1(C(=O)NC(CC=C)CO)CCN(C(C2CCCN2C(c2ccccn2)=O)=O)CC1 98025,Cc1cc(OC(C)C(=O)N(CCCNC(C2CC23CCSCC3)=O)C)cc(C)c1 98026,CC(C)C(C)COCC(=O)NCCOCCC(=O)NC(C1CC1)C1CC1 98027,c1(C(=O)NCC(C)(CO)NC(c2ccc(C(O)CF)cc2)=O)ccnc(Cl)c1N 98028,c1(C(=O)NC(COC)C(=O)NC23CCCC2C3)c[nH]c(=S)cn1 98029,c1(C(=O)NCC2(C)CCN(C(c3scnc3Cl)=O)C2)cncc2c1CCCC2 98030,c1(=O)[nH][nH]c(=O)[nH]1.c1(C(C)Cc2ccccc2)cc(Cl)cs1 98031,Cc1c(Cl)ccnc1C(N1CCC(N(C(=O)CC23CCC(CC2)C3)C)C1)=O 98032,C(=O)(CC(C)CC(C)(C)C)N1CCC(C(F)F)(CNC(c2ccc(C=C)cc2)=O)C1 98033,c1(COC)csc(C(=O)NC2CCCC2CNC(=O)C(C)SC)c1 98034,N1(C(CCC#C)=O)C2CCC1CN(C(=O)Cc1ccc(Cl)nc1F)C2 98035,C12(C(N3CC(O)CC(NC(c4ccncn4)=O)C3)=O)CCCC(CCC1)C2O 98036,C(C)(CCCc1ccccc1)(C(=O)NCS(=O)(=O)C1CCCC1)c1cn(C)nc1 98037,C(=O)(CCC(C)(C)F)NC(COC)CNC(=O)C(c1ccccc1)O 98038,CC1CCC(NC(=O)Cc2cc(Cl)ccc2Cl)CN1C(=O)CCCn1ccnn1 98039,C1(NC(c2c(CNC(c3cnncc3O)=O)cc[nH]2)=O)CC12CCCCCC2 98040,c1(C(N2CCC(NC(C=CCC)=O)C2)=O)c(C)c[nH]c1-c1ccccc1 98041,C1(C#N)(C(=O)NC(Cn2cc(CNC(CN3CC(C)C3)=O)nn2)C)CC12CCC2 98042,C(=O)(CCS(C)(=O)=O)NCC(C)(CO)NC(=O)CSCCc1ccccc1 98043,N1(C(C(CCCC)C)=O)CC(O)(C2CCN(C(C3(C)CC3(F)F)=O)CC2)C1 98044,C1(C)CCC2(CC1)OCCO2.CCCN=C(NCC1CC1)NC1CCNC(=O)C1 98045,c1(C2C(C(=O)NC3(C)CC(NC(C4(Cl)C(C)(C)C4)=O)C3)C2)ccncc1F 98046,c1(C(N(CC(C)NC(=O)C(c2ccc(C(F)F)cc2)C)C)=O)cc(Cl)cn1C 98047,C1(CNC(C(CC)=CC)=O)CN(C(c2nc(Cl)sc2Cl)=O)CCCO1 98048,Cc1nc2c([nH]1)CN(C(=O)C(CC(F)F)NC(=O)NC1CCN1C)CC2 98049,CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)NCc1ncon1 98050,N1(C(c2cc(SC)oc2)=O)CC(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C(C)C1 98051,c1(N2C3(CN(C(C)Oc4ccnc5[nH]ccc45)C3)CC2)cccc(F)c1[N+](=O)[O-] 98052,C1(C(N(CCOC)CCNC(=O)C=Cc2cnccn2)=O)CC2CCCCC2O1 98053,C1(CNC(C2(NC(C(CC3CC3)OC)=O)CC2)=O)CCCCC1(C)C 98054,c1(C(N(CCCCN(C(Cc2cc(C)sc2C)=O)C)C)=O)cc(O)nc(O)n1 98055,c1(C(=O)NCC(CN(C(CSC)=O)C)(C)C)cc(C)nc(N(C)C)n1 98056,C1(NC(C(C)=CC2CC2)=O)CCC(NC(=O)C=CC2CCC2)CC1 98057,Cc1ccccc1-n1nccc1NC(=O)OCC(C1CCC(=O)N1)=O 98058,Cc1cc(C(=O)NC2CC2NC(c2nccnc2C)=O)cc(C)c1Cl 98059,C1(NC(=O)CC2COCCO2)CCOC12CCN(c1ncc(O)cn1)CC2 98060,C(=O)(C1=CC(C)(C)C1)N1CCC(CC(C)NC(=O)CCC2CCCCO2)CC1 98061,c1(NC)c(C(=O)NCC2(F)CN(C(=O)CC(F)(F)F)C2)cccc1C 98062,CC1(C)Cc2c(cnn2-c2ccccc2)CN(C(c2cc(I)cs2)=O)C1 98063,C1(C(=O)NCCCCNC(C)=O)CCN(C(c2ccco2)=O)CC1 98064,O=S(=O)(c1cccc2c(Cl)nccc12)NC1CCC(NCc2cnc(O)cc2O)C1 98065,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C(=O)Cc3cn(C)cn3)C)C2C1 98066,C=CCC(C(=O)N(C(C(=O)NCC1CCSCC1)C1CC1)C)C(C)C 98067,N1(C(C=CC)=O)CCC(C(C)NC(C2(CCS(N)(=O)=O)CCC2)=O)CC1 98068,C1(NC(CCc2nnc(C)o2)=O)CC2CCC1N2C(c1cccc(O)c1)=O 98069,N1(C(CC2(C)CC2)=O)CCC(CCNC(C2CCOC2C(F)F)=O)CC1 98070,C1(OCC)CN(C(C2CCC(=O)N2)=O)CC1CNC(c1ccnc(CO)c1)=O 98071,C1(CNC(CCCOCC)=O)CCC(C)(C)CN1C(=O)CC1CC(OC)C1 98072,N1(C(CC2C(C)CCCC2)=O)CC2CN(C(=O)CCc3cscn3)CC(C1)O2 98073,N1(C(C2C(C=C)C2)=O)CC2CCC1C(NC(=O)CNc1cccc(F)c1)C2 98074,C(CC(C(=O)O)NC(c1nccnc1-c1ccccc1)=O)(c1ccccc1)OCC 98075,c1(C(=O)NC2(CC)CCN(C(=O)CCF)CC2)cccc2c1C(=O)NC2=O 98076,c1(N2CCC(C#N)C2)nc(=NC2C=CCCCC2)[nH]c2c1COCC2 98077,C(c1cccnc1)=C(C(=O)NCCCCCNC(c1[nH]cc(C(=O)OC)c1)=O)F 98078,N1(C(=O)OC(C)(C)C)CCC(C=CC(=O)Nc2ccn(C(F)(F)F)n2)CC1 98079,C1(C(N2C(C(=O)NC(COC)(C)C3CC3)COCC2)=O)CC2(C1)CC2(F)F 98080,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)ccc(F)c(Cl)c1N 98081,N1(C(C2(C)CC(F)(F)C2)=O)CCC(O)C(NC(C2CC3CC3C2)=O)C1 98082,c1(C(N2C(C3(C)CC3(F)F)CC2)=O)ccnc2c1CCC2O 98083,CC1(C)SCCN1C(=O)CCn1cc(-c2ccc(CCC3CCCCO3)cc2)nn1 98084,c1(CNC(C(C(C)NC(C(C)SCCCC)=O)C)=O)cccc(C)c1F 98085,C12(CNC(C3N(CC)CC3)=O)COCCN1C(=O)CN(C(c1cnc(S)[nH]1)=O)C2 98086,c1(CC)ocnc1C(=O)NC(C)C(CO)NC(c1cc(F)n[nH]1)=O 98087,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)Cc1cn(C)nn1 98088,c1(N2C3CN(C(C4(CC)CCOCC4)=O)CC2CC3)ncnc2cc(C#N)ccc12 98089,N1(C(Cc2c(C)ncnc2C)=O)CCC2CN(C(=O)CC3NC(=O)NC3=O)C2C1 98090,c1(N2CCCC3(NC(c4ccsc4Cl)=O)C(C2)C3)nc2cc(F)ccc2o1 98091,C(=O)(C(C)(C)C(=O)NCC)NC(C1CC(NC(C2(CC)CNC(=O)C2)=O)C1)C 98092,c1(OC)cc(OC)cc(C(C(F)(F)F)NC(=O)NCc2cc(Br)cc(Br)c2)c1 98093,C(C)(C)(CC(=O)NC1CC(CCC(N2CCCC(CC(N)=O)C2)=O)C1)OC 98094,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98095,Cc1cc(C(=O)N(CCCN(C(=O)CC2CC2C)C)C)c(C)n1-c1nccs1 98096,C1(C(=O)NC(C)CC(C)NC(C2(O)CCCCC2)=O)CCOC(C)(C)C1 98097,C1(CN(C)C(C2(O)COC2)=O)CCN(c2ccccc2Br)C1=O 98098,c1(C(c2nnnn2C(C)C)NCCCC2C(C)C2)cc(Cl)n(C)n1 98099,c1(C(N(CCN(C(=O)CCCc2cnn[nH]2)C)C)=O)cnn2cccc(Cl)c12 98100,C1(CNC(C2(C=C)CC2)=O)CN(C(c2ccc(-c3csc(C)n3)s2)=O)CCO1 98101,C1(NC(CN(c2cc(N3CCOCC3)ncn2)CCC)=O)CC12CCOC(C)C2 98102,c1(C(=O)NCCN(C(c2ccc(OC)o2)=O)C)cc(C(F)(F)F)nn1C 98103,n1(CCC)ncc(C(=O)NCCNC(C2CCCN2c2nccs2)=O)c1C 98104,CC(CCc1ccccc1F)C(=O)N(C)CC1CC(F)CN1C(=O)C(N)=O 98105,C1(CN(C(c2n(CC)nnc2)=O)C)COCCN1C(c1nncs1)=O 98106,C#CCC(C)(C(=O)N1CC(CC23CC(C2)C3)C1)NC(C1CC(O)(C#C)C1)=O 98107,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98108,C1(NC(c2cnn(CCC)c2C2CC2)=O)CC2CC1N(C(=O)C(C)=CCO)C2 98109,c1(CC)nc(C(=O)N(C(CNC(=O)CC2CCN(C(C)=O)C2)CC)C)co1 98110,N1(C(CCC(C)OC)=O)CCCC(C2CCN(C(=O)CCOC(C)C)CC2)C1 98111,C=CCCCC(=O)NCC1CCCC(CNC(c2cnc(C3CC3)o2)=O)C1 98112,C1(C)(NC(CC2(C)CCC2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 98113,C=CC1(NC(=O)C(F)CC2CN(C(c3cccc(CC)c3)=O)C2)CCOCC1 98114,c1(NCC2CCN(C(CNS(NC)(=O)=O)=O)C2)cc(S(=O)(=O)NCC)ccc1C#N 98115,CC#CCC(C)NC(=O)CN(C(c1cccnc1)=O)CC1CC1 98116,C(=O)(C(C)(C)C(=O)NC1CC1CNC(c1cc[nH]c1-c1ccccc1)=O)N(C)C 98117,C(=O)(C(CN=[N+]=[N-])NC(c1n[nH]c(C)c1C)=O)NCC1CCN(C(C)=O)C1 98118,N1(C2CN(CC(C(=O)NC(C)=O)Cc3ccc(C)cc3)C2)CC(O)CCC1=O 98119,CN=c1ncc(CNc2ncc(C)c(C(N3CC(C)(NC)C3)=O)n2)c[nH]1 98120,CCC1=C(C(=O)NCCC2CCCN(C(c3cnncc3OC)=O)C2)CCCO1 98121,N1(CCC(=O)NC23CC(C2)N(C(c2cnoc2C2CCC2)=O)C3)C(=O)CCC1=O 98122,c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)ccc(P(C)(C)=O)s1 98123,C1(C(N2CC(C)N(C(C3C(C)(C)C3(C)C)=O)CC2)=O)CC2(C1)NC(=O)NC2=O 98124,c1(C(=O)NC2CCCCN(C(C3N(CC)CCC3)=O)C2)c(C)c(C)nn(C)c1=O 98125,c1(CCNC(c2cnn(C)c2OC)c2n(CCOCC)nnn2)ccccc1C 98126,c1(C(N2C(CC=C)CN(C(=O)CSCCCC)CC2)=O)cn(C)c(=O)n(C)c1=O 98127,C(=O)(C#CC1CCOC1)N(CCNC(c1cnc(COC)s1)=O)CC1CC1 98128,N1(C(C2(C)N(C)CCC2)=O)CCCC(CO)(CNC(=O)CCc2cnccn2)C1 98129,c1(CCCCC)cc(C(=O)NC2(CO)CN(C(c3cc(C(N)=O)co3)=O)C2)n[nH]1 98130,c1(C(CC)N(C)C(=O)N(C)CC2CC=CC2)ccccc1 98131,C1(SC)CCCC1CC(=O)NCC1(C(N2CCC2c2cscn2)=O)CCC1 98132,c1(C(C)O)ncc(C(=O)N(C2CN(C(=O)COCc3nccs3)C2)C)s1 98133,CC(N=c1nc(N2CCC(CCF)CC2)c2c([nH]1)CSC2)C1CCCO1 98134,N1(C(=O)Cc2cc(Cl)ccc2Br)CC2(CCCN2C(=O)COCC2CC2)C1 98135,c1(OC)cccc2c1OCCC(C(=O)NCCNC(C13CCCCC1C3)=O)=C2 98136,N1(C(C2CN(C)C(=O)C2)=O)CC2(CCCC(CNC(=O)C(F)=CCCF)O2)C1 98137,c1(NC(c2cccc(OCCO)c2)=O)cc(-c2cn(CCCF)nn2)ccn1 98138,c1(OC(CC2C(COC)CC2)=O)cccc(F)c1C 98139,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98140,N1(C(CCCN(C(C)=O)C)=O)CC2CC2(NC(=O)CCC2CCCCCC2)C1 98141,C#CCC(C)(C(=O)NC1CC1)NC(=O)CCOC1CCCC1 98142,C1(NC(C)Cc2cccc(OC(C)(C)C)c2)C2CCOC2C1(C)C 98143,C(c1c(C)cccc1Cl)=CC(N1C2C(NC(CCC(C)OCC)=O)C(C2)C1)=O 98144,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98145,N1CCC(C)C(OC)C1.C(=O)(C1=C(C)OCC1)Oc1cc(C2CCCC(OC)C2)[nH]n1 98146,c12sccc1NC2=O.N1(C(C(N2CCOC2=O)C)=O)CC(O)(CCN(C)C)C1 98147,C(CC(F)F)(C(=O)N(C12CCC(CC1)CC2)C)n1cc(-c2cncc(C)c2)nn1 98148,c1(CCC(N2CCCC(O)(CNC(C3(F)CCCC3)=O)C2)=O)nc2ccccc2s1 98149,C1(CC(=O)NC2C(CNC(c3n(CC)nnc3)=O)COC2)CC(=O)NC1=O 98150,c1(C(CC(=O)O)C)cn(C)nc1C1CC1.c1(C(=O)OC)cc(C2CC2)on1 98151,c1(C(=O)NCC(CNC(=O)Cc2cc(C3CC3)no2)(C)O)cccc(OCF)c1 98152,c1(C(c2n(C3(C)CC3)nnn2)NCCOC2CCCC2)sc([N+](=O)[O-])cc1Cl 98153,c1(OC)ccn2cc(C(=O)N(CC(C)N(C)C(c3ccnc(C)n3)=O)C)nc2c1 98154,C(C(C(=O)NCCCC(=O)Nc1ccn(C)n1)OC)OC 98155,c1(C(=O)NC2C(CNC(C(C(=O)OC)(C)C)=O)CCCC2)cnc2[nH]nnc2c1 98156,c1(C(=O)NCCOCCNC(C(C(C)SC)O)=O)c(C)oc2ccccc12 98157,CC(CC(=O)N1CCOC(CC(=O)NCC(F)Cl)C1)C(C)(C)C 98158,CC1(C)CC(C(=O)NC(CCO)C2CCC2)CN(CC(=O)N(C)C)C1 98159,Cn1nc(CNCc2ccc(-n3ccnc3)c(Cl)c2)c(I)c1Cl 98160,Cn1cc(-c2cc(C(=O)NCC3(F)CC(NC(C4CC4F)=O)C3)n[nH]2)cn1 98161,C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1CCN(C(c2ccc(OC)cn2)=O)C1 98162,N1(C(C(C)OCCC(C)C)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(C)C1 98163,N1(C(C(C)(C)C2CCCC2)=O)CCC(O)(CNC(=O)CNS(N)(=O)=O)C1 98164,Cc1ccc(C(N2CC(NC(c3nc(O)c(C)s3)=O)CC(C)C2)=O)c(N)c1C 98165,N1(C(CC2CC(SC)C2)=O)C(C)CN(C(=O)CC2CCC(C)(C)O2)CC1C 98166,C(=O)(C#CC1CCOCC1)N(CCN(C(C(Cc1c(C)noc1C)C)=O)C)C 98167,C#Cc1cccc(C(=O)NC(CNC(c2ccc[nH]2)=O)CCOC)c1F 98168,C=CCCCCC(=O)NC(c1ccccc1)CNC(=O)C=C1CCCCC1 98169,C(=O)(C(C)(C)CC(C)(C)C)NC1CCC(CNC(C(C)C(C)(C)C)=O)C1 98170,c1(C(=O)NCC2(NC(c3cc(C#N)c(Cl)cc3)=O)CC2)ccc([N+](=O)[O-])c(N)n1 98171,c1(C(=O)NCC2N(C(c3cc(SC)ncc3)=O)CC2)ccc(N)c(C)c1C 98172,c1(NC(C(CC=C)NC(=O)C(CO)N(C)C)=O)cccc(C)c1C 98173,c1(C(=O)NC(C2CCN(C)CC2)C2(O)CC(OC)C2)cccc2c(Br)cccc12 98174,N1(C(c2ccc(CSC)cc2)=O)CCN(CC2CCC(F)C2)CC1C 98175,c1(C(N(C)CC2(O)CCN(C(Cc3nc(CC)sc3)=O)C2)=O)cccc(N)c1C 98176,N1(c2c(C#N)ccnn2)CCC2(CC1)OCCCC2NC(=O)C(F)OC(F)(F)F 98177,c1(C(N(C(C)CNC(=O)C(C)(O)c2ccccc2)CC)=O)cc(F)c(Cl)cc1Cl 98178,c1(NC(CNC(CC(CCCC)CC)C)=O)ccc2c(=O)n(C)c(C)cc2n1 98179,c1(OC(C)C)ccc(CNc2cc(NC(C3CC(O)C3)C)ncn2)c(F)c1 98180,C1(C(=O)NCCCn2cc(C3CC(=O)C3)nn2)Cc2ccccc2CO1 98181,N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)C(O)C1CCC1 98182,c1(C(=O)NC(CNC(C(CCC)N(C)C)=O)(C)C2CC2)cc(C)c(C)nn1 98183,N1(C(c2cccc(CC)c2N)=O)CC2(C1)OC1(C)CC2(NC(c2ccco2)=O)C1 98184,c1(CC(C(C)(C)C)N2CCCC2)ccc(F)cc1Br 98185,C1(C(N(C2CCOC2)C)=O)(CF)CCN(C(c2ccn(CCF)n2)=O)C1 98186,N1(C(c2cc(C)nnc2)=O)Cc2occ(C(=O)NC(CO)C3(C)CC3)c2C1 98187,CCCC(C)CC(C(=O)NC1CC1)N1CCN(C(=O)OC)CC(C)(F)C1 98188,C1(CCC)CN(C(=O)C(O)COC)CC1C(=O)NCc1cc(C2CC2)no1 98189,C(C)(C(=O)NC1CC(CO)N(C(=O)COc2ccc(C#N)cc2)C1)(C(C)C)OC 98190,C1(CNC(=O)CNC(c2cnco2)=O)CC(CNC(c2ccccn2)=O)CO1 98191,C1(CNC(=O)NC(c2ccc(C)cc2Br)CCC#N)CC(C)c2ccccc2C1 98192,N#Cc1cnc(N2CCC(F)(F)C(CNC(c3cccc(Cl)n3)=O)C2)c(Cl)c1 98193,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(Cc3c(F)cccc3Br)CC12 98194,C(c1ccc(C)cc1)=CC(=O)NC(CC#C)C(=O)NCCc1n[nH]c(C)n1 98195,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cn(C)nn3)=O)c2n1 98196,CC(=O)CCCCC(=O)NCC(CNC(=O)CCc1cc(Cl)no1)C(F)(F)F 98197,CONC(=O)C(=O)N1CCC(C(C)(C)C(=O)NCC2C3CCCCC23)C1 98198,C(CCC1CCC1)(C(=O)NOCCN(C)C)NC(C(C(=O)OC)OC)=O 98199,c1(-c2ccc(CNC(c3nc(Br)cs3)=O)cc2)cc(C(F)(F)F)ccc1O 98200,C(=O)(CN1C(=O)Cc2ccccc21)N1CCCC(N(CC(O)C(=O)O)C)C1 98201,C1(NC(C(C(C)C)(C)O)=O)COC2(CCN(C(=O)C(=O)N(CC)CC#N)C2)C1.C(C(F)F)O 98202,c1(C(N2CC(CC)C(OC)C2)C(=O)NCC(C)C)c[nH]c2cc(Br)ccc12 98203,c1(C(N(C)CC2(NC(C(CCC)C)=O)CC2)=O)ccc2occ(C)c2c1 98204,C1(CNC(C(C)N(C(C)=O)C)=O)CCC(CSC)O1 98205,N1(C(CCCC2C(C)C2)=O)CCC2(CCCC2NC(c2nsnc2O)=O)CC1 98206,C1(C(=O)NCC2CC2(Cl)Cl)CCC(O)CN1C(c1c[nH]nc1Cl)=O 98207,c1(NS(C)(=O)=O)cccc(C(=O)NCC2(NC(C3CCC(O)C3)=O)CC2)c1 98208,C1(C(N(C2CCCCC2O)C)=O)(CO)CCN(C(C2CCOC2C(F)F)=O)C1 98209,C12(NC(C(c3ccn(C)n3)C)=O)CC3CCC(C1C2)N3C(=O)Cn1cnnc1 98210,N1(CCSC)CCCC(CNC(C2CCCS2(=O)=O)=O)CC1 98211,c1(C(N(C)CC2(NC(c3cc(C(=O)OC)sc3)=O)CC2)=O)noc2c1CCCC2 98212,c1(C(=O)OCC)cccc2c1N(C(C(=O)OCC(C)(C)C)c1ccoc1)CCC2 98213,c1(CCC(=O)NC2CCC(NC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98214,C(=O)(CCS(C)(=O)=O)N(CC(N1CCC(C(N)=O)CC1)=O)Cc1c(C)onc1 98215,c1(CC(=O)NCC(CC)NC(=O)C(F)CC2CC2)cc(OCC)cc(F)c1 98216,n1(Cc2nc(C(C)(F)F)sc2)ncc2ccc([N+](=O)[O-])cc2c1=O 98217,C1(C(=O)NCc2n(CC)ncn2)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98218,C1(CC(C)NC(C(=C(C)C2CC2)F)=O)CCN(C(=O)CN(C)C(N)=O)CC1 98219,C(=O)(CS(=O)(=O)CC(F)(F)F)NCC1N(C(C(C)OCC2CC2)=O)CC(C)(C)C1 98220,C(=O)(C1c2c[nH]nc2CN1C(=O)CC(=O)N(C)C)N(CCC)C(C)C 98221,C1(CNC(C2CCCN(C)C2)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 98222,c1(CCCC)cc(C)nc(N2CCOC(CNC(c3cc(=O)cc(Cl)[nH]3)=O)C2)n1 98223,C1(CC)CN(C(=O)Cc2cnns2)CC1NC(c1ccc(C(C)(C)CC)cc1)=O 98224,CC1C(=O)NC2(CCC2)CN1C(=O)CC1CC2(CCOCC2)C1 98225,C#Cc1cnn(C)c1C(N1CCC(C(C)NC(=O)C(CCC)OCC)CC1)=O 98226,c1(SC)cccc(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)c1O 98227,N1(C(C2(NC(CC)=O)CC2C)=O)CCC2(CNC(=O)O2)C1 98228,c1(C(=O)NCCN(C(=O)CNC(c2ccc(Cl)cc2)=O)C)c[nH]cc(Br)c1=N 98229,c1(C(=O)NC2CN(C(C3(OC(C)=O)CC3)=O)CC(C)C2)c(Cl)ccc(OC)c1N 98230,c1(COC)nccc(=NCC(C2CCCC2)OCCNC(=O)CC2CC2(Cl)Cl)[nH]1 98231,C1(C(C2CC2)NC(=O)C=O)CCNCC1.NC1(CC(N)=O)CC1 98232,C(=O)(C1=C(C)CCOC1)N1CC2C(C(=O)NC(c3ccnn3C)CC)(COC2)C1 98233,c1(C(N2CC(CCNC(C3CC(C)(CC)C3)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] 98234,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2cc(N)c(Cl)cn2)=O)C1 98235,C1(CC(=O)NCCC(CNC(=O)CC2OCCCO2)OC)CCCN(C)C1 98236,c1(C(=O)NCCC2CC(C)C2)cc(CNC(c2cscc2Cl)=O)nn1C 98237,c1(CC(=O)NCC(CNC(C(CCCC)O)=O)C)coc2c(Cl)c(Cl)ccc12 98238,C1(C[SH2]C)C(C)N(C)CCN1C.C1C(N)C1C 98239,c1(CC)cccc(C(N2CCC(CNC(C3(C)C=CCC3)=O)C2)=O)c1N 98240,c1(CCC(=O)NC(C(=O)NCCOCCC#C)c2ccoc2)cccnc1 98241,C1(CNC(c2ccc(C(C)(C)C)o2)=O)COC2(CCN(C(c3cc[nH]n3)=O)C2)C1 98242,c1(CC)cc(C(=O)NCC(c2ccccc2)N(C(=O)C=CBr)C)cn(C)c1=O 98243,c12ccc(cc1)S(=O)(=O)N2.CC1CCC(C#N)(NC(C2CCCO2)=O)C1 98244,N1(C(c2cc(C)c(F)cc2)C(=O)O)CC2CCN(C)C2C1 98245,C(S(=O)(=O)C(F)(F)F)c1cn(C(C(=O)NCC(CC)SC)C(C)C)nn1 98246,Cc1c(C(N2CCC(CNC(C3CC4CC3C4)=O)CC2)=O)oc2c(Cl)cccc12 98247,c1(C(N(C2CCC(NC(c3cocc3Cl)=O)C2)C)=O)cc(F)ccc1N 98248,c1(C(C)=O)cc(=NCC2CN(C(C3CCCCC3O)=O)CCO2)[nH]cn1 98249,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(C)O)C1 98250,CC1C(=O)N(C)CN1C(C1CC=CCC1C(=O)OC(C)(C)C)=O 98251,c1(NC(C(C(C)ONC(C2(SC)CCCCC2)=O)(C)C)=O)cccc([N+](=O)[O-])c1 98252,C12(CC)CCC(NC(=O)C(CC3CCOCC3)NC(=O)C=CCN3CCC3)C1C2 98253,c1(C(N2CC(C(C)NC(=O)CCCC(F)(F)F)C2)=O)ccc2nn[nH]c2c1O 98254,C(C)(C)(CC(=O)N(C)CC1OCCC1(C)C)N(C(c1cnc(CC)s1)=O)C 98255,c1(C(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)nnc2ccccc2c1N 98256,CN=c1[nH]cc(C(N2CCCC(N(C(=O)Cc3ccc(F)cc3)CCO)C2)=O)s1 98257,C1(CNC(CC2ON=C(CC)C2)=O)COCCN(C(=O)C(CCO)N(C)C)C1 98258,Cc1cc(C(F)(F)F)nc(N2CC(N3CCN(Cc4ncccc4C)CC3)C2)n1 98259,C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)C3(F)F)=O)C2)CC1 98260,N1(C(Cc2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCCN1CCOCC1 98261,c1(C(N(CC(CC)NC(CSCCC)=O)C)=O)cn2c(Br)cnc2s1 98262,c1(C(N2CC(CNC(CCCC=C)=O)C2)=O)ccnc(C(F)(F)F)c1N 98263,C1(NC(C2CC(C(C)C)C2)=O)CCC(O)CN(C(=O)Cc2ccc(Cl)cc2F)C1 98264,c1(SCC)ccc(C(=O)NC2CC(CNC(=O)COC3CC3)C(O)C2)cn1 98265,c1(C(=O)NCCN(C2CCN(CC)C2)C(=O)C(C)C2CC2)cccc2nsnc12 98266,Cc1cc(-c2cncc(F)c2COC)ccc1Nc1cnn(-c2ccccn2)c1 98267,N1(C(C(Cc2cccc(OC)c2)N)=O)CC(C)(C)CCC1CO 98268,C1(NC(CCN(C)CC)=O)CCN(C(C2(n3cnnn3)CCCCC2)=O)CC1OC 98269,Cc1sc(C(=O)Nc2ccc(-n3ccnc3)cc2)c(C)c1Br 98270,c1(C2N3CCCC(C3)N(CC)C2=O)ccc(F)cc1C.C=CCNC(C)=O 98271,C(C(C(=O)N1CCC(CN(C)C)C1)n1cc(-c2csnn2)nn1)OCC 98272,N1(C(C=Cc2c(C)ncs2)=O)CCCN(C(c2ccc(F)c(N)c2)=O)CCC1 98273,C(=O)(CC(F)(F)C(=O)OC)NCC(CC)NC(=O)CSc1cccc(OC)c1 98274,C1(C)(CC)CC(C(=O)NCCCNC(C2CSCC2c2ccccc2)=O)C1 98275,C1(NC(=O)C(O)C2CC2)CCC2CN(C(c3cc4c(nn3)CCC4)=O)CC2C1 98276,C12CCCN(C1)C(=O)CCC(=O)N2C(C)=O.C1(SC)CCC=C1Br 98277,Cc1c(C(=O)N(C2CC2)Cc2cscc2N2CCOCC2)cc(F)cc1Br 98278,N1(C(CN2CCCC(CC)C2)=O)CCC(F)(CNC(=O)Cc2cnn(C)c2)CC1 98279,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98280,CCC(CC)(CC)C(=O)NCC(C)NC(=O)CCN1C(=O)NC(C)(C)C1=O 98281,c1(-c2onc(C(C)SCC)n2)cc(NC(=O)OC(C)(C)C)cc(C)c1 98282,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsn2)C1 98283,C(C(C)CC(C)C)NC(c1ccn(C)c1)CC 98284,N1(c2cc(NCc3c(C)nccn3)ncn2)CCC(C)C2(CCC2)C1 98285,C1(C)(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CCNc2ncccn2)CCO1 98286,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CCC3C1)=O)CC2 98287,C1(C)(NC(Cc2c(CC)noc2CC)=O)CCCN(C(c2cnn(C)n2)=O)C1 98288,c1(CC)cc(C(=O)NCC(C2CC2)NC2(CC3CCCO3)CCCC2)cnc1C 98289,C12N(CCC1(C)C)C(=O)C2.c1(CNC(c2cc(OC)nn2C)=O)cc(C)nc(C)c1 98290,N1(C(c2cnc(S)nc2)=O)CC(F)CC1C(=O)Nc1nc(=O)o[nH]1 98291,c1(N(C)C)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O 98292,CCCCCC(O)CC(=O)NC(CNC(=O)CC(C)C)C1CC1c1ccccc1 98293,c1(C(=O)NC2CN(C(c3c(C#C)c[nH]n3)=O)C2)coc2cc(F)ccc12 98294,C12(CNCC(C)S(C)=O)COCC(CO)(C1)C2 98295,C(=O)(C(C(C)C)c1cc(C)on1)N1CCC(N(C(C(C)NC(CC)=O)=O)CC)C1 98296,c1(CNC(C(CC)n2ccnc2)=O)cnn2c1CN(c1nnc(C3CC3)o1)CC2 98297,Cc1ccc(C(CNC(=O)C(C)(C)CO)NC(c2cc(C(C)C)n(C)n2)=O)cc1 98298,C1(NC(CCC#CC)=O)CN(C(C2CSCCS2)=O)CC1(C)C 98299,N1(C(C)=O)CCCC(CN2CCCC2c2cc(Br)cs2)C1 98300,S(=O)(=O)(c1c(C)noc1C)NCC(=O)NC1CN(C(CCCC=C)=O)C1 98301,c1(C(N2CC(C)N(C(c3nc(=O)n(C)[nH]3)=O)CC2)=O)cc2c(Cl)cccc2[nH]1 98302,c1(C(C)C)nc(N2CC(OC(C)C)C(F)C2)cc(N2CCC(C(C)O)CC2)n1 98303,N1(C(=O)C2=CCCCC2)CC2OCCN(C(C3CC3C3CC3)=O)C2C1 98304,N1(C(C2C(CCC)C2)=O)CC(N=[N+]=[N-])CC1C(N1CC(N=[N+]=[N-])C1)=O 98305,C(=O)(CC1OCCc2sccc21)N1CC(CC(C)NC(=O)Cc2ccoc2)C1 98306,CC(C)(C)C(O)C(=O)N1CCC(NC(=O)Cc2ccc(O)nn2)C1(C)C 98307,N1(C(C(=O)NC(C(=O)NCC(=C)C)C2CC2)C)CCOCC1 98308,C1(NC(C(C2CCCC2)N(C(=O)COCc2nc[nH]n2)C)=O)(CN)CCCOC1 98309,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2(CC(NC(=O)CC3CCC4CC34)CO2)C1 98310,C(=O)(CCCCNC(C)=O)NCC1(C(C)(C)O)CN(C(c2ccc(CC)o2)=O)C1 98311,c1(NC(C(=O)NC(C)CC2CCOCC2)=O)cccc(S(F)(F)(F)(F)F)c1 98312,CCCC(CCC)=CC(=O)NCC(C1CCOC1)NC(=O)C#CC1CC1 98313,CCS(=O)CC(=O)NC1CN(C(=O)CC2CCN(C(C)C)CC2)CC1O 98314,C1(NC(C(CCSC)NC(N)=O)=O)C2CCC1N(C(c1ccsn1)=O)C2 98315,c1(C(CN(C(=O)Cc2nc[nH]n2)CC)NC(C2CCN(CC)C2)=O)cccc(Cl)c1 98316,N1(C(C(C)CCO)=O)CCN(C(=O)C=Cc2nccs2)CC1C1CCC1 98317,C1(NC(c2c(CC)nns2)=O)CCC12CCCN(C(=O)CC1COCCN1C)C2 98318,c1(C(C(=O)Nc2cn(CCOC)nc2)OC)ccc(C)cc1 98319,C1(C(N2CC(OCC(NOCC=C)=O)C2)=O)CC(=O)N(OC)C1 98320,N1(C(C(C)OC(C)(C)C)=O)CC2CC(NC(c3coc(C(F)F)c3)=O)C1C2 98321,c1(N2CCC(C(F)F)C2)[nH]c(=NCc2cn(C3CC3)nn2)nc2sccc12 98322,C1(NC(=O)C=CCn2cncn2)CN(C(C2CCCCS2)=O)CC2(CC2)C1 98323,C1(C)(CNC(C(F)(F)C2(OC)CCC2)=O)CNC(=O)C1.C12CCCN1C2=O 98324,C(=O)(CCC(=O)c1cnccn1)NC(C(C)C)CNC(C1CC(CC2CC2)C1)=O 98325,C(=O)(C(C)(C)CC#N)NCCCN(C(C1CN(CCC)C(=O)C1)=O)CCSCC 98326,c1(C(N(CCNC(=O)CN(C)C(N)=O)CC)=O)cc(OC)ncc1F 98327,C1(F)(CNC(CN(C2CCCCC2)C)=O)COCCN(C(=O)C(O)CN(C)C)C1 98328,C(=O)(CC(C)c1cccnc1)NCC1(NC(C(C)C)=O)CCC1 98329,c1(N2CCC(c3onc(C)n3)C2)nc(=O)c(Br)c(C)[nH]1 98330,C1(CNC(c2cc(C)n(C)n2)=O)(CO)CCCN(C(C2CCN(C)C(C)C2)=O)C1 98331,N1(CC(=O)NCC2OCCN(CC)C2)CCCN(C(C2(CO)CC2(C)C)=O)CC1 98332,C1(NC(=O)Cn2nccn2)COC2(CCN(C(C34COC(CF)(C3)C4)=O)C2)C1 98333,N1(C(=O)Nc2c(C)cccc2)CC2CC1CN2c1cncc(Cl)n1 98334,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(c2scc(C)c2)=O)C(C)C1 98335,c1(C2CC2)ccc(NC(C2CC(CC(N3CCC(CC)(OC)C3)=O)C2)=O)c(OC)c1 98336,N1(C(C(CC)CO)=O)CCCC(C)(NC(=O)Cc2sc(-c3nc[nH]n3)nc2C)C1 98337,c1(CC)cnn2ccc(C(=O)NCCCC3(O)CCC3)nc12 98338,c1(CC(=O)N(C2CN(C(=O)C=CCO)C2)C)cccc2ccccc12 98339,N12CCCC(C1)c1cccn1C(=O)C2=O.c1(NCCC(=O)NCC#C)ccc(Cl)cc1 98340,C1(C(N2C(C)CC2)=O)CCCC(NC(=O)COCC2CC2)C1 98341,C1(C2(O)CCC2)(CNC(CC2(C)N(C(C=Cc3ccc(C)o3)=O)CC2)=O)CC1 98342,CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOc2cc(CN)ccc21 98343,N1(C(CCCCOC)=O)CC2CC(NC(=O)Cc3ccnc(F)c3F)C2C1 98344,CCCC(C(=O)NC(C(=O)NCCCOCC)C1CC1)NC(=O)CC 98345,C(=O)(C(O)CC(F)(F)F)N1CCC(N(C(=O)COCCOC)CC#C)CC1 98346,c1(OC)ccc(C(=O)C(=O)NC(C)CNC(c2cc(F)cs2)=O)cc1C(F)(F)F 98347,Cc1nnc(Br)cc1C(N1CCCC(O)(CNC(C2CCC23CCC3)=O)C1)=O 98348,c1(C(N2CC(CNC(C3C(C(N)=O)C3)=O)C(O)C2)=O)cn2c(n1)CCC2 98349,N1(C(CC#C)=O)CCC2(CCCN(Cc3cc([N+](=O)[O-])ccc3C)C2)CC1 98350,S(=O)(=O)(c1ccccc1)NCC(=O)NCC1CC(NC(=O)CCc2cccs2)C1 98351,C(CCCCC(=O)NC(Cc1cn[nH]c1)C(N1CC2COCC2C1)=O)SC 98352,C=CCCCCCC(=O)NCCNC(C1CNC(=O)N1C)=O 98353,CC1CCCC(C)N1CC(=O)NC1CN(C(=O)CCc2ccn(C)c2)C1 98354,C1(C(N2CC(N(C(c3c(C)cc(F)s3)=O)C)C2)=O)CC2(CCC2)CCO1 98355,C1(C(=O)NCC2COCCN(C(C(C)C#N)=O)C2)C2CC3CC(C2)CC1C3 98356,c1(SCC(=O)NCCNC(c2ccc(CF)cc2)=O)ccccc1Br 98357,C1(C(=O)NCC2(CCNC(C(CN(C)C)N(C)C)=O)CC2)CC(=O)N(O)C1 98358,C=CC(C)(C)CC(=O)N1CC(C(=O)NCC2(CC)CCCCCC2)C(F)C1 98359,C=CC(CCC)CC(=O)NC1CN(C(=O)Cn2nc(C)c(C)c2C)CC(F)(F)C1 98360,C(=O)(C(O)C1=CCCCC1)N1CC(COC)(CNC(C2CCN(C(C)=O)C2)=O)C1 98361,C(CC1=CCN(C(c2nnc(O)nc2O)=O)CC1)NC(C(C)=CC)=O 98362,C1(C(N(CCC(C)NC(C2N(CC)CCCC2)=O)C)=O)CCC2(CCCC2)CC1 98363,N1(C(COCCCCC)=O)CC(NC(c2cc(C(N)=O)[nH]n2)=O)N2CCC1C2 98364,c1(CC)cc(C(=O)NCCC2CCN(C(=O)CCC3(C)CC3)C2)c(C)o1 98365,c1(C(=O)NCCCNC(C(C(C)(C)C)c2ccncc2)=O)ccc(F)c(Cl)c1N 98366,n1(CC)ccnc1C=CC(=O)NCCCN(CCCNC(C1CC1CSC)=O)C 98367,c1(NC(C2N(C(CSC)=O)CC(C)(C)C2)=O)cc(Br)cc([N+](=O)[O-])c1C 98368,c1(OC)ccc(CC(N2CCCC2CNC(=O)C(C2CCC2)C2CC2)=O)cc1F 98369,c1(C(N2CC3CC(NC(C4(COC)CCOC4)=O)C3C2)=O)ccc2ncnn2c1 98370,N1(C(C2CCC(n3cc(-c4cn(C)nc4)nn3)C2)=O)CCC2CCCC2CC1 98371,c1(-c2nnn(CCC(=O)NOCC(=O)NCN3CC4CC4C3)n2)ccccc1F 98372,C(=O)(C(CC(C)C)N(C)C)NCC(CCCC)NC(C1CC(CF)C1)=O 98373,C(=O)(C(C)(C)CCCF)NCC1(F)CCC(CNC(COC(C)C)=O)C1 98374,C(=O)(C1CC(=O)Nc2ncccc21)N(C(C)C)CCNC(=O)C1CCc2nccn21 98375,C(CC(C(C)C)NC(=O)Cc1cncc(O)c1)NC(C(n1cc(C)nc1)(C)C)=O 98376,C(=O)(CCC(C)(C)F)NC(C)C(c1ccccc1)NC(=O)C1=CSCS1 98377,C1(NC(CC)=O)CN(C)CCN1C(=O)NCc1ccn(C2CC2(F)F)n1 98378,C1(C#N)(OC)CC(C(N2CC(F)(CNC(=O)C=CC3CCCN3C)C2)=O)C1 98379,c1(C(=O)NC2CC(NC(c3csc(-c4ccco4)n3)=O)C2)c(F)c(F)ccc1Cl 98380,c12ccccc1S(=O)(=O)C(CC)=CC=C1C=NN(CCC(C)(C)CNC2=O)C1=O 98381,C1(c2nnnn2CCOCC)(NCCc2cc(CC)no2)CCCS(=O)(=O)C1 98382,CC1(OCCC(=O)NC2COCC2CNC(C2CN(C3COC3)C2)=O)CCCC1 98383,CC1CC(=O)NCC1C(=O)NCC1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O 98384,c1(NC(C(C(C)C2CC2)NC(C)(C)C(F)F)=O)ccc2c(c1)CCC2.CC=C 98385,N1(C(C2CCC(=O)C2)=O)CCC2CC2(C(=O)Nc2cncnc2O)CC1 98386,c1(C(=O)NCC2CN(C(c3cncc(CC)c3)=O)CC2O)c(F)ccc(C)c1N 98387,c1(C(C(=O)NCC(CNC(CC(C)NS(C)(=O)=O)=O)CO)(C)C)ccc(Cl)nc1 98388,C1(NC(c2ccccc2-c2ccncc2)=O)C2CC(O)C1N(C(C1CC1F)=O)C2 98389,c1(C(=O)NCC(CNC(C(C)C(C)O)=O)(C)C)cnc(N)c(O)c1 98390,C1(C(N(CCSCC(=O)N(CCCCC=C)C)C2CC2)=O)CCCC12CCC2 98391,C(=O)(C(C)(C1CCC1)NC(c1cocn1)=O)NC(c1cnn[nH]1)C 98392,N1(C(C(OC)OCC2CC2)=O)CC2COCC2(C(N2CC(c3cccnc3)C2)=O)C1 98393,C1(CNC(C(C)Cc2cnn(C)c2)=O)CCCN(C(c2n[nH]cc2Br)=O)C1 98394,C12(C(N3C(CCC(=O)N(C)CC4CCCN(C)C4)CCC3)=O)CCC(C1)C2(C)C 98395,C1(CC(=O)NC2CC(NC(c3ccc(C(=O)OC)o3)=O)C2)C(=O)NN=C1C 98396,c1(C(=O)NC(C(C)NC(c2ccc(C)nc2)=O)C(C)C)n[nH]c2c1CCOC2 98397,Cc1cnccc1C=CC(=O)NC1CCCC(NC(c2c(C)nn(C)c2Cl)=O)C1 98398,Cc1oc(Br)cc1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCNC1=O 98399,N1(C(c2ccc(CC)cn2)=O)CC(CC(=O)NC2(C(C)O)CCC2)CC1(C)C 98400,CC1C(CN(C(=O)CCC2OCCO2)C(=O)CSC2CCCC2)CCCN1C 98401,C(c1c(Cl)nc2sccn12)=CC(=O)NC1C2CCN(C(=O)C(O)CC(F)(F)F)C12 98402,C(C)(CN=C(NCc1ccccc1)N1CCCC(C(C)C)C1)OCC 98403,c1(OC)cccc2c(N3CCC(NC(c4ccc(Cl)cc4)=O)C(C)C3)ncnc12 98404,C1(CCC)CCC(C(=O)NCCCCNC(c2nscc2N)=O)CC1 98405,C(CNC(=O)C(n1cc(C)cn1)C)(CC(=O)N1CCCC1CCCO)OC 98406,c1(CNC(c2n(CCSC)nnn2)c2cscc2C)ccncc1Cl 98407,CC1CCN(C(C2(CO)COC2)=O)CC1NC(=O)CC(F)(F)Br 98408,c1(OC)ccc(C)c(C(=O)NC2CCN(C(=O)CCC(C)N(C)C)C2)c1 98409,c1(NC(CCCCNC(c2cc(CC)sn2)=O)=O)ccc(F)cc1OC(C)C 98410,C1(CCC(=O)NC(C2CCC2)CSC(C)C(=O)NC(C)C)(N(C)C)CCCCC1 98411,c12ccc(cn1)CC(=O)N1CC(F)(C1)CNC2=O.N1(CC)CCCC1CC 98412,c1(CC)ccc(C=CC(=O)NC2COCCN(C(=O)CC3CC(F)C3)C2)cc1 98413,c1(CC(=O)NCC2N(C(C(C)SC)=O)CCCCC2)coc2ccc(F)cc12 98414,CN1CCN(C(c2cc(Cl)ccc2Cl)=O)C(CNC(c2cnc[nH]c2=N)=O)C1 98415,C1(N(C(CCC)=O)C)CCN(C(c2cc(Cl)ncc2OC(F)F)=O)CC1C 98416,CC1(C)CC(CC(=O)NC2(C3CCCN3C(C3CC=CCO3)=O)CC2)CCO1 98417,C1(C(=O)NC(C)CCNC(=O)C(=O)Cc2ccccc2)CC(C)(C)CCO1 98418,CC(C)(O)C(C(=O)NC1CCCC1O)NC(c1cnn(C2CC2)c1)=O 98419,C(C(C)CC(=O)NCC1(COC)CN(C(=O)Cn2cnnc2)C1)OC 98420,N1(C(CCC(=C)Cl)=O)CC(C(N2CCC(OC)CC2)=O)CC12CCC2 98421,C(C(C(C)C(C)C)NC(=O)CCc1cnccn1)NC(CSCCC(C)C)=O 98422,N1(C(C(C)OCC(C)C)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCCCC2 98423,C1(OC)(CNC(C2CC3CC3C2)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1 98424,C(=O)(CCCNC(=O)CC1CCCN1CC)NC1CC(SC)C1.C(C)=O 98425,c1(COC)ccc(C(=O)NC23CC(NC(=O)CC(=O)Nc4nccs4)(C2)C3)o1 98426,N1(C(C2CCC3CC23)=O)CCOC2(CCCN(C(c3ocnc3C(F)F)=O)C2)C1 98427,c1(C(=O)NCC23C(CN(C(CCC(C)OC)=O)C2)C3)ncc(Cl)cc1F 98428,C12(C(=O)OC)CCCC1(C(=O)NCCCCNC(C1CCCSC1)=O)C2 98429,Cc1n[nH]c(C)c1CNc1ccnc(N(C)CC2CCOC2)n1 98430,C(=O)(CC(O)CC(C)(C)C)NC(C(=O)NCC(C(C)C)O)Cc1ccco1 98431,c1(C(N(C(C)C)CCNC(C2CCCCO2)=O)=O)c(Cl)c([N+](=O)[O-])nn1C 98432,C12(CNC(COCC)=O)CCC(C(N3CCCCC(C(N)=O)CC3)=O)(CC1)CC2 98433,N1(C(c2nn(CC)c(C)c2)=O)CCC(N(C)C(c2cc(OC)nn2C)=O)C(C)C1 98434,N1(C(Cc2cccc(SC)c2)=O)CCN(CCO)CC1C.C12(CC1)NC2 98435,C1(C(=O)OCC(C2CCCC2)C)CSC(c2ccccc2O)=N1 98436,N1(C(CNS(N(C)C)(=O)=O)=O)CCC2(CCCC2NC(=O)CC(C)(F)F)CC1 98437,Cc1ccc2c(C(=O)NCC3(F)CC(CNC(c4ocnc4C)=O)C3)cnn2c1C 98438,c1(C(=O)NC(C)CN(C(=O)CC(C)CN(C)C)C)ccc2oc(N(C)C)nc2c1 98439,c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)CO)c[nH]c(=O)c2ccncc12 98440,c1(N2CCC(c3ccc(N(C)CCn4ccnc4)cc3)CC2)ccnc(S(C)(=O)=O)n1 98441,C1(N(C)C(c2cc(F)cs2)=O)CN(C(=O)CNC(=O)NC2CCCC2)CC1F 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98670,C=CC1(CC(N2CC(N(C(=O)CCC(N)=O)C)C(F)C2)=O)CCCCC1 98671,N1(C(COC)=O)CCN(CC(=O)NC2c3c(-c4ccccc4)noc32)CC1.OC.SC 98672,C=CCC(C(=O)NC1CC(NC(=O)C(C2CCC2)OCC)C1)OC 98673,C1(NC(=O)CC2CC=CCC2)CCN(C(=O)COc2ccc(O)nc2)CC1O 98674,C1(C)(C(N(C)CC2N(C(CC(C)SC)=O)CCCC2)=O)CCC(=O)CC1 98675,C1(NCCCS(CC)(=O)=O)CCCC(CNC(=O)OC(C)(C)C)CC1 98676,CCC(CC(=O)N1CCN(C(c2cccc(C)c2C)=O)CC1C(C)C)C(F)F 98677,Cc1nnc(C(c2ccccc2)NC(c2nnnn2C2CCC2)C2CCC2)n1C1CC1 98678,N1(C(C2(N(C)C)CC2)=O)C(CNC(c2ccc(F)cc2Cl)=O)CC2COCC12 98679,C(CNC(C1CNC(=O)N1C)=O)(CC(C)C)NC(C(C)SCC)=O 98680,N1(C(C(=O)NC(C)=O)=O)CCC2(C1)CO2.C(CCSCC)NC(C)=O.C(C)(C)C 98681,C(=O)(C1=NOC(CNC(c2c[nH]c(=N)o2)=O)C1)N(C)CC1COC(=O)N1 98682,C1(F)(C(N2CCCC(N(C(c3cnn(CC)c3C)=O)CC)C2)=O)CCCN(C)C1 98683,CN1CC2CCCC(C1)N2C(=O)C(CC(N)=O)NC(C1CCCN(C2CC2)C1)=O 98684,c1(CC(N2CCC(Cn3ccnn3)C2)=O)cn(C2CCOCC2)nn1 98685,C1(NC(c2[nH]cc(CC)c2)=O)CC2CCCC(C1)N2C(C1OC2CCC1CC2)=O 98686,O=C(C(O)C(F)F)NCCC1CC(NC(=O)CCc2ccccc2F)C1 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98704,N1(C(C(C)n2cccn2)=O)CC2CN(Cc3c[nH]nc3-c3ccccc3)C2C1 98705,C1(CC)CN(C(c2sccc2OC)=O)CCC1C(F)(F)F.C(=O)(CCCSC)NC 98706,c1(N2CCN(CC(CC)Oc3cccc(C)c3)CC2)cccc(F)c1F.C1(=O)CN1 98707,C1(N(C(Cn2nc(C)oc2=O)=O)C)CC(=O)N(c2cnn(C)c2)C1C 98708,c1(N2C(CNC(CCCC#N)=O)CCCC2)nc(C(F)F)nc2nc(Cl)ccc12 98709,N1(C(C2(NC(C)=O)CCOC2)=O)C2CCC1CN(C(c1cc(COC)c[nH]1)=O)C2 98710,C1(N(C(c2sccc2CSC)=O)CC)CCCN(C(=O)C=C(C2CC2)C2CC2)C1 98711,C1(C(=O)OCC)CN(C(=O)NCC2CS(=O)(=O)C2)C1(C)C 98712,Cc1csc2ccc(CC(C(=O)C(=O)N)=O)cc12.C1(CN)CC2CC(C(N)=O)CC12 98713,c1(-c2ccc(C3(CC(=O)Nc4ccns4)CCC3)cc2)c(F)cccc1[N+](=O)[O-] 98714,CC1CCN(C(C2CC(F)(CO)C2)=O)CC1NC(c1cc(C2CC2)[nH]n1)=O 98715,c1(C(=O)NC(CC(C)C)CNC(C2(C)CCCS2)=O)ccc2ncncc2c1 98716,CCC(CC(C)C)C(=O)NCCCN(C(=O)COCC1CCC1)CCO 98717,C1(CC(=O)N(C2CCN(C(=O)C3=CCSC3)CC2)CC)(CC)CCOCC1 98718,CC(C)CC(C(=O)N(CCCCCC(=O)NC1CCCSC1)C)C(N)=O 98719,N1(C(c2cc(OC)no2)=O)CCC(C(N2CCC(C)(OC)C2)=O)(CO)C1 98720,C(=O)(C(N)CC(F)F)NC1C(c2cccc(-c3nccc(C)c3)c2)C1 98721,C1(=O)CC(C)SCCNC(=O)C(C)N1CCC.C(CCO)NC(N)=O 98722,O=C(C1=CCN(C(c2csc(Cl)c2)=O)C1)Nc1cnn(C(F)F)c1 98723,C(=O)(CC(F)(F)C(C)C)NC(C)CNC(=O)C(C)OCCN(C)C 98724,C12(C(N3C(C)CC(NC(C4CCC=CCC4)=O)C3)=O)CCOC1CC(=O)NC2 98725,CC1(NC(=O)CNC(=O)Cc2cccc(N)c2)CCN(C(=O)C(F)C2CCC2)C1 98726,C1(C(N2CCN(C(c3snc(O)c3Cl)=O)C(CO)C2)=O)CCCC2CCCN12 98727,c1(C(N2CC(NC(=O)CC3CC4(CCC4)C3)CC(C)C2)=O)cccc([N+](=O)[O-])c1 98728,N1(C(C2CC(C)OCC2)=O)CC2CC(NC(C3(N(C)C)CCC3)=O)CC1C2 98729,Cc1oc(C(F)(F)F)c(C#N)c1CNC(=O)NC1(CS(C)(=O)=O)CCC1 98730,c1(CN(C=O)CC)ccccc1CNC(=O)C(C)OCCC1C(C)C1C 98731,C=C(C)CC(C)C(=O)NC1(COC)CCN(C(=O)Cc2nncn2C)CC1 98732,Cn1cnc2c1CC(C(=O)NCc1nc(O)c3ccccc3n1)CC2 98733,C12CN(CCO1)c1nc(ns1)C2.C=C(Br)CC(=O)N(CCCCC)CCOC 98734,C1(CC(=O)NCC(C(C)C)NC(c2ccc(Br)s2)=O)CCC(C)(C)O1 98735,c1(NCC2(CSC)CC2)[nH]c(=NC(C)c2n[nH]c(CO)n2)nc2c1cnn2C 98736,Cc1ccnn1CC(=O)NC(CNC(c1cccs1)=O)C1CCC1 98737,N1(C(CN(C2CC2)CC)=O)CC(C)CCC1C(=O)NCC1(C)CCC(=O)N1 98738,CCC(C)(C)CCCC(=O)NCC(C)(C)CN(C(=O)C(C)(F)C(F)(F)F)C 98739,C(c1ccc(F)cc1)=C(C)C(=O)NC1CCCCN(C(=O)C(C)(C)C2CCC2)C1 98740,C(=O)(C(C)(O)C(C)C)NCC1CC(COC)CN1C(C1CCCCCC1)=O 98741,C1(CS(=O)(=O)N(c2ccc(C(CC)C3CC3)cc2)C)CC2COCC2O1 98742,C1(C(=O)NC(CCOCC)C(=O)NCC(C2CC(C)(C)C2)O)CCC(C)(C)CC1 98743,CCCCCCn1cc(C2CCN(C(=O)Cc3nocc3C)C2)nn1 98744,C1(CC(=O)NCC(CNC(CCC(=C)Br)=O)OC)CCCCC12CC2 98745,C1(N(CC(=O)N(CC(=O)NC(C2CCOC2)C#C)CC(N)=O)C)CCCCCC1 98746,c1(SC)nc(Cl)c(C)c(=NC2CCN(C(=O)CN3CCCNC3=O)C2)[nH]1 98747,c1(C(=O)NC(CNC(C(CC)CO)=O)(C)C)cc(Br)cc2c1OCC2 98748,CC(CCc1ccc(Br)cc1)CC(=O)NCC1CCN1C(c1ccco1)=O 98749,c1(C(=O)NCC(C)=CC(=O)N(CCCC(C)(F)F)C)cc(C)c(C)cn1 98750,c1(C(N2CC(C)C(C(=O)NC(C3CCOC3)CO)C2)=O)cccc(F)c1O 98751,C=C(C)C(C)(C)C(=O)NC1CC(C)(C(=O)N(C)Cc2cnco2)C1 98752,c1(CC(=O)NC2(C)CCN(C(C(CC)C(C)O)=O)CC2)c[nH]c2cccc(F)c12 98753,N1(C(C(=O)NC(CC)(C)C)CCCCC2CC2)CCC2NC(=O)CCC2C1 98754,N1(C(CC(C)(F)F)=O)CCc2ccccc2C1CNC(C1CCCOC1)=O 98755,C1(C(=O)NCC(CCOC)NC(c2c[nH]c(C(F)(F)F)c2)=O)C(C)(C)C1(F)F 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98844,c1(C(=O)NC(CCNC(C2(NC(C)=O)CC2)=O)C)cc(C)cc(C)c1N 98845,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CN(C(=O)Cc1cc2ccccc2o1)C)O 98846,n1(C(C)C)ncc(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2(F)F)=O)c1C(F)F 98847,c1(C(N2CC(CNC(c3c(CC)c(C)sc3)=O)C(C)C2)=O)ccc2c(c1)CCO2 98848,N1(C(C2CCCC(NC)C2)=O)CCC(C(=O)N(C)Cc2ccccc2O)CC1C 98849,N1(C(C2(CC)CC(C)(C)C2)=O)CC=C(C(=O)NCCC2CC3C=CC2C3)CC1 98850,C1(NC(CCNC(=O)NC)=O)CCC(CNC(=O)C(c2cncn2C)O)C1 98851,C(=O)(C(C(C)CCC=C(C)C)N(c1ccc(COC)cc1)C)NCC.C(C)(=O)O 98852,c1(CC)cc(CC(N2CC(NC(=O)COC3(C)CCCC3)C(C)C2)=O)cc(Cl)n1 98853,C#Cc1cccc(CC(N2CC(C(=O)Nc3cnc(CC)nc3C)(CC)C2)=O)c1 98854,c1(C(N2C(CCNC(CC(COC)C)=O)CCC2)=O)cc2occc2[nH]1 98855,CCS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CCCN(C(N)=O)C1)=O 98856,C1(NC(c2n[nH]c(CC)c2Cl)=O)COCCN(C(=O)CN(C)CCO)C1 98857,c1(C(=O)NCC2CCN(C(=O)C(F)(F)c3ccco3)C2)ccnc(Br)c1F 98858,c1(C(=O)NCCCCCNC(Cn2nc(C)n(C)c2=O)=O)ccc2cc[nH]c2c1 98859,Cc1c(CC(=O)NC(C)CN2CCN(C(=O)Cn3cnnn3)CC2)cnn1C 98860,c1(C(=O)NC2CC(CC(=O)NCC(COC(C)C)O)C2)c[nH]nc1C(F)(F)F 98861,C1(NC(C(N2CCCCC2)C)=O)CCCC(NC(=O)C(=O)NCC2CC2)C1 98862,c1(CC)ccc([N+](=O)[O-])cc1C(=O)N(CC(C)(C)NC(c1ccncc1F)=O)C 98863,C1(C(=O)NC(CN(C(Cc2onc(CCC)n2)=O)C)(C)C)CCN(C)C1C 98864,C1(NC(C#C)=O)CCCCCC1C(=O)N(C1CCCCC1)C 98865,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(C)Cc2ccncc2)C)n[nH]1 98866,C#CC1(C(N2CCCC(CCNC(C3COCCN3C)=O)C2)=O)CCCC1 98867,CCC1=C(C(=O)NC(C)CCCNC(=O)CC(C)c2cnn(C)c2)CCCO1 98868,CN1CCCC(O)(CC(=O)NCC(=C2CN(C(c3cc(C4CC4)ns3)=O)C2)F)C1 98869,Cc1cc(N2CC3CN(C(C4CC5CC4C4CC54)=O)CC3C2)n2nc(C)nc2n1 98870,N#CCC(=O)NNC(=O)CC1CC1Cc1ccc(Cl)cc1 98871,c1(C(=O)NC2CN(C(C3(C(N)=O)CC3)=O)C2)ccccc1.c1(C)nc[nH]n1 98872,C1(NC(C(C=C=C)C)=O)CCC2CCN(C(=O)COC3(C)CCCC3COC)C1C2 98873,C1(C)(CC)CCC(NC(=O)C(CC2CC2)NC(C2CC2[N+](=O)[O-])=O)CC1 98874,c1(C(=O)NC2C(CNC(COC(CC)(C)C)=O)C2)sc(CC2CC2)nc1C 98875,C1(C(=O)NCCC2(OC)CCC2)CC12CCN(C(c1cccc(F)c1O)=O)C2 98876,Nc1cccc(CC(=O)OC2CCN(CCOCc3ccccc3)C2)n1 98877,C(=O)(C1Cc2ccccc21)N1CCC(F)(CNC(C(C)CO)=O)CC1 98878,c1(NC)ccc(C(=O)NCC(C)(O)CNC(C2CCCCC2O)=O)cc1 98879,c1(C(=O)NCC(CCCC)NC(C2CC2(C)C)=O)cnc2c(F)ccc(F)c2c1 98880,CC(C)(C)CC(=O)N1CC(C(N2CCC(n3ccnc3)CC2)=O)C(F)C1 98881,N1(C(c2ccc(C(=O)OC)cc2)=O)CC(NC(c2conc2C)=O)C2(CC2)C1 98882,N1(C(c2cocn2)=O)CCN(Cc2nc(-c3cccc(Cl)c3)no2)C2CC12 98883,N12CCCCC1C2=O.CC(C)(C)C(=O)NCC1CCN1CC(c1cc(F)cs1)=O 98884,c1(SC)cc(F)ccc1C(=O)NCCC1CN(C(=O)CN2CCCC2C)C1 98885,C1(C(=O)NC(CC=CC(=O)NCCCN(C)C)(C)C)CCC(C2CC2)C1 98886,C(CN=c1nc(O)c(Cl)c[nH]1)SCc1ccc(Cl)c(F)c1 98887,N1(C(C2N(C)CC(O)CC2)=O)CCC(C(N2CC3(CO)CC3(CO)C2)=O)CC1(C)C 98888,CC1COc2c(C(=O)N(C3CCCN(C(=O)Cn4cnnc4O)C3)C)cccc21 98889,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 98890,C1(C(C)C)CC(=O)N1.c1(CCOCC)nc(CNc2ccccc2)n(C)n1 98891,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(c3ccc(OC)nn3)=O)C(C1)CO2 98892,C1(CNC(C=CCC)=O)CCCC(CNC(=O)C(C)(c2ccccc2)N(C)C)C1 98893,c1(C(N2CCN(CCC(=O)NC(C)C)CC2)C(=O)OC)cc(OC)c(OC)cc1O.CN 98894,N(C(=NCCc1cccs1)NCCCN1CCCC1)Cc1c(CC)nn(C)c1 98895,c1(C(N2CC3CN(Cc4ccc(Cl)nc4)C3C2)=O)ccnc2ccc(O)cc12 98896,CCC(CC(F)F)C(=O)N1CCCC1Cc1ccc(F)cc1.C12CCN(C1)C2=O 98897,CS(=O)(=O)CC(F)(F)CCNC(=O)Nc1nn[nH]c1C(F)(F)F 98898,N1(C(C(CC#C)C2CC2)=O)CCC(C)(C)C1CNC(C1CCN(C2CC2)CC1)=O 98899,c1(C(=O)NC(CC)(C)CNC(=O)C(CC)CCOC)cc(F)c2nc(C)cn2c1 98900,N1(C(c2c(C)cnnc2)=O)CC(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCC1C 98901,c1(COC)nn(C)cc1C(=O)NC12CC(NC(c3cc(C)n(C)c3)=O)(C1)C2 98902,N1(S(C)(=O)=O)CCCC1C(=O)NCC1(NC(=O)CC2CCC2)CCOC1 98903,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)NC(=O)CCc1ccoc1)C 98904,CC(C)(CCCCNC(c1csc2cncn12)=O)NC(=O)CCN1CCCCC1 98905,CC(C)C(C)C(CNC(=O)CCCc1ccncc1)NC(C1CC2(F)CC1C2)=O 98906,S(=O)(=O)(c1ccc(Br)c(OC(F)F)c1)N1C(C)CC(C)CC1C 98907,c1(C(=O)NCCC2(CNC(C(CCOC)C)=O)CC2)cc(C)c(F)cc1F 98908,N1(C(C(CCC#C)O)=O)CCCN(C(c2cnoc2C)=O)C(C(C)C)C1 98909,CC(C)(O)C(F)CNC(C1(C2CCCN2C(=O)CC2CCCO2)CC1)=O 98910,CC1CC(C(=O)NCC2(F)CC(NC(=O)C(=O)NCCNC(N)=O)C2)CC(C)C1 98911,CC1C(NC(c2coc(N(C)C)n2)=O)C(C)CCN1C(c1cnccc1Br)=O 98912,c1(OCC)ccc2c(c1)C(NC(=O)NCC1CC(CCS(C)(=O)=O)C1)CCO2 98913,N1(CCNC(c2ccc(CNC(C3(CCCC)CCC3)=O)o2)=O)CCCC(C)C1 98914,c1(C(=O)NCC2CCCN2C(c2cnn(C3CCOC3)n2)=O)cnn2c1CCC2 98915,c1(C(=O)NC2C(NC(C3CC(C)N(C)CC3)=O)COC2)ccc(Cl)c([N+](=O)[O-])c1 98916,C1(C(=O)NCc2cc(C)oc2)CCCCN(C(C2CC(N(C)C)C2)=O)C1 98917,CCC(C)(O)C(=O)NCCCN(C(=O)CCC1CC(C)(C)CO1)C1CCCC1 98918,CC(C)CCCC(C)C(=O)NC1CCN(CCCNC(c2c[nH]nc2[N+](=O)[O-])=O)C1 98919,N1(C(c2c(OCC)nc(C)cc2)=O)CCCC2(CCN(C(=O)C(C)C(F)F)C2)C1 98920,c1(C(C(=O)NC2CC2)N(C)Cc2n(CCC)ccn2)ccc(Cl)cc1F 98921,Cc1ncc(Br)c(N2CCOC(CNC(c3sc(F)cc3C)=O)C2)n1 98922,c1(-n2cc(C(C3CCCCC3)C)nn2)ccc(C(=O)Nc2cc(F)n(C)n2)c(F)c1 98923,Cc1csc(Cl)c1C(N1CCC1CNC(C1C(c2ccccc2)C1(F)F)=O)=O 98924,N1(C(C2(SC)CN(C(CC(CC)O)=O)C2)=O)CCOC(C)CC1 98925,c1(COC)cncc(C(=O)N(C(C)CN(C(=O)CCc2cncs2)C)C)c1 98926,c1(CC)cc(C(=O)NCC(C)(C2CC2)NC(c2cc(C)[nH]n2)=O)ccc1O 98927,CC1SCCCC1C(N1CCC2CC12CNC(=O)CNC(=O)C(F)(F)F)=O 98928,Cc1cn2ccc(C(N3CCC(Cc4cn(CCO)nn4)C3)=O)cc2n1 98929,N1(C(C(C)NC(CC)=O)=O)CCN(C(c2ccnc(Cl)c2O)=O)C(CCO)C1 98930,Cc1nc(Cl)ncc1NC(C1CCCN(C(C2CC(C)(C)C2)=O)CC1)=O 98931,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 98932,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccns2)=O)C1 98933,c1(C(=O)NCCC2CC(NC(C(C)O)=O)C2)sccc1C(C)(C)C 98934,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 98935,C(CC(C(C)C)(c1nnnn1CC1CCOC1)NCCc1ccc(Cl)s1)OC 98936,N1(C(CCOCC)=O)CC2(C1)CC(=O)NC2.C1(C(COC)OC)CCCO1 98937,C1(CCNC(c2cnn(C)c2Cl)=O)CCN(C(=O)Cc2cc[nH]c2)CCC1(F)F 98938,c1(C(=O)NCCCCNC(C(n2ncc(C)c2)C)=O)cnc(O)cc1C 98939,C1(C(=O)OC)CCC(F)(F)CN1N(C1CCNCCC1C)c1ccnc(OC)c1.C(C)=O 98940,C1(CNC(C(COC)OC)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 98941,S(=O)(=O)(c1c[nH]ccc1=NC(C(C)(C)C)C(F)(F)F)N1CCN(C)C2C1C2 98942,C(=O)(C1CCCn2c(C)cnc21)NCCCCC(C)NC(CN(C)CC)=O 98943,N1(C(C(C)n2ccnc2)=O)CC2CCC(C1)N(C(=O)CCc1cc(F)ccn1)C2 98944,N1(C(C(C)CF)=O)Cc2ccccc2CC1CNC(=O)C(c1ccccn1)O 98945,N1(C(C(CC)(CC)CC)=O)CCC2(CCC(NC(=O)Cc3cnns3)CC2)C1 98946,c1(C(=O)NCC2C(CNC(COC(C)C)=O)C2)cc(C2CC2)cnc1O 98947,C1(C(=O)NC2CC(NC(Cc3ncc(C)s3)=O)C23CCC3)CC2C=CCC(C1)C2 98948,O=C1NC(=O)C(CNC(C2CC23CC(NC(c2cocn2)=O)C3)=O)N1 98949,C1(CNC(c2c(CC)cccn2)=O)CCN(C(=O)C(C)(C)CO)CC1C 98950,CCC1=NOC(CC(=O)NC2(CNC(C3CCNC(=O)C3)=O)CCC2)C1 98951,C(CC(C)NC(=O)CNC(=O)OC1CCCC1)OCC 98952,N1(C(C(C)(CO)OC)=O)C2CCC1CC(NC(=O)CC1CC3CCC(C1)C3)C2 98953,C(=O)(CC(CNC(=O)CCC1CCOC1)C1CC1)N1C(C(=O)NC)CC1 98954,C1(N2C(=O)CC3(CC3)[SH]2C)CCN(C(=O)Cc2cncn2C)CC1.CC(C)C 98955,C(=O)(CCC(C(C)O)NC1CCCN1c1cccc(Cl)c1)OC 98956,c1(CC)conc1C(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)SC 98957,CC1CN(C(c2cnc(C(C)(C)C)s2)=O)CCCN1C(=O)CCSC(F)(F)F 98958,Cc1ccc(S(=O)(=O)NC(c2cccc3nnn(C(C)(C)C)c23)=O)cc1C(=O)O 98959,N1(C(CN(C(C(C)C)=O)C)=O)CCC(CNC(=O)C(C(C)O)N(C)C)C12CC2 98960,C(=O)(CCCC(C)(C)C)N1CC(C(C)C)N(C(=O)C(C)N2CCCC2)CC1 98961,C1(Cn2c(C(=O)Sc3cccs3)ccc2)CCCN1CCSC 98962,c1(-c2nc(C(C)Cn3cccc3)n(C(C)C)n2)ccc(N2CCOC2=O)c(F)c1 98963,Cc1nc(Cl)nc(N2CC3CC2(CNC(=O)CC2CCC(C)(C)CO2)C3)c1[N+](=O)[O-] 98964,Cc1c(C(=O)NC2COCC2NC(=O)Cn2cnccc2=O)[nH]c2c1CCCC2 98965,c1(C(=O)NC2C(C)CN(C(c3cnccn3)=O)C2)nc(C2CC2)ncc1Br 98966,C(C)(C(C(=O)NCC(Cl)=CCl)NC(=O)CC1(O)CCOC1)OC 98967,c1(OCC)ccc(NCC(N2CC(NC(c3sccc3F)=O)CC2C)=O)cc1 98968,c1(C(C)C)c(CNCCO)c(C#N)cn1-c1ccc(F)c(Cl)c1 98969,CC(C)C(C)(Cc1ccccc1)C(=O)Nc1cncn1-c1ccccc1 98970,c1(CC)cnc(C(=O)NCC(c2cccc(F)c2)NC(=O)C(=O)C(C)C)nc1 98971,c1(N(C)C)cccc2c1CN(c1nnc(C3CC34CC4)n1CCCOC(F)F)C2